SMILES C(=O)(CCCCCOCC)NC1C2CN(C(CC(C=C)C)=O)C1C2 N1(C(C2(C)CC2(Cl)Cl)=O)CCC(CNC(=O)CC2C=CCCC2)CC1 C1(C(=O)NCC(C(C)C)(C)NC(C2OCCC2C(F)(F)F)=O)CC(=O)C12CCC2 C(=O)(CCCC(=O)N(C)CC1CC(F)CN1C(C1CC2COCC2C1)=O)OC c1(C(=O)NCCSC2CC2C(=O)NCc2cccnc2)ccncc1C(F)(F)F c1(C(=O)NC(CNC(c2c(OC)cc(C)cn2)=O)C)sccc1S(N)(=O)=O C(=O)(CC(C)(C)CNC(=O)C(C)n1cncn1)NC(c1nc(C)oc1C)C C1(C(=O)NCC(c2ccc(Br)cc2)C)CCC(F)(F)CO1 c1(C(=O)NC2CC(NC(C(C)NC(CC)=O)=O)C(O)C2)cc2oc(C)cc2[nH]1 C(=O)(C(CC)(CC)CO)NC(CC=C)CNC(C1OC2CCC1C2)=O N1(C(CC(c2c(C)noc2C)C)=O)CC2(CCCN(C(=O)Cc3cccs3)C2)C1 N1(CC)CCC(C(=O)NCC(O)CC(=O)N(C)CCO)CC1 C#CC1CCC(C(=O)NC2CCC(NC(C3CC4CC3CC4O)=O)C2)CC1 c1(NC(c2cc(NCCN3CCCC(O)CC3)cs2)=O)ccc2c(c1)OCO2 C12(C(=O)NCC(CCCC)O)COCC1CN(C(C1OC3CCC1C3)=O)C2 c1(C(=O)NCCCC(C)(C)NC(=O)Cn2nccn2)ccn2c(O)nnc2c1 c1(C(=O)NCC(C)(C)OCC(=O)NC(CCC)(C)C)ncncc1N c1(NC(C(=O)O)CCN2CCOCC2)ccc(Br)c2c1CCCC2 C1(COC(CCC(C)Nc2cccc(OCc3ccccc3)c2)=O)CC12CCOCC2 C(=O)(N=c1[nH]nc(-c2ccc3[nH]ccc3c2)s1)NC1C(C)CCCCC1 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c1(C(=O)NC(C)CCN(C(=O)C(CC(F)F)C2CCC2)C)c(N)ccc(F)c1F N12CCC(C1CC)C2=O.C(CCC(=O)OC)NC(CSCCC)=O O=C(CC(C(F)(F)F)NC(=O)CN1C(=O)CNC1=O)NCCN1CCC(O)CC1 CCC(C(=O)N1CC2CCC(CNC(c3c(C)ncnc3C)=O)C2C1)C(F)(F)F c1(C(=O)NCC2CN(C(c3ncc(C)cc3Br)=O)C2)oc2c(C)cccc2c1C c1(CN(CCc2nc(=N)[nH][nH]2)CCO)ccc([N+](=O)[O-])cc1F C12CCC3CN(CC3C1)c1nc(ns1)C1CN2C1.C1(N(C)C)CCC(C)(C)C1 C1(C(C(N2CC(CN(C(CCOC)=O)C)C2)=O)O)CCCCC1 CCCCCC(O)CC(=O)N1CC2CC(C(=O)NCC(=O)NC)CC2C1 c1(C(=O)NC2CCN(C(CCSC)=O)CC2O)ccc2nc(C)c(=O)n(C)c2c1 c1(OC)ccc(C)cc1C(N1CCC(O)C1C(=O)Nc1ncc(O)cc1Cl)=O c1(C(N2CC(N(C(CSCC(=O)OC)=O)C)C(C)CC2)=O)noc2ccccc12 N1(C(CC(=O)NCC#C)=O)CCC2(CCCN(C(c3cc(C(C)C)on3)=O)C2)C1 C#Cc1cc(C(=O)NC(CNC(=O)C(C)(C)n2cnnn2)(CC)CC)cc(F)c1 C(=O)(C(=O)CCC(C)C)N1CCC(CCC(=O)NCC(COC)(C)CO)C1 Cn1cnc2cccc(C(=O)NCC(O)CNc3cncc(Cl)n3)c12 C#CC(C)N(C)N1CCN(c2ccccc2NS(=O)(=O)c2cccc(Br)c2)CC1 CCC(COC)C(=O)NC(c1ccccc1OC)CNC(c1sccc1CO)=O c1(C(CC)C)cc(C(=O)N(CCCCCNC(c2nsnc2O)=O)CC)on1 C1(C(=O)NCC(CN(C(=O)CCC2CC2)C)O)CC12CCSCC2 c1(NC(C2CC(C(N3CC(CNC(=O)C4CC4)C3)=O)C2)=O)cc2cccn2cn1 C1(C(c2ccccn2)NC(COC(C2CC(=O)N2)=O)=O)CC(F)(F)C1 C1(CNC(C(C)OCC)=O)CCC(C)(C)CN1C(=O)CCCc1ccccn1 C1(COC(C2C(C)CC=CC2)=O)CN(C)C(=O)CCO1 N1(C(CCOC)=O)CCN(C(c2cn(C)cn2)=O)C2CS(=O)(=O)CC12 CC1=NC(C)(C(=O)NCC23CC2CCC3(F)F)N1c1ccc(F)cc1F N1(C(CCC=CC)=O)CCC2(C1)CN(C(=O)CC1CCCCC(=O)N1)C2 N1(C(c2cc(CC)[nH]n2)=O)CC2CCN(C(c3noc(CC)c3C)=O)C2C1 C1(C#N)(C(=O)NCc2ccc(CC)s2)CCCO1.C12CC(C1)NC2=O C(CCCCCCC)OCC(=O)N(CCCNC(c1n(C=C)ncc1)=O)CCO N12CC(C)(C)CC1C(=O)NC(CCC)C2=O.C1(C(C)(F)F)(OC)CC1.SCC C(C(=O)NCC(O)CCNC(=O)C=CC(=O)NC1CC1)(C(C)C)NC(C(C)C)=O CC1(C)C(NC(=O)C=Cc2ccc(C(N)=O)o2)CCN1C(=O)C1=NNC(=O)C1 c1(C(=O)OCC)cc(NC(=O)CCn2cc(C3CCCO3)nn2)cnc1O c1(-c2ccc(CN3C(CN)CCCCC3)o2)c[nH]c2ccccc12 C=CC1CN(C(=O)C2=CCSC2)CC1NC(C1CSCCS1)=O C(C)(CCCCNC(c1cncc(N)n1)=O)NC(C1CC(OC)(OC)C1)=O C1(C(C)(C)C)CCCCN1C(=O)NCCC1CCN(CC(F)F)CC1 C12(CNC(c3c(CNC(c4c(C(C)C)ocn4)=O)n[nH]c3)=O)COC(C1)C(O)C2 C1(CC(=O)N(C)CC2CCC2c2ccccc2)Cc2ccccc2C1 c1(NCC2C(C)COC2)ccc(S(=O)(=O)NCc2ccccn2)c2ccncc12 N1(C(c2ccc(CC)cc2)=O)CCN(C(=O)CN(C)C)C(C2CCCC2)C1 c1(C(N2CC(C)C(C)(CNC(c3ccc(F)o3)=O)C2)=O)cc2cccn2c(O)n1 CC(CN(C)C(C1CCCS1)=O)C(=O)N(C1CCC1)C C=CCC(CC(=O)N1CC(CN(C)C)C1)NC(c1cn(CC2CC2)nn1)=O C1(C(N(CCCOCCNC(=O)Cc2ccco2)C)=O)CC2CC1C2 c1(CCC)sc(C(N2CC(CNC(C3(C)CCCC3)=O)CC2C)=O)cc1CC O=C(C1=NOC2COCC12)NC1(C(N2CCCC(CF)C2)=O)CC1 c1(CN(C(=O)CC2(N(C)C)CCCC2)C)cnc2sc(Br)cn2c1=O C1(OC(C)C)CCN(C(C2CC(C)N2C(=O)COc2cccnc2)=O)C1 c1(C(=O)NC2CN(Cc3ccc(N(C)C)nc3)C2)c[nH]c2nccc-2c1Cl N1(C(c2c(-c3n(C)ncc3)n[nH]c2)=O)CCOC(C)(C)C1CO C(c1csc2ccccc12)=CC(=O)N(CCNC(C1(OC)CCSC1)=O)CC C#CCCCCCC(=O)N(C)CC1(O)CCN(C(c2cn3c(n2)CCCC3)=O)C1 c1(CN(CCN)CC)ccc2nonc2c1 N1(C(C(C)SCCCC)=O)CCN(CCN(C)C(C2C(C)(C)C2(F)F)=O)CC1 c1(CNC(C2(CC)COC2)=O)cn(C)c2ccc(OC)cc12 C1(CNC(C2(SC)CC(O)C2)=O)CC(C)(C)CN1C(=O)CNC(=O)NC1CC1 C(=O)(C1SCCc2sccc21)NCC(CO)NC(CCCC)=O C1(NC(c2c(C)nc(C)[nH]2)=O)CCCC(NC(=O)CCN2C(=O)CCC2=O)CC1 c1(N2CC(CNC(CC=C)=O)OCC2)ncc(Cl)c(C(F)(F)F)n1 C1(NC(COC2CN(C(CCOC(C)=O)=O)C2)=O)CCC(C2CC2)O1.CSC c1(C(=O)NC(C(NOC(COC)COC)=O)C2CCCC2)cc[nH]c2nccc1-2 c1(CC(N2CC(O)(C(C(=O)N(CCOC(C)=O)C3CC3)F)C2)=O)cccc(C)c1 c1(C(=O)NC(C(=O)NCCCOCCCC)C2CCOC2)cnn(CCF)c1 C1(CC(=O)N(C2CCN(C(c3cc(Cl)no3)=O)C2)CCC)CCCCOCC1 N1(C(CCSC)=O)CC(=O)NCC1C(=O)NC(c1ccncn1)C C(=O)(CC1=CCOCC1)NC1C(CC)CN(C(=O)C(CO)c2ccccc2)CC1 C(CCCCC(=O)N1CC(C)(C)CC1CNC(C1CC2C=CC1C2)=O)SC N1(S(CC)(=O)=O)CCCC1C(=O)NCC1N(C(=O)Cn2cc(C)cn2)CC=C1 Cn1ccc2c(N3CC(F)(F)CC3C(N3CCN(CC4CC4)CC3)=O)ncnc12 C(C)(C)(CC(=O)N1CC(CCNC(c2sccc2C2CC2)=O)(OC)C1)OC Cc1[nH]c2c(C(=O)NC3CCCC3CNC(=O)Cn3cnnc3)cccc2c1C N1(C(CCOCC#C)=O)CC(CNC(=O)CC2CC(F)(F)C2)N2CCC1C2 C1(C)(CN(C)C(C2CCCC2O)=O)CCCN1C(c1ncoc1CCC(F)(F)F)=O c1(-c2n(CCCC)nc(COC)n2)nn(-c2ccccc2)cc1[N+](=O)[O-] C#CCC(C)C(=O)NC(C)CNC(=O)COc1ccc(C(C)C)cc1 N1(C(c2c(C)oc(Cl)n2)=O)CCC2(C)CN(C(=O)C3=COCC3)CC12 N1(CC)CC2(CNC(=O)C2)C1.N12CCC(CC1)N1CC(OC1=O)C2=O C1(NC(c2cc(CC)no2)=O)CCOCC1NC(c1cc(C)c(Br)o1)=O C1(NC(C2CCCS2(=O)=O)=O)CCC12CCN(C(=O)C(F)(F)CO)CC2 C(=O)(CCCCC(=O)N1CC2(CCC(NC(C3CCCC3)=O)C2)C1)OC N1(C(C2N(C(C)C)CCC2)=O)CCc2c(ccn2C)C1.c12cc(cn1C)NC2=O c1(N2CC(C)OC3(C2)CCCOC3)nc(=NCCC(F)F)[nH]c2cccnc12 c1(C(=O)NC2C(C(N(CC)Cc3cccc(Cl)c3)=O)C2)ccccc1CO N1(C(C=CC2N(C)CCC2)=O)CCCC(C)(C)C1CNC(c1cccc(N)n1)=O C1(C(C)C)CN(C(=O)C(C)n2ccnc2)CCN1C(=O)CCNC(=O)CO c1(C(N2C(CNC(C3CC4C=CC3CC4)=O)CC2)=O)cc(F)ccc1Br C1(C(N2CC(COC)N(C(=O)C(O)P(C)(C)=O)CC2)=O)Cc2ccncc2C1 c1(OC)ccc(C)c(CNc2ncc(CC3CCOC3=O)s2)n1 C1(COC)(CNC(C2CC2c2cccnc2)=O)CN(C(C2CC2(C)C)=O)C1 N1(C(CC(C=C)(C)C)=O)CCC2(CNC(c3coc(SC)c3)=O)CCCCC12 C=CCCC(C)(C)C(=O)N1CCCC(N(C)C(c2ccc[nH]2)=O)C1 Cn1cc(NC(c2ccc(-c3cccnc3C)nn2)=O)c(C(F)F)n1 S(=O)(=O)(c1nc2c(s1)C(=O)CCC2)NC1N(CC2C(C)(C)C2(C)C)CCCC1 Cc1cc2cccnc2nc1C(=O)NC1CCC(NC(=O)Cn2cnnc2)CC1 C1(C(=O)OCC=C)COCCC1N.N1(CC(=O)NCC(C)NC=O)CCOC1=O C(CO)(CC(F)(F)F)NC(CN(CCOC)C(C1CC(OC)C1(C)C)=O)=O c1(CNC(C(C(C)C)F)=O)nnc2n1CCN(C(=O)Cc1nc(C3CC3)cs1)C2 c1(C(=O)NC2CC3(C2)CC3C(=O)NCC2CC3(CCC3)C2)c(F)cccc1F c1(C(N2CC(C=C)C(NC(c3cnc(C)[nH]3)=O)C2)=O)sc2ccccc2c1Cl C1(NC(C2(CNC(c3cc(OC)ns3)=O)CC23CCC3)=O)C=CC(C)(C)CC1 C(=O)(C(C)(C)C1=CCN(C(c2cccnc2S)=O)C1)N1C(C)C(C)(C)CC1 CC(C)C(CCNC(=O)C(C)(C)c1ncco1)NC(=O)Cc1cscn1 C(=O)(C(C(C)C1CC1)N(C)Cc1ccccc1Br)NC(C)C Cc1cc(C)c(C(=O)N(CC(O)CNC(=O)C(c2cccnc2)O)C)s1 C1(C(=O)NCCCC(C)(C)NC(Cc2c(C)nccc2)=O)CC2CCCCN2C1 c1(C(=O)NC(C(C)NC(c2ccc(C(C)(F)F)nc2)=O)C)cccc2c1OCC2 c1(C(=O)NC(CNC(C2CC(CC(F)(F)F)C2)=O)C2CCC2)ccc(Cl)[nH]1 CC1(C)CCOC1C(=O)NCC1(NC(=O)C2=CCSC2)CC1 c1(C(=O)NCCOCCCN(C(c2ccc(CC)cc2)=O)C)cccn(C)c1=O c1(C(=O)NCC2CC(NC(c3ccc(C#C)o3)=O)C2)ccc(Cl)nc1Cl Cc1cnc2c(cnn2CC(N2CC(CCNC(=O)C(F)(F)C3CC3)C2)=O)c1 c1(C(N2CC(NC(C3CCSC3)=O)CC3(C2)CC3)=O)cc2cc(Cl)cnc2o1 c1(OCCCC)cc(C)nc(NC2CC(NCc3cccn3C)C2)n1 N(C(=NCCC(C)C)NCC1CCC2(COC2)O1)CC(c1ccc(Cl)cc1)CC Cc1n[nH]c(C)c1C(C)C(N1CCC(C(C)NC(c2ccc(F)cn2)=O)C1)=O c1(C(=O)NC2(C)CCN(C(C(C(C)C)C#N)=O)C2)ccsc1S(N)(=O)=O C1(C(=O)NCC(=O)OC)CCCN(C(c2cn(C)nc2OC)=O)CC1 Cc1cnc(C(N2CCCC(C)C2CNC(=O)Cc2nocc2C)=O)c(C)c1 CN(OC1CCCC1)C(=O)C(CNC(C1CCCN1C=O)=O)C(C)(C)C C1(c2cccc(OC)c2)CN(C(=O)COCCF)CCN1C(C1(C)C=CCC1)=O c1(N(C)C)cc(C(=O)NC2C=CC(CNC(=O)Cc3cnn(C)c3)C2)ccc1O C1(NC(=O)Cc2cnc(O)nc2O)CCCN(C(=O)CCc2cc(Cl)no2)CC1 c1(C(=O)NC2COCCN(Cc3cc(C)[nH]n3)C2)c(Br)ccc2cccnc12 C1(O)(CNC(CCC2CC(NC(C=CCCC)=O)C2)=O)CC2CCC1O2 C1(CC(=O)NCCN(c2nccc(-n3nc(C)cc3C)n2)CC)CCC2CC2C1 C1(C(=O)NC(Cc2ccn(CC)n2)=O)COCCN1CC1CC1CNC1CCC1 N1(C(C2(C)CC(=C)C2)=O)CCC(O)(C2CCN(C(C3CN(C)C3)=O)CC2)C1 c1(SC)nccnc1C(=O)NC1CCN(C(=O)CC2CCOC(C(C)C)C2)CC1 C1(C(=O)NCC(CN(C(=O)Cn2nnnc2-c2ccccc2)C)O)OCC1(C)C CC(C)CC(C)CC(=O)NC(C1(O)CN(C(=O)C(C(C)C)NS(N)(=O)=O)C1)C c1(C(=O)NC23C(NC(C(C4CC4)SC)=O)CC(CC2)C3)ccn2ccnc2n1 n1(CC(=O)NC2C=CCN(C(c3ccc(CC)[nH]3)=O)C2)[nH]cc2c(=O)ncnc1-2 N1(C(c2c(OC)n(C)nc2)=O)CCC2CCCC(C1)N2C(C1CSC1)=O N1(C(C(c2ccccc2Cl)C)=O)CC2CCC(NC(=O)C(C)CO)CC2C1 C=C=CC(C)C(=O)N1CC(F)CC1C(=O)N(C)OC C12(CNC(C3N(C(C4C(C)C4C)=O)CCOC3)=O)CCN(CC1)CC2 C123CC1CN(C2)NC(=O)C3.c1(CNC(C=CC=CC)=O)ocnc1C(=O)OC Cc1cc(=NCC(C(C)C)N2CCCS2(=O)=O)[nH]c(N2CCC(C)C(C)(C)C2)n1 C1(CNC(C=CC)=O)CC2CC(OC)C2C1.C12(CCCO1)C(=O)NC2 C(=O)(C(C)(F)C(C)(C)F)NCc1ccc(C(C)NC(c2nc(C)nn2C)=O)cc1 c1(CNCC2(C(N3C(C)C(=O)N(C)CC3)=O)CC2)cc(F)c(F)c(Cl)c1F C1(C(F)(F)F)(C(=O)OCC)CCN(C(=O)NCc2cnc(CC)s2)CC1 C1(C(=O)NCC(C)(C)CCO)(COC)CCCCCC1 c1(CC)csc(CC(=O)NCC2CCC(NC(=O)CSc3ccccn3)C2)n1 CCCC(C)(CC)C(=O)N1CC=CC(NC(=O)Cc2ccc(OC(F)F)cc2)C1 C1(C(=O)NCC=C)CC(F)(F)CN1Cc1ccc(C2CC2)cc1 N1(COC2C(SC)CCCC2)C(=O)c2ccccc2C1=O.C1CO1.C1CO1 C1(CC(=O)NCC(CC=C)NC(c2[nH]cc3c2CCC3)=O)CCC(C)(C)CO1 C1(C(=O)NC(C#C)CC2CCCC2)COCCN(C(=O)C=CCN2CCCC2)C1 c1(C(=O)NCC2(C)CCC(NC(=O)CC3CC=CC3)C2)cc(Cl)ncc1O c1(OCCCC(=O)NC(CN(C(C=C(CCC)C)=O)C)C)ccc(C)cc1Br N1(C(C2CN(CCC)C(=O)C2)=O)CCC2(CCC2NC(=O)CN(C)CC)CC1 N1(C(COC2(C#C)COC2)=O)CCC(C)(C2CC2)C1.C1(N)CCOC(C=O)C1 C1(C(N(c2nnc(COC)s2)C2CC2)=O)CCCC(OC(F)F)C1 N1(C(CONC(c2cc(CO)[nH]n2)=O)=O)CCC12CC(CO)C2 N1(C(c2cc(COC)oc2C)=O)CCCN(C(c2nc(O)sc2C)=O)C(CO)C1 N1(C(C(CCF)NC(c2nn(C)c(Cl)c2)=O)=O)CCOCC(C)(C)C1 c1(OC)nc(=NCC2CN(C(c3nc(O)sc3C)=O)CCCO2)[nH]c2[nH]cnc12 c1(C(N2CCC(N(C(c3n(CC)ncc3)=O)C)C(C)C2)=O)cc2c(nn1)CCC2 N1(C(c2ccc(C)c(Cl)c2)=O)CC(NC(=O)Cc2cscn2)C2CCCC12 C(C1CCC(C)CC1)=C(C)C(N1CC(O)(CNC(c2ncoc2C2CC2)=O)C1)=O CC1CC2CN(C(=O)CC3=CCCCC3)CC2N1C(c1cnc(N(C)C)nc1)=O c1(CCCNC(c2nc(CS(C)(=O)=O)no2)(C)C)cccc(F)c1F c1(C(=O)OCc2cc(F)cc(F)c2)c(F)cc(OC(F)F)cc1F.CC1C(=O)N1 c1(C(=O)NC2CCCN2Cc2cn(Cc3ccc(OC)o3)nn2)nn(C)c(C)c1Cl CCCCCC(=O)NCC(N1CC(CNC(=O)COCC(F)F)C(O)C1)=O n1(CC)nccc1C=CC(=O)NCC1(O)CN(C(C2CC(C)OC2C)=O)C1 c1(CC(=O)NC(C)(C)CNC(c2cscn2)=O)cc(F)cc2c1OCOC2 C1(C(=O)NCC2N(C(c3n(CC)c(O)nc3)=O)CCC2)CC1C1CCOCC1 CC1C2CN(C(=O)C(C)(C3CCCO3)C(C3CCC3)N)CC12.C1CC1 N1(C(C2CC(C(C)C)C2)=O)C2CCC1C(F)C(NC(=O)C1=CCOCC1)C2 C1(C(=O)NCC2(CNC(C3(CC#C)CCC3)=O)CC2(F)F)C2CCC(F)(F)C12 c1(CNC(C2=CCCC2C)=O)nn(C)c2c1CN(C(C1CN(C)C(=O)N1)=O)CC2 C(C(CO)C(F)(F)F)NC(C(C1CC=CCC1)NC(c1c(COC)cco1)=O)=O C(=O)(C1=NOC2(CCC2)C1)N1CCCC(F)(CNC(C(C)CC(C)(C)C)=O)CC1 Cc1cc(C(N2CCCC2)=O)cc(N)c1Cl.C1(N)CC1C1CC1 CC1CCN(C(c2cccnc2)=O)CC1NC(C1CNC(=O)N1)=O N1(C(Cn2ncc(C)c2)=O)CCC(NC(C2CC3CCC3C2)=O)CC(C)(C)C1 C1(CC=C)(NC(C2CCC3(CCC3)C2)=O)CCN(C(=O)C(CC)=CCCC)CC1 C1(C#N)(C(N(C2CCN(C(CCOCC#C)=O)CC2)CCC)=O)CC2CCC1C2 N1(c2snc(CCOC)n2)CC2CCCN(C(c3cc(Cl)ccc3F)=O)C2C1 C=CCC(C(=O)NC1COC(C(F)F)C1)NC(=O)Cc1cncs1 c1(C(=O)NCC(C2(O)CN(C(CSCC)=O)C2)(C)C)cscc1C#N N1(C(c2ccc(C)nc2O)=O)CCC2(C1)CN(C(c1ccnnc1)=O)C2 CN1CCN(C)CC(NC(=O)C(Cc2cn[nH]c2)NC(C2CCS2(=O)=O)=O)C1 c1(C(N2CCC(C(C(=O)N(C)CCOCCO)(C)C)C2)=O)cccc2cc[nH]c12 C1(C2CCC2)C(=O)N1.C1(C)(OCCNC(C2CC2)=O)CCC1.CC C1(NC(C=CC(C)C)=O)CC2(C1)CN(C(C1CCC(F)(F)CO1)=O)C2 CN1CCOCC1C(=O)NC1CC1NC(c1ccc(-c2ccco2)o1)=O C(CC1CC1)(C(=O)NC1CC(CCO)C1)OCC=CC(=O)NCc1ccccc1 CC(CCl)CS(=O)(=O)NC1CCCC2OCCC12 c1(N2CCC(O)(C(C)NC(C3CCCNS3(=O)=O)=O)C2)nccn2nnnc12 Cc1ccccc1C1(C(=O)N(C2CC(NC(=O)CC34CC(C3)C4)C2)CCO)CC1 c1(C(=O)OC2CC(NC(COC3(C)CCC3)=O)C2)cccc(OC(F)F)c1 C(CO)(C(=O)NCC1CCC1NC(=O)Cn1nnnc1-c1ccsc1)N(C)C c1(NC(C(C)C)=O)ccc(C(=O)NCC(C)(C2CC2)NC(=O)C2=CCOC2)cc1 c1(N(C)C)ccc(C(N2CCC(O)C(C(=O)NC3(CNC)CCC3)C2)=O)cc1Br N(C1CCCc2ccccc21)C(C12CCC(NC(C3CC(C)C3)=O)(CC1)CC2)=O c1(C(=O)NC(C(C)NC(=O)CCCNC(N)=O)C)cc(C#N)n(C)n1 C(CS(=O)(=O)CCS(C)(=O)=O)C1CCC(C(c2cn(CC(=O)O)nn2)C)CC1 Cc1cncc(C(=O)NC2CCCN(C(c3cc(Cl)ccc3O)=O)C2C)c1Cl n1(C(C)C(=O)NC(C)(CNC(c2cnc(S)[nH]2)=O)C2CC2)ccc(C(F)(F)F)n1 CC(CC(=O)NCc1ncccc1NC(=O)CC1CSCCO1)C(C)(C)C N1(C(CSCC(=O)OC(C)(C)C)=O)CCC(O)C(NC(=O)C2=CCCS2)C1 Cc1ncc(C=CC(=O)NC2CCC(CCNC(c3cnc(S)nc3)=O)C2)s1 c1(C(N2CC3(CN(Cc4ccc(C(=O)OCC)[nH]4)C3)C2)=O)cc(Br)ncc1Cl c1(NC(C)C)nc2ccc(C(N3CC(O)CC3CNC(=O)CC#N)=O)cc2s1 c1(C(C)C)cccc2c1OCC2NC(=O)C(F)(Cl)c1ccccc1 CC1(NC(C2CCC2c2ccc(Br)o2)=O)CN(C(C2(F)CC2)=O)C1 N1(C(C2C(=C)C2)=O)CC2(CC2)CC1C(=O)NCC1(C(C)C)CC1 N1(C(C2OCCC(NC(CSCCCC)=O)C2)=O)CC2(CCOC(=O)N2)C1 Cc1ccc2oc(C(N3CCCC(C(C)(O)CNC(=O)C=CCF)C3)=O)cc2c1 c1(C(=O)NCCC(C)NC(C(CC)COC)=O)cc2cc(Br)cn2c(O)n1 c1(C(N(CCCNC(=O)C(c2cccnc2)C)CC)=O)cccc(C(F)F)c1F C1(C)(C(=O)NCCN(C(=O)Cc2ccsc2)CC)CCCO1 CC(C)C(C)C(=O)NC1CCC(CCNC(C2(CO)CCOCC2)=O)C1 C(=O)(C(C#N)C(C)(C)C)C1CC2(C(=O)NCC(C)CN(C)C=O)C(C1)C2C Cc1cc(C(N2CCC(N(C)C(C3CC(C)(C)CO3)=O)C2)=O)nc(O)n1 CCS(=O)(=O)CCNC(=O)CC1(N(C)C)CC1.C12CCC(O1)CNC2=O C1(n2cc(CCC(C)O)nn2)CC2CCC1(NC(C1(C)CC=CC1)=O)C2 CCC(CC(C)C)C(=O)N1CCC(NC(=O)CC2CSC2)CC1C c1(CC(C)(C)OCC)cn(C2COCC2NC(=O)C(O)COC)nn1 C1(CNC(C(CNC(c2cc(OC)ns2)=O)OC)=O)CC(=O)N(C)C1=O N1(C(C2N(C(CCCCCCC)=O)CC2)=O)CCOC(C2(C)N=N2)C1 c1(OC)ccc(C(=O)NCC2CCC2NC(c2cc(Cl)cnn2)=O)c(F)n1 N1(C(c2ccc(C)o2)=O)CC(NC(c2coc(C)n2)=O)CC2(CC2)C1 C(N=c1cc(NS(C)(=O)=O)nc[nH]1)C1(NCC2OCC(C)(C)OC2)CCOCC1 N1(C(C2(C#N)CCC2)=O)CC2C=CC1C(C(=O)NCC1CC3(CCC3)C1)C2 C(=O)(CCNC(C1CC1SCCC)=O)N(CCCO)CC=C C1(NC(C(C2CC=CCC2)NC(C)=O)=O)CCn2ccnc2C1 C1(NC(=O)C2=CCSC2)CCCN(c2ccccn2)C1.O=C1CCCO1 c1(C(=O)NCCCNC(COCC=C)=O)cc(F)cc(C)c1N c1(C(=O)NCC2C(NC(C(CCC)N(C)C)=O)C2)cc(C)c(CC)nc1O c1(N(C)C)cccc(C(N2CCCC2CCNC(C2CCNC2=O)=O)=O)c1 C(C(CCCC)C(=O)NCC1CCN(C)C1)NC(C(F)=CC)=O N1(C(C(C)N(C(C)=O)C)=O)C(C(N2CC(C)CC(C)C2)=O)C2CC(F)C1C2 c1(C(N2CCC(C(C)(C)NC(C3C=CCC3)=O)CC2)=O)c[nH]c2cccnc12 S(=O)(=O)(c1ccc(Br)cc1Cl)Sc1nnc(-c2ncnc(-c3ccc(C)cc3)c2N)o1 C(=O)(CC(CN(C)C)C(F)F)NCC1N(C(COC(C)C)=O)CC(C)(C)C1 CCC(C)C(C(=O)N1CC(CNC(C2CCN2S(C)(=O)=O)=O)(OC)C1)OC N1(C(C(CC)Cc2ccc(N)cc2)=O)CC2CC(C1)N(C(=O)CNC(=O)OC)C2 C(Cc1cn(C2CCOCC2)nn1)(C(=O)O)NC(c1cc(Cl)cs1)=O C(CCCCC(=O)NC(C)(CNC(c1c(C)c[nH]c1CC(N)=O)=O)CO)SC c1(C(N2CCC(COC)(NC(=O)CC(C)F)CC2)=O)ccnc(OC)c1[N+](=O)[O-] CCCC(C(=O)NCC1(OC)CCC1)NC(N)=O.c12ccsc1C(=O)NC2 c1(C(=O)NC(CNC(c2occ(C(N)=O)c2)=O)C2CC2)csc2c1CCCC2 CCCCCC(C)CC(=O)N1CCCC1C(C)(C)C(=O)NC(C)COC(F)(F)F CCC(C)(C)CC(=O)NC1CC(C)CN(C(c2cccc(CF)c2)=O)C1 Cc1cccc2c(C(=O)NCC3CCCC(NC(=O)C(C)(C)C(N)=O)C3)c[nH]c12 c1(OC)cccc(C(C)C(N2CCN(C(c3sc(Cl)nc3Cl)=O)CC2)=O)c1 C12(NC(c3cncc(C(N)=O)c3)=O)CCN(C(C3CCSCC3)=O)CC1C2 C1(CN(C(c2ccc(C#N)s2)=O)CC)CCN(C(C2CCC(F)C2)=O)CC1 C1(NC(C(=O)NCC(F)F)=O)(CF)CCN(C(C2CC=CCO2)=O)C1 C(=O)(CC(C)C)OCCN(C(CCN(CC)CC)=O)C.C1(=O)CCN1C.C1(CN)CCC1 Cc1nn(CC(=O)NCC2CCN(C(c3ncncc3Cl)=O)C2)c(=O)n1C N1(C(C=CC(C)NC(C(n2ncc(C)c2)C)=O)=O)CCC(N(C)C)C1C C#Cc1cccc(C(C(=O)NC(CC)CC)N(C2CCCCCC2)CCC)n1 Cc1c(C(N2CCC(NC(=O)C=Cc3nnc(C(C)C)o3)CC2)=O)ccn1C C#CC1(N(C)C)CN(C(C2(C(C)NC(C3C=C(C)CS3)=O)CC2)=O)C1 c1(C(=O)NC2CN(C(C(CC)C)=O)CC2CC)nnc2ccccc2n1 C1(OC)CCOCC1C(=O)Nc1ccc(C#N)s1 c1(C(=O)C(N2CCN(C(C3CCCO3)=O)C(CO)C2)=O)ccc(F)c(F)c1F Cc1ccc(C(=O)NCC2(CNC(C3CCN(c4ncccn4)C3)=O)CC2)nc1 CCCC(C(=O)N1CCCC(CCCCNC(c2scc(C)c2C)=O)C1)C(C)C c1(C(C(N)=O)N(CC(Cc2ccccc2)OC)CCO)ccc(Cl)cc1 CC1(NC(C2CN(C3CCOC3)C2)=O)CCCN(C(=O)C(F)(F)C(F)F)C1 Nc1c(C(=O)NC(CNC(=O)CN2CCC2C)CO)cccc1Br c1(C(=O)NC2(C)CCN(C(C3(CC)CC3)=O)C2)cc2c(s1)-c1ccccc1CC2 N1(C(C(C(C)C)NC(C)=O)=O)CC2CC(NC(=O)CC3CCC(=O)N3C)C2C1 S(=O)(=O)(c1ccc2c(c1)CCC2)Nc1ncc(-c2nccc(C)c2)cc1C C(CN=c1cc(NCc2ccc(=N)[nH]c2)nc(C(C)C)[nH]1)OCCOCC c1(NC(c2nn(CC)c(C3CC3)c2)=O)ncn(C)c(=O)c1Br.C1C(C)CN1C C1(NC(CCn2c(C)nc(C)n2)=O)CCN(C(=O)C=CI)C(C)C1 CC1CC(C(N2CCC(N(C)C)(CNC(c3ccn(C)n3)=O)C2)=O)CC(=O)N1 c1(C(=O)NC2C(NC(c3c(C)coc3)=O)COCC2)ccc(C(C)C)nc1O C(=O)(C(C)CS(C)(=O)=O)N1C(CNC(c2ncc(C)c(C)c2)=O)CC1 N1(c2snc(C)n2)CCCC1C1CCCCN1C(C1(F)CCOC1)=O c1(NC(c2ccn(C)n2)C)ccc(OC(F)(F)C(F)F)cc1 O=C1CC(NC(=O)CCn2cc(CN3CCCCCC3)nn2)CCN1 c1(C(N(C2CN(C(c3cc(C(F)(F)F)n[nH]3)=O)C2)C)=O)ncn2c1CCCC2 N1(C(C(C)OCC=C)=O)CC(C)(C(=O)N(CC(C)(C)C)C)CC1(C)C Cc1[nH]c2ccccc2c1C(=O)N(C)CCNC(c1cncc(Cl)c1Cl)=O C1(NC(C2(CC#C)CCCO2)=O)CCCCN(C(=O)C=Cc2cc[nH]c2)C1 C1(NC(C2=C(C)CC2)=O)CC(F)CN(C(c2cccc(C)n2)=O)C1 N1(C(CC2N(C(C3C4CC(=O)CC43)=O)CCC2)=O)CC2(CCC(=O)O2)C1 N1(C(CC)=O)CC2CN(C(c3scnc3COCC(C)(C)C)=O)CC2C1 c1(CNC(C(CC)COC)=O)n[nH]c2c1CN(C(=O)C1=C(C)CCCC1)C2 c1(Nc2ccc(CC)cc2C(C)=O)cc(OC)c(OC)c(F)c1 Fc1cccc2nc(Nc3ccc4c(Br)n[nH]c4c3)oc12 c1(C(=O)NCC(CNC(c2c(=N)[nH]cnc2)=O)CO)ccc2c(c1)CCCCS2 N1(C(C=C(C)C)=O)CCOCC1C(C)NC(=O)Cc1ccc(C2CCC2)cc1 c1(OC)ccc(F)c(C(N2CCC(NC(c3coc(Cl)c3)=O)CC2)=O)c1 CC(C)C(F)(CNC(c1cncn(C)c1=O)=O)C(=O)N1CCC2(CCSC2)C1 c1(OC)nccnc1C(=O)NCC(O)CN(C(=O)CCSCC(C)C)C C(CC(C(=O)NCC1CN(C(N)=O)C1)NC(=O)Cn1nnc(C2CC2)n1)N(C)C CC1(CCO)CCN1C(c1n[nH]cc1CNC(C1CCCSC1)=O)=O c1(C(=O)NCC2CC(COC)CN2C(=O)COC(C)=O)cc(=O)n(C)cn1 c1(C(N2CC(CNC(c3cc[nH]n3)=O)C3C2C3)=O)cc2ccc(Cl)c(F)c2o1 c1(CN2C(CCC(=O)Nc3nccnc3Cl)CCC2)ccc(O)c2ncccc12 c1(C(N2CCC(NC(CCC=CCC=C)=O)C2)=O)ccc(C)nc1Cl c1(C(=O)NC(CN(C)C(c2ccc(N)cc2O)=O)(C)C)c(Cl)cccc1Cl N1(C(CSCC)=O)CC2CCC1C2NC(c1cc(C2(C)CC2)on1)=O N1(C(=O)CCCCC(F)F)CCC2(CCN(C(=O)C(C3CC(F)(F)C3)O)C2)C1 C1(NC(=O)OC(C)(C)C)CC(O)CN(C(C2C3CC4C(C3)C24)=O)C1.CO c1(Sc2cnc(N3CCN(C(=O)CCCCl)CC3)nc2)cnc(O)nc1O Cc1c(C(=O)NC2CC(NC(C34CCN(CC3)C4)=O)C2)ccc(C(F)(F)F)c1F C#Cc1ccc(OC)c(C(=O)NCC2(C)CCC(NC(=O)Cc3cnsc3)C2)c1 N1(C(NC2C(OC)Cc3ccccc32)=O)CC2C3CCC(C3)C2(C)C1 C12(C(=O)NCc3ccncc3)CC3CCC(CC(C3)C1)C2.C12CCC(C1)C(=O)N2 C1(C(=O)NC2CCN(C(C3(C)C=CCC3)=O)CC2)OC2CCC1CC2 N1(C(C(=O)NCCC#N)C2C(C)C2)CCCC(NC(=O)NC(C)C)C1 C1(C(N2CC(C(N)=O)(CNC(c3c(C)c(N)ccc3)=O)C2)=O)CCCCC(C)(C)C1 C(=O)(C1CC(C)(C)C1)N(CC(=O)N(C(c1ccccc1)CC)C)C(C)C CCCC(C)(C)CC(=O)N1CCC=CC1C(=O)NC(C12CCC(CO1)C2)C CCCC(CC)CC(=O)NCc1cc(C2CCN(C(C3CC3CC)=O)CC2)no1 CC1(C)CCN(C(c2c(N)cccc2Cl)=O)CC1NC(c1cccnc1)=O CC1CCC(NC(c2cnn3ccsc23)=O)CN1C(=O)CC12CCCC1C2 c1(CNC(=O)NCC(=O)NCCN(C(C2CCC(=C)C2)=O)C)cccc(C)c1 c1(C(=O)NC(CC)CC(=O)NC2COC(C)(C)C2)ccc(O)nc1C C(=O)(C1CCOc2ccccc21)NCC1C(NC(CCCN=[N+]=[N-])=O)CCC1 C(CN(C)C(C1CN(CC(C)C)C1)=O)(CO)(CO)NC(COCCC=C)=O CCCCC(=O)NCC1(O)CC(NC(=O)C(C2CC2)C2CC2)C1 c1(C(N(C(CNC(CCCCC)=O)C)CC)=O)cc2c(Cl)cc(F)cc2[nH]1 C(=O)(NNC(=O)Cc1ccccc1)NCC(C(C)c1ccccc1)O C1(C(N2CCC(CNC(Cc3c(C)n[nH]c3C)=O)C2)=O)COCC(=O)N1C(C)C CCC(C)CC(=O)NC(C)(CNC(=O)C=Cc1cnccn1)C1CC1 C(C(=O)NC(c1cnc[nH]1)C)(C(C)(C)C)NC(c1c(C)cc(F)s1)=O N1(C(c2c(OC)ccs2)=O)CCCC2CN(C(c3cnc(C)cn3)=O)CC12 N1(C(c2c(CC)ocn2)=O)CCC(CNC(C2(C#N)CCOCC2)=O)C(CC)C1 O=C(CC1COc2cc(O)ccc21)N1CCC(N(CCO)C(C2CC(O)C2)=O)C1 C(C(CNC(C1CC12CCCCC2)=O)S(C)(=O)=O)NC(C(n1c(C)ncc1)C)=O C(=O)(C1CCCc2ncccc21)NCC1OCCCN(C(c2cnc(C)o2)=O)C1 C(=O)(CC(C)CN(C)C)NCCC1N(C(C(C2CCOC2)OC)=O)CCC1 Cc1ncc(CCC(=O)NCC2COC(CNC(c3c[nH]nc3C3CC3)=O)C2)o1 c1(OC)ncc(C(=O)NCCC2CN(C(C3(C(F)F)CC3)=O)CCO2)cn1 C(=O)(CCCC(C)=O)NCC1(NC(C2C(CC)OCC2)=O)CCOCC1 C1(NC(c2cnc(C)o2)=O)CCC(C)N(C(=O)Cc2ccnc(Br)c2)C1 N1(C(C2CC(C)OCC2)=O)C2CCC1CN(C(C1(N=[N+]=[N-])CC1)=O)C2 C(=O)(CC1OCc2ncccc21)N1CCCC(NC(c2scnc2Cl)=O)(CO)C1 c1(C(=O)NCCN(C(C(C=CCCC)O)=O)Cc2ccccc2)ccncc1O N1(C(C)=O)C(C(=O)NC(C)CNC(=O)N(C)CS(=O)(=O)C2CC2)COCC1(C)C C1(NC(C2CCOC2)=O)CCCN(C(c2ccc(-c3ncc[nH]3)nc2)=O)CC1 N1(C(C(C=C)(C)CCOC)=O)CCCC2(CCCN2C(=O)Cc2coc(C)n2)C1 c1(C(=O)NCC(=C)CCNC(C2CN(C)CC(C)O2)=O)ccc2cn(C)nc2c1 c1(C(N2CCN(C(c3nccc(C)c3O)=O)CC2)=O)cccc2ccnn12 n1(CC(N2CC(CCC=C)(C(=O)NCCC3CCCOC3)C2)=O)nc(C)nc1C C1(COC)CN(C(c2ccc(Cl)nc2C)=O)CCN1C(C1CNC(=O)N1)=O CC(C)C(F)(F)CC(=O)N1CC2CCC1C2NC(=O)CN1C(=O)CN(C)C1=O N1(C(C2(CC#C)CCOC2)=O)CCC(CNC(=O)Cn2ccnn2)C(F)(F)CC1 C1(N(C(CN(C(C)=O)C)=O)C)CC2CCC(C1)N2C(=O)COc1ccccc1Cl CCC(C)CC(=O)NCC1CCN(C(=O)C(O)C2CCC2)CC1 n1(CCN(C(=O)C(O)CC2CC2)C)cc(CC2CCOCC2)nn1 CC(C)C(C)CC(=O)N1CCCC1C1CCN(C(=O)C2=CCOCC2)CC1 C1(C(=O)NCC(C)CO)CCCCN1C(=O)CN(C)C(c1ccccc1)=O CN1CCN(C(c2coc(CO)c2)=O)C(CNC(C2CCSC2)=O)C1 c1(C(N2CCC(NC(c3nc(C)c(C)s3)=O)CC2)=O)cnc2n1CCS2 C1(CNC(C2CC(C)C2)=O)C(C2CC2)CCN1C(=O)Cn1cnc(=N)[nH]1 CC(C)CC(=O)C(=O)NC1CCN(C(C2CC2C(C)O)=O)CC1 N1(C(CCSCCC)=O)CC(C(=O)NCCSC(C)C)C(C)(C)C1 c1(C(N2CCN(C(C(=O)N(C)C)=O)C3C2CCC3)=O)ccc2ccc(Br)cc2c1 C(S(=O)(=O)C(F)F)c1scc(CNC(c2coc(CN3CCCC3)c2)=O)c1 n1(C(C)C)ncc(C(=O)NCC2CN(C(=O)CC(C)O)C2)c1C(F)(F)F C1(C(=O)NC2C(C)COCC2)CC2(CC(C(=O)NC3COCCO3)C2)C1 C(C)(CSC)(C(=O)N(CC)CC1CC1)NC(c1n(CC)ccc1)=O CC(CCCc1ccccc1)C(=O)N1CC(NC(C2CC(C(F)F)C2)=O)C(C)C1 C=C=CCC(=O)N1CCC(C(F)C(=O)NCC2(O)CCSC2)C1 c1(C(=O)NC2CC(CCNC(C3C(C=C)OCC3)=O)C2)ccc(C(N)=O)cc1C C1(CNC(C(C(C)C)OC)=O)CN(C(=O)CSCCCc2ccccc2)C(C)(C)C1 CCC(C)(C#N)C(=O)NC(CNC(c1cc(O)cc(F)c1)=O)CC(C)C N1(C(C2(OC)COC2)=O)CCC2(CC1)CN(C(C1CCCN1C(C)=O)=O)CCO2 c1(C(=O)NC2C=CCN(C(C3C(C)CC(C)O3)=O)C2)cnn2c1C(=O)NCC2 CCCCCC(O)CC(=O)NCCN1CCN(C(C2(C)CC2C(F)(F)F)=O)CC1 CC(=O)CC(C)C(=O)NC1CCCN(c2cc(OC(F)F)ncn2)CC1 C(c1cn(C)nn1)=CC(=O)NCC(C1(O)CCN(C(c2ccc(=N)[nH]n2)=O)C1)C C1(CNC(CCCSCC)=O)CCCN(C(c2ccc(CC)s2)=O)C1 N#CC1CCCC(C(=O)NCCCCCCNC(c2ccc(CCF)cc2)=O)C1 C12(N)CC3CC1C2C3O.C12C3CN(CC13)C(=O)C1(c3ccsc32)CC1.CCOC C(CC(F)F)(C(=O)N1CCC(O)(CC(N)=O)C1)NC(c1nc(=N)[nH]cc1)=O C1(C)(C(=O)NCC2(C(=O)OCC)CC2)CCN(C(=O)C#CC(=O)N(C)C)CC1 C1(CNC(C(C(C)C)OC)=O)CN(C(C2(OC(C)C)CCOCC2)=O)CC1(F)F c1(C(=O)NCC2(Cn3cc(-c4cnn(CCl)c4)nn3)CC2)nnc2ccccn12 S(=O)(=O)(c1c(Br)cc(F)c(Cl)c1F)N(CCOC(CC)CC)C c1(CNc2c(O)ccc(C(F)(F)F)c2)cccc2ccsc12 N1(C(c2cc(C)c(O)nc2)=O)CCC(C2CC2)C1CNC(=O)CN(C)S(N)(=O)=O C1(NC(CCC2(C)CC2)=O)CCCC2CN(C(=O)C=Cc3ccccc3F)CC12 O=C(C1=C(Cl)CCC1)NCC12CCC1CN(C(=O)CCc1cncnc1)C2 C(=O)(C1CC2(CCN(C(C3(C#N)CC34CCC4)=O)C2)Oc2ccccc21)OC c1(CNC(c2nn(C)cc2Br)c2n(CCC)nnn2)c(Cl)n[nH]c1C c1(C(N2CC(CCNC(CC(C)(C)C3CCCO3)=O)C2)=O)[nH]nc([N+](=O)[O-])c1Cl C1(C(N(CCCN(CC)CC)C)=O)C(C)OCCN1C(C1CC2(C1)CC21CC1)=O C(=O)(C(=O)C(C)(C)CC)N1CC(CCC=C)(C(=O)NC2CCCN(C)C2)C1 N1(C(C(C)OC(=O)Cc2cccc3ccccc23)=O)Cc2ccccc2CCC1C N1(C(c2n(CC)nc(C)c2)=O)CCC2(CCCN2C(C2COCOC2)=O)C1 c1(NCCNC(c2cc(C)c(F)cc2)C2CC2)nccc(=NCCC(C)N(C)C)[nH]1 C1(CC(N2CC(CCNC(C(N(C)C)C3CC3)=O)C2)=O)CC(F)(F)C1 C1(C(=O)NCCCN(CCCNC(c2c[nH]nc2C(F)(F)F)=O)C)CNC(=O)N1 N1(CC(N2CCN(C(C3ON=C(C(C)C)C3)=O)CC2C)=O)CCc2ccccc21 c1(C(N2C(C)C(C)C2)=O)cc2oc(Br)cc2[nH]1 c1(C(N2CC(NC(=O)Cc3cnccn3)C3C2C3)=O)c[nH]c2cccnc12 c1(NC(C2(OC)CC2)=O)cccc(CC(=O)NCCN(C)C(=O)N(C)C)c1 CCCC(C)(O)C(=O)N1CCOC(CNC(c2ccccc2CCC(C)C)=O)C1 C1(O)(C(N(C2CCN(C(=O)C=CC(C)C)C2)CC)=O)CCN(C)CC1 c1(CCC)sc(C(N2CCOC(CNC(=O)C(C)C3CCC3)C2)=O)cc1CC c1(CC(C)C(=O)NCC2CN(C(=O)C(O)c3ccsc3)C2)cccc(Br)c1 c1(C(=O)NCC2OCCN(C(CN3CC(=O)NC3=O)=O)C2)cnn2c1OCC2 CC(C)CC(CNC(C1(c2ccccc2)CCOCC1)=O)NC(C1CC1C#N)=O C(=O)(C(F)(F)C1=CCOCC1)NCCC1CC(NC(c2cc(C(F)F)cs2)=O)C1 C12(C(=O)NC3(CCNC(=O)Cn4cc(Cl)cn4)CCCC3)CCCCC1OCC2 CCCC(O)(CCC)CC(=O)NC1CCN(C(c2[nH]c(C)nc2C)=O)C1C c1(C(N2CC(NC(c3c(C)cnnc3)=O)C(O)C2)=O)ccc2c(c1)NC(=O)C2 C1(COC)(NC(c2c[nH]c(Br)c2)=O)CCN(C(=O)C(C)c2ccsc2)CC1 C(C1OCCc2sc(F)cc21)NC(=NCC)NCC1CCN(C(=O)CCOC)CC1 N1(C(C(CO)N(C)C)=O)CC(CNC(C2CC(=O)CCO2)=O)C(C)(C)C1 CC(C)C(C(=O)N(C)CC1CCCCC1)C(C)NC(C1CCN(C)C1)=O Cc1cc(C)c(S(=O)(=O)Nc2ncc(CC(=O)Nc3ccncn3)s2)c(C)c1 C1(C(=O)NC(CN(CCCC)C)C)(NC(c2ccns2)=O)CCCCC1 c1(C(=O)NC(C2CC(NC(C(C)OCCCC)=O)C2)C)cccc2c1OCC2 N1(Cc2ccnc(SC)n2)CCCC2(CCCN(C(c3ccncn3)=O)C2)C1 c1(OC)nc(C)c(C(=O)NC2COCCC2NC(C2CCC(=O)N2C)=O)s1 c1(C(N2CC(CCOC)N(C(c3scnc3C)=O)CC2)=O)cc2cnn(C)c2s1 C(=O)(C(C)CCc1ccccc1F)NCC1CN(C(c2cnoc2C(=O)OC)=O)C1 Cc1ccc(Cl)c(C(=O)N(C2CCCCN(C(=O)C#CC3(C)CC3)C2)C)c1 N1(C(C(c2cccc(C)n2)(F)F)=O)CCCCC(CNC(=O)CCC(C)C)CC1 C1(CNC(c2ccc(SC)o2)=O)CN(C(c2cncn2C)=O)CC1C(F)(F)F N1(C(Cc2cc(C)nn2C)=O)CC2CCC1C1CN(C(=O)C=CBr)CC21 N1(C(C(=O)OCC)=O)CCCCC(C(=O)Nc2cc(Cl)ccc2OCC)C1 C(c1ccc(F)cc1F)=CC(=O)NC(C)CCCNC(c1ccn(C(F)F)n1)=O c1(C(=O)OC)cn(C)[nH]c1=NC(=O)N(C)Cc1nc(C2CC2)no1 C1(C(=O)NCC(CC)NC(c2csc(C(C)C)n2)=O)CCCCS1 c1(CNC(c2cnn(C)c2F)c2n(CC)nnn2)cc2ncccc2s1 C=CCC(C(=O)OCC)NC(=O)C(O)C1CCC1.C(C)(C)(C)O N1(C(C=CC(C)C)=O)CCC2(NC(c3cc(Cl)c(Br)[nH]3)=O)CC2C1 c1(NC(C(C)Oc2ccc(OC)cc2)=O)cnc2c(CCC)c1CCOC2 c1(C(N(CC(C)(C)C)CCOC)=O)ccc(Cl)c2c1OCCO2 C1(NC(COCCC=C)=O)CCCC12CCN(C(=O)C(C)C(F)F)CC2 c1(OC)ccc(C(c2nnnn2C2CCC2)NC23CC(F)(C2)C3)cn1 C1(C(=O)NCC2(C)CCCO2)CCC2CCC1N2C(=O)CC(F)(F)F C1(NC(c2cnc(C3CC3)o2)=O)COCCN(C(C23CCCCC2C3)=O)C1 C1(C(=O)NC2CC(n3cc(Cc4nn[nH]n4)nn3)C2)CC2CC3CC(C2)CC1C3 c1(N2C(C(=O)Nc3ccc(C)nc3Br)CCC2C)nc(C)c2cc(Br)ccc2n1 Cc1ccc(C(C)OC(c2c[nH]nc2C2CCOCC2)=O)nc1 C(=O)(CC1COc2ccccc21)NCC1(F)CC(NC(c2c(C)cnn2C)=O)C1 C=C(C)C(CC(=O)NC1CC2C(NC(=O)C=C3CCCCC3(C)C)C2C1)OCC C(=O)(C1OCCc2ccccc21)NCCC(C)NC(C1CC2CC1C1CC21)=O C(=O)(C(C)CCOC)NC(C(CO)NC(c1c(CC)ncs1)=O)C c1(C(N2CC(CNC(C3(C)CCC34CCC4)=O)C2)=O)ncc2ccccn12 C1(C(=O)NCC2CCOC2)(CC)CCCN(C(=O)CC2CCCC2)C1 C(=O)(C(C(C)(F)F)c1ccccc1)N1C(C(C)C)C(NC(=O)CCC(N)=O)CC1 C1(N(C(C(c2ccco2)NC(C)=O)=O)C)CCC(=O)N(C)C1 C#CC1CC2CCC1N(C(c1cc(COC)on1)C(=O)NC1CCCC1)C2 N1(C(c2cn(CCNC(CC(C)(C)C)=O)nc2)=O)CC2(C)CCC2(C)C1 NC1c2ccccc2CC1C(=O)NCc1cn(-c2ncc(Br)cn2)nn1 C=Cn1nccc1C(N1CCC(CCCNC(c2cn(C)nc2C)=O)CC1)=O C1(C)(C(N2CC(CNC(COCC(C)C)=O)C(F)(F)C2)=O)CCCNS1(=O)=O c1(OC)cc(C(N2CCC(N(C)C(C34CCC3CC4)=O)C(C)C2)=O)c(F)c(Cl)c1 N1(C(=O)NCc2n(CCOC)ncc2)CCC2(CC1)CC(n1ccnn1)CCO2 c1(C(N2CCC(NC(=O)CC3CC4(CC4)C3)C2)=O)cc2cccn2c(O)n1 C(=O)(CC(CNC=O)CC(C)C)N(CC)OC(C1CN(c2ccc(Cl)cc2)C1)=O CC(C)C(O)C(C)C(=O)N1CCCC(C)(C)C1C(=O)NCC(Cl)=CCl N1(C(CC2CCCC(C)C2)=O)CCC(F)(C(=O)NC2(C)CCCC2O)CC1 CC(CCC(C)(C)C)C(=O)NCC1CCN1C(c1ccc2c(c1O)CCC2)=O C1(CNC(Cc2cn(C)nc2)=O)CCN(C(c2ccnc(CO)n2)=O)CC1(F)F N1(C(=O)CCCN2CCOC2=O)CC(C2CN(C(=O)CC3COCC3O)C2)C1 c1(CC(=O)NCCN(C(c2csc(Cl)c2)=O)C2CC2)coc2ccccc12 CCC(CC)C(=O)NC1CC1NC(c1nc(C)n(-c2nc[nH]n2)n1)=O c1(C(=O)NC2CCCN(C(=O)Cn3ccnn3)CC2)cc(Cl)cc2c1CCC2 C1(NC(=O)CC2COCC2O)CCOCC1NC(c1cscc1C(F)(F)F)=O CC1=C(C(=O)N2CCC(C(=O)NC3CCN(C)CC3C)CC2)SCCO1 CC(C)C(C)C(=O)NCCC(C(C)C)NC(C1(N2CCCC2)CC1)=O CCN=c1ccc(C(N2CC(NC(=O)CC3COCCN3C)CC(O)C2)=O)c[nH]1 C(=O)(CCCC(=O)NC(C)CNC(=O)CN1CC=CC1)NCCC c1(CC)ccc(F)c(C(=O)NC2CC(C)CN(C(=O)CC3(CO)CC3)C2)c1F c1(C(=O)OCc2csc(CC3CCCC3)n2)cc(O)cc(Cl)c1Cl N1(C(c2cc(C(C)(C)C)no2)=O)CCOCC(C(N2CCC(O)CC2)=O)C1 CC1(C#N)CCN(C(=O)NCC2(c3ccccc3)CCCOC2)C1 c1(CC(=O)NCC(CNC(c2ccc(OC)c(O)c2)=O)C)ccn2cncc2c1 N1(C(c2cc(C(C)C)on2)=O)CCC2(C1)CN(C(c1cnncc1O)=O)CCO2 C1(NC(c2c[nH]c(=N)s2)=O)CCCOC1C1CCN(C(=O)COCCCF)CC1 N1(c2c(C)cncn2)CC2CC(NC(=O)C3=NOCC3)CC1C2 c12ccc(cn1)ON(CCC)CC(=O)NC2.C1(C=O)CC1(C)C(F)F.CC c1(NC(C(CC2CCC2)NC(CC2ON=C(C)C2)=O)=O)c(C)noc1C(C)C n1(CC)ncc(C(N2CCCC(CC(=O)NCc3cnc(C)s3)C2)=O)c1Cl CC1CCC(CC(=O)NCCC2(CNC(c3cn(C4CC4)cn3)=O)CCCC2)O1 CC(C)(C)CC(O)C(=O)NC1CCC1C(N1CCCC(O)(C(N)=O)C1)=O CCC(CC)C(C(=O)N1CC2CC1(C(=O)NC1CC(=O)N(C)C1=O)C2)OC C1(C(=O)NC2C(OC)CN(C(CN(CCC)C)=O)C2)CCc2nn(C)cc2C1 c1(C(N2CCC(F)(C(N3CCCC3CCO)=O)CC2)=O)cc(O)ncc1F C=CCC(CC)C(=O)N1CC(OCCNC(c2cc(C)c[nH]2)=O)C1 c1(C(=O)NCC(CNC(CC2C(C)CCC2)=O)O)cc(-n2ccnc2)ccn1 c1(C(=O)NC2CN(C(C(C=C=C)C)=O)CC(F)C2)occ2c1CCOC2 CCC(CCCC(=O)N(CC(C)(F)F)C)NC(c1cc(CO)n(C)n1)=O CC1(C)OC(C)(C)C1C(=O)NCC(C1CCCCC1)NC(c1cnoc1CCO)=O c1(SCC)ccc(Cl)cc1C(=O)NCCCNC(c1cc(C#N)no1)=O C1(C(=O)NCCOC(C)(C)C)C2CCC1(C)C2(C)C.CN1CCC1=O C1(C(=O)NCC2C3CN(C(C4C(CC)OCC4)=O)C2C3)CCC([N+](=O)[O-])CC1 C1(C)(C(=O)Nc2cccc(NC(C#CC(C)(C)C)=O)c2)CCCNS1(=O)=O C1(C(C)NC(=O)CCN2CCOC2=O)CCCN(C(c2cnoc2C(C)C)=O)C1 Cc1ccc(Br)c(CN(C)CC2CCC(=O)NC2)c1 C(=O)(CC(=O)N1CCCC1CNC(C1CNC(=O)N1)=O)N(C)C c1(C(=O)NCCCCCNC(CSC(C)C)=O)ccc(C2CCCO2)cc1 C(=O)(CCCC(C)(C)C)NC(CCNC(C(=O)NCCOC)=O)C c1(C(N2CCCCC(NC(CC(=O)OC)=O)C2)=O)cc2cc(C)ccc2nc1C CCC(O)(CC)CCNC(C1(NC(=O)C=CC(C)(C)SC)CSC1)=O.C(CN)SC C1(C(N2CCC(OCCNC(c3nc(C)sc3C)=O)C2)=O)CCCC(C)CC1 c1(N2CCC(NC(c3c(CC)c[nH]c3)=O)C(C)C2)ccc([N+](=O)[O-])cc1C(C)=O C1(NC(C=CC=CCC)=O)CC2CCC(C1)N2C(=O)C=CC(F)(F)F N1(C(c2c(N)nccn2)=O)CCN(C(=O)CN2C(=O)CCC2=O)C(C2CCC2)C1 N1(C(c2cncc(C)c2)=O)CCC2CCC(NC(=O)Cc3ccc(F)cc3Cl)C12 C12(CC(=O)NC3CN(CCCC=C)CC3(C)C)CC3CC(CC(C3)C1)C2 C1(NC(Cc2cc(C)no2)=O)CC1C1CCCN(C(C2CC3(C2)CC3F)=O)C1 c1(C(CNC(CC2(C#N)CC2)=O)NC(C2CC2(F)F)=O)cc(F)cc(Cl)c1 S(=O)(=O)(c1ccc(F)cc1Cl)NC1CCC(NC(c2ccc(C)c(Br)c2)=O)C1 c1(C(=O)NCCC(C)N(C(=O)C(C)C#N)C)cccc2scnc12 Cc1c(CCC(=O)N(CCCCC(=O)N(CC(O)CO)C)C)cnn1C C(=O)(CCN1C(=O)CCc2ccccc21)NCC(CC)NC(C1CC(O)C1)=O Cc1ncc2ccccc2c1C(=O)NC1CC(NC(=O)C(N)=O)C12CCC2 Cc1ccc(C)c2c(C)c(C(=O)NC3CCCC(NC(=O)CSC(C)C)C3)oc12 c1(C(C)C)ccc(O)c(C(=O)NCCCOCCNC(C2CCCN(C)C2)=O)c1 c1(C(N(C2CCN(C(C(C)OCCCCCC)=O)C2)C)=O)c(Cl)ccc(F)c1C N1(C(C=CCCC)=O)CC2(C1)OC1(C)CC2(NC(c2ccn3c2CCCC3)=O)C1 c1(C(=O)NCC(C)NC(=O)CC2CC=CCC2)cc2c([nH]1)CCC2 Cc1cc(C(=O)N(C)CC2(CNC(C3CC4CC4C3)=O)CC2)c2c(c1)CCO2 C#CCC(CC)NC(=O)C(C1(O)CN(C(=O)C(C)c2cccs2)C1)F c1(CNCC(=O)NC(C(=O)NC)C)ccc2c(c1)nnn2C C(=O)(CC(C)C(=O)NCCCCC(N1CC(=O)NCC1C(C)C)=O)OC Cc1cn(CC(=O)N(CC(C)NC(C2CCS(=O)(=O)C2)=O)CCO)c(=O)nc1O C(=O)(CC(C)(O)C(F)(F)F)NC(C1CN(C(c2cnc(C(C)(C)C)o2)=O)C1)C CC1CCC(C2CCC2)CN1C(=O)Nc1ccc(I)cc1F C1(CC(=O)NC(C#C)C2CC2)CCN(C(=O)C=Cc2ccccc2C)C12CCC2 C1(C(=O)NC2CCN(C(C3CC(SC)C3)=O)C2C)CC2(CCO1)CC(F)(F)C2 N1(C(CC(=C)C)=O)CCC(c2ccccc2)C(NC(C2(CO)CCCO2)=O)C1 N1(C(CCC2CCC(NC(CSC(C)C)=O)C2)=O)CCC(C)(C2CC2)C1 c1(OC)cccc2c1OCC(C(N1CCCC(C)C1)=O)C2.c12cc(on1)CNC2=O C1(CC#C)(NC=O)CCNCC1.c12ccccc1CO2.S(C)CC c1(C(N2C(CNC(c3c(C)nc[nH]3)=O)CC2)=O)cnn(CC(C)C)c1C N1(C(C(C)NC(=O)Cc2ccc(Cl)s2)=O)CCN(c2nc(C(C)(C)C)ns2)CC1 CCS(=O)c1ccccc1C(=O)NCC1CC(F)CN1C(=O)CN1CC2CC2C1 c1(C(N2CCCC(F)(CNC(CC(C)OC)=O)C2)=O)cc2cc(F)ccc2cn1 C1(C)(C(=O)NCC(CC=C)NC(CC2(SCC)CC2)=O)CCC(=O)N(C)C1 C(CCCCCNC(=O)COC1CCCCC1C)N(C(c1c(C)occ1)=O)C c1(C(N2CCCC(CCNC(C=Cc3occ(C)n3)=O)C2)=O)cc(Cl)n[nH]c1=N CC(CNC(C1CCC(=O)NC1)=O)N=c1[nH]nc(C(C)(C)C)o1 C1(C(=O)NC2CC(N(C)C)C2)CN(C(C2CCS2(=O)=O)=O)CC1(C)C N1(C(C(C)O)C(=O)O)CC2CC(C(=O)NCc3cc4n(n3)CCO4)C2C1 CC#CCCC(=O)N(CC(=O)N(C)CC1CCCS1)C(C)C Cc1[nH]c2c(C(=O)N(c3cc(O)ncn3)CC3CCNC3)cccc2c1C N1(C(C(C)OCCOCC)=O)CC2(CC(NC(=O)Cc3coc(C)n3)C2)C1 CC(O)CC(C)(C)CNC(c1ccc(CNC(C2CC(=C3CCC3)C2)=O)s1)=O C1(O)(CN(C(c2cn(CC=C)nn2)=O)C)CCN(C(=O)C(C)OCCCC)CC1 C(=O)(CCS(C)=O)NCCCCCNC(c1n(CC)ncn1)=O Cc1coc(C(=O)NC(C)CCN(C(=O)CSCc2ccccn2)C)c1C N1(C(C2C(C)CCO2)=O)CC2OCCN(C(c3cc4cccc(F)c4o3)=O)C2C1 Cc1cc(C(N2CC(NC(c3cnn[nH]3)=O)CC(C)C2)=O)c(F)cc1Cl c1(NC(C2(NC(C(C(COC)C)C)=O)CCC(C)(C)C2)=O)cncc([N+](=O)[O-])c1 c1(C2C(N(C3(C(N(CCCOCCN(C(C)=O)C)C)=O)CC3)C)C2)ccccc1 N1(C(c2cc(C)nc(O)c2)=O)CC2(CCN(C(c3ccoc3Br)=O)CC2)C1 N1(C(CCNC(=O)CO)=O)CC=CC1C(=O)NCC1(F)CCC1 C12(C(N)=O)CCN(C(C3CCSCC3)=O)CC1C2.C(CCCC(=O)N)OC c1(C(=O)NCCSCCNC(C2C(C(=O)OC)CCC2)=O)cc(CO)nn1C N1(C(=O)CSc2nc(-c3ccncc3)cs2)CCC(c2cccc(F)c2)CC1 CC1=NOC2(C1)CC(C(=O)NC1CCN(C(C3CCC(=O)O3)=O)C1C)C2 C1(NC(c2c(N)n(CCO)nc2)=O)CS(=O)(=O)CC1NC(c1ccc(F)o1)=O c1(COC)nc(NCc2ccoc2C)cc(N(C)Cc2ncc[nH]2)n1 c1(CCC(=O)N(CC(C)NC(C2(C)CC2C(F)(F)F)=O)C)cc(F)ccc1F C(CC(C)(c1ccccc1)Oc1ccccn1)SC.C1(=O)CCN1 C1(F)(CNC(C(n2ccc(C3CC3)n2)C)=O)CC(CNC(=O)Cn2ncnn2)C1 C#Cc1cc(C(=O)N(C2CCN(C(=O)C=COCC)C2)C)ccc1C Cc1ccc(Cl)cc1C(=O)NC1CCCC1CN(C)C(c1sccc1C1CC1)=O C(C(CC(=O)Nc1csc(C(C)(C)C)n1)C(F)(F)F)c1n(C)ccn1 C(=O)(C(C)(COC)CC)N(CC(C)NC(c1cnc(OC(C)C)c(Cl)c1)=O)CC C12CCC(CC1)C(=O)N2.c1(NC(C2(CC(C)=O)CC2)=O)cncnc1O C1(NC(c2cnns2)=O)CC(F)CN(C(C2CCS(=O)(=O)N2)=O)C1 C1(C(=O)NC(CCOCC)C(=O)NCC2(F)CN(C)C2)CC(=O)NC1(C)C Cc1cc(C(=O)NC2CC(NC(c3cccc(CCCCO)c3)=O)C2)oc1C C1(N(CCCN(C(=O)CC2CCCCC2(F)F)C)C)CCC(=O)NC1=O C1(C(=O)NC(CNC(CN(CCC)C)=O)CC)CCC2(CC1)OCCO2 CS(=O)(=O)C1CCCCN(C(=NCC2CC2)NCC(F)F)C1.c12nc(cs1)CC(=O)N2 c1(N2CCC(C(C)C)C2)nc(N2CC3CC(C2)N(C)C3)c2ncn(C)c2n1 N1(C(=O)CC2CCCN2C(c2cccnc2)=O)CCC(O)C1C(F)(F)F C1(CCNC(C2CC(OC)C2)=O)CCCN(C(=O)CNS(=O)(=O)N(C)C)C1 C1(N(C(COCCOCC)=O)C)CCN(C(C2(C)CC=CC2)=O)C1 N1(C(C2(CO)CCN(C(=O)C(F)(F)F)CC2O)=O)CCCc2cc(CN)ccc21.CO c1(CS(=O)(=O)NC2CC(C(N3CC(C(=O)OC)OCC3)=O)C2)c(Cl)cccc1Cl C1(C)(C(=O)NC2CCN(C(C(=O)NCCCCOC(C)C)C)C2)CCC(=O)C1 c1(NCC(=O)NCC2C(C)CCC2)ccc(C(C)(C)C)cc1 C1(CC)C(NC(=O)CCS(C)=O)CCN1C(=O)C(C)NC(=O)NC1CC1 c12cccc(c1)NC2=O.n1(CC(=O)OC)cc(CNC(=O)COCC(C)C)nn1 c1(C(=O)NC2CC(C(=O)NC(C)C(N)=O)C2)ccccc1Cl C(C(COC)C(=O)NCC1(NC(C2CCC(=O)NC2)=O)CC(F)(F)C1)OC c1(CN(C(=O)C2=CCSC2)C)cnn2c1CN(C(c1ccccc1Cl)=O)CC2 C1(C(=O)NC(C)CCNC(=O)CCCC#N)CCCCC1(C)C CCC(C)C(CC(=O)N1CCC12CC(O)C2)NC(=O)CC1CCCO1 c1(OC)c(C)ccc(NC(c2csc(N3CCCCC3)n2)=O)c1C N1(C(Cc2cccc(OC)c2)=O)CCOCC(NC(=O)CC2(C)CCCCC2)C1 C1(NC(Cn2c(C)ccn2)=O)CCC(C)N(C(=O)CSCCC(F)(F)F)C1 C(=O)(C(CO)C(F)(F)F)N1C(C2(NC(c3cc(SC)oc3)=O)CC2)CCCC1 N1(C(c2c(C)c[nH]c2)=O)CCS(=O)(=O)C(CCNC(=O)CCOC)C1.C1(CO)CC1 Cc1cc(C(=O)NCC2(F)CCCN(C(c3cnc[nH]c3=N)=O)C2)nc(O)n1 Cc1c(F)ccc(CN2CC3CC3(C(=O)Nc3cc(Br)cnc3O)C2)c1F c1(OC)cccc(C(N2CC3CC(NC(c4ccoc4Cl)=O)C2C3)=O)c1N C(=O)(CC(O)CC(C)C)N1CCC(C(=O)NC(c2nn[nH]n2)CC)(CC)C1 C1(C2(CNC(=O)CNC3(CCS(N)(=O)=O)CCC3)CCC2)NC(=O)NC1=O C(=O)(C1CCCc2nncn21)C(c1cnn2ccn(C)c21)=O.C(CN(C1CC1)CC)N C1(O)(C(C)NC(=O)CCN(S(C)(=O)=O)C)CCN(C(=O)Cc2ccccc2O)C1 N1(C(c2ccc(COC(C)C)cc2)=O)CCC(NC(c2cc(F)n[nH]2)=O)C(F)C1 C(=O)(C(CC(C)(C)C)NC(=O)CC1CCCC2CC12)NCC(N(OC)C)=O C1(NC(N2CC(c3c(C)nccn3)C2)=O)CC2CC(N(C)CC3(CO)CC3)C1C2 Cc1ccc2c(C(=O)NCC3(C)CCN(C(=O)C4CC4)C3)coc2c1 CC(CC(=O)NCC1CC(C)N(C(c2n[nH]c3c2CCC3)=O)C1)CC(C)(C)C C(C(C)(C)CC(=O)NCCN1CCN(C)CC1)NC(CCOCC#C)=O N1(C(C2CCCN(C)C2)=O)CCC2(CCCN(C(=O)CCCCBr)C2)C1 C1(NC(=O)Cc2csnn2)CCNCC1CO.C(c1cn[nH]c1)=C(C#N)C#N C(C(N=[N+]=[N-])C(=O)N1CCC(CNC(c2cscn2)=O)(OC)C1)OCC c1(C(N2CC(CNC(c3cccc(C#C)c3F)=O)C2)=O)c(F)c(F)cc(F)c1F CC(=O)C(C)(C)CC(=O)NCc1cc(C(N2CC=CC2CF)=O)n(C)n1 c1(C(=O)NCC(CC(F)(F)F)NC(C(C)CF)=O)ccc2c(c1)NC(=O)CS2 Nc1cc(C(=O)NC(c2ccccc2)CNC(C2(C3CC3)CC2)=O)cc(Cl)n1 Cc1cc(C(=O)NC2CC(F)CN(C(=O)CCCN3CCCC3)C2)ccc1F C(C(CC(=O)ON(C)C)C(C)C)NS(C1(c2n(CC)nnn2)CC1)(=O)=O C(C(=O)N)(C(C)C)N.C(C)(CN(C(=O)C(C)=C1CCCC1)CC)(CC(C)C)C1CCC1 Cc1nc2ccccc2nc1NC(=O)C(O)CC1CCCCC1.N12CC(C1)C2=O N1(C(c2ncc(C)cc2C)=O)CCCC2(CCCN2C(=O)CC2CCC2(C)C)C1 n1(CC(=O)NCC2CCC2C(=O)NCCC23CCCC2C3)c(O)nnc1O [N-]=[N+]=NC1CCCCC1C(=O)NC1(CCC(F)(F)F)CC1.C12CCN(CC1)C2=O N12CCCC(C1C1(OC)C(CC)COC1)CNC2=O.c1(SC)noc(C)n1 Cc1cnn(CCNC(=O)CC2(O)CN(C(=O)CCn3ccnn3)C2)c1 N1(C(c2n(C)cc(C#N)c2)=O)CCC(C2(NC(=O)C=CC=C(Cl)Cl)CC2)C1 C12(NC(Cc3cn(CC)nc3)=O)CCCC1(F)CN(C(C1CC(OC)C1)=O)C2 c1(OCCC(=O)NCCCC2CN(C(=O)CCF)CCO2)ccc(F)cc1F c1(OC)cc(CSc2c(-c3ccc(C)nc3C3CC3)ccnc2OC)ccc1I c1(NC(Cc2cc(C)ns2)=O)cc(Cl)c(I)cc1F c1(N2CCC(CCOC)(NC(=O)CNC(N)=O)CC2)ncnc(C)c1C#N CCC1=NOC(CC(=O)N(CC(C)(C)CNC(c2ccncc2NC)=O)C)C1 CCCC(CC)C(=O)NC1(CNC(c2sc(SC)cc2C)=O)CCCCC1 N1(C(C2ON=C(C(C)C)C2)=O)CCCCC(C2CN(C(c3ccon3)=O)C2)C1 Cc1cc(F)c(CC(=O)Nc2cccc(C(=O)NC(C)(C)C)c2)cc1F c1(C(=O)NCC2C(C)CCN(C(=O)CNC(=O)C3CC3)C2)cn2ccncc2n1 C=CCC(C)(C(=O)NCC(C1CC1)N(C(=O)CCC(C)OC)C)N(C)C N1(C(CC2CC(OC)C2)=O)CC(=O)CCC1C(=O)NC(C)Cn1ccnc1 c1(C(=O)NCC2N(C(COC(CC)C)=O)CCC2)c(OC)nsc1OC C1(NC(CN2CCC(C)CC2)=O)CCC12CCN(C(C1CCS(=O)CC1)=O)CC2 CCCCC(O)C(=O)N1CCC1CNC(c1ccc(Cn2ccnc2)o1)=O C(c1cncn1C)=CC(=O)N(C(C)C(N1CCC(C(=O)OC)C1)=O)C1CC1 CCCCCC(F)C(=O)NCC(C)(C)CC(=O)NCCN(CCC)CCC n1(CC)ncc(Br)c1C(=O)NCC12CC(NC(C3(C#N)CC3(C)C)=O)(C1)C2 N1(C(c2ccc(C)n2C)=O)CCN(C(=O)C(C)Oc2cccnc2)C2COCC12 O=C(N=c1ccc(-c2cccnc2C(F)(F)F)n[nH]1)NC1CC2COCC(C1)C2 c1(C(=O)NC2COCCN(c3ncnc(CC)c3F)C2)ccc2nsnc2c1 Cc1cc(C(N2CC(NC(c3cnn(CC(F)F)c3)=O)C(C)C2)=O)sc1C c1(NC2CCCN(C(c3n(C)ncn3)=O)C2)ccc(C#N)cc1[N+](=O)[O-] Cn1cc(C(=O)NCC23CC2CN(C(=O)COc2ccc(Cl)cc2)C3)ncc1=O N1(C(CCNC(=O)OCC)=O)CCC2(CNC(c3cnn[nH]3)=O)CCCCC12 c1(OCCCOC)ccccc1-c1nc(-c2ccc(OC)nc2)no1 C(=O)(N=c1cc(C(F)(F)F)n(C)[nH]1)c1sc(Br)c(C)c1Br CCCC(C)(C)C(=O)NCC1CCCCC1C(N1CCC2(CC1)N=N2)=O c1(NC2CC(NC(C3C=CCC3)=O)C2)ccc(OC(F)F)cc1 c1(C(=O)NC(C)CC(C)NC(C2(C)C=CCCC2)=O)ccccc1CO Cn1nc(C(=O)NCC2(CCNC(C34CCC3CC4)=O)CC2)c2c1CCC2 C1(C(=O)NC2C=CCC(C(=O)NCc3n(C)cnn3)C2)CC2CC(=O)C1O2 C1(NC(COCC(=O)OC)=O)CCOCC1NC(=O)CCc1ccccc1C Cc1nc2ccccn2c1C(N1CC2CC(C1)N2c1nccc(Br)n1)=O C1(F)(CNC(C(C)NC(=O)NC)=O)CCN(C(c2ccccc2SC(F)F)=O)C1 c1(C(=O)NCC2C(NC(C3C(C)C3)=O)CCCC2)cnc2ccccn12 c1(C(=O)NCC2CC(NC(C3C(COC)C3)=O)C2(C)C)ccc2cccnc2c1 CC1CC(=O)NC1C(N1CCC(NC(c2cc(C3(O)COC3)on2)=O)CC1)=O c1(C(N2C(C=CCC(=O)NC(CSC)C)CCC2)=O)ccc2[nH]ccc2c1 N1(C(C(C)Cc2ccnn2C)=O)CCC2CN(C(C3(Cl)CC3)=O)CC2CC1 c1(C(=O)NCC(C)NC(C2CC2c2cccnc2)=O)cc2c(nc1O)CCCC2 c1(C(N(C(C(=O)OCC)C)C)=O)cc([N+](=O)[O-])cc(C)n1 C(=O)(CC(C)C(F)(F)F)N1C(C(=O)NCc2onc(CC)n2)C(C)(C)CC1 N1(C(c2c(C#C)cnn2C)=O)CCCC(C2(NC(C3CCS3(=O)=O)=O)CC2)C1 c1(C(=O)NC(CCCCNC(C(CC)CCOC)=O)C)cnc2c(c1)COCC2 c1(OC)cc(C)cnc1C(N1CC2CC2(C(N2CCCC(F)C2)=O)C1)=O N1(C(C(CC=C)C)=O)CCCC(CO)(CNC(C2(CCCC)CCC2)=O)C1 C1(CC)CC(C(=O)NCC(C)CN(C(=O)CCn2ncn(C)c2=O)C)CC(=O)N1 O=C1Cc2c(N3CC4CN(c5ncc6c(n5)CCC6)CC34)ncnc2N1 C1(NC(c2scnc2C2CCCC2)=O)CCCCN(C(=O)C=CC2CCCO2)C1 N1(C(c2cc(C)sc2C)C(=O)NCCC2CC2)CCOC(C)C1C N1(CC(=O)NC(CC(=O)N(CC(CC)CC)CCC)C2CC2)CCN(C)CC1 O=C1CCC(C(F)(F)F)(NC(=O)C(=O)NCC2CCS(=O)CC2)CN1 N1(C(C(C(C)C)c2cnc(C)s2)=O)CCCC(NC(=O)COCC2CC2)CC1 O=C1CC(CNC(=O)C(Cc2cn[nH]c2)NC(=O)CN2CCSCC2)CN1 c1(CC)cc(C(=O)N(CC(O)CN(C)C(c2cncnc2)=O)C)cc(Cl)c1 Cn1nc2c(c1C(=O)NC1CC3CN(C(c4ccns4)=O)CC13)CCCC2 C1(F)(CNC(c2ccc(C(C)=O)o2)=O)COCCN(C(=O)C(C)=C2CCC2)C1 c1(C(c2n(CCCC)nnn2)NCCc2cncn2C2CC2)ccc(Cl)c(F)c1 C1(C(N2CCC(N(C(CSCC=C)=O)C)CC2)=O)CC(c2ccc(C)cc2)=NO1 C1(CC(N2CC(C(C(=O)NC3CN(C(C)C)C3)OC)C2)=O)Cc2ccccc2C1 C(=O)(C1=CC2(CCN(C(=O)C(N3CCNC3=O)C)C2)C1)NC1C(C(C)C)C1 C1(CN)CN(C(=O)C=CCN2CCOCC2)CCO1.C1(CC(=O)C=O)C2CCCC12 N1(C(c2n(CC)nnc2C)=O)CCCN(C(=O)CP(C)(C)=O)CC1C C1(O)(CNC(C)=O)CCN(C(=O)C(=O)NC2CCN(C(=O)C3CC3)C2)C1 CC(C(O)C(=O)NCCCOCCN(C(=O)CO)C)c1ccccc1F C1(CC(NOCCC)=O)CC(NC(=O)C(O)C2CC2)C1(C)C N1(C(COCC(=O)NCC)=O)CCN(C(=O)CC2CCCCC2O)C(C(C)C)C1 C1(CC(=O)N(CCN(C(=O)CC2CCCC2)CC)CC)CC(=O)NC1=O C(=O)(CC1CS(=O)(=O)c2ccccc21)N1CCC(N(C(=O)C=CCF)CC)CC1 S(=O)(=O)(c1ccc(N(C)CCOCC)c(Cl)c1)NC1C(C)COCC1.C(C)(C)(C)O CCC(Cc1cccc(C)c1)C(=O)NC1CC1NC(c1ccc(SC)cc1)=O C1(C(=O)NCC(C2CCCC2)NC(CC2(CC)COC2)=O)COCCN1CC N1(C(c2c(CC)non2)=O)CCC(F)(CNC(c2cnc(O)o2)=O)C1 C1(CC(N2C(C(C)NC(=O)C=CC(=O)NC3CC3)CCC2)=O)CCCC12CC2 Cc1nc(C)n(C2CC2)n1.c12cn(nn1)C(C)C(=O)N1CCC21 C1(C(=O)NC2CCOC(C(=O)N(C)Cc3c[nH]nc3C)C2)(CC)CCCC1O C1(NC(C)=O)CCC2(CC1)CN(C(=O)CCNC(c1ccccc1C)=O)CCO2 N1(C(COCCC#C)=O)CCC(C(=O)N(C(C)CCCC)CC)(CC)C1 c1(C(=O)NC2C3CN(C(CCC(C)(C)OC)=O)CC32)c(F)ccc(Cl)c1N c1(OC)ncc(NC(=O)CC(C)NC(C2CCCN2C(C)C)=O)cn1 C1(CC)(NC(=O)CCC2CCC(=O)NC2)CCN(C(c2cc(C)c(Cl)s2)=O)CC1 N1(C(=O)NC2C(C)CN(C)C2)CCC(C)(N2CCCC2=O)CC1 N1(C(C2CC(=C)C2)=O)CCCC1(C(=O)N(CCS(C)(=O)=O)C)CC Cc1ocnc1NC(=O)C(=O)NC(C1CCCCC1)Cc1ccccc1 c1(C(N2CC(NC(C(C)=CC)=O)C(O)C2)=O)cn2cc(Cl)cc(Cl)c2n1 n1(CC(=O)NC(CNC(C2CC(n3cccn3)C2)=O)C2CCC2)ccccc1=O C1(C(N(CCCC)CC)=O)C=CCN(C(C2CC(CCC)C2)=O)C1 C1(C(N2CCCC(NC(=O)CSc3ncccn3)C2)=O)CCCC12OCCO2 C#CC1CN(C(=O)C(O)C=C)CCN1C(=O)COC1CCCC1 c1(OC)cc(C(=O)NC2CC(C)N(C(=O)CCn3cncn3)C2)cnc1C C1(NC(=O)CC2(CO)CC2)CN(C(c2cccc3c2OCO3)=O)C2(CCOC2)C1 C1(COCC)CCCCC1n1cc(CC(=O)NC(=O)C=CS(C)=O)nn1 C(=O)(C1=C(Cl)CCC1)NC1C(C(N(C(C2CCCCC2)C)C)=O)COC1 N1(C(C2OCCN(C)C2)=O)CC(NC(=O)Cc2cccc(O)c2F)CC12CCC2 C1(C(=O)Nc2c(C)cccc2)CC2(CC2)CN1C(c1cccn1C)=O Cc1n[nH]c(=NC2CCCN(C(c3cnc(CO)nc3C)=O)CC2)s1 c1(C(=O)NCCCCN(CCCNC(C2(C)CCCO2)=O)C)cn(C)c(CO)n1 C(=O)(CCC(=O)NN(C)C)NC1CC2(C(C(N(C(C)C)CC)=O)C2)C1 C1(CNC(C2CCS(=O)(=O)C2)=O)CCC2(CCC2)CN1C(=O)COCCF C1(CC)CCCN(C(=O)C(C)OCCC(C)C)C1C(=O)NCc1ccncc1Cl c1(C(C(=O)NC(C(C)NC(c2c(CCC)nns2)=O)C)(F)F)ccc(F)cc1 Cc1coc2ccc(C(N3CC(NC(=O)C(O)CC(N)=O)CC3CO)=O)cc12 C(=O)(CC(O)C(C)C)N1C(CN(C(C(COCC)C)=O)C)COCC1 N1(C(CSCCC(C)C)=O)C(C(N2CCN(C)C(=O)C2)=O)CC2CCCC12 C1(C(=O)NC2CN(C)C2)C2CC1N(C(c1cccnc1Br)=O)C2 c1(C(=O)NCCNC(C2CCN(CC3CC3)C2)=O)ccc(OCF)cn1 C1(C(N2CCC(CCNC(c3ccc(=N)[nH]n3)=O)C2)=O)CCC2(CCC2)O1 N1(C(=O)CO)CCN(C(c2cc3n(n2)CC(O)CO3)=O)C2COCC12 C1(N(C(C2CCCC2SC)=O)CC)CCCN(C(=O)COC(C)(C)C(F)(F)F)CC1 CCC(C)(C)CCCC(=O)N1CCC(=CCNC(C2CC2F)=O)CC1 Cc1c(O)ccc(CNc2ccc(C(=O)NCc3cccs3)cc2)c1C C1(CNC(C(c2cccc(Cl)c2)OC)=O)CC2CC2N1C(=O)C(C)(F)F C#Cc1ccc(Cl)cc1NC(=O)C(C)(C)COC(F)F Cc1ccc(C)c(CCNC(c2ccccc2CNc2ccsc2C(=O)O)=O)c1 C1(c2c(CC)nc(C)nc2)NC(=O)N(CCC2CC2)C(CF)=C1C(=O)OC C(C(C(=O)NC(CC)C(=O)NC(C)CCN1CCCC1)OC)OC Cc1cccc(C(=O)NC(C)(CO)C(=O)N2CCN(CCF)CC2)c1F Cc1ccc2snc(C(N3CC4(CCN4C(c4cnc(O)c(Cl)c4)=O)C3)=O)c2c1 c1(CN2CC3(C(C(N(CC(C)C)CCC)=O)C3)C2)cccc(F)c1C#N C1(N(C(C)C(=O)NCCNC(=O)COCCCF)C)CSCN1C(=O)C(C)(C)C N1(C(C(C2CCN(C(C(C(=O)OC)(C)F)=O)CC2)C)=O)CC2CC(C1)C2(C)C N1(C(C(C)C2CC2)=O)CCC(NC(c2ccccc2-c2ccccc2)=O)C(F)C1 CC(C)CCC(F)C(=O)N1CCC(C(=O)NCC2CC3C=CC2CC3)C12CC2 C1(NC(C2(COCC)CC2)=O)CCC(NC(=O)C(C)n2ccnn2)CC1 N1(C(CC(=O)CSS(C)(=O)=O)=O)CC(N)C(O)C1.C1(NC)CC(=O)N(C2CCCC2)C1 C(c1ccc(OC)cc1OC(C)C)=CC(=O)NC(CNC(CC(CC)SC)=O)C c1(C(N2CCN(C(Cc3nc(=N)[nH][nH]3)=O)CC2)=O)ccc(SC(F)(F)F)cc1 c1(C(=O)NC2CCC(N(C)C(c3ccc(=O)oc3)=O)CC2)cc2ncccc2o1 CCN=C(NCc1cn(C2CC2)cn1)N1CCC(OCC2CCCN2C)CC1 c1(OC)cc(Cl)c(C(=O)NCC(C)(C)NC(c2ncn(C)n2)=O)cc1Cl c1(C(=O)NCCN(C(C=CC(=O)NC2CC2)=O)C2CC2)cc(F)cc2cc[nH]c12 N1(C(C(n2ccc(C)n2)C)=O)C2CCC1CC(N(C)C(c1snnc1C)=O)C2 c1(CONC(Cc2cc(OC)c(Br)cc2)=O)cc(OC)c(OC)c(I)c1 C1(NC(C(C2CC2)NC(C)=O)=O)CC(O)(C(F)(F)F)C1 Cn1nnc2cc(NC(C3(CNC(c4cc(Cl)cnc4F)=O)CC3)=O)ccc12 C1(NC(c2c(C)ncnc2)=O)CS(=O)(=O)C12CCN(C(=O)CC(C)CF)CC2 Cc1ccc(CC(N2CCN(CC(C)NC(c3ccsc3C)=O)CC2)=O)cc1F Cc1ccc(C(=O)NCC2CN(C(C3CCCC(F)C3)=O)CC2(F)CO)c(C)n1 CCC(C)(CNC(=O)CC1(OC)CC1)C(=O)NCc1nc(C2CC2)n[nH]1 c1(C(C(=O)NCCN(C)C(C)=O)N(C(C=C)(C)C)C)cccc(Br)c1 N1(C(CCNC(=O)C=CCl)=O)CC2CC(C1)N(C(C1CCOC1C(F)(F)F)=O)C2 N1(C(c2nc(CC)oc2)=O)CCC(F)C(NC(c2ccccc2CC)=O)C1 N1(C(c2ccc(CNC(C(CC)CN(C)C)=O)cn2)=O)CCCC(F)(F)C1 N1(C(c2cc(C3CCCCC3)[nH]n2)=O)CCC2(CCCC2NC(=O)C(F)(F)Cl)C1 c1(NC(c2nc(C(F)(F)F)n3c2CCCC3)=O)ccc(F)c2ccccc12 c1(C(=O)NCC2C(NC(COCC#C)=O)C2)cscc1S(C)(=O)=O C(=O)(C(C)CC(C)C)N(CC(CNC(C=Cc1cc(C)no1)=O)(C)C)C C1(c2n(C(CC)CC)nc(-c3ccc(Cl)s3)n2)CCC(C)(C)c2ccccc2C1 C1(CNC(CCCC(=C)C)=O)CN(C(C2CN3CCCC3CO2)=O)C2(CCC2)C1 c1(C(N(C)CC2N(C(CC(C)NC(N)=O)=O)CCC2)=O)cc2c(s1)CCSC2 CCC(C)(C)CN1CCC1CC(C)(C)CNC(CC(=O)O)C1CCCCC1 C1(C)(C(=O)NCCOCCCNC(c2ccc(OC)o2)=O)CC=C(C)CC1 c1(C(=O)NCC2CN(C(CC(C)F)=O)C3(C2)CCC3)cc2ccccc2cc1F C=CCCCC(C)(C)C(=O)NCC1C(O)C(O)CN1C(=O)CNS(C)(=O)=O c1(C(N2CC(CC(C)NC(c3cnnc(O)c3)=O)C2)=O)cc2c(O)cccc2[nH]1 C(=O)(CC1COCc2ccccc21)NCC(C)NC(C1COCCN1C)=O C(CC(C)(C)C)(C1CCCCC1)(N)CC.C(C(C(C)C)c1nnnn1C)C1C(C)C1 c1(NC(C2C=CCN2C(=O)Cc2ccccc2)=O)ccc(F)c(Cl)c1F Cc1ccc(C(C)C(=O)NC2CC2NC(c2ccncc2F)=O)cc1 c1(C(=O)NCCN(C(CSC)=O)C(C)C)ccc(N2CCN(C)CC2)c(F)c1 C(C(O)C(C)(C)C)N(C(CN(CC(C)C)C(c1nc(CC)oc1)=O)=O)C c1(C(=O)NCC2OCC(CNC(C3C(=C)C3)=O)C2)cc(N)cnc1Cl c1(C(=O)NC(CC=C)CNC(=O)C(CCC)OCC)ccc(C2CC2)c(Cl)c1 C(=O)(CC(F)(F)C(F)(F)F)NCC12C(CN(C(c3c(SC)nccn3)=O)C1)C2 c1(OC)cnccc1C(=O)NCCC1CC(NC(=O)CC(C)n2ccc(C)n2)C1 N1(C(c2ncn(CC)n2)=O)CC2(C)CC1(C(=O)NC1CCC(=O)NC1=O)C2 c1(C(=O)O)ccc(F)c(S(=O)(=O)N2CC(n3cc(CC4CC5CCCC45)nn3)C2)c1 C1(C2CCN(C(C3CCC3C(C)(C)C)=O)CC2)(NC(CCCC(=C)C)=O)CCC1 C12(CNC(=O)C(F)F)CCCC(CN1C(c1ccc3nc[nH]c3n1)=O)C2 c1(C(=O)NC(C2CCCO2)(C)C)cc(C(=O)NCCCCC2(CO)CC2)[nH]n1 CC1CC(NC(=O)CCc2nnc(C3CC3)o2)CN1c1cc(C(F)(F)F)ncn1 N1(C(N2CCC(C(N)=O)CC2)=O)CCOC(CNC2CCC(=C3CCC3)CC2)C1 N1(C(CC2C(CNC(c3ccc(C)s3)=O)C2)=O)CCc2ccncc21 c1(C(=O)OC)nsc(=NC(CNC(c2ccc(F)o2)=O)C(C)C(C)C)[nH]1 Cc1ccc2c(C(N3CCC(CNC(c4cnn(C)n4)=O)CC3)=O)csc2c1 c1(C(N2CC(NC(C(C)n3cccc3)=O)(CO)C2)=O)cc2c(cn1)CCCC2 C#Cc1cccc(CC(N2CC=C(C(=O)N3CC=CC3COC)C2)=O)c1 Cc1c(C(N2CCC(CN(C)C(C3(Cl)CC3C(F)F)=O)C2)=O)noc1C1CC1 c1(C(C(=O)NCc2ccco2)N(CC(=O)OC)CC2CC2)cc(Cl)ncc1F C(=O)(CCN(OC)C(=O)C(C)(C)C(O)C(C)C)NC1C(OCC)CCC1 c1(C(=O)NC(C(C)NC(COCC=C)=O)C)cc(O)c(F)cc1N C(=O)(C1=CC2CCC(C1)C2)NCC(C(=O)NCC1(O)CCC(C)(C)C1)N(C)C c1(-c2ccc(CNC(C3CCOC3c3nc[nH]n3)=O)s2)ccc(Cl)cc1 c1(CC(=O)N(CC(C)(C)O)C)cnn(C)c1NC(=O)CCCCNC(N)=O c1(C(N(CC)CC2CCN(C(C3(CO)CC3)=O)CC2)=O)cc2sc(Cl)cc2s1 c1(CN(C)C(=O)NCc2cncc(C(F)(F)F)c2)cn2ccccc2n1 c1(NCc2ccc(OCC)nc2)ncnc(N2CCC(F)(CO)C2)c1C CC1(C)CCN(C(=O)COCCc2cccs2)C1CNC(C1CC=CCO1)=O c1(C(=O)NCC(C)(O)C2CC2)cccc(NC(CCC2(C)N=N2)=O)c1.C(N)(=O)N c1(C(N(C2CN(C(c3c(C)nns3)=O)C2)C)=O)cncc2ccccc12 c1(CCN(C)CCO)cn(CC(=O)N(C)CCN2CCOC2=O)nn1 O=C(C#CC1CC1)NCCC1CSCCN1C(=O)CSc1ccccc1 N1(C(CSC(C)C)=O)CCC(C)(C)C1CNC(c1c[nH]c(C(F)(F)F)c1)=O c1(C(C)OC(c2cc(COC)oc2C)=O)ccc(F)cc1F c1(C(=O)NC2CC(N(C)C(C34CC(O)C3C4)=O)C2)c(Cl)cncc1Cl C1(CNC(c2ccc(C)cc2)=O)CCN(C(=O)C(C)C2CCCO2)C1(C)C c1(N(C(c2c(C)non2)C)C(c2cnn(C)c2)=O)ncccc1Br C1(NC(CCC(C)N(C)C)=O)CCC2CN(C(C3C(C)(C)C3(C)C)=O)CC2C1 c1(OC(C)=O)cccc(N(C(=O)C(F)(F)CC2CC2)CC2CCCNC2)c1[N+](=O)[O-] C1(CC=C)(NC(=O)C(C2CC2)OCC)CCN(c2ncc(Br)c(C)n2)CC1 N1(CC(c2cccc(SC)c2)NCC(C)C)CCCC(C)(C#N)C1 N1(c2snc(SC)n2)CCN(C(c2sc(CC3CC3)nc2C)=O)C(C)C1 N1(C(CNc2nccc(-c3c(OC)cnc(F)c3)c2)=O)CCc2n[nH]c(C)c2C1 C(=O)(C1=CCCCC1)NCCc1ccc(CNC(C2CCC23CCCO3)=O)cc1 c1(OC)ncc(Cl)cc1C(=O)N(CCCN(C(=O)Cc1ccco1)C)C C1(CC(C)NC(C2(OCC)CCC2)=O)CCN(C(=O)CC2(C#N)CC2)CC1 N1(C(C2ON=C(C(=O)OC)C2)=O)CCCC2CN(C(C3CC(C(C)C)C3)=O)CC12 C1(NC(C(CC)OCC)=O)CN(C(c2cnc(Br)s2)=O)CC(F)(F)C1 C(CC(=O)NCC12CCC(CC1O)C2)(C(F)(F)F)NC(C1C(C)SCCC1)=O N1(C(C2C(OCC)CCC2)=O)CCC(C)C(NC(c2c[nH]nc2C(C)(C)C)=O)C1 N1(C(CN(C(=O)CCc2cscn2)CCOC)=O)CC(C)SC(C)C1 CC1(C)OC(C(=O)NCC(C)(O)CNC(c2csc(Br)n2)=O)C(C)(C)O1 C1(C)(CNC(CC2C(CC)C2(F)F)=O)CCCN(C(c2c(C)nsc2C)=O)C1 Nc1ccc(F)cc1C(=O)NC1CCCC1CNC(C1CC12CC2)=O N1(C(=O)CC2CC=CC2)CC2(C1)CN(C(C1CC13CCOCC3)=O)CCO2 N1(C(COCCOCC#C)=O)CCC2OCCN(C(c3ccsc3C#N)=O)C2C1 C1(C(=O)NC(C)Cn2cc(-c3ncc(F)cc3F)nn2)CC2CC(C1)C(=O)N2 N1(C(c2cnc(CCC)s2)=O)CC(CNC(C2CC(=O)N(C)C2)=O)C(C)(C)C1 C1(C(N(CC(=O)NCc2nc(COC)sc2)C2CC2)=O)CCCC(F)C1 c1(C(N(C)CC2CCCCN2C(c2ccc(F)cn2)=O)=O)c2c(nn1C)CCC2 c1(OC)c(CC(N2CCOCC(NC(=O)C(O)C3CCC3)C2)=O)cccc1C#N C1(NCC(CN(C)C)O)CC(CNC(c2ccc(O)cn2)=O)C12CCC2 c1(SC)ccccc1C(=O)N(CCCN(C(=O)CCOC1CCOCC1)C)C N1(C(c2sccc2NCc2cnc(O)nc2O)=O)CCC2(C1)CC2(F)F c1(C2(NC(=O)Nc3c(-n4c(C)nc(C)n4)cccc3)CC2)ccc(Cl)c(Cl)c1 c1(C(N2CC(c3n(CC)nnn3)(Nc3ccnnc3O)C2)=O)cc2[nH]ccc2s1 N1(CC)CCC2(CC1)CN(C)C2.C(=O)(C(C)CC=Cc1ccccc1)N Cc1[nH]nc2ccc(NC(=O)C(Cc3cnc[nH]3)NC(=O)OC(C)(C)C)c(Cl)c12 c1(C(C)=O)c(NC(=O)CC2CN(C(C3CC3C)=O)C2)cccc1F CC1CCN(C(C2CCCSS2)=O)CC1CNC(C1CCC(=O)C1)=O N1(C(N2C(C)C(C)(C)CC2)=O)CCC2CC1CN2C(=O)OC(C)(C)C c1(C(N2CCC(NC(CCN(C)CC)=O)CC2C2CC2)=O)cc(C)c(C)nc1C CCC(C)C(C(=O)N1CCC(NC(C2CC(C3CC3)C2)=O)CC1)N(C)C(C)=O O=C(C#CC1CCOC1)NCC1CCCCN(C(c2cc3cnccc3[nH]2)=O)C1 c1(N2CCC(C)(F)C2)ccc(S(=O)(=O)NCCc2cc(Cl)cc(Cl)c2)cc1C#N CC1CC(COc2ccccc2)CN1C(c1ccc(NC(CN(C)C)=O)cc1)=O C1(C(=O)NCCCC(F)(F)F)(CC)CCCN(C(=O)C=CC(C)(C)SC)C1 c1(OCC(=O)NC(C(C)NC(C2(F)CC(COC)C2)=O)C)cc(F)ccc1F CCC(C(=O)NCC#CC(N1CCC(C2CCC2)C1)=O)C(C)(C)CC C(=O)(C#CC(=O)N(C)C)NCC1CCN(C(C(CC)F)=O)C1 c1(C(=O)NC(C(=O)N(CCCCCC)C)C2CCOC2)ccnc(OC)c1 c1(CNC(C2C(C(C)NC(=O)CCn3cncn3)C2)=O)c(O)ncnc1O C#Cc1ccc(C)c(NC(=O)C(CCC=C)NC(=O)CCCCCOC)c1 c1(CC(=O)NCCN(C)C(c2cc(C(F)F)[nH]n2)=O)ccc(-c2ccccc2)o1 CCC(N=c1nc2sccc2c(NC2CC2C2CCC2)[nH]1)C(C)C N1(C(C(C2CCCN(C(C3CC(=O)CC(=O)N3)=O)C2)C)=O)CCCN(C)CC1C N1(C(CN2CC(C)(OC)C2)=O)CCC2CCN(C(=O)CCC(C)SC)C2C1 C(C)(CC(=O)NC(C(=O)NC1(c2cc(C)on2)CC1)C1CCCO1)SC C1(C)(CNC(C2(COC)CCCC2)=O)CCN(C(c2cc(Br)n(C)n2)=O)C1 N1(C(C)=O)CCC(CNC(=O)CCNC(c2ccc(C)cc2)=O)C(C)C1 CC(=O)CCCC(=O)NCC1CN(C(=O)CCOCC2CC2)CC1C CCCCCC(CC)C(=O)N1CCC(CCNC(=O)CN2CCC(C)CC2)CC1 Cc1ccc(C(N2CCN(C(c3coc(Cl)c3)=O)C(C)C2)=O)cc1C1CC1 N1(C(CC2(OC)CC2)=O)CCC2(CCC2)C(NC(=O)CN2CC(=O)NC2=O)C1 c1(C(=O)OCc2cccc(S(C)=O)c2)cc2c(s1)C(C)(C)CCC2 c1(C(N2CCC(NC(C(CCSC)OC)=O)C(C)C2)=O)ncnc2sccc12 N1(C(CCC(=O)NCC)=O)CCCC12CCCN(C(=O)C(C)S(N)(=O)=O)C2 Cc1cc(C(N2CCC(NC(c3ocnc3C)=O)C2)=O)c(C(F)(F)F)o1 CC(CO)C(=O)N(C)CC=CC(N1CC(CN(C)C)C1)=O c1(OC)ccc(C=CC(=O)N(C)CC2CCCN(C(c3csnc3Cl)=O)C2)cc1 c1(C(N2CCC(N(C(C3(C(C)C)CCCO3)=O)C)CC2)=O)cnc2[nH]ccc2n1 c1(C(=O)NCCCCC2CN(C(C3CCN(C)C3=O)=O)C2)cc(Cl)c(F)cc1F C(Cn1cccn1)(C(=O)NCC(C)(C)C1(O)CCC1)NC(C1(CC=C)CC1)=O CC1(NCC2(C(F)F)CC(F)(F)C2)CCOC12CC2(F)F C(C)(CC1CCC1)(C(=O)NC(CNC(c1csc(C2CCC2)n1)=O)CO)OC c1(CCOCC(=O)NCC(C2CN(C(CO)=O)C2)CC)ccc(F)cc1.CC(C)(C)OC N1(c2nccc(C#N)n2)CC(NC(=O)Cn2ccc(C(F)F)n2)C2CCCCC12 c1(C(=O)NCC(C)NC(c2ccc[n+]([O-])c2)=O)c[nH]c2nccc(Br)c12 CCCCC(CNC(=O)CN(C1CCC1)C)NC(=O)C(=Cc1ccc[nH]1)C N1(C(C2CCC(C)CC2)=O)CC(CNC(c2cc(N)cc(O)c2)=O)C2(CCC2)C1 c1(C(N(C2CCCN(C(=O)CCc3ccccc3O)C2)CC)=O)cc[nH]c(=N)c1 c1(C(N2CCCC(NC(C(C)=NOC(C)C)=O)C2C)=O)oc2ccccc2c1CO C(=O)(C(C)(C)C(F)F)N1CC=CC(C(=O)NC(COC)C(C)C)C1 C1(C(=O)NC(CNC(COCCOCC)=O)C(C)(C)C)CCC2(CCC2)C1 c1(C(=O)NC2CCN(C(c3c(C)n[nH]c3C)=O)CC2O)csc2c(O)ccnc12 c1(OC)cc(CN2CCC(C)(C(=O)NCCCN3CCCCC3)CC2)ccc1Cl c1(OC(COCC#C)C)cc(Cl)cc(C#C)c1.N12CCC(C)(C1)CC2=O N1(C(C(CC)CC2CCCCC2)=O)CCCN(C(C2CCCS2(=O)=O)=O)CC1 c1(SC(C)Cc2ccc(NC(CC)(C)C)cc2)cccc(F)c1F C1(C(N(CCC)CCNC(=O)CC(C)C(C)(C)C)=O)CCc2cc(C)ccc2O1 Cc1c(C(N2CCC(F)(CNC(C3(CCO)CC3)=O)C2)=O)ccc2ccccc12 C1(NC(c2c(OC)nsc2)=O)CCN(C(=O)C(C2(O)CCCC2)F)C(C)C1 CCCCC(=O)C(=O)NCC=CCC(=O)NCCC(O)C1CCC1 Cc1[nH]nc(C(N2CC3C(C(N4C(C)CC4(C)C)=O)C3C2)=O)c1Cl Cc1cccc(OCC(=O)NC2CCC(NC(C3CCCC3C(F)F)=O)CC2)c1 CC1(C)C(c2ccc(F)cc2)CN1C(=O)Cn1cc(CN)nn1 CC(c1ccsc1)=CC(=O)NC1COCCC1NC(=O)C(C)(C)c1ncco1 C1(C(C(=O)NCC(CC)NC(C2(COC(C)C)CC2)=O)O)CCOCC1 C1(CC(N2CC(NC(C(C(C)C)(C)C)=O)C2)=O)Oc2ccccc2NC1=O C1(C(=O)OC)(C(N2CCC(C)(NC(=O)C(C(C)(C)C)SC)C2)=O)CC2(CCC2)C1 c1(OC)ccc(C(=O)Nc2nc(C(=O)Nc3cnc(Cl)cn3)cs2)cc1F Cc1cc(C2CCCN2C(=O)NCCSC(C)CCS(C)(=O)=O)cnc1C C1(C(=O)NC2CCSC23CN(C(C2CCOC2)=O)C3)CC(c2cccnc2)=NO1 N1(C(C(n2c(C)ncc2)C)=O)CCOC(CNC(c2n[nH]cc2C(F)(F)F)=O)C1 CC(c1ccccc1)=CC(=O)N(C(C)C(=O)NCC1CCC(C)C1)C1CC1 CC(C(=O)NCC(C)(C)NC(C1CCCC(C#N)C1)=O)C(C)(C)C C#CCC(C)C(=O)NCC=CCNC(c1ccc(Cn2ccnc2)cc1)=O c1(N2C(CCCOC)CCC2)ccncc1C#N.C12(CCC1)C(=O)NC2 c1(-c2cn(C(CC)CC(=O)NCC(C)CO)nn2)cc(F)ccc1N c1(NC)ccc(C(=O)NC2CCCCC2NC(=O)C(C)OCCC(C)C)nc1 C1(CC(=O)N(C(CC(=O)NC)C2CC2)C)CN(C(=O)C(C)OCC2CC2)C(C)(C)C1 c1(C(N2CCC3(C(NC(CN4CC(C)(C)C4)=O)C3)C2)=O)ccn2ccnc2c1 C(=O)(C1=CC2(CCOCC2)C1)N1CC2CC(NC(c3ccc(C)c(O)c3)=O)C2C1 C=CCC(C(=O)N1CC(CNC(=O)C=C(C2CC2)C2CC2)C(O)C1)C(C)C CCC(CCC(=O)NC1(COC)CCN(C(=O)C(C2CC2)OC)C1)OC c1(N2CCC(N(C(=O)C(C3CCOCC3)=O)C)C2)nc(C2CC2)ns1 N1(C(CC(CC)C)=O)CCC(O)C(NC(c2cncnc2)=O)C1 c1(OC)nc(C)ncc1C(=O)NCCC(C(C)C)NC(c1cc(C)cc(Cl)c1)=O C1(CN2CCC(CC(=O)NC3(CC)CC3)C2)CCN(C(=O)OC(C)(C)C)C1CC C1(C(=O)NCc2nccc(C)c2)CC12CCN(C(=O)CN(c1ncccn1)C)C2 c1(OC)cc(C)ccc1C(=O)NCC(C)NC(C1CC(F)C(=O)N1)=O.C1C(=O)N1 N1(C(c2occ(C)c2)=O)CCC(C)C(NC(=O)Cc2cnn(C(C)C)c2)C1 C(=O)(CC(C)(C)c1cccc(Br)c1)NC(C(C)NC(C=C(CC)CC)=O)C C(C(=O)NCC1CC(O)CN1C(c1oc(C)cc1C)=O)(C(C)C)NC(=O)OC N1(C(CCCOC)=O)CCCC12CCN(C(C1CCc3ncccc3C1)=O)CC2 C1(C(N(CCCC)CCO)=O)CCOC1CNC(=O)CCc1nccn1C C1(NC(c2c(C)c[nH]n2)=O)CN(C(=O)C2=CCSC2)CC12CCOCC2 CC(=O)CCCC(=O)NC(CNC(=O)COc1cccnc1)C(C)C C1(C(N2CC(CC(C(=O)NCCC(CC)CO)F)C2)=O)CCC(C)=C(C)C1 S(=O)(=O)(c1nccs1)N1C(C(=O)NC2CC(Oc3ccc(Br)cc3)C2)C(O)CC1 C12(C(=O)NCCCN(C(=O)Cc3c(F)cccc3Cl)CC)CC1COC21CCC1 c1(C(N(C2CCN(C(c3nccnc3Cl)=O)C2)C)=O)cnc(Cl)cc1Cl C1(CNC(C=C(CC)C)=O)CCCN1C(=O)C(C)c1cncs1 CC(F)(F)CCCC(=O)NC1CN(C(=O)C(F)(F)Oc2ccccc2)CC1O c1(C(N2CC(N(C(c3cnc(C)s3)=O)C)C(F)C2)=O)cnn2ccn(C)c12 c1(C(C)NC(=O)NCC(C=C)(F)F)cccnc1F C1(N(C(C=CC(C)NC(=O)CN(C2CCCC2)C)=O)C)CCNC1=O c1(C(C)C)ccc2c(c1)CN(N1CCC(O)C(F)(F)CC1)C2 C1(NC(c2n(CC)ncc2)=O)CCN(C(c2cnc3[nH]cncc2-3)=O)C12CCC2 c1(C(=O)NCC2(F)CC(NC(C(C)OC)=O)C2)cncc(-c2ccoc2)c1 c1(-c2n(C(CC)C)nc(-c3cccc(Br)c3)n2)cc2c(O)ncnc2cn1 CC(=O)CCN=C(NCCCC(F)(F)F)NCC1CC(=O)N(C(C)C)C1 N1(C(c2n(C)cnc2)=O)CCCC(CNC(=O)CCCc2ccc(Br)cn2)C1 Cn1ccc2ccnc(C(N3CCN(C(C4CC5(CCCC5)CO4)=O)CC3)=O)c12 CC(CC(=O)NC12CCC(CC1)N(C(=O)C#CC1CCC1)C2)CC(F)(F)F C(=O)(CCCCCCCCCO)NC1(CO)CCN(C(Cc2nc(C)sc2)=O)C1 N1(C(C(C)NC(C2CCCC2)=O)=O)CC=CC(NC(C2(S(N)(=O)=O)CC2)=O)C1 N1(C(C2CC(C)(F)C2)=O)CCCC2(C1)CN(C(=O)CSCc1ccccc1)C2 C1(C(N(CC(COCC)O)C)=O)(NC(=O)CC(C)(C)C)CCCC1C CC(CCCC(=O)NC1(C)CCCN(C(c2ccncc2N)=O)C1)c1ccccc1 c1(C(=O)NC2CN(C(C34CCCC(CO3)C4)=O)C2)ccc(-n2cccn2)c(F)c1 c1(C(=O)N)cc(C2CC2)oc1C.c1(COC)cn(CC(=O)C2(C(=O)NC)CC2)nn1 C1(NC(C(Br)=C(C)C)=O)CC2CCC(C1C)N2C(c1ccc(CO)cc1)=O C(=O)(C(CNC(=O)CCc1nccn1C)N(C)C)NC(COC(C)C)C c1(COC2(CC=O)N3CCCC(C2)OC3=O)cc2cc(Cl)ncc2[nH]1.C(C)(C)(C)OC c1(C(=O)NCC(CC)(C)Cl)cc(C(=O)N(C)C)cn1C CCCCCCC(CC)C(=O)N1CC2CC1CC2NC(=O)COC(F)(F)F c1(C(N2CCCCC(NC(C3C4CCCC34)=O)C2)=O)cccc2[nH]ncc12 N1(C2CCC(NC(=O)NC(C)C(=O)N(C)C)C2)CCN(Cc2ccccn2)CC1 CCCC(O)CC(=O)NC(C)CNC(c1cn(-c2cccc(F)c2)nc1C)=O c1(C(N(CCCNC(c2ccnc(-c3cc[nH]n3)c2)=O)C)=O)ccc(F)cc1N N(C1CCSc2ccc(Br)cc21)C(c1ccc(COC)cc1)=O C(=O)(C(F)C(F)(F)C(F)(F)F)N1CC(CCNC(Cn2nc(C)n(C)c2=O)=O)C1 C1(F)(C(=O)NCC(CN(C(c2c(C(C)C)[nH]cc2)=O)C)C)CCN(C)CC1 CCCCC(C(=O)N(CCC(C(C)(C)C)NC(=O)C=CC(F)(F)F)C)N(C)C S(=O)(=O)(C(C(F)(F)F)N1CCC(n2ccc3ccccc23)C1)NC(C)C C1(C2CN(C(=O)CCCNC(c3ccsc3)=O)C2)(NC(CN(C(C)C)C)=O)CC1 C#Cc1cccc(C(=O)N(CC(=O)NCC2CC2Cl)C2CC2)c1C CC1Cc2sc(C(=O)NC3CC(NC(c4cnc(O)cc4O)=O)C3)cc2C(C)C1 CC1=CC(C(=O)N(CC(=O)NCc2nc(CO)n[nH]2)CC2CCC2)SC1 c1(CC)ccc(C(=O)NC(C)CC(C)NC(=O)C=CSC)c(F)c1 c1(CSCC)ccc(C(=O)NCC2(O)CN(C(=O)C(n3cc(C)cn3)C)C2)cc1 Cc1cc(C(=O)NC(CNC(=O)C(C)C2CCCC2)CO)nc(-c2cccs2)n1 C(=O)(C(F)(F)C(F)F)N1CCC(C(=O)NCC(O)CC2CCCC2)CC1 S(=O)(=O)(c1cccc(=NCCCC2CC(N(C)C)C2)[nH]1)N1CCN(CCOC)CC1 c1(C(=O)NCC(CC)NC(C2CCCN2S(C)(=O)=O)=O)cccc(O)c1[N+](=O)[O-] Cc1ccc(F)cc1C(N1CCC(C(=O)NC2CCCC(CO)C2)C1C)=O C1(C(=O)NCCC(CC)(C)NC(=O)CCCN(C)N=O)CCC2(CCCO2)CC1 C1(CNC(c2c(C)occ2)=O)C(C)CCCN1C(C1CC(N(C)C)C1)=O.C(C)(C)(C)O C1(NC(C2CC2c2ccco2)=O)CC(N=c2cc(Cl)nc(C3CCCO3)[nH]2)C1 C1(C(=O)NCC2CC(NC(c3c(C)cccn3)=O)C(O)C2)CN2CCCC2CO1 CC(C)C(C)(C)C(=O)NC(C)(CO)C(=O)NCCOC1CC1(F)F c1(OCC)cncc(C(=O)NC2CCC(NC(=O)C(C3CCC3)OC)CC2)c1 C(=O)(C(C)(C)CF)NC1CCC(CCC(=O)NCCCCCN(C)C)C1 c1(C(=O)NCC=CCNC(c2ccc(C3CCOC3)s2)=O)cccc2nc(S)oc12 C(=O)(C(C)(C)C(=O)N(CC(C)N(C)C(c1cc(SC)oc1C)=O)C)NC C1(C(N(CCSC)CC)=O)CC2CN(C(=O)CCCC(=O)OC)CC2C1 c1(CNC(CCC2(NC(CC(C)n3ccnc3)=O)CCCC2)=O)cccc(F)c1 C1(C(N(CCCNC(=O)C(C)(F)F)CC)=O)CCCCC12CCC2 c12ccc(o1)COC2=O.C(CCN(C)C)=C(C)C C1(CC(=O)NC2(CO)CN(C(c3sccc3NS(C)(=O)=O)=O)C2)CCCCC1F C(CN=c1nc2sccc2c(N(CC(C)(C)C)C)[nH]1)c1c(C)ncs1 C1(NC(c2cnccc2Cl)=O)CN(C(=O)CCCCC2CC2)C2(CCCCC2)C1 CC1c2cc(Cl)ccc2CCN1C(c1ccc(-n2c(O)nnc2O)cc1)=O C(=O)(C(F)CC(CC)CC)N1C(C)CCC(C(=O)NCCC(C)N(CCC)C)C1 C1(N2CCN(CC(c3cccc(C(F)(F)F)c3)(C)O)CC2)CC(C)(C)OC(C)(C)C1 CN1C(=O)OCC1C(=O)NCc1nocc1C(=O)NCC(=O)N(C)C1CC1 C1(NC(c2cc(C)nc(C)c2)=O)CCC12CCN(C(c1cc(C)oc1C)=O)CC2 Cc1c(Cl)ccc2[nH]c(C(=O)N(C)CCNC(c3c[nH]c(C#N)c3)=O)cc12 c1(C(N2CC(C(=O)NCc3ccc(C)cc3)(CC)C2)=O)nccc2occc12 C1(CNC(C(c2ccccc2Cl)C)=O)CN(C(=O)CCCN(C)C)CC1(F)CO Cc1cccnc1CC(=O)NC(C)C(CO)NC(c1cc(C(C)(C)C)c[nH]1)=O c1(C(C)C)nc(=NC2CN(C(=O)C=Cc3cnc[nH]3)CC3(CCCC3)C2)s[nH]1 c1(C(C)C(N2CCC(N(C(=O)C=CCOC(C)(C)C)C)C2)=O)cccc(F)c1 C(=O)(C(C)C(C)NC(=O)C(CCSC)NC(c1cc(C2CC2)on1)=O)OC Cc1cccc2[nH]c(C(N3CC(O)CC3C(=O)NCCc3nn[nH]n3)=O)cc12 c1(CC(=O)OC)ccc(C2CC(NC(=O)C(=O)C=Cc3cccs3)C2)nc1 C#CCC(CC#C)C(=O)N(C1CC2CCC(C1)N2C(C12COCC1C2)=O)C N1(C(c2ncc(C)nc2)=O)CC2CC(NC(c3cncc(Cl)c3Cl)=O)CC2C1 Cc1c(NC(=O)CC2CCCC2NC(=O)CNC=O)cnn1CC1CC1 CCC(C(=O)NC1CC(CCNC(=O)Cc2n[nH]c(=NC)s2)C1)C(C)(F)F CN(C1CCCC1S)N(C)Cc1ccccc1-n1cccn1 N1(C(CNC=O)=O)CCN(C(=O)Cc2cccc3c2OCCO3)C2CCCC12 C1(CNC(C2OCC(C)(C)C2)=O)CCN(C(c2cnsc2)=O)C12CCC2 c1(N(C(C)C(=O)OCC)CC)ccc(C(C)(C)C#N)cc1 C1(OC)(CNC(=O)C(C)(O)C2CC2)CN(C(c2cc(-c3cccs3)[nH]n2)=O)C1 c1(C(=O)NCC(=C)CCNC(=O)C(CC)C(C)O)cnc(P(C)(C)=O)cn1 c1(C(N(C(C)CNC(c2csc(C(C)OC)n2)=O)CC)=O)ccnnc1O c1(C(=O)NCC2(F)CN(C(c3ccc(Cl)nc3O)=O)C2)c[nH]c2ccc(F)cc12 N1(C(C2CC2SCC(=O)NC(C)CSC)=O)CCC(Cc2cccs2)CC1 c1(N(C)C)ccc(C(CNC(=O)C=CSC)NC(=O)C(C)(C)N(C)C)cc1 Cc1cc(CC(=O)NCCC(O)CNC(c2cccn2-c2ccccc2)=O)n[nH]1 CCC(CC(=O)NCC1CC2(CC(NC(=O)C(O)CC(C)C)C2)C1)C(F)F CCC(CC)C(=O)NCC1(F)CCN(C(=O)CC2CC(OC)C2)C1 C#Cc1cccc(N2CCN(Cc3nc(Br)nn3CC)CC2)c1 c1(OC)ccc(F)c(C(=O)NCC(F)CNC(C2CCSCC2)=O)c1F c1(C(N2C(CNC(CC(C)c3cccnc3)=O)C=CC2)=O)ccn2ccnc2c1 Cc1ncc2ccc(C(=O)NC3CC4CC(NC(c5ccncn5)=O)CC34)cn12 CC1(C)CC(CNC(c2n[nH]cc2Br)=O)N(C(c2ccc(Cl)cc2N)=O)C1 C(CC(C)CC)(C(=O)N1CCCN(C=O)CC1)NC(c1c(CC)cccn1)=O O=C(CCCCc1ccccc1)NC1CC(F)(CNC(=O)C(F)(F)C2CC2)C1 c1(NC(=O)C(C)N(C)C)cncn1C.C1C(O)CCC(C)=CC(=O)N1C C1(C)(CNC(C=COCC)=O)CCN(C(=O)CC2CC=CC2)C1 C1(N)CN(N2CCCS2(=O)=O)CC2(CCC2)C1.c1(C(=O)O)ccc(C)c(Cl)c1 C1(CC)CN(C(C2CCC(=O)C2)=O)CC1C(=O)Nc1csnc1C1CC1 C(=O)(C(C)(C)C(=O)NCc1cccc(C(=O)NC2CCOCC2(C)C)n1)NC N1(CC(N2CC3C(C2)N3C(c2cocn2)=O)=O)C(=O)CNC1=O C(C(=O)OCC=CC(F)(F)F)(c1cccs1)NC(=O)OC(C)(C)C C1(NC(CSC)=O)C=CCN(C(c2ccc(N3CCCS3(=O)=O)cc2)=O)C1 c1(C(=O)NC(CC)CCOC)cccnc1CNC(=O)CC1CC2CC2C1 c1(C(=O)NC(C2CCCN2C(=O)Cc2ccccc2)C)ncc(Cl)cc1F C(C(CC(=O)NC1CCCNC1=O)C1CCC1)NC(c1cc(C2CC2)on1)=O N1(OCC)CCC(C(N2CCC(n3cc(CCc4ccccc4)nn3)C2)=O)CC1 c1(C(C(=O)NC2CC2)N(CCOCC2CC(SC)C2)CC)ccn(CC(F)F)n1 n1(CC)nc(C)cc1C(=O)NCC1(F)CCN(C(=O)COCC2CCCCO2)C1 c1(C(N2CCN(c3ccncc3)C(=O)C2)=O)cc2c(s1)-c1ccccc1CC2 C1(NC(C=C(COC)C)=O)CCN(C(c2c(F)cncc2Br)=O)CC1C N1(C(CCCCC#C)=O)CCC2CC2(C(=O)N(CCCCN=[N+]=[N-])CC)CC1 N1(C(c2c[nH]c(=NC)s2)=O)C2CC=C(C(=O)NCC(C)(O)CC(C)C)C1CC2 C=CC1(C(N2CC(O)CC2CNC(C2CC=CCO2)=O)=O)CCCCC1 C1(NC(CCNS(CC)(=O)=O)=O)CC2CC1CN2C(c1cccn2cnnc12)=O C(C(=O)N(C1CC(C)C1)C)(C(C)(C)C)NC(CC(C)(C)SC)=O c1(NC2CCC(C(=O)NCc3c(OC)cccc3)C2)cccc(Cl)c1OC c1(CC2C(C(=O)NCCCOCC(F)(F)F)C2)ccc(Br)c2nsnc12 c1(OC)cc(C(N2CC(NC(c3cccc(Cl)c3)=O)CCC2C)=O)cc(C)c1 c1(C(N2CC3C(CC(N4CCC(F)CC4)=O)C3C2)=O)cc(F)cnc1O C=CCC(CNC(C1(C)CCC1)=O)NC(c1conc1C1CCC1)=O C(Cc1cn[nH]c1)(C(=O)NCC(F)F)NC(CCOCCOC)=O c1(C(=O)NC(CNC(C(CC)SC)=O)(C)CC)cc2c(C)c(C)ccc2[nH]1 C1(C(N(C2CCN(C(c3ccc(Cl)c(Br)c3)=O)C2)C)=O)CCc2nn[nH]c2C1 c1(CC)cnn(C)c1C(C(=O)NC1CCCO1)N(C)CCOCC1CC1 C1(c2nnnn2CC(F)F)(NC(CC)(C)C)CCC(P(C)(C)=O)C1 c1(C(=O)NCCC(C)NC(CS(CC)=O)=O)nc2ccccn2c1F CC1CN(C(=O)CCc2cnn[nH]2)CC(C)N(C(=O)CC23CCC(CC2)CC3)C1 c1(SC)c(C(=O)NCC23CC(NC(=O)C(C)C(F)F)(C2)C3)[nH]c2ccccc12 c1(OC)nc(C(=O)NCC2CCCCN2C(=O)C=Cc2nnn(C)n2)sc1C N1(C(c2nn(CC)c(O)c2)=O)CC2CCCC(C1)N(C(c1ccns1)=O)C2 C(CC(O)C(F)(F)F)N.N1(C(=O)OC(C)(C)C)CCC(NC(N2CC(CF)C2)=O)CC1 CCC(C)CC(C)C(=O)N1C2CC1CN(C(C1SCC=C1C)=O)C2 C(=O)(C1=NNC(C(F)(F)F)C1)N(CCC(C)NC(C1CC(CCC)C1)=O)C N1(C(C(c2c(C)cccc2C)O)=O)CCOCC(F)(CNC(=O)C2CC2)C1 C12C(C1(C)C)CNC2=O.C(=O)(CCOC1CCC1)NC(C1(O)CCC1)C C1(NC(CC)=O)CN(C(c2ccc(C)c(C)n2)=O)C2(CCCOC2)C1 c1(C(N2CCC(O)(C(C)NC(c3ccnn3C)=O)CC2)=O)ccc(F)c(Cl)c1N CC(CCC(C)(C)C)C(=O)NC1CCCCCC1C(N1CCC([N+](=O)[O-])CC1)=O Cc1cnc(C(=O)NCC(CO)NC(c2csc(C)c2C)=O)cc1Br N1(C(c2c(C)cc[nH]2)=O)CCN(C(=O)CCC(N)=O)C(CC(C)(C)C)C1 C12(C(=O)NCC3(CNC(C(C)NC(N)=O)=O)CC3)CCC(C)(CO1)C2 c1(C(N(CCCCCCNC(=O)CC2COCCO2)C)=O)cncc(C(F)F)c1 C1(C(N(C(C)C)CCN(C(=O)C(F)(F)c2cscn2)C)=O)CCC(C2CC2)CC1 Cc1cc(C(=O)NCC2CCCN2C(=O)COCCF)c(C(F)(F)F)o1 C1(NC(C(C)C2CC2)=O)COC2(CNC(c3c[nH]ccc3=N)=O)CC1C2 c1(CC2CCN(C(NOC(CC)CC)=O)C2)cccc(Cl)c1 CC1(CNC(c2ccncc2)=O)CCN(C(=O)COC2CC2(F)F)C1 C12(CNC(CCSCC)=O)CC(NC(c3cnc(SC)[nH]c3=N)=O)(C1)C(C)(C)O2 c1(CCCC(=O)NCC2CCC(NC(COCC=C)=O)CC2)ccc(CC)cc1 C1(C(=O)Nc2c(C)ccc(F)c2)CCC2(CN(C(C3(C)CCC3)=O)C2)O1 C12(CNC(CCCNC(C)=O)=O)COC(CNC(=O)C(c3cccs3)SC)(C1)C2 Cc1cc(C(=O)NCC(C2CC2)NC(C2CCCC23CC3)=O)nc(O)c1 Cc1c(CC(N2CC=CC(NC(c3cc(Br)cn3C)=O)C2)=O)ncn1C Cc1cc(F)ccc1CC(=O)N(CCCNC(C1CC1C(F)(F)F)=O)C c1(OC)ccc(F)c2[nH]c(C(=O)NC3C4CC3CN(C(=O)C(C)C3CC3)C4)cc12 CC1CC(NC(c2ccc(F)o2)=O)CCN1C(C1CC2CC2CC1C)=O c1(C(=O)NCCC2CCCN(C(=O)C=Cc3cc[nH]n3)C2)cc(O)nc(O)c1 C(=O)(C(O)C(C)(C)C)N(C)CC1CN(C(=O)C(N2CCOCC2)C2CC2)C1 CCCC(C)CC(=O)N1CCCC(N(C)C(c2c[nH]nc2OC)=O)C1 Cc1ccc(C(=O)NCCC2(O)CCN(C(=O)C(C)P(C)(C)=O)CC2)nc1O C1(NC(c2cncc(N)n2)=O)CCCCN(C(=O)Cc2cc(C(F)F)no2)C1 O=C(C1=CCCCO1)NCc1csc(CNC(c2cccc(Cl)c2O)=O)n1 c1(CC(=O)N(CCCNC(C2CC2[N+](=O)[O-])=O)CC)cccc(OC)c1Cl N1(C(C2(CO)CC(C)(C)C2)=O)CCCN(CCNC(C23CC(C#N)(C2)C3)=O)CC1 c1(C(=O)NC(C(=O)N(C)Cc2c(CC)noc2)COC)cncc(OC)c1 c1(CNC(=O)NC(C)CCC(F)(F)F)cnc2ccccn12 O=C(C1OCCn2ccnc21)NC12CC1CN(C(=O)CCn1ccnc1)C2 C1(C(=O)NC(c2csnn2)C)CC2(CCN(C(=O)CN3CCOC3=O)C2)C1 N1(C(C(C2CCN(C(=O)CC3OCCOC3C)C2)C)=O)CC2(CCC2)C1 c1(C(N(CC(C)NC(c2ccc(C(C)C)o2)=O)CC)=O)ccccc1SC(F)F CC1CCC(CNC(=O)CCSC(F)(F)F)CN1C(c1nnc(O)cc1O)=O C1(CNC(C(CCN(C)C)O)=O)(NC(=O)Cc2ccc(C)s2)CCCCC1C n1(CC(=O)NC(CC)CN(C)C(C2Cc3nccn3C2)=O)c(C)cc(O)cc1=O C(=O)(C(O)C1=CCCCC1)NC1CC(NC(C2CCC2(F)F)=O)C(O)C1 c1(CC)nc(C(=O)NCc2cc(C)sn2)co1.C12(CCCC1)CCC(=O)N2 c1(OC)cccc(Cn2nnnc2C(c2csc(-c3ccco3)n2)NC(C)C)c1 C(=O)(C(CCC1CC1)Nc1cccnn1)OCC(N)=O C1(C(=O)NC(CNC(C(C(C)C)C2CCC2)=O)(C)C)CCC2(CCC2)O1 C1(C(=O)NCC(CNC(=O)C(F)(F)C2(O)CCC2)OC)CC2CCCC12 c1(OCC)ccc(C(=O)NCC2(N(C(=O)C=CCO)C3CC3)CCOC2)cc1 N1(C(Cc2c(C)cc(Cl)cc2)=O)CC2CCN(C(C3SCCS3)=O)CC12 C(CCOC)(C(=O)NCCN1CCC(N(C)C)C1)NC(C1CC(=C)C1)=O c1(OC)ccc(CCC(N2CCC(C)(CC(=O)Nc3cc(O)ccn3)C2)=O)cn1 c1(OCC)cncc(-c2cn(CCCNC(=O)C=C(C3CC3)C3CC3)nn2)c1 CCCCCCC(C)CC(=O)N1CCCCC(NC(=O)C(F)(F)c2nccs2)C1 N1(C(CC=C=C)=O)CCC2(CC(NC(=O)C(C)CSC)C2)C1 c1(SC)ccc(N)cc1C(=O)N(C)CC1(O)CCN(C(=O)C2CC2)CC1 c1(CC)cc(C2CC(N)C2)ccc1NC(N1CC(c2ccc(Br)cc2)CC1C)=O c1(C(C)NC(=O)CCC2CC(NC(=O)CCCC3CC3C)C2)cc(O)ncn1 CC1CCN(C(C2CCC=CC2NC(=O)CCc2cnccn2)=O)CC1O c1(CSC(C(C)O)C)nc2cc(Cl)ccc2n1C C(=O)(NN1CCCC1C(=O)NCc1nnn(C)c1C)c1cc(C)c(C)o1 Cc1cc(N)c(C)nc1C(N1CC=CC(NC(=O)CCOCC2CCCO2)C1)=O c1(CC)c(C(=O)NCC2(O)CCN(C(=O)C=CC3CCCO3)C2)cnn1C C1(CCC)CN(C(=O)C(F)C(C)(F)F)CCN1C(=O)C(C(C)C)C1CCC1 C#Cc1ccc(F)c(NC(CC(C2CC2)SC)c2nnnn2CCCSCCC)c1 C=Cn1nccc1C(=O)NCC1CC1CNC(C1(Cl)CC12CCC2)=O S(=O)(=O)(c1cccc(C(=O)NC2CC(C)(C)OC2=O)c1)N(C1C(C)OCC1)C C12(NC(C(COC)OC)=O)CCC(CC1NC(C13CCC(CC1)C3)=O)C2 Cc1ccc(C(N2CC(NC(=O)CC3CCCC34CC4)CC(C)C2)=O)c(F)c1C c1(CNc2cccc(C(=O)Nc3nc(C)c(C)s3)c2)cccc(F)c1Br C(=O)(C(C)(CO)NC(c1ccc(C)cn1)=O)NCC(CCC)O C1(CC=C)(NC(=O)C=Cc2ccsc2)CN(C(c2csc(COC)n2)=O)C1 c1(C(N2C(CN(C(=O)C=CS(C)=O)C)CCC2)=O)ccc2oncc2c1 CC(c1ccccc1)=CC(N1CCN(C(=O)CCCC(=O)N(C)C)CC1)=O C1(O)C=CCS1.C(C(=O)NCC=CC)OCCCOCCOC.C1CO1 Cn1cc(C(N2C(CNC(C3CC=CC3)=O)CC3CC23)=O)c2ccccc2c1=O C1(NC(Cc2ccc(C)cc2)=O)CN(C(c2cnc(C)cn2)=O)C2(CCC2)C1 N1(C(c2c(Cl)cn(CC)n2)=O)CC2CC(NC(c3ncccc3OC)=O)CC2C1 C(=O)(CC(C)CCCCCCCC)NC(CCN(C(CCCOCC=C)=O)C)C c1(C(=O)NCC(N(C(C2ON=C(CC)C2)=O)C)C2CC2)ccc(=O)n2c1CCC2 C12(C(=O)NCC3C4CN(C(C=CSC)=O)CC43)CCCN(CCC1)C2 CCC(Cc1ccccc1)C(=O)N1CC(NC(c2cc(=O)cc[nH]2)=O)C(F)C1 c1(CN(C)C(C2(CCO)CNC2)=O)cc(F)ccc1F N1(C(C(C(=O)OCC)(C)C)=O)CCC2CN(C(C3(CO)CC3(C)C)=O)CC2C1 C1(NC(C(CC)COC)=O)CC2CC1CN(C(C1(C(F)F)CCOCC1)=O)C2 C1(CC(=O)NC2C(CSC)COC2)CN(C(=O)CN2CCCCC2=O)CCC1C c1(OC)nc(N2CCC(CNC(C3CCC(=O)N3)=O)C2)cc(C)n1 c1(C(N2C(C(=O)Nc3nnc(C)o3)CSCC2)=O)ccc(Br)cc1C(F)(F)F C(=O)(CC(C)(C)c1cccc(Br)c1)N(CCCNC(C1C(C)C1C)=O)C C1(CCNC(=O)C=CC(F)F)CCCN1C(=O)COC1CCOC1 N#Cc1ncc(C(=O)NCCN(C2CCCCCC2)C(c2ccoc2Cl)=O)s1 CC1(NC(c2ncsc2Br)=O)CCN(C(=O)Cn2cnc(C#N)n2)C1 c1(NC(CCC)Cc2nccn2C)nc2ccc(Br)c(C)n2n1 CC1CN(C(=O)C=Cc2ccc[nH]2)CCN1C(C1CC(=C2CCC2)C1)=O CCCCC(CC)CC(c1nnnn1-c1ccccc1CC)NC1(CCF)CC1 N=c1ccc(C(=O)NCC2CCC2NC(C2CCC2(F)F)=O)c[nH]1 c1(NC(=O)C(C)C(C)(C)C)nc2ccccc2s1.C1(=O)CCCN1C(C)C C1(NC(COc2cn(C)nc2)=O)CCC(C)(CNC(=O)C2=CCCCO2)CC1 c1(C(=O)NCC2(C(F)F)CCN(C(C34CC3C4)=O)C2)ccc2ccncc2c1 c1(CC(=O)NC2CC(NC(c3ccsc3Br)=O)C2)cnc2[nH]ccc2c1 C1(NC(C2(CC)CCCCO2)=O)CCN(C(=O)C=C(C)C)CCC1CO C1(C(N2CC3C(NC(=O)C(O)C4CCC4)(C3)C2)=O)CC2(CCCCC2)C1 C1(CCN(C(c2c(C)noc2)=O)C)CCCN(C(=O)CC2CCN(C(C)C)CC2)C1 c1(OC)ccncc1C(=O)NC1CC1NC(=O)CC(C)c1cccnc1 N1(C(C2(C)CCCC2)=O)CC2(CC(=O)NCc3cncc(F)c3)CC1C2 N1(C(C(C)CF)=O)CCC2(CC1)CN(C(=O)Cc1cccc(CC(F)(F)F)c1)C2 c1(CCC=C)n[nH]c(=NC(=O)c2cn(C)nc2OCC(F)(F)F)s1 c1(C(=O)NC(CNC(CC(C)CF)=O)(C)C2CCC2)cccc2ncccc12 C(=O)(CCCC(C)(C)C)NCC1CCN(C(c2n(C)nnc2)=O)CC1O C(CCCCC(C)C)NC(C1N(C(C2C(CSC)C2)=O)CC1)=O c1(C(N2CCC(NC(C(C)C(C)(C)C)=O)C(C)(C)C2)=O)nn2cccnc2c1Cl c1(N(C(c2cccs2)C)C)c2ccccc2nn1C C1(C(N2CCC(CC)C2)=O)(CC)CCN(C(c2csc(CO)n2)=O)C1 N1(C(C)C)CCCC1C(=O)NC(C(=O)NCc1cccnc1)C1CC1 c1(-c2c(C(=O)NCC3CN(C(CCC)=O)C(C)C3)cccn2)ccc(F)c(F)c1 c1(CC(=O)NCCN(C(C)C)C(C2CCC(C)O2)=O)cccc(Cl)c1Cl C12(C(N3CC(CCNC(CNS(NC)(=O)=O)=O)OCC3)=O)CCC(CC1)C(C)O2 CC(C)CC(C(=O)NC1CC(c2ncc[nH]2)C1)ONC(=O)C(C)N1CCCCC1 CN=c1[nH]c(=NCc2cc(Cl)cc(F)c2)[nH]c(=NC2CCC3C4CCC(C4)C23)[nH]1 c1(C(N2C(C)CCC(NC(CC(=O)NC)=O)C2)=O)cccc2c(C)c(C)[nH]c12 c1(CC)cc(NC(C2(NC(=O)C(C)C(O)CC)CCCC2)=O)cc(C)c1 C1(C(=O)NCC2(C)N(C(CN(C)C3CC3)=O)CCC2)CC(c2ccccc2)=NO1 C1(c2nnnn2Cc2ccc(OC)nc2)(NCC)CCCC(C(=O)OCC)C1 Cc1cc(C)n(CC(N2CC(CC(C)NC(c3cnn(CCO)c3C)=O)C2)=O)n1 CCC(CC(=O)N1CCCCC1c1cn(Cc2ccccn2)nn1)C(C)C N1(C(=O)Cc2ccc(Br)s2)CCC2(CCCN(Cc3c(Cl)cc(Cl)cc3Cl)C2)C1 c1(OC)cc(OC)cc(CN2CC3CC3(C(=O)NCCc3cccc(Br)c3)C2)c1 c1(OC)cc(C(=O)OCCCNC(=O)C(C23CCC(CC2)C3)O)ccc1OC Cc1cccc(C(=O)C(c2noc(Cc3ncc(-c4ccsc4)n3C)n2)C)c1 C1(CNC(C2(C)CC2)=O)CC(CNC(c2cnoc2C2CCOCC2)=O)CO1 C(C1=NOC(C)C1)NC(C1N(C(CCc2cc(C)[nH]n2)=O)CC1)=O.C=CC c1(C(=O)NCC2CC2NC(C2CCOCC2)=O)cccc(Cl)c1F c1(CC(N2CCC(O)C2c2ccccc2OC(F)(F)F)=O)cc(Cl)nc(Cl)c1 c1(CC)oc(C(=O)NCC2(F)CCC(NC(c3n[nH]cc3OC)=O)C2)cc1C N1(C(c2cncc3c[nH]nc23)=O)CCOC2(C1)CN(C(CC(F)F)=O)C2 S(=O)(=O)(c1ccc(NC(C)CCCCN)c(Cl)c1)NCc1c(C)ccnc1C c1(SC)ncc(C(N2CCCC(NC(=O)CC3CC4(CC4)CO3)C2C)=O)c(O)n1 c1(CN(C)C(=O)NCc2cccc(F)c2)ccccc1OC(C)(C)C C(=O)(CC(F)(F)CBr)NC(C)CC(C)NC(=O)CCC1OCCO1 c1(SCC)cccc(C2CC2C(=O)NC(C)CCNC(C2(CO)CCC2)=O)c1 Cc1ccc(-n2nc(Cc3ccccc3C)nc2CCc2cn(C)nn2)cc1Cl N1(C(CCNC(=O)OC)=O)CCC2(NC(=O)CCc3cccs3)CCCCCC12 N1(C(CC2CC(C)(C)CN2C(=O)CSc2cn[nH]c2)=O)C2CCCC1COC2 N1(C(c2ccc(OC)cc2C)=O)CC2CCC1CN2Cc1ccnn1CC(C)C C1(C(F)(F)F)(NC(N2C(c3ccc(C)nc3)CCC2)=O)CCCCCCC1 Cc1cnc(C(=O)NC(C)CNC(=O)C(C)n2cnnn2)cc1C#N C1(NC(CSc2cn(C)nc2)=O)CC2(C1)CC(NCc1cc(Br)co1)C2 Cc1ccc(O)c(CNC(=O)CC2CCC(C)(C)O2)c1 c1(C(N2CCCC(CNC(=O)C(=O)C3CC3)C2)=O)cc(Br)c(O)c(Br)c1 C1(C(=O)NCCC2(CNC(=O)C(c3ccc(F)cc3)(F)F)CC2)CCS(=O)(=O)C1 N1(C(c2nccc(CC)c2)=O)CCC2C(CCCN2C(=O)CC2CNC(=O)C2)C1 N1(C(c2c(CCC)nco2)=O)CCC(CC(=O)NCCC(C)C(C)(C)C)C1(C)C CC(CC(=O)N1CC(O)(CNC(C2(CF)COC2)=O)C1)c1cnn(C)c1 c1(C(=O)NC2CCCN(C(CCc3c(C)noc3C)=O)C2)ncc2n1CCCC2 C1(OC(c2nc(CCOC)[nH]n2)=O)CCCN(CSc2ccccc2)C1=O N1(C(CCN(S(C)(=O)=O)C)=O)CCCC(C2CCCCN2C(=O)Cn2ccnn2)C1 c1(N(CCS(N)(=O)=O)C)nc(N(C)Cc2cc(Br)cn2C)c2c(n1)CSC2 c1(OC)ccc(CN2CCSCC2C(=O)NCC2CNC(=O)CO2)c(Cl)c1OC Cc1nc(CNC(=O)NCC(C)(C)CCOC(F)(F)F)ccc1C(C)O C1(C)(CNC(c2cc(COC)on2)=O)CN(C(c2cc(Cl)cn2C)=O)CC1C N1(C(Cc2c(SC)cccc2)=O)CC(NC(c2cc(O)nc(Cl)c2)=O)CC(F)C1 c1(C(=O)NCC2CNC3(CCOCC3)CO2)cc(Cl)c2ccccc2c1 c1(C(N(C(C)CNC(c2c(Cl)cccc2Cl)=O)C)=O)cc(F)cc2ccncc12 C(=O)(CC(C(F)(F)F)c1nccn1C)NC(CC)CNC(=O)CCOCC(C)C C1(C(=O)NCC2N(C(C3=C(C)OCCC3)=O)C3C(C2)C3)CCOCC12CCCC2 Cc1ncccc1CN1CCOCC1C(=O)Nc1cnn(-c2cccc(Br)c2)c1 C1(NC(C(COC)C)=O)CN(C(C2(Cc3ccc(F)cc3)CCC2)=O)CC1O N1(C(C(=O)NCCC)CCCc2ccccc2)CCc2c(F)ccc(O)c2C1 Cc1cc(C(N2CCC(O)C2)=O)c(-c2ccc(C3CCCC3)cc2)cc1C C(=O)(C(C)C(CC)CC)NCC1CN(C(c2cc(CC)c(C)cc2)=O)C1 N1(C(COC)=O)CCC(CCC2CCCN2C(=O)Cc2ccsc2Cl)CC1 c1(CC)ccc(CC(C)C(N2CC3C(CNC(=O)CC4CSC4)C3C2)=O)cc1 C1(NC(=O)CCOCC(F)(F)F)CN(C(C2CCCNS2(=O)=O)=O)CC1C1CC1 c1(C(=O)NC2C(NC(CC3(CSC)CCC3)=O)CCC2)cccc(C2CC2)c1 N1(C(=O)Nc2cn(C)nc2-c2ccoc2)CCOC2COCCC12 C1(NC(C=C(C)C(F)F)=O)CCCC12CCN(c1nccnc1C#N)CC2 N1(C(C2C3(CC(NC(c4c[nH]c(=NC)s4)=O)C3)C2)=O)CCn2c(cnc2C)C1 N1(C(C(CC)C)=O)CC(OC)CC1CCNC(=O)COC1CCCC1 CC(C)C(C(=O)N(C)C)NS(=O)(=O)CC1(C(F)(F)F)CCC1 C(=O)(CCCCC(=O)N1CC2(COC(CNC(=O)CSCC(N)=O)C2)C1)NC N1(C(C2CC(C#N)(O)C2)=O)CCc2ccccc2C1CNC(C1CC=CCC1)=O N1(C(C(=O)NC2CCC(C(=O)O)CC2)=O)CCC2NCCCC2C1 C(C1CCCCCC1)=CC(=O)NCC(CC(C)C)NC(=O)COC(=O)CO c1(C(N(C)CC2CN(C(Cc3c(C)ccs3)=O)C2)=O)ccnc(OCCOC)c1 C1(C(=O)NCC(C#C)CC)CCN(C(=O)C2=CCCCC2)CC1C N1(C(C(C)OCC=C)=O)CCN(C(=O)C(C)(C)CF)CC1C1CCCC1 C1(C(=O)NCC(CNC(C(CCC)OC)=O)OC)Cc2cscc2C1 N1(N2CCC(C)C(CC=O)C2)CCC(C)(C#N)CC1.C(=O)CN(CCO)C1CC1 C(CC(CC)C(=O)N(C)CC1(NC(c2oc(C3CC3)nc2C)=O)CC1)=CC C1(CC(=O)NC(c2ccc(F)c(Cl)c2)C)(OC)CC2NCCC12 c1(C(N2CCN(C(=O)CO)C(c3ccccc3)C2)=O)[nH]c2ccccc2c1CO C(=O)(CCCCC(F)(F)F)NC(C)CCCCNC(C1CC2C(C1)C2(F)F)=O N1(C(C(=O)NC(C)CCCc2cccs2)=O)C(CO)CCC12CCC2 C1(NC(C=CCC(C)(C)NC(c2c[nH]nc2C2CC2)=O)=O)CC2CC1CC21CC1 Cc1c(C(=O)NCC2CC2NC(=O)C2=COCCO2)nc2sccn12 C1(NC(CN(CC)Cc2cscn2)=O)CCCCC1n1ccnc1 C(C(=O)NC(C)CCCCNC(c1[nH]nnc1C)=O)(C(F)(F)F)OC(C)=O C1(C(=O)NCc2occ(C(=O)OCC)n2)(NC(=O)C(C)O)CCC(F)(F)CC1 N1(C(C(=Cc2ccccc2)C)=O)CCN(C(=O)C2CC2)CC1c1cccs1 C1(O)(C(=O)NC(C2CC(C)(C(=O)OC)C2)=O)CCN(Cc2ncc(C(C)C)s2)C1 N1(C(COCCC)=O)CC2CC(NC(=O)C(C(C)C)c3ccncc3)C1C2 C1(c2n(C)cnc2)CN(C(C2CCCO2)=O)CC1NC(c1ccc(C2CC2)s1)=O Cc1ncnc(C)c1C(=O)NCc1ccoc1C(=O)NCCn1cccn1 c1(CNC(N(C2CCCC2)CCN(C)C)=O)ccoc1C1CC1 N1(C(CNC(CCC)=O)=O)CC2(CCC2)CC1C(=O)NC(c1ccc(C)cc1)C c1(C(=O)NCCCN(C(=O)COCC2CCCC2)C)c(N)sc2c1CCC2 C1(NC(C(C(C)OC)O)=O)CN(C(c2ccc(F)cc2F)=O)CC12CCC2 c1(N2CC(CC)SCC2)nc(NC2CC3CCCC23)nc2c1cnn2C c1(OC)cc(F)c(C(C(=O)O)NCc2cc(C)sc2C)cc1F Cn1cc(C(=O)NCC2(NC(C3C4CC4C4CC34)=O)CC2)c(O)nc1=O C1(NC(C(C)(C)CO)=O)CN(C(=O)CCn2cncn2)CC2CCCC12 C(CSC)(C(=O)N1CC(=C(F)CNC(=O)Cc2cc(C)cs2)C1)OC C1(NC(CCN(C)CC)=O)CCOC2(CCN(C(=O)CCCOC(C)C)CC2)C1 c1(C(N(CCCNC(c2n(CC)ccc2)=O)CC)=O)cc(C)c(F)cn1 c1(C(=O)NCCN(C(C2C(OC)CCC2)=O)C)cccc(NC(C)=O)n1 c1(C(=O)NCC2CCC(NC(c3c(C)cc(Br)o3)=O)C2)ccc2n[nH]cc2c1 C(=O)(C(=O)N1CC(C(C)NC(=O)CNC(=O)CNC(C)=O)C1)NCC c1(OC)c(Br)ccc(CNC2CCC(C(=O)Nc3ccc(C#N)c(Cl)c3)C2)c1F C1(NC(CCC(=C)Cl)=O)CCCC12CN(C(=O)C(C)OC)C2 C1(CNC(c2cnc[nH]2)=O)C2CCC(C2)N1C(=O)C=CC1CCCCC1 C1(CNC(C2C(COC)C2)=O)CCCC2CN(C(c3cc(F)n(C)n3)=O)CC12 O=[N+]([O-])c1cc(I)c(N2CCN(CC(CO)Oc3ccc(F)cc3)CC2)cc1F CN1C(=O)CSC1=CC(=O)NC1CC(C)(NC(C2CC3(C2)C(F)(F)C32CC2)=O)C1 CC(C)S(=O)(=O)CC(=O)N1CC(NC(=O)CCS(=O)(=O)N(C)C)CC(C)C1 C1(C(=O)NCCN(C(C(CC)NC(N)=O)=O)CCOC)CCCC1(C)C c1(C(N2CC(NC(C3C(=C)C3C(=O)OC)=O)C2)=O)ccc(F)c(C(F)F)c1 C1(C)(C(N2CCC(N(CCC)C(c3ncoc3COC)=O)C2)=O)CCC(=O)N1 c1(-c2cc(NC(=O)COC)cc(OC)c2)ccc(C(=O)O)c([N+](=O)[O-])c1 c1(C(N2CC(C3N(C(C(CC)SC)=O)CCC3)(O)C2)=O)cc(F)ccc1Cl C1(NC(=O)CCCNC(C2CCC2)=O)CN(C(c2ccsn2)=O)C2CC12 C1(C(=O)NCC2CCCN(C(C=COCC)=O)C2)Cc2ccc(F)cc2C1 C1(C(=O)NC(CN(C(c2c(C(C)C)ccs2)=O)C)C)CNc2ccnn2C1 c1(C(=O)NC2CC(F)(CNC(C(C)NC(=O)NC)=O)C2)nn(C)cc1[N+](=O)[O-] C1(C(=O)OC)CC(C)CN(C(c2cccc(-c3ccc(C(=O)O)cc3)c2)=O)C1 N1(C(c2n(C)ncc2)=O)CCC(C2CCCN(C(=O)C(O)c3ccsc3)C2)C1 CCC(O)CC(=O)NC1(C(N2CCN(C(C)=O)CC2)=O)CC1 C1(C(=O)NCCCO)CN(C(=O)CSc2ccccn2)CCO1 N1(CC(N2CC(N(C(C=Cc3n(C)cnc3)=O)C)C2)=O)CCCC2(CC2)S1(=O)=O c1(OCCC(=O)NC2CC(CCNC(=O)CC3CC=CCC3)C2)cccc(F)c1 C[Si](C)(C)CNC(=O)C(CC1CC1)NC(c1cnn(CCF)c1)=O C12(NC(CS(=O)(=O)N(C)C)=O)CCCC1CN(C(C1(F)CC3(CCC3)C1)=O)C2 CCC(C)C(O)CC(=O)N1CCC(C(=O)N(CCC(=O)NC)C)C1 N1(C(C=C(CC)C)=O)CC(C)(CNC(c2cc(C3CC3)ccn2)=O)CC1(C)C N1(C(c2cnn(CC)n2)=O)CCN(C(=O)C=Cc2cccc(F)c2)CCC1C c1(NCCN2C(C)COCC2)ccc(S(=O)(=O)NCCN2CC=CC2)cc1C#N c1(C(N2C(CNC(CC(CC)C)=O)CC2)=O)ccc(S(=O)(=O)N2CCCCCC2)o1 CCC(C)(C)C(C(=O)N1CCC(NC(c2cnc(C)n2C)=O)C1)OC c1(NC(COC)=O)ccc(C(=O)OC)c(Cl)c1.C12CCC(C)N(C1)C(=O)C(=O)N2 c1(C(=O)NC2C(CNC(C(C)OCC)=O)CC2)cnnc(C2CC2)c1 CCC(C(=O)N1CCC(NC(=O)CC2CC(F)C2)CC1C)C(C)O C#CCCCC(C)C(=O)NC(C(=O)NCC(C)(C)C1CC1)C(C)(C)O Cc1cc(N(CC(C)NC(c2cn(C3CCOC3)nn2)=O)C(N)=O)nc(Cl)n1 C1(C(N2CCC(CCN(C)C(C3CC(=O)NC3=O)=O)CC2)=O)C(F)(F)C12CCC2 c1(CS(=O)(=O)NC(c2cccc(OCOCC)c2)=O)cccc(OC)c1F Cn1nc(C(F)(F)F)c(CN2CCC3(CC3C(N3CCC(C)(C#N)C3)=O)C2)c1Cl C(=O)(CCC(c1nnnn1CCCSCC)NC(C)Cc1ccc(C)nc1)NC c1(C(N2CC(NC(C3(CCC)CCC3)=O)C(C)CC2)=O)oc2ccccc2c1Cl C1CC(=O)N1.C(C(CNC(=O)CCNC(C)=O)OC)N(CCC)C N1(C(C23CCC(C)(C2)CO3)=O)CCC(C2CC2NC(=O)C=Cc2ccoc2)CC1 N1(C(CCC(C)NC(CN(C(=O)OCC)C)=O)=O)CC2(CC(C)CO2)C1 C(=O)(OC)NCC=CCNC1CC1 c1(OC)cccc(Cl)c1CC(N1CC(NC(=O)C(C)(C)CN(C)C)CC(C)C1)=O C(C(=O)NCC1CN(C(=O)Cc2ccnn2C(C)C)CC1O)(C(C)(C)C)OC Cc1cc(COCC(=O)N(C)CC2CCN(C(=O)Cc3ccon3)C2)n(C)n1 C1(C(=O)NCC2(c3ccccc3F)CC2)CC2(C1)C(F)(F)C21CC1 C1(C)(CC)C=C(C(=O)N2CCC(O)(CCNC(=O)CCC(F)F)CC2)C1 c1(COC)ncc(C(=O)NC2CCCC2CNC(=O)CCc2ccn(C)n2)s1 N1(C(C2(c3cc(OC)oc3)CCC2)=O)CCN(C(C)=O)C(C2CCCC2)C1 N1(C(C(C(C)C)N(C)C)=O)CCC(O)(CCNC(=O)C=Cc2cn(C)nn2)CC1 c1(OC)ccnc(OC)c1C(=O)NC1CC2CC1N(C(=O)C=CC(C)=O)C2 C(=O)(CC(O)C(Cl)(Cl)Cl)NC(CC)CN(C(=O)C=Cc1ccc(C)nc1)C C12(C(=O)NCCN(C(c3c(OC(C)C)nccc3)=O)C)CCCN(C1)S(=O)(=O)C2 C1(NC(CSCC)=O)CC2(C1)CC(CNC(C1(C)CCCN1C)=O)C2 C(=O)(C(C)C(O)C(C)C)NC1C(CNC(c2cc(C)ncc2C)=O)COC1 c1(C(=O)NCCN(C(C2C(C)CCOC2)=O)C2CC2)ccc2c(c1)CN(C)CC2 c1(CNC(=O)OC(C)(C)C)ccc(Cl)c(F)c1Cl.N12CC(C13CCC3)CC(=O)NC2 N1(C(CCOCCC)=O)CCC(CCNC(C2CCC(c3cc[nH]n3)O2)=O)C1 c1(CCCNC(C(C)(C)NC(=O)Cn2cc(C3CCC3)nn2)=O)ccc(O)cc1 C(C(CC(=O)N1CC(OC)C(O)C1)N)NC(c1ccc(CO)o1)=O.COC N1(C(c2ccc(C#C)cn2)=O)CC(NC(C2CCCN2CCC)=O)CC(C)(C)C1 C1(NC(c2ccccn2)=O)CCN(C(C2CCC3(CC3)C2)=O)CC1 N1(C(Cc2nc(CC)sc2)=O)CCC(NC(c2n[nH]cc2Cl)=O)C1(C)C c1(N(CCNC(=O)NC(C)CCC2CCCC2)C)cccc2ccccc12 C(=O)(C1=CC2CCC(C1)C2)N1CC(C)(CNC(C(CSC)OC)=O)OCC1 c1(NCCNC(C(CC(C)C)NC(C)=O)=O)ncnc2c1nnn2C1CC1 CCC(C(=O)NCCC1CCN(C(=O)C(C)(C2(C)CC2)OC)CC1)C(F)(F)F n1(CCC(C)C)cc(C(N2CC(O)(CNC(=O)CCOCC3CCC3)C2)=O)nn1 CN1N=C(CC(=O)NC2CC3CC(NC(C4CCC(C)(C)OC4)=O)CC23)CC1=O C1(C(N(C)Cc2cn[nH]c2)=O)COCCN(C(=O)C2=CCSC2)C1 c1(C(N2CC(OC)(CNC(=O)Cn3nc(C)cc3C)C2)=O)cnc2c(c1)CCC2 Cc1cc(N2CCCC2C2CC(NC(C3(O)CCSCC3)=O)C2)nc(S(C)(=O)=O)n1 c1(N(C2CNCCC2(F)F)C(C2CC3(CCC3)CN2)=O)ncnc2c(Br)c[nH]c12 C1(C)(CC)C=C(C(=O)NCC(C)N(C(c2ccc(C(C)=O)c(C)c2)=O)CC)C1 CC(C)CC(CNC(=O)COC1CC1)NC(c1ccoc1)=O Cc1nn(CC(=O)NCc2cccc(CNC(C3CCCN3C)=O)c2)c(C)c1Br c1(CNC(c2cscn2)=O)cccc(C(=O)NC2CCC(F)CC2)n1 c1(C(=O)NC(c2coc(C(C)NC(CCC=C(C)C)C)n2)=O)csc(C)c1C n1(CC)nccc1C=CC(=O)NC(C)C(C(C)C)NC(=O)COC CC1(C#CC(=O)NC2CN(C(=O)C(O)c3ccsc3)C2)CCCO1 C(=O)(C1=CC2CCC(C1)C2)NCCC1CC(NC(CSc2n(C)ccn2)=O)C1 C1(C(=O)NC(C2CN(C(C=C(C)C(C)(C)C)=O)C2)C)CCC2(CC1)COCCO2 c1(C(=O)NC2CC3(CN(C(CC(=O)OCC)=O)C3)OC2)cnc2snc(C)c2c1 C(C(O)CC(=O)NCC1CC(NC(=O)C(c2cccc(Cl)c2)O)C1)N(C)C C=CCC(CC(F)F)C(=O)N1CCCC1Cc1cn(Cc2ccccc2)nn1 C1(C(N(CCOCC)C)=O)C2CCN(C(c3cc(OC)cnn3)=O)CC12 CC1(C(F)(F)F)CN(C(=O)CC2CNC3CC2C3)CC1C(=O)O N1(C(c2c(C)csn2)=O)CC(C(=O)NCC(c2ccncc2)C)C2(CC2)C1 CCC(CC(=O)NC(Cc1cn(-c2ccncc2)nn1)C(=O)OC)c1ccccc1 C(c1ccnc(Cl)c1)=CC(N1CC2C(CC(N3CCC(F)C3)=O)C2C1)=O CCC(C)(C)C(=O)Nc1ccsc1C(N1CCC1C(=O)NC)=O CC1C2CCC(C2)C1C(=O)NCCC(=O)NCC=Cc1ccc[nH]1 CC1CCC(Cl)=C(C(=O)NC2C=CCN(C(=O)CC3CCCCCO3)C2)C1 Cc1nc(C#N)c(NCCC(=O)N(C)CCN(C)C(C2CC2C(F)(F)F)=O)o1 c1(OC)cc(C(=O)NC2COCC2NC(=O)CCC(C)(F)F)ccc1C#N N1(C(=O)OC(C)(C)C)CC2(COC(CNC(C34CCCN3CCC4)=O)C2)C1 C(=O)(C1=CCS(=O)(=O)C1)NC(CN(C(C(c1ccccc1)OCC)=O)C)C c1(OC)ncc(C(=O)NCC(C2CCCN2C(C2CC2CN(C)C)=O)(C)C)s1 c1(C(N2C(C)CN(C(c3cnc(C#N)c(F)c3)=O)CC2)=O)cc(F)c(F)cc1Cl C1(CNC(C2C(CC)CCC2)=O)(NC(c2cccc(NC(C)=O)c2)=O)CCCCC1 N1(C(c2ccc(CC)cc2F)=O)CCCN(C(C2CC2C(F)F)=O)CCC1 n1(CC)cc(NC(=O)CC2CCCN2Cc2n[nH]cc2Cl)c(C)n1 N1(C(=O)CC2(C3CC3)CC2)CC2CN(C(C3CC4CCCCC34)=O)CC2C1 CON(C(=O)C12COC(CNC(C3CC(=O)C34CCC4)=O)(C1)C2)C(C)C c1(C(N(CC(CNC(c2cc(OC)ncc2)=O)(C)C)C)=O)cn(C)c(=O)cn1 c1(C(=O)NCC(CC=C)NC(C2CC(C(=O)OC)C2)=O)cc(C)ccc1Br c1(CNC(c2cccc3occc23)=O)cc([N+](=O)[O-])cc([N+](=O)[O-])c1 c1(C(=O)NCC2N(C(c3ncc(C)s3)=O)CCC2C)ccc2ccccc2c1 n1(CC(=O)NC2C(NC(c3c(C)oc(Cl)n3)=O)CCC2)ccc(=O)n(C)c1=O C1(O)(CNC(C(CC=CC)C)=O)CC2CCC(C1)N2C(C1(O)CCCCCC1)=O c1(CCC(=O)N(C2CCCC2)CCCOCC)ocnc1CNC(=O)CC1CCOC1 C1(CC(N2CCC(N(C(COCC)=O)C)C3(C2)CC3)=O)Cn2ccnc2NC1=O CCCC(O)CC(=O)NCC(C)N(C)C(C1CC(O)(C#N)C1)=O C(=O)(CC1=NNC(=O)C1)NC(CC)CN(C(=O)CCn1c(C)csc1=O)C N1(C(C2CC(OC)C2)=O)CCC(CO)(CNC(C2(C)CCCO2)=O)C1 C(=O)(C1=NOCC1)N1CCC(C(C(=O)NCCN(CCO)CC)F)C1 Cn1cc(CN2CC3CC2C3C(=O)NC(CCO)c2cccs2)c2ccccc12 C12(CNC(Cc3cccc(COC)c3)=O)CCC1CN(C(C1(C#N)CC1)=O)C2 C1(OC)CCC2(C(=O)NC3(CNC(=O)Cn4cnnc4)CCC3)CC12 C1(C(C(=O)OC)(C)C)CCN(C(=O)Nc2cccc(-c3cccnn3)c2)CC1 C(CNC(c1ncoc1C(C)C)=O)(C(C)(C)C)NC(C1C(CC(C)C)C1)=O Cc1cc2nc(NCC(C)(C3CC3)NC(C3CCCS3)=O)cc(=O)n2o1 O=S(=O)(c1ccc2ncsc2c1)N1CCN(c2ncnc3sccc23)C2CC12 n1(CC(=O)NCc2cn[nH]c2)ccc2ccc(-c3c(O)cccc3F)cc12 c1(OC)ccc(CN)cc1O.C1(C(=O)OC)(CO)CCCN1C(c1cc(C)c[nH]1)=O N1(C(COCC)=O)CCCC(C2CCCN(C(C)C(=O)NCc3ccco3)C2)C1 N1(C(c2n(C)cc(C(N)=O)c2)=O)CC(NC(=O)CCC(F)(F)F)C2(CCC2)C1 c1(C(=O)NC(CNC(c2cccc(N)c2)=O)CO)cc(F)cc(F)c1 C1(CN(C(C(=O)NCCC(=C)C)=O)C2CCC2)CN(C)CCO1 C1(C(=O)NC(C2(O)CN(C(=O)Cc3cnc[nH]3)C2)C)CCC2(CCC2)C1 C1(N(C(C(CC)O)=O)CCO)CCCN(C(c2oc(C(F)F)cc2C)=O)C1 c1(CC)ccc(CCN(C(c2cc(C)on2)C(=O)NC2(C)CC2)C2CC2)cc1 O=C(CCCCCn1cc(CC2C3CCCCCCC23)nn1)N1CCOCC1 CC1CCN(C(C2C3(CC3)C23CC3)=O)CC1NC(=O)CCC(N)=O c1(C(N2CCOC(c3n[nH]c(-c4ccccc4)n3)C2)C(=O)NC)ncc(Br)cc1C C=CC(C)(CCOC)C(=O)N1CCC(CNC(C2(N3CCCC3)CC2)=O)C(C)C1 C1(NC(=O)CCc2cscn2)CCN(C(C2CCOCC2)=O)C12CCCC2 Cc1ccc(Cl)c(N)c1C(N1CC2CCCN(C(C3CCCS3)=O)C2C1)=O N1(C(CNc2cn(C)nc2)=O)CCCC(CCNC(=O)CC2(C(=C)F)CC2)C1 c1(C(N2C(CNC(c3c(C)nsc3)=O)C=CC2)=O)nc2ccccc2[nH]1 Cc1ccc(S(=O)(=O)N(C(=O)CN2CC34CCCCC3(CNC4)C2)C)cc1 N1(C(c2cc(OC)no2)=O)CCC(CC(C)NC(C23CSCC2C3)=O)CC1 C1(F)(CNC(C2C(CC)C2)=O)CN(C(C2CCN2S(C)(=O)=O)=O)C1 c1(CN(C2CCN(C)CC2)Cc2c(C)nn[nH]2)cccc(Cl)c1 C(C(C)(O)C(C)(C)C)NC(C1(C#C)CN(C(=O)C2=NOC(C)C2)C1)=O C1(C(=O)NC(CNC(CCCC#C)=O)C(C)C)CC2C(C1)C2(C)C Cc1cccc2c1CC(C(=O)Nc1cc(F)cc(F)c1CO)N2 C1(CC(N2CCC(CCNC(C3C(C(C)C)C3)=O)C2)=O)CCN(C)CC1 C1(NC(c2cccn2C2CCCC2)=O)CN(C(=O)Cc2ncccc2F)CC1F C#Cc1cccc(CNC(=O)NC(CN2CCCC2)CC)c1F N1(C(CNC(=O)C2CC2)=O)CCC2(CCN(C(C3CCCCNC3=O)=O)CC2)C1 C1(NC(c2ccc(CC)[nH]2)=O)CCCN(C(=O)C(C)Cc2ccccc2)C1 C(=O)(CCCCN=[N+]=[N-])N1C(C(=O)NCCCCC=C)CC(O)C1 Cc1ncc(CC(=O)NC2(CCCNC(C3COC(=O)N3)=O)CC2)[nH]1 c1(CNC(=O)CC(C)COC(C)=O)cncc(F)c1C.C12(CC)CCCN1C2=O C1(CNC(c2cc(Cl)cs2)=O)CN(C(C23CCCC2C3)=O)CCO1 c1(C(=O)NC2CN(C(C=CC)=O)C2)c[nH]c2ccc(OC(F)F)cc2c1=O c1(C(N2CCN(C(CNC(C)=O)C(F)(F)F)CC2)=O)cc(N)c(F)cc1F N1(C(c2cc(C(C)(C)C)on2)=O)CCC(CNC(=O)Cn2cc(CO)nn2)C12CC2 N1(C(C2OCCC(C)C2)=O)CC2(CC2)CC1C(=O)NC1CC1CN(C)C c1(C(=O)NC(CC)CN(C)C(c2cnsc2C)=O)cc(Cl)cn1C C(=O)(CCN(C(=O)CSCCC#N)CC1CC1)NCC(C)OC C1(O)(CNC(c2cc(C)sc2C)=O)CCCN(C(c2ccc(C(F)(F)F)s2)=O)C1 c1(CNC2CC(C(=O)NC3CCS(=O)(=O)C3)CC2O)ccc(Cl)c(F)c1F CCCCCC(F)C(=O)NCCOCC(=O)N(C)Cc1cnn(CC)c1 CC(CN=C(NCc1ncccc1N(C)C)NCC1CCOC1)C(F)F c1(C(N2CCC(N(C(c3c(N)nccn3)=O)CCO)C2)=O)cc2n(n1)CCCC2 Cc1nn(C)cc1CCC(=O)NCC(C(C)C)NC(C1CC1(C)C(F)(F)F)=O c1(C(=O)NCc2cc(C(=O)NC(CC)C)n[nH]2)ccccc1NC(=O)C(C)(C)C C1(C(N2CC(C)C(CNC(=O)C(C#N)C3CC3)C2)=O)C2C3CC4C1C1C2CC3C41 C(=O)(C(O)(CN(C)C)C(F)(F)F)N1CC(CNC(c2c(OC)scc2)=O)C1 N1(C(C(CC)NC(N)=O)=O)CCN(CC2(NC(=O)C(CC)SC)CC2)CC1 C=CC(C)(CC)C(=O)NOCC(=O)NC(C)CC C12CCN(CC1(C)C)C2=O.c1(CN2CCC(COC)C2)cc(F)c(Cl)c(Cl)c1 C(=O)(C(C)(C)N=[N+]=[N-])N1CCN(CC(N2C(CSC)CC2)=O)CC1 C(CC(C)CC)(C(=O)NC(c1nccc(O)n1)C)NC(C1CC(CCC)C1)=O N1(C(CCOC)=O)CC(C(=O)NCc2ccnc(C(N)=O)c2)CC1(C)C C1(C(=O)NC(CC)C(N)=O)CN(C(c2ccc(O)cc2)=O)CC1F C#CC1CN(C(c2nccn2C)=O)CCN1C(c1cscc1C)=O Cc1c(CN=c2[nH]c(N3CC(CO)CC(C)C3)nc(=N)[nH]2)[nH]c2ccccc12 C(=O)(C(C)(C)C(C)C)NCC(C1CC1)NC(C1CN(CC(C)C)C(=O)C1)=O C1(C(=O)NC(C)C=CC(=O)NCC(=O)N(C)O)CCCC(=O)CC1 CC(C(C)(C)NC(c1cnn(CCO)c1)=O)NC(=O)CCOC1CCOC1 C1(NC(c2c(-c3c(CC)scc3)ncs2)=O)CC=C(C)CC1 c1(SCC(=O)N(C2CCN(C(C3(C#C)CC3)=O)C2)CCC)ccc(F)cc1O CCCC(C)(CC)C(=O)N(C(CNC(=O)COC(F)F)CC)CC Cc1ccn2c(C(=O)NCC3CN(C(c4ccnc(O)c4)=O)CCO3)cnc2c1 c1(C(C(=O)NCCC(C)N(C(C2CC(C(=O)OC)C2)=O)C)OC)ccncc1 N1(C(C(C)(C)CF)=O)CCC2C(CCCN2C(c2cc[nH]c(=N)c2N)=O)C1 C1(C)(CC)CC(C(=O)NCC(C2CCCN2C(=O)CN(C)C)(C)C)C1 C(=O)(C(=O)CCC(C)C)NCCOC1CN(C(C(c2c(C)nn(C)c2C)C)=O)C1 n12nc(CS(C)(=O)=O)nc1CC2.N1(CCOC)CCCCC1 c1(C(=O)OC)cccn(CC(N2CCC(SCC(C)N(C)C(C)=O)CC2)=O)c1=O N1(C(C=Cc2n(C)cnc2)=O)CCC(C)(C)C1C(=O)NC1CC2CCCC2C1 C1(NC(CCC=C(C)C)=O)CCCCCC1NC(=O)CC1CC2CC2C1 C1(C(=O)NCC(N2CCN(C(C(C(C)C)C)=O)CC2)=O)CCN(C)S1(=O)=O C1(NC(c2nn(C)c(OC(F)F)c2)=O)CCN(C(c2cc(F)n[nH]2)=O)CC(C)(C)C1 Cc1ccc(O)c(C(N2CCC(CNC(=O)CCC3(C)CC3)C2(C)C)=O)c1 C1(NC(c2c(CC)c[nH]c2)=O)CC2CCC(C1)N2C(C1CCC(=O)N1C)=O C1(C(N2CCC(C)(NC(C3CCC(C)(C)C3)=O)C2)=O)(COC)CCCCC1 C#Cc1cc(C(=O)NC2CCN(C(=O)CN3CCCC(N(C)C)C3)C2)cc(F)c1 Cn1c(=O)ccn(CC(=O)NC2C=CCN(C(C3CCNC3=O)=O)C2)c1=O C1(CCCNC(C2(C)CC2(F)Cl)=O)CCN(C(C2(NC(C)C)CC2)=O)CC1 C(=O)(CCCCCNC(C)=O)N(C(CN(C(c1ccc(COC)s1)=O)C)C)C N1(C(CN(C)C)=O)CCC1CNC(C1CCS1)=O c1(CC)c(C(=O)NC2(C3CCCN3C(=O)CC(C)(C)OC)CC2)cccc1C C1(CC(N2CCC(CO)C2)=O)CCCCN1C(=O)Cc1ccsc1.C(CS)O c1(C(C(=O)N(CCN(C(C)C)C(C2CC2C#N)=O)C)(F)F)c(F)cccc1F N1(C(C2C(=C)C2)=O)CCCCC(C2CN(C(=O)C(O)C(C)CC)C2)C1 c12ccc3c(c1)CN(CC3)C2.C=CCS(=O)(=O)NC(=O)C(C)(F)F c1(OC)cccc(C(C)(C)C(=O)N(CC(C)CNC(c2ncccc2F)=O)C)c1 C1(CC(=O)NCCC(C)NC(c2cn3c(n2)SCC3)=O)CC2C=CC1CC2 C(=O)(C1CCCc2ccnn21)NC1C(NC(C(C(C(C)C)O)C)=O)CS(=O)(=O)C1 C1(C(=O)NCC(CCOC)NC(=O)C=CCN2CCOCC2)CC2(CCCO2)C1 C1(C(=O)NCCC(C)NC(C(CC)NC(C)=O)=O)CCC2(CC2)C1 N(C1CCCc2ccc(Cl)cc21)Cc1n(CCc2c(O)cccc2)nnn1 S(=O)(=O)(c1cc(C(=O)OC)co1)N1C(COC)CC(O)C1 C1(NC(c2c(C)ccc(C)c2)=O)CCN(C(C2CCC2)=O)CC(C)(C)C1 CCCC(O)C(=O)NC1CN(C(=O)CN2CCOCC2)CC1C(F)F c1(NCC(CNC(C2CCC(C(C)C)CC2)=O)C)ncc([N+](=O)[O-])cc1Cl CC1(NC(c2ccnc(-c3ccco3)c2)=O)CC2CCC1CC2=O C1(C(=O)NCCN(C(=O)CSC)CCC)CCOCC12CCCCC2 N1(C(c2cnc(CNC(C(C)N(C)C)=O)o2)=O)CC2C(C)C2C1 CN=c1nc(C(=O)NCCCCNC(=O)C(c2cncn2C)O)cc(C)[nH]1 C1(CNC(C(CSC)OC)=O)(CNC(C2(C(C)C)CCOCC2)=O)CC12CCC2 c1(N)cc(=NCC2CC2)[nH]cn1.c1(OC)ccc(CCCN(C)CCF)cc1N N1(C(C(CC)Sc2ncccn2)=O)CC(S(=O)(=O)NC(C)(C)C)C1 c1(C(=O)NC2CCN(C(CC(C)OC)=O)C2C(C)C)ccc(Br)c(F)c1C C#CCCCC(C)C(=O)NCc1cc(C(=O)N(C(C)CC)C)n(C)n1 c1(C(N(C2CCCN(C(C3(C(F)(F)F)CCC3)=O)C2)C)=O)nnn2ccccc12 C1(NC(c2cnc3cc(C)nn3c2)=O)C2Cc3cc(F)ccc3C12 C(=O)(C(C)(C)C(N)=O)NC1CCN(CCCNC(C(c2ccccc2)C)=O)C1 c1(SCCNC(c2c(C)[nH]c(=NCC)s2)=O)cnc(O)c(C(C)=NO)c1 N1(C(CC2(CC)CCC2)=O)CCC2CN(C(=O)C(C(=O)OC(C)(C)C)OC)C2C1 CCC(C(C)C)C(C(=O)Nc1cccc(OC)c1)N1CCSC(C)C1 C(CC(CNC(C1CCS1(=O)=O)=O)NC(c1ccc(N)s1)=O)OC.C(C)(=O)N C12(O)CCN(C1)C(=O)CS2.c1(C(N(C)CC2CC2)=O)ccc(-c2ccccc2)s1 Cc1[nH]c(=N)ccc1C=CC(N1CCC1CNC(c1cc2c([nH]1)CCCC2)=O)=O N1(C(C2(COC)CCC2)=O)CC2(CCCC(CNC(C3(F)CC=CCC3)=O)O2)C1 C=C=CC1CCCCN1C(=O)C(CC(=C)C)OC CCCCC(F)C(=O)NCCCC(O)C(=O)NCC1CC2(CCC2)CO1 C(C(C)C(=O)NNc1ccc2[nH]ncc2c1)c1c(C)ccc(OC)c1 c1(OCc2scc(C(=O)NC(C)CCCNC(=O)C(N)=O)n2)cccc(F)c1 c1(NCC2CN(C(C(CCC)CCC)=O)CC23CC3)ccc([N+](=O)[O-])c(OC)c1 S(=O)(=O)(c1cn2c(n1)CCC2)N1CCC(F)(C(=O)OC)CC1 Cc1ccc(-c2nnco2)cc1C(=O)NCc1cc(C(=O)O)co1 Cc1cc2c[nH]nc2cc1C(=O)NC1CCCCCC1NC(=O)C(=O)NC1CC1 N1(C(c2ccc(-c3scc(C)n3)cc2)=O)CC2CC(NC(C3CCOC3)=O)C2C1 C1(C)(C(N2C(CNC(C3N(C(C)C)C(=O)CC3)=O)CCCC2)=O)CCN(C)CC1 c1(CNC(C2C(C)(C)C2)=O)nc2c(s1)CCN(C(C1CC3C=CC1C31CC1)=O)C2 Cc1cncc(C(N2CC=CC2(C)C(=O)NCC[Si](C)(C)C)=O)n1 N1(C(C(CCSC)O)=O)CC2CCCC(NC(C3CCC(C)C(C)C3)=O)C2C1 N1(C(c2c(CC)cccc2F)=O)CC(NC(=O)CC2CSCCS2)C(N=[N+]=[N-])C1 N1(C(c2[nH]cc(CC(C)C)c2)=O)CC2C(CNC(c3cnoc3C3CC3)=O)C2C1 CC1CCC(C(=O)NCC2CCCC2NC(=O)CCc2ncc(C(C)(C)C)o2)O1 N(C1CCC(NC(=O)CCCC2CCC2)c2ccccc21)C(=O)CCC1CCC1 c1(C(=O)NCC(Cn2cc(-c3cccc(O)c3)nn2)OC)cc(Cl)c(Cl)cn1 N1(C(Cc2ccc(C)o2)=O)CCC(C)N(C(c2cc3cscc3s2)=O)CC1 CCC(C)(CNC(c1csc(C#N)c1)=O)C(=O)NCC(=O)NC1CC1 C1(NC(c2c(C)ccs2)=O)CN(C(=O)Cc2ccc3nc[nH]c3c2)CC1C1CC1 c1(C(=O)NC(c2cccnc2)CC)ccc(CNC(=O)CC2CCCC2)cc1 C1(NC(c2c(CC)nsc2)=O)CCOC(C(=O)NCCCn2cnnc2C)C1 C12(C(=O)NC3C(C)CN(C(C4CCCCC4)=O)C3)CC3CC(C1)CC(O)(C3)C2 O(N(C)C(=O)CN=C(NCC1CC1)N1CCC(CC2CC2)C1)CC c1(C(N2CCC(CNC(C(CCC)OC)=O)CC2)=O)nnc(O)c(Br)c1O CCC(COC)C(=O)N1CCC(F)(CNC(=O)CCc2ccnc(Cl)c2)C1 C(C(CN=c1[nH]cc([N+](=O)[O-])c(=N)[nH]1)C(F)(F)F)NC(C1N(C)C(=O)CC1)=O C1(C(=O)NCCNC(C2C(C)C2)=O)CCCN(C(=O)CC2COC(=O)N2)C1 C12(C(=O)NC(C=CC(=O)NCCC(C)OC)C)CC(C#N)(C1)C2 NS(=O)(=O)c1ccc(C(=O)NC2CCN(C(=O)CC34CCC(CC3)C4)C2)[nH]1 c1(OC)cc(N)c(C(=O)NCC2CCCCN2C(C2CC3CC2C3)=O)cc1F c1(C(=O)NCC(CNC(Cc2cccc(SCC)c2)=O)O)cccc(F)c1O c1(C(N2CC3(F)C(NC(C=CC)=O)(CCC3)C2)=O)ccc2c(c1)C(=O)N(C)C2=O C(=O)(C1CCc2nccn21)NC1CCCCCN(C(C(CC)(CC)CO)=O)C1 C1(NC(=NCC)NCC(c2ccc(F)cc2)(F)F)CC1C1CCCC1 C(=O)(CC(C)CC(=O)N1CCN(C(c2[nH]cc(C)c2C)=O)CC1C(F)F)OC C#Cc1ccccc1CC(N1CCC(C)(CCNC(=O)C(N)=O)C1)=O c1(C(=O)NC2CN(C(=O)CCc3ccco3)CCC2CO)nnn2c1CCC2 c1(OC)cc(C(=O)NCC2CCC(NC(c3cc(C(F)F)n(C)n3)=O)C2)ncn1 C1(NC(CC2N(C)CC=CC2)=O)CCCCCC1NC(c1ccc(Cl)cc1)=O c1(C(=O)NCC(C2CCCC2)NC(c2c(C)ocn2)=O)c(F)ccc2c1OCC2 CC1(C)CCCN(C(c2ccc(C#N)cn2)=O)C1C(=O)NCC1C=CCCC1 Cc1ccc(C)c(C(c2nnnn2C(C)C)NCCC2(C(F)F)CC2)c1 Cc1nc(N(C)C)sc1-c1ccc(C(=O)NOCC)cn1.N1CCOC(CC)C1 c1(C(=O)NC2CN(C(c3cccc(NC)n3)=O)CC2O)ccc(C)c([N+](=O)[O-])c1 c1(C(=O)NC(C)C(C)(C)C(=O)N(CCN=[N+]=[N-])C)cc2cccnc2[nH]1 C1(CC)CCN(C(=O)Cc2cnns2)C(CNC(=O)CCC2CC2(C)C)C1 N1(C(CC2(C)N(C(c3c(C)c(F)ccc3)=O)CC2)=O)CCC2(CCCO2)C1 C1(NC(C2N(C(C)=O)CC2)=O)COC2C(NC(c3cccc(CC)n3)=O)COC12 c1(C(=O)NCCCN(C(CNC(C)=O)=O)C2CC2)cscc1C#N Cc1nn(C)cc1CNC(CCN(C)C(c1ccc(OC(F)(F)F)cc1)=O)=O C1(=CCNC(c2c(OC)c[nH]n2)=O)CCN(C(C2CCOC2C)=O)CC1 Cc1cc(C(=O)NCC(O)CNC(=O)C=CSc2nc[nH]n2)cnc1OC(F)F c1(CNC(c2n[nH]c(C)c2O)=O)cnn2c1CN(CCS(C)(=O)=O)CC2 c1(CC)cc2c(N3CCC(C4(NC(=O)C(CSC)OC)CC4)C3)nc(C)nc2s1 C1(CS(=O)(=O)NC(C(c2ccc(OCC(=O)OC)cc2)(C)C)=O)CCC12CCCO2 CC1(C)CC(C(N2CCCC(CO)CC2)=O)CCN1C(=O)Cc1cccnc1 C1(C(=O)NCCN(C(=O)C(C)Oc2ccccn2)CC)CCCN2CCCC12 C#CCC(C(=O)OC)NC(=O)CCCCNC(=O)CCn1cnc(=N)[nH]1 c1(C(N2CC3CC3(NC(C3(Br)CC3(F)F)=O)C2)=O)ccc2[nH]ccc2c1 c1(C(=O)NC2CC(NC(CCc3scc(C)n3)=O)CC2O)cc(C)c(C)c(C)c1 c1(C(=O)NCCn2cc(C(C)(C)S(C)(=O)=O)nn2)sc2c(Br)cccc2c1N C1(NC(c2ccc(C#N)o2)=O)CN(C(c2coc(Br)c2)=O)CC2CC12 C12(NC(CCCc3onc(CC)n3)=O)CCN(C(c3c[nH]nc3C)=O)CC1C2 c1(C(=O)NC2C(OC)CN(C(c3ccc(=O)oc3)=O)C2)c(F)cc(Cl)cc1Cl C12(C(N3CC(C)N(C(=O)C(CO)N(C)C)CC3)=O)C3C4C1C1C2C3C41C(N)=O c1(C(=O)NC2CC(CN)C2)cnn2c1S(=O)(=O)NCC2 C1(C(=O)NC2CC3CC2N(C(=O)C2=CCOCC2)C3)CC2CCCN2C(=O)N1 C(C(CNC(c1c(OC)noc1C)=O)S(C)(=O)=O)NC(c1ccc(OC)cc1)=O N1(C(c2c(C)coc2C2CC2)=O)CC2(C1)CN(C(=O)CCNC(N)=O)CCO2 C(=O)(N=c1cc(C)n(CCO)[nH]1)NC1CC(CC(=O)NCc2ncc(C)o2)C1 C12(C(N3C4CC(CC(C(N5CCCCC5)=O)C4)C3)=O)CCCC1CS(=O)(=O)C2 C1(NC(c2ccc(C#C)o2)=O)CC2CC1N(C(c1c(Cl)cnn1C(C)C)=O)C2 c1(C(=O)Nc2c(Br)ccc(OC)c2)cc2c(s1)CCN(S(=O)(=O)C(F)(F)F)C2 C1(OCC)CCN(C(c2nc(CCNC(CCC(C)OCC)=O)oc2)=O)CC1O C1(CNC(C2=CCN(C)C2)=O)N(C(C2CC(=O)N(O)C2)=O)CCCC1(C)C c1(C(=O)NC2C(NC(C(N3C(=O)CCC3=O)C)=O)CC2)c(N)sc2c1CCC2 C(=O)(C1OC(=O)c2ccccc21)NCC1CC(NC(c2ccncc2)=O)C(O)C1 C1(O)(CC(=O)NCC2C(C)CCN2C(c2cc(C(N)=O)[nH]n2)=O)COC(C)(C)C1 N1(C(C(C(C)(C)C)OC)=O)CCN(C(c2csc(C)c2C)=O)CC(C)C1 N1(C(C(=O)NC2CC23CC3(F)F)=O)CCC(C2CCOCC2)C1 CC1(C)COC(C)(C(=O)NC2CCN(C(=O)C=C3CCCCC3)CC2F)CO1 C(C)(C(CC(=O)N1CCSCC1)NC(C1(C)CC1C)=O)OC C1(CN(C)C)C(=O)N(OC)CCC(=O)N1.C#CCC(O)C(=O)OC C1(NC(c2nnc(O)nc2O)=O)CCCCN(C(c2cn[nH]c2)=O)C1 C#CC1(C(=O)NC(CO)CCC=C)CCN(C(c2nc(C)sc2C)=O)C1 c1(C(N2CC(OCCNC(CC3CCN(C)C3)=O)C2)=O)ccn2[nH]c(=N)nc2c1 c1(C(N2CCC(C)C(NC(=O)CC=CC(C)(C)C)C2)=O)cc2c(s1)CCC2=O c1(C(N2C3CN(Cc4cc(C(=O)O)c(Br)nc4)CC32)=O)ccc2c(c1)C(=O)OC2 N1(c2n(CCCOC)c(-c3ncnn3C)nn2)CCOC(C)(C(F)(F)F)C1 C(=O)(CS(=O)(=O)c1ccccc1Cl)N(C)CC1N(C(C(CC)F)=O)CC(F)C1 c1(C(=O)NCC2(O)CC(NC(c3n(CC)nnc3)=O)C2)cc(Cl)ccc1F c1(C(=O)NCC(=C)CCNC(C2COC(C)C2)=O)cc(Cl)cc(Cl)c1Cl N1(C(Cc2c(C)occ2)=O)CCC(NC(C23CC(CN2C2CC2)C3)=O)CC1C C(=O)(N=c1cc(C(F)(F)F)[nH][nH]1)c1cccc(NCc2ccc(C)c(C)n2)n1 N1(C(C2C(C)(C)CC2)=O)CCC(C)(CNC(=O)C(C)(C)C2CCCC2)C1 CN1CCN(C(c2ccsc2Cl)=O)CC1C(=O)NC1(CO)CC1 C1(OCSCC)CC2(CCC(C(N3CCN(S(=O)(=O)C4CC4)CC3)=O)CC2)C1 C1(CCCNC(c2coc(C3CC3)n2)=O)CCCN(c2cc(O)ncn2)C1 C(C(C)(F)C(C)(C)F)n1cc(N2CCCC(NCc3n(C)c(O)nn3)C2=O)nn1 c1(C(=O)NCC2CC(C)N(C(C3CCCS(=O)(=O)C3)=O)C2)nc(=O)cc(N)[nH]1 c1(OC)ccc(C)c(C(=O)NCCNC(=O)CN(C)C(=O)C(C)C)c1N c1(C(=O)NC(C2(O)CN(C(c3nc(C(C)OC)sc3)=O)C2)C)ccccc1Cl C12CN(CC13CC3)C2.C1(CC(=O)OCCOCCC)(SCC)CC1 S(=O)(=O)(c1ccc(Cl)c2cnccc12)N1C(CC(=O)OC)COC(C(F)(F)F)C1 CC1(NC(c2cnc(O)c(C(F)(F)F)c2)=O)CCN(C(c2cncs2)=O)CC1 N12CCOC(C1)C2=O.c1(CCC)nc(C(=O)NCCC(C)=CCC)co1 N1(CC)CCCCC1C(N1CC(C(=O)NCC(C)(C)NC(=O)COC(C)C)C1)=O N1(C(C(CC2CCC2)OC)=O)C2CCCC1CC(N=c1ccnc(CO)[nH]1)C2 N1(C(C2CN(C(=O)NC)C2)=O)C(=O)NC(c2cncn2C)C2=C1C(C)N(C)C2=O Cc1ccc(C=CC(N2CCC(CNC(C3CCCCO3)=O)C2(C)C)=O)cn1 c1(C(C)C(N2CCC(NC(=O)CN(C)CCO)C2)=O)ccc(F)cc1F c1(C(=O)Nc2c(OC)ncc(C3CC3)c2)cc2ccc(Br)cc2s1 CCC(CC(F)F)C(=O)NCC#CCNC(=O)CCc1ccccc1Br Cn1nc(CNC(C2C=CCC2)=O)c2c1CCN(C(C1(C#N)CCCCC1)=O)C2 C1(CC(=O)N(C)CCn2cc(CCCCS(C)(=O)=O)nn2)CCC2(CCC2)O1 c1(C(N2CCC(C(=O)Nc3c(C)cc(C(=O)OC)[nH]3)C2)=O)cc(Cl)c(Cl)nc1Cl C1(NC(c2n[nH]c3c2CCSC3)=O)CC2CC(C1)N(C(C1CCCCO1)=O)C2 CC1CCCC(C(=O)NCC2CN(C(c3cccc(F)c3)=O)C2)CC1 CC1CN(C(c2nccnc2Cl)=O)CCC1CNC(c1c(Cl)cnn1C)=O C1(NC(c2nc(CCC)oc2)=O)CC2CCC(C1F)N2C(C1CC(C)(O)C1)=O CC(C)CC(C(=O)NC(CN=[N+]=[N-])C(=O)NCC1CC12CC2(F)F)C(C)C c1(C(=O)NC2CN(C(C(C(C)C)(C)O)=O)CC2O)noc2c1CC(C)(C)CC2 N1(C(=O)CCC2CCCC2)CC2C(NC(=O)C(F)(F)c3cccnc3)C2C1 c1(OC(C(=O)N(C)CCNC(c2coc(C(F)F)n2)=O)(C)C)ccc(F)cc1 c1(C(C(N2CCC(NC(CC3(C)CC3)=O)(CF)C2)=O)(F)F)c(F)cccc1F n1(CC(=O)NCCCNC(=O)CC2CCCCC2F)c(=O)cnc2ccccc12 C12(CC(=O)NC(C(=O)NC)(C)C)CCC1CN(C(C1CC(C(N)=O)C1)=O)C2 Cc1ccsc1C=CC(=O)NCC(F)CNC(=O)CCNc1nnnn1C N1(C(C2CC(NC(c3cnn(CCO)c3)=O)C(O)C2)=O)CCOCC1CO N1(C(C2(CC)CCC(O)CC2)=O)CCN(C(=O)COC2(C)CCC2)CC(C)(C)C1 c1(C(N(C2CCN(C(C(C)CN(C)C)=O)C2)C)=O)ccc2c(c1)N(C)CC2 c1(OC)ccc(C(c2nnnn2C(C)C)NC2CS(=O)(=O)CC2OC)cc1Br CCC(C)(CNC(c1sccc1C)=O)C(=O)N(CC(C)COC)C C(=O)(CC(C)(C)N(C)C(C1CCNC(=O)C1)=O)NC(C)C(=O)N(C)C CCCCC(CCCC)C(=O)NCCC(C)NC(C1C=CC1C(=O)OC)=O n1(CC)cccc1C(=O)N(CC(=O)NCC1CC12CC2)C C(CCCC(=O)NCC(=Cc1cnc[nH]1)NC(c1ccc(C)cc1)=O)(OC)OC c1(OCC)cccnc1C(=O)NCC1CCCN(C(C2(O)CCOC2)=O)C1 c1(OCC(=O)NC(CNC(C(C)=C2CCCC2)=O)CC(C)C)c(F)cccc1F CCCCCC(O)CC(=O)NC(C)C(C)C(=O)N1CC2(CSC2)C1 N1(C(c2cccc(N)c2N)=O)CCC2(CCN(C(c3cccc(O)n3)=O)CC2)C1 c1(C(=O)NC(C(=O)NC2C(OC)CC2)CCF)cc2cccnn2c1 N1(C(Cc2scc(C)n2)=O)CCCC2(CCN(C(c3cn[nH]c3)=O)C2)C1 C1(NC(=O)NCC2(C(=O)OC)CC2)CN(C(=O)CC2(O)CCCC2)CC(C)(C)C1 C1(COC(C2CC(C)OC2=O)=O)CCS(=O)(=O)C(C)C1 C(=O)(C1Cc2c(Cl)cccc21)NCC1C(C)CN(C(=O)CCOCC2CC2)CC1 C1(NC(C(CC=C)(C)C)=O)CCC2CN(C(=O)C(C)NC(=O)COC)CC12 c1(C(=O)NCC(CC)NC(=O)C(C(C)C)c2cnc(C)s2)ccc(C2CC2)cn1 CC(CC(=O)NC(C(N1CCC(CCCO)CC1)=O)c1ccoc1)CC(C)(C)C O=C1NCC2(CCN(C(=O)CN(C(=O)Cc3ccns3)CC3CC3)C2)N1 Clc1cccc2c(CNC3CCC(c4cccc(Br)c4)C3)csc12 c1(C(C)C)ccccc1OCC(C)COC1CC(N2CCOC(C)C2)C1 C1(NC(CNC(CC)=O)=O)CCCC(N(C(=O)CN2CCN(C)C2=O)C)C1 c1(C(=O)NC(CNC(C(COCC)(C)C)=O)CC)cc(F)c2[nH]nnc2c1 C1(CNC(c2oc(C)c(CO)c2)=O)CN(C(c2cc(C(N)=O)co2)=O)C(C)(C)C1 n1(CC)ncc2c1CC(C(N1CCC(CNC(=O)CN(C)C)C1)=O)CC2 c1(OC)ccc(C(=O)N(C(CNC(c2coc3c2CSC3)=O)C2CC2)C)cc1O c1(C(=O)NCCC2CCN(C(=O)C=CBr)CC2)cc2c(=O)[nH]ccn2n1 C1(N(C(CC)=O)C)CCCN(C(=O)C=Cc2ccc(I)o2)CC1 CCC(C)(COC)C(=O)N1CCCC(CO)(CNC(=O)C(O)CC2CC2)C1 c1(NC(C)=O)ccc(C(N2CCN(C(=O)CC3=CCCC3)CC2CF)=O)cc1F C(C)(CCC(=O)N(CCCC(=O)NCC1CCN(C(C)=O)CC1)C)OC c1(NC(CC(CC)C2CCC2)=O)cc(C)c(Br)cn1 C1(CCN)CCCN(C(=O)NCC(c2ccccc2Cl)O)C1 c1(C(=O)NC(CNC(C(C)=C2CCC2)=O)C(C)C(C)C)nn(C)cc1[N+](=O)[O-] c1(OCC(N2CCN(C(C(C)C)=O)CC(C)(F)C2)=O)cccc2c1OC(C)(C)C2 c1(C(=O)NC2CCN(C(CCC=C)=O)C(C)C2)cc2c(nc1N)CCC2 c1(C(=O)NC2C(NC(C(=O)NC(C)C)=O)CC2)cocc1Br c1(OCC)ccnc(O)c1C.c12nc(C)c(s1)CNC2c1nnnn1CCSC C1(CNC(c2ccsc2C(F)F)=O)CC2(CCN(c3nnc(O)s3)CC2)CO1 Cc1cc(Br)c(C(=O)NCC2C3CN(C(c4coc(C#N)c4)=O)CC23)s1 CC(C)S(=O)(=O)CC(=O)NCC1CSCC(CO)C1 C1(NC(C(c2cccc(F)c2)(C)O)=O)CC2(C1)CC2CNC(=O)C1=CCCC1 C(=O)(C(C)C(C)(F)F)NCCC1CCN(C(CCCn2c(C)ccc2C)=O)C1 C(C(C)C(F)C(=O)Nc1cncc(CO)c1)NC(C(CC)C#N)=O C=Cn1nncc1C(=O)NCC1C=CC(NC(=O)C(CC(C)C)NC(=O)OC)C1 C(N=c1nc2sccc2c(N2CCC(C#N)C2)[nH]1)c1cnc(C)o1 N1(CC2(NC(Cc3nnc(C)o3)=O)CC2)CCN(C(=O)C(C)(Cl)Cl)CC1 Cc1ccc(C(N2CC(O)(C(C)NC(=O)C(C(C)C)C3CCC3)C2)=O)cc1C Cn1ncc2c(NCc3cn4c(n3)SCC4)[nH]c(=NCCC3CCOC3)nc12 C(CC(C)(C)C)N(CC(=O)NCC(CC)NC(=O)CCC1CCCN1C)C c1(OC)ccc(S(=O)(=O)NC(C(=O)O)C2(CC(C)C)CC2)c(C(C)(C)C)c1 c1(CC)ccccc1NN1CCN(C(=O)OC(C)(C)C)CC1.C12CN(C1)C2 S(=O)(=O)(c1cc(Nc2sc(-c3ncnc4c3CCCC4)nc2C)n(C)c1)NC Cc1ncc(C(N2CCCC2CCNC(=O)CC(O)C(C)C)=O)cc1N C=CCC(C)(C)CC(=O)N(C(CC(F)F)C(=O)NCC1CCCN1C(C)=O)C C123CCC(CC1)(CO2)C(=O)NC3.C1(C(=O)NC2C(COC)C2)CC(C(C)(C)C)C1 C1(NC(CC=CCCCCC)=O)CCCC(NC(=O)COCc2scnc2C)C1 C(N=c1nc(OC)c(F)c(C)[nH]1)C1C2CN(C(c3c(CC)cncc3)=O)CC21 C1(C(N2CCC(OCC(=O)N(C)CC3(C)CCC3)C2)=O)C(C#N)C1(C)C N1(C(c2c(CC)noc2)=O)CCCC(C(=O)NCC(C(C)CC)OC)C1 N1(C(Cn2cnc(=N)[nH]2)=O)CCOC(C(=O)NCCOCCC(=O)NC)C1 c1(C(N2CCC(C(=O)NCCC(C)F)CC2)=O)cnc(C)c(C)c1 Cc1nn(Cc2ccc(CCCN3CCCC3c3cnn(C)c3)cc2)c(C)c1Br c1(CCCC(=O)NC2CN(C(C3C(C)C3)=O)C2)ccc2c(c1)Cc1ccccc1-2 c1(-n2c(-c3c(C)cncc3)nc(-c3ccco3)n2)cc(F)ccc1C CC(C)C1=CCC(NC(c2occc2CNC(C2(C)CC3CC3C2)=O)=O)CC1 c1(NC(C2CCN2Cc2cnccc2Cl)=O)cccc(Br)c1Cl C1(C(N2CC(NC(CC3(CC)CCC3)=O)C(OC)C2)=O)CCC(C2CCC2)CC1 c1(C(=O)NCC)ccc(F)c(F)c1F.C1(COCC)C(=O)N1.C(C)(C(=O)OC)(OCC)CO C1(C(N2CCC(O)(CNC(C3CCN(C(=O)NC)C3)=O)C2)=O)(CC)CCCCC1 c1(C(N2C(C(C)NC(c3cnc(OCC)s3)=O)CCCC2)=O)ccc(F)cc1C N1(C(CCC2CCC(C)O2)=O)CCN(CCNC(=O)Cn2ncccc2=O)CC1 CC#CC1CCN(C(C2CCCCC2(C)NC(c2cc(CC)[nH]n2)=O)=O)CC1 c1(C(=O)NC2CC(C)CN(C(=O)C(C)(F)F)C2)c(Cl)oc2ccccc12 C(=O)(NNc1cc(I)ccn1)NC(CCC(=O)O)c1ccc(F)cc1 C(=O)(C1=COCCO1)NC1CCC(OC2CCN(C(COC)=O)C2)C1 c1(OC)ccc(Cl)cc1CC(=O)NC(c1c(C)nn(C)c1C)C N1(C(CCC(=O)NC)=O)CC(C)OC2(CCN(C(=O)C(C)(C)c3cnc[nH]3)C2)C1 N1(C(c2c[nH]nc2C(F)F)=O)CC(NC(=O)C(F)(F)c2ccco2)C(C2CC2)C1 C=CCC(CC(=O)N(C1CN(C(C)C)C1)C)NC(=O)C(C)COC c1(NC(C2C(C)(C)CCN(C(C(CCC)C)=O)C2)=O)cnc2ncnn2c1N CC(C)(C)C(CNC(=O)CCN1CCCCC1)NC(C12CCCC1(C(N)=O)C2)=O C(CC(F)CN=[N+]=[N-])NC(C(C)(CO)NC(CC1ON=C(C)C1)=O)=O c1(C(=O)NC2(COC)CCN(C(C(CCC)OCC)=O)C2)cccc2c1COC2 c1(OC)cc(C)c(C(N2CC3CC2CC3CNC(c2cnoc2)=O)=O)cc1OC c1(CC(C)NC(=O)NC2N(S(CC)(=O)=O)CCC2)ccccc1Cl.C1(C)C(=O)N1 N1(C(c2c(C)nns2)=O)CCC(C)(C(=O)N(CC(=O)NC(C)C)C)C1 C1(C(=O)NC(C#C)C)CC12CCN(Cc1ncc(Cl)cc1Cl)CC2 C1(CNC(CC(CC)C)=O)CC2CN(C(c3ccc(C)nc3)=O)CC12 c1(C(N2C(C#N)C3CC3C2)=O)csc2c1CCN(C(c1ccc(Br)cc1Br)=O)C2 C1(C(=O)NCC2(N(C(=O)CSc3cnn(C)c3)C)CC2)CC2(CCO1)CC2 c1(C(N2CC3C(C(=O)Nc4ncc(C)c(Cl)n4)(C3)C2)=O)ccc2c(c1)NC(=O)C2 N1(C(CCC(=O)NCCc2cccc(C)c2)=O)C2C=CCC1CC2 C(CCCCCC(=O)N(C1COCC1O)C)NC(CCC(C)(C)N(C)C)=O C1(CNC(C2CC(N(CC)CC)C2)=O)CCN(C(c2conc2C)=O)C12CCC2 Cc1cccc(N2CCC2NC(=O)C(C)(C)NC(=O)CCSC(F)(F)F)c1C C(=O)(C(F)C(C)(C)O)N(C1CCN(C(CN2CCN(C)CC2)=O)CC1)CCO C(C)(C)(C(=O)NCC(O)CNC(C1(O)CC(c2ccccc2)C1)=O)OCC C1(CC)CCCCC1OCC(N1CC2C(NC(=O)Cn3cc[n+](C)c3)C2C1)=O c1(C(N2CCC(NC(CC(=O)N(C)C)=O)CC2C2CC2)=O)ccc([N+](=O)[O-])cn1 C1(N(C(=O)C=Cc2cscn2)C)CCCCN(C(C2CCC23CCC3)=O)C1 C12(CNC(C=CCC)=O)CCC(CC1)N(C(=O)C(C)(Cl)Cl)C2 c1(COCC(C)N(C(C2C(C(=O)OC)C2)=O)CCN(C)C)ccc(Cl)nc1 CC1CCN(C(=O)CC2CCSC2)C1CNC(c1nccc(C(F)(F)F)n1)=O c1(CN(C)C)ccccc1NC(=O)NCC=C(Cl)Cl C(c1c(C)noc1C)=CC(=O)NCC(CCOC)NC(c1cc(C(N)=O)c[nH]1)=O C1(C(N(C)CCNC(c2ccc(C(F)(F)F)cc2)=O)=O)CC2CCCCC2O1 CCC(CC(=O)N1CC(C2CC2)C(F)(C(=O)O)C1)C(C)(C)C C(=O)(C(CC)CC)Nc1cn(CC2N(C(C(C)(C)OCC)=O)CC=C2)nn1 Cc1ccc(F)c(C(=O)NC2(CNC(=O)Cc3cc(Cl)cs3)CCC2)n1 CCCCCCCCN(C)C(C1(CNC(c2cnc(C)[nH]c2=N)=O)CC1)=O c1(C(=O)Nc2cc(C(F)(F)F)ccc2C2CC2)c[nH]c(=O)c2ccnn12 c1(C2C(CNC(C(C)N(CC(=O)NCC(C)C)C)=O)C2)ccccc1 c1(C(=O)NCc2nocc2C(=O)NCCC2CCCS2)cncc(O)c1 c1(N(C)C)c(C(N2CC=CC(NC(c3csnn3)=O)C2)=O)cnc2ccccc12 N1(C(COCC#C)=O)CCOCC(C)(CNC(c2nc(C)sc2CC)=O)C1 c1(C(C(=O)NCc2nccs2)N(C2COC2)C2CCC2)cc(Br)cs1 C1(NC(c2cc(F)cc([N+](=O)[O-])c2)=O)CC2CC1C1CCCC21 c1(C(=O)NC(COC)CNC(=O)CC2CC=CCC2)cc([N+](=O)[O-])no1 Cc1cn2cc(CC(=O)NCCCNC(=O)C(C)(C)c3cnsc3)nc2s1 CC1CCCc2nc(C(=O)OCC3CCC3=O)cn21 C1(CC(=O)NCC2(CCC)CC2)CC(C)(C)CN1C(=O)C(CC)C(C)C Cc1[nH]nc(C(F)F)c1C(=O)NC(C)C(CO)NC(C1(CCO)CC1)=O C1(N(C(C)Cc2ccccc2)C(c2cc(C)no2)=O)C2CCC1CNC2 Cc1nnccc1C(=O)NC1COCCC1NC(c1cc[nH]c1C1CCCC1)=O c1(OC)cc(C(=O)N(C)CC2CN(C(C3CC3C(F)(F)F)=O)C2)ccn1 Cc1ccnc(O)c1C(=O)NCC1CCCCC1NC(c1csc(C2CC2)n1)=O CC1(C(=O)N(C2CCN(c3cc(-c4cccs4)ncn3)CC2)CC2CC2)CCNC1=O C(=O)(CCC(=O)NCCC1CC1NC(c1coc(C(=O)OC)c1)=O)NC C(CN=C(NCC1(C(C)(C)C)CCCO1)NC1CCNC(=O)C1)N(C(C)C)C N1(C(CN(C)C2CC2)=O)CCC(CNC(=O)COCC2CCCO2)C12CC2 C12(CNC(C3CN(C(=O)NC)C3)=O)CC1CN(C(c1cccc(F)c1)=O)C2 C(=O)(C1CCCc2ccnn21)NCCN(C(CC(C)P(C)(C)=O)=O)C n1(C2CC(COC(F)F)C2)nnnc1CC1CC1CF c1(N(CCNC(C=CCC)=O)CCC)cc(C(=O)NC2CC2)ncn1 c1(C(=O)NCCC2CC(NC(c3c[nH]c(Br)c3)=O)C2)ccc(C(F)F)o1 C(C(C(=O)NCC1CC(F)(F)CO1)C(C)C)NC(CCCOCC)=O Cc1scc(C(=O)NC(C)CNC(=O)C(c2ccc(Cl)cc2)C)c1N CCC(CNC(C1CN(C2CCC2)C1)=O)NC(C1(c2cnoc2)CC1)=O c1(C(=O)NCCC2CC(NC(CC(=O)OC)=O)C2)c(F)cccc1Br CCCC(CC)C(C(=O)NC1CCC(F)(F)CC1)N(C)Cc1ccc(F)cc1C CC1(NCC(c2cccc(-c3cccnc3)c2)C(=O)O)CCOC1C1CC1 c1(C(=O)NCC2CC(F)(CNC(=O)Cc3ccoc3)C2)cc2cccnn2c1 c1(CCN(C)C(=O)N(CCCn2ccnc2)C2CC2)ncc(C2CC2)o1 c1(C(=O)NC(CN(C(=O)CS(N)(=O)=O)CC)C)ccc(-n2cccn2)c(Cl)c1 C1(CNC(C2ON=C(C)C2)=O)CC2CCCC2N1C(c1ccn2ccnc2n1)=O c1(C(=O)NCC2(F)CC(CNC(=O)CNC(c3ccco3)=O)C2)cc(Cl)cnn1 c1(CN(C)CC2CCS(=O)CC2)nc2ccccc2[nH]1 Cc1ccc(SCC(N2CCOCC2c2ccccc2Br)=O)cc1 C1(C(N2C(CNC(c3nc(C)n(C)c3)=O)C=CC2)=O)CC(O)c2ccccc2O1 O=C(CCCCCF)NC1(CNC(=O)CC2CCC3CC23)CCCOCC1 C12(C(=O)NC3C(NC(COCC#C)=O)COC3)CCN(CC1)CC2 C1(CNC(C(C)(C)CO)=O)COCCN(C(=O)CCc2ccc(N)cn2)C1 c1(C(=O)NC(C2CC2)C2CC2)cccc(C2CC2)c1.CCO CC1CC(C(=O)NCC2CCCN(C(C3(Nc4ccc(Cl)cc4)CC3)=O)C2)=NO1 Cn1ncc(C(N2CC(NC(=O)C=Cc3cc[nH]n3)C(O)C2)=O)c1N c1(C(=O)NC2(CNC(c3ccc(CC(N)=O)cc3)=O)CCOC2)cncc(O)c1 N1(C(CCC=C)=O)CCCC1(C)CNC(c1cc(C(F)(F)F)nn1CC)=O C1(CNC(=O)Cn2ncnn2)CCCN1C(=O)Cc1nncs1 N1(C(C2(C#C)CC2)=O)CC2C3CCC(C(NC(c4cccc(Cl)c4Cl)=O)C3)C2C1 c1(OC)cc(S(=O)(=O)NCC(N2CCc3ccccc32)=O)cc([N+](=O)[O-])c1C N1(C(C(C(C)C)OC)=O)CCC(NC(c2ccncc2C(F)(F)F)=O)C(O)C1 C(CCN=C(NCc1cccc(C(C)C)n1)N1CCC(c2cccnc2)C1)SC C1(c2nnnn2CCO)(NCCc2c(C)ccnc2)CCCC2CC12 CC1(C)CCN(c2nc(Cl)ncc2C2CC2)CC1NC(=O)CC1CC2CCC1C2 CCCCCC(O)C(=O)NCCCN(C1CCCCC1)C(C)C(=O)OCC c1(C(=O)OC)cc(O)nc2c1CCCN2C(=O)COc1cccc(Cl)c1 CC(C)(F)C(C)(F)C(=O)N1CC(NC(c2cc(N)cnc2Br)=O)C(C)(C)C1 Cc1cccc(OCC(N2CC(C)(NC(=O)C(C)(C)C3CCC3)C2)=O)c1 C1(O)(CC)C=C(c2cccnc2C(=O)Nc2ccc(SC)nc2)CCC1 CC1(F)CCC(C(=O)N(c2ccc(F)cc2)CCO)CC1.N12CSCC1C2=O c1(CNC(=O)NCc2nnnn2CC2CCOC2)cc(C2CC2)ccn1 c1(C(=O)NCC2CCC(CNC(COCC)=O)CC2)[nH]c2cc(C)ccc2c1C c1(NC2C3N(C(c4ccc(C)cn4)=O)CC(CC3)C2)nc(C)c([N+](=O)[O-])cc1Cl C1(C(N2C(C(=O)OC)CC2C)=O)CC2CC2N1C(c1ccc(C)cn1)=O CCCC(C)(CCC)C(=O)NC1CCC1C(N1CC2(CCNC(=O)O2)C1)=O CCS(=O)(=O)CC(=O)NCCC1CCCN(C(=O)COC(C)C)C1 CCC(CC(=O)N(C)C(c1cc(C)on1)C)N(C)C(C1CCOC1)=O N1(C(C2(C)CC2)=O)CCCC(CCNC(C2(O)CC2(C)C)=O)C1 N1(C(c2c(OC)ccs2)=O)CCC(C(F)(F)F)C(NC(c2cnn(C)c2C)=O)C1 N1(C(CC2CN(C(c3c(C)nn[nH]3)=O)CC2C)=O)CC2C=CC1CC2 O=C(N=c1[nH]oc2cc(Cl)ccc12)NC1CC(c2cc(F)ccc2F)=NO1 CC1=NNC(=O)C1CC(=O)NC(CNC(C1(C(F)F)CCOCC1)=O)C(C)C C(=O)(C1Cc2ccc(Cl)cc21)NCC=CCNC(c1ccc(N)c(Cl)c1O)=O C(=O)(CCCCC(N)=O)NCC(CNC(c1ccc(OC)c(O)c1)=O)(C)F n1(CC)nncc1C(=O)NC1COCC1NC(=O)COC1CCOC1 Cc1sc(Cl)nc1C(=O)NCC(C1CCOC1)NC(=O)CCc1ncco1 N1(C(CCOC)=O)CC2CCN(C(c3cnn(-c4ccccc4F)c3)=O)C2C1 Cc1cn(C)nc1C(=O)NC(C1CCN(C(=O)CCc2nc(C)c(C)[nH]2)CC1)C C1(C)(C(=O)NCc2cn(CC(=O)OC)nn2)CCN(C(=O)CC2CCCCO2)C1 c1(N2CCC(NC(c3c(CC)ncnc3)=O)(COC)C2)c(Cl)cncc1[N+](=O)[O-] C(C(C)(C)C(=O)N1CCC(CN(C(=O)CC(C)c2ccco2)C)C1)SC C1(F)(CNC(C(CC)(C)CO)=O)CCCN(C(c2cc(Cl)cc(Cl)c2)=O)CC1 C1(SC)CCCN(C(=O)C(=O)NC2CC(c3cnc(Cl)c(C)c3)C2)C1C c1(C(=O)NC(CC(C)NC(CSCCCC)=O)C)cc(C)c(C)c2ncccc12 C1(CNC(C2CCN(C3CCN(C(C)=O)C3)CC2)=O)CC2(C1)CC(C)(C)C2 c1(C(N2CC(F)(CNC(CN(S(CC)(=O)=O)C)=O)C2)=O)cnc2c(ccn2C)c1 c1(C(C)(C)C)ocnc1C(=O)NC(CNC(C12COCC1C2)=O)C1CC1 CC1CCOCC1(c1nnnn1-c1ccccc1)NCc1cc(Br)cn1C CC(C)C(C)CCNC(C1CCC(C2CC2)N1C(=O)C=Cc1ccn(C)c1)=O N1(C(C2(OC)CC2)=O)CCCC2C1CCN2c1nc(SC)ncc1Br Clc1cccnc1C(c1ccccc1)NC1CCC2CCC12 CC1=C(C(=O)N2CCSCC2C(=O)NCC(N2CCOCC2)=O)CCO1 CCC(C)(C)C(=O)NC1(C(=O)N(CC(O)CN(C)C)C)CSC1 Cc1cnc(C(N2CCN(C(c3cccnc3C)=O)C(C3CCC3)C2)=O)c(F)c1 C1(C(C(=O)NC2CC(c3cn(CCOC)nn3)C2)C)CC2CCC1CC2 N1(C(c2cc(C)c(F)cc2F)=O)CCOC2(C1)CN(C(c1ccc[n+]([O-])c1)=O)C2 C1(C(=O)NCC2C(NC(C3(SC)CCC3)=O)CCCC2)CCC2(CCC2)O1 c1(NC)cnncc1C(=O)N(C(C)CCNC(c1sc(CO)nc1C)=O)C c1(CNC2CCCN(CCOC)C2)ccc(OC)c2oc(C)cc12 c1(NC(C2CN(C(c3cc(Br)cnc3Br)=O)CCC2O)=O)ccc(Br)c(Cl)c1Cl c1(C2CC(CC)C2)ccc(F)cc1.c12occc1C1(CC1)C(c1nnnn1C)N2 c1(C(N2CCN(C(C3C(=C)C3)=O)CC2CCO)=O)ccc2c(c1)B(O)OC2 c1(OC)cc(OC)c(C(N2CCOC(C(C)NC(=O)CCC(C)SC)C2)=O)cn1 c1(C(N2CCC(C3CCCN3C(C3CCCS3)=O)C2)=O)cc2c(Cl)nccc2o1 c1(C(=O)NCCCNC(C(C(=O)OCC)OC)=O)cncc(Cl)c1C C1(NC(=O)NCc2cc(C(C)C)on2)CCC2(CC1)CNCCO2 C1(C(N(C2CCN(C(C3CN(C(C)C)C3)=O)CC2)CC)=O)C2CCC1CC2 Cc1cc(C(=O)NCCOCC(N2CCCCCC2)=O)ccc1O CC1C(C(=O)N2CC(C)C(NC(=O)CCS(C)(=O)=O)C(C)C2)=NOC1C Cc1cnccc1C(=O)NC1CCC(N(C(=O)C(C(C)O)NC(N)=O)C)CC1 c1(C(N2CCC(OC)(CNC(C3COCC(C)O3)=O)C2)=O)cnc(O)n(C)c1=O Cc1cncc(-c2cccc(C3CN(CC(N4CCCCCC4)=O)C3)c2)c1 C1(C(=O)NC2CC(CNC(c3cc4sccc4s3)=O)C2)CCc2[nH]nc(O)c2C1 c1(OC)ccc(C(c2nnnn2C2CCCC2)NCCCCS(C)(=O)=O)c(C)c1 CCS(=O)(=O)C=CC(=O)NC(C1(O)CCN(C(=O)Cc2sc(O)nc2O)C1)C C1(C(=O)NC2CN(C(c3ccc(C)cc3F)=O)CC3C2C3)CCc2c[nH]nc2C1 c1(C(N2CC(C3CN(C(c4cc(Br)cs4)=O)C3)OCC2)=O)ccc(F)c(Cl)c1 C1(C#N)(C(N2CCCC(O)(CNC(CCC(C)OC)=O)C2)=O)CCN(C)CC1 c1(C(=O)NCC2CCC2NC(=O)C(c2cccc(Cl)c2)O)ccc(Cl)c(F)c1 Nc1c(Cl)c(C(=O)NCC2CCC2NC(=O)C=Cc2ccco2)cc(F)c1Cl c1(C2CC(C(=O)ON3CCC(OC(F)F)C3)C2)ccc(F)cc1 C1(C(N(C(C)CN(C)C)C)=O)CCN(C(=O)C(C)(C)C)C1C C1(C(N2CC(C)C(C)C2C)=O)CC2CCC(C1)N2C(C1CCCOC1)=O c1(C(=O)NC(C)CNC(=O)CCSc2ccccc2Cl)cc(O)cc(O)n1 N1(C(C(c2cccc(C)c2)O)=O)CCN(C(c2cc(C3CC3)nn2C)=O)C2(CC2)C1 C1(C(N2CCC(C)CC2)=O)CCN(CC2CC2)CCC1c1ccccc1 c1(OC)cccn2ncc(C(=O)NC3CN(C(=O)CCC4CC4)CC(C)(C)C3)c12 N1(C(C(C=C)(C)CC)=O)CCC(C2(O)CC(NC(=O)C(C)=C3CC3)C2)CC1 C1(CNC(C2CN(CC)C(=O)C2)=O)CC2(CO1)CN(C(c1ccc(=N)[nH]n1)=O)C2 C1(C(C)C)CN(C(=O)CN(C)C(=O)C2CC2)CCN1C(=O)C(C)N(C)C C(=O)(C(C(C)(C)O)NC(C1CC1F)=O)NCc1nnn(C)n1 C(CCNC(C1C2CCCC12)=O)(C(=O)N1CCC(C(C)(C)O)CC1)OC N1(C(c2n(CC)ccn2)=O)CCN2C(=O)C(NC(C3CCN(C)C3C)=O)CC2C1 CC1(C)C(NC(=O)C(=O)NCC2CC3C=CC2CC3)CS1(=O)=O Cc1cc(C(=O)NC2CCOC(C(=O)NC3(C#N)CCCCC3)C2)nc(O)n1 C1(C(=O)NCC2(C(C)NC(c3c(C)nccc3)=O)CC2)CC2CS(=O)(=O)CC2C1 N1(C(C=C(C)C(F)F)=O)CCN(C(c2ccc(C(C)(F)F)cn2)=O)CC(O)C1 c1(CNC(C2C=CCN2C(c2cn(C3CC3)cn2)=O)=O)cc(F)cnc1O C(=O)(C1OCCc2ccccc21)N1CC(CN(C(COC(CC)C)=O)C)C1 c1(C(=O)NC2CCN(C(C=CCC)=O)CC2CC)nn(C)c(=O)cc1C C(C1=NOC2CN(C(c3cnsn3)=O)CC12)NC(c1cn(C)nc1Cl)=O N1(C(CC2CCCC(NC(C3C(C)CC3)=O)C2)=O)CCC2(CSC2)C1 C1(C(=O)Nc2c(C)ccc(-c3ccccn3)c2)CCN(C)C12CCCNC2 CN=c1cc(C(=O)NC2CCC(CCNC(=O)CCC3CCCCC3)C2)cc[nH]1 C12(C(=O)NC3(C#C)CCCOC3)CCC(CC1)N(C(C1(OC)CC(CO)C1)=O)C2 CC(C)(C)C(CNC(=O)C=Cc1cnc[nH]1)NC(=O)CSCc1csc(=N)[nH]1 C12(CNC(C(CC)SC)=O)CCC(CC1)N2C(c1cn(CC(=O)OC)nn1)=O N1(C(c2ccc(CC)cc2)=O)CC2(C1)CN(C(=O)Nc1c(OC)cccc1Cl)C2 N1(C(C)=O)CCC(NC(=O)C=CCC(C)(C)NC(=O)CC2CCOC2C)C1 C1(c2n(CCCC(=O)NCc3c(C(=O)OCC)nsc3)nnn2)CCCC(OC)C1 N1(C(c2cncc(CC)c2)=O)CC(CC(=O)NCCC(C)C(F)(F)F)CCC1C C(CCCC(=O)NC1(CCCNC(c2cccnn2)=O)CC1)(OC)OC N1(C(c2c(CNC(Cc3n(C(C)C)cnn3)=O)noc2)=O)CC(C)CCC1C C1(NC(c2c(CNC(=O)CC3CCOC3)cco2)=O)CCCC2(CC2)C1 n1(CC(=O)NC2C(NC(CC3(NC(C)=O)CC3)=O)CCC2)ccccc1=O c1(C(C(=O)Nc2ccc(N3CCOCC3)nc2)=O)cc(F)cc(Cl)c1 C1(NC(C(c2c(C)noc2C)CC)=O)CCN(C(=O)C(C2CCCCC2)C)CC1 c1(CC(=O)NC2CC(CNC(C=C(C)Cl)=O)C2)ccc(OC(F)(F)F)cc1C c1(N(CC)Cc2ccccc2-c2cn[nH]c2)nc(C)cc(=NCC2CCOC2)[nH]1 n1(CCNC(C2(CNC(=O)Cc3cn[nH]c3)CC2)=O)ncc2ccccc12 c1(C(N2CC(OCC=C)C(C=C)C2)=O)ccc2nc[nH]c2n1 C12(C(=O)NCC(CNC(C3C=CCS3)=O)OC)CCC(C1)S(=O)(=O)CC2 C12(C(=O)NC34CC(C(=O)NCC5C(C)COC5)(C3)C4)CCCN(CC1)C2 N12CC3CC1C(C3)C2.C1(NC(=O)CC2CC3CCC2O3)CNC(=O)C12CC2 C1(C)(C(=O)NCC(CNC(CCc2c(C)nccc2)=O)CO)CCN(C)CC1 Cc1cc(C(=O)NC2CCC(NC(=O)CNC(C3CC3C)=O)CC2)c(C)[nH]1 c1(OCC)ccc(NC(=O)CC(O)CC)c(OCC)c1.N12CCC(C1)NCC2 NS(=O)(=O)CCCC(=O)N1CCC(O)(CCNC(C2CCC2CF)=O)CC1 C1(C(=O)NCC2(C)CCC(NC(C3C(CC)C3)=O)C2)CC2(CCCCC2)C1 C1(C(CNC(=O)C(O)Cc2cnc[nH]2)F)CCN(C(=O)C=CC2CCOC2)CC1 N1(S(CC=C)(=O)=O)CCc2sc(C(=O)Nc3cc(Br)c(F)cc3O)cc2C1 c1(C(=O)NCC2CCCN(C(C3C=CCC3)=O)C2)c(Cl)ccc2ncccc12 N1(CCCOCC)CCC2(CC1)CN(C(=O)CCNC(N)=O)CC(C)O2 C1(C(=O)NC2CCCC(NC(c3c(OC)c[nH]n3)=O)C2)CCCCC(F)(F)C1 c1(CNC(C(c2ccc(F)cc2)NC)=O)nn(C)c(Cl)c1Br CCC(C)CCC(=O)NC1(CCC)CCCN(C(c2ncc[nH]c2=O)=O)C1 C1(NC(C2C3COCC23)=O)CCC12CCN(C(c1[nH]nc([N+](=O)[O-])c1Cl)=O)CC2 C(=O)(C(O)CCCNC(=O)Cc1cncc(C)c1)NC(CC(C)(C)OC)C C(=O)(C(CC)C(C)C)NC1(CC=C)CCN(C(c2cnc(Cl)[nH]2)=O)C1 N1(C(C(CCOC)NC(CC(C(CC)C)O)=O)=O)CC2CCCCC2C1C c1(C(C)(C)C)ccc([N+](=O)[O-])cc1NC(=O)CCCCCF CCCCCCC(C)C(=O)NC1CC(CCC(N2CCC3(CC2)CC(O)C3)=O)C1 Cc1ccn(CC(=O)NC23CC2CN(C(=O)CC2(C)CCS(=O)(=O)N2)C3)c(=O)c1 C(=O)(C1=CNC2=NCCC2=C1)NC1(CN(C(=O)Cc2cnns2)C)CC1 c1(SC(C2CCN(C)CC2)C(=O)OC)cc(Br)ccc1C.C1(C)(C)CC(=O)N1C c1(C(=O)NCC(CC)NC(=O)C(C2CCCCC2)O)cc(C)co1 C=C(C)CCCC(=O)NC1CCCC1NC(=O)Cn1nc(C)n(C)c1=O CC(C)(C)C(CNC(=O)CC1CC2(CC2)CO1)NC(=O)CCc1ccco1 C1(NC(=O)C(Cl)=CCl)COC2(C1)CN(CC1(NC(C(C)NC(N)=O)=O)CC1)C2 c1(OCCOC)cccc(CNC(c2cccc(C(C)OCCO)c2)=O)c1 CN1C2CCC1CC(CC(=O)NC13COC(C1)C(NC(=O)Cc1ccon1)C3)C2 C1(NC(Cc2cc(C)sc2C)=O)CCN(C(C2(CO)CCC2)=O)CC1F C1(C(=O)Nc2c(C)scc2)CN(C(=O)CNC(N)=O)CC1C C=CCC(C)(CC)C(=O)NC1CCCC1NC(=O)CCC(C)(F)F Cc1ccccc1C(C)CC(=O)NCCN(C(c1cnc(C2CC2)s1)=O)C1CC1 C(CCC(=O)N(CCNC(=O)CNC(=O)CC1CCCCC1)CC)OCC C1(NC(c2nnn(CC)c2C)=O)CC=C(C(=O)NC2COCC(C)(C)C2)C1 N1(C(C)=O)CC2CC1CC2NC(=O)Cn1nc(-c2cccs2)oc1=O C1(NC(COCCOC)=O)CC2CC(C1)N(C(c1cccc(C(C)C)c1N)=O)C2 c1(C(=O)NC2COCCN(C(c3nncc(C)c3)=O)C2)cccc2oc(O)nc12 C1(NC(C(C)OC2CC2)=O)CN(C(=O)Cn2cnc3ccccc23)C2(CCC2)C1 C1(C(F)(F)F)CCC(N=c2[nH]c(-c3ccccc3)nc(=NCCC#N)[nH]2)C1 c1(CC)c(C(=O)NC2CC2C(=O)Nc2cnn(CCOC)c2)ccn1C C1(CNC(c2cc(Cl)sc2Cl)=O)CC2CCC1N2C(c1cnns1)=O C1(NC(c2cc(COC)no2)=O)CN(C(=O)CC(C)=C(C)C)CC1SC c1(NCC23C(O)CCC2C3)nc2ccccc2nc1NC1(CCO)CCCCC1 C1(CCC)CN(C(=O)CSCCC#N)CCN1C(=O)CC1(OC)CC1 c1(C(N(CCC)CCNC(=O)C#CC2CC2)=O)ccc(F)c(C)c1C#N c1(OC)cc(CN2CCC(C)(C(=O)NCc3cccc(F)n3)C2)c(Br)cn1 O=C(C1CCCc2ccccc21)NC1CC(NCc2cn3cc(F)ccc3n2)C1 N1(C(C=CC)=O)CCC(CO)(N(C(=O)CCC2CCC(C(N)=O)O2)CCN(C(C)(C)C)C)C1 N1(C(C23C(C)(C)OCC2C3)=O)CCC2CCN(C(=O)C(N)=O)C2C1 c1(OCC)cnc(C(N2CC=CC(NC(C34CC(C)C3C4)=O)C2)=O)c(Cl)c1 N1(C(C(CCC)N(C)C)=O)CC2CCC2(N(C(=O)C=CCOCCOC)C)C1 C1(C(=O)NC(CNC(c2cn(CC)nc2OC)=O)C2CC2)CC(C2CC2)=NO1 CCCCCCC(C)C(=O)N1CC2(CC(CC(=O)NC3CCCCCC3C)C2)C1 C1(C(N2CC(CCCCNC(C3CCCC(=O)C3)=O)C2)=O)C2CCCCCC12 c1(C(=O)NCCCN(C(c2[nH]cc3c2CCC3)=O)CC)ccc(C)c(Cl)c1N c1(C(=O)NC(CC)CNC(c2cnnc(O)c2)=O)ccc2oc(O)nc2n1 C1(NC(=O)Cc2ccnc(O)c2)CCCC(NC(C23CCCC2C3)=O)C1 C(=O)(C(C)N=c1ccn2ncc(C#N)c2[nH]1)N1CCCC(C(=O)NC(C=C)C)C1 N1(C(CC=C)=O)CCCCC1C1CCCN1C(c1cc(OC)ccc1N)=O c1(C(=O)NCCN(C(c2c(CCC)nns2)=O)CC)cn(C(F)F)c(C)n1 C=Cc1cncc(C(=O)N(CCC(C)N(C)C(C)=O)C)c1.C12CCCN(C1)C2=O C(=O)(CN1C(=O)CSc2ccccc21)NC(C(C)(C)C)CNC(c1ccoc1)=O C1(CCNC(CC2(N(C)C)CC2)=O)CC(NC(=O)C(F)C2CCOC2)C1 c1(SC)ncc(N)c(C(=O)NC2COCCC2NC(=O)COc2cccnc2)n1 c1(C(N2CC(NC(C(C(CC)(C)C)O)=O)C(C)CC2)=O)sc2ccccc2c1C c1(CSC(C)C)cccc(C(=O)Nc2nccc(N3CCOCC3)n2)c1 C12(CNCC(c3ccc(F)cc3)CO)CC1CCC2(F)F c1(OCC)ccc(CNC(=O)NC2(n3cc(Br)cn3)CCCC2)c(Cl)n1 c1(CNC(c2n(CC)ccn2)=O)cccc(CNC(=O)CC2CN(C)CC2O)c1 N1(C(CC(C)OC)=O)CCOC(C(=O)NC2(C)CC(O)C2)C1 CN1CC(N=c2[nH]c(N3CCC(F)(CO)C3)nc3ccsc23)CC12CCOCC2 c1(C(=O)NC(C2CCN(C(C(C)SC)=O)C2)(C)C)nnn(C)c1C(F)F C1(C(=O)NCC(C(=O)NC2C3(CC(OCC)C3)C2)O)CC2(C1)CC(O)C2 C(CC(C)(C)C(=O)NCc1nn(C)cc1CO)NC(COCC(=O)NC)=O C(=O)(C1=NN2CCCN=C2N1)NC1(CNC(c2cc(C)cc(C)c2)=O)CCCC1 C1(C(=O)Nc2nc(-c3cnn(C)c3)cs2)(CC)CCNC1=O c1(C(=O)NCCCC(C)NC(c2c(C)n(C)nc2Cl)=O)cc2cc(Cl)sc2[nH]1 C(C(=O)NC1CCCC1CSC)(C(C)C)NC(c1nc(OCC)sn1)=O O=C(NNc1ccc2ncsc2c1)c1cccnc1C1CCCC1 c1(OCC)cccc(C(=O)NCC2CC2CNC(c2cc[nH]n2)=O)c1N C(C(C)(C)CC(=O)N1CCCC(F)C1)NC(CCc1ccn(C)n1)=O C1(CNC(C(C)NC(CC)(C)C)=O)CC2(CC2)CN1C(=O)C(C(C)(C)C)OC N1(C(C2CCCN(C(C=CC(C)C)=O)C2C)=O)CCN2CC(F)CC2C1 N1(C(Cn2nc(C)c(Cl)c2)=O)CCC(NC(C2CC(C)(C)C2)=O)C12CC2 C1(C(=O)NC(CN(C(=O)CN=[N+]=[N-])CC)C)C2CCC(C2)C1C Nc1cnc(Cl)cc1C(=O)NCCOC1CN(C(c2c(O)noc2C)=O)C1 C12(NC(c3ccnc(OC)n3)=O)CCC(CC1NC1CCC1(C)C)C2 C=CC(O)C(=O)N1CC(=C(F)CNC(C2CCCN2C(=O)OC(C)(C)C)=O)C1 c1(CC)noc(C)c1CNC(=O)CN(C1CC(C#N)C1)C(C1C2CCC(F)C12)=O n1(CC)ncc(CN(C=O)C(C2CCOC2)C)n1.N1CCC1 c1(SCC(=O)N(CCC(C)NC(C(C)OCCC#C)=O)C)ccccc1Cl.NCC c1(C(=O)NCC(CNC(C2C(CCC)C2)=O)OC)cccc(C2OCCO2)c1 c1(C(=O)NCCCN(C)C(C2(CO)CC2)=O)cc(C(F)F)nn1C c1(C(N2C3CN(C(C(C)(C)SC)=O)CC2CC3)=O)ccnc(S(N)(=O)=O)c1 CCCC(C)(O)CC(=O)N1CCC(N)C(O)C1.c1(C(=O)C=O)ccnn1C1CC1 Cc1cc(O)ccc1C(N1CC(NC(c2cnn(CCF)c2)=O)C(C)C1)=O Cc1c(C(N2CCCC(CNC(=O)CC3CNC(=O)O3)C2)=O)cnn1C c1(-c2c(C(=O)OC)nccc2)ccc(S(=O)(=O)N2CCC23CCCCC3)cc1 CC1CC2CN(C(=O)Cc3cscn3)CC2N1C(C12CCC(CC1)C2(C)C)=O C1(C(N2CC(N(OC)C)C2)=O)CCC2CCC1N2C(=O)C(C)(C)C(=O)N(C)C C1(CN(CCN(CCCOC)C)C)CCCN(C)C1c1cncn1C CC(C)C(F)(CNC(=O)C(C#N)C(C)(C)C)C(=O)NC1CC2CC1C(O)C2O c1(N2CCC(Cc3ccc(C)cc3)C2)ncnc(NCCC2CCOCC2)c1C c1(CNC(COCC)COC)c2c(nn1C)CCC2 CC(C)C(C)C(CNC(c1cccc(F)c1)=O)NC(c1coc(Cl)c1)=O c1(SC)ccccc1C(=O)NC1CCCCC1CNC(=O)CCS(C)=O Cc1nc(C#N)ccc1C(=O)OC1Cc2cscc2C1 Cc1cc(-n2cc(CNC(C34CC=CC(C3)OC4)=O)nn2)ccc1Cl c1(CC)cc(C(=O)NC2(CC(=O)NCCC3CCCCC3O)CCC2)n(C)n1 c1(C(=O)NCC(CNC(C(C)OCCC(C)C)=O)O)csc2cccnc12 C(=O)(C(F)(F)C(F)(F)C(F)F)N1C2C(CNC(=O)Cc3cncnc3)CC(C2)C1 c1(C(=O)NC(CCCNC(C(C)OCOC)=O)C)cc2c(C)cc(Cl)cc2[nH]1 C(=O)(C1=NN(C)C(=O)CC1)NCC1CCC(NC(c2onc(C)n2)=O)C1 C12(CNc3cc(C(=O)OC)cc(Cl)c3)CCC1C1(CC2)OCCO1 N1(C(C)=O)CCCCC1CC(=O)NC(C)C(CO)NC(C1CC=CC1)=O C1(C(N2CCC(CCC=C)C2)=O)CCCN(C2CCN(C)CC2)C1 c1(-c2cc(C)cc(C)c2)ccc2c(c1)CCN(C(=O)CNC(N)=O)C2 C#CCCCCCC(=O)N1CCC2(NC(C3CC(OC)C3)=O)CC2C1 N1(C(Cn2c(C)cc(C)n2)=O)CCC(CO)C(NC(c2cnc(S)n2C)=O)C1 N1(C(C(C)(C)O)=O)CCc2c(-c3nn[nH]n3)cccc2C1 C12(NC(C(CC#C)O)=O)CCC(CC1)N(C(c1cc(O)ncc1Br)=O)C2 c1(CC(=O)NCCC(C)N(C(c2cccc(C)c2)=O)C)oc2ccccc2c1C Cc1nn(C)c(Cl)c1C(N1CCC12CN(C(c1ccnc(CC(C)C)n1)=O)C2)=O C(CCCCOC)(C(=O)NCCC1CC1)N(C(c1cc(CO)oc1C)=O)CC Cc1cnn2ccc(C(=O)NC3CC3NC(=O)C(C)(C)c3ccc(Cl)s3)nc12 N1(C(C(C)C#N)=O)CCC2(C1)CN(C(=O)NC1(c3ccc(F)cn3)CC1)C2 C(CCCN=c1[nH]c(=NCC23COCCN2CCOC3)c2ccccc2[nH]1)OC C1(OC)CC(NC(C2CSC2)=O)C12CCN(C(c1c(C)[nH]c(C)c1C)=O)CC2 C(CN=C(NCCCCO)N(C)CCSc1ccoc1C)=CC C1(NC(C2CCn3ccnc3C2)=O)CC2CCC(C1)N2C(C1(C2CC2)CC1)=O c1(C(=O)NC(CNC(CN(CCC)C)=O)C)cc(=O)c2ccc(Cl)cc2o1 c1(C(N2CCN(CCCCCNC(=O)C=CI)CC2)=O)coc2c1C(=O)CCC2 c1(C(N(CCCCN(C(=O)CCCC2CCC2)C)C)=O)cnn2ccn(C)c12 N1(C(C2CCC3C(C)(C)C2C3)=O)CCNC(=O)CC12CCOCC2 C12(C(CNC(=O)COc3ccccc3)NC(C3CCCO3)=O)CCC(CC1)C2 c1(C(C(=O)NCc2ccnn2C)N(CCCSC)C)cc(Cl)ncc1Br N1(C(c2c(CC)onc2)=O)CCC(C2(O)CCN(C(=O)C(C)(C)C)CC2)CC1 CCC(C(=O)N1CC2CCC(C1)N2C(=O)C(O)C1CC1)C(C)(C)CC C(=O)(CCCC(=O)NC1CCC(CCNC(C2(CCF)CCC2)=O)C1)NC(C)C C1(NCc2ccc(-c3c(C)n[nH]c3C)cc2F)CCNC2(CCC2)C1 c1(N2C(c3scc(C)n3)CCC2)cc(F)c(NC(=O)NC(C)C)c(F)c1 N1(C(CN2C(C)CC2)=O)CC2C(CNC(=O)C=Cc3ccc(C(N)=O)o3)C2C1 Cc1nc2c(C(=O)NC(c3ccccc3)Cc3ncc[nH]3)ccnc2[nH]1 CCS(=O)(=O)C=CC(=O)NCCCCC1CN(c2ncc(C#N)cc2F)C1 c12ccnc(n1)N2.N1(C(C2CC(OCCOCC)C2)=O)CCC(OC)CC1.C(=O)OC n1(CCC)ncc(C(=O)NC(C)(C)C(C)NC(c2cn(C)nc2Cl)=O)c1C c1(C(N2CCC(CNC(CNC=O)=O)C2)=O)cc(NC(N)=O)ccc1Cl N1(C(c2scc(COC)c2)=O)CCC(CCN(C)C(C2(F)CCOC2C)=O)CC1 c1(NC(N2CC(O)C=C(C)C2)=O)cc2c(C)cccn2c1 c1(N2CCC(CCOC)(NC(C(CC)n3ccnc3)=O)C2)nc2cccnc2s1 c1(OC)ncnc(OC)c1C(=O)NC1CC(NC(c2cc(C)c(CO)cn2)=O)C1 Cc1nc2c(C(=O)NC(CO)C(C)NC(=O)CCC(C)C)ccnc2[nH]1 CC(C)C(O)C(=O)NCCCC(C)NC(=O)CC1CC2(CC2)CO1 Cc1cc(C(N2CCCC3C2CCCN3C(=O)C=C(Cl)Cl)=O)c(N)c([N+](=O)[O-])c1 CN1CCCC1C=CC(=O)NC1CC(O)(CNC(c2nnn(C)c2C(F)F)=O)C1 C(=O)(C(F)Cc1ccccc1)N(C(=O)CN1CCC1)C1CCC1 N1(C(c2c(C)nsc2N)=O)CCC2(C1)CN(C(=O)COCCCF)C2 c1(OC)cc(NCC2N(C(=O)OC(C)(C)C)CCCCC2)nc(C(F)(F)F)n1 C1(CCNC(C(CCOC)C)=O)CCCN(C(c2ncn(C(C)C)n2)=O)CC1 c1(CC)onc(C(N2CC3C(C(=O)NCC4CC(n5cnnc5)C4)C3C2)=O)c1C C(=O)(C#CC1CCCCC1)N1CC2N(C(CCCCCCC)=O)C(CC2)C1 N1(C(c2c(C)nc(C)o2)=O)CCC(C(=O)NC2CCCC2CN(C)C)CC1(C)C C1(CNC(C(C)=CC2CC2)=O)CC(C)CN(C(=O)Cc2ccnc(C)c2)C1 N1(C(CCN(C)CCO)=O)CC2(C1)C(NC(C1CC3CC3C1)=O)CCS2(=O)=O c1(C(=O)NC(CC)(C)CNC(C2CCCN2C)=O)cnccc1Cl N1(C(C2(C#N)CCCOC2)=O)CCC(NC(=O)C=CC2CCC2)C(CO)CC1 c1(CNC(=O)NC2C3CCCC23)ccnc(-c2ccccc2)n1 N1(C(C2(F)CCN(C(c3ccnc(O)c3F)=O)C2)=O)CCCN(CC)C(=O)C1 c1(OCC(=O)N(CCCCCNC(=O)CNS(C)(=O)=O)C)cccc(F)n1 C1(CCN(C(=O)COC2CC=CC2)C)CCN(C(C2CCCCC2O)=O)CC1 C1(CC)CN(C(C23COC(CCO2)C3)=O)CCN1C(=O)Cc1ccoc1C N1(C(CCc2n(C)cnc2)=O)CC(O)CC1C(=O)NCCc1cccc(F)c1 N1(CCCOCC)CCC(C(C)NC(=O)C(C2CCCC2)OC)CC1 c1(OCC)cccc(C(=O)NC2CC(O)CN(C(=O)CCC=C(C)C)C2)c1N c1(C(=O)NC2C(CNC(c3c(Br)cn(CC)n3)=O)C2)cccc2[nH]ncc12 N1(C(C2CCC(NC(c3nc(C)sc3)=O)C2)=O)CCN2CCCC2C1 c1(C(N2C(C(C)(C)NC(CCC3CC(OC)C3)=O)CCC2)=O)ccc(N)cc1 C1(C(C)C)CN(C(c2cnn(C)c2)=O)CCCN1C(c1cnc(O)c(F)c1)=O C1(C(=O)NC2CCN(C(N)=O)CC2)CCN(C(c2nsnc2O)=O)CCO1 c1(NC(C)=O)ccnc(CC(=O)N(C)C)c1 C1(NC(C(C(C)C)C)=O)CN(C(=O)CC2(c3ccccc3)COC2)CC1(C)C C1(OC)CN(C(C2(S(N)(=O)=O)CC2)=O)CC1NC(c1coc(C)n1)=O c1(C(=O)NCC(=C)CCNC(C2(C)CCOC2)=O)cc(Br)cc(Cl)c1F C1(NC(c2cncc(N(C)C)c2)=O)CC1C1CCN(C(C2(CCO)CC2)=O)CC1 C(=O)(C(C(=O)NC1(CO)CN(C(=O)Cc2ncc(C)s2)C1)OOC)OCC.N C1(CNC(C(C(C)(C)C)OC)=O)CC2CCC(C1)N2C(=O)C(C)(C)c1cncs1 N1(C(c2cccc(CC)c2)=O)CCC(CNC(=O)Cn2ccccc2=O)C(C)C1 CCC(CC(=O)N1CCN(C(=O)Cc2cnns2)CC1C(C)C)CC(F)(F)F C12(NC(C(c3cccc(Cl)c3)CC)=O)CCCC1N(C(=O)CCC(N)=O)CC2 N1(C(C)=O)CCc2c(NC(c3cc(-n4nnnc4O)cc(F)c3)=O)cccc2C1 N1(C(=O)NCc2ccc(O)nc2)CCC(O)C(O)C1 c1(C(N2C3CN(C(C(C)=CC4CC4)=O)CC2C3)=O)cc(C)cc([N+](=O)[O-])c1 C(=O)(C(CO)NC(=O)CCOCC(C)NC(C1CCCOC1)=O)OCC c1(OC)cc(Cl)ccc1C(=O)NCCCOCCNC(=O)Cc1oc(C)nc1C c1(C(N2C(C)CNCC2)=O)ccc(S(=O)(=O)N2CCC3(CC(F)C3)C2)cc1 C1(CNC(C23CC(CCC)(C2)C3)=O)(CO)CCN(C(=O)CC(C)SC)CC1 Cc1ccc(-n2nnnc2C(CCCN(C)C)NC2CCC3(CC2)CC3)c(C)c1 CCCCCC(O)CC(=O)OC.N12CCOC(CC1)C(=O)NOC1CC(C1)C2=O C1(C)(CNC(CCOCCN(C(c2ccc(CC)o2)=O)C)=O)CC=CCC1 CCC(C)CCCCC(=O)N1CCCCNC(C(C)OC)CC(=O)N(C)C(C)C1 c1(SC)cc(N2CCCC(CNC(C3(C(F)F)CC3)=O)CC2)nc(SC)n1 c1(C(=O)NC(C)CCCNC(c2ccoc2)=O)ccnc2ccccc12 C1(C(=O)NC2C(C)(C(F)F)C2)(NC(c2ccc(CCF)cc2)=O)CC(F)(F)C1 c1(-c2onc(-c3cc(C)cc(C)c3)n2)cnn2c1CCCC2 Cc1ccc(C(N2CC(NC(=O)C(C)(C)c3cnc[nH]3)CC(C)C2)=O)c(O)c1C Cc1nc(C(=O)NOCC(=O)NC2(Nc3ccccc3)CCSC2)co1 C1(C(=O)NCCN(CC(C)O)C(c2ccc(Cl)[nH]2)=O)CCCCC1 N1(C(C2C(C=C)C2)=O)CC(NC(=O)C(c2ccc(CC)cc2)(F)F)CC1(C)C c1(CC(=O)N(C)CC2N(C(C(CC)=CC)=O)CCOC2)cccc(C)c1Cl C1(NC(c2cc(C(C)=O)[nH]n2)=O)CC(C)CN(C(C2CC3CCC(C2)S3)=O)C1 c1(COC)cc(C(=O)N(CC(C)NC(=O)C(n2ccc(Br)n2)C)C)no1 c1(C(=O)NCC2C(NC(=O)CSc3n[nH]c(O)n3)CC2)ccc(Br)cc1F C(=O)(C(F)(F)C1=CCOCC1)NCC1(O)CN(C(C=COCC)=O)C1 c1(C(=O)NC2CCC(C(=O)NCCC)C2)c(-c2ccccc2)nn2ccccc12 c1(C(=O)NCC(c2ccccc2)CNC(C=C(C)C2CC2)=O)ccnnc1O CC1CN(C(=O)C=Cc2ccc(Cl)cc2F)CCCN1C(=O)C(CO)N(C)C N1(C(C2N=C(C)SC2)=O)CCC2(CCN(C(=O)CN3CC4CC4C3)C2)C1 N1(C(=O)Cc2cncnc2)CC2CCCC(C1)N2C(c1ccc(Br)cc1CO)=O C1(CNC(C(CC)N(C)C)=O)CCN(C(=O)C(F)(F)C2(OC)CC2)CC1 c1(C(N2CCN(C(CC=C=C)=O)C3C2C3)=O)cnc2c(c1)CCCO2 N1(C(C2(CC)CC2)=O)CC(C2CCCN(C(=O)C(C)SC(C)C)C2)C1 C(N=c1nn[nH]n1C)C1(F)CC(NC(C(c2ccc(Cl)s2)C)=O)C1 N1(C(c2c(C)c(=O)cc[nH]2)=O)CCC(C)(C)CC1C(=O)NCCC12CCCC1C2 N1(C(C(C)=C(C)C)=O)CCN(C(c2cc(C)[nH]n2)=O)CC1c1nccn1C c1(CC(=O)NCC(C(C)C)NC(CC(CC)C2CC2)=O)ccc2ncccc2c1 N1(C(CCCCCOC)=O)CC2CC(NC(=O)C(n3nc(C)cc3C)C)C(C2)C1 c1(C(=O)NCC(CO)NC(C2(OCC)CCCC2)=O)cccc2c1NCC2 CN1C(=O)CCCC1C(=O)NCC1CN(C(c2ccc(CO)nc2)=O)CC1(C)C N1(CCOCC)CC(C(=O)N(C)CCN(C)C(c2sccc2C)=O)CC1=O C1(Cc2n(C3OCCC(C)C3)nc(C(=O)NC)n2)COc2ccccc2O1 c1(C(N(CCNC(C(C2CCC2)OC)=O)C)=O)csnc1C c1(C(N2CC(NC(C3(OC)CCCOC3)=O)C2)=O)ccc(C)c(F)c1N C(=O)(CCC(=O)NCC1CCN(C(=O)CC2C(C)(C)C2(C)C)C1)N(C(C)C)C C(=O)(C1=CCS(=O)(=O)C1)NCC1N(C(c2nn(CC)nc2C)=O)CCC1C C(CC)(C(=O)NC(C)C(CO)NC(c1ccc(C2CC2)s1)=O)=CC C(=O)(C(O)C(F)(F)F)N1CCN(CCNC(C(C)CC2CCCC2)=O)CC1 C1(CCNC(CCC)=O)CSCCN1Cc1cc(-c2cccs2)[nH]n1.C1CC1 c1(N2CC(OC)C3(C2)CC3)nc2c(c(=NCC3(C4CCCO4)CCC3)[nH]1)CCC2 CC(C)C(F)(F)CC(=O)N(C)CCOCCN(C(=O)CC1CC=CCN1C)C Cc1cc(C(=O)NC2CCN(C(=O)Cc3ccc(Cl)cc3)C2)c2c(n1)CCCC2 c1(C(C)(C)C)ncc(Br)cc1C(=O)NCC1CCN1C(c1ccc(O)cn1)=O c1(C(N2CC3(COC)CC2(CNC(C2(F)CC2)=O)C3)=O)cc(F)c(F)c(F)c1F c1(NC2(c3n(CCSC)nnn3)CCCSCC2)ccc2[nH]ccc2c1 C(CC(=O)NCC1N(C(=O)Cc2csc(=N)[nH]2)CCCC1(C)C)(C(F)(F)F)OC c1(C(C)=O)cn(C)nc1C(=O)NC1COCCC1NC(=O)C(C)c1cncs1 N1(C(c2ccc(C(C)=O)cc2)=O)CCC(C)(NC(=O)C(O)CC2CC2)CC1 CC1CCCCC1CCNC(C1CN(C(=O)Cc2ccccc2F)CCO1)=O C(CCS(C)(=O)=O)(C(=O)NCC(C)CNC(=O)CN(C)C)OC c1(C(=O)NC2C(NC(c3cn(C)nn3)=O)CCC2)cccc2c1CCCC2=O c1(CNC(C#C)C(C)CC)sc(S(N)(=O)=O)c(OC)c1OC C1(NC(Cc2nc(C(C)C)sc2)=O)CC2(C1)CN(C(=O)C(F)CC1CCOC1)C2 C(CC(=O)N1CC(C)CC(O)C1)(C(F)(F)F)NC(C(CCC)C)=O CC(CNC(c1n[nH]c(O)n1)=O)CN=c1cc(C(C)(C)C)nc(Cl)[nH]1 C=C=CC(C)C(=O)N1CCN(C(=O)Cn2cnc(-c3nc(C)no3)c2)CC1 N1(C(c2occ(C(N)=O)c2)=O)CCC(O)(C2(NC(=O)Cc3ccsc3)CC2)CC1 CCC(CC)(C(=O)N(C)CCOCCNC(C1CC2CCCC2C1)=O)OC c1(OC(C)C)ccc(CNC(=O)Nc2cc(O)n[nH]2)cc1 Cc1cccc(C)c1NC(=O)C(C(C)CC1CC1)N(C)C(c1ccccn1)C CCC(F)C(=O)NCC1CCC1NC(=O)C(C)(C)c1ccccc1 CCC(CCC(=O)NC1CC(=O)NC1=O)NC(c1sc(F)cc1C)=O c1(CNC(=O)CN(C(=O)Cc2ccsn2)C2CC2)ccc(O)c(F)c1 N1(CCCC=C)CCC2(CC1)CC2(C)C(N1CCNC(=O)C1)=O N1(C(c2c(C)ncs2)=O)CC2CC1CCN2C(c1cnn(C(F)F)c1)=O c1(C(N2CC(N(C)C(c3cnc(Cl)s3)=O)C(C)(C)C2)=O)ccc(S(N)(=O)=O)o1 C(C)(C)(C(=O)NCC1(F)CN(C(C2CCCO2)=O)C1)OC(C)=O C(=O)(CCCCCC(=O)NCCCC(C)(C)NC(=O)CCCC1CC1)OC c1(C(=O)NC2C=CC(C(=O)NCc3c(C)nn[nH]3)C2)c[nH]c2cnccc12 N1(C(c2nc(C)nn2C)=O)CCCC2C1CCN2C(C1CCCCN1N=O)=O N1(C(C(C#C)(C)C)=O)CCC2CN(C(c3c(C(F)(F)F)cccc3F)=O)CC2C1 Cc1ccn(CC(=O)NCC2(O)CN(C(=O)Cc3ccccn3)C2)c(=O)c1 C12(NC(C(CCC#C)O)=O)CC(C)(C1)OC21CN(C(=O)C(CC)SC)C1 OC1CCNCCC1[SH]=CCSc1ccc(Br)cn1 Cc1ccc(C(F)CNC2(CNc3ccc(C(=O)C(C)C)cc3)CNC2)cc1C C(C1COCc2ccccc21)NC(=NCC=C)NC1CC(OC(F)F)C1 c1(C(N(CC(CNC(C(C)(C2CC2)OC)=O)C)C)=O)cc2cc(N)ccc2s1 N1(C(C2(SC)CCC2)=O)CCC2(CC(NC(c3ccnc(C(C)C)n3)=O)CO2)C1 C(=O)(C(C)(F)C(=O)NC1CCC(CNC(c2scnc2C(C)C)=O)C1)OC c1(C(=O)NCC(CO)NC(=O)Cc2c[nH]nc2O)nn(CC(F)(F)F)cc1Cl N1(C(C=CCC)=O)CCC2(COCC(CNC(=O)CCC3CCCCCC3)O2)C1 C(=O)(C(CCC(C)C)NC(=O)CC(C)C(F)(F)F)N(C)Cc1ccc(C)o1 C1(C(=O)NC2(CNC(=O)C(C)Cn3ccnc3)CC(OC)C2)CCCCCCC1 c1(O)ccccc1C.C12COCC1NC(=O)C1CC(C)(C1)C(=O)N2.C1(OC)(C)CC1 c1(CC)nc(C)c(CC(=O)NCC(O)CNC(c2cn(C)cn2)=O)c(C)n1 N1(C(C(C)OCCOCC)=O)CCC(C)(CNC(C2CC3CC2CC3O)=O)CC1 C(CC(C)C(F)F)NC(C1C(CNC(c2c(C)snn2)=O)OCC1)=O c1(C(=O)NCC2CC(NC(CC=C)=O)C2)nnn(C2CC2)c1C(F)F C(C(C)(C(=O)NCC(O)(CO)CO)NC(=O)Cn1cnnc1)SC N1(C(c2cc(CC)[nH]n2)=O)CCC(CC(=O)NCC2CC2(C)C)CC1 c1(C(=O)NC2CN(C(C(CC(C)C)OC)=O)C(C)C2)cc2c(cc1F)NCCC2 C(=O)(C(C)(C)C(=O)N(C)C)NCC(CCC)NC(c1cnn(C(C)C)c1F)=O n1(CC(=O)NC2CN(C(COCC=C)=O)C(CO)C2)ncc(C)cc1=O Fc1cc(Cl)c(Cl)cc1-c1noc(C2CC(c3cncc(Br)c3)C2C(F)(F)F)n1 C1(C)(CCNC(CNC(=O)OC)=O)CCN(C(=O)C=C2CCN(C)CC2)C1 CCCCCCC(=O)NCC(C)CNC(c1ccc(F)cc1NS(C)(=O)=O)=O C1(CC(N2CC(NC(c3n(CC)ncc3)=O)C2)=O)CCCC2(CC2)C1 c1(C(=O)NOC2COC2)c(-c2ccccc2)nn2ccccc12 N1(C(C(C)O)=O)CC2CN(C(=O)CCn3cncn3)C2C1 c1(C(N2CC(OCC)C(CNC(C3CC3(C)C)=O)C2)=O)ccc([N+](=O)[O-])c(Cl)c1 C1(CNC(C2(CCCC)CC2)=O)CCCCC1NC(C1(SC)CC1)=O c1(C(C)=O)cncc(C(N2CSCC2C(N2CCC(n3ccnc3)C2)=O)=O)c1 c1(CNC(N2CC3(C2)CC3(F)Br)=O)ccc2nccn2c1 c1(C(=O)NC23CC(NC(C(CC=C)C)=O)(C2)C3)ccc(OC(C)=O)c(OC)c1 CCC(CC)(CC)C(=O)N1CC(NC(=O)CS(=O)(=O)CC)C(C)C1 c1(C(=O)NCC(C)NC(C(CC(CC)C)C)=O)cn2c(n1)C(C)CCC2 C1(CNC(C2C(OCC)C2)=O)CCCN(C(=O)CN(C2CCSC2)C)CC1 c1(C(=O)NCCCCC(C)NC(c2nc(OC)c(C)s2)=O)cc(N)c(O)c(F)c1 c1(C(=O)NC2CCN(C(C3CCNC3=O)=O)CC2F)nc2ccccc2[nH]1 C(=O)(C(C)CCCC(C)C)N1CCC(C(=O)NC(CC#C)C)C1(C)C C(CO)(C(=O)NC(CC1CCCC1)C(=O)NCCOC(F)F)OC N1(C(CCOCCOCC)=O)CCC2(CCCN(C(=O)CN(C)CC)C2)CC1 O=C(CC(F)(F)Br)NCC(CO)NC(c1cc(C2CCOC2)[nH]n1)=O c1(C(=O)NCC#CC(=O)N(C)Cc2n(CC)cnn2)ccnnc1C CCC(C)CCC(=O)N1CC2CC(N(C(=O)CCc3cnn(C)c3C)C)C1C2 c1(C(N2C(C)CC(CNC(C=Cc3ccc(C)s3)=O)C2)=O)cnc2[nH]cnc2c1 c1(C(C(N2CC(CCNC(CCCCOC)=O)C(C)C2)=O)=O)ccc(F)c(Cl)c1 c1(C(N(CCNC(C2CCCC(OC)C2)=O)C(C)C)=O)cncn(C)c1=O C1(n2cc(CCCNC(c3nn(C)c(C(N)=O)c3)=O)nn2)CCCC(F)(F)CC1 C1(C)(C(=O)OC)CC(OC)CN1C(=O)CCc1ccncc1 C12(C(=O)NCCCCCCNC(c3ccc(C#N)cn3)=O)CCCC(=O)N1CCC2 c1(C(N(C2CCCC(N(C)C(c3cc(=O)cc[nH]3)=O)C2)C)=O)cc(N)cc(F)c1 n1(CC(=O)NC2CCN(C(C(C)(C)CF)=O)C2)sc2ccccc2c1=O C1(C(N(C)CC2CCCN(C(c3csnn3)=O)C2)=O)CCCNS1(=O)=O CC1CN(C(c2ccc[n+]([O-])c2)=O)CC1CC(=O)NC1CCN(C2CC2)C1=O C1(C(=O)Nc2ncc(C#N)s2)CN(Cc2cccc(-c3ccco3)n2)CCC1O c1(C(=O)NCCOC2CN(C(C3(CC)COC3)=O)C2)cc2ccccc2n1C Cc1ccc(C(=O)NCC2(C)CCCN2C(=O)C(C)S(N)(=O)=O)c(C)c1 C=CCCC(C(=O)NC1(CO)CN(C(c2ncn(CC)n2)=O)C1)c1ccccc1 c1(C(C)C)cccc(-n2nc(C3CC=CCC3)nc2C2C(C)C2(F)F)c1 CC1CC(=O)NCC1C(=O)NCCCCCNC(c1cscc1C(N)=O)=O C1(CC(=O)NC2CCN(C)C2=O)CC(C)(C)CN1C(=O)Cc1csnn1 N1(C(c2c(CCC)[nH]cc2)=O)C(C(=O)NCC(C(C)CC)OC)CC2CC12 CCC(C)CC(=O)NCC(CC(=O)N1CCC(F)C1)NCc1cccnc1 c1(OC)cc(C(C)Nc2cc(NCC3OCCC3(C)C)ncn2)ccn1 c1(OC)ccc2cc(C(=O)NCCN(C(=O)C=CCO)C)c(Cl)nc2c1 C1(C(=O)NCCN2CCNC2=O)CC12CCN(C(=O)CC1COCC1O)C2 C1(CNC(Cn2c(C)ncc2)=O)CCC(C)(C)CN1C(=O)CC1COC(=O)N1 CC1(C)Cc2cc(Br)ccc2C1NC1C(C)(C)C1(C)C N1(C(=O)NC2CCCN(c3cccnc3)C2)CC2(CCSCC2)C1 Cc1cc(C)c(NC(=O)CC2CCCCC2NC(=O)COCCCN=[N+]=[N-])cn1 N1(C(C2N(CC)CCOC2)=O)CC2(CCC2NC(=O)CSc2n[nH]c(O)n2)C1 c1(C(=O)NC2CCCC(O)C2)ncc(C(=O)NCCNC(C2CCCC2)=O)cn1 Cc1cc(C(=O)NC2CC2NC(=O)CC23CCCC2C3)no1 Cc1cc(NCc2ncoc2-c2ccccc2)c(F)cc1[N+](=O)[O-] C=C1CCN(C(=O)C=CC(C)(C)SC)C(C(=O)NCCC(C)(C)COC)C1 c1(C(=O)NCC2CC(C)SCC2)cnc2sc(Br)cn12 c1(C(N2CC(C(C)NC(Cc3c(OC)cccc3)=O)C2)=O)ccc(=O)n(C)c1 Cc1ncc(N)cc1C(=O)NCC(C1CCOC1)NC(c1csnn1)=O CCCCC(F)C(=O)NC(CCC)C(=O)NCCC(=O)N(CC)CC C1(CN(C(CN(C)C(=O)OC(C)(C)C)=O)C2CC2)CCCN1C(=O)Cn1cccn1 C(=O)(CCN=[N+]=[N-])N(C(C(=O)NCCCN1CCOCC1)C1CC1)C N1(C(c2ccc(NC(C)=O)c(F)c2)=O)CCCCC(C(F)F)C1 S(=O)(=O)(CCc1cnn(CC(F)(F)F)c1)N(C)C(C1CC(CF)C1)=O Cn1cnn(CC(=O)NCCCNC(C2CC2C(F)F)=O)c1=O c1(-c2scc(NC(C(C)N(c3cnc(Cl)s3)C(C)=O)=O)n2)cc(O)nc(O)n1 N1(C(C(C(C)C)CNC(C23CC2CNC3=O)=O)=O)CCC2CC1C(=O)O2 CC1CCOCCN1N1CCCC(Oc2ccc(F)cc2)C1 C12(NC(c3nc(OC)oc3)=O)CCC(C(=O)NC3C(CCOC)C3)(CC1)C2 C1(NC(c2c(C)c[nH]n2)=O)CN(C(c2cncc([N+](=O)[O-])c2)=O)CC12CCCC2 C1(C(=O)Nc2cc(O)nc(CO)n2)CC12CCN(Cc1cccnc1O)CC2 C(C(=O)N1OC2C=CC1CC2)N(CC#C)C(c1ccc(F)c(F)c1)=O C1(CNCC(=O)NC2CC(OCC(c3ccccc3)C)C2)CCC2(CCC2)O1 c1(CNCC(CNC(C2CC(=O)C2)=O)O)cccc(Cl)n1 N1(C(=O)CCC2CC2)CC(CNC(C2C3C4CCC(C4)C23)=O)C2(CC2)C1 C(=O)(CC(C(C)C)C(C)C)N(CC(CNC(C(CC(C)C)OC)=O)C)C c1(C(=O)NC2(C)CCN(C(c3c(COC)noc3)=O)C2)ccc(N)c(SC)c1 c1(Cn2cc(C(C(N3CCOCC3)=O)N3CCCC3)nn2)cnn2c1CCC2 c1(N2CCC(N(C)C(c3cn(CC4CCCCO4)nn3)=O)C2)ncnc(O)c1Br C(CC(C)C)(C(=O)NCCc1nncs1)NC(C(CC)OCC)=O N1(C(c2ccn(C(F)F)n2)=O)CC2CN(C(c3ncccc3Br)=O)CC2C1 CC1(C)CCC(C(N2CCCC(O)C2)=O)CN1C(=O)CCC1OCCO1 CC1CC2(CCN(C(=O)CCCN3CCCC3)CC2)CN1C(C12CCC1C2)=O C1(C(=O)Nc2cccc(NC(c3n(CC)ncn3)=O)c2)CC12CC(C)(C)C2 Cc1cc2[nH]c(C(=O)NCC3CC(C(=O)NC4COCC4CO)=NO3)cc2o1 C(CN=c1[nH]c(=NCCNC2CCOCC2)[nH]c2c1CSC2)c1n[nH]c(=N)s1 C1C(C)(CO)CN1.N1(c2c(C)ccs2)C(=O)CCC1C(=O)O N1(C(c2n(C)nnc2)=O)CCC(O)(CCNC(=O)CCOCC2CCCO2)C1 Cc1nc(=NCC(CC(C)C)NC(=O)CCC2CCCC2)s[nH]1 CC1CC(F)(F)CN1C(=O)COC1CCN(C(C2CC2c2cccnc2)=O)C1 CCC(C)C(O)C(=O)N1CCCC1CN(C(=O)C(c1ccc(C)s1)C)C1CC1 c1(C(=O)NCC2CN(C(C3C(=C)CC3)=O)CC23CC3)cc2cnccc2cc1F CC1CN(N2CCCCC2c2ccccc2C(F)(F)F)C1 c1(C(N2CCCOC(CC)C2)C(=O)NCCCSCC)cc(F)c(F)c(F)c1F Cc1cc(C(F)(F)F)nc(NC2CC(F)CN(Cc3ccc(Cl)cc3C)C2)n1 Cc1nc(C(C)C)ccc1C(=O)NCC12CCC1CN(C(c1cccc(N)n1)=O)C2 c1(C(N2CCCC2CNCc2ccc(Cl)s2)=O)ccc(Br)cn1 CN1CCN(C(C2CCC(C)(C)CC2)=O)C(C(=O)Nc2ccc(O)cc2)C1 C=C(Br)CCC(=O)N1CC2C(N(C)C(c3cc(-n4cccn4)ccn3)=O)C2C1 Cn1cc(CC(N2CCC(NC(=O)Cn3cc(C(F)F)cn3)CC2)=O)c(Cl)n1 N1(C(C(CN(C)C)(F)F)=O)CC2CCC(Nc3nc(C#N)ncc3Cl)C2C1 C1(NC(C(C)(C)OC(C)=O)=O)COCCC1NC(c1cnc(C(F)(F)F)nc1)=O N1(C(C(C)NC(N)=O)=O)CC2CCC1CN2C(c1ccc(SC2CC2)cc1)=O N1(C(C=CC(CC)=CC)=O)CCC2CCN(C(c3ccc(O)nn3)=O)CC12 c1(C(N2CCC(NC(C(CC)(C)C)=O)C2)=O)ccc(NC(C)=O)cc1O c1(NS(CC)(=O)=O)cccc(F)c1C(=O)Nc1cc(OC)cc(Br)c1 C1(C(=O)NCCC(CCNC(c2n(CC)cnn2)=O)C)CCCC(C)(C)CC1 c1(SC)cccc(C2CC(N3CC4(CCC4)C3)C2)c1 c1(C(N2CCN(C(CC(C=C)C)=O)CC2C)=O)cc(C)c(C)cc1C c1(OC)cc(CC(=O)NC23CCN(C(c4cn(C)c(C)n4)=O)CC2C3)ccc1C C1(NC(CC2CCN(C(CC3CCC(C)CO3)=O)CC2)=O)CC2CCC1N(C)C2 Cc1nc(C)n(CC(=O)N(C)CC2CC2CC(=O)NCc2cnco2)n1 C12(C(=O)NCC3CCCN(C(Cn4cc(C(C)O)nn4)=O)C3)CC3CC1C2C3O C1(C(N2CC3C(CNC(c4cc(Cl)ccn4)=O)(C3)C2)=O)CC2CCC(C1)C2 C1(C(=O)NC2CC(NC(c3c(C(=O)OC)c[nH]c3)=O)C2)COCCN1C(C)=O N1(CCCNC(=O)N(CCO)Cc2ccoc2)CCCCC1 CN1CCCC1c1cc(C(=O)NCC(CNC(=O)CCc2cnn[nH]2)CO)n[nH]1 C1(C(N(CCN(C)C(C2CC(NS(C)(=O)=O)C2)=O)C)=O)CC(C2CC2)=NO1 C1(CC(=O)NC2CC(C(C)NC(C(C)CN(C)C)=O)C2)OCCCC1(C)C C1(C(=O)NC(c2ccc(O)cc2)C(C)C)C(O)CCN1C(c1ccc(F)cc1)=O c1(NCC(CC2CC2)OC)ncccc1S(=O)(=O)NCC1C2CCCCCC12 N1(C(C(c2ccccc2)OC)=O)CCC2(CCC2)C(NC(=O)CCC2CC2)C1 CC(C)C(=O)C(=O)NC1CCOCC1C(=O)NC(C1CCCC1)C CON=C(C(=O)NCC1CCN(C(=O)CC(C)(C)O)C(C)C1)c1ccco1 C(C(CCC)C(=O)NCC1COCC(=O)N1C)NC(CC=CCCCCC)=O C=CC(C)(CC)NC(=O)C(C)(C)NC(c1ccnn1COC)=O c1(CC)c[nH]nc1C(=O)NCCCN1CCC(NC(c2cc(Cl)c[nH]2)=O)C1 c1(NC(CN(c2nnc(C)s2)C2CCCC2)=O)ccc(C(F)C(F)(F)F)cc1 n1(CCCOC)nc(-c2cccc(OC(C)C)c2)nc1C1CC1CF N1(C(c2c(C)nc(O)cc2)=O)CC(C)CN(C(C2(F)CC=CC2)=O)CC1C c1(C(C(=O)NC2COC2)N(C)Cc2c(C)noc2C)ccc(S(N)(=O)=O)s1 C(CC(C(C)(C)C)NC(=O)C(c1ccc(C)cc1)F)N(C(CSC)=O)C C1(C(=O)NCc2nc(CNC(C(C)n3ccnn3)=O)sc2)CC(=O)NC(=O)C1 C1(NC(c2cccc(OC)c2F)=O)CC2CC(NC(C3CC=CCC3)=O)CC2C1 O=C(NNc1ccnc(Cl)c1)NCCCCCCc1ccccc1 C1(NC(C2CCO2)=O)CN(C(C2CCC(C(F)(F)F)CC2)=O)CC2(CCC2)C1 N1(C(c2cc(F)c(F)c(F)c2)C(=O)NC(CC)(C)C)CCC2CC(CC)CCC12 C1(NC(C(CCOCC)NC(C2C(C#N)C2(C)C)=O)=O)CCOCC1(C)C C(C(N=[N+]=[N-])C(=O)NC1CCCCC1NC(c1cncc(Cl)c1)=O)OCC C(CC(=O)NCC(O)CNC(=O)CCCOc1ccc(C)cc1)(C(F)(F)F)OC C(CN=c1ccnc(N2CCC(n3ccnc3)C2)[nH]1)OC1CCN(C(COC)=O)C1 CN1CCCC1C1COCCN1C(c1cc2cc(Br)cc(Cl)c2[nH]1)=O C1(C(N(C(C)C)CCN(C)C(c2cc(Cl)n(C)n2)=O)=O)CCN(C)C(=O)C1 C(=O)(C1=CC2(CCOC2)C1)NCC(CCCC)NC(CCCC#C)=O C1(C(N(C)Cc2nnc(CC)o2)=O)CCCN1NC(=O)COCCC(C)C n1(CC)ccc(C(c2nnnn2-c2ccccc2)NC2CC(CF)C2)n1 CCC(C)(C)C(C)CC(=O)NCC1CC(C)(C)CN1C(=O)CCc1ccco1 C1CC(=O)N1CCO.C1(C(N(CC(N)=O)C)=O)(CCF)CC1 C1(C(N(CCCOCCNC(c2c(CC)cco2)=O)C)=O)CCCCS1(=O)=O CC(C)(C)C(C(=O)NCC(O)C1(Cl)CC1)NC(c1cn[nH]c1)=O C1(C(=O)NCCC(C)N(C)C(C2CCCO2)=O)CCN(C(N)=O)CC1 C1(NC(c2ccc(CC)o2)=O)CCCCC1C(=O)NC1(CCOC)CCC1 c1(OC)ccc(CC(=O)N(C)CC2CN(C(c3c(C)nn(C)c3C)=O)C2)cc1O c1(C(N2C3CC(NC(c4cc(C(F)(F)F)n[nH]4)=O)C(C3)C2)=O)ccc(Cl)cc1F C1(NC(C2N(C(=O)OCC)CCC2)=O)CN(C(C2C3CCCC23)=O)CC2(CCC2)C1 c1(C(=O)NCC(C(C)C)NC(=O)CN(C2CCC2)C)c(F)c(F)c(F)c(F)c1F c1(C(N2CC(C(C)NC(c3ccc(C)cc3Br)=O)C2)=O)cc(F)c(C)cc1N C(=O)(C1CC(NCc2nnnn2CSc2ccccc2)c2ccccc21)OC N1(C(CC=CC=C)=O)CCCC(N(C(=O)CCOCC(C)(C)C)C)CC1 Cc1nn(C)c(Cl)c1C(=O)NC1CC(O)CN(C(=O)Cc2cc(Cl)cc(Cl)c2)C1 Cn1nccc1CCNC(=O)CCC1(NC(C2CCC2C#N)=O)CCC1 C12(NC(c3sc(C)c(C)c3C)=O)CCCN(C(=O)C(N)=O)CC1C2 C(CC(C(=O)NCCCCC1CC1C)NC(C1CCS1(=O)=O)=O)OC c1(NC)ccc(C(=O)NC2CCC2NC(=O)C(c2c(C)cccc2C)O)cc1F C12(CNC(C(C)(CO)OC)=O)CN(C(c3cncnc3C)=O)CC1(C(F)(F)F)C2 Cc1cc[nH]c1C(=O)NCCC1CCC(NC(=O)CSc2n[nH]c(O)n2)C1 N1(C(COC)=O)CC2CCC2(C(=O)NCc2cc(C(N)=O)co2)C1 C1(C2CCC2)(CNC2CCN(C(C(C)C)=O)C2)CCNCC1 N1(C(C(CC)N(C)C(c2cccnc2N)=O)=O)CCOC(CNCC)C1 c1(C(=O)NCC2N(c3nnc(C)s3)CCC2)ccc2c(c1)CN(C)CC2 C1(C)(CNC(c2cnc(CC)[nH]2)=O)CCC(NC(c2cnc(Cl)s2)=O)C1 N1(C(c2ncn(CC(C)C)n2)=O)CC(C2CN(C(c3coc(C4CC4)n3)=O)C2)C1 c1(C(=O)NC2(C)CCN(C(CN(C3CCC3)C)=O)CC2)nc2ncccn2n1 S(=O)(=O)(c1ccc2c(c1)C(=O)NC2=O)Nc1ncc(C)[nH]1 c1(C(N2CCC(CNC(c3cnc(CC(C)C)s3)=O)C2)=O)cccc2c1OCC2 C=C1CN(C(=O)OC(C)(C)C)C1C(=O)N(C)CCNC(=O)CC1CCCN1C C(C(C)(C(C)C)NC(c1cnn[nH]1)=O)NC(C(Cc1ccccc1)OC)=O c1(NC(c2nnnn2C(C)C)CCOC)nc2ccccn2c1C C1(C(N2CC(NC(C(CCSC)O)=O)C2)=O)N(C(=O)OC(C)(C)C)CCC12CC2 C=C(C)CC(C(=O)NCC(c1ccco1)O)NC(c1sccc1C)=O C12(CNC(c3cc(C)sc3)=O)CCCN(C(=O)COc3cccc(C)c3F)C1C2 C1(C(N2CC3(CN(C(C4CCCC(C)C4)=O)C3)C2)=O)Cc2ccccc2N1 CCC(CNC(c1ccc(CO)s1)c1nnnn1C1CCCC1)CCO C1(C(N(CC(CN(C)C)O)C)=O)COCCN(C(c2ccc(C#N)cn2)=O)C1 C1(NC(=O)CCn2ccnn2)CCC2(CC1)CN(C(c1cnco1)=O)CCO2 c1(NC(C(CCCNC(C)=O)O)=O)cc([N+](=O)[O-])ccc1C.C12(CC1)C(=O)N2 N1(C(C(C2(O)CN(C(c3c(C)noc3C)=O)C2)F)=O)CCCN2CCCC2C1 c1(CC(N2CC(n3cc(C(C)O)nn3)C(C)C2)=O)ccc(OC(F)(F)F)c(Cl)c1 C1(CC#C)CN(C(=O)C(C2CC2)NC(=O)C(=O)Nc2ccccc2)CCO1 c1(NCC(Cc2ccccc2)NC(c2ccc(C)[nH]2)=O)cc(O)ncn1 CC1CN2CCN1C(C(=O)NCC#CCNC(C1CCOC(=O)N1)=O)C2 N1(C(c2cc(C)oc2C)=O)C2CCCC1CC(NC(c1ccnc(C)c1N)=O)C2 c1(C(N2C(C(=O)NCCCN(CC)CC)C(C)(C)C2)=O)nc(C)ncc1Br N1(C(CCOCCCNC(c2ccc(C)nn2)=O)=O)CCCC(C)(C(C)C)CC1 c1(SC)ccc(C(=O)NC(C)C(C)NC(c2ncnc(O)c2F)=O)cc1[N+](=O)[O-] c1(C(N2CC3(CC)CC2(CNC(C2CC2(C)C)=O)C3)=O)ccc2oc(S)nc2c1 c1(C(=O)NC2CCCC(NC(c3ccc(F)s3)=O)C2)csc2ncnc(O)c12 N1(C(C(c2cccc(OC)c2)OC)=O)CCC2CC2(NC(c2ccsc2)=O)CC1 C(C)(CC)(CCNC(c1cnsn1)=O)NC(C(CC)n1nccc1C)=O C1(NC(C(C2CCC2)OC)=O)COC2(C1)CN(C(=O)COCCn1cncn1)C2 N1(C(Cc2ccc(OC)cn2)=O)CC(C)CCC1CNC(c1sc(C)cc1Cl)=O N(C(=NCC(C)C)NCc1ccnc(Oc2ccccc2)c1)CC1(CC)CCC1 C(C(=O)Nc1ccc(-n2cnnn2)cc1)(C(C)C)OCC(C)C c1(CC(C)(NC2(C(=O)OCC)CC2)SC)ccc(C(F)(F)F)c(Cl)c1 C1(C(C)C)CN(C(=O)C(F)(F)c2ccccc2)CCN1C(=O)CC1CCC2CC12 c1(CC)cncc(C(=O)NCCC(C(=O)NC(c2cncs2)C)OC)c1 Cc1cccc(C)c1C(=O)NC(C)C(=O)NC1(CNC(=O)C(C)S(C)(=O)=O)CC1 c1(N2CC(C)CC(CO)C2)nc(N2CCC(CN3CCCC3)C2)c2sccc2n1 C1(C(N(CC(C)NC(C2CSCN2C(=O)OC(C)(C)C)=O)C)=O)COCCO1 c1(OC)cc(OC)cc(CCC(=O)NC(c2ccc(NC(=O)C3CC3)cc2)C)c1 Cc1cccc2[nH]cc(C(=O)NC3(C)CN(C(=O)Cc4n[nH]c(=N)s4)C3)c12 c1(C(=O)NC(C(=O)NCCN2CCCCC2)C2CC2)ccc(O)cc1 c1(C(=O)NCC(CN(C(C(CC=C)(C)C)=O)C)O)cc2nc[nH]c2cn1 C1(OC)CC2CCC(C1)N2C(c1coc(C(C)NC(c2ccc(C)o2)=O)n1)=O O(NC(=O)CC1CC(NC(c2c[nH]cc2C2CC2)=O)C1)C(C(C)C)C C(=O)(C#CC1CCOCC1)NCC1N(C(c2ccc(OC)c(N)c2)=O)CCC1 CCC(CC)(CCNC(=O)C(SC)SC)NC(=O)CCSc1ccccn1 N1(CC2(C)N(C(=O)NCc3ncn(C)c3)CC2)CCC(OCC(F)F)CC1 C(=O)(C(C)CC1CCCCC1)NC(c1ccccc1)CNC(C1(CC)CC1)=O c1(C(=O)NC2C(F)CCN(C(CCCC(C)C)=O)C2)cc2ccccc2nc1O c1(OC)cnc(C(=O)NC(C)(C)CCNC(C2(CO)CC2(F)F)=O)nc1 CC1CN(C(C2CC3(C2)CC(F)C3)=O)CCC1NC(C1Cc2cscc2C1)=O C1(NC(c2cc(OC)ns2)=O)CN(C(=O)NC2CCCC2)CC12CC2 C(C1(O)CCc2cc(F)ccc21)NC(=O)NCC1(C#N)C(C)(C)C1C#N Cc1nc(C)c(CC(N2CCC2CNC(=O)C=CCF)=O)c(O)n1 Cc1cc(NC(N2CCCC(C)(CC(C)C)C2)=O)c(F)cc1Br CCC(C)(CC)C(=O)N1C2CCC1CN(C(C1(F)CCS(=O)(=O)C1)=O)C2 N1(C(c2ccc(OCC)cn2)C(=O)NC(C)(C)CC)CCOCC12CCC2 C#Cc1cc(C(N2CCC(O)(CNC(=O)C3=COCC3)C2)=O)ccc1C C#CC1(O)CN(C(C2N(C(C3CC3=C)=O)CCC2(C)C)=O)C1 N1(C(c2cccc(CCC(=O)Nc3cccc(OC)n3)c2)=O)CCCC(C)(F)C1 CCCCC(C(=O)NCC12CC1CN(C(=O)C(CO)N(C)C)C2)N(C)C Cn1ccc2cc(SCC(=O)N(C(CN=[N+]=[N-])C3CCCC3)C(C)(C)C)ccc12 c1(C(N(CCNC(=O)Cn2c(C)ccc2C)CC)=O)nc(C)ncc1Br CN1CCN(C(C2CCCN2C(N2CC3CC2CN3C)=O)=O)C(CO)C1 N1(C(C=CC(C)(C)NC(C(C)n2cccc2)=O)=O)CCOCC12CC2 C1(C(=O)NC(c2cc(C)[nH]n2)(C)C)C2CCN(C(c3cc(C(C)C)on3)=O)CC12 c1(NC(N2CC(O)(C(=O)OC)C2)=O)cc(Br)c(C)nc1O C(=O)(C(COC)CC(C)C)N(CC(=O)NC1(COC)CCOC1)CCOC C1(NC(c2ccnc(C(F)(F)F)c2)=O)CCN(C(c2nc(Cl)cs2)=O)CC1O C1(CNC(C(C)(C)c2cc[nH]n2)=O)CN(C(=O)Cc2n[nH]c(=N)s2)C2(CCC2)C1 CN1N=C(CC(=O)NCCCC2CCCN2C(C2CC3(CSC3)C2)=O)CC1=O C12(C(N3C(CNC(=O)C(C)(C)SC)CC(OC)C3)=O)CCCC1C2(F)F c1(C(=O)NC2CC(CNC(C=CCOCCOC)=O)C2)c[nH]c2nc(Cl)ccc12 N1(C(=O)CC2CCCN(C(c3ccc(O)cn3)=O)C2)CCC2(CCCO2)CC1 N1(C(C2CC(=O)NC2)=O)CC(NS(=O)(=O)Cc2c(Br)cncc2Br)C(F)(F)C1 C(CC(C)C)(C(=O)NC1CCN(CCNC(C2(C)CC(C)(C)C2)=O)CC1)OC C(=O)(C1=CCCSC1)NC1CC(CNC(c2ccc(=N)[nH]c2)=O)C1 N1(C(CCCC#C)=O)C(CC(=O)NC2CC3CCC2C3)C2CCCC12 CC1=NN(C)C(=O)C1CC(=O)NC(C)CCN(C)C(c1cc(Cl)cs1)=O N1(C(Cc2n(C(C)C)cnn2)=O)CC(NC(=O)CN2CCS(=O)CC2)C(C)(C)C1 C1(CC)CN(C(=O)C(O)C2CC2)CCN1C(c1ccc(C(C)(F)F)cn1)=O c1(C2C(CC)N(C(=O)NCCCNC3CC3)CCC2)ccc(F)c(C)c1F C1(NC(c2c(C)ncn2O)=O)CC2CC(C1)N(C(c1scnc1Cl)=O)C2 N1(C(CCCCCCNC(CCC(C)N(C)C)=O)=O)CC(=O)N2CCCC2C1 C1(C)(CNC(c2c(C)n(C3CC3)nc2)=O)COCCN(C(=O)C2=NOC(C)C2)C1 C1(C(=O)NCC2COCCN2C(C23CCC(F)C2CC3)=O)CCC(F)(F)CC1 c1(CC(=O)NCCC2CN(C(C3C(CC)OCC3)=O)C2)ccc(C(C)C)cc1F C(=O)(CC=CCNC(=O)C(C)c1cccs1)NC1(C(C)C)CC1 C(CC(C)CC)(C(=O)N1CCn2nccc2C1)NC(c1cncc(C#C)c1)=O c1(C(=O)NCC(CC=C)NC(=O)C(F)F)ccc(F)cn1 C(=O)(C1=NN(C)C(=O)CC1)NCC(C(=O)N(CC#CC)C(C)C)CC(C)C c1(CCC(N2C3C(OCCOC)C(C3)C2)=O)nc2cc(C)cc(C)c2[nH]1 O=C1CCC(C(=O)NCC2C3CN(c4nccc(C(F)(F)F)c4[N+](=O)[O-])CC23)=NN1 CN1CCN(C(c2cccc(N3CCCC3)n2)=O)CC1CNC(C1CCO1)=O c1(C(=O)NC2CC(NC(C34OCC(C(C)C)(C3)C4)=O)C2)ncc(Cl)cc1Cl C1(NC(C2(C)CCC(F)(F)CC2)=O)Cc2ccccc2C1NC(C1CCC1)=O C(=O)(C(C)CC(C)C(C)=O)NCCN(CC(=O)NCC(=O)NCCC)CCOC c1(SC)ccccc1C(=O)NCC1CCN(C(C2C3CCCC23)=O)C1 N1(C(C2N(C(c3cc(C)sc3N)=O)CCCCCC2)=O)CCC(C2=NOCC2)C1 C(N=c1[nH]c(Cl)ncc1Cl)C1CC(NC(c2cc3nc(C)sc3[nH]2)=O)C1 CC(C)C(CNC(=O)Cc1ccc2c(c1)CC2)C(=O)NCc1ccncc1 N1(C(C(=O)NCCSC2CC2)C2C(C(=O)OCC)C2)CC(OC)CC2CCCCC12 CCC(C)C(O)C(C)C(=O)N1CCC(NC(c2c[nH]nc2C2CC2)=O)CC1C C(C)(CCC(=O)N1CCCC1(C)CNC(=O)CC(C)c1ccco1)SC C1(C(=O)NC2CCC(NC(C(C)(F)c3ccon3)=O)C2)CCC(N=[N+]=[N-])C1 CN1CCc2nc(O)c(C(=O)NCC(O)CCNC(C3CC3C(N)=O)=O)cc2C1 C(=O)(CC(C)C(F)(F)F)N1C(CC)(CC)CC1.C123CCCC1CN(C2)C3=O C1(C(N(C(C(N2CC(O)(C(C)C)C2)=O)C2CC2)C)=O)CC2(CC2)CN1C N1(C(CC(C)C2CC2)=O)CCN(C(=O)CC2CC2)C(CO)C1 C1(NC(c2c(OC)nccc2)=O)CCCC(N=c2[nH]nc(-c3ccon3)s2)C1 c1(C(N2CC(F)(CNC(C3=CCCCC3C)=O)C2)=O)cnc2c(ncn2C)c1 C(=O)(C(CC)CC(F)F)NCCCCCCNC(c1ccc(NCC)cc1F)=O C#CCC(C(=O)N(C1CCN(C(C2(C3CC3)CC2)=O)CC1)CC(C)C)C1CC1 c1(C(=O)OC)cc2c(s1)CN(CC1(Cl)CCC1)CC2 C1(C(N2CC(CC(C)NC(=O)COCC3CCC3)C2)=O)CCOCC1(C)C N1(C(c2snc(O)c2Cl)=O)CCC(N(CCO)C(c2[nH]nnc2C2CC2)=O)CC1 C1(N(C(CCn2c(C)csc2=O)=O)C)CN(C(=O)C(F)C(F)(F)F)CC1(C)C c1(C(NOCC(=O)NC(CC#C)(C)C(=O)NCCOC)=O)ccc2cccnn12 C(=O)(C(F)(CNC(C1(O)CC1)=O)C(C)C)NC1C(C(C)C)CCC1 C1(CNC(C(c2cccc(OC)c2)O)=O)CN(C(=O)COC2CCCC2)CCC1C C=CC(CCC)CC(=O)NC1(C)CCCC1NC(c1cc(Cl)cn1CC)=O CC1CCC(CC(=O)NCC2CC2CNC(=O)Cn2ccc(C3CC3)n2)O1 C1(CCNC(C(CC)OC)=O)CCCN(C(c2cn(Cc3cccs3)cn2)=O)C1 C(=O)(CC(C)(O)C1CC1)N(C(C)C(=O)N1CC(ONCC2CC2)C1)C1CC1.C.O CON(C)C1CCN(CC2CCS(=O)(=O)C2)CC1 Cc1nc(CNC(=O)C(C2CCN(C(=O)CN3C(=O)CCC3=O)C2)C)c(C)s1 Cc1cn2c(n1)CCC(C(C(=O)NCc1nnn(C)n1)NC1CNC(=O)C13CC3)C2 C1(C(=O)NC(CN(C(C(C)=C(C)C)=O)C)C)(CF)CC1(F)F C1(NC(c2cc(Cl)ccn2)=O)COC2(CNC(C3(CO)CCNC3=O)=O)CC1C2 c1(C(N2CC=C(C#N)CC2)C(=O)NC)cnc(OCC(F)(F)F)c(Cl)c1 Cn1c(C(N2CCCCC2C2(NC(=O)C=CBr)CC2)=O)ccc1C1CCCO1 CCC1=NOC(CC(=O)NC(CO)C(=O)NCc2ccon2)C1 c1(C(=O)NCC2N(C(C3(C)CC4CC4C3)=O)CCC2)cnc2[nH]nnc2c1 c1(CC)cc(C(=O)N(CC(C)(C)CNC(=O)CC2(C)CC(F)(F)C2)C)n(C)n1 S(=O)(=O)(c1cccc(=NCC(=O)NC2CC2)[nH]1)NCC1(C)C(C)C1 N1(C(c2c(C)coc2)=O)CCC2(CCCN(C(=O)CC3CCCOCC3)C2)C1 c1(OC)ccc(CN2CCCC(C(=O)NC3CCC(F)(F)C3)CC2)c(Br)c1 c1(CN2CCC(CC(=O)CCn3c(C)ncc3)C2)nc(-c2ccccc2)nn1C C1(NC(C2C(C)C2)=O)CCC1NC(=O)CSC1(C)CCC1.C1CN1 c1(C(=O)NC2(c3cn(C(C)CO)nn3)CCCOC2)cc2n(n1)CC1(CC1)C2 C=CCCC(C(=O)N1CC(N(C)C)C(C)(C)C1)NC(C1CC2CC2C1)=O N1(C(Cc2nc(C)oc2)=O)CCC(F)CC1C(=O)NCC1(C)CCC(=O)N1 C1(NC(COC)=O)CN(C(c2cccc(C#N)c2)=O)Cc2ccnn2C1 C1(C(=O)NCC)(CCF)CCCN1C(C1CCCN1C(C)C)=O C1(C(=O)NCCCCOCC)CC(NC(C2CC2(C)C(F)F)=O)C(O)C1 C(CS(=O)(=O)CC(=O)NC(C1(NC(=O)CC2CCC(=O)N2)CC1)C)OC C1(CCC)(NC(c2cc(CSC)on2)=O)CCN(C(=O)CC(C)C)CC1 C1(CNC(c2cc(C)oc2)=O)CC(F)(F)CN1C(c1coc(C)n1)=O N1(C(CC2(OC)CC2)=O)CC(F)(F)CC1CNC(c1cnc(-c2cccs2)s1)=O C1(CC(=O)N(CCN(C(=O)CNC(=O)NC)CC)CC)CC=CCC1 N1(C(C(C2CN(C(=O)CCCc3ncco3)C2)OC)=O)CC2CCC(C1)C2C#N c1(C(N2CCC3(CCN(c4ncccn4)C3)C2)=O)cc(Br)cc2cn[nH]c12 C1(C(N)=O)(NC(=O)OCC2CC2c2ccccn2)CCOCC1.C1CC(=O)N1 N12CCC(C1C1CC1)NC(=O)C1C(CCC1)CC2=O.C1(CF)CC(CC2CC2)C1 C1(NC(c2c(OC)oc(C)n2)=O)CCN(C(=O)CC(C)c2ccncc2)C(C)C1 CC(C)C(O)C(F)(F)C(=O)N1CCC(=CCNC(C2CCC(=O)N(C)C2)=O)CC1 N1(C(C2(OC)CCOC2)=O)CCC(c2cncn2C)C1.c1(C=O)cccs1 C1(NC(CCC#C)=O)CCN(C(=O)C(O)CC(C)C)CC1F C1(C(F)(F)F)(C(c2n(CCC)nnn2)NCCCN2CCCC2=O)CCCCC1 c1(C(CNC(C2CC(O)C2)=O)NC(C(c2ccccc2)C)=O)ccc(Cl)cc1.C(C)(=O)O C1(C#N)(C(N2CCC(N(C)C3CC3)CC2)=O)CC2CC2C1.C12CN(C1)C2=O C12(C(=O)NCCCCCN(C(CC(=O)NCC#C)=O)C)CCC(CC)(C1)OC2 c1(C(N2CCC(N(c3ncccc3C(=O)C(F)(F)F)CCO)C2)=O)cccc(F)c1 C(C)(CO)(C(C)(C)O)NC(c1c(C)nc(CNC(=O)CN2CCCCC2C)o1)=O c1(C(N(CCCCCNC(c2cnc[nH]2)=O)C)=O)cc(N)c(F)c(F)c1Cl c1(CC(N2CC3CC(CNC(C4(CCC)CC4)=O)C3C2)=O)c(C)nc(O)nc1C c1(CC)ccc(Br)cc1C(=O)NCCC1CCCCN1C(=O)C=CCO C(=O)(C1COc2cc(C)c(C)cc21)N(C(c1ncccn1)(CC)C)CC(C)C c1(N)ccc(C(C)(C)C)cc1.c1(C(=O)NC2C(C(=O)NCC(C)C)C2)cscc1CO c1(CC)nonc1C(=O)N(CC(C)(C)CNC(c1cnc(C2CC2)o1)=O)CC N1(C(Cc2cc(CC)no2)=O)CC(C2(NC(=O)OC(C)(C)C)CC2)CC1CO Cc1cc2cc(C(=O)NC3CN(C(=O)Cc4ccc(F)cc4)CC3F)ccc2[nH]1 C(N=c1[nH]c(N2CCCC2c2ccc(Cl)cc2)nc2c1CSC2)c1cc(C)no1 CC(C)CCC(=O)NCCC1(NC(C2CC2(C)C)=O)CCOCC1 CC1C2CCC(C2)C1C(=O)NC1CC2(C1)CC2NC(C1CCC(C)(C)C1)=O C(CCCC(C)(C)C(=O)NNC(=O)N=CC1CCOC1)NC(C(C)S(C)(=O)=O)=O C1(C(N(CCOC)CCNC(=O)CSc2nccs2)=O)CCSCC1 c1(C(=O)NC2CCC(CNC(=O)COC(F)F)C2)cc2c(cc1Br)OCO2 C(=O)(C1=C(Cl)CCCC1)C(=O)CC1CC(O)C12CCC2.C1(N)CC2CCC1N2 C(=O)(C1=CC2C=CC1C2)NCC1CCN(C(CCc2c(C)cccn2)=O)C1(C)C c1(C(N2CC(CNC(CCC=C=C)=O)C3C2C3)=O)ccc(F)c(F)c1F C1(NC(C2(OC)CC2)=O)CCC(C)(C)CC1CNC(=O)CN1CSCCSC1 N1(C(c2cncc(C)n2)=O)CCN(C(c2ccc(C(C)(C)C)nc2)=O)C2CC12 C1(OC)CCCCC1N=c1cccc(S(=O)(=O)NCc2cncn2C)[nH]1 CN1CCOC(C(=O)NC2C3CC2N(C(=O)CSCc2cccnc2)C3)C1 CN1CCC(C(=O)NC2CCCCC2CNC(=O)Cc2ccc(O)cn2)S1(=O)=O N1(C(C=C2CCC(C)C2)=O)CCC2CN(C(=O)C(C)Cc3ccco3)C2C1 C(C1(C)CCOCC1)=CC(=O)N(CC(CC)NC(C1COCCN1CC)=O)C C12(NC(c3n(CC)ncc3)=O)CC3CC(C1)CC(CNC(=O)C(C)C(C)O)(C3)C2 c1(OCCC#C)ccc(Cn2cc(C(N3CC(C(N)=O)C3)=O)nn2)cc1.O C12(C(N3CC4C(CNC(c5c(C)cnn5C)=O)C4C3)=O)CCC(N=[N+]=[N-])(CC1)C2 C(CNC(=O)Cc1ccc(OC)cc1C)(C(C)C(C)C)NC(CCC=CC)=O C=CCC(CN1CCOCC1)C(=O)N1CCCC1c1cn(C)c(=O)cn1.C(=O)OC Cc1ccc(F)cc1C(=O)NC1(C)CC(NC(=O)CN2CCCCS2(=O)=O)C1 c1(NC(C(CCNC(CC2CC(CC)C2)=O)OC)=O)ccc(O)c(Cl)c1 N1(C(c2c(C)nn(C3CCC3)c2)=O)CC(CNC(C2CS(=O)(=O)C2)=O)C(F)(F)C1 CC1OC(=O)NC1C(=O)N(C1(C(=O)NCC23CC(CN2C)C3)CC1)C CC1CC(C(=O)OCCOc2ccc(Cn3cccn3)o2)CCC1=O C#Cc1ccc(C(=O)NC(C)(C)C(C)NC(=O)C(O)Cc2ccccc2Cl)nc1 C(=O)(CCC(=O)C(C)(C)C)N1CC(C=C)(CC(=O)Nc2ccc(C)c(CO)c2)C1 c1(C(=O)NC2CCC(CNC(=O)C=Cc3cc[nH]c3)C2)cnnc(O)c1 N(CCC=O)CCC(=O)OCC(=O)NC.OC C1(NC(c2cn(CC)nc2C)=O)CCCC12CN(C(c1sccc1COC)=O)C2 CC1CCCN(C(C2C3CCC2CC3)=O)C1CNC(=O)CN(C1CCC1)C C1(CNC(c2ccc(NC(C)=O)s2)=O)CC2CCC1N2C(=O)CCCF N1(C(CC2CCC(C)(C)CO2)=O)CC2(CC(NC(C3(O)CCCC3)=O)CO2)C1 c1(C(N(CCN(C(=O)CCC2CCC(=O)N2)C)C)=O)nc2ccccc2s1 C1(C(=O)NC(CNC(CCCCC)=O)CO)CC2(CCC2)CN1C(=O)OC(C)(C)C N1(C(C2(C)CC2Br)=O)CCC2(COC(CNC(c3c(F)cccc3F)=O)C2)C1 C1(COC(c2c(N3CC(C)OC(C)C3)cc(C(N)=O)cc2)=O)CC(F)(F)C12CCC2 c1(NC(C(C)N(C(c2c(C)n[nH]c2)=O)C)=O)ncccc1C(C)C c1(C(=O)Nc2ccc(N(C)C)nc2)ccc(F)c2occc12 C1(NC(=O)Cc2ccncc2)CCC2(CC1)CCN(C(=O)CC1CC1)CC2 c1(C(=O)Nc2cccc(NC=O)c2)ccc(CCF)cc1.C(=O)(C=C1CC1)NCO c1(C(N2CCC(NC(C3CC4(C3)CC4(F)F)=O)C(F)C2)=O)cc[nH]c2nccc1-2 C1(OC(=O)N(C)CC(F)F)(Cc2ccccc2)CC2CCC1CC2 C(=O)(C1=CC(O)CCC1)N1CCC(C(C)(C)NC(CNC(=O)OC(C)(C)C)=O)C1 C(=O)(C(CC=CC)NC(c1c[nH]c(=NC)o1)=O)NCCOCCCCC CCC(O)C(C)C(=O)NC1CC2(C1)CC(NC(=O)C(O)COC)C2 C1(CNC(Cc2ccc(CC)cc2)=O)COCCN(C(=O)Cc2cnc(C)s2)C1 c1(CCCNC(=O)COC2CN(C(c3ccccn3)=O)C2)nc(CO)n[nH]1 C1(C(N(CCOC)CCNC(C2CCN(C(C)=O)C2)=O)=O)CCc2c(ncn2C)C1 CCCC(C(=O)NCC(CCOC)NC(c1nncn1C1CC1)=O)NC(N)=O N1(C(CSc2nc(C)[nH]n2)=O)CCC2OCCN(C(c3sccc3C)=O)C2C1 Cc1nonc1S(=O)(=O)N1CCC(c2n[nH]c(=N)o2)C1 C1(CC(=O)N(CC=C)CC2CC2)CC(NC(=O)C(C2CC2)OC)C1 C(=O)(C#CC1CCCCC1)N1CCC(=CCNC(=O)Cc2csc(Cl)c2)CC1 C(C1=NOC2(COC2)C1)NC(CCc1c(-n2cc(COCC)nn2)cccc1)=O c1(OCCCC)ccccc1C(=O)C(C1CC(N)C1)=O.c1(C(=O)N)n[nH]cc1Cl C(C1CN(C(=O)C(N2CCNC2=O)C)CC1C(=O)NC(C)CCCCCO)=CC C1(NC(CCCCC#C)=O)CCCCCN(C(=O)CCC2CC2(Cl)Cl)C1 c1(COc2ccc(NC(CC(=O)OC)=O)cc2)ccc(I)c(Cl)c1 C1(C(N(C(C)CO)CC)=O)COC2(CCN(C(c3ccno3)=O)CC2)C1 C12(C(=O)OC)CCC(CN(C(C3(C)CCCC3O)=O)C1)C2 C(c1nnn(C)n1)=CC(=O)N(CCCCN(C(=O)CCCN1CCCC1)C)C Cc1cc(C)c(CNC(C2C=CCN(C(=O)C(=O)C3CCCC3)C2)=O)s1 C1(CNC(C2CCN(C(CC)=O)C2)=O)CC(F)(F)CN1C(C1CCC=CO1)=O N1(C(C(CCCC)O)=O)CCC2CN(C(=O)CCCNC(C)=O)CC2C1 N1(CC(=O)N(c2cc(C(F)F)ccc2F)C2CCOC2)CCC2(CCNC2=O)CC1 C(=O)(C(C)(CC)CCCC)N1CCC(CNC(C2CCN(CC)C2)=O)C1 C1(C(=O)NC(CCCOC)(C)C)CC(C)CN(C(c2sccc2C)=O)C1 C1(OC)CC2CC(C1)N(C(C1C3CC1N(C(c1cnnn1C)=O)C3)=O)C2 c1(CCNC(C(C)C2CCCO2)=O)ccc(CNC(=O)Cn2ccnn2)cc1 C(C(C)C(C)C(=O)NCCCOCCNC(=O)CCP(C)(C)=O)SC Nc1ccc(C(=O)NC(CNC(C2CC2c2ccccc2)=O)CO)nc1 O(NC(=O)C(C)CNC(C1(F)CCOCC1)=O)CCC C12(C(=O)NCC(C)(NC(c3cc(C4CC4)[nH]n3)=O)C3CC3)CCCC(C1)C(=O)NC2 C1(C(=O)NCC(C)(C)OCC(=O)NCCC2(CC)CC2)CCCCN1C C1(c2nnnn2C(C)C)(COC)CN(Cc2cccc(F)c2)CC1C Cc1cc(C(N2CCCCC2C(C)NC(=O)CCN2CCC2)=O)ccn1 c1(NC(C2(COC)CN(C(=O)C(C)N3CCCC3)C2)=O)cc(C)c(F)c(C)c1 C(C(NC(=O)NCCOCC1CCC1)OC1CC1)OC C1(CCNC(CS(=O)(=O)N(C)C)=O)CC2CCC(C1)N2C(=O)COc1ccsc1 C1(CC(=O)N(CCC(=O)OC)C)C2CCCC2N1C(=O)CC1CC(O)C1(C)C c1(CCC(=O)NC(C2CN(C(C3CCCN3C)=O)C2)C)ccc(F)cc1 C1(C(F)(F)F)(CC)CN(C(=O)C(=O)NC(C)CC(=O)NC)C1 N1(C(c2cc(C(C)(F)F)on2)=O)CCC2(CCCN(C(C3CC3F)=O)C2)C1 CCCCCCC(C(=O)N1CCC2C(NC(=O)CC3(OC)CC3)CC12)NC(C)=O c1(CN2C(C(=O)NCC#N)CC(O)C2)cnc2cc[nH]c2c1 N1(C(c2ccc(C(=O)OCC)o2)=O)CCC(C(=O)NC2(CO)CCOCC2)CC1 C(=O)(C(CNC(=O)Cc1ccccc1C)C(C)C)NCC(C#C)C(C)C N1(C(c2ccncc2F)C(=O)Nc2c(C)cccc2)CC2CC2C2CC12 c1(C(=O)NCC(CNC(C2(c3c(C)ccs3)CC2)=O)CO)cnc2nccn2c1 CCCC(C)(CC)C(=O)NOCC(=O)NC1CN(C(=O)OCC)C1 C1(C(N2CC(O)(CNC(C3CC(C4CCC4)C3)=O)C2)=O)CCCC1C1CC1 CCCCN=C(NCCC1(O)CCCOC1)NC(C)CC C1(C(C(=O)NCCC(C)NC(c2cc(C)nn2C2CC2)=O)C)CCC(C)(C)CC1 C1(C)(C(N2CC(OCCNC(C=CC(=O)N(C)C)=O)C2)=O)CCC(=O)NC1 C1(NC(c2cncc(C)c2)=O)CN(C(C2CS(=O)(=O)C2)=O)CC2(CCOCC2)C1 CCCC(C)(CCC)C(=O)NC1CN(C(c2ccc(F)cc2Cl)=O)CC1C1CC1 C1(C(=O)NC(COCC)C)CCN(C(=O)CSC2CC2)C12CCC2 Cc1cc(C(=O)NC2CCN(C(=O)C=CBr)CC2(C)C)cc(N)c1O N1(C(C(C)n2ccnc2)=O)CC2CCCC(C1)N2C(c1cc(Cl)on1)=O C1(C(=O)NC(C2CCOC2)CO)(SC)CN(C(=O)C(C)c2cccs2)C1 C1(N(C(=O)CC2COCCO2)C)CN(C(c2cccc(CO)c2)=O)CC12CC2 c1(OC)cc(C)c(C(=O)NCC2(Oc3cccnc3)CCN(C(=O)C)C2)cn1.OC Cc1cccc(N2CCN(C(=O)C(=O)N(CCO)CC3CC=CCC3)CC2)n1 C(=O)(C1CCCc2scnc21)N(C1CCN(C(c2cc(C)ncc2Cl)=O)CC1)C Cc1nn(C)c(Cl)c1C(=O)NC1CC(CO)N(C(C2CC23CC3)=O)C1 c1(CC(N2CCCC(Cn3cc(C4(C)CCCC4)nn3)C2)=O)cc(F)cc(F)c1 C1(OC)CN(C(=O)C=C(C)C(F)F)CC1NC(=O)C(C)CCC1CCCCC1 C(CC(C)C)(C(=O)NCCC1(NC(C2CCCC(C)(C)C2)=O)CCC1)OC N1(C(c2c(CC)cccn2)=O)CCCC(NC(C23CSCC2C3(F)F)=O)CC1 C1(NC(c2c(OC)nc(C)cc2)=O)C(C)(C)CN(C(C2CC2C)=O)CC1(C)C S(=O)(=O)(CC(=O)N1CCC(CCNC(C2CCC(OC)C2)=O)CC1)NC C(CC(=O)N1CCC(NC(c2cc(F)cc(F)c2)=O)C1(C)C)(C(C)C)OCC N1(CC(=O)NCC(CC(F)(F)F)NC(CC(C)F)=O)C(=O)c2ccccc2C1=O N1(C(CCOC(C)C)=O)CCCC(C)C1CCNC(c1cnc(O)n1C)=O c1(CC(N2CC(CNC(c3ccc(NC4CC4)cc3)=O)C2)=O)ccc(F)c(F)c1 C(=O)(CCCCCC(C)O)NC(CC(C)C)CNC(c1ccc(C(N)=O)o1)=O C1(CC(=O)N(CCC)C)C2CN(C(=O)C3CC3)CC12 N1(Nc2ccc(C)cc2-n2cc(OC)nn2)CC(C)OC2(CCC2)C1.c1(C)cn(C)nc1C c1(C(N2CCC(O)(CCNC(C3C(C)CCO3)=O)C2)=O)cc(O)nc(C2CC2)n1 CC1CCCCC1C(=O)NC(C)CNC(=O)CCc1csc(=N)[nH]1 C(=O)(C(F)(F)C(F)(F)C(F)F)NCCCCCCNC(=O)Cc1cnoc1 S(=O)(=O)(c1c(C)cccc1Cl)NC1C(C(=O)NC(C=C)C)C1 C1(CNC(CNS(CCCC)(=O)=O)=O)CN(C)CCN1C(c1cccnc1Cl)=O c1(C(=O)NC2C(C)CN(C(C3CCC(=O)N3C)=O)C2)cc2c(F)c(F)ccc2[nH]1 c1(CC(=O)N(CC(C)NC(CNC(C(CC)C)=O)=O)C)cccc(OCC)c1F c1(NC(=O)CC2CCN2C(c2nccs2)=O)csnc1-c1ccccc1 Cc1cc(C(N2CCCC2CNC(=O)CSc2cnn(C)c2)=O)on1 C(=O)(C(C(C)C)N1CCCC1=O)NCC(CNC(C(C)C)=O)F C#CCCCCC(=O)NC(C(=O)NCc1ccc(F)c(C)c1)C1(O)CCC1 C1(COC)(NC(=O)CCCF)CCN(C(c2cnn(CCC(=O)OC)c2)=O)C1 c1(C(N(CCCN(C(=O)CC2CCC2)C)C)=O)ccc2c(c1)CCC(O)C2 N1(C(C2C(C)CCC2)=O)CCCN(CCNC(c2cccnc2C(F)F)=O)CC1 Cc1cocc1C(=O)NC1CC(C(=O)NCCNC(c2ccc[nH]2)=O)C1 Cc1cccc(CC(=O)NCC(C2CC2)NC(c2conc2C)=O)c1Br Cc1cnc(C(N2CC3C(N(C)C(c4cc5n(n4)CCC5)=O)C3C2)=O)cc1C c1(N(C)Cc2cc(Cl)cc(Cl)c2F)nc(N2Cc3ncsc3C2)nc2c1CSC2 C#CCCCCC(=O)NCC(CNC(=O)CCc1cc(F)ccc1F)C(F)(F)F Cc1noc(C)c1C(C)C(=O)NC1CN(C(c2conc2C2CCC2)=O)CC1C Nc1cncc(C(=O)NCC(C2CCCC2)NC(c2c[nH]nc2F)=O)c1 Cc1ccnc(N(C(C)CCNC(C2CCCOC2c2ccco2)=O)C)n1 CCC(C(=O)N1CCC(O)(CN(C)C(c2c[nH]c3nccc-3c2)=O)C1)C(F)(F)F Cc1cc(F)cc(Cl)c1NC(C1CC(C)CN1C(=O)Cc1ccccc1I)=O C(=O)(C(C)C(=O)OC)NCCN(C(C1CCC(c2ccccc2)CC1)=O)CC c1(NC(C(C)C)=O)cc(Cl)c(C(=O)NCC(c2ccc(Cl)cc2)O)c(Cl)c1 Cc1ccnc(C)c1C(=O)NCC1(NC(=O)CCP(C)(C)=O)CCCC1 C(=O)(C(C)(C)C(F)F)NC(CCC(=O)NC(C(C)NC(C)=O)C(C)C)=O C12(CNC(C3CN(C(C)=O)C3)=O)CCCN(C(c3cnccc3Cl)=O)C1C2 N1(C(CC=C)=O)CCC2(CC1)CC(NC(=O)C(C)C(O)CCCC)C2 c1(OC)cccc(C(C)C(=O)N(CCCNC(=O)C(C)N2CC(C)C2)C)c1 c1(C(N(CCCNC(C2Cc3nncn3C2)=O)CC)=O)cc2sccc2n1C C(=O)(C(F)(F)Cc1ccccc1)NC(=O)OCC(c1nc(C)sc1)=O c1(OC)ccc2cc(-c3nc(C(C)O)nn3-c3ccc(OC(F)F)cc3)[nH]c2c1 C1(CC(N2CC(NC(c3cncc(Br)c3)=O)C2)=O)Cc2ccccc2NC1=O c1(NC(C23CCC(C(N4CC5CC5C4)=O)(CC2)CC3)=O)cccc2c1OCCO2 c1(C(=O)NCC2CCCN(C(CCC#C)=O)CC2)cc(F)c(CC)cc1F C1(CNC(CC2(C)CC2)=O)CCCN(C(c2cnc(C(F)F)s2)=O)C1 N1(C2CCCN(C(C3C(=C)C3)=O)C2)CCN(C(=O)COCC(=O)OC)CC1=O C1(CC(=O)N(C2CCCC2)CCCNC(C(COC)C)=O)CCN(C)C1=O c1(C(=O)NC2CC(C)N(C(=O)CC3=NNC(=O)C3)CC2)ccc([N+](=O)[O-])cc1O c1(C(C)C)cc(C(=O)N(CCCCNC(=O)C=C2CCN(C)C2)C)cc(O)n1 c1(SCCNc2c(C(=O)OC)cccc2)c(Cl)cc(OC)cc1Cl c1(C2C3CCCN(C3)C(=O)N2)cccc(C(F)(F)F)c1C.Cc1ncccc1Cl C1(CNC(C2(C)CN(C(c3cc(CC)sn3)=O)C2)=O)COCCOC1 C1(C(=O)NC2CC(C)(NC(=O)CCCc3cnccn3)C2)(OC)CCSC1 C#CC1(C(=O)NC2CC(O)(CNC(c3nccnc3C)=O)C2)CCOCC1 C12(C(N(CC(C)(C)C)C)=O)CC(CCO1)N(C(c1sccc1Cl)=O)C2 CC(CNC(=O)C=Cc1ccsc1)CC(=O)N1CCC1CC(N)=O C1(C(=O)NC(C)(CNC(=O)Cn2cnnn2)Cc2ccccc2)CC12CC(O)C2 N1(C(c2scc(COC)c2)=O)CC(NC(C2(C)CCC2)=O)CC12CCCCCC2 C(=O)(C(C)N(OC)C(=O)CC1C2CN(C(=O)CC3CCC=CCC3)CC12)OC c1(OC)cnc(C(N2CCC(CC(=O)Nc3c(Cl)n[nH]c3C)C2)=O)cn1 N1(C(c2cccc(C#C)c2Cl)=O)CCC2CN(C(C3CCCS3(=O)=O)=O)CCC12 c1(OC)ccc(CC(C2CC(F)(F)C2)NC(C)C(C)C)c(F)c1 N1(C(C2(OC)CCC(C)C2)=O)CCC12CN(C(c1cccc(C)c1N)=O)C2 c1(C(N(C2CN(C(c3cc(Br)cnc3F)=O)C2)C)=O)cc(F)c(Br)cc1F N1(C(CCOC)=O)CCC(C)(C(=O)NCc2ccc(N3CCCC(O)C3)cc2)C1 CCCCC(C(=O)NCc1cc(C)nn1C)NC(=O)CC1CCCCO1 C12(CNC(CC(C)(C)N(C)C)=O)CCC(CC1NC(c1nn(C)cc1Cl)=O)C2 C1(NC(c2c(OC)cccc2)=O)CCCN(C(=O)CCCc2ccc(C)s2)C1C C(=O)(C1CCCc2nncn21)N1CC(COC)(CNC(=O)C2=COCC2)C1 CC1(CNC(=O)CC2CCNC2=O)CCCN(C(C2CC(C#N)C2)=O)C1 c1(CN(C(=O)CCC2CCC2)C)ccccc1CNC(c1cncn1C(C)C)=O C(=O)(C(CC)C(=O)NC1(C)CCCN(C(c2ccn(C(C)C)n2)=O)C1)OCC CCCCC(CC(=O)NCCc1cnccn1)OCC.c1(CC=O)cnsc1 CCC(CC(=O)NCCCCCNC(c1cncc(N(C)C)c1)=O)NC(N)=O N1(C(=O)NC2C(c3onc(C)n3)C2(C)C)CCC(C2CC2)C1SC(C)(C)C C(=O)(C1=CCC2CCC1N2C(C1(CC)CCNC1=O)=O)N1CC(C(=O)OCC)C1 C1(NC(=O)CC2CSC2)CN(C(C2COCCC2(F)F)=O)CC1C1CC1 CCCCC(CC)C(=O)NC1CCCC(NC(=O)C2=CC(C)(C)C2)C1 CC(C(=O)NCC(C1CCCC1)NC(c1ccc(-n2cnnn2)cn1)=O)C(F)F C1(CNC(C(C(C)C)n2ccc(C)c2)=O)CN(C(c2cc(F)c[nH]2)=O)CC12CC2 c1(CC(=O)NC(CC)(C)CNC(=O)CCNC(=O)CO)ccc2c(c1)CCCC2 C1(C(=O)NC(CCOC)CNC(c2[nH]nnc2C2CC2)=O)CCC2(CCC2)OC1 c1(SC)cc(C)ccc1C(=O)NCC1(O)CCN(C(C2C3CCC(=O)C23)=O)CC1 C1CCCN(C(C2CC23CCC3)=O)C1.CC1(C)CC(CC(=O)NC(C)(C)C)C1 N1(C(CC2C(C)OCC2)=O)CCC2(CC2C(N2CC=CC2(C)COC)=O)C1 Cc1c(NC(=O)CC2CC(C)N(C(=O)COCC(F)(F)F)C2)cccc1F C1(F)(CSCC)CCN(C(=O)C(=O)NCc2cnn(C)c2C(=O)OC)C1 Cc1cc(CN2CCSC(C(N3CC(N4CCCCC4)C3)=O)C2)nc(O)n1 c1(NC(=O)CN2CC(C)(C)C2)cnc2[nH]cnc2c1.Cn1ncc2c1C(=O)NC2 CCCCC(C)CCC(=O)NC(C)(CSC)C(N1CC2CC(C1)C2(C)C)=O c1(OC)ccc(CC(=O)NC2(C(N)=O)CC(F)C2)cc1O.C1CC(=O)N1 c1(C(=O)NC2C(CNC(C3(C)CCCCO3)=O)COC2)ccc2cccnn12 c1(CNC2C(C)CC=CC2)ccc2nc(O)oc2c1.C12=CC=C(C=C1)C2 C1(NC(c2ccc(C(C)C)o2)=O)CN(C(=O)CC2NC(=O)NC2=O)CCC1(F)F CC(C)(C)CC(=O)NCC(c1cccc(Cl)c1)NC(=O)CN1CSCCSC1 N1(C(COCC(=O)OC)=O)CCC(C)C(NC(=O)Cc2cc(Cl)cs2)C1C N1(C(CCC)C)CC(C(=O)NCC2CCCN2C(C2CC=C(C)CC2)=O)CC1=O c1(-c2cc(C(=O)Nc3scc(C(F)(F)F)n3)n[nH]2)cc(O)c(F)c(F)c1 N1(C(c2cc(OC)cc(Cl)c2F)=O)CC(NC(C2(F)CC2)=O)CC12CCCCC2 C1(NC(CC2CC(NC(C(C(C)C)N(C)C)=O)C2(C)C)=O)CC2(CCCCC2)C1 CCCC(F)C(=O)N1CCSCC1CCNC(c1ncsc1C(C)C)=O Fc1ccc2ncnc(N3CCCC(n4ccnn4)CC3)c2c1 N1(C(C2C(CC)CN(C(C3CC=CC3)=O)C2)=O)CC2(CCC2)OCC1C CCC(C)C(O)C(=O)NC1CN(C(c2cccc(C3OCCO3)c2)=O)CC1O c1(C(=O)NCc2ncc(OC)nc2)c(C)ccc(C)c1O N1(Cc2scc(C(=O)OC)c2)CCC(F)(C(=O)Nc2ncccc2C)CC1 N1(C(C(N)=O)=O)CCC(c2ccccc2)(NC(C2(C(O)C(F)(F)F)CCC2)=O)CC1 CN1C(=O)CC(NC(C2(F)CCN(C(C3CC4(CC4)CO3)=O)CC2)=O)C1=O Cc1cc(CNCc2ccc(-c3cccc(CO)c3)cc2C(F)(F)F)ncc1Cl C1(C(C)C)CCCN(C(=O)CNC(C2CCC3(CC3)C2)=O)C1 c1(CC(=O)N(C2CN(C(C3CC(C)C3)=O)CC2O)C)ccc2[nH]ccc2c1 c1(C(N(CC(O)CNC(C2CCSC2)=O)C)=O)ccc(C#N)c([N+](=O)[O-])c1 N1(C(c2nc(-c3ccc(OCC)cc3)sc2)=O)CCc2occc2C1C(=O)O c1(OC)ccc(C)cc1C(=O)NC(CCNC(C1CCCCC1C)=O)C(C)C c1(C(=O)NC(CNC(CSC(C)C)=O)CO)cc(F)c(Br)c(F)c1N c1(C(=O)NC2(C)CCN(C(C34CC(F)(C3)C4)=O)C2)cccc(Br)c1Cl c1(N2CCC(CNC(C(C)OC)=O)C(C)C2)cnc(C#N)c(C#N)n1 C1(C(C)C)(C(N2CC(O)(CCNC(c3ccns3)=O)C2)=O)CNC(=O)C1 C1(C(N2C3(C#C)CC(C2)C3)=O)CN(C(c2cc(C)c(O)nn2)=O)CCC1(C)C C1(NC(C2(COC)CCCC2)=O)CCCC(CNC(=O)Cn2cc(Br)cn2)C1 CCCC(C)C(=O)NC1CCN(C(c2ccccc2COC)=O)C1C c1(C(=O)NCC(C)(C2CC2)NC(CCCOC)=O)cc2ccoc2cc1F N(C1c2ccccc2C2CCCC12)c1n(C)c(CC(c2ccccn2)O)nn1 c1(CNC(c2ccccc2C2CCCCN2)=O)ccnc2c(C(=O)O)cnn12 C1(C(n2cc(CO)nn2)=O)COCCN1NC(=O)CCC(O)C1CCC1 N1(C(C2(COC)CN(C(CCSC)=O)C2)=O)CCCC(C)(C)C1C C1(N(C(c2c(C)cn(C)c2)=O)C)CCC2CN(C(=O)CC3CSC3)CC12 C1(C(=O)NCC(C)CC(C)O)(CNC(c2c(CC)ocn2)=O)CCCCC1 COn1cnc(C)c1C(N1CC(NC(c2coc(C3CC3)n2)=O)CC(O)C1)=O C12(C(=O)NC(C(=O)OCC)CC)CC1CN(C(C1CC13CCCC3)=O)C2 C1(NC(=O)Cc2ccsc2)CN(Cc2ccc(-c3ccc(O)cc3)cc2)CC1O c1(C(=O)NC(CNC(=O)COc2cccnc2)CO)cn(C(F)F)nc1C(F)F Cc1c(C)c(NCC(=O)OCCCS(N)(=O)=O)c(C)c(C)c1Br C(C)(CCC(=O)NCC(CC(C)C)NC(=O)C(O)Cc1ccccc1)OCC C1(CNC(c2ccccc2)=O)CCCN1C(c1csc(C(F)F)n1)=O C(=O)(C1=NN(C)C(=O)CC1)N1CCOCC(CN(C)C(=O)C2CC2)C1 CC(CC(=O)N1C2CCC1CN(C(c1cnn(C)c1Cl)=O)C2)CC(F)(F)F C1(C(N(CCCNC(CCCC(=C)C)=O)CCO)=O)CCC2CCCCN12 C1(NC(=O)CC(C2CC2)NC(=O)CN2CCNC(=O)C2)CCC12CCCC2 C#CCC(O)C(=O)N(CC(C)C(=O)NC(CC)CCO)C c1(C(N(CCCCN(C(C=C(CCC)C)=O)C)C)=O)c[nH]nc1-c1cccs1 c1(SCCC(=O)N(C2CCC(NC(=O)Cn3nccc3F)C2)C)ccccn1 C(CC(=O)NC1CC(F)CN(C(=O)C=C2CCCCC2)C1)(C(F)(F)F)OC C1(CC)(NC(=O)CC(C)(C)O)CCN(C(=O)COC2CCOC2)CC1 CC(C)CC(CC(=O)N1CCC(CO)CC1)NC(C1(C)COC(=O)N1)=O CC(O)C(C)C(=O)NC(C)(C)CCCNC(c1cc(OC(F)F)n(C)n1)=O N1(Cc2ccc(C#C)s2)CCC2(CC1)CC2C(=O)Nc1cccc(I)c1 C12(CNC(c3ncn(C(C)C)n3)=O)CCC(CC1)N2C(C1(CO)CCCCC1)=O c1(C(C)C(=O)NC2CC(NC(=O)C(F)(F)c3cscn3)C2)ccc(F)cc1F C12CCN(CC1(F)F)C2.c1(N(C)C)ccc(CCNC2COCCN2CCO)cc1 C(=O)(C(F)(F)C(C(C)C)OC(=O)C1CC1)NC1C(OC)CCCC1 C=CC(CC)CC(=O)N1CC(CNC(=O)CC(=O)NCC(F)(F)F)C(C)C1 N1(C(c2c(CC)cnn2C)=O)CCC(C(N2CC(O)C(O)C2CO)=O)C(C)C1 N1(c2c(C(=O)OC)c(Cl)ncn2)CCC2CCC(C1)N2C(=O)CCF C1(C(=O)NC2C=CC(CC(=O)NC3(C#C)CCOC3)C2)CCCCCN1C CC1(c2nnc(N3CCC(OCC4CCC4)C3)n2CCN2CCCC2)COCCO1 C1(C(=O)NCC(C)Cn2ccnc2)CCN(C(c2cncnc2)=O)C1 C(=O)(CC(CC1CC1)NC(c1c[nH]c(=NC)o1)=O)N(CC(C)OC)CC CC1(NC(c2cc(C(N)=O)co2)=O)CCN(C(c2cnc(C(C)(F)F)s2)=O)CC1 c1(SC2CC(OCC(=O)OCC3CCC(F)(F)C3)C2)c(CC)nc(=N)[nH]c1C c1(C(=O)NCC2CCCCN(C(C(C)SC)=O)C2)c(C)cccc1[N+](=O)[O-] C1(NC(C(C)CF)=O)CCOC12CCN(C(=O)C(=CC(F)(F)F)NC(C)=O)CC2 CCC(O)C(C)C(=O)NC1(CCNC(c2c(C)coc2C2CC2)=O)CCCC1 C1(C(=O)NCC2(O)CCN(C3CCC(C)C3C(=O)O)CC2)Cc2ccccc2O1 N1(C(C(C2CC2)OC)=O)CC(NC(c2cnn(CC3CCCC3)c2)=O)C(SC)C1 c1(CNC(C)(CCC#N)c2n(CCCSC)nnn2)ccc(F)cc1Br c1(CC)cc(C(N2CCCC2CNC(=O)C(C)(C)CNC(C)=O)=O)ccc1OC C1(CC)CN(C(=O)Cc2ncc(F)cc2F)CCC1CNCC1CC(OC)C1 c1(C2(C(=O)NCC(C3CC3)NC(CN(C(C)=O)C)=O)CCC2)c(F)cccc1F N1(C(C2N(CC)CCC2)=O)CCCC(CC(=O)NCc2ccc(F)c(C)c2)CC1 c1(C(N2CCCC(C(N3CCCC(CC)C3)=O)C2)=O)cc(C)c(O)nn1 c1(C(N(C)CC2OCCN(C(CC(C)O)=O)C2)=O)ccc(F)cc1C1CC1 C(CCCCCC(=O)NC1CC12CCC(NC(=O)CCc1cnco1)CC2)SC n1(SCC(=O)OCCC(c2ccc(O)cc2)O)c2ccccc2c2ccccc12 N1(C(c2snc(C)c2N)=O)CC(C(=O)NCC2CC(C)CC(C)C2)C(C2CC2)C1 N1(C(c2c(C)nc(COCC)s2)=O)CCN(C(c2cc3occc3s2)=O)CC1C C1(SCc2n(C)nnn2)CCN(Cc2nc(CN3CCOCC3)no2)CC1 Cc1nc2cccc(C(=O)N(CCCN(C)C(C3CCCS3)=O)C)c2[nH]1 c1(OC)ccc2c(c1)CC(NC(=O)NCC(c1ncccc1C)(C)C)CC2 C1(CNC(CC2(CC=C)CCCC2)=O)(NC(c2nnc(C)s2)=O)CCCCC1C c1(CCCC(=O)NCCN(C(=O)CCCN(C)C(C)C)CC)ccc(C#N)cc1 c1(NC(C2(F)CN(C(C3CC3(F)Cl)=O)C2)=O)ccc2nn[nH]c2c1 C1(C2CN(C(C=C(C)C)=O)C2)CN(C(=O)C(C2(O)CCCC2)F)CCO1 C1(C)(CC)CC(NC(C2(C(C)(C)C)CCCC2)=O)CN1C(c1cccn1C)=O c1(CN(C)C)cnc(O)c2ccccc12.C12CCCN(C1)C(=O)C(=O)NC2 C1(CCNC(CCC=C)=O)CN(C(=O)CCCn2cccc2)CCS1(=O)=O C(=O)(CCC(=O)NC1CC(CCNC(C2(C)COCCO2)=O)C1)NC c1(C(c2noc(C3CCCCC3)n2)N)ccccc1.c12ccc(s1)CNC2=O C1(CC=C)(NC(c2cc[nH]c(=O)c2)=O)CCN(C(=O)Cc2ccsn2)CC1 n1(CC)ncc(C(=O)NC2(C)CCN(C(C3CS(=O)(=O)C3)=O)C2)c1C1CC1 C(C(C)(O)C(C)C)NC(=O)NC(c1ccncc1)CC CCC(C)C(=O)C(=O)NC(CCC1CCC1)C(=O)NC(c1nc(C)cs1)C N1(C(c2n(C)cc(Cl)c2)=O)CCCN(C(=O)C(C#N)CC2CC2)CC1 N1(C(CN(C(=O)OCC)C)=O)C(C)CC2CN(C(C3OCC4CCCC34)=O)CC12 c1(CNC(C2C(C(N3CCC(OC)C3)=O)C2)=O)cccnc1Br C(CCCCC(=O)N(C)CCNC(c1ccc(N(C)C)nc1)=O)NC(C)=O c1(CC(=O)NC(C2CCN(C(c3c(C)ccnc3)=O)C2)C)cccc(O)c1F C1(NC(C2CC(NC(=O)CN3CC4C=CC3C4)C2)=O)CCCCC12CCC2 c1(OCC=C)cccnc1C(N1CC(CNC(C2CCCC2(C)C)=O)C1)=O C(=O)(CC1OCc2ccccc21)N1CC=C(CNC(Cc2c(C)ocn2)=O)CC1 C1(c2cn(C(COC)COC)nn2)CN(C(C2CCCC2SC)=O)CCO1 C(=O)(C(C)CC(=O)N1C(CNC(c2ccc(F)cc2F)=O)CC2CC12)OC c1(C(=O)NC(CC)CNC(=O)C(C)c2ncco2)cc(C)ccc1Br C1(CNC(C(C(C)C)NC(N)=O)=O)CN(C(C2C3CCOCC23)=O)C(C)(C)C1 C1(O)(CNC(=O)CC(F)F)CCN(C(c2ncc(Cl)cc2Cl)=O)CC1 Cc1cc(C(=O)NCC2(CNC(c3nc(C4CC4)cs3)=O)CC2)n(CCO)n1 C#CC1(C(=O)NCc2cc(C(=O)NCC(C)(O)C(F)F)n(C)n2)CC(=O)C1 C1(NC(c2cc(CCC)nn2C)=O)(CO)CCCN(C(c2ccc(C)nn2)=O)C1 CC(C)C(O)CC(=O)NC1CN(C(=O)CN2CCCCCC2)CC1C N1(C(CCC(C)OCC)=O)CCC(C)CC1C(=O)NCC=Cc1ccccc1 CCC(CC)C(C(=O)N1CCCC1CNC(=O)C(=Cc1ccccc1Cl)C)OC c1(CC(=O)NC2CCN(Cc3cc(Br)ccn3)CC2O)ccc(F)cc1Cl C1(NC(=O)NC(C)(Cc2ccccn2)C(=O)O)NCCC1C1CC1 C1(CC(=O)N(CCCNC(C(C)C(C)(C)C)=O)C)CCCCCC1(F)F c1(NS(C)(=O)=O)cccc(C(=O)NC2CCC(NC(c3csnn3)=O)C2)c1F c1(C(=O)NC(C)CNC(=O)C(F)(F)CN(C)C)ccc(NC(N)=O)cc1Cl c1(C(=O)NC2CN(Cc3nccc(N(C)C)n3)C2)cnc2cccc(Cl)c2c1 C1(C(=O)N(CC(=O)NC2CC(N(C)C)C2)Cc2ccncc2)CC2CCCC2C1 c1(CCC(=O)N(C)CC2(O)CCN(C(=O)C3=NOCC3)C2)cccc([N+](=O)[O-])c1 CC1CCCC=C1C(=O)NC1(CO)CCN(C(=O)CC2(O)CCCC2)C1 c1(C(=O)NC2CCC(CNC(C(CNC(C)=O)(C)C)=O)C2)cccc(C#N)c1 C(=O)(CC(CC)N(C)C(c1ccsc1C#N)=O)N(CCCO)CC#C C=CCC(CC(C)C)C(=O)N1CC(C=C)(CC(=O)NC2N(CC)CCC2(C)C)C1 C(C(CC)N=c1nc(CC)[nH]s1)NC(Cc1c(SCC)cccc1)=O c1(CNC(=O)CCCCCSC)c(Cl)ccc(N2C(C(=O)OC)CC3CC32)c1F C(=O)(C(C)C(C)(F)F)NC(CC)CNC(=O)Cn1cc(Cl)c(C(F)(F)F)n1 C(c1ccccc1C#N)=CC(N1CCCN(C(C2CCC(C)(C)O2)=O)CC1)=O C(=O)(C1CCCc2cncn21)NC1CN(C(CC=CCC)=O)CC1(C)C c1(NC(C(C)(F)CNC(=O)C2=CCOC2)=O)cc(C(N)=O)cc(F)c1 C12(CNC(C=Cc3nc(C)sc3)=O)CCCC1N(C(C1C3CCCCC13)=O)CC2 N1(C(c2c(C)nsc2)=O)CCCCC1C1(CNC(=O)CCOC2CC2)CCOCC1 C1(CC)(NC(=O)C(C)COC)CCCN(C(=O)CN2CCC(=O)NC2=O)C1 c1(OC)cncnc1C(=O)NCC(CC1CC1)C(=O)N1CC2(CC2)C1 N1(C(C2C(C)N(C(c3nocc3Cl)=O)CC2)=O)CCCC(N=[N+]=[N-])CC1 c1(OC)ccc2ccccc2n1.C1(C(CNC(=O)C(C)(C)C)=O)CCN(C)CC1 C1(C(NOCCCC#C)=O)CCN(C(C2C(C#N)C2(C)C)=O)CC1(C)C c1(NC(C(CN(C(C2C(C(=O)OC)C=C2)=O)C)(C)C)=O)cc(C)cnc1C C#CCCN=C(NCCc1ccccn1)NCc1ccc(CN2CCCC2)cc1 C=C(C)CCCC(=O)NC(C1CCCCC1)CNC(c1cncc(O)c1)=O N1(C(c2occ3c2CCC3)=O)CCC2(NC(=O)COC3CCC3)CCCCCC12 N1(C(c2c(OC)cccc2F)C(=O)NCCSC)CCCOCC1(C)C C(=O)(C=C1SCC(=O)N1C)N1CC(N(N2CCC(c3cnn(C)c3)C(C)C2)C)C1 Cc1cccc(C)c1CNC(=O)C(C)(C)NC(=O)Cc1cn(C)cn1 N1(C(CSC(C)(C)C)=O)CCC2CCC(O)C1C2.C1(=O)CCOCCN1 c1(C(N(C2CC(NC(=O)CCc3csc(Br)c3)C2)C)=O)cnccn1 C#CC1CCC(NC(c2nnnn2-c2ccc(OC)cc2)=O)C1 Nc1ccc(NC(=O)Cc2ccc(Br)cn2)cc1 N1(C(CC(=O)OC)=O)CCc2ccc(C(=O)C3CC3)cc2CC1 C1(CNC(C(COC)N(C)C)=O)CN(C(=O)C(C)(C)CSC)CCO1 Fc1c(CNCc2oncc2-c2ccc(C(F)(F)F)cc2)ccnc1Br Cc1cnc2n1CC(C(=O)NCC(C1CCC1)NC(=O)C(F)(F)C(F)(F)F)CC2 CC1(C)CC(NC(=O)C=CC2CCOCC2)CN1C(c1cc(C(F)F)ccn1)=O c1(C(N(C2(CO)CN(c3ccnc(-c4nccs4)n3)C2)C)=O)nnc(O)nc1O Cc1nc(C(=O)OC(C)(C)C)ccc1NC(=O)NC1CC(=O)N1.C12CC1C(=O)N2 Cc1cc(C(=O)NC2CCCC23CN(C(c2cccnc2)=O)C3)n2ncnc2n1 c1(C(N2CC(N(C(c3c(C)nncc3)=O)C)C(C)(C)C2)=O)cnc2ccnn2c1 Cc1cc(C)n2nc(C(N3CCCC(N(C(=O)CSC4CC4)CCF)C3)=O)cc2n1 c1(C(C)=O)cc(CCC(=O)NC(C)(C)C(C)NC(=O)C=Cc2cc[nH]n2)on1 C(=O)(C1=C(Cl)CCCC1)N1CCN(C)CC1C(=O)NC1COCC1C(N)=O n1(CCC)ncnc1CN(C1CCN(C)C1)CCNOC(C)=O C#Cc1cc(C(N2CCC(NC(=O)COc3ccc(C)cc3F)C2)=O)cc(F)c1 c1(NC)ncc(C(=O)NCCCC(C)NC(c2ccncn2)=O)cc1Cl c1(C2C(=O)N2C(C)C(C)F)cccc(C(F)(F)F)c1.CC(C)C(=O)N(C)C(C)=O c1(C(c2n(CCC(C3CCC3)=O)nnn2)OC)ccc(F)cc1.C(C(=O)N)NCC(C)C N1(C(C2(CC(=O)OC)CC2)=O)CCOC(C)C1C(N1CC(F)(F)CC1C)=O C1(C(N(C)Cc2cscn2)=O)CCC2CCC1N2C(c1ccncc1)=O Cc1cscc1C(=O)NCC1CCN(C(c2nnc(C(C)(C)C)s2)=O)C1 C(C(=O)N(CCNC(=O)CCOc1cccnc1)CC1CC1)(C(C)(C)C)SC C1(C(N2C(Cn3cc(-c4nc(C)sc4)nn3)CC2)=O)CCC2CC2CC1 C1(N(C(c2cnc(Cl)[nH]2)=O)CC)CCCN(C(=O)Cc2c(Cl)cnn2C)C1 C1(CCCSCC(=O)NC(C(N)=O)C2CC2)CC=CCC1 n1(C(C)(C)C)cc(C(=O)NC2(CCCNC(C3CC(=C4CCC4)C3)=O)CC2)nn1 CS(C)(=O)=NCCN(c1ccccc1)C(=O)NC1CC1C(O)C(F)(F)F N1(c2ccnc(OC)n2)CC2CCC(NC(=O)CO)CC2C1 C(=O)(C(C)C(C)S(C)(=O)=O)N1CCC(O)C1.Cc1cccc(C2CCNC2)c1 CN(OCc1ccco1)C(=O)C(c1ccco1)NC(=O)CCc1ccsc1 C1(NC(C2C(C(C)O)C2)=O)CN(C(c2ccc3ncnn3c2)=O)CC(C)(C)C1 Cc1nn(C)c(C)c1C(=O)C(=O)NCC(CO)NC(=O)C(O)CC1CCCCC1 c1(C2(NC(C3(CNC(c4n(C)nnc4)=O)CC3)=O)CCCC2)cc(F)cc(Cl)c1 Cc1cc(O)c(C(=O)NC2CCCN(C(c3cc4c(s3)CCC4)=O)C2C)nn1 C1(CNC(C2CC3C=CC2CC3)=O)CCCN(C(=O)CCc2csnn2)CC1 Cc1ccc2nsnc2c1C(=O)NCC(C)(C)NC(=O)CCCC(C)C CN1CCCCC1CC(=O)NC1CN(C(=O)CCc2cccc(O)c2)CC1O C1(=O)C(C(C)(C)C)NCCN1.c1(C(N(C)C)=O)cccc(C(=O)NS(C)(=O)=O)c1 CC(C)C#CC(=O)NC(Cc1cn[nH]c1)C(=O)NC(c1cccnc1)C c1(OCC)cc(CC(=O)NC2CC(CC(=O)N(CC(C)CC)C)C2)[nH]n1 N1(c2cc(OCC)ncn2)CC2CC1CCC2NC(C1CCC(C)=C(C)C1)=O C#CC1(C(=O)NCC(O)CC(=O)NCC(c2ccccn2)C)CCCCC1 C1(CNC(C(C)CF)=O)CN(C(c2cccc(Br)c2Cl)=O)CC12CC2 C(=O)(CC1=CCN(C(=O)C(C)(C)OCCF)CC1)NCC1(CSC)CC1 N1(C(C)=O)CCC(C(N2CC(O)(Cn3cc(CSc4ccccc4)nn3)C2)=O)C1 CCCCC(O)C(=O)N(C1CCC(NC(=O)CCCNS(C)(=O)=O)CC1)C N1(C(C2C(OCC)C2)=O)CC2CCC(C1)N2C(=O)C=Cc1cccc(F)c1F N1(C(CCCC(C)C)=O)CCN(C(=O)C(CC(C)C)n2ccnc2)CC12CCC2 C1(CC(N2CC(c3onc(C)n3)C2)=O)CC2(CC2)CN1C(=O)C=Cc1cncn1C CC1COC2(CCC2)CN1CCC(=O)NCCCc1ccc(N)cc1 CCC(C)(CC(=O)NCC(C1CC1)NC(c1cncnc1)=O)C(=O)OC Cc1cc(=NC(=O)C(=O)N2CC(O)(C(C)NC(=O)CC(C)C3CCCC3)C2)[nH]o1 c1(C(=O)NC(N(C2CCOC(c3ccncc3)C2)CCCC)=O)ccc(Br)cc1 CC(C)(CCC(=O)N1CCC(NC(=O)COc2ccc(Cl)nc2)C1)[N+](=O)[O-] C(=O)(C1CCCc2sc(C)nc21)NC1C2C(NC(C(F)=CC)=O)CC(CC2)C1 c1(OC)ccc(-c2cccc(C(N3CCC(O)(SC)C3)C3CC3)c2)c(CO)c1 c1(C(N2C3(CN(C(CC(=O)NCC)=O)C3)CC2)=O)ccc(S(C)=O)cc1 CCCC(C(=O)NC1CCCC(CNC(=O)CCC2CC2)C1)S(N)(=O)=O c1(C(C)NC(Cc2ccc(Cl)cc2)C(C)C)coc2ccc(Cl)cc12 C(CC(C)(C)C)(C(=O)NCC1CC1Cl)NC(C(CC)CCOC)=O Cc1nc2cncc(C(N3CC=CC3CNC(=O)COCC3CCCC3)=O)c2[nH]1 c1(C(=O)NC2C(NC(C(C)(C)OC)=O)CC2)ccn2ccnc2c1 CC1CN(C(=O)C(C(C)O)NC(c2cc(Cl)cn2C)=O)CC1F N1(C(C)C)CCCCC1C(=O)NCCNC(C1CC1C(N1CCOCC1)=O)=O C1(C)(CNC(c2c[nH]c(=O)cn2)=O)CN(C(C2(c3ccccn3)CC2)=O)CCO1 C(c1ccc(Cl)cc1)=CC(=O)NCC(CCOC)NC(c1ccncc1F)=O c1(OCCOC(CC2CCCC(C)(C)O2)=O)ccc2c(c1)OCO2 C12(NC(C3C(C)(C)COC3)=O)CCCC(NC(=O)CN3CCCC3=O)(C1)C2 N1(CC=CC(=O)NC2CCC2CNC(c2ccc(CO)s2)=O)CCOCC1 C=C(C)C(C)(C)C(=O)N(CCC(=O)NCc1cnco1)CC1CC1 S(=O)(=O)(c1cccnc1)NCCC(=O)NC(c1ccc(F)cc1F)(C(=O)OC)C C(=O)(C1=CC2(CCN(C(c3c(F)cccc3F)=O)C2)C1)N(C(C(C)C)C)C N1(C(C(CC)(C)F)=O)CCC(CNC(=O)CC2CCC2)C(F)(F)CC1 c1(NCC(C(C)C)CO)[nH]c(=NCc2cnccn2)nc2sccc12 C1(CC)(NC(C2CCC3CC23)=O)CCCN(C(c2ccc(C3CCCO3)[nH]2)=O)C1 CC1(C2CN(C(C3CCCC3NCC3CCCNC(=O)C3)=O)C2)CC1 Cc1ccc2c(c1)CC(C(=O)NC1(C)CC(NC(C3CCCO3)=O)C1)S2 C1(CNC(C(CC)OCC)=O)C(C2CC2)CCN1C(c1cc(C)no1)=O C=C(C)CC(C(=O)Nc1cccc(C)n1)NC(=O)CCCN(C)C(C)=O C(C(C)(C(=O)OC)C(=O)NOC1CCOC1)OC(CC)C c1(C(=O)NCC2CC(C)N(C(=O)CC3CN(C)C3)C2)cc2c(F)c(F)ccc2[nH]1 Cc1cc(C(=O)NCCC2CCCN(C(c3cc(O)n(C)n3)=O)C2)nc(Cl)c1 N1(C(C(C)(C)c2cc[nH]n2)=O)CCC(F)(F)C(CNC(C2CC3CC3C2)=O)C1 CC1CC=C(C(=O)N2CCC(CC(=O)NCC3OC(=O)CC3(C)C)C(O)C2)CC1 N1(C(c2c(C)nc(C)s2)=O)CCN(C(=O)CCOC(C)CC(C)C)CC(C)C1 C(=O)(C(C(C)CC(C)(C)C)N(CC1CC1)Cc1ccccc1)NCCCSC c1(OC)cc2c(c(OC)c1CN1CCC13CC(F)(F)C3)C(C)CCC2 c1(C(=O)NCC2(O)CCN(C(C3C(C)CC3)=O)CC2)cc2ncccc2o1 Cc1ccc2c(C(N3CCCC(NC(C4CCCS(=O)(=O)N4)=O)C3)=O)csc2c1 c1(OCC(N2CC(CC(NOCCC=C)=O)OCC2)=O)c[nH]c(C)cc1=O C1(NC(CCC)=O)CC(F)CN(C(C2(CC(=O)OC(=O)NC)CCCCC2)=O)C1 CC1=NOC(C(N2CCC(CC(=O)NC(CO)CCN(C)C)C2)=O)C1 CN1CCN(CCN(C2CCS(=O)(=O)C2)C=O)CC1.c1(C(CO)=O)cc[nH]n1 C1(C)(NC(C(C)OCCOC)=O)CCCC12CCN(C(=O)C(=O)NC1COC1)CC2 c1(CC(=O)NC(CN(C(c2csnc2Cl)=O)CC)C)coc2cc(OC)ccc12 N1(Cc2ncc(NC(=O)Nc3ccc(C(C)(C)C)cc3)s2)CC2(CC(CO)C2)C1 C1(CC(=O)NC(C2C(C(N(CC(C(=O)OC)C)C)=O)C2)C)CC(C)(C)CO1 N1(C(C(c2ccccc2)C)=O)CC(F)CC1CN(C(=O)C=CSc1nc[nH]n1)C c1(C(N2CCN(C(C(C3CCOCC3)C)=O)C(CF)C2)=O)cc(F)cc(Cl)c1N CC1CC2(CCN(C(=O)CC3(O)CCOC3)CC2)CN1C(=O)CCc1nc[nH]n1 c1(C(=O)NC2C(NC(c3cc(C)sn3)=O)C2)ccc(SC2CCOCC2)cc1 c1(CC)ccc(C(=O)N(C)CCNC(c2cccc(CS(C)=O)c2)=O)nc1 c1(C(=O)NC(CC)CO)cn(C(C)(C)C)nc1C c1(C(=O)NCC2(C(C)(C)C)CCN(C(=O)CCCF)C2)cc(O)nc(C2CC2)n1 C(=O)(CCC(=O)NC(C1CCCN(C(=O)CC(C)(C)OC)C1)C)NCC c1(C(=O)NCC=C(Cl)Cl)cnc(O)c2c1NCCC2 N1(C(CCCNC(C)=O)=O)CCC2CCN(C(=O)C3CC3)C2C1 c1(C(N2CCN(C(C3CCN(CC#C)CC3)=O)C(C)C2)=O)ccc(Cl)c(C)c1O C(=O)(CCCCCSC)NC(CC#C)CC(=O)NC(CO)CC(F)(F)F c1(NC(=O)NC2CCN(CCOCC)CC2)c(C)cc(C)nc1Cl Cc1cnc2c(C(=O)NC(C)CC3CN(C(C4CCC(C)(C)C4)=O)C3)cccn12 c1(C(=O)NC2CC(NC(c3c(Cl)cn(C)n3)=O)C2)nc2cnccc2s1 C1(COC)CN(C(=O)CNC(=O)CN(C)C)CCN1C(=O)C1=NNC(=O)C1 N1(C(=O)CC2CCCOCC2)CCN(C(c2cnc3n2CCS3)=O)C(CF)C1 C12(CC#C)CCCN(C1)C(=O)N2.c1(CO)ccc(-c2nc[nH]n2)cc1 c1(C(=O)NC(C2CCCN2C(c2ccc(CCF)cc2)=O)C)ccnc(O)c1 N1(C(C(c2ccc(Cl)cc2)C)=O)CCC2C(CCCN2C(c2cncnc2)=O)C1 C1(C(=O)NCCCOCCNC(C=C2CCN(C)C2)=O)CCCN(CC(F)F)C1 c1(CNC(C23CC(NC(=O)CCc4cnc[nH]4)(C2)C3)=O)c(F)cncc1F N1(C(C(C)OCc2ccccc2Cl)=O)CCC2CN(C(=O)C(C)(C)CO)CC2C1 C1(N(C(=O)CC2CCC2)CC)CCN(C(C2CCOC2)=O)C1 c1(OC)ccc2c(c1)CC(C(N1CCC3(C1)CN(C(=O)C=C1CCC1)C3)=O)CC2 n1(CCC)c(C)cc(C=CC(=O)NC2(C)CN(C(C3CC3Cl)=O)C2)c1C C1(NC(C)=O)CCC12CN(C(c1ccn(-c3cccc(F)c3)n1)=O)C2 Nc1cc(F)c(O)cc1C(=O)NC1CCC(CCNC(=O)CC(=O)NC2CC2)C1 N1(C(C2OCCN(C(c3ccc(C)c(C)n3)=O)CC2)=O)CCCC(C)(C)C1C CCC(CC(C)O)NC(C1CN(C(=O)OC(C)(C)C)CC1OC)=O C1(C(N2CC3C(NC(C4C5(CC(OCC)C5)C4)=O)C3C2)=O)CC(=O)NC(=O)N1 CCC(CC)(C(=O)N1CCC(C)N(C(=O)CC23CCCC2C3)CC1)C(C)C CCCC(CNC(=O)C(C)c1ccco1)NC(c1cnc(C)[nH]1)=O c1(C(N(c2c(F)cccc2[N+](=O)[O-])C)=O)ccc2c(S(N)(=O)=O)cccc2c1 C1(C(=O)NC2C=CC(CNC(c3nn(CC)c(O)c3)=O)C2)CCC(C)=C(C)C1 c1(CC(=O)NCC(C)N(C)C(c2cccn2C)=O)ccnn1-c1ccccc1 N1(C(C(C)N(C(C)=O)C)=O)CCC(C(=O)NCC2(F)CCCCC2)CC1 C1(CC(=O)NC2CC(NC(c3cccc(CN(C)C)c3)=O)C2)CCCCC12CC2 C1(C(=O)NCCC2CCCC2O)CCCCN1C(c1c[nH]nc1Cl)=O C1(C(=O)NCC2CSCCO2)CCN(C(=O)C2CCCCCCC2)O1 C1(CC)CCN(C(=O)CCOC(C)C)CC1.c12sccc1NC2=O C(=O)(C(CC(C)C)n1ccnc1)NC(CC)CNC(=O)C=CCc1cccnc1 C(=O)(CC(O)CC(C)(C)C)N1CCC(CN(C(c2cc(C)n(C(C)C)n2)=O)C)C1 c1(C(N2CC(CC)C(N(C)C)C2)=O)ccc(OC)cc1C.c12nc(cs1)NC2=O C1(N(C(COCCOC)=O)C)CN(C(c2cn(C(F)(F)CO)nn2)=O)CC1F C1(N(C(CCCC)=O)C)CCCC2CN(C(c3ccncc3N)=O)CC12 C1(C(=O)NCCCN(C(c2c(OC)nsc2)=O)C)CCC(=O)N(C2CC2)C1 O=C(C#Cc1ccccc1)N1CCN(C(C2CCCC3CC23)=O)C(CCO)C1 Cc1cc(Cl)c(C(=O)NC2CCN(C(=O)C(c3ccc(Br)cc3)O)C2)cn1 c1(C(CNC(c2nnsc2C)=O)NC(c2n(CC)ccn2)=O)cccc(C)c1 c1(C(CC)C(=O)NCCOCCCNC(=O)C=CCCC)cccc(Cl)c1 C(=O)(C(CNC(=O)CCc1nc(C(C)C)no1)N(C)C)NC(CCSC)C C12(C(N(CCCNC(C3CCCN3c3ncccn3)=O)C)=O)CCCN(CC1)C2 N1(C(CCC2CC(C)C2)=O)CCC2CCN(C(=O)C=CCF)CC12 c1(OC)cscc1C(N1C(C(=O)NCCCN(CCC#N)C)C=CC1)=O Cc1cc(C(=O)Nc2cc(C(F)F)cc(Br)c2)c2c(C3CC3)noc2n1 c1(C2(C(=O)Nc3nc(C)[nH]n3)CC2)cccc(C#N)c1.C12CCC(C1)N(C)C2=O C1(NC(C2(C)C=CCC2)=O)CCN(C(c2ccc(O)cc2)=O)C12CCC2 N1(C(c2ncn(CC)c2)=O)CCC(CNC(C2CCCN2C)=O)C(O)C1 C1(O)(CNC(=O)CCN2CCCCC2)CCCN(C(=O)CCc2cnc[nH]2)C1 C1(NC(C2CCN(CC)C2)=O)C2CC3C1C3C2C(=O)NCCN1CCCCC1=O C1(NC(C(CC)NC(C)=O)=O)C2CC1CN(C(c1cc(C)nc(C)n1)=O)C2 C(=O)(CC1=CCN(C)CC1)NC(CC)(C)CNC(=O)C(C)N(C)C Cc1n[nH]c(C)c1CC(C)C(=O)NCC1(NC(=O)CC23CCC(CC2)C3)CC1 N1(C(c2c(C(C)C)occ2)=O)CC(CNC(=O)C(F)(F)c2nccs2)C(C)(C)C1 C1(C(=O)NC(C2N(C(Cc3c(C)n[nH]c3C)=O)CCC2)C)CCC=CCCC1 C1(C(=O)NCC#CC(=O)NCCCn2cncn2)CC2C=CC1O2 CCCC(C)(CCC)C(=O)NCC1CC(O)(CNC(=O)CSC(F)(F)F)C1 CC1CCOC(C(=O)NCCCN(C(=O)CSc2cccnc2)C2CC2)C1 CC(C)(C#CC(=O)N1CCC(CC(=O)CNC(=O)OC(C)(C)C)CC1)SC1CC1 c1(C(=O)NCCN(C(C2CCCC2COC)=O)CC)cncn1C c1(OC)cccc(Cl)c1NC(c1n[nH]cc1NC(c1ccc(Cl)nc1)=O)=O c1(CNC(N2CCC(C3CCCO3)C2)=O)noc2c1CCCCC2 c1(CNc2nccc(SC)c2)cc(C)nc2ccnn12 c1(C(=O)NCCCC2CCCN2C(=O)C=Cc2nccs2)cc(F)c(F)cc1O C1(C(C)C)C(C(=O)NCC2CC3CCCC23)CCN1C(=O)Cc1ccccc1 N1(C(c2[nH]c(C)c(C)c2C)=O)CC2CC1CN(C(c1ncc(F)cc1F)=O)C2 C1(CN(C(C2CC2C)=O)CC)CCCCN1C(=O)CCSc1ccc(F)cc1 C(=O)(C(C)COC(c1csc(C2CCCN2)n1)=O)OC C1(C(N2CC2)=O)CCCC(CC)C1.C(=O)(C(C)SCC=C)N.C#CCONCC#C.N C1(CC)CN(C(=O)C(C)CC(F)F)CCN1C(c1ccnc(OC2CCC2)c1)=O C(CNC(=O)C(C)(C)C1CCN(C(c2cnn(CCO)c2)=O)C1)(C(C)(C)C)OC C(=O)(CCCCCC(=O)NC1CC1NC(=O)C(O)Cn1cncn1)OCC CCCC(C(=O)NC1CC1=O)OCC.C(C(C)(C)C)C(CN)C.OCC CCCCC(CC)C(=O)N1CCC(CNC(=O)C=Cc2nccs2)C1(C)C N1(C(CCCC(C)O)=O)CC2CCCC(NC(=O)CCc3ccn(C)n3)C2C1 CCC(CO)(C(=O)NC1CC=C(C(=O)N(C2CCCCCCC2)C)C1)OC c1(OC)ncc(C(N2CCC(N(C(=O)OC(C)(C)C)CCO)C(C)C2)=O)cc1Cl C1(C(=O)NCC(=O)NCC(=O)OCC)(OCCC(C)c2cn[nH]c2)CCC1 C1(C(=O)NC2(CNC(=O)CCC3CCCC3)CC2)CCn2c(O)nnc2C1 N1(C(c2n(CC)cnn2)=O)CC(CNC(=O)CCc2nnc(C(C)C)o2)CC1C N1(CC)CCN(c2ncnc(SC)c2I)CC12CCC2 C1(C(C)C)C(C(=O)N(C)Cc2cccnc2)CCN1C(=O)C(C)C1(O)CCC1 C1(NC(C2(C)CC2(Cl)Cl)=O)CC(NC(=O)Cc2cnsc2)C12CCC2 N1(C(C(C(C)C)N(C(=O)C2CC2)C)C=O)CC2CN(OC(C(C)(C)C)=O)CC2C1 CC(O)C(C)(C)C(=O)N1CCC(NC(=O)OC(C)(C)COCCOC(C)(C)C)C1 c1(C(=O)NC(CN(C(C2C(C=C)CC2)=O)CC)C)cc(N)ccc1SC c1(OC)c(C(=O)NCCN(C(C2CCOCC2C)=O)C2CC2)cc(F)cc1F c1(C(=O)NC2CN(C(CSc3nc(C)on3)=O)C2)snc(O)c1Cl Cc1cc(F)cnc1-c1cn(C2COCC2NC(C2CC2c2ccsc2)=O)nn1 c1(OC)ccc(C)cc1-n1cc(CCCNC(=O)C(C)NC=O)nn1 C(C(=O)N1CCC(=CC)CC1)(C(C)C)NC(C)=O.c1(OCC(=O)N)nc(O)nc(O)n1 C(=O)(C1CCC(=O)c2ccccc21)NCC1N(C(CNC(N)=O)=O)C2CCC1C2 C1(CC)CCC(C(N2CCC(C)(CNC(C3CN(C(N)=O)C3)=O)C2)=O)CC1 N1(C(C23CC(CN(C(C4(CC=C)CC=CC4)=O)C2)C3)=O)CC2(COC(C)(C)C2)C1 c1(C(N2CCC(C(C)NC(c3cc(C)no3)=O)C2)=O)c(O)cc(F)cc1F c1(C(N)=O)cc(Cl)ccc1-n1cc(CONC(C2CN3CCC2C3)=O)nn1 N1(C(Cn2c(C)ccn2)=O)CC2(CC2)CC1CNC(=O)C=CC(C)C Cc1cc(Br)cc(C)c1C(c1nnnn1-c1ccccc1)NC1CCC(F)(F)C1 N1(C(C2CC(CC)C2)=O)CCCC(C)C1CCNC(c1cnc(O)cc1OC)=O C1(F)(C(=O)NC(C(C)OC)C)CCN(C(c2cc(C)ccc2C)=O)CC1 C#CCCC(O)C(=O)NCC1CCC1NC(c1cccc(CCC=C)c1)=O n1(CCc2ccccc2)nc(C2CC2)nc1C1CCCCS1.C1(C)CCCCO1 c1(CC)cc(C(=O)N(C(C)CN(C)C(C2CC(CF)C2)=O)C)c(Br)s1 c1(NC(CC2CCCN(C(c3c(C)ocn3)=O)C2)=O)ccc(O)c(CO)c1 C1(C(=O)NC(c2cccc(C)c2)CNC(=O)CP(C)(C)=O)CCCC2(CC2)C1 CCC(C)CCCC(=O)N1CC2(CC(C(=O)NCC3Cc4nccn4C3)CO2)C1 c1(SC)ncc(N)c(C(N2CC3C(NC(C4(C)CC4)=O)C3C2)=O)n1 c1(N(C2CCNC(OC)C2)CCC=C)ncnc2[nH]ccc12 C1(C(=O)NC2CCC(NC(c3n(CC)ccc3)=O)C2)CCCS1(=O)=O N1(C(c2ccc(C)o2)=O)CCCCC1C1(NC(c2cnn(C(C)C)c2)=O)CC1 CCCCCCC(=O)NC1CN(C(C2C=CCCC2)=O)CCC1C C(=O)(N=c1c(Br)c[nH]cc1I)C1(F)CCN(C(C(N2CSCSC2)C)=O)C1 N12CCC3(CC1)CC3CNC(=O)CC2.C(CC(=O)NC1CC1C(F)F)=C(C)C N1(C(C2CC(OC)C2)=O)CC2CCCC1(CNC(=O)C(C)(C)c1ccns1)C2 C1(CN=[N+]=[N-])CCCN(C(c2cc(CNC(=O)Cn3ccnn3)no2)=O)C1 Cc1cnc(Cl)c(C(=O)NCC2(O)CCCN(C(=O)C(C)NC=O)C2)c1 Cc1nc(C2CCC2)oc1C(=O)NC(C1CCCN1C(c1ccc(CO)s1)=O)C C1(C(C)C)CN(C(=O)C(C)c2cc[nH]n2)CCN1C(=O)C1=CCCC1 c1(C(N2CCC3(CC2)CC(O)C3)C(=O)NC(CC)C)ccc([Si](C)(C)C)cc1 C1(C(N2CCC(n3cc(CCN4CCSCC4)nn3)C2)=O)(CO)CCCO1 Cc1ccc(C(N2CC3(CNC(=O)Cc4csc(S)n4)CC2CO3)=O)nc1F c1(C(N(C2(CC)CCNCC2)Cc2ncsc2C)=O)ncnc2cc(I)sc12 Cn1cnc2cc(C(=O)NCCCOCCCNC(c3ccsn3)=O)ccc12 C1(CCC(=O)NCC2N(C)CC(O)C2)CCN(C(=O)Cc2nccn2C)C1(C)C C1(CNC(c2n[nH]c(C)c2C)=O)CC2(CC2)CN1C(=O)CCc1nc(O)n[nH]1 C1(c2n(C)ccn2)CN(C(=O)CC#N)CCN1C(c1cnc(C2CCOC2)s1)=O c1(OC)ccc(CNC(=O)NC(CC(N)=O)c2ccccc2)cn1 c1(OCC(=O)N(C2CN(C(CCN(C)CC)=O)CC2F)C)ccc(Cl)cc1F C(=O)(C1c2ccccc2C2CC1C2)NCC(C)CNC(=O)C(S(C)(=O)=O)C1CC1 c1(C(=O)NCC2N(C(COC)=O)CCC2C2CC2)ccc2[nH]c(=O)c(=O)[nH]c2c1 C1(CNC(C(C)OCCOC)=O)CC(=O)N(C)C1.C12(CC1)CCNC2=O c1(C(C)=O)ccc(S(=O)(=O)N2CC(NCc3cnc(O)c(Cl)c3)C(C#N)C2)cc1 CCCC(CC(=O)NC(C)CF)NC(c1cnc(O)c(C)c1)=O N1(C(=O)OC(CC=C)CNC(=O)CCCCN(C)C)CCC(C(F)F)(CO)C1 N1(C(CCC(=O)NC)=O)CCC2(CC1)COC(CNC(=O)C(C)(C)C)C2 Nc1ccc(F)c(C(N2CC3OCC(NC(=O)Cn4nccn4)C3C2)=O)c1F c1(N2C(C)CCN(C(C3N(CC(C)C)CCCC3)=O)CC2)cc2nncn2cn1 N1(C(c2c(CC)cns2)=O)CC2CC(C1)CN(C(=O)CN1CC(CC)C1)C2 C(CCCCC(=O)N(CC(O)CN(C)C(c1cn2ccsc2n1)=O)C)=CCCC Cc1ccc2nc(C)cc(C(N3CC(CNC(=O)CCCC(C)C)C3)=O)c2c1 CCCS(=O)(=O)CC(=O)NCC1(NC(c2cn(C)c(C(F)F)n2)=O)CCCCC1 CCCCCC(F)C(=O)N1CCC(NC(=O)CCC=CC(C)C)C1C(C)(C)COC C(C(C)C(=O)NCC1(O)CN(C(=O)Cc2ccc(Cl)s2)C1)OC c1(C(N2C(CSC)CC2)=O)ccc(F)c(NC(c2c[nH]nc2-c2cccs2)=O)c1 c1(C(=O)OC)ccc(C=CC(=O)NC(C)CCNC(C2CCS2(=O)=O)=O)o1 C1(C(=O)NCCOCCCNC(CC(C)(C)O)=O)Cc2c[nH]cc2S1(=O)=O CCCC(C)CC(=O)NOCc1cc(C(N2CCC2C)=O)ncn1 C1(C(=O)NCCOCCNC(c2c(C)nc(Br)o2)=O)CCOCC12CCCC2 C1(C(=O)NCCCCCN(C)C)CCC(C2CC2)N1C(C1CCC=CCC1)=O C1(N(C(CCc2ccc(C)cc2)=O)C)CCN(C(C2CCCOC2)=O)CC12CC2 CCC(CNC(=O)C(C)NC(c1ccc(CO)s1)=O)C(C)(F)F N1(C(C2C3(CCN(Cc4cnc(C)nc4)CC3)C2)=O)CCC(C2CCN(C)C2)C1 C1(N(C)C(C2(CO)CCOCC2)=O)CN(C(=O)C=C(Cl)Cl)CC1(C)C N1(C(C2CC(C)=C(C)CC2)=O)CC2CCC1CN(C(c1cc(Cl)cn1C)=O)C2 N1(C(C2(C(=O)OCC)CC2)=O)CCC(O)(CNC(c2cc(Cl)c(C)cn2)=O)CC1 c1(C(=O)NCC(CN(C(=O)CN(C)C)C)O)ccc(F)c2occc12.C1(=O)CN1 c1(C(CNC(COCC=C)=O)NC(c2cc(CC)[nH]n2)=O)cccc(Cl)c1 N1(C(CC(C)(C)CNC(c2ccoc2)=O)=O)CC2(C)CC1CCO2 c1(C(N(CCN(C(C2C(CC)C2)=O)C)C(C)C)=O)cnc2cc[nH]c2c1 CC(C)CC(=O)C(=O)Nc1cc(C(N2CCOC(C3(C)CC3)C2)=O)[nH]n1 N1(C(c2ccc(OCC)nc2)=O)CCN(C(=O)C(C)c2ccon2)CC(O)C1 Cn1cc(NC(c2ccoc2CNC(=O)CC(C)(C)O)=O)c(O)n1 CC(C)(C)S(=O)(=O)CC(=O)N1CCOCC1C1CCN(C(C2CCCC2)=O)CC1 c1(OCC)cnc(C(N2CCCC(N(C(=O)CC3CCCC3(F)F)C)C2)=O)cn1 O=C(C1=CC2CCC=CCCC12)NCC1CC(O)CN1C(=O)C=Cc1nccs1 C(=O)(CCN=c1[nH]ccs1)NC(CNC(c1ccc(N=[N+]=[N-])cc1)=O)C1CC1 c1(OC)cc(C(N2CCC3(NC(=O)C4=NOCC4)CC3C2)=O)cc(C(F)(F)F)c1 N1(C(C=CCOC)=O)CCC2CC1CN(C(=O)C1=CCCOC1)C2 c1(C(=O)NCC(CNC(c2scc(C)c2)=O)F)snc(O)c1Cl C1(C)(NC(C2CCC(CNC(c3ncn(CC)n3)=O)O2)=O)CC2(CCC2)C1 C=C(Br)CCC(=O)N1CC(NC(=O)CN2CCCCC2=O)C(SC)C1 N#CC1(C(=O)NCCCCCNC(=O)CSCc2cccc(Cl)c2)CCCO1 c1(OC)nsc(OC)c1C(=O)NC1CCC(CNC(C2OCCOC2C)=O)CC1 C(=O)(C(C)(C)C(=O)NCC1COCC1NC(=O)C1=CCCCO1)N(C)C C(=O)(C#CC1(C)COC1)NC(C(=O)NCC(C#C)CC)C1(C)CC1 c1(NC(C(C(C)OC)C)=O)ccc(C)nc1O.c12ccsc1C(=O)N2 N1(C(CCN(C(CN2C(C)CCC2)=O)C)=O)CCC2CC12CO C1(C(C)(C)NC(c2cnc(C)[nH]2)=O)CCCCN1C(c1nnsc1C)=O c1(C(N2CC(C)C(NC(c3ccccc3Cl)=O)CC2)=O)ccc2nnn(O)c2c1 CC1c2cc(Cl)cc(Cl)c2CCN1C(=O)NCCc1ccnc(Cl)c1 c1(OC)ccc2c(c1)C(C(=O)N1CCN(C(C)C)C(=O)C1)CC2 c1(C(=O)NC2CC(=C)C2)cc(CNC(c2cc(OC)n(C)n2)=O)ccn1 C1(O)(CC(=O)NCC2CC3CCC2N3C(C2CC2C2CCC2)=O)CCCCCC1 C(N=c1[nH]c(=NC2CCCC(C)C2)[nH]c2cccnc12)c1ccc(CC)cc1 c1(C(N2CCC(NC(c3c(CC)ccs3)=O)C(O)C2)=O)cc(F)cc(F)c1O CC1COC2(C1)CN(C(C13COC(C1)C(NC(=O)Cn1cc(C#N)cn1)C3)=O)C2 N1(C(C2CCCOC2)C(=O)NCCC#N)CCC(C2CC2)CC1 CC1Cc2ccccc2N(C(c2ccnn2C2CCCC2)=O)C1C c1(C(=O)NCC(=O)NC2(C(=O)NCC)CCC2)cnc2ccccc2c1OC C1(CNC(C=CC=CCC)=O)CCC2(CN(C(=O)CN3CC(C)(C)C3)C2)O1 c1(NC(C)=O)cccc(C(=O)NC2CN(C(=O)CNC(N)=O)C3CC23)c1 C1(C(N(C(C)C)SC)=O)CC(=O)N(c2ccccc2F)C1.c12ccc(o1)CC2 Cc1ncccc1C(=O)NC(Cc1cn[nH]c1)C(=O)N1CC(CN(C)C)C1 N1(C(CC2CC(C)(C)OC2)=O)C2CCC1C1CC1(NC(=O)CNC(N)=O)C2 CC1CC(C)CN(CCCCNCc2nc(C(C)(C)C)n[nH]2)C1 N1(C(C(c2ccc(C)o2)C)=O)CCC2OCCN(C(c3nc(C)sc3C)=O)C2C1 C1(C(=O)NCC(C(C)O)C)CCC(C)(C)N(C(C2CC2(C)C)=O)C1 Cc1ccc([N+](=O)[O-])cc1C(=O)NC(Cn1cc(CC(C)(C)C)nn1)CC(C)C C1(NC(C2CC=CC2)=O)CCCCN(C(=O)Cn2nccc2-c2ccccc2)C1 c1(CN(C)CC2CCCN(C(C(=O)NC)=O)C2)cc2ccc(Cl)cc2[nH]1 CN(C)NC(=O)CCC(=O)NC1CN(C(C2C(F)(F)C23CC3)=O)C1 c1(C(N(C(C(CC)C)CO)C)=O)ccc(-c2c[nH]nc2C(F)(F)F)cc1[N+](=O)[O-] c1(NCC2CCC(C(N3CCCC3C=O)=O)CC2)ncc([N+](=O)[O-])cc1Br.CO C(=O)(CC(C)CC(C)(C)C)N1CCC2(C(NC(c3c(C)c(Cl)cnc3)=O)C2)CC1 Cc1cc(OCC(C)NC(=O)NCCOc2nc(Cl)ccc2CO)cc(C)c1 C(C(CCNC(=O)C(C)NC(=O)C(C)CN1CCOCC1)OC)OC C(N=c1[nH]c(=NCc2cnn[nH]2)c2c(F)cccc2[nH]1)C12C(F)(F)C1CCCC2 CS(=O)(=O)CCCC(=O)N1CC(CNC(C2CCC3(CCC3)O2)=O)C2(CCC2)C1 c1(N2CCC(SC)CC2)nc(=NCc2cc(C)on2)[nH]c2c1COCC2 CC#CCCC(=O)NCc1cn(-c2c(CCN3CCCC3)cccc2)nn1 N1(C(CN(C)C(=O)C2CC2)=O)CC2(CCCN(C(c3cc[nH]c3)=O)C2)C1 N1(CCC(=O)NC2c3cc2co3)CCN(C2CCC2)CC1.CC(C)(C)N.C(=O)OCF c1(C(N2CC(CCO)(NC(CC(c3ccc(F)cc3)C)=O)C2)=O)cc(F)n(C)n1 C(=O)(CCCC(C)(F)F)C(=O)Cc1n[nH]c(=N)s1.C1(C2CC2)CC(=O)N1C.N C12(NC(=O)CC=C(Cl)Cl)CCC(n3cc(CN(C(=O)C4CC4)CC)nn3)(CC1)C2 C#Cc1ccc(N(C)C)c(C(N2CC(NC(=O)COCCSC)CC2(C)C)=O)c1 c1(-c2cc(C(N3CCC(C)(C(=O)OC)C3)=O)sc2)cc2cn[nH]c2cc1OC C1(CNC(=O)Cn2cc(C3CC3)cn2)CN(C(C2CSC2)=O)CCCO1 c1(CC)cc(C)c(C(=O)NC23CC2CN(C(C2(Cc4cnn[nH]4)CCC2)=O)C3)s1 c1(C(N2CCC(C(=O)NCCCCC#C)(CO)C2)=O)nccc(C)c1N C1(NC(C(OC)OC)=O)CC2(C1)CN(C(c1cc(F)ccc1C(F)F)=O)C2 Cc1ccc(C(=O)NCC2(F)CC(NC(=O)Cc3ccnn3CSC3CCC3)C2)s1 N1(C(C2CCN(C(c3cnns3)=O)C23CC3)=O)CCc2ccccc2C1 c1(C(=O)NC(C2CN(C(=O)C(C)(C)C(F)(F)F)C2)C)cc(C(N)=O)c(C)nc1C n1(C(C)C)cc(Br)cc1C(=O)N(CC(=O)O)Cc1noc(-c2ccccc2)n1 N1(C(C(c2ccc(C)o2)C)=O)CCN(C)CC1CNC(c1nscc1C)=O C(=O)(CS(=O)(=O)C(C)C)N1CC(F)CC(NC(c2[nH]c(=NC)sc2)=O)C1 N1(C(=O)CSc2nncn2C2CC2)CCCCC(NC(C2CC23CC3)=O)C1 N1(C(c2ncc(C#C)cc2C)=O)CCOC2(C1)CN(C(=O)C(CC)SC)C2 N1(C(C2(SC)CC2)=O)C2CCC1CC(F)(CNC(=O)C(C1CC1)SC)C2 C1(CNC(C2CC(C(F)(F)F)(OC)C2)=O)CCN(C(=O)C=C(C)C(F)F)CC1C C(CN=c1[nH]c(C(F)F)nc(=N)[nH]1)(N1CCCC(C)C1)C1CC1 C12(C(N(CCN(C(C)C)C(C3CCC(O)CC3)=O)C)=O)CC(C)(CCO1)C2 c1(NCC2CC(NC(=O)C=Cc3ccncn3)C2)c(Cl)cc([N+](=O)[O-])cc1Cl C(=O)(C(C)(C)C(N)=O)NCC(C(C)C)NC(c1cc(C(C)=O)sc1)=O C(=O)(C(CCC1CC1)NC(=O)CC)NCc1ccc(CC)s1.C1(C)CCC1 C12(CNC(C(C)=CC3CC3)=O)CCCCC1CN(C(=O)Cc1ccc(Cl)nc1)C2 c1(N2CC(NCc3cc(Br)cc(C)c3O)C(F)(F)CC2)[nH]cnc2nc(Br)cc1-2 c1(C(=O)Nc2cccc(OCCC=C)c2)cccc(Cl)c1-n1cncn1 CC1(C)CC(C(N2CCCC2CC(N)=O)=O)CN1C(=O)CC1CCCCC1 C1(NCC(COC(C(C)NS(CC)(=O)=O)=O)(C)C)CCC(C)CC1 C1(C(=O)NCCC2CCN(C(C(C(CC)C)O)=O)CC2)CCC(C2CCC2)CC1 n1(C(CCS(C)(=O)=O)=O)nc(Cc2ccccc2)c2ccccc2c1=O c1(NC2CC(CNC(c3ccc(C(=O)OC)nn3)=O)C2)ncnc(O)c1Br c1(C(C)C)[nH]ccc1C(N1CC(O)(CNC(c2ncoc2C(C)(C)C)=O)C1)=O N1(C(C(CC)OCC)=O)CCC2(CC1)CCN(C(=O)C(C)=CC1CC1)CC2C C12CCCC(CC1)CNC2=O.c1(C(=O)NCCO)cncn1C1CC1.C1(S)CC1 c1(COC(=O)CC2CC3(C(F)(F)F)COC2C3)n[nH]c2c1CCCC2 Nc1c(Cl)ccc(C(=O)NC2CCC3(CCCC3)C2)c1Cl C1(C(=O)NCC2C3CN(C(c4nonc4N)=O)CC23)(CC)CCCCC1 N1(C(C(C2CC2)OC)=O)CC2(C1)CN(C(=O)CCc1ccc(Br)c(Cl)c1)C2 Cc1cc(Br)cc(C)c1CCSC(F)F.C12C=CCN1C2 C1(CNC(c2ccc(OC)nc2Cl)=O)CN(C(=O)CCS(C)=O)CCC12CCC2 C1(Cc2cn(CC(CC)C)nn2)CCCCN1C(C1(C(F)(F)F)CC(=O)C1)=O C1(NC(c2c(C)coc2)=O)CCC2(CC1)CC(NC(=O)CN1CC(C)(C)C1)C2 c1(C(=O)NCC2C(NC(CCC3N(C)CCC3)=O)CCCC2)ccc(C#N)cn1 NS(=O)(=O)c1cc(C(=O)NC2CC2C(=O)N(CC#N)CCN(C)C)c(F)cc1Cl C1(CNC(CCC#C)=O)C2CCCC1N(C(C1CNC(=O)O1)=O)C2 c1(NCC(C)(CSC)OC)cc(N2CCC=C(Br)C2)nc(C)n1 N1(C(C2CC=C(C)CC2)=O)CCCC2CN(C(c3ccc(NC(C)=O)o3)=O)CC12 c1(C(=O)NC(C)CNC(C2(C)CCCC2C)=O)ccc2c(O)n[nH]c2c1 N1(C(c2cnc(OC)s2)=O)CCC2C(C1)NC(=O)CCN2C(=O)CSCCOC C(=O)(CCCCC(=O)NCc1ccoc1C(N1CCC(C)(O)CC1)=O)OC CC(C)(C)C(O)C(=O)NC1C2CC3C(C2)C13C(N1CCC(CC2CC2)C1)=O c1(CNCC2CN(C(CC)=O)C2)nc(-c2ccccc2)no1.C1(C=O)SCCS1 c1(C(CC)O)cn(C2CC(NC(=O)Cc3ncoc3-c3ccccc3)C2)nn1 c1(NC2CCC(CCCC)C2)ncc(C)cc1S(=O)(=O)N1CC(OC)C1 N1(C(=O)NC2(Cc3ccc(C(F)(F)F)cc3)CC2)CCNC2(CCC2)C1 c1(C(=O)NC2(C)CN(C(c3cc(CC)ncn3)=O)C2)cn(C)c2ncccc12 C1(C(=O)NCCCN(C(C(C)N2CCC2)=O)C)CC12CCC1(CC1)CC2 c1(SCC(C(=O)NCCOC)N2CCCC2CCN(C)C)ccc(F)cc1 N1(C(=O)OC)CCCC(C(=O)NC2CC(NC(C3(O)CC3(C)C)=O)C2)C1 c1(C2(N(C(CC(c3scc(C(=O)OC)n3)NC3CC3)=O)C)CC2)ccc(Br)cc1 C=CCCC(C)(C)C(=O)N(CC(C)NC(=O)C(c1ccccc1F)C)C C1(C(N(C)CC2(NC(C34CCCCC3C4)=O)CC2)=O)CCCN1C=O CC1CCCC1CC(=O)NC(CNC(=O)CCn1ccnc1)Cc1ccccc1 C1(C(=O)NC(CC)CNC(C23CC(C)(C2)C3)=O)CC2(C1)CC2(F)F CC1CC(C(=O)NCC2(C(=O)N(C3(CCO)CC3)C)CC2)=NO1 N1(C(C2C(C)CCS2)=O)CCN(C2CCN(C(c3coc(N(C)C)n3)=O)C2)CC1 C1(CNC(C2(C)CCC2)=O)CN(C(=O)CCCc2ccccc2)CCC12CCC2 Nc1ccnc(C(=O)NCC(C2CCCC2)NC(=O)CC2CCC3CC23)c1Cl CC(O)CCCCCC(=O)NCC1(O)CN(C(c2cnc3[nH]c(=N)sc3c2)=O)C1 C12(CNC(C3CC(NC(CCc4ccn(C)n4)=O)C3)=O)CCC(CC1)CC2 c1(CNC(C2C(NCc3cc(C)oc3C)C2)=O)ccc(Cl)c(Cl)c1 N1(C(=O)Cn2cnnc2)CCN(C(=O)C2=CCCC2)C(c2cccs2)C1 C=CC(C)(C)C(=O)NC(C)CCNC(=O)CC1CCC(C2CC2)O1 C12(CNC(CC3CCCN(C(C(C)C)=O)C3)=O)CCC(CC1)CN2C(=O)CC#N N1(C(COC)=O)CCCC2(CCC(CN3CCCCC3)C2)C1 N1(C(c2ccncc2)C(=O)NC)CCN(CC(C)O)CC1 C(C(COC)CC(=O)N1CCC(C)(C(N2CC3(CC(F)C3)C2)=O)CC1)OC c1(C(=O)NCC(CNC(C(C#C)(C)C)=O)CO)ccc(S(=O)C(C)C)cc1 C(N=c1[nH]c(Cl)nc2c1CCCC2)C1CC(NC(CC2CC(C)OC2C)=O)C1 C=CC(C)CC(=O)NCc1cccc(C(=O)NCC2CC(OCC)C2)n1 C1(NC(c2cc(C3CCCC3)no2)=O)CCN(C(=O)Cc2ccsc2)C1 N1(C(C(C)CCN(C)C)=O)CCC(C(=O)NC2CCCC2O)C(O)C1 N1(C(C2CC(C)(C)OC2)C(=O)NC(C)(C)C)CCCSCC1C1CC1 c1(OC)c(CC(N2CCC(N(C)C(c3cnn(C)c3Cl)=O)C2)=O)cccc1C#N c1(C(N2C(C(=O)Nc3c(C)nccc3)CSCC2)=O)ccc([N+](=O)[O-])cc1 CC1CC(NC(C2(CCF)CC2)=O)CCN1C(=O)CCN1CCCS1(=O)=O CC1=NNC(=O)C1CC(=O)NCc1cn(CC(=O)N(C)CCn2cncn2)nn1 c1(C(N2CC(C(C)NC(c3cccc(C(C)(F)F)c3)=O)C2)=O)cncc(N)c1 C(=O)(C(CC(F)F)N(C(=O)CC(C)F)C)NC(CSC)C C(=O)(CC(C)C(=O)N1CCN(C(=O)C=Cc2cocn2)CC1CF)OC c1(CC)noc(CC)c1CC(=O)NCC1C2CN(C(=O)CN3CCOC3=O)CC12 N1(C(c2ccc(C#C)s2)C(=O)NC2CC(C(=O)OC)C2)CCCC(C=C)C1 C=CC1OCCC1C(=O)NCC1CC(NC(c2cn(CC)nc2C2CC2)=O)C1 N1(C(Cc2ncn(C)c2)=O)CC(C2CC2)(C(=O)NCCC2(CO)CC2)C1 CC1CC(NC(=O)CC2OCCCO2)CCN1C(C1C=CCC1)=O C#CC1(O)CCCN(C(C2CCCCC2(C)NC(=O)CNS(=O)(=O)CC)=O)C1 C1(NC(CCCC#C)=O)CN(CC(=O)Nc2ccc(CC)cc2)CC1C#N c1(OCC(=O)N(CCCNC(C(CC)(C)CO)=O)C)cccc2c1OC(C)(C)C2 c1(NC(C)(C2CC2)C2CC2)ncnc2c1cnn2CCO C(=O)(CCCC(=O)OC(C1CN(C(C2CC3C(C2)C3(C)C)=O)CCO1)C)NCC C(CCCCCNC(=O)C(F)(F)C1(O)CCC1)NC(c1ccnc(O)c1)=O CCC(C(C)C)C(C(=O)NCCC1CC1)N1CCCCC1Cn1ccnn1 CC1(C(=O)NCC2COCCN2C(=O)Cc2nc([N+](=O)[O-])n[nH]2)CCC(=O)NC1 C1(C(=O)NC(CC#C)C)CN(C)CCN1C(C1CC(O)CN1C)=O C1(C(=O)NC(CC#C)CO)CN(C(C2(Cl)CC2(F)F)=O)CCO1 c1(C(N2CCC(C)SCC2)=O)cc(O)nc2c1CN(C(=O)CCCF)CC2 N1(C(Cc2n(C)cnn2)=O)CC(CNC(=O)C(O)CC(F)F)CC12CCC2 N1(C(Cc2ccc(C#C)cc2)=O)C2CCC1C(C)C(NC(C1(CCO)CC1)=O)C2 C1(C(C(C)(F)F)NC2CCOC2C2CC2)CCCCCC1 Cc1ncc2n1CCN(C(=O)CC1CCCC1NC(C1(C)CCC3CC3C1)=O)C2 CCCC(CCCNC(=O)Cc1cc(Cl)n(C)n1)NC(=O)C=CSc1nc[nH]n1 c1(CC)ccc(O)c(C(=O)NCC2(O)CC(CNC(C3CCCC4CC34)=O)C2)c1 C1(C)(COC)CC(NC(c2csc(Cl)n2)=O)CN1C(c1cn(C)nc1OC)=O N1(C(C=CCNC(C2(C(C)N(C)C)CC2)=O)=O)CC(S(N)(=O)=O)C1 Cc1ccc(C(=O)NCCCNC(=O)C(O)C2CCC2)o1 C12(C(N3C(C)CC(NC(=O)CSCCN(C)C)C3)=O)CCCN1CCC2 c1(C(=O)NC2CC(NCc3c(O)cccc3F)C2)ccc([N+](=O)[O-])s1 Cc1cc(NC2(CNC(c3ncn4ccccc34)=O)CCC2)n2ncc(C)c2n1 C=CCC(CC=C)NC(=O)CC12CC(NC(=O)CCC(C)SC)(C1)C2 C1(N(C(C(C(C)C)F)=O)C)CN(C(c2ncc(C(F)(F)F)s2)=O)CC1(C)C N1(C(c2c(C)coc2)=O)CCC(CO)(CNC(=O)CC2CCSC2)C1 c1(NC(c2ccc(C(=O)OC)[nH]2)=O)n[nH]c2c1CN(C=O)C2.C(C)(C)(C)O O=S(=O)(c1ccc(Br)cc1)N1CCC(O)(c2ccc(F)c(F)c2)CC1 c1(N(C(c2cc(F)ccn2)C(=O)NCCC2(C)CC2)C)cc(Br)cc([N+](=O)[O-])c1 N1(C(CC(C)CNC(C2CCS2(=O)=O)=O)=O)CCC2(CC1)CC2C#N C(=O)(C(C)(C(F)F)c1ccccc1)N(CC(C)NC(=O)Cc1cccs1)C Cc1ncc(N)cc1C(=O)NCC(C)(O)CNC(=O)CC(C)N(C)C Cc1nc2ccc(C(=O)NC(C)CNC(C3CCC(C)CC3)=O)cc2[nH]1 N1(C(C2C(C)CCC2)=O)CCCC(C2(NC(C34CC(C)(CCO3)C4)=O)CC2)C1 C(C)(N=c1[nH]c(=NCc2nonc2C)[nH]c2c1COC2)c1n(CC)ncc1 Cc1cc(C(=O)NCC2CCCC(NC(c3oc(C)cc3C)=O)C2)cc(O)c1 c1(C(N(CC(C)N(C(c2c(SC)csc2)=O)C)C)=O)cnn2ccc(C)cc12 C(=O)(C(F)CCC(C)(C)C)N1CC=C(CNC(C2(OC)CC2)=O)CC1 CCCC(C)CCCC(=O)NC(C)CN(C(=O)Cn1nc(C)cc1C)C C1(CCC)C(=O)NCCN1C(=O)C(C)CN(C(=O)CS(=O)(=O)NC1CC1)C C1(C)(C(=O)NC(CC)CNC(C2(N(C)C)CCC2)=O)CCC(C(C)(C)C)CC1 C1(N(C)C)CCC(C(=O)NCC(CNC(c2cccc(Cl)c2)=O)CO)CC1 c1(C(=O)NC23C(CN(C(C4N(CC)CC4)=O)C2)C3)cc(N)ccc1Cl c1(C(N(C2CCN(C(c3cnco3)=O)C2)CCC)=O)ccc2c(c1)NC(=O)C2=O c1(C(=O)NCCSCc2cn(CC3COCCO3)nn2)[nH]nc2ncnc(O)c12 N1(C(c2n(CC)nc(C)c2)=O)CC2CCCCC2(NC(=O)Cc2[nH]cnc2C)C1 C(C(C)(C(F)(F)F)c1ccccc1)OC.N12CCC(CC1C)NC2=O C1(C(=O)NC2CCC2NC(=O)CC2CCCCC2)(OCC)CCOC1 c1(CNC(C2CC(C(=O)NCCc3c(CCC)n[nH]c3)C2)=O)ncc[nH]c1=O C1(CC)CCCCC1C(=O)NCC(C)N(C(=O)CSc1cccc(F)c1)C CC1(CNC(=O)CC2CCC(=O)N2)CCCN(C(C23CCC2CC3)=O)C1 C=C(C)CCCC(=O)N1CC2(CC2)CC1CC(N1CCCCC1SC)=O Cc1ncc(C(=O)NC2CC(C(C)NC(=O)CCC3CCCC3)C2)o1 C(=O)(CC(C)(O)C(F)(F)F)NCC1N(C(c2cccc(C)c2N)=O)CC2(CC2)C1 C1(CNC(C(C)CC2CCCC2)=O)CC(C)CCN1C(=O)C#CC1(C)CC1 C1(C(=O)NC2(C)CCCN(C(C3=C(C)CCC3)=O)C2)COc2ccccc2O1 c1(CC(=O)NC2CN(C(=O)CC3CCC3)CC2F)cc2ccccc2s1 N1(C(COCCC)=O)CCN(C(=O)CC(C)(F)F)CC1c1ccccc1Cl N1(C(CCCCNC(N)=O)=O)CC2ON=C(CNC(c3coc(Cl)n3)=O)C2C1 C1(NC(C2(C)CCNC2=O)=O)CC(C(N2CCC3(CC2)N=N3)=O)C12CCC2 c1(C(N2CC(SC)C(NC(c3ccccc3F)=O)C2)=O)c(F)ccc(F)c1N Cc1nn(C)c2sc(C(N3CCC(NC(=O)C(C)C(F)(F)F)C3)=O)cc12 N1(C(c2cccc(CNC(C3CN(C(C)C)C3)=O)n2)=O)CCNC(=O)C1C C(C1=CCCN(C(C2C3CC4C(C3)C24)=O)C1)NC(COC1(C#C)COC1)=O C1(NC(C2ON=C(C)C2)=O)C2CC3CN(C(=O)CCP(C)(C)=O)C1C3C2 n1(CCC)nc(C)cc1C(=O)NC1CC(NC(=O)C(C)C(C)O)C(O)C1 c1(CNC(c2n(CCC)ncc2)c2nnnn2CC(F)F)ccc(Br)cc1NC c1(OCCC(=O)NC2CN(C(C3CC(C=C)C3)=O)C3C2C3)cc(F)cc(F)c1 N1(C(c2cc(C)nc(C)c2)=O)CCC2(CC1)CC(C(N1CCOC3CC13)=O)CO2 CC1CN(C(=O)CN2CCCC2C)CC1NC(C1CC1C#N)=O CC1CN(C(c2ncc[nH]c2=O)=O)CC(C(=O)Nc2cccc(CCF)c2)O1 N1(C(=O)Cc2csc(Cl)c2)CCN(C(=O)CC2(O)CCCOC2)CC(O)C1 c1(C(=O)NC2C3CN(Cc4cc(C)c(Cl)c(C)c4)CC32)oc2ccccc2c1C N1(C(COC(C)=O)=O)CC2OCCN(C(C3CN(C4CCC4)C3)=O)C2C1 C1(OC)(CNC(=O)C(F)=C(C)C)CCN(C(=O)CC2CCCO2)C1 S(=O)(=O)(CCC(=O)NCC1CC1NC(=O)COc1cc(C)cc(C)c1)NCC Cc1n[nH]c(=NCCCN(C(=O)Cc2csc(C(C)(C)C)n2)C(C)C)s1 C(C)(C)(CCC(=O)NC1CN(C(=O)CCCc2cccc(Br)c2)CC1C)OC C1(C(=O)NCC(O)CO)CCC(CNC(C2CC2(F)Cl)=O)CC1 C1(NC(=O)CSc2ccccc2)CCN(C(C2(O)CCSC2)=O)CCC1(F)F c1(C(C)C)ccc(-n2nc(COc3ccccc3)nc2C2CCCOC2)cc1 C1(CN(C)C)CN(C(c2cocc2Br)C(=O)NCC2CCCO2)CCO1 c1(CN(C(=O)NC2CCC(C)=C(C)C2)CC2C(C)=NOC2=O)cnc(O)c(Cl)c1 CN1C(=O)CCCC1C(N1CCCN(C(=O)Cn2cc(N)cn2)CC1)=O N1(C(C(c2ccc(OC)cc2)OC)=O)CC2CC(C(=O)Nc3cn[nH]c3)C(C2)C1 Cn1cc(S(=O)(=O)N(C)C(c2ccccc2)c2cnccn2)cc1C(=O)O N1(C(C2C(OC)C2)=O)CCC2(CCCN(C(c3cnn(CCF)c3)=O)C2)C1 C(=O)(C(N=[N+]=[N-])C(C)C)NC1(C(=O)NCc2c(C)nsc2)CCOCC1 Cc1[nH]nc2c1CN(C(c1cccc(Br)c1C)C(=O)NC1CCCC1)CC2 c1(N(C(=O)CN2CC(C)(C)C2)C)ccc(OCC(O)CSc2cccnn2)cc1 C1(CC)(NC(C2CCN(C(C)=O)C2)=O)CCN(C(c2cccc(N(C)C)c2)=O)C1 c1(OC)ccccc1OCC(N1CC2CC2(CNC(=O)CC2COCC2O)C1)=O c1(C(N(C2CC(NC(c3[nH]cc(CC)c3)=O)C2)C)=O)c(C)cnnc1O Cc1c(O)c(=O)ccn1CC(=O)NCCOCCN(C)C(C1CC=CCC1)=O CC1CN(C(=O)CSCCN(C)C)CC1NC(C1CC(O)(c2cccnc2)C1)=O Cc1ccc(NC(=O)C(=O)NCc2cccc(C(=O)N=S(C)(C)=O)c2)nc1C c1(OC(=O)NC)coc2ccccc12.C(Cc1ccccc1)(CCN1CC1)OC N1(C(C2C(NC(c3c(C)nccc3)=O)CCCCC2)=O)CC(C)c2ncccc21 CC(C)C(C(=O)N(C(C)CNC(=O)CCCn1ccnn1)C)NS(N)(=O)=O N(C(=NCC#Cc1ccccc1)NC(C)C)CCC(=O)NC.c12ccc(cc1)[nH]2 C1(NC(c2cn3cccnc3n2)=O)CC(N=c2nc[nH]c3[nH]c(Br)cc23)C1 CC1CN(C(c2c[nH]nc2[N+](=O)[O-])=O)CC(C(=O)NCC(c2cn(C)cn2)O)O1 N1(C(Cc2cccc(C)c2F)=O)CC2CCN(C(c3ncccc3C)=O)C2C1 N1(C(C(C)OCC(C)C)=O)CC2(CC(NC(C3CCCC34CC4)=O)C2)C1 c1(C(=O)NC2CC(F)(CNC(c3sccc3Cl)=O)C2)cc(Br)ccn1 c1(C(C(=O)NC(C)C)N(C)Cc2ccc(CC)s2)cc(C(F)(F)F)cc(Br)c1 N1(C(c2ncn(C(C)C)n2)=O)CC2(C(=O)NCC3CCCC(C)(C)C3)CC1CO2 c1(SC)cc(C(=O)NCC2COCC2NC(=O)C(F)(F)C(C)O)ccc1F C(CSC)(CCC(F)(F)F)NC(CCC)(c1nnnn1CCCOC)C1CCC1 c1(OC)ccc(CCNCCCCNCCS(=O)(=O)N(C)C)c(C)c1 c1(C(N2CCC(C(C)NC(COCC=C)=O)C2)=O)cccnc1N(C)C N1(C(c2c(O)ncc(CC)c2)=O)CC(NC(C2CCC(=O)NC2)=O)CC(C)(C)C1 N1(C(C(SC)C2CC2)=O)CC(NC(=O)COC2(C)CCC2)CC12CCOCC2 CCCC(CC)N=c1[nH]c(=NCCC2CCCCC2)[nH]c2c1COCC2 N1(CCN(CCN(c2ccon2)C)CC)C(=O)c2ccc(C)cc2C1=O c1(C(=O)NC2CC(F)(CNC(COCCC)=O)C2)cc(C(N)=O)ccc1C C#Cc1ccc(C(=O)N(CC(CC)NC(=O)COc2c(F)cccc2F)C)nc1 c1(NC(C(N2C(CNC(CCC(=O)NC)=O)CC2)C)=O)ccc(F)c(F)c1 Cc1cc(=NC(=O)C2CCN(CC(=O)NC=O)CC2)[nH]n1C c1(C(CN(C)C)CN)ccccc1.c1(CCCN(C(C(=O)NC)=O)C)ccc(Br)s1 C1(NC(C=COOCC)=O)CC2CCC(C1)N2C(=O)Cc1ccccc1O N1(C(c2cscc2Cl)=O)CCC(F)(F)C(CN2CCCC2Cn2ccnc2)C1 C1(CNC(CSCC)=O)CC2CC2N1C(=O)C(C)Cc1cnc[nH]1 Cc1nc(C)c(C(=O)N(C2CCCN(C(c3nn(C)nc3Br)=O)C2)C)o1 N1(C(c2cn(CCCC)nc2C)=O)CCC(NC(c2cc[nH]c2)=O)C(CC)C1 C(=O)(C(F)(CNC(=O)C(C)CC(F)(F)F)C(C)C)NCCC(=O)NC c1(C(N2CCN(C(CSC)=O)CC2CCO)=O)ccc2ncccc2c1Cl c1(NCC2CCN(Cc3ccc(C)cc3)C2C)nc(C)n2ccccc12 C1(C(N(CCN(C)C)Cc2cccc(OC)c2)=O)CC12CCCCC2 c1(C(C(N2C(CNC(c3c(C)scc3)=O)CCCC2)=O)=O)cc(F)c(F)cc1F C1(C(=O)OC(C)(C)C)CC(C)(C)CCN1C(=O)C1CC1.Cc1noc(C2CC2)c1 N(C1CCc2cccc3cccc1c23)C(=O)NCC1CCC(O)C1 c1(N2C3CC(NC(c4c(C)nco4)=O)CC2CC3)nc2ccc(O)cc2s1 C1(C(=O)NCC2CCN(C(c3n(C=C)nnc3)=O)C2)CC2(C1)CC(C(=O)OC)C2 C(CCN=C(NCC(F)F)N1CCOC(C2CCCO2)C1)OC(C(F)(F)F)(F)F Cc1nn(C)c(C)c1CC(=O)NC1(C2CN(C(=O)C=Cc3ccncc3)C2)CC1 C1(NC(=O)Cc2ncccn2)CN(C(=O)CC2CCCCO2)CC12COC2 C1(C)(C(N2CC3C(NC(C(C)C)=O)(C3)C2)=O)CCCCC1(F)F C#Cc1cc(C(=O)NC2CCCC2NC(C2CN(S(=O)(=O)CC)C2)=O)cc(N)c1 Cc1nn(CC(C)C)c(C)c1CC(=O)NC1CCN(C(C23CCC2C3)=O)C12CC2 C(=O)(C1CCCc2cncn21)N1CCC(NC(CC2=NNC(=O)C2)=O)(CO)CC1 S(=O)(=O)(c1cccc(F)c1)N.c1(C(=O)NCCN(C2CC2)C)nc2ncccn2n1 c1(CC(=O)NCCN(C(=O)C=CC2CC2)CCOC)csc(Br)c1 N1(C(CN(CC#C)C(c2n[nH]cc2Cl)=O)=O)CCCNC(=O)CC1 C(=O)(C1=NOC(C)(C)C1)NCCC1(NC(CC2CCCC(C)C2)=O)CCCC1 N1(S(CC=C)(=O)=O)CCC(NC(c2ncccc2Br)=O)C(C)(C)C1 n1(C(CC)C)nc(C(N2CCC(CNC(c3c[nH]nc3C(C)C)=O)C2)=O)cc1C N1(C(c2n(C)cnn2)=O)CC(C(N2CC([N+](=O)[O-])C2)=O)C2(CCC2)C1 c1(C(N2C(CN(C(C(C=C=C)C)=O)C)CCC2)=O)ccc2ncnn2c1 c1(OC)cc(C(F)(F)F)[nH]c(=NCC2CN(C(=O)C(C)(C)OC)CC2C(F)F)n1 C(N=c1cc(Cl)nc[nH]1)C1N(C(C(C2CCCCC2)C)=O)CC1 C(=O)(CC(C)(C)N(C(=O)C=CCOCCOC)C)NCCC(C=C)C c1(OC)cccc(C(=O)NC2CN(C(=O)CC3CC(C)=NO3)CC2O)c1C c1(C(N2C(C)(CNC(C(CC)F)=O)CC(F)(F)C2)=O)cc2ccncc2cc1F C1(CC(N2CCC(C)(NC(CC(CC)C)=O)C2)=O)CCS(=O)(=O)CC1 N1(C(c2ccc(OC)o2)=CCBr)CC2CCC1CN2C(=O)CC1(C)CC1 Cn1cc(C(=O)NCC(CO)NC(c2ccccc2C2(C)CC2)=O)c(O)nc1=O c1(C(N2CC(SC)C(NC(C3CC34CCC4)=O)C2)=O)ccc(Cl)c2ccccc12 Cn1cccc(C(N2CCOCCC2C(N2CC3C(C(N)=O)C3C2)=O)=O)c1=O Cc1csc(C(C(F)(F)F)NC(=O)CCC2CCCO2)n1 c1(C(c2n(CCCC)nnn2)NCCC2CCCOC2)ccc(Cl)cc1OC C1(N(C(=O)C(Cl)=CCl)C)CCCCN(C(C2(CF)CC2)=O)C1 C(=O)(CC1=NNC(=O)C1)N1CC(C(C)NC(c2cnccn2)=O)OCC1 CCCCC(CNC(=O)Cc1c[nH]nc1C)NC(C1CCC(=O)N1C1CC1)=O C(=O)(CC(C)CN(C)C)NCC(CNC(c1cnc[nH]c1=N)=O)OC C1(F)(C(=O)NCCc2cnc(C)[nH]2)CCN(C(c2sncc2C)=O)CC1 C1(c2n(C)ncc2)CC(=NO)CC1CNC(=O)NCCC(C)(C)N1CCOCC1 c1(CC(=O)NCC(C)NC(c2scc(C(=O)OC)c2)=O)ccc(C(C)(C)C)cc1 N1(C(CNC(CCC)=O)=O)CCC(NC(=O)CCc2nc(C)no2)C(CO)CC1 C1(C(F)F)(CNC(c2cc(C)[nH]n2)=O)CCN(C(=O)CCc2ccccn2)C1 C1(C(=O)NC2CCC(C(=O)NCC3CN(CCC)C3)C2)C2(CC2)C12CC2 C(=O)(C(CN)c1ccccc1)NCCNC(=O)CN1CCCC1.C1(Cl)(C(=O)O)CCC1 CC1CCNC(=O)C1NC(c1cc(CNC(c2cc(Cl)ns2)=O)ccn1)=O N1(C(C(=O)OC(COc2cccc(OC)c2)=O)=O)CCCC2(CCSC2)C1 c1(COC(c2cn(C)nn2)=O)c(Br)ccc2c1OCO2 c1(C(=O)NCC(C)(C)NC(C(COCC)C)=O)cc2c(C)cc(Cl)cc2[nH]1 C(=O)(CCN1C(=O)COc2ccccc21)N1C(CC(C)C)CC1 C1(NC(CC(C=C)(C)C)=O)CN(C(=O)CCCOCCOCC)C2(CCC2)C1 CCC(C)CC(=O)C(=O)NC(CCF)C(N1CCCCC(C)(F)C1)=O C(=O)(CC(CC(C)C)NC(c1cccn(C)c1=O)=O)NCCC(C(C)C)O C1(C(N(CCCO)CCOC)=O)CC12CCN(C(=O)CSc1ccccn1)C2 Cc1coc2c(C(N3CC(=C(F)CNC(=O)C=CC4CC4)C3)=O)cccc12 C#CC1CC2CCC1N(C(=O)CC1CC1CNC(=O)Cc1cc(C)[nH]n1)C2 C1(NC(c2cccc(C)c2F)=O)CC2CC(C1)N(C(=O)CC1CC=CC1)C2 c1(C(N(C2CCN(C(C(CC)(C)COC)=O)C2)C)=O)cc2oc(C)cc2[nH]1 C(=O)(CCC1=CCCCC1)N1C(C)(C(N(CCCC#C)C)=O)CCC1 C(C(=O)N1CC(CNC(=O)CNC(=O)CCC2CC2(F)F)C1)(C1CCOC1)OC N1(C(CCCC#C)=O)CCN(C(c2ccc(Cl)c(OC)c2F)=O)C2COCC12 c1(C(N2CC(NC(C(C)(C)F)=O)CC23CCC3)=O)cc2c(Cl)cccc2s1 C1(=O)C(F)(CC)C(=O)ONCC2(C)CCN1C2.c1(C(C)SC)ccccc1O c1(C(=O)OC)cncc(C(=O)NCC2CC2CCO)c1.c12sc(nc1Cl)[nH]c2=O C(C(=O)N(C(C)C(C)C)C)(C(C)(C)O)NC(Cc1cnc(C)s1)=O N1(C(CCSCCC)=O)CCC(C(=O)NCCOC2CC2)C1 C1(CCC)CCC(C(=O)NCC=CCNC(=O)C(n2nccc2C)C)CC1 C(=O)(C1=CSCCO1)NCCC1N(C(c2cc(C3(C)CC3)on2)=O)CCC1 C(N=c1[nH]cnc2ccsc12)C1(F)CCN(C(C2CC23CC3)=O)CC1 c12oc3ccccc3c1-c1c(CC)cc(o1)C(=O)NC1(CC1)CNC2=O.C(CO)SC CC1(C(=O)NOCC2CC2)CC(c2ccccc2)=NO1 Cc1cc(N2CCC(CNC(c3sccc3C(=O)O)=O)CC2)nc(C)n1 c1(CSC)ccc(C(=O)NC(C)(CNC(C2(C)CC(C)=NO2)=O)CO)cc1 N1(C(C2C3CCC(F)(F)C23)=O)CCCN(C(c2cc(Cl)cc(Cl)c2)=O)C(CO)C1 C1(NC(Cc2cc(C)no2)=O)CC(F)CN(C(=O)CNc2cnn(C)c2)C1 N1(C(C(Cc2c(C)nc[nH]2)O)=O)CCOC2CCN(C(c3cc(Cl)no3)=O)CC12 c1(OC)cccc(C(N2CC3CCC(C2)N3C(=O)CCCCC(C)C)=O)c1[N+](=O)[O-] c1(OCC(=O)N(CC(CNC(C)=O)O)C)cccc(C(=O)OC)c1F c1(C(N2CCC(O)(C(C)NC(COCC#C)=O)C2)=O)cc(CC)nnc1C C=C(Cl)CCC(=O)NC1CCOCC1C(=O)NCCCn1ccnc1C c1(CC)ccc(F)cc1C(N1CC(OC)CC1CNC(c1nocc1C)=O)=O CON1CCC(C(=O)NC2(C(=O)NCc3noc(C)n3)CCSC2)CC1 c1(-c2ccc(OC(CC)(C)C)cn2)ccc(CNC(=O)C(=O)C(C)(C)C)c(C)c1 C1(C#N)(C(N2CC(N(C)C(c3cn(C4CCOC4)cn3)=O)C2)=O)CCCO1 C(=O)(C1c2ccccc2-c2ccccc21)N1C2CN(C(C(C)CBr)=O)C(C2)C1 c1(OC(C)C(=O)Nc2cnc(-c3cccnn3)cn2)cccc2ccccc12 c1(C(=O)NC(C2(O)CN(C(C(C=C)(C)C)=O)C2)C)sc2ccc(C)cc2c1C Cc1ccc(NC(=O)CN2CCC(CNC(=O)CCSC(F)(F)F)CC2)cc1 C=CC1CN(C(=O)COC(F)(F)F)CC1NC(C1CCCC1(F)F)=O C1(NC(C(C)=C(C)C)=O)CN(C(=O)CCC(F)F)CC1C1CC1 C(=O)(C(C)(C)C(O)C(C)C)NC1CCCN(C(c2c(OCC=C)cccn2)=O)C1 N1(C(c2[nH]cc(COC)c2)=O)CCC2(CCCN(C(=O)CN3CCC3C)C2)C1 C(=O)(CCCCCC(C)O)N1CC(C2CN(C(c3c(CC)nc(C)n3C)=O)C2)C1 C(C(N=c1[nH]nc(C2CC2)o1)c1ccccc1)NC(c1ccc2cc(C)oc2c1)=O c1(OC)ncc(CN2CCCC2CCC(=O)NCCCc2cccnc2)cc1Cl C1(NC(c2c(SC)scc2)=O)C=CCN(C(=O)CSCCC(F)(F)F)C1 C1(NC(C(N2CCc3ccccc32)C)=O)CC(N=c2c(Cl)c[nH]cc2[N+](=O)[O-])C1 n1(CC(=O)NCC2(COC)CN(C(=O)C=CC3CCOC3)C2)ccccc1=O CCC(C)(C)CC(=O)NC12CCC1CN(C(=O)CCCN(C)C)C2 C(N=c1ccc(-c2ccc(CO)c(F)c2)c[nH]1)c1scc(COC)n1 N1(C(C(C=C)O)=O)CC2(CCC2NC(c2cc(SC)oc2C)=O)C1 C1(C(N2CC(CNC(c3c(=N)cc[nH]c3)=O)OCC2)=O)CCC12CCOCC2 C=CCC(C)(C)CC(=O)NCC1CCCC(CNC(c2cc(F)ccc2F)=O)C1 N1(C(c2ccn(CCC)n2)=O)CC2CC(C(N3CCN(C)C(=O)C3C)=O)C(C2)C1 c1(CNC2CCN(c3cccc(C)c3)C2)cc(Cl)c(Cl)c(Cl)c1 C1(CNC(C2CC(OCC)C2)=O)CC(NC(c2cncc(C(N)=O)c2)=O)CC1O Cn1nc2ccccc2c1CN=c1ccnc(NCCCN2CCCC2)[nH]1 C(=O)(C1=NOC(CCCNC(=O)C(F)(F)CC#N)C1)NCC(C)F.C1CCN1 N1(C(c2c(COC)onc2)=O)CCC2CN(c3ncnc4cc(Br)sc34)CC2C1 CCC(CC(=O)N(C1CN(C(=O)CC2C(C)(C)C2(C)C)CCC1O)C)C(F)F N1(CCCNC(C(C)c2cncs2)=O)CCC(NC(=O)CCc2cnccn2)C1 c1(C(=O)NCCCCCNC(C2CC3CCCC3C2)=O)ccc2ncccc2n1 c1(CCC)ccc(C(=O)NC(CNC(=O)CN(C)C2CC2)C(C)C)[nH]1 N1(C(C2(C)CC3CCC2O3)=O)CCC2(CC1)CN(C(c1ccc(N)c(Cl)c1)=O)C2 C(=O)(CC(=O)N1CCCCC1)OCC(C1(C(CO)O)CCOC1)=O.C(F)(F)F N1(C(CCOC(C)C)=O)CCCCCCC1C(=O)NCc1nc(C2CC2)no1 C1(C)(CNC(c2ccc(OC)cc2)=O)COCCN(C(=O)CC(O)C(C)C)C1 C1(C)(CNC(c2nccc(C)c2)=O)CCN(C(c2coc(Br)c2)=O)CC1 CC1(C)CCCC(C(N2CC(NC(=O)CCNC(N)=O)C(F)C2)=O)O1 c1(C(N2C(CO)CC(NC(=O)CCOCC3CC3)C2)=O)cnc2ncccn12 N1(C(c2n[nH]c(=N)s2)=O)CCCC(NC(c2conc2C2CCCC2)=O)C1 N1(CCC(=O)N(C)Cc2c(OC)cc(Br)cc2)CCC2CCC(C1)S2 N1(C(CN(C(=O)C(CC)CC=C)CC#C)=O)CC(C)CCCC1C Cc1ccc2ncccc2c1C(=O)NC1CN(C(=O)CCC(C)CN(C)C)C1 CN1CCN(C(=O)C(O)C(F)(F)F)CC1CNC(c1scnc1Cl)=O c1(C2(C)COC2)ccc(C(=O)NCC2(O)CN(C(=O)C=CCc3cccs3)C2)o1 c1(C(C)C(=O)NC2CC(CO)N(C(=O)C=Cc3ccco3)C2)ccc(F)c(Cl)c1 c1(C(N2C(C(C)NC(c3c(C)cc[nH]3)=O)CCCC2)=O)n[nH]c2nccc(Cl)c12 Cc1cc2c(C(=O)N(C(C)CNC(c3ccnc(Cl)c3N)=O)C)cccc2o1 CCC(C)(CCNC(c1ccc(O)cn1)=O)NC(C1C2CCC(=O)C12)=O N1(C(c2cc(C)c(C)o2)=O)CC2CCC1CN(C(c1c(C(C)C)cnn1C)=O)C2 c1(C(N2CCC(NC(C(CSC)C)=O)(CF)C2)=O)ccc(N)c(N)n1 N1(C(c2c(O)ncc(C(C)C)c2)=O)CC2CCC1C(NC(C1(C)CC=CC1)=O)C2 C1(C(=O)NC(C=C)(C)CC)CCCN1NC(=O)Cn1cc(COC)nn1 Cc1c(F)ccc(C(=O)NCC2CCN2C(c2ccc(Cl)c([N+](=O)[O-])c2)=O)c1F C1(OC)CN(C(=O)CCC(F)F)C(C)(CNC(c2cccc(Cl)c2)=O)C1 N1(C(CC(=C)C)=O)CC(CNC(c2noc(C3CC3)c2C)=O)OC2(CCC2)C1 c1(C(=O)NCC(C2CCOC2)NC(C(C)=C(C)C)=O)n[nH]c(C)c1C N1(CC)CCN2CC1C2=O.c1(CO)sc(N(C)C)nc1C c1(C(=O)NCC(CC(C)C)N(C)C)cc2cccnn2n1.C1=CC(=O)NC1(C)C n1(CC(N2CCN(C(=O)Cn3nccn3)C(CF)C2)=O)ccc2ccccc12 c1(NCc2c(OC)cc(F)c(C)c2)c(-c2cccc(F)c2O)ccc2c1OCO2 N1(C(CCOC(C)=O)=O)CCOC(CC(=O)NCC(O)C2CC2)C1 C(=O)(CS(=O)CCC(F)(F)F)N1CC(C(C)NC(CSCC)=O)C1 N1(C(c2n(CCOC)ncc2)=O)CCOC(C)(CNC(c2cccnc2O)=O)C1 c1(CNC(C(C)CC2CCC2)=O)ccccc1CN(C(=O)C(C)OC1COC1)C N1(C(CC=CC(C)(C)C)=O)CCCC(CCNC(=O)CN2CCCC2CO)C1 Cc1nc(C(C)C)oc1C(=O)NC(c1ccccc1)CNC(=O)CC(C)C C(=O)(C(C)(C)Cc1nn[nH]n1)N(C)CC1(C)CCC1 N1(C(C2N(C(C)=O)CCC2)=O)CCN(CCNC(C2(CC(F)F)CCC2)=O)CC1 Cc1cc(Cc2nc(-c3ccn(C)n3)nn2-c2cccnc2)ccc1Br C(=O)(C#CC1(C)CC1)NCCCN(C(=O)C(C1CCC(C(C)(C)C)CC1)O)C CC1C2CC(C2NC(=O)C=Cc2cn(C)cn2)N1C(=O)CCC(C)(F)F N1(C(C=C(CC)CC)=O)CCC(NC(=O)CSc2cc(C)ccc2C)C(O)C1 C1(C(N2CC(F)(CNC(C3CC=C(C)CC3)=O)C2)=O)Cc2ccncc2N1 N1(C(c2cn(CC)nc2C)=O)CCC2(CC2C(=O)NOCC2CCCO2)C1 c1(OC)cn(C)c(C(=O)NCCC(C)N(C)C(c2c(C)[nH]c(C)c2C)=O)cc1=O C(=O)(C(F)(F)C(F)(F)F)N1CCCC(CC2C(C)C2)CC1.c1(N)cc(=O)n(C)cn1 N1(C(c2nccc(C)n2)=O)CCN(C(c2nc(Br)cnc2N)=O)C(C)C1 C(=O)(C1CCCc2ccccc21)NC1C(C)N(C(=O)CC2COC(=O)C2)CC1 c1(C(=O)NC2CN(C(C3C(C)CCO3)=O)CC23CCC3)cc(Cl)ccc1[N+](=O)[O-] CC1(C)CC(C)(CNC(C2C(C)(C)C2(C)C)=O)CN1C(C1CC(=O)CCO1)=O N(C1CCCn2nccc21)C(C1C(NC(=O)Cc2cnsc2)C2CCC1C2)=O Cc1cn2c(n1)CCC(C(N1CCCN(C(c3cnc(C4CC4)s3)=O)CC1)=O)C2 C1(OC)CC2CCC1(C(=O)NCC1(C3CC3)CC1)C2 c1(C(NOCC(=O)NC2C(C(C)(C)C)CC2)=O)ccc([N+](=O)[O-])[nH]1 c1(NC(=O)NCC(=O)OCC=C)ccc2c(c1)CCN2C(=O)OC(C)(C)C C1(C)(CNC(C(c2cn(C)nc2)O)=O)CCCN(C(=O)CC(C)c2ccco2)C1 C(CC(=O)NC(C1CCOC1)CNC(C1CC(N2CCCC2)C1)=O)SC n1(C2(C(=O)NCC3(NC(c4c(C)[nH]cc4)=O)CCOC3)CC2)cc(C#N)cn1 CC(C)C(O)C(C)(C)C(=O)N1CCC(NC(=O)CC2CCC2)C(O)C1 N1(C(C(CC#C)C)=O)CCC2CN(C(=O)C(c3nc(C)cs3)C)CCC12 Cn1nccc1C(=O)NC(c1ccccc1)CNC(C1CCC1(F)F)=O N1(C(C(C2CCC2)OCC)=O)CCC(CCCNC(c2c[nH]nc2CC)=O)CC1 C1(CNC(CCNC(=O)CO)=O)CN(C(c2cc(O)nc(O)n2)=O)C2CCN1C2 C(=O)(CCC(=O)NC(C)CNC(=O)CN1CCSCC1)OC O=C(C1=CC2(CCOC2)C1)N1CCN(C(c2ccccc2CO)=O)C2(CC2)C1 CCCCCS(=O)(=O)CC(=O)NC1CCN(C(c2cc3cc(F)ccc3[nH]2)=O)C1 N1(C(C2(SC)CCC2)=O)CC(C)(C)C(N(C(C2CCC(C)S2)=O)C2CC2)C(C)(C)C1 C(=O)(C1CCc2ccccc21)NCC1CC2N(C(C3ON=C(C)C3)=O)C(CC2)C1 N1(C(C(CC)(C)CNC(c2cscn2)=O)=O)CCCC(O)(C2CC2)C1 c1(-n2cc(CCNC(C(CC=C)OC)=O)nn2)c(C(F)(F)F)cccc1C c1(NC(c2ccc(C)o2)COC)ncccc1S(=O)(=O)NCC1CCC(CO)O1 c1(C(=O)NCC2C(NC(c3cc(COC)on3)=O)CCCC2)ccc(C)c(C)c1 Nc1c(Cl)cc(C(N2CC(CCCCNC(=O)Cc3ccncc3)C2)=O)cc1Cl N1(C(C2(c3cc(C)no3)CC2)=O)CCCC(NC(=O)CCC2CCOC2)C1C c1(N(CC(F)(F)Cl)C)nc(N2CCC3CCC(C2)S3)nc2scnc12 C=CCCC(CO)NC(C1CCN(C(=O)CN(C)CCC)C1)=O CC(C)C(O)C(C)(C)C(=O)N1CCOC(CNC(c2ccc(C(F)(F)F)s2)=O)C1 C(=O)(CCCS(C)(=O)=O)N1C2CC(NC(c3cn(C)c(Br)c3)=O)(C2)C1 N1(C(N2CC(N3CCOC3=O)C2)=O)CCCCC1C(F)F.O=C(CCN)OC c1(NC(c2c(OCCOC3CC3)ccc(C)c2)=O)ccc(F)c2cnccc12 c1(C(C)C(=O)NCCCC2(NC(=O)CC3CCC3)CC2)cc(F)cc(F)c1 C=CCCCNC(=O)C(=O)SCCOCCOC.C1CCN1.C(COCC)N C1(CNC(=O)C=CC2CCC2)CN(C(c2cc(C3CC3)cc(Cl)c2)=O)CC1(F)F C=C1CCN(C(=O)CCN(C(c2cnn(C(F)F)c2)=O)CC)C1 c1(OC(CC)(C)C)ccccc1C(=O)N(CCC(C)NC(=O)C(C)(C)CF)C C(=O)(CC1=NNC(=O)C1)N(C(C)CNC(C1CC(F)(F)CS1)=O)CC Cc1ccc(Cl)cc1C(=O)NCC(CO)NC(=O)C(C)(C)CO N1(C(CCC(C)O)=O)CCC(C)(CNC(c2cnnn2-c2ccccc2)=O)CC1 C1(C(C)NCc2ccc(F)cc2)CC2(CC2)C(=O)O1.C1(C)(C)C(=O)N1 CC1CN(C(=O)CC(C)(C)C)CCC1NC(c1cc(CN(C)C)on1)=O CCC(C)CCCC(=O)N1CC2CN(C(=O)C(=O)NOC)CC2C1 C12(NC(CNC(CCC)=O)=O)CCOC(CNC(=O)C=Cc3sccc3C)(C1)C2 c1(CCCC=C)ccc(C(=O)NC2CN(C(=O)CC(CC)SC)CC2OC)cc1 N1(Cc2cccc(OC)n2)Cc2c(C(=O)N(CCO)CC#N)n[nH]c2C1(C)C c1(NC(=O)CONC(=O)C2(C(C)OC)CC2)ccn(C)c1 C12(C(=O)NCc3cccc(C(N)=O)c3)CCCC1N(C(=O)Cn1cccn1)CC2 c1(C(=O)NCC(C(C)C)(C)NC(=O)CCF)cnc2c(c1)NCC2 c1(CC(=O)NC(CCN(C(C2(CC#C)CCCC2)=O)C)C)c(F)cccc1Cl c1(NC(=O)OC2CC(SC)C2)ccc2cc(OC(C)C)ccc2c1 c1(C(N2CC3C(NC(c4ccc(CC)s4)=O)(C3)C2)=O)ccc(S(N)(=O)=O)o1 C=CCCCC(C)(C)C(=O)NCC(C(=O)NC1CC2CC1CC21CC1)C(C)C c1(C(C)C)c(C(=O)NCC(C2CC2)NC(c2cn(C)c(O)n2)=O)cccc1F c1(CCC)cc(C(N2CC(C(C(=O)NC(C)Cc3nncn3C)OC)C2)=O)no1 c1(C(N2CCN(Cc3ccc(C(=O)O)cc3)CC2)=O)cc(O)nc(O)n1 CCC(C)C(CNC(=O)CCCNC(=O)CCCCCC)CO C1(C(N2CCN(C(C=C(C)C)=O)C(C3CCC3)C2)=O)CC(C)CC(C)(C)C1 c1(CC)ccc(CNCC2NCCC2(C)C)nc1C C1(CNC(COC(C)C)=O)CC(F)CN1C(=O)CCC(C)c1cccc(F)c1 c1(CC(=O)NCC(CNC(c2ccc(CC)s2)=O)(C)C)cc(C)nn1CC.C1(C)CC1 C(C(=O)NCc1ccsc1C)(C(C)C)NC(c1cc(C)[nH]c1)=O C1(NC(C(C(C)C)SCC)=O)CCCC2CN(C(=O)C=Cc3cccnc3)CC12 c1(NC2CN(C(C=Cc3n(C)cnc3)=O)CC23CCC3)ncc2c(n1)CCOC2 N1(C(CCOCC)=O)CCC(CO)C(NC(=O)C(C(C)O)NS(C)(=O)=O)C1 C1(Sc2cccc(NC(=O)Nc3cc(C(=O)OC)n(C)n3)c2)CCC(C)(C)CC1 c1(COCCC2(NC(C(CC)C)c3nnnn3C)CC2)cc(C)ccc1Cl c1(C(=O)NCC(CCCC)NC(C2CC2C)=O)coc(=O)c2ccccc12 C(C(C)(CC(C)C)NC(C1CN=C2N=CNN2C1)=O)NC(c1c(OC)n[nH]c1)=O c1(OC)cc(NC(C2CCCN(C(C3CC3c3ccccc3)=O)CC2)=O)ccc1F C#Cc1cccc(C(=O)NC2CN(C(c3ccnc(Br)c3Cl)=O)CC2F)c1 Cc1cc(Cl)ccc1OCC(=O)NC(C)CNC(=O)C(n1cnc(C(N)=O)n1)C C1(NC(C2N(CCC)CCCC2)=O)CC1C1CCCN(C(=O)CCC2CC2)C1 CCCC(CCCNC(C1CC12CC(O)C2)=O)NC(=O)CC(=O)OCC C1(NC(=O)Cc2ccnc(CCC3CC3)c2)CC(F)CN1C(=O)C(=O)N(C)C c1(C(=O)NC2CN(C(C3CCN(C4CCCCC4)C3)=O)C2)ccnc(C2CC2)n1 Cc1cccc2c(C(=O)NCCC3CN(C(c4cnn5c4CCC5)=O)C3)c[nH]c12 CC1(C)CN(C(C2CC23CC(NC(=O)CCc2ncccn2)C3)=O)CCO1 C1(NC(C(c2n(C)ncc2)(F)F)=O)CCC(CNC(=O)C(F)C2CCCC2)CC1 c1(CC(=O)NC2(CNC(Cc3ccc(C)o3)=O)CC2)ccc(O)c(F)c1 c1(C(=O)NC(C2CN(C(c3ccc(Cl)cn3)=O)C2)C)cc2cccnc2[nH]1 C1(CNC(c2c(C)cc(=O)oc2C)=O)CN(C(=O)C(C)O)CCC12CCC2 Cc1cnc(NCc2cnc(F)cc2C)c(S(=O)(=O)NCCN2CCCOC2)c1 Cn1c(=O)[nH]c2cc(C(=O)NOC3CCOCC3)ccc12 c1(-c2cc(C(N3CC(n4cc(CC(C)(C)O)nn4)C3)=O)sn2)cccc(Cl)c1 C(C)(N=c1[nH]c2c(c(=NC)[nH]1)CCC2)c1n(C(c2c(Cl)cccc2Cl)C=C)nnn1 CC1=NN(C)C(=O)C1CC(=O)N(C)CCNC(c1nccn1C(C)C)=O C1(CNC(COCC#C)=O)COCC2(CCN(C(c3cccc(F)c3F)=O)C2)O1 C(=O)(NNC(=O)C(F)(F)c1cccc(O)c1)C1C(N)CCOC1 N1(C(c2c(CNC(CCCSC)=O)ccs2)=O)CCCC(C)CC1 c1(NC(=O)NC(Cc2cnc[nH]2)CO)cccc(NC(C2CCC(F)C2)=O)c1 N1(C(C(C)OC)=O)CC(F)(F)CC1CNC(C1(C)CCNC(=O)C1)=O c1(CNc2ccc(C(N)=O)c3c2cccc3)nccc2c(Br)cccc12 c1(CC)ccc(C(=O)NC2(CF)CCN(C(c3sc(F)cc3Cl)=O)C2)cc1F N1(CCC(=O)NCC2C=CC(NC(C3(CC)COC3)=O)C2)CCCCC1C C1(NC(=O)Cc2cnccc2Cl)CN(C(=O)CC23COC(CF)(C2)C3)CC12CCC2 C1(NC(C(c2cn(C)nc2)(F)F)=O)CCCN(C(=O)CCc2cnccn2)C1 C1(CN(C(=O)C#CC(=O)N(C)C)C(C)C2CC2)CCCCN1C(c1cocn1)=O C(CN=c1cc(C)c(S(=O)(=O)NCC2CCN2C)c[nH]1)=CCCC CC(C)S(=O)(=O)CC(=O)N1CCN(C(c2cc(Cl)cnc2O)=O)C(CO)C1 n1(CC)cccc(C(=O)OCCNC(=O)C(C)(C)Nc2ccccn2)c1=O C(CC(C)(C)CC(=O)N1CCC(NC(C2CN3CCC2CC3)=O)C1C1CC1)OC N1(C(CCN2C(=O)COCC2)=O)CCCCC(NC(=O)COC2CCC2)CC1 CC1CN(C(=O)CS(=O)(=O)CCO)CCCN1C(=O)C=C1CC1 C1(C)(CNC(C2C(c3onc(C)n3)CCC2)=O)CCCN1C(=O)CC(C)(C)C C(=O)(C(C(C)(C)C)NC(C1CC(=O)CCO1)=O)N1CCC(C(C#C)C)CC1 c1(C(N(CCC(=O)NC(CC)CN2CCCC2)CC2CC2)=O)cc([N+](=O)[O-])n[nH]1 C1(C(N(CCN(C(c2c(C)c[nH]n2)=O)C)C)=O)CCCN(c2cc(O)ncn2)C1 N1(C(C(C=C)C)=O)CCN(C2CN(C(c3conc3COC)=O)C2)CC1 c1(C(=O)OC)cocc1C(=O)NCCCCCNC(=O)Cn1ncc(Br)n1 CC(C)CC(CNC(c1cc(Cl)no1)=O)NC(=O)Cc1ccn(CC(F)(F)F)n1 Cc1ccc(CCC(N2CCC(NC(c3c(C(F)F)n[nH]c3C)=O)C2C)=O)cc1 C(CC(=O)N(CC(=O)NCCCC1CCC1)C)N(CC)CC c1(C(N2CCC(C(C(=O)NCc3cc(C)ns3)(C)C)C2)=O)cccc2nccn12 C1(C(N2C(C3(O)CN(C(C4CCCO4)=O)C3)CCC2)=O)CCc2nnc(O)n2C1 CCC1C(=O)Nc2ccc(C(=O)NC3CC(NC(C4CN(C)C(=O)N4)=O)C3)cc21 c1(C(N2CCN(C(c3c(OC)c[nH]n3)=O)CC2)=O)c(C)oc(C)c1C c1(C(N(CC(=O)NCC2CC3CCCC3C2)CCOC)=O)ccc2ccoc2c1 c1(CC)ccc(F)cc1C(=O)NC1CC2CC1N(C(c1cc[nH]c1C)=O)C2 CC(C)CC(C)C(=O)N(CC(=O)N(CC(C)(C)O)C)CC(C)C n1(CC)cc(C(=O)N(CC(C)NC(c2coc(C(C)C)n2)=O)CC)c(C)n1 c1(N2C(=O)CCC2)ccccc1S(=O)(=O)N1CC23CCCC2(C1)C3 c1(C(=O)NCC2C3CN(C(c4c(OC)n(C)nc4)=O)CC32)nccc2cc[nH]c12 c1(C(N(CC(O)CNC(C2(Br)CC2(C)C)=O)C)=O)ccc2c(c1)COCO2 Cn1cc(C=C(F)C(=O)NC2CCC(F)(CNC(=O)Cc3cncs3)C2)nn1 c1(C(=O)NCCC23C(CN(C(CC(=O)OC)=O)C2)CC3)cnc2n1C(C)CCC2 c1(C(c2nnnn2CC(F)F)NCC(=C)Br)c(Br)sc2ccccc12 C1(C(=O)NCCCNC(CC23CC(C)(OC2)C3)=O)CC1C1CC(F)(F)C1 C(=O)(CCCN(C)N=O)NCC1CCN(C(c2cnc(C(C)C)n2C)=O)CC1C CC1CN(C(=O)C(F)(F)C2(O)CCC2)CC(CCNC(C2CCCC2)=O)O1 c1(C(N2CCC(O)(C(F)(F)F)C2)C(=O)Nc2c(C)cccc2)cc(Cl)nc(Cl)c1 C#CCC(C(=O)N1CCC(OCCF)C1)NC(=O)Cc1csnc1C N1(C(C2C(C)C2C)=O)CCN(C(c2cn(Cc3ccccc3)nn2)=O)CC1C CP(C)(=O)C(O)C(=O)NCC1(O)CCN(C(c2cnc(N3CCOCC3)s2)=O)C1 N1(C(C2(N(C(=O)C(F)C3CCCC3)C3CC3)CCOCC2)=O)CCOC(CO)CC1 N1(C(C2CC(OCC)C2)=O)CCCCC(NC(c2sccc2SC)=O)C1 CC1CN(C(C2(Cl)CC2)=O)CCC1NC(=O)C=Cc1cn[nH]c1 C#CCCCCC(=O)NCC1(F)CCN(C(=O)C(F)OC(F)(F)F)C1 c1(C(=O)NC2CC(CC(=O)Nc3c(OC)nsc3)C2(C)C)cc[nH]c2nccc1-2 c1(C(N2CCCC2CNC2CCC2)C)ccccc1F N1(C(C(COCC)C)=O)CCC(O)C(NC(=O)C(C)(C)CSC)C1 c1(C(N2C(C(=O)NC(c3nc(C)on3)C)CCCC2)=O)coc2ccccc12 c1(NC(C2CN(Cc3ccc(Br)c(F)c3)CCO2)=O)cnc(O)c2ccccc12 C(=O)(C(C)(C(C)C)OC)N(CCCNC(c1cccc(CC)n1)=O)C(C)C c1(OC)cccc(Cl)c1NC(N1CCN(CC(C)C)C(C)C1)=O C1(NC(C2(CCCC)CC2)=O)CC2CC1N(C(c1nn(C)c(C)c1Cl)=O)C2 C12(NC(=O)C=CCN3CCCCC3)CCCN(C(=O)CCC3CCOC3)CC1C2 c1(C(N2CC(NC(C(CC)SC)=O)(COC)C2)=O)cc(=O)c(OC)cn1C N1(C(CC2CN(C)C2)=O)CC2CCN(C(c3cn(C)c(=O)n(C)c3=O)=O)C(C2)C1 N1(c2c3ncn(CCC(CC)O)c3ncn2)CC=CCC2(CCCC2)C1 n1(CC(=O)NC(C(C)NC(=O)C(C)NC=O)C)cc(CO)nn1 CC(C)C(C)(CNC(=O)Cc1nc(C2CC2)cs1)NC(C1CC2CCC1C2)=O C1(NC(c2nc(C(N)=O)sc2)=O)(CNC(c2cncc(F)c2)=O)CC2CCC1C2 C=C1COCC(C)(C)N(C(c2cccc(F)c2OC)C(=O)NCCC#N)C1 C1(CCNC(c2cc(OC)n[nH]2)=O)CN(C(c2ccncc2OC)=O)CCO1 CC1CC=C(C(=O)NCC(Cc2ccccc2)NC(C2CCOC(C)C2)=O)CC1 Cc1ccccc1C(C(C)(C)C)NC(c1ccccc1OCC(N)=O)=O c1(CC)ncc(N(C(=O)CCSC)CC(=O)OCC(C)(C)CC2CCOCC2)[nH]1 C(=O)(C(C)(C)C(=O)NC1CC(C)N(C(c2cc(C)n(C(C)(C)C)n2)=O)C1)OC CCCCC(C(=O)NCC(C1CCC1)NC(c1csc(COC)c1)=O)N(C)C CCCC(C)(O)CC(=O)NC1CC2(C1)CC(C(N1CCOC(C)(O)C1)=O)C2 O=C(C1=COCCC1)NC1CC2CN(C(=O)CC(O)C3CCCC3)CC12 C(=O)(C(C)(O)CCC)N1CC(CC(C)NC(c2c(C)nsc2C)=O)C1 c1(CC(=O)NCC(CCOC)NC(=O)CN(C)C(C)=O)cnn(C)c1.C(F)(F)F C1(C)(C(N(CC(C)O)C)=O)CCN(C(=O)CN2CCC(O)CC2)C1 C1(NC(C(C=C)C)=O)CC2CC(C1)CN(C(c1cccc(C)c1)=O)C2 Cc1ccc(C)c(C(=O)NC2(C(=O)NCC3CCCCCC3)CCCC2C)n1 CC1CCN(C(=O)CC2(CO)CC2)CC1NC(=O)Cc1nc(-c2cccs2)n[nH]1 c1(C(=O)NC2C(NC(C(C(CC)C)O)=O)CCCC2)cc(F)cc(Cl)c1O Cc1nn(C)c(=O)c(C(N2CC3(C2)CN(C(C2(C)CCC2)=O)C3)=O)c1C N1(C(COCCOC)=O)CCCC(C)(CNC(=O)CC(C)SC)C1 CC(C)CC(C(=O)N(CC(O)CNC(c1ccn2ccnc2n1)=O)C)C(C)C C1(NC(c2c(CC)n(C)nc2)=O)CC2CC(NC(=O)C(F)(F)C(O)C3CC3)C1C2 N1(C(CC2CN(C(C)=O)C2)=O)CCCC(C(C)C(=O)NCCC(Cl)Cl)C1 CC(C)C(O)CC(=O)NC(C)(C(=O)NCCC1CCC1)C1CC1 c1(C(C)C(=O)Nc2ncc(C(C)(C)C)cc2C#N)c[nH]c2ccccc12 C1(C(N(C2CCCC2)C)=O)C2CN(C(=O)CC3CC=CCO3)CC12 C12(CCNC(C3CCCC3O)=O)CCC(CC1)N(C(C1Cc3cscc3C1)=O)C2 C1(CNC(C2C(C)(C(C)C)C2)=O)CC2CCC1N(C(c1ncccc1N)=O)C2 Cc1cnc2n1C(C(=O)N(CC(O)CNC(=O)CSCC(C)C)C)CCC2 c1(CC(=O)NCC(CC)NC(c2cn3c(n2)CCCC3)=O)c[nH]c2ncccc12 C(CCC(=C)Br)NCC(=O)NCCN(CCOCC#C)C.C(C)(=O)O c1(NC(=O)NC(C)CC(c2ccc(Cl)cc2)O)ncc([N+](=O)[O-])cc1O C12(NC(=O)COC3CC=CC3)CCCN(C(c3cc(O)nc(O)n3)=O)CC1C2 C(CCN=c1nc(C(=O)NC)cc(CC)[nH]1)N(C(C(C(CC)CC)C)=O)C C1(C(N(C)CC2(CNC(c3cccs3)=O)CC2)=O)CCN2CCOCC12 Nc1ccc(C(N2CCCCC(CNC(C3CC4CCC(C3)O4)=O)C2)=O)c(F)c1 C(=O)(C(C)(C)CN(C(=O)CC#N)C)NC(C)CN1CCOCC1 C=CCC(C(=O)N1CCC(CNC2CCN(c3ccccc3)C2)CC1)NC(C)=O C1(C(=O)OC)(CNC(c2cc(CO)c(C)o2)=O)CCNC1=O.C12CC(C1)CCC2 C(=O)(C1=NOC2(CCN(C(=O)Cc3ccccn3)C2)C1)NC(CC)C(F)(F)F c1(C(N(CC(=O)NCCN(CCCC)C)C2CC2)=O)sccc1Cl C=CCC(CNC(=O)CCCF)C(=O)N(C(C)C=CCCC)C1CC1 c1(NCC(=O)NC2CC(NC(CC)=O)C2(C)C)ccc(C)c(S(=O)(=O)NCC)c1 C#CCC(CC(=O)NC(c1cnsc1)C)NC(=O)C(C)=C(C)CC N1(C(=O)NC(c2cc(C)[nH]n2)CC)C2CCC1CC(F)C2 C1(CNC(CCN(CCC)C)=O)CC(C)(C)CN1C(=O)CC1C=CS(=O)(=O)C1 C1(NC(CC(C)(F)F)=O)COC2(CCN(C(c3sccc3C(F)F)=O)C2)C1 Cc1ccc2n[nH]cc2c1C(=O)NC(C)CCNC(=O)CC1CCCC1(F)F N1(C(C(=O)NC2C(COC)C2)=O)CCCc2sccc2C1 Cc1cc(Cl)c(C(=O)NCC2CC3(CO2)CN(C(C2CC4CC4C2)=O)C3)cc1C C1(NC(c2cc(C)[nH]c2C)=O)CCCCCN(C(C2CCCCCC2)=O)C1 Cc1cccc(S(C)(=O)=NC(=O)C(C)(C)N(C)C)c1 N1(CCC)CCCN(C(C2(NC(=O)CC(C)O)CSC2)=O)CC1 C1(NC(c2ccsc2)=O)COC2C(NC(C3CC4CCC3CC4)=O)COC12 c1(C(=O)NC(C)CCN(C(=O)CC2(C(F)(F)F)CC2)C)ccsc1Cl c1(C(N(C)CCOCCNc2cnccn2)=O)cnnn1C CC1(C)CC1(C#N)C(N1CC=CC(C(=O)NCc2ccc(Cl)nc2)C1)=O C1(O)(CCNC(c2cc(CF)on2)=O)CCCN(C(C2COCCC2(F)F)=O)C1 c1(C(=O)NC(c2cn(C3CCCCC3)nn2)C)csc2c(F)cccc12 N1(C(c2ccc(C)nc2O)=O)CCC2(C=C(C(=O)N3CC4CC3C4)C2)C1 C=C(C)c1cccc(NC2CN(C(=O)C(=O)NC34CCCC(C3)OC4)C2)c1 S(=O)(=O)(c1cn(C)nc1C)Nc1ccc(C(=O)Nc2c(C)ccc(Br)c2)nc1 C(=O)(CC(F)(F)F)NCC1CC(F)(CNC(C(C)OCC(C)C)=O)C1 C1(C(C)NC(=O)N(CC(N2CC(C(C)(C)C)C2)=O)CC2CC2)CCCCC1 C#CCCCCCC(C(=O)NC1CCOCC1)N1CC2CCC1C(O)C2O N1(C(C2CC(C(C)C)C2)=O)CC=CC(NC(c2cc(-c3cnn(C)c3)no2)=O)C1 c1(N(C)C)c(CNC2C(F)CCN(S(=O)(=O)CCCl)C2)ccc2ccccc12 c1(CC(=O)NC(CC)(C)CNC(C2CC(COC)C2(C)C)=O)ccc(Cl)cc1Cl C1(C(N2CCC(CCNC(CC(C)(C)F)=O)CC2)=O)Cc2nncn2C1 C#CCC(C)(C(=O)NCC1CC12CCCCC2)NC(=O)CCN(C)CC C1(CC)CN(C(=O)CC2(C)CCC2)CCN1C(c1cc(COC)cc(Cl)c1)=O C1(C(=O)NC2(C(N3CC=CC3)=O)C(C)C2)(CF)CC(=O)C1.C1(N)C=CCCC1 Cc1cc(F)c(C(N2CCC(NCc3cn4ccsc4n3)C(C)C2)=O)c(F)c1 Cc1ccc2sc(C(N3CCCC3CNC(C3CCCSS3)=O)=O)c(C)c2c1 c1(C(N2CCC(NC(c3nc(CC)oc3)=O)C2)=O)cccc(NC(=O)OC)c1 CCC(CCC(=O)N1CCC(C)(C(=O)NCc2cc(C)cc(C)c2)CC1)OC C1(CNC(CCNS(CC)(=O)=O)=O)COCC1NC(=O)Cc1ccsc1C C1(C(=O)NC(C2CCCN2C(c2ncc[nH]2)=O)(C)C)(CO)CCCC1 N1(C(COCC)=O)C2CCC1CC(CNC(=O)CC1(C)CCOC1)C2 c12cc(F)ncc1C(=O)N2.C12(C(N)=O)CC(NC(=O)NC3CCCC3)(C1)C2 O=S1(=O)CCCN1C(c1ccc(Cn2cc(C3(O)COC3)nn2)cc1)=O C1(CC)(NC(c2cn(C)c(=O)cn2)=O)CCN(C(=O)CSc2nccn2C)CC1 C(=O)(CCCCCc1ccccc1)NCC(=C1CN(C(C(C)=CC)=O)C1)F CC(CCNC(=O)NCC=C1CCSCC1)C(C)(C)C c1(NC(C2(OCCC(=O)NC(C)CCC)CC2)=O)ccncc1 CCC(C)CC(C)C(=O)N1CCC(NC(C23CC2COC3(C)C)=O)C1(C)C C1(NC(CN(C)C(=O)C2CC2)=O)CCCCN(C(C2(n3cc(Cl)cn3)CC2)=O)C1 C(C(=O)N(CC1CCCCC1)OC)C1C(CNC(CN(CCC)C)=O)C1 N1(C(CN2CCC(C)C2)=O)CCC(O)CC1C(=O)NCC1(O)CCCCCC1 CCCCC(CC)CC(CNC(=O)NCCOC1CCOC1)CC O=C1CN(C(=O)C(=O)NC2COCC2N2CCCC2=O)CC2(CCCC2)N1 C1(C(N2C(C3(NC(C4C(=O)NCC4)=O)CC3)CCC2)=O)Cc2cccnc2C1 CN1N=C(C(=O)N2CCC(C(=O)NCCn3ncnn3)C2C2CC2)CCC1=O c1(NC(C)=O)cccc(C(C)NC2CCOC(c3ccccn3)C2)c1 c1(OC)ccc(Br)cc1CNC(C1CCC(NC(=O)CN2CCOC2=O)C1)=O N1(C(c2cc(CCC)on2)=O)CCC(C)(NC(c2cn(C)nc2SC)=O)CC1 C1(C(N2CC(OCC(=C)C)C2)=O)CCC2CCC1N2C(C1(OC)CC1)=O C=CC1CCN1C(=O)C(C)N(C(=O)CC1CCC(C)O1)C C1(NC(c2csc(-c3ccccc3)n2)=O)C2CN(C(=O)COCCCF)CC12 Cc1noc(C)c1CN1CC(CNC(c2cnc(C3CCOCC3)s2)=O)C1 C1(CC(=O)NCC2C(NC(=O)COCC3CCOC3)C2)C=CS(=O)(=O)C1 N1(C(C2C(C)C2)=O)CCC(F)C(NC(c2ccc(CCF)cc2)=O)C1 C1(C(N(CCN(C(C(c2cc(F)cc(F)c2)C)=O)C)C)=O)CCC2(CCC2)CC1 N1(C(CCOC)=O)CC(F)(F)CC1(C)CNC(=O)CNC(N)=O CC1(C)CC(NC(C2CCn3cnnc3C2)=O)CCN(C(=O)CC2OCCO2)C1 c1(C(N2CC3C(C2)N3C(=O)CC2CCCCO2)=O)cccc([N+](=O)[O-])c1O CC1COCCN(C(=O)CC2(NC(C3CC(=O)CS3)=O)CCC2)C1 Cc1cc(Cl)c(C(=O)NCC(CC(C)C)NC(C2CCN2S(C)(=O)=O)=O)s1 C(=O)(C(C)(C)CCS(C)(=O)=O)NC12C(CN(C(CCC=CC(C)C)=O)C1)CCC2 c1(C(=O)NCC(CC(C)C)N(C)C)ccc2nn[nH]c2c1 N1(C(c2[nH]cc(C#N)c2)=O)CC(NC(c2cc3ccncc3[nH]2)=O)CCC(O)C1 CCCCC(O)CNC(=O)C(CC1CC1)NC(c1ccc(CC)s1)=O CCC(C)(C(=O)N1CC2CCC(C1)N2C(=O)Cc1ccc2sccc2c1)C(F)F N1(C(c2c(OC)noc2C)=O)Cc2[nH][nH]c(=NC(=O)c3ccc(SC)cc3)c2C1 C12(C(=O)NCC(C)CN(C(=O)C(c3ccc(C#N)cc3)O)C)CCC(C)(CO1)C2 c1(C(=O)NCC2C(NC(C3CC(C)(C)OCC3)=O)COC2)cc(F)cc(N)c1F N1(C(c2cc(OC)ncc2)=O)CC2CCC(C1)C(NC(C1CC13CCC3)=O)C2 C(=O)(C(Cc1c(C)cc(C)cc1C)C(F)(F)F)OCc1ccn(CC)n1 c1(C(=O)NCCC2CC(NC(c3nc(COC)oc3)=O)C2)cccc(Br)c1 c1(C(N2CC(NC(CNC(=O)NC)=O)C(OC)C2)=O)cc(Br)c(C)cc1F C(=O)(C1CCc2nnc(C)n21)NC1CC(NC(CC(C(=O)OC)(C)O)=O)C1 Cc1cc(-c2cn(CC(C3CN(C(=O)CCN4CCCC4)C3)F)nn2)ccn1 c1(CC)cc(C(N2CC(NC(=O)CCSc3ccccc3)C3CC23)=O)sc1C C=C(C)CC(C(=O)NC(CCO)C(C)C)NC(C(CC)CN(C)C)=O CC(CNC(C1(C)CC(NC(C2CN(C)CCN2C)=O)C1)=O)CC(F)(F)F Cc1cn2c(n1)C(C(=O)NC1CC13CC(NC(=O)CSC(C)C)C3)CCC2 N1(C(c2c(NC)cccc2)=O)CC2CC1CN2C(=O)CCc1ccn(C)c1 C12(C(=O)NCCCCC3C(C)C3)CCC(CN(C(=O)C(C)(C)C(=O)N(C)C)C1)C2 n1(CC(N2CC3C(CNC(c4ncn(C)n4)=O)(C3)C2)=O)ccc(O)nc1=O c1(OCCOC)ccccc1CN(C)C.c1(C(=O)N)ccc(-c2n[nH]c(SC)n2)cc1 N1(C(CCc2scc(C)n2)=O)CCCC(N(C)C(C2CC(=C3CCC3)C2)=O)C1 C#CC1CN(C(=O)C(C)C(C)O)CCN1C(=O)Cc1cc(F)ccc1Cl C(N=c1[nH]c2c(c(=NCC3(C)CCN(C)CC3)[nH]1)COC2)C1(SC)CCCCC1 C(CN=c1[nH]c2cc(F)c(F)cc2s1)(CC(C)C)NC(C(CC)C)=O c1(C(N2CCC(N(C(CSCCOC)=O)C)CC2)=O)cnc2n1CCC(C)C2 N1(C(CCCc2scc(C)n2)=O)CCC2C(NC(c3coc(C)n3)=O)C2CC1 N(C(=NCC1CC12CC2)NCC(C)C)C(C#C)CCC C(=O)(C1=NOCC1)NCCc1cc(C(N(C(C)C2CC2)CC)=O)no1 c1(C(=O)NC(C(C(C)C)NC(c2c(C)c(Cl)ccc2)=O)C)ccn2c1CSCC2 N1(C(C(C)NC(Cn2nnc(C)n2)=O)=O)CCc2cccc(C)c21 C1(C(N2C3(C(=O)NCCC(C=C)C)CC(C2)C3)=O)CC2CCCC2C1 C(=O)(C(F)CC(C)(C)NC(=O)Cc1ccccc1C#C)N1C(C#C)CC1 N1(C(COCCOC)=O)CCN(C)C(C(N2CCCC2CF)=O)C1 C(C(O)C(F)(F)F)N(C)C(=O)NCc1nc(-c2cc(Br)cs2)cs1 C1(C(=O)NCc2[nH]nc(COC)n2)CCC(O)CN1C(c1ccccc1F)=O CCC(CC(=O)NCC1CN(C(C2(C)NC(=O)NC2C=O)=O)CC1(F)F)C(C)C c1(C(C)C)nc(C(=O)NC2COCC2NC(=O)C(C)CN(C)C)co1 C1(C(=O)NCC2CC(NC(C(C)(C)c3ccccc3)=O)C2)Cc2ccccc2S1 C1(C(C)NC(=O)NCCOC)CCCN(C(N(c2scnc2C)C(C)(C)C)=O)C1 CCCC(F)(F)C(=O)NCCC(N1CCC(C)C1C)=O CC(=O)CC(C)(C)C(=O)N1CC2C(C(=O)NCC(C)OCCO)C2C1 c1(C(N(C2CCCN(C(C(C)Sc3ccccc3)=O)C2)C)=O)cccc(O)c1Cl C1(C(=O)NC(c2nc(C(N3CCC(C(F)(F)F)C3)=O)co2)C)(CC)CCCC1O O=C(CCS(=O)(=O)c1ccc(Br)cc1)NC1COCC1N1CCCC1 c1(C(=O)NCC(CCOC)NC(c2nnn(C)c2C)=O)ccc2oc(S)nc2c1 CCCCCC(CC)C(=O)N1CC(C(=O)Nc2cc(Cl)ccc2F)CC(C)(C)C1 c1(CC(=O)NCCC(C)(C)NC(c2cncc(OCF)c2)=O)c(F)cccc1Cl Cc1c(CC(=O)NCC(C)CNC(=O)CCc2ccc(O)nc2)cnn1C CCCC(C(=O)N1CC(C)(CCC(N2CCC=C(Cl)C2)=O)C1)N(C)C c1(CCOC(CNC(CNC(C(C)CC)=O)=O)CNC(=O)COC)nccn1C CC(C)CC(=O)C(=O)NCc1ccc(SC(F)F)cc1 CCCC(C)(C)CC(=O)N1CC2CC2(C(=O)NCc2cnnn2C)C1 c1(C(N2C(C(CCC)C)CCC2)=O)cc(Br)c(I)s1 c1(C(=O)NC(CC(C)C)CNC(=O)C=C2CCCCC2)ccc(N)cc1Cl N1(CC)CCC(C)(C2CC2)C1.c1(C(=O)NC2CC(NC)C2(CO)CO)cc(C)nc(C)c1 c1(C(=O)NC2COCCN(C(c3ccc(CC)s3)=O)C2)cc2ccccn2c1 CC(C)(CCCNC(C1CCN(C(N)=O)CC1)=O)NC(=O)C=Cc1ccccn1 C1(NC(C2C(NC(c3ccc[n+]([O-])c3)=O)CCO2)=O)CCn2ccnc2C1 Cc1cc(F)cnc1C(N1C2CCC(C2)C1CC(=O)NC(C)CC(C)C)=O c1(C(=O)NC(CC)C(O)C(=O)OC)c2c(nn1C)CCC2 c1(C(C)C)ccc(NNC(=O)C2CC3(CCCC3)CN2C(=O)OC(C)(C)C)cc1 c1(C(N(CCCNC(c2ccc(SC)o2)=O)CC)=O)cc2cc(F)c(F)cc2[nH]1 c1(C(=O)NCC2C(NC(C3(CC=C)CCOC3)=O)CC2)ccc(C)nc1C N1(C(C(COC)(C)O)=O)C2CCC(C2)C1CNC(=O)Cc1cccnc1C(C)=O N1(C(c2n(CCC)ncc2)=O)CCC2(C1)CN(C(=O)C(C)CSC)C2 C1(C(=O)NCC2(CNC(c3ccc(Cl)o3)=O)CC2(F)F)CCC2(CC1)CC2 Cc1nn(C)c(Nc2cccc(COCCc3ccccc3)c2)c1Cl c1(-c2onc(-c3[nH]c4ncn(C)c4c3)n2)c(F)ccc2[nH]ccc12 C1(CNC(C2CC(NC(C(C)Cn3ccnc3)=O)C2)=O)COCC1(C)C C1(C(N2CCC(NC(c3cc(O)ncn3)=O)C(F)C2)=O)CC1C1CCOCC1 C1(CC)CN(C(=O)CC2CC2(C)C)CCC1Nc1nc(-n2cccn2)cc(C)n1 C(=O)(C(C)(C)O)C(=O)CC1CC(C(N(CCC(N)=O)CC)=O)C1.N CC1CC(NC(C2(S(C)(=O)=O)CC2)=O)CN(C(c2ccc(C(O)CF)cc2)=O)C1 c1(CC(=O)NCc2cccc(NC(C(C=C)(C)C)=O)c2)ccc2c(c1)CC(=O)N2 C1(COCC(N2CC(OC(=O)COC(C)C)C2)=O)CCC(F)C1 C1(O)(CC)CCCN(C(C(=O)NCCCF)C(C2CCC2)OC)C1 C(=O)(CC(C(C)C)NC(=O)CC1CC2CCC1O2)NC(c1cccnc1)CC C1(CNC(COCC(=C)C)=O)CC2CCC1N2C(=O)CC1CCN(C)C1 c1(CN(C2CCCC2)C(C=C(C)C)=O)nc2sc(C)cn2c1C(=O)OC(C)(C)C C=CCC(CC(=O)NC1CN(c2ncco2)C1)NC(=O)CCCC(OC)OC CCC(C(C)C)NC(=O)C#CCNC(C1CN(C(C)C)C1)=O C(=O)(C1=NOC(C2(O)COC2)C1)NC1(CCOC)CCN(C(c2ccco2)=O)C1 c1(C(=O)NCCOCCNC(C2C(C=C)C2)=O)ccc(OCCOC)cc1.CCC c1(NC(C(c2ccc(Cl)c(Cl)c2)N(C(CC)C#N)C)=O)ccc(C)cc1C N12CCCC(O)(C1)C2=O.c1(C(=O)OC)cc(CNn2cc(Cl)cn2)cs1 C(=O)(C(F)C(F)(F)F)NCC1CN(C(c2c(C)sc(O)n2)=O)C1 N1(C(CCC(N)=O)=O)CC2CCN(C(=O)C(O)CC3CCCCC3)CC12 c1(C(=O)NCCN(C(c2c(CCCC)onc2C)=O)C)cc2c(C)cccn2c1 c1(C(=O)NC2CC(C(C)O)C2)cccc2nn(C)cc12 C1(CNC(C=CC=CCC)=O)CCN(C(c2cc(C)[nH]n2)=O)CC1(F)F C1(NC(c2ccn(C(C)(C)C)n2)=O)CN(C(=O)Cn2ccnn2)CC1n1ccnn1 c1(CNC(C2N(C(=O)CNS(=O)(=O)C3CC3)CC2)=O)cc2ccsc2s1 c1(C(C(C)NC(C2(C)CN(Cc3ccns3)C2)=O)=O)cnc2ccccn2c1=O N1(C(C2C=CCN(C(C(C=C)(C)C)=O)C2)=O)CCc2nncn2CC1 c1(C(N2CC(N(C(C(C)OC)=O)C)C(C)(C)C2)=O)cc(O)nc2[nH]c(=N)ccc12 C1(CC(N2CC(NC(c3cnc(CC)[nH]3)=O)C(F)C2)=O)CCC2(CCC2)O1 N1(C(c2ccnc(O)c2)=O)CCN(C(c2ccc([N+](=O)[O-])o2)=O)C2CCC12 C=CC(CC)CC(=O)N1CCOC(CN(C(=O)C(F)(F)CC2CC2)C)C1 C1(C(=O)NCC(C2CC2)NC(C2(COC)CCCO2)=O)CN2CCCN1CC2 C(C)(C)(CC(=O)NCCNC(=O)C(CC#N)c1ccccc1)OC C(=O)(CC(C)CNC(C1(C)CC(C)=NO1)=O)NC(C#C)(C)C c1(C(=O)NCC2C(NC(=O)COc3cccnc3)C2)ccc(F)c2ccsc12 Cc1ccnc(O)c1C(=O)NCC(C)(C)NC(=O)C(c1cccc(Cl)c1)C C1(N(C)C)CC(CC(=O)OC(C2CC(=C3CCC3)C2)C#N)C1(C)C N1(C(COCc2n(C)ccn2)=O)CCOCC1CNC(C1CNC(=O)C1)=O C(=O)(C(C)(C)C(F)(F)F)N1CC(C)(C)C(CNC(=O)C(F)=C2CCC2)C1 CN1CCN(C(c2scnc2C2CC2)=O)CC1CNC(C1CC1C(N)=O)=O N1(C(CNC(CC)=O)=O)CC(NC(=O)C(=O)NC(C)CSC)C1 C1(NC(C(C)OCC#C)=O)CC2CN(C(c3ccc(C(F)F)cn3)=O)CC2C1 C(=O)(C(CC(F)F)NC(=O)OCC)N1CC(OC(C2CCC(CC)CC2)=O)C1 C1(CC(=O)NCCCCCN(C(c2cc(COC)sc2)=O)C)CCCNC(=O)C1 C(c1ccc(Cl)cc1F)=CC(N1CCC(NC(C2CCC(=C)CC2)=O)C(F)C1)=O C1(C(=O)Nc2c(SC)noc2)CN(C(=O)CSCCC(C)C)CCO1 c1(NC(CN(CCCC)C)C)ccc(S(=O)(=O)NC2CCCC(F)(F)C2)cc1F c1(CC(=O)NC23C(NC(C4=C(C)CC4)=O)CC(CC2)C3)cccc2c1CCC2 N1(C(C2(CC)CC2)=O)CCC(NC(c2ccc(Br)c(C)n2)=O)C(O)C1 c1ncccc1[N+](=O)[O-].Cc1nc(C(=O)NCC2(CO)CN(C(C)C)C2)[nH]c1C N1(C(CC2CC(C(C)C)OCC2)=O)CC2(CCN(C(=O)C=Cc3cn[nH]c3)C2)C1 c1(C(N2CC3CC(NC(C4(O)CCSC4)=O)C(C3)C2)=O)cnn2c1OCCC2 C1(C#C)(C(=O)NC(C2CCCC2)C#C)CCN(C(=O)C(CC(C)(C)C)OC)CC1 C1(C(=O)NC2C=CCN(C(c3c(C)cns3)=O)C2)SC2C=CC1CC2 N1(C(C(C)C(F)F)=O)CC2CC(C1)CN(C(=O)C(C)Oc1ccccc1F)C2 N1(C(Cn2c(C)nc(C)n2)=O)CCCCC(NC(=O)CN2CCS(=O)CC2)CC1 c1(C2(C)CC2)ccc(C(N2CC3CC2C3NC(C2(CO)CCCC2)=O)=O)cc1 C(N=c1[nH]cnc(Cl)c1Br)C1OCC(CNC(c2ccc(CN(C)C)[nH]2)=O)C1 N1(C(C2(OC)CC2)=O)CCC(=CCNC(=O)Cn2cnc(C#N)n2)CC1 C1(C(N2CCC(NC(=O)CCc3ccc(Cl)s3)(CO)C2)=O)CCC(F)(F)CC1 C12(C(N(CC(CNC(C3(COC)CCC3)=O)(C)C)C)=O)CCCC1C2(F)F O=C1CC(CC(=O)NC2CN(C(=O)Nc3ccccc3)C2)CCCN1 c1(SC)ccc(C(N2CC(N(C(=O)C(C)C(C)C)C)C2)=O)cc1[N+](=O)[O-] C1(C)(C(=O)NCC2C(C)(C)C2C(=O)NCCCCOC2CC2)CCCC1O C12(NC(c3cc[nH]c3C3CCC3)=O)CCC(CNC(C3(CF)CC3)=O)(CC1)CC2 C1(CNC(C2C(CCC)CCC2)=O)CCC(C(N2CCSC(C)C2)=O)CC1 c1(C(=O)NC(C)CCCNC(=O)CC2(CC3CCO3)CC2)ccc(F)cc1 Cc1cc(C(N2CC(NC(c3cccn3C(C)C)=O)C(O)C2)=O)cc(C(F)F)c1 C1(C(=O)NCC2=CCN(C(c3ccc(C)o3)=O)CC2)Cc2ccccc2N1C N1(C(C)C)CCCC(C(=O)NCC2CC(NC(=O)C(C)(O)C3CCC3)C2)C1 C(=O)(CCCCN=[N+]=[N-])NCC(C(=O)N1C(CC)CCCC1)(C)CC c1(C(=O)NCC(CCNC(=O)CN2CSCC2=O)O)c(F)cccc1F Cc1ccn2cc(C(=O)NC3CCCCC3NC(C3(C)C=CCC3)=O)nc2c1 c1(CC)noc(C(=O)N(C)CCN(C)C(C2CCN(C(C)CC)CC2)=O)c1C CC1CN(C(c2cnsc2)=O)CC(C)CN1C(=O)CCc1nnc(O)nc1O c1(C(N2C(C)CC(NC(CCNC(=O)NC)=O)C2)=O)snc2ccccc12 c1(C(=O)NC2CN(C(c3cn[nH]c3)=O)CC2F)cc2c(nn1)OCCS2 Cc1nc(C)c(C(=O)N(C2CCN(C(C3CCOC3)=O)C2)C)o1 C1(C(=O)NC2C3CN(C(C(c4ccccc4)OC)=O)C2C3)CC2CCC1CC2 C1(CC)C(C(=O)NCCSC(F)F)CCCN1C(C1CSC1)=O N1(C(c2nc(CC)oc2C)=O)CCC(NC(c2coc(C3CCC3)n2)=O)CC1C c12cnn(c1)CC(=O)NCCC1(CC1)NC(=O)CC1CCN(C1)C2=O.CC.CC C(CC(C(=O)NCCn1cnc(C(N)=O)n1)NC(=O)C=CC(F)F)SC c1(C(=O)NCCCC(C)NC(C2(Cl)CC23CCC3)=O)cnc2ccoc2c1 Cc1cc(C(=O)NC2CCCC(C(=O)NC3CC4C=CC3C4)CC2)cc(C)c1 Cc1ccn2cc(C(=O)NC(C3CCN(C(=O)C(F)CC4CCC4)C3)C)nc2c1 Cc1cc(=NCc2nc(N(C)C)n[nH]2)[nH]c(N2CC=C(Cl)CC2)n1 C1(C(N2CCC(NC(c3cnn(C(C)C)n3)=O)C2)=O)CC2(CCCC2)C1 c1(N(C2CCN(C(c3c[nH]nc3C3CCC3)=O)CC2)C)ncc2c(ncn2C)n1 c1(CC)ncccc1C(=O)N(CC(=O)Nc1ccc(OCC=C)cc1)CC C1(O)(CN(C(=O)C=Cc2cn(C)cn2)C)CCN(C(=O)C=Cc2ccoc2)C1 [N-]=[N+]=NC1CC(C(N2CCC(CC3CC3)CC2)=O)N(C(=O)C(O)C(F)(F)F)C1 Cc1cn2cc(C(N3CCC(CNC(=O)CCCCC(N)=O)C(O)C3)=O)sc2n1 C1(CNC(CN(C)C(c2ccccc2)=O)=O)CCCC1NC(c1nonc1N)=O C(C)(C(F)(F)C(F)(F)F)NC(C(C)Oc1ccc(Cl)cc1)=O Cc1cnc(CN2CCN(Cc3cccs3)CC2)cc1Br N1(C(C2CCCC(C)(C)O2)=O)CCC2CCCC(C1)N2C(=O)C=C(Cl)Cl c1(C(=O)NC2COCCN(C(=O)C(O)C3CC3)C2)ccc2c(c1)S(=O)(=O)NC=N2 C1(N(C(c2c(SC)ccs2)=O)C)CCCN(C(=O)C(C2CC(F)(F)C2)O)C1 Cc1nc2ccc(C(N3CC4CC(C3)N4C(c3c(Cl)c(C)nn3C)=O)=O)cc2[nH]1 C(CC(C)C(=O)NCC(CC(C)C)NC(c1c(Cl)n[nH]c1C)=O)OC C=CCC(CCC=C)NC(c1ccc(CC)cc1NC)c1nnnn1CCCC C1(CNC(CC2COCC(C)O2)=O)CC2(C1)CN(C(=O)C1=NOCC1)C2 C1(C)(C(N(CCCCCC=C)C)=O)CCCN(C(=O)C(C(C)C)NC(C)=O)C1 Cc1nn(C)c(Br)c1C(N1CCCC1C(c1ccccc1)C)=O CS(=O)(=O)c1ccc(C2CCCN2C(CCCCCCCCCCO)=O)cc1 Cc1coc(C)c1NC(C1(NC(=O)COC(C)C)CC(O)C1)=O CC1(C)CCCCC1C(N1CC(C2CC2C(N2CC(C(C)(C)O)C2)=O)C1)=O N1(C(C(CCOCCO)NC(C(c2cnn(C)c2)C)=O)=O)CCOC(C)(C)CC1 N1(c2nccc(=N)[nH]2)CCC2(CC1)CC2C(N1CCCC1c1cccnc1)=O C1(NC(CC(C)OC)=O)CN(C(=O)CCSc2nccn2C)CCC1C(F)(F)F C(CNC(C1CC1CNC(=O)CC1OCCC1C)=O)(C(F)(F)F)OC N1(C(C2(C#C)CCCC2)=O)CCCC(NC(=O)C(C)(O)c2ccccn2)CC1 c1(C(=O)NCCOCCNC(c2ccn(C)c2)=O)cncc(P(C)(C)=O)c1 C12(OCC)CCC(C(=O)N(CC(C)NC(c3ccc(=O)n(C)n3)=O)CC)(CC1)C2 c1(N(C(C2C(C=C)C2)=O)C)ccc(C(=O)NCCNC(=O)C(C)CCOC)cc1 C1(O)(C(=O)NCC2C(NC(C3(O)CC(c4ccccc4)C3)=O)C2)CCSCC1 c1(C(=O)NC(CN(C(C(C)C(F)F)=O)C)C)cc(N)c2ncccc2c1 C1(CNC(C=CC(CC)C)=O)(CNC(=O)Cc2ccccc2)CCCC1 C=C(C)C1OCCC1C(=O)NCC1CN(C(c2ccc(F)c(C)c2)=O)CC12CC2 Cc1ccnc(O)c1C(N1CCN(C(c2cccc(Br)c2Cl)=O)CC1)=O C1(OC)CCC2(C(=O)NCC(C(=O)N(CCF)C(C)C)OC)CC12 C1(CNC(C(C)OCCOC)=O)CN(C(c2ccc(C3(C)CC3)cc2)=O)CCO1 C1(NC(Cc2c(C)con2)=O)CCN(C(c2nnsc2C)=O)C(C)C1 c1(C(=O)NCCC(C)NC(=O)Cc2cscc2F)n[nH]c2ccc(Cl)cc12 N1(C(C(C)CO)=O)CCCC(O)(Cn2cc(CCn3cncn3)nn2)CC1 S(=O)(=O)(c1ccc(NCc2cnc(C)n2C)c(Cl)c1)NC1C2(CC(OC)C2)C1 C(=O)(C1=CC(C)CC1)NCC1(C)CC(NC(COCCC=C)=O)C1 CC1CC(NC(c2cccc(=O)n2C)=O)CCN1C(=O)Cc1cc(F)ccc1O N1(C(c2oc(CC)c(C)c2)=O)CCC(CO)(NC(c2cc(CF)on2)=O)C1 C1(C(N(C(C(=O)NCc2c(C)nco2)C)C)=O)CC(O)CN1C c1(C(=O)NCC=CCNC(C2(O)CC(C)(C)C2)=O)cc(C2CC2)nc(O)c1 Cc1nn2ncccc2c1C(N1CC2CCC(C1)N2C(=O)CN1CCC(C)C1)=O C1(NC(c2n(CC)ncc2Cl)=O)CN(C(=O)CCOc2cccnc2)CCC1C C1(CSc2c(OC)ncc(C(=O)OC)c2)CC(C)CC2(CC2)C1 N1(C(c2cccc(OC)c2)=O)CCC(N=c2ccnc(CC3CC3)[nH]2)CC1C O=C1CN(CC(=O)NC2(C(N3CCC(C(F)F)C3)=O)CCCC2)CCN1 Cc1cccc(Cl)c1CC(=O)Nc1cccc(NC(=O)C(C)CSC(F)(F)F)c1 c1(C(=O)OC)c(NC(C2CC2NC(=O)Cn2cncn2)=O)cccc1Br C(=O)(C(F)C(F)(F)F)N1C(C2(NC(CC=C)=O)CC2)CCC1 c1(CSCCC(=O)NC2CCC(CNC(c3ccns3)=O)C2)ccccc1 C1(NC(C2CCC(=O)N2)=O)CC2CN(C(=O)CC3CC3(Cl)Cl)CC12 N1(CCC)CC(C(=O)N(CC(CC)NC(=O)CCCc2ccncc2)C)CC1=O C1(NS(C(=O)NCC2CC2)(=O)=O)COCCN(C(=O)COc2ccccc2Cl)C1 c1(C(=O)NC2CC(C(=O)Nc3cccc(OC)c3)C2)ccc(C)cc1Cl c1(OC)ccc(CC(=O)NCC2(O)CN(C(C3CC(=C(F)F)C3)=O)C2)c(Cl)c1 C1(C(=O)NCC2N(C(c3nccc(C#C)c3)=O)CC(O)C2)CCC2(CCC2)CC1 C(=O)(C(CC1CCOCC1)NC(=O)CCOCC1CC1)NC(C#C)C1CCC1.CN c1(OCCC)ccc(Cl)cc1C(=O)NCC1CCN(C(=O)C=C2CCC2)C1(C)C n1(CCC(=O)NC(C(C)C)CCNC(=O)C=Cc2cc[nH]n2)ccc(O)nc1=O c1(C(N2CC(C)(NC(Cc3ncc(CC)[nH]3)=O)C2)=O)ccc2ncsc2c1 c1(C(=O)NC2CC(O)(CNC(C3C(C)OCC3)=O)C2)ccc(C2(F)COC2)cc1 c1(CC(C(=O)N2CC2)NC(=O)CNC(=O)C2CC2)ccc(Cl)cc1Cl.CCS C1(C(N2CCC(NC(CC)=O)C2)=O)CC2(CCN1C(=O)C#CC1CCC1)CC2 C1(N(C(C2CC2(Cl)Cl)=O)CC)CCCN(C(=O)C(c2ccccc2)N(C)C)C1 Cn1cc2c(n1)CCC(C(=O)NC13CC(NC(c4cncc(Br)c4)=O)(C1)C3)C2 N1(C(c2c(C)cccc2F)=O)CCC2(CC1)CC2(C)C(=O)N(CCC#N)C C=CC(C)(O)C(=O)NCC(C)NC(c1ccc(-c2cscn2)nc1)=O c1(COC(C23CCC(OC)C2C3)=O)ccccc1[N+](=O)[O-].N12CCC(C13CC3)C2=O c1(OCC(=O)NC(c2c(C)cc(Br)cc2)C)cc(Cl)c(Cl)cc1Cl C1(NC(CCCNC(=O)NCCC)=O)CC2(CN)CC1C1CC21 N1(c2n(CC)c(C3CCC4(CCC4)O3)nn2)CCC(F)(F)CC1 O=C1CCC(CNC(=O)CC2CC(O)CN2C(=O)Cc2ccoc2)CN1 C(=O)(C(F)(F)C(F)F)NC1CC(N(C(C(c2cccc(O)n2)C)=O)C)C1 CCC(CC(C)C)C(=O)N1CCC2C(C1)CN2C(c1cncc(C)c1)=O c1(C(=O)NCCCC(C)NC(C2CC(=O)OC2(C)C)=O)ccc(C2CC2)cc1F c1(C(N(CC(C)N(C(CCNC(COC)=O)=O)C)C)=O)nccc(Cl)c1O C1(CNC(COC(CC)C)=O)CCC(CNC(=O)C(c2ccc(Cl)cc2)O)CC1 C1(CNC(C2(CCOC)CCC2)=O)CC2(CC2)CN1C(=O)CCc1cc(C)no1 Cc1nc2c(s1)C(N(C)CCCC(O)CNC(c1ccccc1)C)CCC2 Cn1ncc2nc(SCCCN=C(N(C)C)N(C)C)c(C(F)(F)F)cc12 C(=O)(C(CC)C(C)(F)F)NC1(CO)CCN(C(CC(CC)SC)=O)CC1 c1(C(=O)NCC2C(NC(CCC(=O)OCC)=O)C2)cn2ccnc2cn1 CCCC(CC)CC(=O)NC1(CCNC(c2cc(C)c(CC)o2)=O)CCCC1 C1(NC(C(c2ccoc2)SC)=O)CCCC1CC(=O)NC1(C(F)F)CCCC1 c1(C(=O)NC2C(NC(CCOCCOCC)=O)CCCC2)cc2nnn(C)c2s1 c1(C(N2CC3CC(CNC(=O)C4=COCC4)C3C2)=O)cccc2cnnn12 C(CCC1CCC1)(C(=O)NOCC(O)CO)NC(c1ccc(OC)cn1)=O C=C1CC(C(=O)NC2CC(O)(CCC)C2)(CNC(=O)Cc2ccccn2)C1 C1(NC(=O)CN2CC3CC3C2)C=CCN(C(C2(c3ccccc3)CC2)=O)C1 N1(C(C(CC)n2cccn2)=O)CCC(C(O)CNC(C2CCC23CCC3)=O)CC1 C1(C(N(CCC(C)NC(c2ccc(SC(F)(F)F)o2)=O)C)=O)CCCOC1 c1(C(=O)NC(CNC(CC2CC(OC)C2)=O)C)ccc(CO)cc1 C1(CN=C(NC(CC)CC)NC2CCc3nccn3C2)CC(F)(F)CCC1(C)C C1(C(=O)NCCc2cc(C(N3CC(OCC(N)=O)C3)=O)no2)CC(F)(F)C1(C)C C1(CCNC(C=CCC)=O)CN(C(c2cc(N)ccc2Cl)=O)CCS1(=O)=O c1(NC(=O)NCc2ncc(C(C)(C)C)o2)ccc(-c2cn[nH]c2)cn1 Cc1cc(=NC(C)c2nncs2)[nH]c(=NCc2cnc(C(F)(F)F)s2)[nH]1 CC1CCC(CC(=O)NCC2(CNC(C3COC(=O)N3)=O)CCC2)CC1 c1(OC)ccc(OC)c(C(N2CC3(CC3)CC2CNC(c2c[nH]c(Br)c2)=O)=O)c1 Cc1cc(F)cc(C(N2CCC(C(C)NC(=O)CCCc3cnn[nH]3)C2)=O)c1C N1(C(C2C(C)CC=CC2)=O)CCC(F)C(NC(=O)C2=COCCC2)C1 S(=O)(=O)(c1ccc(F)cc1)N1C(C(=O)Nc2c(OC)cccc2)CCCC1 c1(CC(N2C(CNC(C3CCCS3)=O)C=CC2)=O)ccc(F)cc1Br C(=O)(C1=C(c2ccccc2)CCCC1)NC1C(NC(c2csc(C)c2C2CC2)=O)C1 c1(C(=O)NC(CC)CN(C(=O)Cc2cnns2)CC)coc2c(C)cccc12 C1(F)(C(N(CCN(C(C(C)CSCc2cccnc2)=O)C)C)=O)CC2(CCC2)C1 CC1CCn2ncc(C(=O)NCC3CCN3C(=O)C#CC3CCCO3)c2C1 c1(CNC(=O)Nc2c(C(=O)OC)nc(C3CC3)o2)ccc(O)c([N+](=O)[O-])c1 c1(C(=O)NC2C(OCC)CN(C(=O)COCCSC)C2)ccc2[nH]ccc2c1F N1(C(c2cc(-n3ccnc3)no2)=O)CCOCC1c1cn(CC2CCCO2)nn1 N1(C(C(C)C(C)O)=O)CCC(F)(F)C(CNC(=O)CC2CCCCN2C)C1 CCC(CC)(CCNC(=O)C1=CC(C)(C)C1)NC(=O)CC1CCCC1C c1(-c2cn(CCNC(=O)Cc3ccc(Cl)c(F)c3)nn2)ccc2c(c1)NC(=O)C2 c1(C(N2CCC(C)(NC(C3C(C(C)O)C3)=O)C2)=O)ccc(Cl)c(C#N)n1 S(=O)(=O)(CCC(=O)NC1COCC1NC(=O)COCP(C)(C)=O)N(C)C Cc1ncc2n1CC(C(N1CCCCC1CN(C)C(c1cnco1)=O)=O)CC2 C(c1ccco1)=CC(N1CSCC1C(=O)O)=O.N12CCC1C2=O Cc1cc(C(N2CCCC(C(N3CCN(C4CCOC4)CC3)=O)C2)=O)cnn1 c1(CC)c[nH]cc1C(N1CC(N(C)C(c2cc(CO)[nH]n2)=O)C1)=O N1(C(C2C(OC)CC2)=O)CCN(C(c2c[nH]c(C#N)c2)=O)CC1c1cnn(C)c1 C1(C#N)(C(=O)NCC2C(C(=O)NCCC=C=C)CC2)CCOC1 CC(C)C(C)CC(=O)NCc1ccc(C(=O)NC2CC(=O)N(C3CC3)C2)cc1 N1(C(C)C(=O)Oc2ccccc2)CC(COC(c2cnccn2)=O)OCC1=O c1(CC(=O)OCc2cnn(CCNC(C)(C)C)c2)cncc(C(F)(F)F)c1 N1(C(C2(CN(C)C)CCCC2)=O)CCC2CCCN(C(c3cc[nH]n3)=O)C2C1 c1(CN2CCC(CNC(c3nn(C)c(O)c3)=O)C2)ccc(F)c(S(C)(=O)=O)c1 C1(C(=O)NC(c2ncc[nH]2)C)CN(C(=O)CC2CC2(C)C)CC1F c1(C(=O)NCC2CC(CNC(C3C(C)CC3)=O)C2)cc(C(N)=O)co1 C(C(C(=O)NCC(C(=O)N1CCC(N(C)C)C1)C1CCC1)OC)OC.C(C(N)=O)O c1(C(N2CC(CO)CC(C)C2)=O)cnc2ncn(C)c2n1 S1(=O)(=O)c2cccc(c2)CN1C.c1(NCc2onc(CC)n2)ccc(C#N)nc1 C1(C(=O)NC(C(N2CC(COC)C2)=O)C2CCCO2)CC(C)(C)CCO1 c1(OC)ccncc1-c1nc(-c2ccsc2)nn1CCc1ccccc1 c1(C(N(C2CCCN(C(=O)C(C)(C)C3CCCO3)C2)CC)=O)cn(C)nc1O c1(NC(C2(C)CCN2C(=O)CSc2ccccc2)=O)cccc2c1OCC2 C(=O)(C1=CCC(NC(C2C3CCCCC23)=O)C1)NC1CC(C(C)C)OCC1 c1(Nc2ccc(C(=O)NC3CCC3)cn2)ncc(Br)nc1Cl.C12CC1NC2=O S(=O)(=O)(c1ccc(NC2CC(NCCc3ccccc3Br)C2)c(F)c1)N(C)CC C1(C(=O)NC(C(C)NC(c2ccc(CC)o2)=O)C(C)C)C2CCC(F)(F)C12 N1(C(CN(C)C(c2nc(Cl)cs2)=O)=O)CCN(C(c2cnc(S)nc2)=O)CC1 Cc1cccc(F)c1C(=O)NCC1CC(C)N(C(=O)Cn2cc(N)cn2)C1 CCCS(=O)(=O)N1CCC(C(C2CC2)Nc2ncn(-c3ccccc3)n2)C1 N1(C(c2nc(COC)oc2)=O)CC2(CCCC2NC(C2CC3(CCC3O)C2)=O)C1 C(=O)(C1=C(C)N(C)c2ncnn2C1)N1CCCC(CN(C(C(C)(C)SC)=O)C)C1 c1(NCCNC(c2c(OC)c(Cl)sc2)=O)cc(O)nc(C2CCC2)n1 C1(C(N(C(c2cn(-c3cccc(C)c3N)nn2)C)C)=O)CN(C)C(=O)CCO1 C1(C)(C(=O)NCc2ccc(C)nc2)CCCN(C(=O)CN2CCCC2)C1 c1(CNCC2CN(C(=O)OC(C)(C)C)C2)ccc(C2CCOC2)cc1 c1(CC)cccc(NC(COCC2(C)CCC(NC(=O)Cc3cc[nH]n3)C2)=O)c1 C(=O)(C(CC(C)C)NC(=O)NCC1CC(OC(F)(F)F)C1)NCC C(=O)(C(C)(C)C(O)C(C)C)N.Cc1nn(CC(=O)N(Cc2ccccc2)C)c(=O)o1 Cc1cc(C(=O)NC(C2CCOC2)CNC(c2ccnnc2O)=O)cc(C)c1F N1(C(C(C)c2ccco2)=O)CC(C)(NC(=O)C(F)Cc2ccccc2)C1 c1(CC)ccc(C(=O)NCc2ccccc2Cc2n[nH]c(C)n2)nc1 c1(C(=O)OCC)ccc(NCC(C)CNC(=O)Cc2ccoc2)nc1 [N-]=[N+]=NCCCCNC(c1csc(CNC(=O)C(O)C2CC2)c1)=O N1(C(c2ccn(CC)c2C)=O)CCCC(C2CC2NC(c2ccc(F)s2)=O)C1 c1(N2CC(F)CC(NC(C3CCS(=O)(=O)N3)=O)C2)nc(Cl)nc2ccccc12 C1(CN=c2nc(N3CCN(S(C)(=O)=O)CC3)cc(C)[nH]2)CCC2(CCOCC2)N1 c1(C(N2C(CCNC(c3[nH]cc(CC)c3)=O)CCC2)=O)nccc(C(C)(C)C)n1 N1(C(CCC(C)N)=O)CC2OCCN(Cc3ccccc3)C2C1 N1(c2nccc(SC)n2)CC2CCCC(NC(C3(C)CC3)=O)C2C1 CC1(C(=O)NC(CNC(c2ncc(F)cc2N)=O)C2CC2)CCCCC1(F)F C1(CNC(c2c(F)ccc(C)c2)=O)CN(C(C23CC(C2)C3)=O)C2(CCC2)C1 C12(C(N3CC(NC(C(C)c4cncs4)=O)C3)=O)CC1COC21CCC1 c1(OC)csc(C(=O)NC(C2CN(C(C3(C)CCC3)=O)CCO2)C)c1OC C1(NC(c2c(OC)n[nH]c2)=O)CN(C(c2ccnn2C(C)C)=O)C(C)(C)C1 N1(C(CCCNC(=O)OC)=O)CCCCC1C(C)(C)CNC(=O)C(F)F n1(CCC=C)c(N2CCC(c3cc(O)n[nH]3)CC2)nnc1C1CCCC1 N1(C(CN(Cc2ccsc2)CC2CC2)=O)CCC(C)(NCC(C)C)C1 c1(C(N(C2CCCN(C(C3C(C)C3C)=O)C2)CC)=O)ccncc1Br c1(CC(N2CCC(O)(CN(C(=O)CC3(O)CCCC3)C)C2)=O)cc(F)cc(F)c1 CC1CN(C(C2(NC(=O)C(C)n3ccnc3)CCC2)=O)CC2(CCC2)O1 C(=O)(C(C)(C)C(=O)OC)NC(CN(C(CCCC=C)=O)CC)C c1(C(CC)NC(=O)C(CC)NC(C)C)ccc2c(c1)OCO2 S(=O)(=O)(c1ccccc1C1(C)N=N1)NCC=CC(=O)NC c1(C(=O)NC(C2CN(C(c3ccnc(CO)c3)=O)C2)C)cncc2[nH]ccc12 C1(OCCNC(=O)Cc2cscn2)CCN(C(c2cnc(-c3ccsc3)s2)=O)C1 CC1(C)C(C)(C(N2CCOC(CNC(=O)CC3CCC(=O)N3)C2)=O)C1(C)C C1(C(=O)NCc2ccc(CNC(c3nc(C)[nH]n3)=O)cc2)CC2(C1)CC(C)(C)C2 CCCC(CC)CCC(=O)NCc1nc(C(=O)N(C(C)C(=O)OC)C)c(C)o1 CC(C)C(F)(CNC(=O)CCC(C)(C)C)C(=O)NCC(C)F N1(C(C2C3CN(C(c4cc(NC(C)=O)ncc4)=O)C2C3)=O)CC(F)C(F)(F)C1 C1(OCC)CCCCC1.C12(CCC1)C(=O)COC2.C1(C)CCN(C)C(=O)N1 C(=O)(C1Cc2ccccc21)N1CC(=O)N(C(=O)CCC2CCCCO2)CC1 CC(C)C(C#N)C(=O)NC(CC(=O)N1CC=CCC1)C(C)C c1(C(=O)NC(c2occ(C(N(CC(C)CO)C)=O)n2)C)ncccc1Cl CC1(CNC(c2cc(C3CCC3)on2)=O)CCCN1C(c1sccc1F)=O N1(C(CCOC)=O)CCCC1CC(=O)NCc1cnn(CCF)c1 c1(C(CNC(N(C)Cc2ccn(C)c2)=O)(F)F)cccc(Cl)c1 N1(C(C2CCC(c3nnc(C)o3)C2)=O)CCC(O)(Cc2nc(C)sc2C)CC1.O c1(C(=O)N(Cc2c(C)nccn2)C2CC2)ccc(Br)cc1O c1(C(N2CCCC(N(C(CC(=O)OC)=O)C)C2)=O)cc(C)nc2c1cnn2C CC1COc2ccc(C(=O)NC3CC4CCC(C3)N4C(=O)C3=CCCSC3)cc21 C1(O)(c2cn(-c3c(OC)cccc3)nn2)CCCN(C(c2ncon2)=O)CC1 c1(OC)cnc(C(=O)NCCC2(O)CCN(C(C3CC3F)=O)C2)nc1 c1(CNC(=O)NCC2(C)C(N(CC)CC)CCC2)csc(CCP(C)(C)=O)n1 N1(C(C)=O)CS(=O)(=O)CC1C(=O)NCCN(C(=O)CCN1CCNC(=O)C1)C1CC1 c1(C(=O)NC(CC2CC2)C(=O)Nc2ccc[n+]([O-])c2)cccc(Cl)c1O n1(CC)c(C(=O)NCc2csc(C(N3CCCC3C(C)C)=O)c2)cnc1O c1(C(=O)NC(CNC(C(c2cnccn2)C)=O)(C)C)cc(-c2cccs2)on1 c1(CC)cc(C(N2CCC(NC(=O)CC(C)n3cccn3)C2)=O)cc(Cl)c1 Cc1nsc2ncc(C(=O)NC(C)(C)CN(C)C(C3(C)CCCC3O)=O)cc12 C12=CNC(=NCCOC1=O)C=C2.c1(OCC)ccc(NC(=O)COCC)cn1 Cc1cc(-c2cn(-c3cccc(C(=O)NC4C5C=CC(C5)C4N)c3)nn2)ccc1F Cc1ccc(CC(N2CCC(C)CC2CNC(=O)CC2COCCO2)=O)cc1C C(C(C)(COc1ccccc1F)CO)NCCSCCC N1(C(C(C)C#N)=O)CC2(CCN(C(=O)C(C)(C)N(C)C)C2)C1 N1(C(C(c2cn(C)nn2)NC(C(CC=C)C)=O)=O)CC2(CCOC2)C1 C(=O)(C1=C(C)CCOC1)NCC(CCNC(C1CC(C)=C(C)CC1)=O)O N1(C(COCc2ncc(C)o2)=O)CCC(O)C(NC(c2ccccc2C)=O)C1 N1(C(C(=O)NCCCOC)CC2(C)CCC2)Cc2ccccc2N2CCCC2C1 c1(C(C)=O)cc(NC(C2CC3CC3N2Cc2cn(C)cn2)=O)ccc1F c1(NC(C2CC(NC(C3C(OC)C3)=O)C2)=O)cc(Cl)nc2ccccc12 CCC(C)(O)C(=O)N(C)CCC1CCN(C(C23COC(C2)C3)=O)CC1 C#CCC(C)(C(=O)NC1CCN(C2CC2)C1)NC(=O)C(C)N=[N+]=[N-] N1(C(c2c(C)n[nH]c2)=O)CCC(NC(C2(N(C)C)CCCOC2)=O)C(F)C1 C(c1c(C)cc(C)cc1C)=CC(=O)NCC1CN(C(CC(C)SC)=O)C1 c1(C(C)=O)ccc(OCC(=O)NCC(CO)NC(=O)CSC2CC(C)(C)C2)cc1 c1(CCCSCC(=O)NC2CC2C(=O)NC(c2ccccc2)COC)ccccc1 c1(C(=O)NCC2C(NC(c3cc(N(C)C)n(C)n3)=O)C2)cc(F)cc([N+](=O)[O-])c1 CCCC(CCC)=CC(=O)NC1(C(=O)N(c2ncccn2)CC)CC1(C)C N1(C(C(CC#C)C2CC2)=O)CCN(C(=O)CC(O)C(C)C)C2(CCC2)C1 Cc1nc(C(=O)C(=O)NC2CCC2NC(c2ccsc2Cl)=O)cs1 C1(C(N(CC(CNC(C(C)OCC)=O)C)C)=O)Cc2cc(C)ccc2S1 C(=O)(CC(O)Cc1ccccc1)NCC1(O)CC(CNC(C(C)SCC)=O)C1 Cc1cc(CCC(=O)NC(C)CCNC(=O)CCc2ncc(F)cn2)cc(C)n1 CC1=CCSC1NC(C(CNC(C1CCCSC1)=O)N(C)C)=O CCCCCC(CC)C(=O)NC1CCCCC1NC(c1cn(C)c(C)cc1=O)=O Cc1cccc(CN2CCCCC2C2(O)CC2)c1.C1CCC=CC(=O)N1 C(=O)(C1CCCc2nc[nH]c21)N(CCC(C(C)(C)C)NC(c1cncs1)=O)C C1(CNC(Cc2c(CC)cccc2)=O)Cc2ccccc2C1N=c1[nH]nc(C)o1 C1(C(=O)OCC)CCN(S(=O)(=O)NC2CCC3CCCCC3C2)C1 c1(C(C)NCCCCC2CC2C)ccccc1O C1(=O)CCCCCN(C)C(=O)CCCN1.C1(OC)(CO)CC=CC1 N1(C(C2(CNC(C3C(CC)CCCC3)=O)CC2)=O)CCCN(C=O)CC1 C(C)(CC1CCC1)(C(=O)N(CCNC(=O)CCCCO)C1CC1)OC C#Cc1ccc(C(=O)NC23CCN(C(=O)Cc4nocc4C)CC2C3)nc1 c1(C(=O)NCC(CNC(C(C)(C)OCC)=O)(C)O)cnn(CC)c1C c1(CC2CC(OCC3CCCC(=O)N3)C2)ccc2c(c1)OCO2 c1(OC)cc(SC)ccc1C(=O)NC(C)CNC(=O)Cn1nccc1C c1(C(=O)NCC2OCCC(NC(c3ncn(C)c3)=O)C2)cc(S(N)(=O)=O)co1 c12cc(c3c(c1)OCO3)O2.C1(OCC(=O)OCCC)CCN(C(=O)NCC#N)CC1 Cc1c(CC(=O)NCC(n2cc(C(C3CC3)N(C)C)nn2)C)cnn1C c1(C(N2CCN(C(C(CC)CO)=O)CC2)=O)cccc2cccnc12 C1(C(=O)NCC2C(NC(Cc3n[nH]c(=NC)s3)=O)C2)CCS(=O)(=O)C12CCC2 CC1=CCC(CN(C(=O)CC2CCN(C(=O)C(c3ccccc3)C)C2)C2CC2)CC1 c1(NC(=O)NC(C)C)ccc(S(=O)(=O)N2CC3CC(CCCC3)C2)cc1 CC1(C2CCC(=O)N2)N=C2NC(CC(C)OC(C)(C)C)C(Cl)=NCCCC1(C)N2 C1(C)(NC(C(CC)C)=O)CCN(C(=O)CNc2ccccn2)CC1 C(CCF)(C(=O)N1CC(O)C(O)CO1)NC(C1C(C)(C)OCC1)=O c1(C(N(C2CCN(C(C(C(C)(C)C)N(C)C)=O)C2)CCO)=O)cc(Cl)c(F)cc1F C(=O)(C1=CC2CCCCCC12)NC1CN(C(CCOC)=O)CC1C C1(C(N2CC3C(CNC(c4cnn(CC(F)F)n4)=O)(C3)C2)=O)CC12CCSCC2 c1(C(=O)NC(CN(C(c2n(CC=C)ccn2)=O)C)C)ncn2cccnc12 c1(C(C(=O)N(CCOCC)CCO)N(C)C(=O)OC(C)(C)C)ccc(F)cc1F c1(C(=O)NCCN(CC(=O)NC(=O)NCCCC)C)ncn(CCOC)n1 C1(C(=O)NCC(C)N(C(=O)Cc2cc(C(F)(F)F)n[nH]2)C)CCCC12OCCO2 c1(C(=O)NC(C2CCN(C(=O)CCC#N)C2)C)cccc(NC(N)=O)c1 C(C(C)(C)C(=O)NC(C1CCOC1)CNC(=O)CCc1cccc(Cl)c1)OC c1(C(N2CC(=C(CNC(C(COC)C)=O)F)C2)=O)cnc(OC)cc1C c1(C(=O)NCC=C(C(=O)N(C(CC)C)CC(C)O)C)ccoc1C C1(NC(C=C(C)Cl)=O)CC2CCC(C1C)N2C(C1CCCCCC1)=O N1(C(C(N2CCC(O)CC2)C)=O)CC2(CCCC2NC(=O)CCC(C)(C)C)C1 Cc1cn2cc(NC(C3CCN3C(=O)C(C)n3ccnc3)=O)ccc2n1 c1(N(C2CN(C(c3cn[nH]c3)=O)C2)C)ncccn1 C(CCCC(=O)NCC1CCCC(CNC(=O)CC2(O)CCCC2)C1)OC CC1(C)CN(C(=O)C2=COCCO2)CCC1NC(c1[nH]nc2ncccc12)=O c1(N(C)C)ccc(N)c(C(=O)NC2CCCC2NC(=O)CC2CCCOC2)c1 Cc1cnc2nccc(C(=O)NC3CC(C)N(C(=O)Cc4sccc4C)C3)c2c1 n1(CC#C)cccc1C(=O)NC(C1CCCCC1)C(C)NC(c1cscc1Cl)=O CCC(Cc1ccccc1)CC(=O)NC1CC(CNC(c2cccc(Cl)c2)=O)C1 C1(CC(=O)NC2CC(F)(F)C2)CCCN1C(C1CC1(F)Cl)=O C=CC1CCN(C(C2CN(C(=O)CCCCSC)CC2CCC)=O)C1 C1(C)(CNC(C(CCC)C)=O)CCCN(C(=O)CC2(C3CC3)CC2)C1 C1(CNC(C2C(C)CC2)=O)CC2(CO1)CN(C(=O)OC(C)(C)C)C2 CCC(C)C(=O)NCC(=O)NC(CNC(=O)COC1CC=CC1)Cc1ccccc1 c1(SCC)cccnc1C(=O)NC1CN(C(=O)C(C)OCC2CCCCO2)C1 C12(NC(c3cc(CC)c(CC)o3)=O)CCC(C1)N(C(=O)COC(C)CC)C2 C1(C(=O)NC(CNC(c2oc(CC)c(C)c2)=O)CC)CC2C(C1)C2(F)F CC(C(F)(F)F)NC(=O)C(F)CC1CN(C(c2cc(C(C)C)on2)=O)C1 CCCC(CCC)CCCC(=O)NC(C)CC(C)NC(=O)C(C)(C)COCC N1(C(COCC)=O)CCC2(CCCN2C(c2cn(C3COC3)nn2)=O)C1 Cc1c(NC(=O)CC2CN(Cc3ccccc3C(=O)O)C2)[nH]c2ccccc12 N1(C(CCC=C=C)=O)CC23CCCC2(C1)CN(C(=O)CC1CNC(=O)C1)C3 c1(CC(C)C)ncccc1C(=O)NC(C)CN(C)C(c1cncc(N(C)C)c1)=O N1(C(CCC)=O)Cc2ccccc2CC1CNC(c1nnn(C)c1C(F)(F)F)=O c1(NCc2c[nH]c(=N)s2)cc(NCC(C2CCC2)C2CCC2)ncn1 N1(C(C(CCC)CC)=O)CCC2CCN(C(=O)C(O)CC(C)C)C2C1 N1(C(c2cn(C(C)C)nc2)=O)CCCC(C)(CNC(=O)C(C)(C)CF)C1 CCCCC(C)(F)C(=O)N1Cc2[nH]nc(C(=O)NCC3(O)CC3)c2C1 N1(C(CCC(C)OCC)=O)CCCC2(C1)CN(C(C1CCOC1)=O)C2 C1(C(=O)NCCC(C)(C)CNC(c2cc3n(n2)CCC3)=O)CCC2(CCC2)C1 CC1CCSCCN1C(=O)C(c1ccc(F)cc1Br)C C(=O)(CC(C(F)F)NC(C1CCCN1C)=O)NCC1(C)N=C(C)SC1 C=CCC(C)(C)C(=O)NCC1CN(C(c2cncs2)=O)CC1(C)C N1(C(C2C(C=C)CC2)=O)CC(NC(c2ncc(C)cc2OC)=O)C(S(C)(=O)=O)C1 c1(NCC(=O)NCC2(F)CC(NC(c3cc(OC)n[nH]3)=O)C2)cccc(O)c1 C1(CNC(C2(CC#C)CC2)=O)(OC)CCN(C(C2CCS2(=O)=O)=O)C1 Cc1ccc(CC(=O)NC23CC(C2)N(C(=O)CNC(=O)CCCCO)C3)c(F)c1 c1(C(=O)NC(CCCNC(C2CCC(C)C2)=O)(C)C)cc2ncccc2[nH]1 C(CC(=O)NCc1cc(C2CC2)on1)(CC(C)C)NC(CSCC#C)=O c1(NC(=O)Nc2cccc3c2CCCC3)ccc(Cl)c2ccncc12 C1(C(=O)Nc2c(CCC(=O)OCC)nn[nH]2)CCCCC1CC.C1(NC=O)CC1CC C1(NC(C(COC(C)C)NC(C)=O)=O)CN(C(=O)C(F)(F)CO)CC1C Cc1ncc(NC(C2CCN(C(=O)Cc3ccccn3)C2(C)C)=O)c(C)c1C CN=c1[nH]c(C(N2CCN(CCNC(=O)CC3CCCC3C)CC2)=O)cs1 c1(CC)ncc(NC(N(C)C(C)C2CC2)=O)o1 N1(C(c2nc(CC)sc2)=O)CCCN(C(=O)CCCC(C)(F)F)CC1C N1(C(=O)OC(C)(C)C)CCN(C(N2CCCC(CF)C2)=O)CC1CC(F)(F)F CCCCCCC(C)C(=O)N(CCC(=O)NC(c1ccccc1)CF)C(C)C C1(NC(=O)NC2C(C(C)C)(CC)C2)CCC(=C(F)F)CC1 c1(CC(=O)CC)ccccc1.C1(C(=O)O)COCCO1 CN1CC=C(CC(=O)N2CC3CCC(CNC(=O)CNC4CCCC4)(C3)C2)CC1 c1(CC(N)=O)ccc(C(=O)NCC(O)CCNC(=O)CSc2ccccc2)cc1 C(=O)(C(C(C)(C)C)OC)NC(C(=O)NC1CN(CC)CC1C)CCOC C(=O)(C1COc2ccc([N+](=O)[O-])cc21)NCCC(C)(C)NC(C=C(C)C(C)C)=O c1(C2CS2)ccccc1.C1(CC(CN(CC(C)O)C)C)CCOCC1 N1(C(CC=C=C)=O)CCCC2C1CCN2C(=O)C(N)=O c1(CC(=O)NC2CN(C(c3c(C(C)C)cccc3)=O)C2)cc2c(cc1Br)OCO2 n1(CC)ccc2ccc(NC(=O)C(n3cc(CC4CCCCN4C)nn3)C)cc12 N1(C(C(=O)OCC23CCC(C(=O)OCC)(CC2)C3)C)C(=O)c2ccccc2C1=O C1(CC(=O)NCC(C2CCN(C(=O)Cc3ccns3)CC2)(C)O)CC2(CCC2)C1 c1(C(=O)NCCN(CCOC)C(C2C3CCC2CC3)=O)cccc(C)c1Br N1(C(CN(C)C(=O)C2CC2)=O)CCC2(C1)CN(C(C1CCCC3CC13)=O)C2 c1(NC(c2n(C)cc(Nc3c(C)nn(C)c3C)n2)=O)ccc(C#N)c(Cl)c1 c1(OC)ccccc1C(C)C(=O)NCc1ccc(C(C)(C)C)nc1 N1(CCCC(C)(C)C)CCCCC1c1cccc(C(=O)O)c1 N1(C(c2c(OCCC)cccc2)=O)CCN(C(=O)C(C)OCCC)CC1CO C1(C)(C(=O)NCC(C)N(C(C2CCN(CC)C2)=O)C)CCNC1=O C12(C(=O)NCC3(O)CC(CNC(C4CS(=O)(=O)C4)=O)C3)CCC(CC1)CO2 C(=O)(C(CC(C)C)C(N)=O)NC1C(CNC(c2cc(C)c(O)nn2)=O)CC1 CC1CC(CC(N2CC3(C2)CN(C(=O)C=CCO)C3)=O)CC(C)(C)C1 c1(C(N2CC3C(CNC(CN4CC(=O)NC4=O)=O)C3C2)=O)c[nH]cc(F)c1=O CC1(C)CC(O)(CC(N2CCC(F)(CNC(C3(C#N)CCC3)=O)CC2)=O)CO1 N1(C(C(c2cncnc2)C)=O)CC2CCC(NC(=O)CN3CCC3)CC2C1 Cc1cc(C(=O)N(C)CCN(C(c2c[nH]nc2C)=O)C(C)C)ccc1Cl c1(NC(c2cccc(NCc3c(OC)c[nH]n3)c2)=O)c(C)ccc(C)c1O N1(C(c2c(C)oc(C#N)c2)=O)CC2CN(C(=O)C=Cc3cncc(F)c3)CC2C1 C(=O)(C(F)(F)C(F)(F)C(F)F)N1CC2(C(NC(c3cnccn3)=O)CCS2)C1 N1(C(CC(C)CF)=O)CCN(C(C2CCCCCCC2)=O)CC(O)C1 Brc1ccccc1C1(NCc2noc(Cc3ccco3)n2)CC1 C1(C(N2CC(CN=[N+]=[N-])OCC2)=O)CCN(C(=O)CC2CSCCO2)O1 c1(CC(C)NC2CC2)ccc(Oc2ncncc2Br)cc1 C1(NC(CC2(OCC)CCC2)=O)CCN(C(=O)C(C)OC)CC1F N1(c2snc(C(C)C)n2)CC2(COC(CNC(c3cnc(Cl)s3)=O)C2)C1 n1(CCC)cc(CNC(C2CCN2C(C2CC(OC)C2)=O)=O)nn1 N1(C(CCCCCC)=O)CCOC2(C1)CN(C(C1CCC1n1cccn1)=O)C2 C(C)(C(CC)CC)NC(c1ccc(CNC(c2ccc(CC)s2)=O)o1)=O N1(C(C(C(C)NC(C(C)NC(COC)=O)=O)(C)C)=O)CC2C3C=CC(C3)C2C1 CC(CNC(=O)CCc1cnn[nH]1)C(=O)NCc1nc(C2CC2)n[nH]1 C1(NC(=O)Cc2cnsc2)CN(C(c2cnc[nH]2)=O)CC1C1CC1 c1(C(=O)NC(C2CC(NC(=O)CC34CCCC3C4)C2)C)cccc(C2CC2)c1Cl N1(C(CSCCCC)=O)CC2(CC(NC(C3(C)COCCO3)=O)C2)C1 C1(NC(Cc2nn(C)c(Cl)c2)=O)CN(C(=O)CCc2cccc(O)n2)CC1(C)C CC1CCCCCC1NC(C1OCCC1NC(C1CCCC1O)=O)=O Cc1ccc(F)c(N)c1C(=O)NCCC(C)NC(=O)C=Cc1ncc[nH]1 N#Cc1ccc(C(=O)NCC2(F)CCN(C(c3ccc(Cl)s3)=O)CC2)cc1Cl CCC(CCC(=O)Nc1cnccc1CO)NC(=O)C=Cc1cc[nH]n1 N1(C(C2(C(F)F)CC(=C)C2)=O)CCC(CN(C)C(c2c(Cl)n[nH]c2C)=O)CC1 C(=O)(C(C#N)C(C)(C)C)NC(C)CN(C)C(C1(n2cccc2)CCCC1)=O c1(OC)ccc(N=c2scc(NC(C3CCCCC3C(C)C)=O)n2C2CC2)cc1C C(=O)(C(F)CC(C)(C)C)N1C(CNC(C(C2CCOCC2)OC)=O)COCC1 C=CC(C)(O)C(=O)NC1CC(NC(C2CC(=O)C2C(C)(C)C)=O)C1 c1(C(=O)NC2CC(C)CN(C(c3cncn3C)=O)C2)cc([N+](=O)[O-])cnc1O C1(c2c(C(=O)NCC(CC)CCC3CCCC3)c[nH]n2)CCC(F)(F)CC1 C1(O)(CC(=O)NCC(C)N(C(CNC(C(CC)C)=O)=O)C)CCOCC1 C1(NC(=O)CCCC2CCCCC2)CN(C(C2CC(O)C2)=O)CCC1C(F)(F)F c1(C(=O)NCC(CO)NC(CC2CC(SC)C2)=O)ccc2cccnc2n1 C(=O)(C#CCNC(=O)CN(C)C)NC(C#C)(C)C1CC1 c1(C(C)(C)C)ccc(NC(=O)NCC2CCCN2CCCc2ccccc2)cc1 C1(NC(CCNC(=O)NC)=O)CCN(C(c2cc(C)[nH]n2)=O)CC(C)(C)C1 C1(=CC(=O)NCC(C)NC(C(CC)(C)C(F)F)=O)CCc2ccccc2C1=O CC(C)C(CNC(=O)C=Cc1ccncn1)C(=O)N1CC2CC2C2CC12 c1(N(Cc2ccccn2)C)ccc(SCC(C)C)o1.CCCCCN(CCCC)C=O C(=O)(C1Cc2c(Cl)cccc21)N1CC2N(Cc3ncc(C(C)C)o3)C(CCC2)C1 N1(C(c2c[nH]c(=NC)s2)=O)CC2(CO)CC1(C(=O)NCC(O)CC1CCC1)C2 c1(NC(C2(C(C)C)CCN(C(COCCC#C)=O)C2)=O)cnc(F)cc1C O(NC(=O)C(C)Cn1ccnc1)CCC(C)O.C1(=O)C=CCN1C N1(C(CCNS(CC)(=O)=O)=O)CCC2CCN(C(=O)CC3CC=CC3)CC2C1 c1(C(C(=O)NCC(C)CNC(=O)C(F)(F)CC2CC2)=O)c[nH]c2ccccc12 CC1(C)CC(=O)OC1CNC(c1conc1CNC(=O)CC1CC2CC2C1)=O c1(OCC)ccccc1CNc1cncc(-c2ccccc2)n1 C1(C(C(=O)NC(C=CC(=O)N(C)CC2(CC(C)C)CC2)C)F)CCOCC1 N1(C(C(n2cc(CCN(C(C)(C)C)C)nn2)C)=O)CCCN(S(N)(=O)=O)CC1 Nc1sc2c(c1C(=O)NCC1CC1CNC(c1ccc(=O)oc1)=O)CCC2 C=C(C)C(C)(C)C(=O)N(C)CC1CN(C(c2cc(C)n(CCO)n2)=O)CCO1 C1(CNC(C(C)(C)S(C)(=O)=O)=O)CC(N=c2[nH]c3ccc(F)cc3o2)C1 C(=O)(C(=O)CCC(C)(C)C)NCCN(C(=O)C=Cc1ccncc1)CC N1(C(c2cccc(C)c2N)=O)CC2CC1CCC2NC(c1nccnc1C)=O n1(CC)nc(C(=O)NCC2(CCNC(=O)C(CC)OC(C)C)CC2)c(C)n1 CCC(CC)C(=O)NCc1ccc(-c2ccc(Cc3ccccc3)s2)o1 c1(OC)cc(C)ccc1C(N1CC(F)(C(=O)NCc2cncs2)C1)=O N1(C(=O)NCC2(F)CCOCC2)CC2(CCC(Sc3cc(Br)ccc3Cl)C2)C1 Cn1ccc2ccc(C(=O)Nc3ccc(I)cc3)cc12.c12nc(cs1)C(=O)N2 c1(C(N2CC(NC(C(CC)(C)CC)=O)C(N=[N+]=[N-])C2)=O)ccc(F)c2c1CCC2 C1(NC(C(CSC)O)=O)C2CN(C(=O)CC(=O)NCC(F)(F)F)CC12 C1(O)(C(C)NC(C(C)C)=O)CCN(C(c2cccnc2-c2ccnn2C)=O)C1 C1(C(N2CCC(=CCNC(COCCCCC)=O)CC2)=O)CC2(C1)CC(C)C2 N1(C(CN(CCC)C)=O)CCC2(C1)CN(C(=O)Cc1sc(C3CCC3)nc1C)C2 Cc1nc(-n2nc(C(F)F)nc2C2CC(=O)N(C(C)(C)C)C2)n(C)n1 N1(C(=O)Nc2nc3ccccc3s2)CCC2CCCN(Cc3ccccc3)C2C1 N1(C(c2cnc(CC)s2)=O)CCC(C(=O)N(C)CCOC)(CO)C1 C(=O)(CC(CF)NC(c1c[nH]c(=O)n1C)=O)OC c1(C(=O)NC(C)CN(C)C(c2ocnc2C2CC2)=O)cccc2ncnn12 c1(CNC(N2CCC(c3c(F)cccc3F)(C)C2)=O)ccc2c(c1)C(=O)CC2 N1(CC=C)CCN(CCNS(C)(=O)=O)CC1.c12nnnn1C(C)(C)NC2C1CC1 CCCC(O)(CCC)CC(=O)NC(C)CCCCNC(c1nn(C)cc1C)=O C1(C(N2C(CC)(CC)CCC2)=O)(CC)CCCN(C(C2CC2CCOC)=O)C1 C1(C2CCCC2)CC(C(=O)O)ON=C1C.CN=C(N)NC1CCCC1 C1(NC(=O)CN2CSCCSC2)CC2CC(NC(C3CC4CC4C3)=O)C2C1 c1(OCC(=O)NCC2C(NC(=O)Cn3ccnn3)CC2)ccc(O)cc1 c1(C(=O)NC23CCC(C(=O)NCC4CCC(F)C4)(CC2)C3)c(F)cccc1Cl C(=O)(C(F)C(C)CNC(=O)C(C)(C)F)N1CC(C=C)(O)C1 N1(C(C(CCOC)OC)=O)CCCCCC(NC(c2cc(C(F)(F)F)n[nH]2)=O)C1 Cc1noc(C)c1C=CC(=O)NCC(F)CNC(=O)C(C)Sc1ccc(F)cc1 C(CC(=O)NCC1COC(C)(C)C1)(C(F)(F)F)NC(CC=CC(C)(C)C)=O C1(CCC)(NC(C2CCS(=O)(=O)C2)=O)CCCN(C(c2cc(C3CC3)cs2)=O)C1 CC(CN(C)C(C1CC2(CC2)C1)=O)C(=O)NC1(C)CC1(C)C CCS(=O)CC(=O)N(C)CC1(O)CN(C(=O)COc2cccc(OC)c2)C1 C(=O)(C(=O)N(C)C(c1ccco1)C)NCCOCCCC N1(C(CC2N(C(C(C)(C)C3CCCO3)=O)C3C2CCC3)=O)CC2COC(=O)C2C1 CC1(C)CCN(c2ccnc(NCC3CC(C)(C)CCO3)n2)CCS1 Cc1ccc2c(c1)CC(C(N1CCCC(O)(CNC(c3coc(C)n3)=O)C1)=O)S2 c1(OC)ccnc(O)c1C(=O)NC1CC2(C1)CN(C(=O)CC1CCC(C3CC3)O1)C2 c1(-c2ccc(OC)c(C)n2)cccn2ncc(C(N3CCOC(C)C3)=O)c12 n1(CC)nnc(C)c1C(=O)NCC1COCCN1C(c1cn(C)[nH]c1=N)=O C(=O)(CC(F)(F)C(C)C)NCC(CC(C)C)NC(c1cncc2c1CCC2)=O C1(CCC)CCOCC1(c1nnnn1-c1ccccc1)NC1CCC(=O)N(C)C1 N1(C(C(c2cccnc2)NC(CC(CC)C2CCC2)=O)=O)CCC(O)C(C)C1 c1(OC)ccc(C)cc1C(=O)NC1CCN(C(=O)CC2CCCC(O)C2)C(C)C1 c1(C(N(c2scc(C)n2)C(C)C)=O)ccnc(N2CCOCC2)c1.C1(C)CN1 C=CCCCCC(=O)N(CC(C)NC(C1CC2(CC(OC)C2)C1)=O)C C(C)(CCC(=O)N1CC(=C(F)C(=O)OC(C)(C)C)C1)NC(CCOCC(C)(C)C)=O c1(C(=O)NCCCOCCNC(=O)COc2cn[nH]c2)cccnc1S C1(CC=C)(C(=O)NC(c2cnc(F)cn2)C)CNCCO1 CCC(CC(=O)NCCCCc1ncc[nH]1)NC(c1cn(C)nn1)=O C(=O)(CC1CC(=O)Nc2ccccc21)N(CCCNC(C1CC=CCC1)=O)CC O(NC(=O)C1CCc2ccccc21)C=O.c1(C(C)(C)NC)ccncc1 N12CC3CCCN(C3C1)C(=O)C2CCCC.C1(CNC(=O)OC)CCCCC1 C12(C(N(C3CCN(C(=O)Cn4nnc(=N)[nH]4)CC3)CC)=O)COCC(C1)OC2 C1(C(=O)NCCOCC)CCCC2(CC2)C1.n1(CC(CC)C)cc(CC2CC2)nn1 N1(C(CCC)=O)CCC2C(NC(c3ccc(C4(C)CC4)cc3)=O)C12 C=CCC(C(=O)N1CC(CNC(c2scc(C)c2OC)=O)C1)C(C)C c1(CCO)nc(-c2cncc(F)c2)nn1-c1cccc(Cl)c1 n1(C(CC)C)nccc1C(N1CCCC1CC(=O)NC1CC(F)C1)=O C12CC3(CCN(C3)C1)CO2.C12(CO)CC3CC1C2C3.N1(C(=O)C2CC2)CC(C(=O)N)C1 C(=O)(C(CCC1CCC1)NC(C1CC2(CC2)CO1)=O)NCC1CCC(C)C1 N1(C(CCc2onc(C)n2)=O)CCC(O)(CNC(C2CC(=O)C2)=O)CC1 N1(C(CC2N(C)CCC2)=O)CCN(C(c2ccnc(C(C)(C)C)n2)=O)C(C#N)C1 N1(C(c2ccc(C(F)F)cn2)=O)CC2CCCC1C2Cc1cn(C(C)(C)C)nc1 c1(OCC)ccc(CN2CC(NC(C3CCCC3C)=O)C(F)C2)cc1Br Cc1nc2ccnn2c(C)c1C(N1CCN(C(=O)C(F)CC2CC2)CC1C)=O N1(C(Cc2c(C)nc(C)s2)=O)CCCC(NC(C2COC(C)C2)=O)C1C Cc1cc(Cl)c(C(N2CCCC2CN(C)C(C2CCC(=O)N2C)=O)=O)s1 C(=O)(C1=NOC2(CCC2)C1)N1CCC(C=C)(C(N2CCOC3CCCC23)=O)C1 C1(C(=O)NCC(CNC(C(C)C2CCC2)=O)F)CCn2c(O)nnc2C1 C(=O)(C(C)C(C)S)NC(C)C.C1(C(=O)NC(CN(C)C)C)CC(OC2CCC2)C1 C(CCCC(=O)NCc1nc(C2CC2)co1)N(C(=O)NOC1CC1(F)F)C c1(C(N(CC(C)CNC(=O)C(C)(C)C2CCCCO2)C)=O)ccnc2ccsc12 C1(C(N(C2CC(F)(F)C2)C)=O)CCCCN(C(=O)Cn2cccn2)C1 C1(CNC(c2c(C)coc2)=O)CCN(C(c2cn(C)ccc2=O)=O)CC1C CC1(C)CCC(CNC(=O)C2=CCCCC2)(NC(=O)Cn2ccnn2)CC1 CCC(CC)CC(=O)N(C1CCN(C(c2cc(C(F)(F)F)cs2)=O)CC1C)C N1(C(C(CC(C)C)OC)=O)CC2CC(NC(c3cn(CCO)nn3)=O)CC(C2)C1 c1(OC)cccc(CCC(=O)NC(CNC(c2ccc(SC)o2)=O)CO)c1F C1(CCC)CN(C(c2ncoc2C(C)C)=O)CCN1C(c1ccc(CO)nc1)=O c1(OC)ccc(C(=O)NC(C)CCNC(c2c(C(C)C)cccc2F)=O)c(F)c1 c1(OC)ccc(C(=O)N(CCN(C)C(c2ncnc(O)c2Cl)=O)C(C)C)c(C)c1 N1(CC(=O)NCC2(CCNC(C=CCCC(C)C)=O)CC2)CCSC(C)(C)C1 N1(C(C2(COC)CC2(F)F)=O)CCN(C(c2cc(C(=O)OC)[nH]n2)=O)C(CF)C1 C1(c2n(CCC3(C)CC3)nnn2)(NCC2(CO)CCC2)CSCCSC1 C(=O)(C#CC1CC1)NCC(CNC(c1oc(Br)cc1C)=O)OC Cc1[nH]nc(C(=O)NCC2CC2NC(c2cc(C(C)C)oc2C)=O)c1C c1(OCC)cccc(CC(=O)NCCC(C)NC(=O)CCc2ccoc2)n1 c1(C(=O)NCC(C)(CO)NC(c2sc(F)cc2Cl)=O)c[nH]nc1S(N)(=O)=O C(=O)(CCCC(=O)NCCOCCCNC(c1sc(C)nc1C)=O)N(CC)CC c1(C(N2CC(NC(Cn3c(C)cc(C)n3)=O)C(F)C2)=O)c(Cl)cccc1Cl Cc1nc(C)c(C(=O)NC2(c3ccccc3)CC(NC(c3csnn3)=O)C2)s1 N1(C(C(=O)NCC(F)F)=O)CCCC2(CNC(=O)C3=CCCS3)CCCC12 N1(C(C(CCC)(C)C)=O)CC2CCOCC2(NC(c2sccc2OCC)=O)C1 c1(C(=O)NC(CNC(CCCCOC)=O)(C)C)nc2ccccc2[nH]1 N1(C(c2c(C)cc(F)nc2)=O)CCCC2CN(c3cc(O)nc(C)n3)CC12 C1(CC)CN(C(C2CCCC(C)C2)=O)CCC1NC(c1occ(C)c1C)=O C(=O)(N=c1nc(Cl)nc2[nH][nH]cc1-2)c1ccc(CNC(c2cccc(C)c2)=O)cn1 c1(C(=O)NCC2(C)CCN(C(C3(C)CCC(=O)C3)=O)C2)cc2n(c1)CCCC2 CCC(O)C(C)C(=O)N1CCC(NC(=O)C(C)(C)Oc2ccc(F)cc2)C(C)C1 C1(CN(C(COC)=O)C)C2CN(C(C3CC(C(F)(F)F)CO3)=O)CC12 N1(C(C(C)OC)=O)CCC(NC(=O)CC2CCSCC2)C(OC)C1 c1(NCC)cccnc1C(N1CCC(C)(NC(=O)Cc2ccco2)C1)=O Nc1c(C(N2CCN(C(c3cnccn3)=O)C3CC23)=O)cccc1F C(C(=O)NOCc1ccccc1)(c1ccoc1)OCCNC(C(CC)N(C)C)=O C1(NC(CS(=O)(=O)NCC)=O)COCCN(C(=O)C(N2CCCCC2=O)C)C1 c1(C(=O)NCC2C3CN(C(C(C)(C4CC4)OC)=O)CC32)c(C)[nH]c2ncccc12 C1(C(N2C(CN(C(c3sc(CC)c(C)c3)=O)C)CCC2)=O)CC2(CCCC2)CO1 c1(C(=O)NC2CC(CNC(CCSC)=O)C(O)C2)ccc2c(C)noc2n1 c1(C(=O)NCC(=O)NCCN(C(Cn2c(C)ccc2C)=O)C)c(F)cccc1F Cc1cc(C)c(C(=O)NCCC2(NC(c3cc(Cl)ncc3N)=O)CCC2)c(C)n1 C(=O)(C(C)(C)CN(C)C)N(C(CSCC)C(N1CCC(C2(C)N=N2)C1)=O)C1CC1 C1(C)(C(=O)NC2CC(NC(c3ncn(C)c3)=O)C2)CC2(CC2)C1 C1(CN(C(C=CC)=O)Cc2cccs2)CCCCN1C(=O)C(C1CC1)OCC C(=O)(N=c1ccn(-c2nc(C)cc(C)n2)[nH]1)C1(c2cccc(OC)c2F)CC1 C1(NC(CC(CC)C)=O)CCCCCC1NC(c1ccc(OC)c(C)c1)=O C=CC1(C(=O)N(C)Cc2nc(CC)no2)CCN(C(=O)CCn2ccnc2C)C1 C(=O)(C(F)(F)C(F)(F)F)NC1CCCC(NC(c2ccncc2F)=O)CC1 Cn1ccc(=O)c(C(N2CCN(C3CCN(C(=O)Cc4cc[nH]n4)C3)CC2)=O)c1 C1(C(=O)NCC(C)CNC(c2nnc(C(C)(C)C)s2)=O)CCCC(C)CC1 CCCCCC(C)(C)C(=O)N(C)CCNC(c1c(C)sc(Br)c1C)=O N1(C(C2ON=C(C)C2)=O)C2CCC1CN(C(c1ccnc(N3CCCC3)n1)=O)CC2 c1(C(=O)NCCN(C(=O)COCC(F)F)CC2CC2)cccs1 c1(C(=O)NC(C)CCNC(C2CC3(C2)CC3(F)F)=O)ccc2n[nH]cc2c1Cl C(CCCCNC(=O)CCSC(C)C)N(C(=O)C(C)N(C)C)C(C)C.CO c1(C(N(CCCNC(c2ccc(N(C)C)cc2)=O)CC)=O)ccc(C)c(O)n1 c1(NC(C2(CC)CCN(C(C3CC(OCC)C3)=O)C2)=O)nc(OC)ccc1C CN1CCCC1(C)C(N1CCCC(Nc2cccc(O)n2)C1)=O c1(C(C(=O)NC2CCN(C(Cc3ncc(C)s3)=O)C2)O)ccc(F)cc1 N1(C(C2OCCC(C)C2)=O)CCOC2CN(C(c3ccc4nc[nH]c4n3)=O)CC12 c1(C(=O)C2CC2)cnn(C)c1.C1(CC(=O)NC2(CCCNC3(CO)CC3)CC2)C=CCC1 C1(C(=O)N(C2CC2)CC2CCCCN2C(c2ccc(CO)o2)=O)CCCCC12CC2 N1(C(C2=CCCC2C)=O)CCC(C2(O)CN(C(c3cc[nH]c3)=O)C2)CC1 c1(C(=O)NC2CCC(C(=O)NC(CS(C)(=O)=O)CO)C2)cc(Br)ccc1[N+](=O)[O-] C(=O)(CC(C)CC(C)(C)C)NC1CN(C(c2nc(CC)sc2N)=O)CC1O c1(NCCC=CC)ccc(S(=O)(=O)N2CCC(C3CCCCO3)C2)cc1F C12CCCN(CC1)CC(=O)N2CCCN1CC2CCC1C2.C1(OCC)CCCC1 N1(C(C(C)N(C(c2cccc(C#C)c2C)=O)CC)=O)CCc2ncncc2C1 C1(C(=O)NCC2CCCN2C(=O)C=CCF)CCCN(C(N2CCC2)=O)C1 C12(OC)CCC(C(=O)NCCCCN(C(=O)C=CCF)C)(CC1)C2 C1(NC(c2c(CCC)n[nH]c2)=O)CC(F)CN(C(C2CCCSC2)=O)C1 N1(C(CSC)=O)CC(N(C(=O)CCCOc2ccccc2C#N)C)C(C)(C)C1 CC(C#N)C(=O)NCC(C)(C)CNC(=O)CC1CS(=O)(=O)C1 C1(NC(CCCC(=O)OC)=O)CN(C(=O)COC2CCCCC2)C2(CCC2)C1 c1(C(c2n(CCC(=O)OC)nnn2)NCC2(C)CC2)ccnc(-c2ccco2)n1 CC1(NC(=O)CC(c2cc(Cl)cc(Cl)c2)O)CCC(N2CCCC2=O)CC1.CCCF C1(CCNC(C2CCC(CC)O2)=O)CSCCN1C(=O)CCC1CCC(=O)NC1 Cc1csc(Cl)c1C(=O)NCC(O)CN(C(=O)C(C)C1CCCC1)C c1(CNC(C(=O)NC2C(OCCC)CCCC2)=O)nc2cc(Br)ccc2s1 N1(C(c2cc(C)nc(O)c2)=O)C2CCC1CC(NC(c1cn(C)nc1O)=O)C2 N1(C(CCCSC)=O)CC2CCC2(CCNC(c2c(O)cccc2F)=O)C1 c1(C(=O)NCCCN(C(CCCSC)=O)C)ccc(-n2ccc(C)n2)cc1 CCC(CNC(c1cnc(C(C)O)s1)=O)(CC)NC(=O)C(C)N1CCC1 C1(C(N(CC(C)CNC(C2(C(N)=O)CC2)=O)C)=O)CCS(=O)(=O)C(C)C1 Cc1cnc(C(=O)NC(CCC2CCC2)C(=O)Nc2cc(Cl)ccc2C)c(F)c1 c1(C(N2CCN(CC(C)(C)NC(CC(C)SC)=O)CC2)=O)ccc2sccc2c1 C1(O)(CNC(C2C(C(N)=O)C2)=O)CCN(C(c2c(Cl)cccc2Cl)=O)CC1 C#CCC(O)C(=O)NCCCN1CCC(CNC(c2ccc(CO)nc2)=O)C1 C1(NC(C(C2CCN(C(c3c(CC)nns3)=O)CC2)C)=O)CC2(C1)CN(C)C2 Cc1oc2ccccc2c1CNC(=O)CNC(=S)NNC(=O)c1ccco1 CCS(=O)CC(=O)N1CC(C(C)(C)O)(CNC(=O)Cc2cccc(Br)c2)C1 C(=O)(C1=CCN(C(C2(N(C)C)CCCC2)=O)C1)NC1C(CC=C)COC1 C(=O)(C(CC1CCCCC1)CC)N(CC(C)(C)NC(C(C=C)O)=O)C N(C(=NCCN1CCOC1=O)NCc1cnc(-n2cccn2)s1)C(CC=C)C N1(C(c2c(C)nn(C)c2)=O)CCCC(C2CN(c3ccnc(C(C)(C)C)n3)C2)C1 c1(C(=O)NC2CC(NC(C3=NOC(C)C3C)=O)C2)cc2ccncc2c(O)n1 Cc1nc(CC(=O)NC2(C)CC(NC(C34CC(C)(C3)C4)=O)C2)n[nH]1 N1(C(CSCCCC)=O)CCOCC1CNC(C1CCC(C)C1)=O C1(NS(CC)(=O)=O)CCOC12CCCCC2.c12cn(nn1)CC(=O)N2 c1(C(=O)NC2CCCC(NC(C3(CO)CCC3)=O)C2)coc(=O)c2ccccc12 c1(C(=O)NCCNC(C(=O)N(C(c2ccncc2)CC)C)=O)cccc(Cl)c1O c1(CCC(=O)NCC(C)NC(C(C(C)C)SCC)=O)cnc(C)nc1O C=CCC(C)(C)CC(=O)N(C)CC1CCCN1C(C1(C)CC=C(C)CC1)=O N1(C(c2cccc(COC)c2)=O)CC2CCOC2(CNC(c2ncn(C)n2)=O)C1 c1(C(c2nnnn2C2CC2)NC(c2nccn2C)CC)csc(-c2ccsc2)n1 c1(CC)ccoc1C(=O)NC(CC1CCCC1)C(=O)NCC=CCl C(=O)(C1=CCCO1)N(CC(C)O)CCNC(C1(C#C)CCC1)=O C1(C(=O)NC2CN(C(=O)Cc3ccccn3)C2)CCCCN1C(N)=O c1(SCC(=O)NCC(CO)NC(C2C(C)(Br)C2)=O)nnnn1C1CC1 C1(CNC(Cc2c(C(C)C)con2)=O)CC(C)(C)CN1C(C1CCSCC1)=O C(=O)(CC(CN)C(F)(F)F)Nc1c(C)c(-c2ccno2)ccc1 N1(C(C(CC(C)C)N(C(=O)CCC2OCCO2)C)=O)CCC(CO)C(C)(C)C1 CC1OC2(C(=O)NCC3CCC4(CN(C(C5CCCO5)=O)C4)O3)CCC1CC2 c1(OC)ncccc1C(C)NC(C1CCN(C(c2n[nH]c(C)c2C)=O)CC1)=O CCCCC(C)C(=O)N1CCC(CCC(=O)Nc2cn(C)nc2OCC)C1 n1(C(C)C)ncc(C(=O)NCCC(C)NC(c2nn[nH]c2C(F)(F)F)=O)c1F c1(C(c2nnnn2Cc2ccco2)NCCCCSC)ccn(CC(F)(F)F)n1 Cc1c(C(=O)NC2CCCC(C(N3CCC(n4ccnn4)C3)=O)C2)c[nH]c1C#N Cc1c(CC(=O)N(C2CCC(C(F)F)CC2)C)nnn1C(C)C CCCCC(CNC(C1CC=CCO1)=O)NC(c1ccnc(-c2ncc[nH]2)c1)=O C(C(C)(C)n1cccn1)NC(CN(C)C(C1CCOC1)=O)=O N1(C(CC2C(C)CCC2)=O)CCC2(CC2)CC1C(=O)NCc1ccnc(CO)c1 N1(C(c2cn(CC)nc2)=O)CCN(C(=O)Cc2cnc(O)n2C2CC2)C(C)C1C C(=O)(C#CC(C)(C)CNC(=O)CCc1nc(=N)[nH][nH]1)NCC(=O)NCC Cc1sc(C)c2sc(C(=O)N(C3CC(NC(=O)C(C)n4ccnn4)C3)C)cc12 N1(C(CCC#C)=O)CC(NC(=O)Cc2sc(C3CCC3)nc2C)C(C)(C)C1 n1(CCCC)ncc(NC(=O)Cc2nonc2CC)c1C1CC1 C(=O)(CC(C(C)C)C(C)C)NCC1N(C(c2ccc(C(=O)OC)cn2)=O)CC1 N1(CC=CC(N2CCC(C)C2)=O)CCN(C(=O)NC2(C3CCCCO3)CCC2)CC1 c1(CN2C(C(=O)Nc3cc(Br)ncc3F)CC3(CC3)C2)c[nH]c2ncccc12 C1(CC(=O)N(C)Cc2ccnn2C)C2CCCC2N1C(C1(Cl)CC1)=O c1(C(=O)NC2CC3CN(C(COCCC)=O)C(C2)C3)ccc2c(c1)C(=O)NCC2 CCC(C)CC(=O)NC1CCCN(C(=O)Cc2cnn(CC)c2)C1 c1(C(=O)NCCn2cc(-c3c(C(=O)OCC)n[nH]c3)nn2)c(C)cccc1Cl C1(C(=O)NC2(C3CCCN3C(C3(C(=O)NC)CCC3)=O)CC2)C(Cl)(Cl)C12CC2 N1(C(c2c(C)cc(C)c(Br)c2)=O)C(C)Cc2cc(F)ccc2C1C C1(C(=O)NCCCCC(C)NC(CCc2nc(C)c(C)o2)=O)CC1C1CCCC1 C1(NC(C)=O)CS(=O)(=O)C12CCN(C(C1C(C#N)C1(C)C)=O)CC2 C1(CCNC(c2cnc(C(F)F)[nH]2)=O)CSCCN1C(c1cc(Cl)ccn1)=O CC1(C)COCCC1NC(=O)C=CC1CCCN1C(=O)CN1CCCCCC1 C(=O)(C1CCCc2ccc(O)cc21)N1CCN(C(c2nc(C)[nH]n2)=O)CC(O)C1 c1(C(N2C(CNC(C3CC3(F)F)=O)CC(COC)C2)=O)ccc2c(n1)OCCO2 C1(NC(CCC(=O)NC)=O)CCN(C(=O)C(CC)C(C)C)CC1C N1(C(C(C2CC2)OCC)=O)CCC=C(C(=O)N(CC(C)C)CC)C1 C(=O)(N=c1cc[nH]c(C)c1C)C1N(C(c2c(OCCC)cccc2)=O)CCC1O C(=O)(C(C)C(C)NC(c1cnnc(C)c1)=O)Nc1occ(C)c1 N1(C(C=C(C)C2CC2)=O)CCC(n2cc(CNC(C34CSC(C3)C4)=O)nn2)CC1 c1(CN(C(=O)COC(F)F)C)cnn2c1CN(C(=O)CCCn1cncn1)CC2 C(=O)(C1CCCn2cc(C)nc21)NC(CC)CNC(C1(O)CCCCCC1)=O N1(C(CN2CC(C)C2)=O)CC(CNC(=O)C(C)(C)c2ccncc2)CC1C c1(C(=O)NC2CN(C(CC(CC)SC)=O)CC2C)cnc(Cl)cc1N N1(C(c2ccc(C)s2)=O)CCN(C(=O)C(C)c2ncco2)CC1C(F)F c1(N2CCC(C)C2)nc(N2CCCC(N3CCCC3)C2)nc2c1CCCCC2 c1(C(=O)NCC(CNC(C(c2c(OC)cccc2)OC)=O)OC)coc2c1CSC2 c1(OC)ccc(C(=O)NCC2(NC(=O)C3=NNC(=O)CC3)CC2)c(F)c1Cl CC(C)C(CO)C(=O)NC(CNC(c1cc(F)cnc1Cl)=O)CC(F)(F)F N1(CC)CC(C(=O)NCC2CN(C(C3(C(F)F)CCCO3)=O)CC2C)CCC1=O C1(c2ccc(Cl)cc2)CCC2(CCC2)CC1.N12CCCC1CNC(=O)C2=O C(=O)(CCC(C)(C)F)NCC1C(NC(c2ccc(C(N(C)C)=O)cc2)=O)COC1 CC1=C(C(=O)N2CCN(C(=O)CCCOc3ccccc3)C3CCC23)CCCC1 C12(CNC(=O)CSC(F)(F)F)CCCC1CCN2C(=O)Cn1ccc(O)nc1=O N1(C(C=CCCC)=O)CCC2(CC1)CC(NC(=O)Cc1ccnc(C)n1)CCO2 O=C(C1=NN(Cc2ccccc2)C(=O)CC1)N1CC2OCCOC2C1 C1(NC(c2n(CC(=C)C)nnn2)c2cc(Br)no2)CCOC12CCC2 c1(OCCNCC(C2CCCC2)OC)ccc([N+](=O)[O-])cc1C c1(CN2CCCC(CNC(=O)NC34CC(C)(C3)C4)C2)ccc(S(C)(=O)=O)cc1Cl Cc1nc(CC(=O)NCCC2CCC(NC(c3cc(F)cs3)=O)C2)cs1 N(C(=NCCC(C)(C)C)NC1CCC2(CC2)C1)CCSC c1(C(=O)NC(C)C(C)NC(=O)CN(n2cncn2)C)c[nH]nc1C(F)(F)F N1(C(C2ON=C(C)C2)=O)CCC(NC(c2cc3n(n2)CCO3)=O)C(F)C1 C1(NC(c2cc(CCC)on2)=O)CCN(C(=O)Cc2cc(F)ccc2C)C(C)C1 S(=O)(=O)(c1cccc2c1OCC2)NC1C(C)COCC1 C1(C(=O)NCC(n2cc(CC(OC)OCC)nn2)C)CC2(C1)CS(=O)(=O)C2 n1(CC(=O)NC(CCN(C(C2=CCCC2C)=O)C)C(C)(C)C)cnc([N+](=O)[O-])n1 CC(CNC(=O)Cc1cccs1)CC(=O)NCC(=O)NC1(CO)CCOC1 Cc1cccc(N(C(c2cc(Br)ccn2)C(=O)NCCCC2CC2)C)c1 C(=O)(CCCC(C)(C)NC(=O)CCc1cnn[nH]1)NCC1(CC)CCOC1 C1(CNC(c2c(C)nccc2)=O)CCC2CN(C(C3COC(=O)N3)=O)CC12 n1(Cc2ccc(NC(=O)NCC3CN(CC)C(=O)O3)cc2)ncc([N+](=O)[O-])n1 CC1(O)CCCN(C(c2cc(N3CCCC(C#N)C3)nc(C(F)(F)F)n2)=O)CC1 C1(N(C(c2cnc(C(C)C)o2)=O)C)CN(C(c2ccncc2N)=O)CCC1O C(=O)(CC(CC)C(C)C)NCCCCC(C)NC(c1ccc(OCC)nc1)=O N1(c2n(Cc3ccccn3)c(-c3nsc(C4CC4)n3)nn2)CCCC(O)CC1 C1(C(C2CCCC2)C2CCCO2)CN(C(=O)COC)CCN1C(=O)CN=S(C)(C)=O c1(N2CCC(NC(CC)=O)C2)nccc(=NC2C=CCCCC2)[nH]1 C12(NC(c3cc(SC)oc3)=O)CCCC1N(C(C1CCc3nccn3C1)=O)CC2 C1(C(N2CCC(N(C(c3cc(OC)ns3)=O)CCO)C2)=O)CC2(CCCC2)CO1 c1(OC)coc(C(=O)NCC2CC2CNC(=O)Cc2ccccc2O)cc1=O C(C)(C(=O)N=c1ccn(CC(=O)NC2CCCC(C3CC3)C2)[nH]1)NC(C)=O C1(C(=O)NC23CC(NC(C4CCC5(CC4)CC5)=O)(C2)C3)CCC2(CCOC2)O1 c1(OC)ccc(C(N2CCOCC(CNC(c3sccc3C)=O)C2)=O)c(OC)c1 C1(NC(C(C)Sc2ccccn2)=O)CCCN(C(c2cnn(C)c2N)=O)C1C N1(C(c2onc(COC)n2)=O)CC(NC(=O)C(O)C(F)(F)F)CC2(CCC2)C1 CC(C)C(O)C(C)C(=O)N(CC(N1CCCC1C)=O)C C1(S(=O)(=O)N(c2ccccc2)CC23CC(CO2)C3)(C(=O)OC)CC1C CC1CC(NC(c2cnccn2)=O)CN1C(C1(NC(N)=O)CC1)=O N1(C(C2N(C(C(OC)OC)=O)C(C)C2)=O)CC(C)(C#N)C1 Cc1cnc(NCC2C3CCCC23)[nH]c1=N N1(C(CCC#C)=O)CCCC2(C1)C(NC(=O)CC1CCCCC1)CCN2C c1(N2CCN(Cc3c(C)nc(C)[nH]3)CC2C)ncnc2cnn(C)c12 C(C(C)(C)CNC(=O)CC(C)C1CC1)N(C(C=C(COC)C)=O)CC N1(C(C(CCC)CCC)=O)CCC(C2CCCN(C(c3cncn3C)=O)C2)CC1 C1(C(N(CCCNC(CCSCC)=O)C)=O)CCCN1C1CCCC1 c1(OC)cc(Cl)c(C)cc1C(=O)NCC1CCC1NC(=O)CC1CCCCCC1 CN1CCN(CC(=O)NCCC2CN(C(C3(C(F)F)CCCO3)=O)CCO2)CC1 C1(NC(c2cnc(CC(C)C)s2)=O)CN(C(c2nccn2C)=O)C2CC12 c1(OC)cccc2o[nH]c(=NC(=O)N3CCCCC(C)(F)C3)c12 C(CC(C)C(=O)NCC(CO)NC(c1cccn1Cc1ccccn1)=O)OC C=CC1(COC(=O)C2CC2)CCCCC1.C12(CC1)C(=O)N2 CC1C2CCC(C2)C1C(=O)NCc1nc(C(=O)N(c2ccccc2)C)co1 N1(C(C2CCC(OC)C2)=O)CCC(C2CN(C(C3CC34CCOCC4)=O)C2)CC1 c1(NCC(C)CCCO)ncccc1S(=O)(=O)NCC(O)Cc1nccn1C c1(CC)ncoc1C(=O)N(CC(=O)N(CC(O)CO)CC)C c1(SC)cc(C(=O)NCC2CC2CNC(=O)CCc2ccncn2)oc1C C(c1cc2ccccc2o1)=CC(=O)NC1CCCCN(C(=O)C2=COCC2)CC1 C1(C(=O)Nc2cccc(NC(C3C(CCOC)C3)=O)c2)CCC2(CCCCC2)C1 c1(C(=O)NC2CC(Cn3cc(CCNC(C)=O)nn3)C2)ccc(Cl)cc1Br c1(N(C)C)nc(C(N2CC(CNC(c3cnc(N(C)C)cn3)=O)C2)=O)[nH]c(=N)n1 C(=O)(CC(C)CC(C)(C)C)NC(C(C)C)CNC(=O)C=CCN1CCOCC1 CCC(C)CC(=O)C(=O)N(C)CC=CC(=O)NCC1CCC2(CCC2)O1 C1(N(C(C2CC(OC)C2)C(=O)NC(C)(C)C)CC2CC2)CCC2C(CC1)C2(F)F c1(NC(C)=O)ccc(Cl)c(C(=O)NC2C=CCN(C(c3cnc(C)[nH]3)=O)C2)c1 CC(C)(CNC(=O)C(N1CCCC(CC(N)=O)C1)=O)C(F)F CC1CN(C(c2cn(C)nn2)=O)CCC1C(=O)NCCc1nccc(O)n1 C=CCC(C(=O)NCC(C(C)C)NC(C1CCCC1CC)=O)OC C(C1CCN(C(C2(F)CCCOC2)=O)CC1)=CC(=O)NCCCc1cccnc1 c1(C(N2CCC=C(C(=O)NCc3cc(Br)co3)C2)=O)ccc2ccccc2c1 C#CC1CCC(CNC(=O)C(=O)NC2CC2(c2cccc(Br)c2)F)CC1 N1(C(=O)NCc2nc(-c3ccncc3)no2)CC2C=C(Br)C2C1 c1(C(=O)OC)cccc(OCC(C)NC(=O)C(=O)NC2CCOC2CC2CC2)c1 C1(NC(C2C(C(N)=O)C2)=O)CCCCCC1F.C1(C(=O)N2CC2)CCC1 CC(CC(=O)N(C(C)CCNC(c1[nH]ccc1C1CC1)=O)C)c1ccco1 CCC(C)(CNC(C1CC2(CC2)CO1)=O)C(=O)NC(CO)CCO Cc1c(N)ccc(C(=O)NC2CCCC2NC(C2CCS2(=O)=O)=O)c1C C1(NC(C=C(COC)C)=O)CC(F)CN(C(C2CC(=O)N(C3CC3)C2)=O)C1 C1(NC(C(CC)n2ccnc2)=O)CN(C(=O)CN2CCCCC2=O)CC1N=[N+]=[N-] c1(CCC=C)ccc(C(=O)NCCN(C)Cc2nccnc2C)cc1 CC(C)CC(C(=O)N(C1CCC(OC)CC1)C)N(C(=O)C(C)OCC1CC1)C c1(C(N(C2CCCC2)CCC)=O)ccc(CF)cc1.c12ccc(o1)CNC2=O CCC(CC(F)(F)F)C(=O)NC1CC(Cn2cc(-c3cnn4c3NCC4)nn2)C1 Cc1ccc(N2CCCCC(CNC(C3C4CCCC34)=O)C2)c([N+](=O)[O-])c1 C(=O)(CC(F)(F)C(C)C)N1CCCC(CCNC(C(c2nc(C)sc2)=O)=O)C1 Cc1cc(C(F)F)nn1CC(=O)NC1(CNC(C2(C)CCC(=O)C2)=O)CC1 c1(-c2cncc(C)c2)cccc2c1CN(C(c1ccc(Br)cc1I)=O)CC2 N1(C(C2ON=C(C(C)C)C2)=O)CCCC2CN(C(C3CCCS3)=O)CCC12 C1(NC(CCCC(C)=O)=O)CCN(C(=O)C=CC2CCCN2C)CC1(C)C C1(CCCN2CCC(CSC)C2)COC(C)(C)O1 c1(C(N2CC(Cc3ccc(CCO)cc3)C2)=O)cc2cccnc2s1 c1(C(=O)NCCCC(C)(C)NC(c2cncc(C)n2)=O)cc(C)c(C)c(C)c1 c1(OC)ccnc(OC)c1F.c12cc(Br)cnc1O2 c1(SC(C(=O)NCC(CO)NC(CC)=O)C)ccc2ccccc2c1 N1(C(CCCOC(C)C)=O)CCC(NC(=O)C(C)CC2CC2)CC(C)(C)C1 C1(C)(C(N(C2CC3CCC2CC3)C)=O)CC12CCN(Cc1ccccc1)CC2 C1(C(=O)NCC(CNC2CCC2C)OC)CCN(Cc2ccccc2)CC1 C12(CNC(C(CO)N(C)C)=O)CC(C1)C(NC(c1ccsn1)=O)CO2 N1(C(C2(C)CCCS2(=O)=O)=O)CCCCC(NC(=O)CSCC(N)=O)CC1 c1(N2CCC(CC=C)(NC(c3coc(C4CC4)n3)=O)C2)ccc([N+](=O)[O-])c(O)n1 c1(C(=O)NC(C2CC(NC(=O)COC3CC(C(F)(F)F)C3)C2)C)ncc(F)cc1F C(C1=CN(C(=O)OC(C)(C)C)CCC1)=CC(=O)N(c1cccc(F)c1Br)CCOC C(=O)(C#Cc1ccccc1)NC1CCCC(C(N2C(CC)CC(O)C2)=O)C1 C1(NC(CC(=O)N(C)C)=O)CC2CN(C(c3c(F)cccc3Cl)=O)CC2C1 CC1CN(C(c2c(Cl)cnn2C)=O)CCC1CNC(=O)CN(S(C)(=O)=O)C N1(C(C2(C)CC(NC(C(C)CC(F)(F)F)=O)C2)=O)CCN2CC(O)CC2C1 N1(NC(C2N(Cc3nc(C(C)C)sc3)CC(F)C2)=O)CCOC(C)(C)C1 C(C(CNC(c1ccc(C2CCOC2)s1)=O)C(F)(F)F)NC(c1cnsc1)=O c1(C(N2CCC(CNC(C34CC(F)(C3)C4)=O)C(F)(F)C2)=O)ccc2oncc2c1 CC(F)(F)CCC(=O)NC1CCCC1NC(c1cnsn1)=O S(=O)(=O)(c1c[nH]c2ccc([N+](=O)[O-])cc12)N1CCN(c2cc(C)[nH]c(=N)n2)CC1 c1(C(=O)NC(CC=C)CNC(=O)Cc2ccon2)ccnc(CC(C)C)n1 CC(C)C(O)C(C)C(=O)NCCCN1CCC(NC(C2(C)CCC(=O)CC2)=O)C1 n1(C(C2CC2)C)nc(-c2ccncc2)nc1-c1ccc(-c2ccccc2F)n1C C(=O)(C(CO)C(C)(C)C)N(C)CC1CCCCN1C(c1cnc(O)o1)=O CCCC(C)(O)CC(=O)N(C)CC=CC(N1CCOCC(C)C1)=O c1(NC(CCC)CO)ccc(S(=O)(=O)NCC2(C)CC2(F)F)c(Cl)c1 c1(OC)ccc(C(=O)OCCC(N)=O)cc1OC.C12CCN(C1)C(=O)N2 C(=O)(C(COC)C(F)(F)F)NCC1(C)CC(NC(C2C(CC)CCC2)=O)C1 c1(OC)cccc(C(=O)N(C2CC2)CC2CCCCN2C(c2ncnn2C)=O)c1 c1(N(CC(N2CCCCC2)C2CCC2)C)nccc(=NCCN(C)C)[nH]1 C1(CC(=O)NC2CCN(C(=O)CCCC3CC3)C2C2CC2)CC2(CCC2)CO1 c1(C(=O)NCC(CNC(CC(C)N2CCCC2=O)=O)F)ccc2sccc2c1 C(=O)(C(C)(CC#C)NC(=O)CC1CCCC12CC2)NCCC(=O)NCC#C C1(COC)(NC(c2cc(OC)ns2)=O)CCCN(C(c2ccc(C)n2C)=O)C1 C(CC(C)(C)C(=O)N1CC2(NC(=O)CNC(C3CCCCC3)=O)CC1C2)SC N1(C(c2cc(CC)no2)=O)CCC2(CC1)CC2C(=O)NC1C=CCCC1 c1(N(C(C)=O)C)ccccc1C(N1CCC(CNC(c2scnc2Cl)=O)C1)=O N1(C(=O)NCc2cc(O)cc(Br)c2)CCC(=C(F)F)CC1 Cc1cc(NC(c2conc2CNC(=O)CC2CCC(C)C2)=O)ccc1O c1(CC(=O)N(CCNC(c2c(F)cc(C)cc2F)=O)C)cn2cccc(C)c2n1 N1(C(C(CCCC)=O)=O)CC(CNC(=O)CCSCC(C)C)C2(CCC2)C1 CC1=NOC(=O)C1CC(=O)NCC1(O)CC(NC(C2(O)COC2)=O)C1 C1(CNC(C(COC(C)C)(C)C)=O)CCN(C(C2CC2C(N)=O)=O)C12CC2 S(=O)(=O)(C1CCOC1)NC(CC(=O)OC(C)(C)C)Cc1ccccc1 C12(C(N(C)CCC3CCN(C(c4ccc(C#N)o4)=O)CC3)=O)CCC(C)(C1)OC2 N1(C(C2C(CNC(C=C(CC)CC)=O)OCC2)=O)CCOCC1CCC CCS(=O)(=O)CC(=O)NCC1(n2cc(COc3cccc(C)c3)nn2)CCCC1 N1(C(c2cc(C(C)=O)[nH]n2)=O)CCC2(CC1)CC2NC(=O)C(C)(C)c1cc[nH]n1 n1(Cc2cn(CCC(N3CCOCC3)=O)nn2)cnc([N+](=O)[O-])n1 c1(CC)noc2ncc(C(N3CCN(C(=O)CS(=O)(=O)NC)C4CC34)=O)cc12 C1(NC(Cc2c(C)occ2)=O)CCCN(C(=O)Cn2cccnc2=O)CCC1 N1(C(CSCC=C)=O)CCOC(C(C)NC(c2csc(COC)n2)=O)C1 c1(C(=O)NCC(=O)OC)cc2c(C)cc(OC)cc2[nH]1.C1CCCN(C=O)C1 N1(CCCC)CCC2CCN(Cc3cnc(C(C)(C)C)s3)C2C1 c1(OC(C)C(=O)Nc2ccncc2C(F)(F)F)ccc2c(c1)C(=O)CC2 c1(C(N2CC(CNC(c3cc(C(F)(F)F)cs3)=O)C2)=O)csc2nccn12 c1(C(N2CC(NC(c3n(CCC)ccc3)=O)C(O)C2)=O)c(N)cc(Cl)cc1F C(C)(C)(CCCCC(=O)NC1CN(C(C2(COC)CC2)=O)CC2(CCC2)C1)OC c1(NC(c2ccc(C)cc2)C(=O)OC)nc2cnc(Cl)cc2s1 C(CN=c1[nH]c2c(c(=NC3CCCC3OC(C)C)[nH]1)CCCCC2)SC Cn1c(C(=O)NCC2CN(C(C3CS(=O)(=O)C3)=O)CCO2)cnc1Cl c1(C(=O)O)cc2[nH]c(C(F)(F)F)cc2c(Cl)c1Cl.c1(-n2ccnn2)ccc(F)nc1 CC1CCN(C(C2CC(N=[N+]=[N-])C2)=O)CC1CC(N1CCCN(C2CC2)CC1)=O c1(C(=O)NC(C(=O)N(CC=C)CC=C)c2ccoc2)ccnnc1O c1(C(N2C(CCNC(c3c(CC)c[nH]c3)=O)CCC2)=O)ccc2snnc2c1 C1(C)(CNC(C2C(OCC)CCC2)=O)CCCN(C(c2conc2C(C)C)=O)C1 c1(NC(c2c(C)cccc2F)c2nnnn2C2(C)CC2)ccc2c(c1)OCC2 Cc1cc(C(N2CC3CN(C(C45CC(C4)C5)=O)CC23)=O)ccc1O CC(=O)CCCC(=O)N1CCCC(CNC(=O)C(O)Cc2[nH]cnc2C)C1 C12(NC(COC)=O)CC(CNC(=O)C(C)NS(=O)(=O)CC)(C1)OC2(C)C N1(C(Cn2ncc(C#C)c2)=O)CCN(C(c2cnns2)=O)CC1C(F)F c1(C(N2C(C)(C(=O)NC(C3(CO)CC3)C)CCC2)=O)ccc2cncn2c1 c1(C(=O)NC2CC(O)CN(C(=O)Cn3cnccc3=O)C2)cccc2cc[nH]c12 CC(N=c1nc(O)c2cc(Br)ccc2[nH]1)C1(C(=O)O)CC1 N1(C(c2cc(C)c(F)nc2)=O)CCC(C2CC2)C1CNC(c1c(C)noc1C)=O c1(OC(=O)CCn2ccnn2)ccc(Nc2ccccc2)cc1 C1(CC(=O)NC(C(C)(C)NC(Cc2cc(CC)on2)=O)C)CN(C)CC1O c1(OC)cc(C)c(CN2CCC(O)(C(=O)NCc3ccc(CBr)cc3)C2)cc1OC c1(C(=O)NCC2(C)C(C)CN(C(c3cc(C)sn3)=O)C2)cc(Cl)c(N)c(Cl)c1 c1(OCC)nccc(C)c1C(N1CCC(NC(c2csnc2Cl)=O)C(O)C1)=O C1(C(C)CCSC)CC2CCC1C2.C(CCNS(C)(=O)=O)N C1(C(N(C)Cc2ccc(C)s2)=O)CCCN(C(C2(C)CC3(CCC3)C2)=O)CC1 N1(C(c2ccn(C)n2)=O)CCN(C(=O)CC2CC2c2ccccc2)CC1CCO CCCN=C(NCCC1CCCSC1)NCC(C)Oc1ccccc1 c1(C(=O)NC2(C)CCN(C(=O)C(Cl)=CCl)C2)cc2c(Cl)cncc2s1 CC1(C(=O)NCC2CCCC2NC(=O)CNc2ccc(Cl)cn2)CCC(=O)N1 N1(C(C(c2ccc(C(F)F)cc2)C)=O)CCC2CN(C(c3cnn[nH]3)=O)CC2C1 N1(C(c2c(CC)scc2)=O)CCN2CCOCC2(CNC(=O)CC2CC23CC3)C1 c1(C2(SCC3CN(CC(=C)C)C3)CC2)cn(C2c3c(Br)cccc3NC2=O)nn1 N1(C(C(C(=C)Cl)(C)C)=O)CCC(O)(C2(NC(C3CC34CCC4)=O)CC2)CC1 C(c1ccncc1)=CC(=O)N(C1CCC(NC(c2cncn2C(F)(F)F)=O)C1)C c1(C(C)C(=O)O)ccc(S(=O)(=O)N2CCC3CCCC3C2)cc1 C(=O)(C(F)(F)CC(C)C)NCCC1CCC(NC(C(C)=C2CCCC2)=O)C1 C#CCCC(O)CCNC(c1ccc(C)nc1OC)=O C1(NC(c2cccc(CO)c2)c2n(CCOCC)nnn2)COCCC1(F)F C1(CCC)(NC(=O)COC(C)CC)CCN(C(C2CCOC(=O)N2)=O)CC1 Cc1n[nH]cc1CC(N1CCC(N(C(C2CCOC2C2CC2)=O)CC2CC2)C1)=O C1(C#N)(CNC(C(Cc2cnc[nH]2)NC(C2N(C)CC(F)C2)=O)=O)CC(C)(C)C1 C1(C(N(CCNC(=O)COc2ccc(Br)cn2)C2CC2)=O)COCCC1(F)F N1(C(CSC)=O)CCC(CO)C(N(C(c2ccco2)=O)Cc2ccccc2F)C1 C(CN=C(NC1CCCSC1)NC1CCS(=O)(=O)C1)OC.C1CO1 Cc1cc(C(=O)NC2(CCNC(C3CC(C)C3(C)C)=O)CCC2)c2c(c1)CCO2 c1(C(=O)NC2CC(NC(c3c(OC)cc(Cl)cc3)=O)C2)ccc(OC)c(C#N)c1 n1(CC)nc(C)c(CC(N2CC(C(C)NC(c3cccc(O)c3Cl)=O)C2)=O)c1C c1(C(=O)OC)cn(C)nc1C(=O)NCC1(NC(C2CCCC2(C)C)=O)CC1 c1(C(=O)NC(C2CC2C(=O)NCC2(SCCO)CC2)C)cc(Cl)no1 N1(C(c2cc(CC)no2)=O)CCC(O)(CNC(C23CCC(CC2)O3)=O)C1 CC(C(C(=O)NC1CC(=O)N(C)C1c1ccc(F)cc1)N(C)CCF)C(C)(C)C N1(C(c2c(C)nsc2)=O)CCC(O)(CN(C)C(c2cc(C(C)(C)C)n[nH]2)=O)C1 c1(OC)cc(N)ccc1C(=O)NCC1(C(F)F)CCN(C(C2C=CCS2)=O)C1 Cc1nn(C)c(C)c1CC(=O)NCc1ncccc1CNC(C1CCCO1)=O CC(C(=O)NC1CCCCC1CNC(c1cc2c(s1)CCC2)=O)C(C)(C)C C12(NC(c3cccnc3O)=O)CCOCC1CN(C(=O)C(F)(F)CF)C2 Cc1cc(F)cnc1C(=O)NC12COC(C1)C(NC(c1ccncc1F)=O)C2 c1(C(=O)NC23CC(NC(c4ccnn4C(F)F)=O)(C2)C3)cc([N+](=O)[O-])ccc1O CC1=NC(C(=O)NCC(C)(C)OCCNC(c2ocnc2C)=O)CS1 c1(SCC)cnc(O)c(C(=O)NC2CCN(C(=O)C(F)OC)C2C)c1 N1(C(c2ccc(C(C)=O)cc2)=O)CCCC2CCCNCC12 N1(C(CC2(OCC)CC2)=O)CC(C)CN(C(C2CCOC(C(C)C)C2)=O)CC1C C1(C(N2C(C(=O)NC3CCC(O)C3)CC3CC32)=O)CCc2ccccc2C1 N1(C(C2CC(CNC(C(=Cc3cccnc3)C)=O)OC2)=O)CC2(CCN(C)CC2)C1 c1(C2C(C(N3CCC(C(N(CC)Cc4cccnc4)=O)C3)=O)C2)ccncc1Cl C=CCCCC(C(=O)NCc1noc(C(C)C)n1)NC(=O)Cc1cnns1 N1(C(COCCC#C)=O)CC2CC2(C(N2CCOCC2CC)=O)C1 C(=O)(C1CCCc2nncn21)NCCOCCNC(Cc1cc(C)c(O)cc1)=O C1(NC(C2C(Cl)(C(=O)OCC)C2)=O)CCC(NC(CCN=[N+]=[N-])=O)CC1 C1(N(C(C(COC)C)=O)C)CCCN(C(c2cc(C3CCOCC3)no2)=O)C1 N1(C(C(=O)NCCOC)c2ccsn2)CC(C)C12CCOCC2 N1(C(CCCSC(C)(C)C)=O)CCC(C)(NC(=O)Cn2nnc(C3CC3)n2)C1 c1(C(N2CCCC(N(C(CCCSC)=O)CCO)C2)=O)cc(N)cnc1C C(CCC[Si](C)(C)C)NC(C(C)C)Cc1ccc(Br)cc1 Cc1cccn2cc(CC(=O)NCC(C(C)C)NC(C3CC(=O)C3)=O)nc12 N1(C(C2CCCCS2)=O)CCC2(CCCN2C(=O)CSc2ccc(Cl)cc2)C1 N1(C(CC)=O)CCc2c(CNC(c3cc(Cl)c(C)cn3)=O)cccc2C1 C(CCCCC(=O)N1CC2C(NC(c3cccc(C(C)C)c3)=O)C2C1)OC(C)C C1(CC(=O)NCC2CC(NC(=O)CCSC3CCCC3)C2)(OC)CCC1 c1(C(N(C2CCN(C(C3(CCCC)CC3)=O)C2)C)=O)ccc(Cl)cc1C c1(C(=O)NCCCC2(NC(c3n(CC#C)ccc3)=O)CC2)cc(C)c(C)nn1 c1(C(=O)NC2C(NC(c3cccc(C(=O)NC)c3)=O)CC2)cnc2occc2c1 c1(OC)n[nH]cc1C(=O)N(C1CN(C(C2(C)CC2Br)=O)C1)Cc1ccccc1 N1(C(CCSC)=O)CC2CC1CN(C(C1OCCC1C(C)C)=O)C2 c1(C(=O)NCC2(CNC(C(CO)OC)=O)CC2)[nH]c(C)nc1C CC1OC2(CNC(C3CCCS3)=O)CC1(NC(=O)C(C(C)O)N(C)C)C2 c1(CN(C2CN(C(c3cc(OC(C)C)ncc3)=O)C2)C)cc(I)cc(I)c1O C(=O)(CC1=NNC(=O)C1)N1CCOCC(NC(C(C(C)C)N(C)C)=O)C1 C1(C(N(C(C)(CC(=O)O)c2cn(CC3CCOC3)nn2)C)=O)CCC2(CC1)CC2 C(CCN=C(NC1CC1C#N)NC1CCC2(CC2)C1)OCC c1(OCCOC(C)C)ncc(C(=O)NCC2CCCOC2)cc1Cl c1(C(N(CC(N2CC(CSc3ccccn3)C2)=O)C)=O)cccnc1S C(=O)(CCC(C)(F)F)N(C1CCN(C(C(C)C)=O)CC1)CC1CCCO1 N1(C(C(CC)N(C)C)=O)CCC2(CC1)CC(NC(C1CCN1CC)=O)CCO2 C(=O)(CCC(C)N(C)C)NC(c1cn(CCOCC2CCCC2)nn1)C N1(C(c2onc(C)n2)=O)CCC(NC(c2ncc(Cl)n2C)=O)C(CO)CC1 c1(C(=O)NCCF)ccc(C(N(C)Cc2cn(CC3CCCC3)nn2)=O)nc1 c1(CC(=O)NCC(C)NC)cc(Cl)cc(Cl)c1F CCCCC(C)C(=O)N(C1CC2CCC(C1)N2)C(C)(C)C(N)=O C1(NC(CCc2ccn(C)n2)=O)CCN(C2CCN(C(=O)C(F)=CC3CC3)C2)CC1 CC(C)CC(CN(C)C)CC(=O)NN(C)C(=O)C1CC1.C12(CCCC1)CC2 C1(CNC(CCCCN(C(C2CC(C#C)(O)C2)=O)C)=O)OCC2CCC1C2 C12(CNC(CCCCC=CC)=O)CCC(CC1)N(C(=O)C(C)OC)C2 c1(C(N(CC(C)(C)C2CCCO2)CCC2CCCC2(F)F)=O)ccc(Cl)c(N)c1 C1(C(=O)Nc2c(C)cc(Oc3ccccc3)cc2)CN2CC3CC2(CO1)C3 C1(COCCn2c(-c3ccc(-c4c(C#N)c[nH]n4)s3)ncc2)CCS(=O)(=O)CC1 N1(C(C2CNC(=O)N2)=O)CCC(C(=O)NCCN2CCOCC2)(CO)C1 c1(NC(Cc2c[nH]c3cccc(C)c32)=O)cc(Br)c(C)c([N+](=O)[O-])c1 C1(NC(c2ccc(CNC(c3cccc(C)c3)=O)cn2)=O)C(C)CCCC1C C1(CNC(c2scc(OC)c2)=O)CCN(C(=O)CC(C)(C)SC)CC1C c1(C(N(C)CC2(NC(=O)Cc3cc[nH]c(=N)c3)CC2)=O)cnc2ncccc2c1 C1(C(=O)NC2(C(N3CC(O)C(F)C3)=O)CSC2)CC(C2CC2)C1 c1(C(=O)NCCOC2CCN(C(c3c(C)scc3)=O)C2)ccc2c(c1)NCC2 N1(C(c2c(C)noc2C)=O)CCC2(CC1)CC(NC(=O)C1=CCCOC1)CO2 N1(C(c2c(C#C)cn(C)n2)=O)CCC2C(C1)CN2C(C1CC(C(C)C)C1)=O c1(CNC(C2(CNC(CCC3(C)N=N3)=O)CC(F)(F)C2)=O)cnc2ccccn12 CCCC(C)(CC)C(=O)NCC12CCC(NC(=O)CNC(=O)NC)(CC1)CO2 N#Cc1ncccc1NC(C1CC(F)CN1Cc1ccco1)=O N1(C(C2C=CC(NC(CSS(C)(=O)=O)=O)C2)=O)CC2COC(=O)C2C1 C1(C(=O)NCc2scc(C(=O)NC3(C(O)CO)CCC3)c2)C2CCC3C(C2)CC13 c1(OC)ccc(C(=O)C(=O)NCCc2c(C)cccc2C)cc1Br N1(C(c2scc(C)c2Cl)=O)CC2CCC2(CNC(c2cc3ccsc3s2)=O)C1 C1(N2CCCC(NC(C=NOC)=O)(CO)C2)CC2CCCCC2NC1=O N1(C(c2n[nH]c(C)c2O)=O)CCN(C(=O)C(C)CCN(C)C)CC(O)C1 c1(C(=O)NC2CN(C(c3n(C(C)C)ccn3)=O)C(C)CC2)cnn2cnnc2c1 Cc1cccc(C(N2CC(C)(NC(=O)COc3ccccc3O)C2)=O)c1F Cc1cc(NC(C2CCN(C(=O)CC(C)C)C2)C)c(F)cc1[N+](=O)[O-] C(=O)(C(C)C1=CCCC1)NC1CC2CN(C(c3n(CC(C)C)ncc3)=O)C1C2 c1(C(N(CC(C)C#N)C2CC2)=O)cncc(CNC(C2CC2C#N)=O)c1 C1(C)(C(=O)NC(CC)CNC(c2cc3scnc3[nH]2)=O)CCC(C)=C(C)C1 CCCCC(C)CCC(=O)N(C)CC1OCCC1C(=O)OC.C12(CC1)C(=O)NC2 c1(SC)cccnc1C(=O)NCCC1CC(NC(C2CC2c2ccccn2)=O)C1 c1(NC2C(C)COCC2)ccc(S(=O)(=O)SCCOC(C)(C)C)c(Br)c1 CC(C)(O)CC(=O)N1CCCC(C(=O)NCc2nc(-c3ccnc(O)c3)no2)C1 N1(C(CC(CC)O)=O)CCCC(N(C(c2cc(F)ccc2N)=O)CC)CC1 C1(NC(COC(C)C)=O)CC2CN(C(c3cc(C4CC4)[nH]n3)=O)CC12 Nc1cnc(C(=O)NC2CCCC(CNC(=O)C(F)(F)C3CCCC3)C2)cn1 C1(C(=O)NCC(C)(C)CNC(=O)C=CCO)COc2cc(F)ccc2O1 C1(CC(=O)NC2CC(NC(C(CCC)OC)=O)C2)CC2(CCOCC2)CO1 C(=O)(CC(C(C)C)NC(=O)C(C)=C(C)C)NCC=CC N1(C(C=CC(N)=O)=O)CC(C(F)(F)F)OCC1CNC(c1occc1C1CC1)=O Cc1[nH]cc(C(=O)NC2CC3CCC2N3C(C2CC=CC2)=O)c(=O)c1Cl CN1CC2CCN(C(c3ccc(CNC(c4cc(O)n(C)n4)=O)o3)=O)C2C1 C1(N(C(=O)Cc2ccn(C)c2)C)CN(C(C2(CO)CC(F)(F)C2)=O)CC1(C)C Cc1ccn(CC(=O)NC(C)C(C)NC(c2cccs2)=O)n1 c1(C(C)OC(=O)C(C2CCCO2)NC(=O)OCC(F)(F)F)ccccc1 Cc1cc(O)c(C(=O)NCC(c2ccccc2)NC(=O)CCc2cn[nH]c2)nn1 C(CCC(C)(C)C(=O)NCC1CC(C(=O)NCC2CCCC2)=NO1)OC N1(C(C=CCCC)=O)CC2(CCN(C(c3cnn(C(C)C)c3F)=O)CC2)C1 c1(C(=O)OC)ccc(N(CC(C)NC(=O)CCn2ccc(=N)[nH]2)C)nc1 c1(C(N2CCC(O)(C(C)NC(C3(C)CCCN3C)=O)C2)=O)ccn(C)c(=O)c1 C1(C(=O)NCCc2cc(C(=O)NCC(C)F)no2)COCC1(C)C N1(C(c2c(C)c(Cl)ccn2)C(=O)NC2CCC2)CCc2ccsc2C1 C1(C(N2CCC(C(=O)N(C)C)C2)=O)(NC(c2c(C)n[nH]c2)=O)CCN(C)C1 N1(C(C(C2CCOCC2)C)=O)CCCC2(NC(C3CC34CCC4)=O)CC2C1 c1(SC2CN(C(=O)OC(C)(C)C)C3C2C3)ccccc1NC(c1ccccc1)=O CCC(C)(CNC(=O)C(Cc1cnc[nH]1)NC(c1ccc(=N)[nH]n1)=O)C(N)=O N1(C(c2c(C)n[nH]c2)=O)CCC(C)C(NC(C2CCCS(=O)(=O)C2)=O)C1C C1(C(CC(=O)OC)C(=O)OCC(C)C)CCCN(C(=O)C(=O)N(C)C)C1 C1(c2ccccc2)CCCCC1NC(=O)NC1CN(C(N)=O)C1 C1(C(=O)NC(CCC=C)C)C=CCN(C(=O)C=CCOC)C1 N1(C(c2cc(OC)n[nH]2)=O)CCC2C1CCCN2C(C1CCS1(=O)=O)=O CCC(CN(C)C)C(=O)NC(C(=O)NCC(O)C1CCC1)C1(C)CC1 C1(NC(Cc2nnc(C)s2)=O)CC2CCC1C(NC(c1csc(C)c1C1CC1)=O)C2 n1(CC(=O)N(C)Cc2cn(-c3ccn(C)n3)nn2)ccc(O)nc1=O N1(C(=O)NCc2nc(C)on2)CCC(O)C(NC(C)(C)CC(C)C)C1 C(c1ccccc1)=CC(C(=O)NC1CC(C)(NC(c2cc(C)on2)=O)C1)C c1(C(N(C)CC2CN(C(CCC)=O)C2)=O)ccc2oc(O)nc2c1 c1(OC)cc(F)ccc1C(c1nnnn1C1(C)CC1)NCc1noc(C(N)=O)n1 C=C(C)C1OCCC1C(=O)NCCOCCNC(c1ncoc1-c1ccon1)=O CN1CC(C(N2CCC(CCNC(c3ccc(O)nn3)=O)C2)=O)NC1=O c1(C(N2CCC(C)(CNC(c3ccc(C(C)C)cc3)=O)C2)=O)cc2sccc2s1 N1(C(C2ON=C(CC)C2)=O)CC2CCCC1(CNC(=O)Cn1cccnc1=O)C2 C1(c2n(C3CC(OC)C3)nnn2)(OCC2CCC3CCC23)CCCOC1 CCCCCC(=O)NCc1nocc1C(=O)NCC1(C)CC1(C)C C(=O)(CCCC(F)(F)CO)N1CC(NC(C(c2cccc(C)c2F)O)=O)C(O)C1 C1CC(O)C(=O)N1.c1(C(C)NC(CSCCC(C)C)=O)c[nH]ccc1=O c1(OC)cc(C(=O)NCC2CC3CC3N2C(=O)CCc2scnc2C)c(F)cn1 c1(C(=O)NC(C)CCCNC(C2COCCC2(F)F)=O)ccn2ncccc12 C(=O)(CCC(=O)N1CC(F)(CNC(C2(C3CCCO3)CCCCC2)=O)C1)OC Cc1ccc(Cl)c(S(=O)(=O)N2CCC(Oc3ccccc3F)C2)c1 c1(CN2CC(CC#N)N(Cc3cc(Cl)cnc3Cl)CC2)cc(Br)cc(Br)c1O Nc1c(F)cc(F)c(F)c1C(=O)NC1CCN(C(C2(C3CCC3)CC2(F)F)=O)C1 CC1CCC(CNC(=O)Cc2ccsc2Cl)N(C(=O)COc2ccc(O)cc2)C1 Cc1cnc2cc(C(=O)NC(CNC(=O)C(C(C)C)N(C)C)C(C)C)ccn12 c1(CC(=O)NCCN(C(C=CC)=O)CC)ccc(F)cc1CC.c1ccc(Cl)cc1 c1(C(C(=O)NCC(=O)NCC(CNC(=O)OC)C)C)ccc(Cl)c(Cl)c1 Cc1cc([N+](=O)[O-])cnc1C(=O)NCC(C)NC(c1ccc2[nH]c(=N)oc2c1)=O C1(CNC(c2n(CC)ncn2)=O)CCC2(CN(C(=O)CC3CCCCN3C)C2)O1 C1(NC(C2(OC)CCCC2)=O)CCN(C(=O)C=C(Cl)Cl)CCC1c1ccccc1 c1(C(=O)NCC2N(C(C=CC)=O)CC=C2)ccc(S(=O)(=O)C(F)(F)F)cc1 C1(CNC(CC(CC)C)=O)CCN(C(c2ccnc(C)c2)=O)C1(C)C c1(NC(CN(C(CCCC)=O)C)C)ccc([N+](=O)[O-])cc1Cl CN(CCCC(=O)N1CC(CO)(NC(=O)Cc2cccnc2Cl)C1)N=O c1(C(=O)NC2C(O)CCN2c2ncc(C3CC3)cn2)c(Cl)cncc1Cl c1(C(=O)NC(c2cccnc2)C(=O)N(CC)Cc2ccccn2)ccnnc1O C(=O)(C(C)(C)C1CCCCO1)N1CC(CN(C(C=C(C)C(C)C)=O)C)C1 c1(CC(=O)NC2CCCN(C(C(C=C)O)=O)C2C)nc(F)c(F)cc1F Cc1cc(N)c(C(=O)NC(CNC(c2cc(C)c(C)o2)=O)C(C)C)c(F)c1 n1(CC)cc(Cl)c(C(c2nnnn2C2(C)CC2)NC(c2ccccc2F)C)n1 c1(C(=O)NC2CC(CNC(C3(C)CC3(F)Cl)=O)C2)ccc(F)c2[nH]ccc12 c1(CC(=O)NCC2CCCN(C(CNC(=O)OC)=O)C2)cccc(F)c1O O=S(=O)(CCCCCl)N1CCCC(c2ocnc2C(F)(F)F)C1 c1(-n2cc(-c3cccc(C(=O)NCCN(OC)C)n3)nn2)cc(F)ccc1F S(=O)(=O)(c1[nH]c(=NCC2CC3CCC2CC3)ccc1Br)N1CCCN(C=O)CC1 CCCCC(C)C(=O)NCC(O)CCNC(c1cccc(C(=O)NCCC)c1)=O C1(C(N2CCC=C(CNC(C3CC(=O)NC3)=O)C2)=O)CCC([N+](=O)[O-])CC1 Cc1ccc(CC(=O)NCC2(C(=O)Nc3ccc(OC(F)F)nc3)CC2)c(C)c1 N1(C(Cn2c(C(C)C)ncc2)=O)CC2CC1CN2C(=O)C(=O)Nc1ccccc1 c1(OC)cc(C)c(Cl)cc1C(N1CC2CCCC1(CO)C2)=O N1(C(CCSCCC)=O)CCOC(CNC(C2(c3ccccc3)CCCO2)=O)C1 C=C1COCC1NC(=O)C(=O)N(c1ccn(-c2ccccc2)n1)C C(=O)(CC(C(F)F)C(C)(C)C)NCCN1CCN(C(C2OCC(C)(C)C2)=O)CC1 c1(CC(=O)NCC2CCCN(C(CC(C)(O)C3CC3)=O)C2)ccc(Cl)cc1F c1(NC)ccc(S(C)(=O)=O)cc1C(N1CCN(C(=O)CN2CCC(C)C2)CC1)=O C1(NC(C2N(C(=O)NC)CCC2)=O)CN(C(c2c[nH]ccc2=N)=O)CC12CCC2 CCCC(C)CC(=O)NCc1cc(C)c(C(=O)NCC(C)(CO)OC)o1 C1(CNC(Cn2c(CC)nnc2S)=O)CC(C)(C)CN1C(=O)Cc1c[nH]nc1O c1(NC)ccc(C(=O)NCC2CC2CNC(c2sc(C(C)C)nc2C)=O)cc1 C#CC1(C(=O)NC2CCC(O)CC2)CCN(C(=O)CC2CC=CC2)C1 c1(C(=O)Nc2ccc(-c3cn(C4CCOC4)nn3)c(F)c2)cc(Cl)c(Br)cc1F Cc1ccc(C(N2C(C(=O)NOCC(F)F)CC2C)=O)o1 C(CC(C(=O)NCC(O)CN(C)C)NC(=O)CC1CCCCC1)=CC O=C(C1CCCc2scnc21)NC1CN(C(C2CCC3CC23)=O)C1 C(=O)(C(C)(O)CC(F)F)N1CCN(CCN(C)C(C2CCCN2C=O)=O)CC1 C1(c2cn(-c3ccc(OC)cc3)nn2)C2CCCC1N(c1cc(F)ncn1)C2 c1(CNC(CCN(CCC)C)=O)cnn(C)c1C(=O)NCCC(C)CO c1(C(=O)NC(C(=O)NCC(CCOC)O)C2CCCO2)cc(C2CC2)oc1C c1(C(N(C2CN(C(c3ccc(C4CCCO4)[nH]3)=O)C2)C)=O)cc(N)cc(O)n1 c1(NC(=O)Nc2c(NS(C)(=O)=O)nccc2)nc2c(cc1C#N)CC(C)CC2 C1(CNC(c2c(C)nn(C)c2)=O)N(C(=O)CSc2nncn2C(C)C)CCC1(C)C CCCCCS(=O)(=O)CC(=O)N1CCCC(NC(=O)C(c2cnn(C)c2)O)C1C C1(NC(C(CC)N(C)C)=O)CC(F)CN(C(=O)CCc2cn(C)cn2)C1 S(=O)(=O)(c1cnn(CC(F)(F)F)c1)NC(C(=O)NC)CC(C)C C1(CC(=O)NC2(C)CCN(C(=O)C(C)(C)c3cc[nH]n3)C2)CCC(=O)NC1=O N1(C(Cn2c(C)ccn2)=O)CCN(C(c2ccc(Br)c(C)c2N)=O)C(C)C1C C1(NC(C(CN(C)C)N(C)C)=O)COCC1C(=O)NC1CC(O)C1O N1(C(C2CCC(CC)CC2)=O)CCOC(C(=O)NCCCCCCF)CC1 CC(C)(C)CCCCC(=O)N(CC(C)O)CCNC(C1(C)CC2CC2C1)=O C(=O)(C1CCc2c[nH]nc21)N(C(C)CNC(=O)CNC(c1ccco1)=O)C.C(C)S C(=O)(CC(C)(C)CN(C)C)NCC1N(C(C2C(=C)C2)=O)CCC1C C1(C)(C(=O)OCC)CCCCC1NC1CC(=O)NC(=O)N1.c12cc(ccn1)S2 c1(C(=O)NC2CN(C(CC(=O)OC)=O)C2)cn2c(n1)CCCC2 C1(C(N2CC(CC)C(NC(c3ccoc3C)=O)C2)=O)C2CCC3(COC(=O)C13)O2 c1(C(=O)OCCOC2(c3ccc(OC)cc3)CC2)nc(F)ccc1Cl C1(C(=O)NCC2N(C(C(c3cccc(O)c3)(C)C)=O)CC2)CC2C=CC1CCC2 c1(C(=O)NC2COCC2F)cnc2c(c1)CCN(S(=O)(=O)c1cccnc1)C2 N1(c2[nH]c(=NCC3CC=CCC3)ccn2)C2CCC1CC(N1CCCCCC1)C2 Cc1cn(C)nc1C(=O)NC1CCC1NC(=O)Cc1ncccc1C C12(C(N3CCC(N(C(C(CC=C)C(C)C)=O)C)C3)=O)C3CCC(CC13)C2(F)F N1(C(c2c(NC(CC)=O)cccc2)=O)CCCC(N=c2[nH]nc(O)s2)CC1 C1(NC(c2ncn(C(C)C)n2)=O)CCCN(C(c2ccnc(C(F)F)c2)=O)C1C Cc1cc(C(=O)NCCC(Cc2ccccc2)NC(c2cc(F)n[nH]2)=O)cs1 N1(C(CCc2cc(C)no2)=O)CCN(C(=O)CC2COCCOC2)C(C(F)F)C1 CCC(CC)N(CCC(=O)N(C)CCNC(c1cscn1)=O)C C12(NC(CNC(=O)OC)=O)CCC1CN(C(C13CCC(OC)C1CC3)=O)C2 Cc1ccc2[nH]cc(C(N3CC4CN(C(=O)CSC5CC5)CCC34)=O)c(=O)c2c1 c1(C(N2CCC(C)(C(N3CCC(C#N)C3)=O)C2)=O)cccc2[nH]ccc12 C1(CNC(C(CC)OC)=O)COCCN1C(=O)CC1CCC=CCC1 C(=O)(C(CNC(=O)C=CC=C(C)C)C(C)(C)C)NCC1(C)ON=C(C)C1 c1(C(=O)NCCNC(C=C(CC)c2ccccc2)=O)cn2ccc(OC)cc2n1 N1(C(C(=C)CC(C)NC(C)=O)=O)CC(C)(C)C(O)C(C)(C)C1 C1(NC(CSCC(C)NC(CN(CCC#C)C)=O)=O)CCCC(C)(C)C1 N1(C(C2(CNC(C=C3CCC(C)CC3)=O)CC(C)(C)C2)=O)CC2CC1CS2=O N1(C(c2cc(C)oc2C)=O)CC2(CCNC(c3sc(=N)[nH]c3C)=O)CCC1C2 CC(C)CC1C(=O)N2CC(C3(CC3)C2)NC(=O)N1.C1(C(=O)N(C)C)CC1(C)C c1(NC(c2cnc3n2CCC3)c2n(C(C)C)nnn2)cc(Cl)cc2c1OCC2 C1(NC(Cn2c(C)nnn2)=O)CC2CC1CN(C(c1cccc(F)c1Br)=O)C2 C12C(C)CCN1C2=O.c1(C(CC)CNC(C(COC)O)=O)ccc(F)cn1 Nc1c(C(=O)NC23CCC2CN(C(=O)CCCn2cccn2)C3)cc(F)cc1Cl c1(C(N2C(CC)CN(C(c3cnccn3)=O)CC2)=O)cnc2[nH]nc(O)c2c1 c1(C(=O)NC)ccc2c(c1)CN(C(=O)C(=O)N(C)CC1CC1)C2 N1(C(c2c(C)onc2)=O)CCC2(COCCN2C(c2cccc(F)n2)=O)C1 c1(CC)c(C(N2CCOC(C(C)Nc3n[nH]c(CC)c3Cl)C2)=O)cnn1CC c1(CC(=O)NC2CC3(CN(C(CNS(NC)(=O)=O)=O)C3)C2)cn2c(C)csc2n1 c1(C(=O)NCCc2c(C(N(CC)CC)=O)c[nH]n2)[nH]ccc(=O)c1C Cc1ccc(C(=O)N(C(C)CNC(c2ccc(Cl)c(C)c2O)=O)C)c(F)c1F CC1(C)CCCCC1=CC(=O)NC1CCCC1NC(=O)CCOCC1CCC1 c1(CNC(=O)Cc2ncc(-c3ccccc3)o2)ccc(OC(F)(F)F)cc1 C1(CC(=O)NC2CCC(C(=O)NC3CCC4(CC4)C3)C2)CC2CCC1O2 C1(N(CC(C)NC(c2cc(CC)on2)=O)C)CCN(c2cc(C)nn2C)C1=O C1C(=O)N2CCC(O2)O1.N1(C(C=C2CCC(C)CC2)=O)CCCC12CCNC2=O c1(-n2ccc(CCS(=O)(=O)N(CCCOC)CCO)n2)ccccc1 O(NC(=O)C(CC1CC1)NC(C1CC=CC(O)C1)=O)CC N1(C(c2nc(CCCC)sc2)=O)CCN(C(c2ccc(=N)[nH]n2)=O)C2CC12 S(=O)(=O)(c1ccc(F)c(N2CCCC2)c1)NC1CN(C(NOCC(C)C)=O)C1 C(C)(CC(C)CC)N(C1CCN(Cc2nc(Cc3ccccc3)cs2)C1)CC c1(NCc2n(CC(=O)OCC)c(S)nn2)ncc(C)c(-c2ccccc2)n1 c1(NC(CCC(CC)NC(C2(C#C)CC(=O)C2)=O)=O)ccc2c(c1)OCC2 c1(C(N(C2CN(C(CCCN(CC)CC)=O)C2)C)=O)ccc(CC2CCC2)cc1 c1(CC)cccc2sc(NC(c3cn(C)c(O)n3)=O)nc12 C(=O)(C(C(C)CC)N(C)C(C1CCCC(CF)C1)=O)NCCCCCC#C c1(CC)cc2c(CC(=O)N(CCCN(C)C(c3c[nH]nc3C)=O)C)csc2s1 C1(NC(C2(CC)CCC2)=O)CC(F)CN(C(c2occc2CN(C)C)=O)C1 C(CC(F)F)(C(=O)NCCc1nn[nH]n1)NC(C=C(C)C)=O CC1(CNC(C2CC3(CC3)C2)=O)CC(F)(F)CN1C(c1ccc(Cl)cn1)=O C(=O)(C1=NOC(c2ccccc2)C1)NCC(C)NC(C=C(CC)C)=O N1(C(C2N(C(=O)CCN3CCCCC3)CCN(C)C2)=O)CC2(CNC(=O)OC2)C1 Cc1noc2ncc(C(=O)NC3CC(CCNC(=O)CCNS(C)(=O)=O)C3)cc12 C1(CCC)C(=O)NCCN1C(C1(NC(=O)CC(C)F)CC1C)=O c1(C(N2CC(C(=O)NCc3cc(Cl)ccc3Cl)OCC2)=O)c(F)ccc(Cl)c1Cl C1(C(N(CCN(C(CCCc2c(C)cccc2)=O)C)C)=O)CC2COCCN2C1 C1(CCC(C)(C)NC(=O)C(C)(F)F)CCCCN1C(=O)C=CC1CCCC1 c1(C(=O)NCC2(COC)CN(C(c3ncn(C(C)C)n3)=O)C2)cc(Cl)c(Cl)n1C N1(C(CNS(N(C)C)(=O)=O)=O)CCC=C(C(=O)NCC2(CO)CC23CCC3)C1 c1(OCCNc2ccc(-c3cccc(N)c3)o2)ccc(F)cc1Cl N1(C(C(C(C)C)OCC)=O)CCCC2C(NC(=O)CCSC3CCCC3)CC2C1 Cc1cc(N(C(C)(C)CNC(c2nnn(C(C)(C)C)n2)=O)C)nc(CO)n1 C12(C(=O)NCC(=O)NCC3N(C(CC4(C)CC4)=O)CC3)CCCCC(=O)N1CCC2 C1(NC(=O)NCCCC)CC12CN(Cc1ccc(C(F)(F)F)nc1)C2 C(C(C)(C)C(=O)NCCOCC)NC(CC1C(C(=O)OCC)C1)=O N1(C(c2c(CC)occ2)=O)CC(O)(C2CCN(C(=O)CC3CCCC3O)CC2)C1 N1(C(CC(C)OC)=O)CC2(C=C(C(=O)N3CC4(CC(F)C4)C3)CO2)C1 C(C(=O)NCc1ccnc(C(=O)NCC(c2cccnc2)O)c1)(C(C)C)OC C1(NC(CC(CCC=C(C)C)C)=O)CS(=O)(=O)C2CN(C(c3cn[nH]c3)=O)CC12 C1(C(N2C(C)(COC)CCC2)=O)CC(NC(=O)Cn2nc(C)cc2C)C12CCC2 CC(C)(O)C#CC(=O)NCC1(NC(=O)CN2CCn3nccc32)CCC1 Cc1nc(NC(C2C3CC2N(C(=O)Cc2nc(C)sc2C)C3)=O)ccc1Br CC1CCN(C(C2CCC(C)CC2)=O)C(C)C1NC(=O)CN1C(=O)CCC1=O C1(CNC(C2(CCOC)CC2)=O)C(C)CCN1C(c1ccc(CC#N)cc1)=O C(CC)(CCC(=O)N1CCC(CC(C)C)C1)NC(C(CC)=CC)=O c1(OCC)ccc(CNC2(c3ccc(F)cc3)CC2)cc1.N1(C(=O)COCC)CCC1 C1(C(=O)NC(C2CCCCC2)C(=O)NCC2(SC)CCC2)CC(O)C(F)C1 C1(C2(O)CCC2)(C(=O)NCC(C)(O)CNC(c2cc(C3CCC3)no2)=O)CC1 N12CCC3(CCCN3C(=O)C(=O)C1c1ccc(I)cc1)C2.C(C)(C)(C)O.CN C1(NC(C2(C)C=CCC2)=O)CN(C(c2cc3c(s2)CCC3)=O)C(C)(C)C1 N1(C(CCSCC)=O)CCC(C=CC(=O)NC2CC(C)(C)C23CC3)CC1 CC1(C)CCn2cc(C(=O)NC3CN(C(C45CC(F)(C4)C5)=O)CCC3F)nc2C1 c1(C(N2CCC(CN(C)C(C3CCCN3C)=O)C2)=O)ccn(C)c(=O)c1 N1(C(c2cc(C)c(I)cc2)=O)CCC2(C)C(C1)C2(Cl)Cl c1(N2CC(NC(C3C(C)=C3)=O)C(C)C2)cc(Cl)nc(C2CCOCC2)n1 C1(C(=O)NC2CC(CNC(CSCC(N)=O)=O)C2)C2COCC12 c1(C(=O)NCCN(C(C(c2nccc(C)c2)(C)C)=O)C(C)C)ccc(C)nc1N.C C1(NC(CC=CC=C)=O)C=CC(C(N2CCC(C(CC)CC)C2)=O)C1 C1(NC(c2cc(CNC(C3(C4CCCCO4)CC3)=O)on2)=O)=CC=C1 Cc1cnn(C)c1CC(N1CCCC1C(C)NC(C1CCN1C)=O)=O C1(CNC(C(C#C)(C)C)=O)COCCN(C(c2cccnc2OCC)=O)C1 CC1(C)CC(C2CCC2)N(CC(=O)Cc2ccc(F)cc2F)C1 c1(CN2CC(CNC(c3ncn(C)c3)=O)C2)nccc(OCC(F)(F)F)n1 C1(NC(c2ccc(C(=O)OCC)nc2)=O)CCN(C(=O)C(F)F)CC1F c1(C(N(CC(C)N(C)C(c2ccc(Cl)cc2)=O)C)=O)ccc(Cl)nc1N CC(C(C)(C)C)=CC(=O)N(CCC(=O)NCC(CC1CC1)CO)C1CC1 c1(C(N2C(C)C(C(=O)NC3CC(n4cccn4)C3)CCC2)=O)cc2cccnn2c1 C1(NC(CC2COCC(C)(C)O2)=O)CC2CCC(C1F)N2C(c1coc(Cl)n1)=O C1(CC=C)(NC(=O)CCC2CC2(Cl)Cl)CCN(C(C2(CO)CCCCC2)=O)C1 N1(C(C2CC(=O)OC2)=O)CCC(O)(Cc2cccc(Cl)n2)C1.n12cc(nn1)C2 N1(C(CCC(=O)OCC)=O)CCCC(C2CC2NC(=O)Cc2cnco2)C1 C1(C)(CCNC(Cc2cn(CC)nn2)=O)CCCC1NC(C1CC(C)OC1=O)=O c1(CC)[nH]nc(C(=O)N(CCCCNC(=O)CC2C(C)(C)C2(C)C)C)c1Br N1(C(C2(F)C(C)C2)=O)CC2OCC(NC(c3ccsc3-n3cnnn3)=O)C2C1 N1(C(CCC=CC)=O)CCN(C)CC1CNC(c1cnccc1Cl)=O C12CCCN(C1)C(=O)CCN(C)C2=O.c1(C2(C(=O)NC)CC2)cncn1C CC(C)CC(CNC(=O)CCc1ccccn1)C(=O)NCC(N1CCCCC1)C N1(C(c2ccc(-c3nc4c(s3)CCCC4)s2)=O)CCC(C2(O)CC2)C1 C1(C(N2CCC(CNC(=O)Cc3ccon3)C2)=O)(SC)CCC(C)(C)C1 C(=O)(CCCCCN(C)C)NCCC(C)NC(c1n[nH]c(=N)[nH]1)=O CCN=c1nc(C(N2CCCC2CN(C(=O)CC(C)F)C)=O)cc(C)[nH]1 C1(CC)CN(C(C2(COC)CCCC2)=O)CC1C(=O)NCCOC(F)F c1(C(N2CCC(C)(NC(CCOCC#C)=O)C2)=O)cc2c(s1)CCC(C)C2 CCCC(CCNC(C1(F)CCN(C(C2COCC(C)O2)=O)CC1)=O)CCC c1(CC(=O)N(C(C)CNC(C2(C(N)=O)CC2)=O)C)cc(F)ccc1F C1(C(N2CCC(N(C(c3c(CC)cns3)=O)C)C2)=O)(OC)CCCCCCC1 C1(CNC(c2ccc(CC)nc2)=O)COC(C)(C)CN1C(=O)C=C(C)C(C)(C)C c1(NC(C)=O)ccc(Br)nc1CS(=O)(=O)N.c1(N)nc(C(F)(F)F)cs1 C1(c2ccccc2)(Cc2nc(CS(=O)(=O)CCN3CCCC3)no2)CCOCC1 CC(C)CS(=O)(=O)CC(=O)NC1CC1NC(C1CC(O)C1)=O.C(C)(=O)O C1(C(C)C)CN(C(=O)C(C)C2(O)CCC2)CCN1C(C1CC1C(C)(F)F)=O C(=O)(C(C)(C)C1CCCO1)NCC1C(NC(CN2CC(C)C2)=O)CC1 c1(NC(C2OCCN(Cc3ccc(C)cc3F)C2)=O)cccc2nc(O)oc12 S(=O)(=O)(c1cc2sc(=NC(CCO)C3CCC3)[nH]c2cc1Cl)N(CCCCC)C N1(C(C(CCC)(C)C)=O)CCC(NC(C2(C)CCCS2)=O)CC(O)C1 c1(C(=O)OC(C)C(=O)NCc2ccc(F)cc2)cc(S(C)(=O)=O)cs1 N1(C(C(CC)OC)=O)CC(CNC(c2cccnc2NC)=O)C(C)(C)C1 c1(OCC(=O)O)ccc(CCNC2CCC(CNC(c3ccc(Cl)cn3)=O)C2)cc1 c1(OC)c(C)ccc(C(=O)NC(C)CN(c2nccc(SC)n2)C)c1F c1(OC)ccc(C(=O)NCC2CC(F)(CNC(=O)C=Cc3ncc[nH]3)C2)nc1 N1(C(C2C(C(N)=O)C2)=O)CCN(C(=O)COCc2ccccc2)C2(CC2)C1 c1(C(N(CC(=O)NCC(C)(F)C(C)C)CCC)=O)ncnc2cc[nH]c12 c1(CC(=O)N(CCNC(C2CC(CC)C2)=O)C)ccc(OC)c(OC)c1Cl c1(C(N(C2CCC2)C)=O)cc(OC)c(-c2cn(CC(C(=O)OCC)O)nn2)nn1 c1(C(=O)NC(C)CN(C(=O)Cc2nccs2)C)c(C#N)cnn1C C1(NC(C2CC(F)(F)C2)=O)CC2CCC1N(C(=O)C(c1ccc(F)cn1)(F)F)C2 c1(OC)c(C)cc(CN(C=O)CC2CC23CC3)cc1C C1(C(=O)NCC(C)NC(=O)C(C)Cc2ccccc2F)CCCC(C)(C)C1 C1(NC(C(CNC(C2(CC(C)C)CC2)=O)O)=O)CCN2CCC1C2 c1(C(C)C)cc(F)ccc1NC(=O)C(=O)NCc1nccn1-c1ccccc1 C(C)(C)(CC(=O)NC1CC(C)OC1=O)N(C(COCCN(C)C)=O)C c1(CC(=O)NC2C(NC(C(C)=CC)=O)C2)ccc2nn[nH]c2c1 c1(C(N(CCC)CCNC(=O)C(C)Cn2ccc(C)n2)=O)ccc(O)c(Cl)c1 c12cc(on1)C2.C1(Cn2ccnc2)CCN(C2CC2)C1 CC1CN(C(c2cc(O)cc(O)n2)=O)CCC1NC(c1ccc(C(N)=O)nc1)=O c1(N2CC(NC(C(CCCC)C(C)C)=O)(CO)C2)nc(Cl)nc2c1COCC2 C1(CCNC(=O)CC(F)(F)F)CN(C(=O)COC2CCCOC2)CCCO1 Cc1cc(NC(=O)CC2OCCC2(C)C)ccc1NC(=O)C(c1csc(C)n1)=O C(=O)(CCCCN1CCCC1)NC(CC(C)NC(C1C2CCC(=O)C12)=O)C c1(OCC#C)ncccc1C(=O)NCCNC(C1CC(=O)N(CC(C)C)C1)=O CN1CCOC(C(=O)NC2CCN(C(c3cnns3)=O)C23CC3)C1=O Cc1ccc(C2CCCN2C(c2nc(C)cs2)C(=O)NCC2CC2)cc1 c1(C(=O)NC2C(NC(c3cc(C)sn3)=O)CCC2)cc2ccccc2o1 N1(C(c2c(C)coc2)=O)CC2CCN(C(C3CCC(=O)N3)=O)CCC2C1 c1(CC)cccc(CC)c1C(=O)N(C)CC1CN(C(c2cncc(O)c2)=O)C1 C(C(C)(C1CC1)NC(C1CC(CF)C1)=O)NC(CC1(OC(C)C)CC1)=O CCCC(C)(C)CC(=O)NCC(CC(F)(F)F)NC(c1cnn(C2CC2)c1)=O C=CC1OCCC1N=c1nc2ncn(C)c2c(NCCCC2CCOC2)[nH]1 C(=O)(C(Cc1ccccc1)N(C)C)N(CCC(C)NC(=O)C(C)(C)F)C CC(C)C(CCN(C)C(c1occc1C1CC1)=O)NC(=O)C=CCO C1(CN(CC(=O)NCCCO)C)CCCO1 C(=O)(CC(C(F)F)C(C)(C)C)N1CC(NC(CSCC)=O)C(c2nccn2C)C1 C1(CNC(c2cc(OC)no2)=O)CN(C(C2CCC3(CC2)CC3)=O)C2CCN1C2 C1(C(=O)NCCC(C(C)C)C)CN(C(c2cccc(CO)c2)=O)CCN1C N1(C(c2c(C)c[nH]c2)=O)CCC2CC12C(=O)NCCC(C)C(F)F C(C)(CCC(=O)N(C)C(C1CCOCC1)C)NC(C(C)=C(CC)C)=O N1(C(C(C)(O)C2CCC2)=O)CCCCC(CNC(c2ncsc2Br)=O)C1 C12(C(=O)NCC3(COC)CCN(C(CCC(=C)C)=O)C3)CCCC1CCC2 CC(CC(=O)NCCC1(C)CCN(c2nnn(C)n2)C1)CC(C)(C)C C=CCC(C)(C)NC(=O)C(C1CN(C(=O)C(C2CCCC2)OC)C1)OC Cc1nonc1CC(=O)NCc1cn(CCNC(=O)CN2CCCC2C)nn1 C=CCC(C)C(=O)NCc1cc(C(=O)NC(C2(OC)CCC2)C)n[nH]1 C1(C(=O)NCCCOCCC(=O)N(CC(C)CO)C)(CC)CCOC1 N1(C(c2ccc(C)cc2Cl)C(=O)NC(CC)C)CCNC(=O)C1(C)C C1(NC(Cc2c(C)n[nH]c2C)=O)CC2(C1)CC(NC(c1cocn1)=O)C2 C#CC1(C(N2CCN(C(=O)NC)CC2)=O)CCN(C(=O)C=CC(C)C)C1 C1(C)(C(=O)NCCC(C)CCNC(=O)CCCn2ccnc2)CCCC(F)(F)C1 c1(C(N2CC(NC(C(C)O)=O)C(c3ccccc3F)C2)=O)nc2c(s1)CCC2 c1(OC)ccc(CN2CCCC(C(C)NC(=O)C(N)CO)C2)c(Br)c1 CC(C(C)(C)CN(C)C)NC(=O)CC1(NC(=O)Cc2cccnc2)CC1 N1(C(c2cc(CC)sn2)=O)CCCC(C)(C)C1CNC(C1(C2CCCO2)CCC1)=O c1(C(=O)NC(C)CNC(=O)CCNC(c2ccco2)=O)cccc(Br)c1O c1(CC(=O)NCc2cccnc2)ccnc(O)c1.C1(=O)NOCC(=O)OCC2C1C2 c1(CC)ccc(C(N2CC(CC)C(CNC(=O)CN3CCCC3C)C2)=O)cc1 Cc1c(C(N2CCCC2C(N2CCSCC2)=O)=O)cccc1O CC(CC(N)=O)C(=O)N(C)CC1CCN(C(=O)Cc2cc(F)ccc2O)C1 C1(NC(C2(C)CCN(C(c3ncn4ccccc34)=O)C2)=O)CCc2n[nH]cc2C1 N1(C(C(C)OCC)=O)CC=CCC1C(N(C)Cc1cn(C)cn1)=O C12(C(=O)NC3(C)CCCN(C(Cc4nc(C)sc4)=O)C3)CCCCC1OCC2 c1(OC)ccc(Cl)cc1C(N1CC2CC(NC(C3CC(=O)NC(=O)N3)=O)C1C2)=O c1(C(C(=O)N(c2ccccc2)CCN2CCC(N)C2)N(C)C)ccc(Cl)s1.CO C(CCS(C)(=O)=O)(C(=O)OC)n1cc(C2CCN(C(CC(CC)O)=O)C2)nn1 n1(CC(=O)N(C(CNC(c2cn(C3CCC3)nn2)=O)C2CC2)C)cccnc1=O C(c1ccccc1C)=CC(=O)N(CC(CNC(CCC(C)SC)=O)O)C CC1(C)CC(CO)CN(C(=O)C(C2(C)CC2)NC(c2ccc(C#N)cn2)=O)C1 C1(NC(C2C(C)OC(=O)N2)=O)CN(C(=O)Cc2ccco2)CC2CCCC12 c1(OCCC)ccc(CC(C2C3COCC23)c2nnnn2C2CC2)cc1OC Cc1cc(Cl)c(C(=O)NC2CCC2NC(C2CC2C(c2ccccc2)=O)=O)cc1N c1(OC)c(C(=O)NC(CNC(C2CC2F)=O)C(C)C)ccc(Br)c1F c1(C(N(CC(C)N(C(CCOC(C)C)=O)C)C)=O)cn(C(C)(C)C)cn1 c1(C(=O)NCCOCCCNC(C2(CCOC)CCC2)=O)ccc(C)c(C)n1 N1(C(c2ccn(C(C)C)c2)C(=O)NCCC)CC2CCCC2(C(N)=O)C1 C(COC(C)(C)C)(C(=O)NC(C)CC(C)NC(=O)Cc1cnsc1)N(C)C C(=O)(C(C(C)C)c1ccc(Cl)cc1)Nc1c(C(=O)OC)ccs1 CCCC(CC)CC(=O)N1CC(C2CN(C(C3(OC(C)=O)CC(O)C3)=O)C2)C1 c1(SC)cccnc1C(=O)NC(C)CC(C)NC(c1csc(-c2cn[nH]c2)n1)=O N1(C(c2ccc(N)cn2)=O)CC2(NC(C3OC4CCC3C4)=O)CCC1C2 n1(CC(=O)N(C)CC2COCCN2C(=O)C(F)n2cccn2)cc2ccccc2n1 C1(CC)CN(C(c2coc(C(F)F)n2)=O)CCC1NC(c1nc(=O)n(C)[nH]1)=O C1(C)(C(=O)NCCC2(O)CN(C(COC(CC)(C)C)=O)C2)CCC(C)=C(C)C1 C1(CNC(c2c(C)c(N)ccc2)=O)(NC(=O)C=C2CCC2)CCC(F)(F)CC1 C(=O)(CCCCCSC)N(C(C)CO)CC.C1C(=O)N1 CC(C#N)CCC(=O)NC1(C)CN(C(=O)CCc2ccc(Cl)c(F)c2)C1 C1(NC(C2CC(OCC)C2)=O)CCCC(C(=O)NCC2(CO)CC=CC2)C1 c1(C(N2CCc3ccc(Br)cc32)C(=O)NC)ccc2c(c1)OCC(=O)N2 C(=O)(C(Cc1cc[nH]n1)NC(=O)CC1CC(C)=NO1)NC(C)Cn1cccn1 Cc1cc(N)c(C(=O)NC2CC(NC(=O)COc3ccccc3)C(O)C2)nc1C Cc1nc(C(N2CCCCCC2CNC(=O)C(F)C(C)(F)F)=O)ccc1C#N c1(C(N2C(C(=O)Nc3c(SC)ccnc3)CC(F)C2)=O)csc2ccccc12 N1(C(CCCOCCC)=O)CCN(C(=O)C#CC2CCC2)CC1CF C(=O)(C1=CCCC1)N(C1CN(C(C2(C)CCCO2)=O)CC1F)C CCC(CC)C(=O)NCC1(F)CCC(NC(c2ncoc2-c2cccs2)=O)C1 CC1C(C)N(C(c2nocc2Br)=O)CCN1C(c1ccc(C#N)n1C)=O c1(CCCCN(C2CCCCC2)C(=O)CCc2ccccn2)cn2c(n1)SCC2 C1(C(=O)NCC2OCCCN(C(c3nc(C)n(C)n3)=O)C2)CCC(N=[N+]=[N-])CC1 C1(NC(CS(N)(=O)=O)=O)CC1C1CCCN(C(c2ccnc(C3CC3)c2)=O)C1 C1(NC(Cc2c(C)nn(C)c2)=O)CCN(C(=O)Cc2ccno2)C12CC2 c1(C(N(C2CCN(C(=O)CO)CC2)CC#C)=O)ccc2cc(C)ccc2n1.NCC n1(CC)c(CNC(=O)C(C)N(C(=O)CCC2(C)CCC(=O)N2)C2CC2)cnc1C c1(CNC(c2c(C)[nH]nc2F)c2nnnn2C2CCOCC2)cccc(Cl)c1O c1(OC)cc(C(=O)Nc2ccc3nc(C)cn3c2)cc(F)c1OC C1(NC(C2CCC3(CCC3)O2)=O)CN(C(=O)CCSC2CCCC2)CC2(CC2)C1 CC1CCCC(C)N1C(=O)CN1CCC(N(C)C(C2CCC2(C)C)=O)C1 C=CCC(C(=O)NC1CN(C(=O)CC23CCC(CC2)OC3)C(C)(C)C1)C(C)C C=Cc1cnn(C)c1C(=O)NCC(C1CCCN1C(=O)Cc1ccn(C)n1)(C)C N1(C(C(CO)N(C)C)=O)CCC2C(C(=O)NCCCN3CC=CC3)C2C1 C1(C(C)C)CCNC(=O)O1.c1(COCC)ccc(OCCCl)cc1 CC(C)CC(F)C(=O)N1CCCCC1C1CCCN(C(=O)C=CC2CCC2)C1 C1(CNC(c2[nH]cc(C)c2)=O)CCCCC1NC(=O)Cc1conc1C C1(NC(=O)Cc2ccccc2Cl)CCN(C(c2coc3c2COC3)=O)CC(O)C1 CCC(CNC(C1CCN(C(C2C3CC4C(C3)C24)=O)C1)=O)(CC)C(N)=O C1(NC(c2n(C(C)C)ncc2)=O)CN(C(C23CCCC2C3(F)F)=O)C2CCCC12 C(=O)(CC(C)(F)F)N(C1CCCCC1)CCNC(C1N(C(C)=O)CCC1)=O C1(NC(COCCNC(Cc2cc(C)sc2)=O)=O)CC2C=CC1C2 C1(CC(=O)N(C2CC2)CC2C(C)C2)COCCN1C(c1cc(=O)cc[nH]1)=O Cc1ncsc1C(=O)NCCC(C)NC(c1ncoc1C1CCCO1)=O Cc1cn2cc(C(=O)N(CC(C)(C)CNC(=O)Cn3ncnn3)C)nc2s1 C1(NC(CCCOC(C)C)=O)COC2CN(C(=O)CCc3cccnc3F)CC12 c1(C(=O)NC(CC)CN(C(=O)C(O)CC(C)C)C)cc2c(s1)CCCCC2 Cc1c(F)c(C(N2CC3CC2CN3C(c2cncs2)=O)=O)nn1C C#CC1CC2CCC1N(C(c1cnn(CCNC(C3CCCOC3)=O)c1)=O)C2 C1(OC)CC(NC(=O)CCC(=O)N(C)C)CN(C(c2cn(CCO)nn2)=O)C1 N1(C(c2cn(C)nc2)=O)CC2CC1CC2NC(c1cccn(C2CCC2)c1=O)=O CC(C)(C)C(C(=O)NCCc1ccc(F)c(F)c1)n1cc(-c2ccccc2)nn1 Fc1ccc(C(C(F)F)NCc2ccc(C(F)(F)F)o2)cc1F N1(C(C)=O)CC2CC1CN2C(=O)C(C)N(C(=O)CC(C)C(F)F)C1CC1 C(=O)(CCCCC(N)=O)NCCC1(NC(C(c2ccccc2F)OCC)=O)CC1 c1(C(=O)NC(C2(O)CCN(C(C3(CC4CCC4)CC3)=O)C2)C)cc2ccsc2s1 N1(CCNC(CCN(C(=O)CCc2ccc(C)s2)CC)=O)CCOCC1=O C1(CCC)(NC(c2ccsn2)=O)CCN(C(c2ccc(O)c(Cl)n2)=O)CC1 C12(NC(CCCCCN(C(C(C(C)(C)C)OC)=O)C)=O)CCC(CC1)C2(C)C N1(C(c2scc(C(=O)OC)c2)=O)CCCCC(NC(c2conc2C)=O)C1 C(=O)(CCC(F)(F)F)NC(C(=O)NCCOC)C.CCC(C)N(C)C N1(C(c2ccn(CC)n2)=O)CC2CCC(C1CO)N2C(C1(OC(C)=O)CC1)=O C1(C(N2CCC(OCC#C)C2)=O)CC(NC(C2CCC2C)=O)CCO1 C1(CNC(c2n(CCOC)ncc2)=O)C2CC2CN1C(c1nccnc1N)=O C1(NC(C2N(C=O)CCC2)=O)CCN(C(=O)CSc2cn[nH]c2)CCC1(F)F Cc1ccc(F)c(C(=O)NCc2nnn(C)c2C(=O)NC2CCCCC2CO)n1 c1(CN(C2CCCC(C)C2)CCC)cc2ccccc2n1C C(C(CC(C)C)C(=O)NCC1CCCCC1(C)C)OC.c12n[nH]cc1C(=O)N2 c1(C(=O)OCC)noc2c1CN(C(=O)NC1CCCC13CCCO3)CC2 N(C1CS(=O)(=O)Cc2ccccc21)c1cc(NC2CC(C3CCC3)C2)nc(C)n1 Cc1nn(C)c(Cl)c1C(=O)NC1CCCC1CNC(=O)CCN1C(=O)CCC1=O N1(C(c2c(CC(C)C)onc2)=O)CC(C)N(C(C2C3CCCCCC23)=O)CC1C N1(C(c2c(OC)nc(Cl)cc2)=O)CCC2(CCC(NC(=O)C(C)C3CC3)C2)CC1 N1(C(CSCC)=O)CCCC1(CO)CNC(c1ccccc1CC)=O O=C(CC(C(F)F)NC(c1ccccc1F)=O)NCCCC1CCCCO1 Fc1ccc(CNC(=NCCN2CCCC2)NCC2CCC23CCC3)c(F)c1 C(C)(C)(C(=O)NC1(C)CC(C(=O)NCC(N2CCOCC2)C)C1)NC(=O)OC N1(C(CCCNC(=O)OC)=O)C2CCC1CC(CNC(C13CCN(CC1)C3)=O)C2 N#Cc1nccc2cc(NC(c3ccc(Cl)c(Cl)c3)CO)ccc12 C(=O)(C1=CCC(NC(=O)CC2CCCOC2)C1)N(CCOC)CCO CCCCC(=O)C(=O)NCC1CC1CC(=O)N(CC)Cc1nncn1C C(=O)(CCCC(C)(C)C)NC(CNC(C(C)Cc1ccncc1)=O)CC(F)(F)F C=CCC(CC(C)C)C(=O)N1CCC(N(C(=O)C(CC)(CC)CC)C2CC2)CC1 N1(C(c2cc(C#N)[nH]c2)=O)CCOC2(CCN(C(C3CC3(F)Cl)=O)CC2)C1 c1(OC)cccc(Br)c1C(N1CCN(Cc2cccc(O)c2C)C(C(C)C)C1)=O n1(CC(=O)NCC2CC2NC(c2ccco2)=O)ccc(Br)n1 C(C(C)(C)CC(=O)N1CCOC(C(N2CCC(C)=C(C)C2)=O)C1)OC C1(CCC(=O)NCCCCC#CC)CCCCN(C(=O)C(CC(C)C)N(C)C)C1 C1(O)(C(C)NC(=O)CCc2cnccn2)CCN(C(C2CCCOC2C)=O)CC1 N1(C(CCOCC#C)=O)CCC(=CCC)CC1.C(=O)(C(F)=CC)NCC=C CCCCC(C(=O)NCC(C1CCCC1)NC(=O)C(F)(F)CC)NC(N)=O C1(C)(CC)CC(NC(=O)C(C)(C)c2cccs2)CN1C(C1CN(C)C1)=O C1(CNC(CCCOCCC)=O)CCN(C(C2(O)CCOC2)=O)CC1(F)F C1(CNC(c2cc(CC)no2)=O)CC2CN(C(=O)Cc3cccnc3OC)CC12 C1(C(=O)NC(CC(C)NC(=O)CS(N)(=O)=O)C)CCCCC1N=[N+]=[N-] C(=O)(C1CCCc2scnc21)NC1CC(CNC(c2nc(OC)c(F)cn2)=O)C1 N1(C(C(CC)OC)=O)CCC2(CC1)CC2C(N1CC(OC2CCCC2)C1)=O C1(C(=O)NC(C(=O)NC2CN(CC)CC2C)Cn2ccnn2)CC(C)(C)CCO1 C1(CN2C(C)CCC2C(=O)NC(C2(C)CC3CCC2C3)=O)Cc2ccccc2C1 c1(C(N(CC(CC)NC(=O)C#CC2(C)CC2)C)=O)cccc(Br)c1Cl C12(CC)CCCN(C1)C2=O.C1(CNC(CCOCC#C)=O)CCCC1CCC C(=O)(C(C#N)C(C)(C)C)N1CCCC(C)(C(=O)NCC2CC=CCC2)C1 N1(C(C=C(C)C)=O)CC(F)(F)CC1C(=O)NCCCC1(O)CC1 N1(C(c2cccs2)=O)C(c2ccccc2)CC12CCC2.CC1CCCNC(=O)N1 C(C(C)(O)CNC(=O)COCCc1ccccc1)NC(C1C(CN(C)C)C1)=O C(=O)(C(CNC(=O)CC1COCCO1)C(C)(C)C)NCc1cncc(CC)c1 c1(C(N2CC(C(=O)NC(CCN(C)C)(C)C)C(O)CC2)=O)cnn2cccnc12 c1(C(C)=O)cc(C(=O)N(CC(C)NC(c2ccc(C(F)(F)F)o2)=O)C)oc1C Cc1cc(C(N2CCCC2(C)CNC(=O)Cn2ncnn2)=O)cc2ccoc12 C1(C(=O)NCC2CCN(CC=C)C2)CCc2ncnc(C)c2C1 O=C(C1=C(Cl)CCC1)NCCOC1CCN(C(=O)CCSc2ccncc2)CC1 N1(C(CC2(C)CCC2)=O)CCN(C(=O)CCC2CC2)C(CC(F)F)C1 c1(C(=O)NCC(CCNC(C=CCCC)=O)O)cc(CC)c(C)s1 CC(N=[N+]=[N-])C(=O)N(C)CC1CCCCN1C(=O)CCCC1CC1 CCC(O)C(C)C(=O)NCc1ccc(CNC(=O)C2=CC(C)(C)C2)cc1 C1(CC)CC(C(=O)NCCCCCOC)CN(C(=O)C(F)(F)F)C1 Cc1cc(CC(=O)NC(Cc2cn[nH]c2)C(=O)NC2CC(OCF)C2)nn1C N1(CCCC(=O)NC(CNC(C2C(C)C2)=O)(C)CO)CCc2ccccc21 C1(SCCn2c(-c3c(-c4cc(C)nn4C)cccc3)ncc2)CCCCCCC1 C1(O)(CNC(C(C)OC)=O)CCN(C(c2ccc(C(=O)NC(C)C)cc2)=O)C1 C1(NC(c2cc(C)c(C)s2)=O)CCCN(C(c2ccccc2F)=O)CC1F c1(OC)cc2ccccc2cc1C(=O)NCCN(C(C1CCNC1=O)=O)C1CC1 O=C(C1COc2ccccc21)NC12CC(CNC(=O)CN3CCCCS3(=O)=O)(C1)C2 C(=O)(C(C)C(C)NC(c1oc(CNC(C2CC(=O)C2)=O)nc1C)=O)OC Cc1cc[nH]c(=N)c1C(=O)NC1CC(NC(=O)CS(N)(=O)=O)C12CCC2 C(c1ccc(Cl)s1)=C(C#N)C(=O)NC(CC(N)=O)c1cn(C2CCC2C(=O)O)nn1 c1(C(=O)NCCCn2cc(COC3CCS(=O)CC3)nn2)ccnc(F)c1F C1(NC(C(C)C2CCCO2)=O)Cc2ccccc2C1NC(=O)CCc1nc[nH]n1 c1(C(C(=O)N(CC(C)NC(C2C=CCN2)=O)C)C)ccc(Cl)cc1 C1(CNC(c2cnc3nccn3c2)=O)CN(C(c2ccco2)=O)C2COCC2O1 C(CC(=O)N1CC(OC(=N)O)C1)N(C(=O)C(C)C1CCC1)CC=C N1(C(c2c(C)nc(CO)o2)=O)CCCC(NC(=O)CC23CCCC2C3)C(F)C1 C1(NC(C2C3CC4C(C3)C24)=O)CC2CC(C1)N(C(c1ccn3nncc3c1)=O)C2 c1(OC)cc(F)c(F)cc1C(=O)NCc1cnc(OC)nc1 N1(C(C2=C(C)CC2)=O)CC2CC(CNC(c3ncccc3Cl)=O)CC1C2 C1(NC(CC2(OC)CC2)=O)CC(C)CN(C(C2(C)COC(=O)N2)=O)C1 C(=O)(C(F)CCC(C)C)N1C(C(=O)NC(CCC(=C)C)C)CCC1C(C)C C(CO)(C(C)(C)CO)NC(C1C(C(C)NC(C2C=CCCC2)=O)C1)=O c1(N2C(CNC(C3CC(=O)NC3)=O)CCC2)ccn2nccc2n1 C1(NC(C(C)OCC(F)(F)F)=O)COC2(C1)CN(C(c1cccn1C1CC1)=O)C2 C=CC1(CC(=O)NC2CC(NC(=O)CC34CCCC3C4)C(O)C2)CCOCC1 CCC(C(=O)N1CC(CNC(c2ccc(F)cc2F)=O)C2(CCC2)C1)C(F)(F)F C=CC(C)(CCOC)C(=O)N1CC(CN(C)C(c2cncc(C3CC3)c2)=O)C1 C1(CNC(c2ccccc2)=O)CCC(C(N2CCC(N(C)C)C2)=O)O1 CC1=NN(C)C(=O)C1CC(N1CCC(NC(C2COCCO2)=O)C12CC2)=O C1(C(N(C2CCN(C(=O)Cc3cccc(SC)c3)C2)CC)=O)(CF)CCOCC1 CCCCCCCNC(=O)CCn1cnnn1.c12nnc(s1)CN2.OC C(=O)(N=c1ccn(CCCO)[nH]1)C1CC2(CC(NC(CCC(=O)OC)=O)C2)C1 c1(C(N2CC(C(C(=O)NCC3CCC3CO)OC)C2)=O)csc(Cl)n1 N1(C(c2c(CC)ncs2)=O)CCC(CNC(C2(O)COC2)=O)C(C)C1 C(=O)(C(C)CCNC(=O)OC(C)(C)C(=O)OC)NC1CN(C(CCOCC)=O)C1 C1(CNC(=O)CSc2nc[nH]n2)CCCCN1C(=O)Cc1ccco1 N1(C(C(C=CC)O)=O)CC(O)CC1(C)C(=O)NOC(c1ccccc1)C Cc1cc(N)ccc1C(=O)NC(C)CNC(C12CC(CO)(C1)OC2C)=O CC1(C)OC(=O)NC1CNC(C1(CO)CCN(C(=O)C(C2CCOCC2)=O)C1)=O C(CCC(C)CN(C(C)=O)C)=CCNC(=O)C(=O)N(C)C(C)C c1(CNC(C(CC)(C)OC)=O)ccc2c(c1)CCC2NC(c1cscc1F)=O CC1OC2CCC1(C(=O)Nc1ccccc1-c1ccccc1OC(F)F)C2 Nc1cccc(C(N2C3CCC2C(NC(=O)CCc2ccccc2Cl)C3)=O)c1O N1(C(C(C)OCC(C)C)=O)CCCC1(C)CNC(=O)CNC1(C)CCC1 C(=O)(C(C(C)C)C(C)C)N1C(CC)C(NC(c2cccc(C)n2)=O)CCC1 C(N=c1nc2ncn(C)c2c(NCC(CO)C(C)C)[nH]1)c1c(C)cco1 c1(OCC)cc(CN2CCC(CNC(=O)CC3CCC3)C2)ccc1OC C(N=c1[nH]c(=NC2CCCCC2C#N)c2ccccc2[nH]1)c1c(C#N)scc1 c1(C(=O)NC(CC(C)C)CNC(=O)C(C2CCCCC2)F)cccc2cnnn12 c1(CNC(N(CCC(=O)OC)CCC)=O)nc(C)[nH]c1C(F)(F)F C(C#Cc1cn(CC(C)C)nn1)NC(C1C(C)CC(=O)NC1)=O c1ccc(C=C2CC3CN(C(C=C)=O)CC32)cc1.c1(C(N)=O)ccccc1 N1(C(Cn2ccc(C)n2)=O)CCC(F)(CNC(C2CCN2S(C)(=O)=O)=O)C1 N1(C(C(C)O)=O)CC(S(=O)(=O)N2CCN(C(c3n[nH]c(=N)s3)=O)CC2)C1 c1(C(N2CC(CCC)C2)=O)ccc(CNC(C2(OC)CCC2)=O)cn1.O(C)CC C1(CNC(C(C)(C2C(C)C2)NC(CCS)=O)=O)C2CCCCCC12.C1CCC1 CN1CCCC(O)(CC(=O)NCC(C)(C2CC2)NC(c2ccnc(CO)c2)=O)C1 c1(C(N2CC(OCCNC(C3(C)C=CCCC3)=O)C2)=O)cc2c(s1)CCC2=O Cc1ccc2c(C(=O)NCC3CCCCC3NC(=O)CS(C)(=O)=O)coc2c1 N1(C(CCSCC)=O)CC(CNC(=O)CCCCN(C)C)CCC1C Cc1cc(C(=O)NC2CCCC23CN(C(C2CCN(C)C2=O)=O)C3)c(O)nc1C Cc1ccc2snc(C(=O)NCCC(O)CNC(=O)CCc3nc[nH]n3)c2c1 C1(NC(C2CC(NC(COC3(C#C)COC3)=O)C2(C)C)=O)CCCCC1N=[N+]=[N-] c1(CC(=O)N(CCN(C(CCN(CCOC)C)=O)C)C)nc(C)sc1Cl c1(CC(=O)N(CCC(C)NC(C2(CF)CC2(F)F)=O)C)ccccn1 N1(C(C2(OC)CCCCC2)=O)CCCCC(NC(C2OCCOC2(C)C)=O)C1 C1(NC(=O)Cc2ccccc2)CCN(C(=O)CCCF)CCC1CO C1(CC(=O)NCCCSCC)CN(C(C2(c3cc[nH]n3)CC2)=O)CCO1 N1(C(C(c2cccc(F)c2)C)=O)CCc2[nH]nc(CNC(=O)COCCF)c2C1 c1(C(=O)NC(CNC(C=Cc2n(CC)ccn2)=O)C2CC2)ncc(Cl)cc1Cl C(=O)(C(=O)CC(C)C)N1CCC(OCC(N2CCC(N(C)CC)CC2)=O)C1 N1(C(CCC2N(C)CCC2)=O)CC(C)(C(=O)Nc2ccc3c[nH]nc3c2)CC1(C)C C1(CNC(C(CC=C)c2ccccc2)=O)CN(C(C2(CC)CC2)=O)CC(C)(C)C1 C1(CNC(c2c(C(C)(C)C)ncs2)=O)C2CN(C(c3cc(Br)n[nH]3)=O)CC12 c1(N(CC(=O)NC(C2(O)CN(C(C(COC)O)=O)C2)C)C)ccccc1[N+](=O)[O-] c1(C(C(=O)NC(CCCNC(C2C(OCC)C2)=O)C2CC2)CO)ccc(Cl)cc1 CN1CCCCC(NCC2CCCN(c3cc(CC4CC4)ncn3)C2)C1 Cc1cc(CNC(C2(N(C(C3CC4CC3CC4O)=O)C3CC3)CCC2)=O)cc(C)n1 C(=O)(C(C)(C)CC(=O)OC)N1CCN(C(COCCCCC)=O)CC1CO N1(C(CC=CCC)=O)CC(NCc2cc(Br)c(C)cn2)CC(C)C1 CCCCCC(=O)NCC(N1CC(CNC(=O)C(C)(C)C2CC2)C(C)C1)=O C1(CNC(C(CCC)OC)=O)COCCN(C(=O)CC2COCC2(C)C)C1 C=CCC(C(=O)NC1CC1CNC(c1ccnn1C1CC1)=O)C(C)C c1(OC)ccnc(C(=O)NCCCCC(C)NC(c2cncc(F)c2)=O)c1OC Cc1cnc(N2CC=CCCC2)c(S(=O)(=O)NC2CCc3nccnc32)c1 N1(C(C(C)NC(C)=O)=O)CC2CC(C1)N(c1ncc3ccsc3n1)C2 C1(CC)CCN(C(c2ccc[nH]2)=O)C1C(=O)Nc1ccccc1O C(=O)(C(C)(C)CC(=O)N1CCCC(N(C(=O)CC2(C)CCCO2)C)C1)OC N1(C(c2ccnc(Br)c2Cl)=O)CCCC2(CCCN(C(C3CCCCC3)=O)C2)C1 C1(C2(O)CCN(C(=O)Cc3cccc(CO)c3)CC2)(NC(=O)C=CC2CC2)CC1 N1(C(C(=Cc2ccncc2)C)=O)CCC(N=c2c(Br)c[nH]cc2[N+](=O)[O-])(CO)C1 C1(C(=O)NCCCOCC)CCN(C(=O)C2(C)CC2(C)C)O1 c1(-n2cc(C(CCC)NC(C3CCC(C)(CC)C3)=O)nn2)cc(Br)ccc1OC c1(C(N2C(C3CCN(C(CSC(C)C)=O)C3)CCC2)=O)cc2cc(N)ccc2s1 C(=O)(CC(F)(F)C(F)F)N1C(CNC(C2CC2Cl)=O)CC1 n1(CC(=O)NCC(Cn2cc(CC(C=C)O)nn2)(C)C)cc(S(C)(=O)=O)cn1 C1(C(=O)NCCCC(C)O)NC(=O)OC1(C)C.c12coc(n1)CONC2=O Cc1cc2c(C(N3CCC(C)(CNC(=O)C(C)O)C3)=O)nccn2n1 N1(C(c2cnc(C(C)C)o2)=O)CC(C(=O)NC2CC23CCOCC3)C2(CC2)C1 C12CCCC1CNC2=O.C(C(C)C#N)N(CC)CC.C(=O)(C(C)n1cnnn1)NC C1(NC(CCOC(C)C)=O)CCCN(C(=O)CCC2NC(=O)NC2=O)C1 C12(NC(=O)OC(C)(C)C)CCN(C)CC1CN(C(=O)COc1ccon1)C2 C1(C(=O)NCCC2CCN(C(C(C)NC(C)=O)=O)C2)C(=O)ON=C1C CC(CC(C)(C)C)C(=O)N1CC2CCC(NC(c3cc(CO)[nH]n3)=O)(C2)C1 CC(CS(C)(=O)=O)C(=O)NCc1cccc(NC(=O)CCC2CCCN2C)c1 C1(c2cn(CC(C)(C)C)nn2)(C(=O)OC)CCN(C(=O)CO)CC1 N1(C(C(C)(C(C)C)OC)=O)CCC2(COCCO2)C1 N1(C(C2=NOC(C)C2C)=O)CCCC(NC(=O)C(C)N(C)C)CCC1 C1(NC(C=Cc2cc(OC)ns2)=O)COC2(CCN(C(C3OCCO3)=O)C2)C1 C(=O)(C(F)(F)C(F)(F)C(F)(F)F)NCCC1N(C(CC(C)(C)SC)=O)CCSC1 CC(CCN(C)C)C(=O)NC1CC(C(=O)Nc2ccccc2)CC1O N1(C(COCCOC)=O)CCCC(C(N2CCC(C)(C)C2C)=O)CC1 C=CC1CN(C(=O)CC(CC2CC2)NC(C2CCC2C)=O)CC1O c1(C(N(CCCCC)C2(C(=O)NC3CC(C)(F)C3)CCC2)=O)ccn(C(F)F)n1 c1(COC)ccc(NC(Cc2ccc(Br)cc2)C(=O)NC2CCOC2)cc1F C1(NC(C2(OCC)CCOCC2)=O)CC2CC1N(C(=O)CC1CC(F)C1)C2 Cc1cc(C(=O)NC2CC3(C2)CC3C(N2CCOC(C)(C3CC3)C2)=O)cc(C)n1 N1(C(C2(F)C(C)C2)=O)CCCC(O)(CNC(C2(C)CC=CCC2)=O)C1 c1(C(=O)NC(C)C(CO)NC(c2ccc(Cl)o2)=O)ccccc1Br CC1CCN(C(=O)CC(CC2CC2n2nccn2)NC(C2(CO)CC2)=O)CC1 c1(C(=O)NC(C)CCCNC(=O)C=Cc2cc[nH]n2)cccc(-n2cccn2)c1 N1(C(c2n(C)c(C#N)cc2)=O)CCC2CCCC(C1)N2C(C1CCC(=O)O1)=O c1(C(=O)NCCN(C(c2cncc(OC)n2)=O)C)cc(O)ncc1F C1(C)(CC(=O)NCCCC(C)NC(=O)CCn2cc(Cl)cn2)CC(F)(F)C1 Cn1cc(Br)c(C(N2C3CCC2CC(CNC(=O)C=CC2CC2)C3)=O)cc1=O N1(C(c2ccc(C#C)o2)=O)CCN(C(c2csnn2)=O)C(CCCC)C1 C(=O)(C(C)c1ccsn1)N(CCCNC(C1(C(F)(F)F)CC1)=O)CC C1(SC)CN(C(C23CC(c4ccccc4)C2C3)=O)CC1NC(=O)CSCC(=O)NC C1(NC(C2CC(C(F)F)(OC)C2)=O)CN(C(C2CC(C)(O)C2)=O)CC1O c1(C(N2C(CNC(c3nn(CC)c(C)c3)=O)CC(O)C2)=O)nc(C)n(C)c1C c1(C(C(=O)NCC2C(CNC(c3cncnc3C3CC3)=O)C2)O)ccc(Cl)cc1 N1(C(c2c(C)cccn2)=O)CCCC2C1CCN2C(C1CN2CCN1C(C)C2)=O C1(CC)CCCCC1NC(=O)NCC(O)CNC(c1ccccc1)=O C1(C(N2CCC(CC)(CC)C2)=O)CN(C(c2cc(C#N)cs2)=O)C(C)(C)C1 c1(C(N2CCCC(NC(C(CC)CO)=O)C2C)=O)cnc(O)c2ccsc12 C1(C(N(C(C#CC(C)C)=O)C)=O)CCCC1P(C)(C)=O C(=O)(CC(COC)COC)N(C1CCN(C(=O)CC2CCOC2C)CC1)CC#C O=C1Cc2cc(C(N3CCC4(C3)CN(C(C3CC3(F)Cl)=O)C4)=O)ccc2CN1 C=C1CCC(C(=O)N(CCC(=O)N2CC(CCCCC)C2)C2CC2)CC1 c1(C(=O)NC2CCN(C(C=NOC)=O)C23CC3)cccc2c1ncn2C N1(C(C=Cc2c(C)ccnc2)=O)CCC(NC(c2ncn(C)n2)=O)CC(C)(C)C1 C(C1CN(C(c2cc(CO)c(C)o2)=O)Cc2ccccc21)NC(CCCC=C)=O C(=O)(CCCC(C)(C)C)NC1(CC)CCCN(C(c2c(C)cccc2F)=O)C1 C(=O)(C(C)C(F)(F)F)N(C1CCN(C(c2nc(CC)oc2)=O)CC1)CC C1(CNC(CC)=O)CN(C(C(C)CC(=O)NC2CCN(C)CC2)=O)C2CCCC2O1 c1(NC(CS(CC)=O)=O)ccc(NC(c2cnncc2O)=O)cc1C N1(C(C2(C)CCCCCC2)=O)c2ccccc2S(=O)(=O)c2ccccc21 N1(C(c2ccc(CC)cc2)=O)CC(NC(=O)CCn2cc(C)cn2)CC(C)C1 c1(OC)ccc(CC(C)C(N2CCC(O)(CNC(=O)C(C)=CC3CC3)C2)=O)cc1 N1(c2ccnc(COC)n2)CCC(C2CC2)(CNC(c2cnc(SC)s2)=O)C1 c1(C(=O)NC2(F)CC=CCC2)ccccc1Sc1ccccn1 c1(C(CC)(OCC)CC)nnc2n1C(C)CN(c1ccc(OC)c(OC)c1)C2 c1(OC)ncc(Cl)cc1C(C(=O)NC1CCCC1)N(C(C)C(C)C)C c12oc3ccccc3c1C2.c1(C(C)O)ccccc1C(N1CCCC1C(C)O)=O C(=O)(C1CNC(=O)c2ccnn21)NC(C)(C)Cc1ccc(Br)cc1 C1(CNC(C2C(C)(C(C)C)C2)=O)C2CN(C(=O)Cc3ccc(F)cn3)CC12 C1(CNC(c2c(C(C)C)nns2)=O)COCCN(C(c2nncn2C2CC2)=O)C1 C1(NC(=O)NCCOCCC2CCC2)CSC(CC2CC2)C1 c1(C(N2CC3(C(NC(=O)C(F)CC4CC4)CC3)C2)=O)ccc2c(c1)nc(O)n2CC C(=O)(C(C(C)O)N(C)C)N1C(C(=O)NCc2nc(C)[nH]n2)CCC1 C1(CC)CN(C(c2cc(C3CC3)n(C)n2)=O)CCC1NC(=O)CC1(C(F)(F)F)CC1 Cc1cc(Br)c(C(=O)NCC2CN(C(=O)Cc3cccnc3C)C3CC23)s1 C1(CCOC)CC(N=c2cc(NCCc3ccccc3C)nc(C(C)C)[nH]2)C1 Cc1ccn2c(C(N3CCC4CCN(C(=O)C=CC=C(Cl)Cl)CC34)=O)cnc2c1 c1(C(=O)NCCC2CN(C(C3(C(C)C)CC3)=O)CC2C)nc2cc(O)ccc2[nH]1 c1(OC)cc(NC2CC(NC(=O)Cn3nc(O)ccc3=O)C23CCC3)nc(OC)n1 C12(NC(C3CCCC3)=O)CC(CNC(c3cnc(C4CCCO4)s3)=O)(C1)C2 c1(C(=O)NCC2(O)CC(NC(CCNC(=O)NC)=O)C2)c(Cl)c([N+](=O)[O-])nn1C c1(NC(C2(C)N(C(CC3N(C)CCC3)=O)CCC2)=O)cccc2cncn12 CCC(C(=O)N1CC(F)(CNC(=O)CCSc2ccc(F)cc2)C1)C(C)C Cc1cc(C)c([N+](=O)[O-])c(C)c1C(=O)NCCCNC(=O)CCCc1cncs1 N1(C(C(C=C)(C)C)=O)CCC2C(NC(c3ccccc3OCC)=O)C2C1 N1(C(C(CCC)NC(C)=O)=O)CCC(NC(=O)C(C)=C(C)CC)C(C)C1 C(C(O)CN=c1ccn2nccc2[nH]1)NC(c1cc(CC)no1)=O n1(CC)ncc2cc(C(=O)NC3CC3NC(=O)CC(=O)NCC3CC3)c(C)nc12 c1(CCC(=O)NCC2COCCN2C(=O)CCOCC(F)F)ccc(F)cc1F C(=O)(Nn1cnn(C)c1=S)C1(C)CCN(C(C(C=C=C)C)=O)C1 c1(C(N(C2CCN(C(=O)C(C)(C)c3cncs3)C2)C)=O)cc2n(c1)CCC2 C(C)(C(C(C)C)NC(=O)CCc1cccc(O)c1)NC(CCOCCC)=O N1(C(c2c(CC)nc(C)[nH]2)=O)CC(NC(C2CCC3CC2CO3)=O)C(C2CC2)C1 C12C(NC(=O)C(C3CC3)OCC)CCCN1C2=O.C1(CC)CCCCCC1 N1(C(C2CC2c2cccnc2Br)=O)CCC(=C(F)F)CC1 c1(C(=O)NC(C2CCN(C(Cc3c(CC)cccc3)=O)C2)C)cc(C)ncc1C N1(C(CCc2ccc(C)cc2)=O)CC2CC1CCC2NC(C1CC2C=CC1C2)=O CC(C)C(C)(O)C(=O)N1CC(CC(F)C(=O)NC2CN(C)CCC2O)C1 c1(C(N(C2(CCO)COC2)C)=O)sc(F)cc1Br N1(C(C=C(C)c2ccco2)=O)CCC2CC2(NC(=O)Cc2ccc(Cl)s2)CC1 c1(CNC(C2CC(C)(NC(=O)CCc3cccc(Cl)c3)C2)=O)ccc(F)nc1F C1(C(=O)OC)C2CCCC2CN1Cc1coc(C#N)c1 C(C(CO)(CO)NC(=O)CC1CCCOCC1)N(C(COC1(C)CCC1)=O)C CCC(CNCCCN(C(C)(C)C(F)(F)F)C)C(=O)NC(C)(C)C N1(C(c2c(C)nsc2N)=O)CCC(O)(C(C)NC(C2C(C)C2C)=O)CC1 n1(CC(N)=O)cc(NC(C2CCN2C(=O)CC2CC2)=O)cn1 CN1CCC(CC(N2CCC(C)(NC(c3cn(CC(N)=O)nn3)=O)C2)=O)C1=O c1(SC)ccccc1C(=O)N(CCC(C)NC(c1cccc(C)c1)=O)C C1(C(=O)NCC2CCCC(CNC(C(C(C)C)O)=O)C2)CN2CCCC2CO1 C(=O)(CC(O)CC(C)(C)C)NCC1(F)CCN(C(C(CCC#C)O)=O)CC1 CC1CN(C(C2CC(C)(NC(=O)C#CC(=O)N(C)C)C2)=O)CC1CO c1(C(=O)NCC(CNC(C(c2cccnc2)C)=O)C)ccc2c(c1)N(C)CCO2 C1(CC)(CNC(=O)C(C)CN(C(=O)CCOCC(C)C)C)CCC(=O)N1 C1(C#N)(C(=O)OC(C2CCC(F)(F)CC2)C(=O)N(CC)CC)CC12CCC2 N1(C(CCCN(C)C(C2CCCN2C2CC2)=O)=O)CCN(CC(N)=O)CC1 C1(NC(c2cc(OCC)ns2)=O)COCCC1C(=O)NOC1CCCC1(F)F c1(C(=O)OCc2ccc(C#C)cc2F)ccc(Br)c(S(N)(=O)=O)c1 N1(C(C(CN(C(C2C(=C)C2)=O)C)(C)C)=O)CC2CC(C)C2C1 N1(CC(=C2CN(C(=O)CSC)C2)F)CC(C)(OC(C2(C#C)CC2)=O)C1 c12cccc3c1CN(C3)c1nccc(n1)O2.C(CCNC1CC1)OC c1(C(N2CCN(C(C(CCC)C#N)=O)C(CCC)C2)=O)nsc2ccccc12 C(C(CC(C)C)C(=O)NCC(C(C)(C)C)NC(C1CC(=O)C12CCC2)=O)OC c1(C(N2CCC(C(=O)NCc3cc(C)cc(F)c3)C2)=O)cc(F)c(Cl)cc1C C1(C(=O)N(CCNC(C2CC2c2cscn2)=O)CC)(OCC)CCOC1 C=CCCC(C(=O)Nc1cc(C)cnc1OC)NC(C1CC2CCC(C1)O2)=O c1(C(=O)NCCCCC(C)NC(=O)CC2CC=CCC2)nnc2ccccc2n1 C=CC(C)(CC)CC(=O)NCCC(C(=O)N(CC(C)O)CC)OC N1(C(C(CC)n2cncn2)=O)CCCN(C(c2cc(C)c(C)nc2C)=O)C(C)C1 c1(C(N2CC(c3cn(C(=O)OC)nn3)C2)=O)cc(Br)cc2scnc12 C1(CC)C(=O)N(C)CCN1CC(=O)N(C1CCOC1C)CCO C1(C(=O)NC(CC)CSC)(C(C)C)CCN(C(=O)C=Cc2ccoc2)C1 c1(-c2ccc(C(=O)NC(c3cccnc3)CC)nn2)ccc2c(c1)CCN2 CC1(C)CCC(C(N2CC(CC(F)C(=O)NCCSc3ccoc3)C2)=O)CO1 N1(C(CC(CC)CC)=O)Cc2n[nH]cc2C1C(=O)NCCC1(C)CCCC1 CCC(C)C(O)C(C)C(=O)N1CCCC1CCC(=O)NC1(C)CSC1 c1(CNC(c2csc(C#N)c2)(C)C)ccc2c(c1)CCCO2 c1(-c2cn(C3CCN(C(=O)NCCC=C)C3)nn2)cc(C)cc(Br)c1 Nc1ccc2nccnc2c1C(=O)NCC1CCN(C(C2(O)CCSC2)=O)CC1 C1(CCN(C)Cc2c(OC)cc(Br)cc2)CN(C(=O)OC(C)(C)C)CC(C)(O)C1 C(=O)(C(CC)CC=CC)NC1(CC=C)CCN(C(c2occc2C)=O)C1 c1(C(=O)NCC2(CN(C(c3n(CC)ccc3)=O)C)CC2)cnn(C)c1C(F)F C(=O)(CC(O)(C(F)(F)F)C1CC1)NCC(C(C)C)NC(CN(CCC)C)=O c1(C(=O)NC23CC(NC(c4c(CC)con4)=O)(C2)C3)cc(Br)ccc1C C(=O)(CCCCCC#N)N1CC(C)OC(CCNC(=O)C(=O)NC2CC2)C1 Cc1ccc(C(=O)NCC2CC(F)CN2C(=O)CC(C)(O)C2CC2)cc1[N+](=O)[O-] CC1=C(C)CC(C)(NC(=O)C(CO)NC(=O)CCc2ccccn2)CC1 Cc1[nH]c2ncnc(NCc3nncn3-c3ccccc3)c2c1C C=C1CCN(C(c2c[nH]nc2OC)=O)C(C(=O)NCC(C)C(F)F)C1 C(CN=c1[nH]ccc(=NCCCc2cccnc2)[nH]1)C1(CC(N)=O)CC1 C1(NC(C2N(C(C)=O)CCC2)=O)CCN(C(c2ccn(C(C)C)n2)=O)C(C)C1 C(=O)(CCCCCS(N)(=O)=O)N1C2CN(C(c3c(C)nc[nH]3)=O)C(C2)CC1 C(C(=O)NCC)(C(C)C)NC(=O)CC(=O)OCC.C(=O)(C(CO)N(C)C)N1CC(O)C1 CCCS(=O)(=O)CC(=O)NC(C)(C)CNC(=O)CN1CCC(C)C1 C1(NC(CC(=O)NC)=O)CCCN(C(C2CC(OCc3ccccc3)C2)=O)C1 c1(NC(=O)Nc2nc(COC)nc(N3CCCCCC3)c2)cc(C#N)ccc1Br N1(C(C2N(C)CSC2)=O)CCN(C(c2ccc([N+](=O)[O-])s2)=O)CC1CCO N1(C(c2cc(C(C)C)no2)=O)CCN(C(=O)CCC2CCCOC2)CC1CCO N1(C(c2c(COC)cco2)=O)CCC(NC(C2(C)COC2)=O)C(C)C1 N1(C(CCn2c(C)ccc2C)=O)C2CCC1CN(C(c1cnn(C)c1Cl)=O)CC2 N1(C(CCn2ncc(C)c2)=O)CC2(C1)CN(C(=O)CC(C)C(C)(C)C)CCO2 C1(CCC=C)(C(=O)NCC(O)CCOC)CN(C(=O)C(c2ccccc2)F)C1 n1(CC(=O)NCC2CN(C(C3C(C)COCC3)=O)C2)cnc2ccccc2c1=O c1(C(N(C)CC2(C)CCN(C(C)=O)C2)=O)ccc(F)cc1Cl C1(C(=O)NC2C=CCN(C(C3CCOC3)=O)C2)CC2CCCCC12 c1(NC(C(C)N(C)C)=O)ncc([N+](=O)[O-])cc1I.c12cnc(Cl)cc1CN2 c1(C(N2CCC(O)(CNC(=O)C3=CCCCC3)C2)=O)cc(Cl)cc2ccccc12 C1(n2cc(CCCC)nn2)CN(C(C2(C#N)CCCO2)=O)CC1O CCCC(C(=O)NC1CCC(NC(=O)C(C)NC(=O)CC2C=CCC2)CC1)OC CC1(CCNC(c2cc(C3CCC3)[nH]n2)=O)CCN(C(C2CCO2)=O)C1 c1(CC(C(N2CCC(N(c3snc(C(C)C)n3)CCO)C2)=O)C)ccc(F)cc1 N1(C(CC(=O)N(C)C)=O)CC2CC2(NC(c2cnn(C3CCCC3)c2)=O)C1 c1(C(N2CCN(C(CCC(C)OC)=O)C(CF)C2)=O)ccc(Cl)c(C)c1Cl c1(C(=O)NCC(CNC(C2CCC(C)(C)OC2)=O)(C)O)cc2cccnc2[nH]1 C(CNC(=O)COCCCOC)(C(C)C(C)C)Nc1ccc(C(CC)=O)cc1 C1(C(C)C)C(NC(=O)COC(F)(F)F)CCN1C(C1CC(C)N(C)C1)=O c1(C(=O)NC2CCC(CNC(C3(SC)CC3)=O)C2)cc2cc[nH]c(=O)c2s1 N1(C(c2c(C(C)C)[nH]cc2)=O)CCC(NC(=O)CC2CC=CCN2C)C(C)C1 c1(NC(C(CC)OC)=O)ccc2c(C(=O)Nc3cnsc3)ncn2c1 C(=O)(C#CC1(C)CC1)NC(CNC(CC(C)SC)=O)C1CCC1 c1(C(C(=O)NC)N(C)CCC2CC(SC)C2)ccc(Br)cn1 c1(C(N(C)CC2(NC(=O)CC3CCCOC3)CC2)=O)nccc(-n2ccnc2)n1 N1(C(c2n(C)c(-c3ccccc3)cc2)=O)CC2CC(NC(C3(C)CC3)=O)CC1C2 N1(C(c2cc(C)nn2C)=O)CCN(C(c2cc(CO)oc2C)=O)C(CO)C1 N1(C(C2(C)CC(C)C2)=O)CCN(C(=O)Cc2ccc(C(N)=O)cc2Cl)C(C)C1 C1(C)(C(=O)NCCN(C(c2cnc(C3CCCCC3)s2)=O)CC)CC(C(C)C)=NO1 N1(C(C(CC(=O)OC)C)=O)C(C)CC2CN(C(C3CC4CCC3C4)=O)CC12 N1(Cc2ccc(CC)cc2O)CCC2(CC1)CC2C(=O)NC(c1cc[nH]n1)CC C(CN=c1[nH]c(N2CCOCC(C)(F)C2)nc2c1CSC2)c1c(C)cccc1 CC1(C)C2CN(Cc3c(F)cc(F)cc3F)C(C(=O)Nc3cnncc3Br)C12 C1(CNC(C23N(C(C4(C(=O)OC)CC4)=O)CC(C2)C3)=O)CCCC(C)CC1 CC(C)(C)C(C)(C)C(=O)N1CCC(NC(c2cccc(I)c2)=O)C(F)C1 C1(CC(N2C(C(C)(C)C)COCC2)=O)C2CCCC2N1C(=O)CC(Cl)Cl c1(C(C(=O)NCCOC2CN(C(CCSCC(C)C)=O)C2)C)cccc(Cl)c1 CC(C)(CC(=O)N1CCN(C(=O)C=C2CCC2)CC12CCC2)C(F)(F)F c1(CNC(C(C)NC(=O)Nc2c(CC)con2)=O)cccnc1O Cc1cc(C#N)sc1C(N1CCC(N(C)C(C2CCC(C)(C)OC2)=O)C1)=O N1(C(Cc2n(C)ncc2)=O)CCOCC1CC(N1CCOC(CN=[N+]=[N-])C1)=O Cc1cccc(C(N2CCCC2CCCNC(c2cnc(N(C)C)nc2)=O)=O)n1 CCC(C)CCC(=O)NCC(CNC(c1ccnn1CC(C)C)=O)C(F)(F)F C(=O)(C1CCCn2ccnc21)N1C(CNC(CC(CCC)C)=O)CCC1 c1(SC)cnn(C)c1C(=O)NCC1CC(C)N(C(=O)C(C)N2CCC2)C1 N1(C(C(CC)n2cncn2)=O)CCC(CCC(N2C(C)CC2(C)C)=O)CC1 c1(C(=O)NC2CCN(C(C3(c4ccn(C)n4)CC3)=O)CC2)occ2c1CCOC2 CCC(C(C)(F)F)NC(=O)CC1CCCC1NC(c1cc(OC)nn1C)=O N1(C(=O)CC2CCOC2)CCC(CO)C(NC(c2ccnc(CO)c2)=O)C1 N#Cc1cc(=NCC2CCCCN2C(c2cccc(F)c2)=O)[nH]cn1 c1(C(=O)NC2(C(=O)Nc3c(O)ccc(C(N)=O)c3)CCC2)n[nH]c2cccc(F)c12 C=CC1(CC(=O)NC2CCN(C(c3nc(C)c(C)[nH]3)=O)C2(C)C)CCCCC1 C=C=C(C)CC(=O)NC(C)CN(C(=O)CCCc1ccc(Cl)cc1)C Cc1cc(S(F)(F)(F)(F)F)ccc1NC(C1CCCN1NC(=O)C1(C)CC1)=O C=CCCCCCC(=O)NCC1(F)CC2CCC(C1)N2C(=O)Cc1ccco1 c1(C(N2CC(=C)C2)=O)ccc(N(C(c2n[nH]c(C)c2C)=O)C(C)C)cc1O c1(C(N2CCCCC(NC(C3N(C)CCOC3)=O)C2)=O)ccc2ccsc2c1 c1(CC)cnoc1C(=O)NC(c1cccnc1)C(=O)NC1COC(=O)C1 c1(CC(=O)NC(CNC(C2(OCC)CCCC2)=O)C2CC2)cnccc1Cl C12(CNC(C3=NOC(C)C3)=O)CCCC1N(C(=O)CC1(C)CC1)CCC2 c1(CC(=O)NCC(CN(C(c2n(CCOC)ncc2)=O)C)O)noc(C)c1C#N c1(C(=O)NCC(C2CCCC(C)C2)(C)O)ccc(OC(F)F)c(F)c1 C1(NC(c2ccc([N+](=O)[O-])s2)=O)CN(C(=O)CC(F)F)C2(CCOC2)C1 C1(C(C(=O)N(CC(C)C)C2CC2)C)CCCN(C(=O)C(C)(C)CF)C1 Brc1cn2c(C(c3nnnn3C3CCOCC3)NCc3cnns3)cnc2s1 c12ccc(cc1)C(=O)NCCN(C(=O)C(O)c1ccsc1)CCO2.CCCCOC N1(c2[nH]c(=NCCc3c(C)cccn3)[nH]c(=N)n2)CC(C)(C)C12CCOCC2 C#Cc1ccc(C(=O)NC(C2CCN(c3nccc(OCCC)n3)C2)C)nc1 N1(C(CCc2n(C)c(S)nn2)=O)CC2CCCCC2(CNC(=O)C(N)=O)C1 C1(NC(CCC=CC)=O)CN(C(=O)C=C(CCC)CCC)C2(CCOCC2)C1 C1(C(C)C(=O)NC2CCN(C(=O)CCC=C(C)C)C2C)CCC2(CC1)OCCO2 c1(CNC2CCC(C(=O)Nc3n(CCC)ncc3)OC2)cc(C)c(F)c(F)c1 c1(CC(N2CCCC(CNC(C(C)=C(C)C)=O)C2)=O)ccc2cnccc2c1 N1(C(c2c(C)oc(Br)c2)=O)CC2CC(NC(c3ncncc3Cl)=O)CC2C1 C=C(CC1CCCC1)C(=O)N1CCC(C(C)OC)C1 c1(C(=O)NC2C(C)CN(C(=O)COCCc3ccc(Cl)s3)C2)cccn(C)c1=O c1(C(N(C2CN(C(CNC(C(CC)C)=O)=O)C2)C)=O)cnc2c(c1)NC(=O)CS2 C(=O)(C1CC(C)Nc2ccccc21)NCC(C)NC(c1c(C(C)=O)cccc1)=O Cc1cc(=NC(=O)C(=O)N2CC(NC(C3COCCN3C)=O)CC2C)[nH]o1 C(=O)(CC(C)C(C)C)NC(CN(C(c1c(C(=O)OC)nccn1)=O)C)C C1(CC(=O)OCC)COCCN1C(c1ccc(COc2ccc(O)cc2)cc1)=O N1(C(CC(=O)NCC)=O)CCC(NC(c2ccoc2C)=O)C(O)C1 Cc1ccc(CC(N2C(C(=O)NCCC3CCCC4CC34)CC3CC23)=O)cc1O C(C(C)(C(=O)NC1CC12CC(OC)C2)NC(=O)Cc1cncc(C)c1)SC CC1CN(C(=O)NCCCC2CCOC2=O)c2ccc(Br)cc2O1 CCCCC(C(=O)NC1C=C(C)CCC1)NC(c1ccc(=N)[nH]c1)=O c1(OC)ccc(C(=O)N(CCCNC(C2CC23CC3)=O)CCO)cc1C(C)C c1(C(N(CCN(C(=O)C2=CC(C)(C)C2)C)C)=O)cc2sccc2n1C c1(OC)cc(C(=O)NC(C)C(C)NC(c2ccc(=N)[nH]c2Cl)=O)ccc1Cl c1(C(N(CC(O)CN(C)C(c2c(C(F)F)cccc2N)=O)C)=O)c(O)cccc1O Cc1ccc(S(N)(=O)=O)cc1NC(=O)C(C1CCC(C)(C)CC1)N C(C(CNC1CC1)C(F)(F)C(F)(F)F)OC(c1c(C)c(=O)cc[nH]1)=O C(=O)(C1CN(CCC2CCC2)Cc2n[nH]cc21)OC O=S(=O)(c1ccc(NC2CCN(CCF)C2)c(F)c1)N1CCCC(F)(F)CC1 C1(NC(Cc2nnn(C(C)(C)C)n2)=O)(CO)CCCN(c2nnco2)C1 CC(C)CC(C)(CO)CC(=O)OCN.C1(C(=O)OC(C)(C)C)CN(C(N)=O)C(C)(C)C1 c1(OC)cc(C(N2CC(OC)CC(NC(c3c(C)n[nH]c3C)=O)C2)=O)cc(Cl)n1 Cc1ccc(C(=O)NC2(C(=O)NCCN3CCN(C)C(C)C3)CCSC2)nc1C C(CCCCC(=O)N(C)CC1CCCN1C(C1CC2CC1CO2)=O)SC c1(C2C(C(N(CCNC(CCCC#C)=O)CCC)=O)C2)ccc2ccccc2c1 N1(C(CCOC)=O)CCC(C)(C)C(NC(=O)CC(C)c2ccncc2)C1 C1(CNC(c2c(Cl)cnc(C)n2)=O)CC2(CO1)CN(C(=O)Cc1ccnn1C)C2 C1(CC(=O)NC(c2cn(Cc3ccc(Cl)cc3)nn2)CCC)CC2C=CC1C2 C(CC(C)CCNC(c1c(C(=O)Oc2ccccc2)c[nH]c1)=O)NC(C(C)C)=O Cc1cc(CNC(C2SCCS2)=O)oc1C(=O)N(CC(C)C)CCO C(=O)(CCCCCOC(C)(C)C)N(C1CCN(C(=O)C=CCOC)CC1)CC#C N1(C(C2N(C(C)C)CCCC2)=O)CC(NC(c2ccncc2Cl)=O)C(C2CC2)C1 N1(C(COC2(C)CCC2)=O)CCCC(CC(N2CC(CN=[N+]=[N-])C2)=O)C1 c1(CCC(=O)NC(CCNC(C(CCSC)OC)=O)(C)C)ccc(F)cc1Cl c1(OC)cc(CCNC(C2CC2c2ccc(C(F)(F)F)cc2)=O)ccc1C c1(C(=O)NCC2(C)CCN(C(CCC#C)=O)C2)cc(S(N)(=O)=O)c(C)cc1C Cc1cc(C(=O)NCC2CC3(C2)CN(C(C2CC(C)CO2)=O)C3)cc(N)c1 N1(C(CSC)=O)CCCC2(CNC(C3CCC(C(N)=O)CC3)=O)CCCC12 C(C(=O)N=c1ccc2cc(Br)ccc2[nH]1)OCCCCSC N1(C(=O)NCCc2cccc(Br)c2F)CCC2CS(=O)(=O)CC2C1 C(=O)(C1=CCCN(C(C2C3CCC(F)C23)=O)C1)N(CC(C)C#N)C c1(OC)nc(C(=O)NC(C)CNC(c2cn(C3CCOC3)cn2)=O)ncc1F CCC(CC(=O)NC1CON(CC)C1=O)NC(=O)Cc1ccccc1 C(=O)(C(C)(C)CC(C)(C)C)N1CC(CC)(NC(c2cncc(-n3ccnc3)n2)=O)C1 c1(NC(c2c(C)nc(-n3cncn3)cc2)=O)ccc2cnn(C(F)F)c2c1 c1(C(C)NC(=O)C2=COCC2)ccnc(F)c1.N12CCCC1(C)C2=O c1(CC(=O)N(C2CCCN(C(C(C)OCCC#C)=O)C2)C)ncc(F)cc1F c1(C(=O)NC2C(C)N(c3ccc4nnnn4n3)CCC2)cccc2cncn12 N1(c2nc(C(C)C)nc(N3CCC(c4ccco4)CC3)c2)CC2CC(O)CC1C2 C1(C(N2CCCC(c3ccccn3)C2)=O)CCn2cnnc2C1 C12(OCC)CCC(C(N3CCCC(CN(C)C(c4nnsc4C)=O)C3)=O)(CC1)C2 N1(C(c2c(OC)cncc2)=O)CCC2CCCC12C(=O)N(C)Cc1nnc(C)s1 C(N=c1[nH]c(N(C)CC2CCCC2O)nc2c1SCC2)c1c(C)cn(C)n1 CCCCCC(O)C(=O)N1CCN(C(c2ccn(CC)n2)=O)CC1C1CC1 c1(C(N2CCC(OC)(CNC(C3CCCC3O)=O)C2)=O)cc(F)ccc1F c1(C(=O)NCCCCCN(C(=O)C(F)C2CCOC2)C)nccc2ncccc12 C1(CNC(c2c(C)cncc2C)=O)CC2CCC1N2C(=O)CC1NC(=O)NC1=O C1(CC(=O)N(CCOCCNC(c2cc(NC)no2)=O)C)CCC(=O)NC1=O C1(C(=O)NC2CC(NCc3c(N(C)C)nccc3)C2)C2CC3CC(C2)CC1C3 c1(C(N2CC(N(C(c3c(C)coc3)=O)C)C(O)C2)=O)cncc2cc(Cl)ccc12 c1(C(=O)NCC(Cn2cc(C(C)NC)nn2)(F)F)cc2sc(C)cc2s1 c1(CNC2CC(O)C2)nc(Cl)cs1.C1(C(C(=O)C)=O)CCCO1 C1(NC(=O)C=CC(F)(F)F)CCC(F)(CNC(=O)C=CCN2CCCCC2=O)C1 C=CC(C)(CC)NC1(c2nnnn2CCC2(C)CC2)CCOC1 C(c1ccccc1)(C(F)(F)F)=CC(=O)NCC1CC(NC(C2CC2(F)Cl)=O)C1 C1(C(=O)NC(COCC)C)CC(NC(c2cc(NC)ncn2)=O)C(O)C1 C#CCCCCC(=O)N1CCC(C(C)C(=O)NC2CC3CCC2C3)CC1 CC1CCN(C(c2cnc(Cl)n2C)=O)C1C(=O)N(CC(O)CO)C N1(C(=O)CCc2ccncc2)CC(F)CC1CNC(C12CCCCC1C2)=O C1(CC(=O)N(CCN(C(=O)CCCOc2ccccc2)C(C)C)C)C=CCCC1 CC1=CCN(c2cccc(NC(C3(C)CN(S(C)(=O)=O)C3)=O)c2)CC1 C1(O)(CNC(CCN(CC#C)C(C2C[SH](C(C)C)C2)=O)=O)CCCC1 Cc1cc(NC(=O)NC2CCC(c3ccccc3)C2)n(C2CCOCC2)n1 N1(C(=O)CN2CCOCC2)CC2CCC1CN2C(c1cc(Cl)ncc1Cl)=O C(=O)(CCCC(=O)NC1CCOC1C(=O)NCc1ncc[nH]1)N(C)C Cc1ncccc1C(N1CCC(C)C1C(=O)NC(CCO)C(C)C)=O c1(-c2nc(-c3ccc(CC)nc3)on2)ccc(C(C)(C)C)c(C)c1 c1(C(CC)(C)C)ccc(C(N2CCN(C(C3C4(CC4)C34CC4)=O)CC2)=O)cc1 N1C2CCC1CC(n1cc(-c3sc(C)cc3Cl)nn1)C2.C1(NC)CCCC1 c12cccc(c1)OO2.c1(N(C(CCn2c(C(C)C)ncc2)=O)CCO)ccccc1F C(=O)(CCC(CF)CF)N1CCC(C(C(N2CCC(CC(=O)NC)C2)=O)C)CC1 N1(C(CCC=CC(C)C)=O)CCC2(CC1)CN(C(c1cc3c([nH]1)CCOC3)=O)C2 S(=O)(=O)(c1ccc(OC)c([N+](=O)[O-])c1)N(C(Cc1ccc(F)cc1)C(C)C)CC c1(C(N(CCN(C(C(COCC)(C)C)=O)C(C)C)C)=O)cnc2cc[nH]c2c1 C(c1ccc(C)nc1)=CC(=O)NC(CC=C)CNC(c1ccc(C2CC2)nc1)=O c1(N2C3C(NC(C=CCCC)=O)(CCC3)CCC2)c(F)cc(C#N)cc1[N+](=O)[O-] Cc1cc(C#N)ccc1C(=O)NCCC(C)NC(c1cnc(O)c(C)c1)=O C1(NC(C(c2cccc(C)c2)O)=O)CC2CC1N(C(c1[nH]nnc1C)=O)C2 Cc1cc(Cl)cc(N)c1C(N1CC(NC(=O)CSC(F)F)CC(F)(F)C1)=O c1(NCC2(F)CCN(C(C(C)=CC)=O)CC2)cc(C)c([N+](=O)[O-])cn1 C(=O)(C1c2ccccc2C2CC1C2)N(CC(C)O)CCNC(Cc1c(C)non1)=O n1(CC)nc(C)cc1C(=O)NC1(CC(=O)NC2CCCC2(C)CO)CCC1 c1(OC)cc(C(N2CCC(NC(=O)C(F)OC(F)(F)F)C2C)=O)c(F)cc1N C=CCCCCCCCC(=O)NCC(CC=C)NC(=O)CC12CC(C1)C2 c1(C(N2CC(CC#C)OCC2)C(=O)NCCC)ccc(N2CCCC2)c(Br)c1 N1(Cc2c(OC)ccc(Br)n2)CCOC2(CCCN(C(c3nccs3)=O)C2)C1 CCC(C)(CO)C(=O)NCC(C)CN(C)C(c1cnc(=N)[nH]c1)=O c1(C(N2CC=C(CNC(c3c(C)nncc3)=O)CC2)=O)cccc2cc[nH]c12 C1(C(=O)NCc2cc(C)c(F)cc2)CCN(C(=O)C(O)CCC(C)C)C(C)(C)C1 C1(CC)CN(C(c2cncn(C)c2=O)=O)CCN1C(c1cnc(C(F)F)s1)=O C#Cc1c(C(=O)OC2(C(F)(F)F)CC(OC)C2)cc(COC)cc1C(F)(F)F.C(C)O N1(C(C(C)OCCOC)=O)C2CC1CN(C(c1ccc(O)cc1OC)=O)C2 c1(CC)ccc(C=CC(=O)NCC2(NC(=O)C(C3CCCCC3)OC)CC2)cc1 Cc1cc(=NC(=O)C(=O)NCCCCC(C)NC(=O)C(C)(C)c2cnco2)[nH]o1 CCCC(CCC)C(=O)NCC1CCC1NC(c1cc(OC)c(F)c(F)c1)=O c1(NC(c2cnn(C3CC3)c2-c2ccccc2)=O)cc2cccc(O)c2[nH]1 C(C(CC(F)(F)F)NC(c1cncc(N)c1C)=O)NC(C(CC)C)=O CCCCCCC(=O)N1CCCCC(N(C)C(c2cnc(OCC)cn2)=O)C1 N1(C(c2c(C)nco2)=O)CCN(C(C2CCC(=O)N2C)=O)C(CC(F)(F)F)C1 c1(OC2CCN(C(=O)NCc3cnc(COC)s3)C2)ccc2c(c1)OCO2 C1(C(N2C(C(=O)NCc3cccc(CC)c3)CC2)=O)CC2C(C1)C2(F)F CC1CCC(NC(=O)Cc2ccc(Cl)c(Cl)c2)CN1C(c1cc(O)ccc1N)=O C(=O)(CS(=O)(=O)C(C)C)N1CC(CC)C(NC(=O)C=Cc2ccccn2)C1 C1(C)(CCNC(C(COC)N(C)C)=O)CCN(C(c2c[nH]nc2F)=O)C1 C(=O)(C1CCc2nccn21)NC(c1ccc(C)cc1)CNC(C1(C)CC(C)(C)C1)=O c1(CNC(C2C(C)C2)=O)n[nH]c2c1CN(C(C1(C)COC(C)(C)OC1)=O)CC2 C1(CC=C)(NC(c2cn(CCCC)nn2)=O)CCN(C(=O)C(COC)OC)CC1 C(=O)(C1=CC(O)C(NC(=O)C(C2(O)CCCC2)F)C1)NCc1cc(C)on1 c1(SC)ccc(Cl)c(C(N2CCC(CNC(=O)C(CO)NC(=O)C(C)C)C2)=O)c1 N1(C(CCN(C(c2cc[nH]n2)=O)CC)=O)CC2CC1C2N(C)C Cc1cccc(C)c1C(N1CC(CN(C(=O)Cc2c[nH]nc2C)C)C2(CC2)C1)=O c1(C(N2C(C)COCC2)=O)ccc2c(c1)C1(CCCC1)CN2C(c1nccs1)=O C1(NC(c2c(OCC)cccc2)=O)CN(C(=O)C=C(CC)CC)CCC1CO C1(C(=O)NCC2(CNC(=O)CCc3ccc[nH]3)CC2(F)F)CC(=O)NC(=O)N1 CN1CCC(N=c2cnc(CO)c[nH]2)(C(F)(F)F)C1 C(=O)(CC(CNC(=O)CC(C)OC)OC)NC(CCOCC)(C)C N1(C(=O)NCc2nccc(OC)c2)CC2CCCCN2CC1C c1(OC(C)C)cnc(C(=O)NC(C)CC2CN(C(=O)C=Cc3cnc[nH]3)C2)cn1 C(=O)(C1=COCCO1)N1CC(CNC(c2c(C)nc(CCCC)s2)=O)C(O)C1 Cc1n[nH]c(C)c1CC(N1CC(NC(c2cc(Br)ccn2)=O)C(O)C1)=O O(NC(=O)C(Cc1cnn(C)c1C)OC(C)=O)C(COCC)C c1(OC)cc(Cl)c(Cl)cc1C(=O)NC(CNC(C1CCCCO1)=O)C1CC1 N1(CC(N2CCn3c(Br)nnc3C2)=O)CCCC2(CCNC2=O)C1 c1(C(N2CC(N(C(CSCCC)=O)C)C3(C2)CC3)=O)cc2cccc(C)c2o1 N1(C(C2C(C)C2)=O)CC2(CC(NC(c3cc(-c4cn(C)nn4)on3)=O)CO2)C1 c1(C(N(C)CCNC(=O)C=Cc2ccccn2)=O)ccc(Cl)c2c1OCCO2 c1(C(=O)NC2CCN(C(Cc3c(C)n[nH]c3)=O)CC2C)cc2c(nn1)CCC2 CCCC(C)CC(=O)N1CC2(CC2)CC1CNC(=O)CCn1ccnc1 c1(C(N(C(C)(C)C)CCN)=O)cc(C(=O)O)cc2cc[nH]c12 N1(C(C2(C(C)C)CC2)=O)CCCC(N(C)C(c2cnn(C)c2Br)=O)C1 C1(CNC(CCNS(CC)(=O)=O)=O)CN(C(c2cc3[nH]ccc3s2)=O)CC1(C)C c1(C(=O)NCC(C2CCCC2)NC(c2coc(Br)c2)=O)ccc(F)cc1F N1(C(CCCOCC)=O)CCC2(C1)CN(C(c1nccc3occc13)=O)C2 C1(CNC(c2c(C)cc(F)s2)=O)CC(NC(c2ccnnc2)=O)C12CCC2 c1(N2C(=O)CC(C(=O)NC(c3cnn[nH]3)CC)C2)ccc(OC)cc1C CC1(C)C2CCC1(C(=O)NC1CCCCC1NC(C1CC=CCO1)=O)CC2 N1(C(c2ccc(C)c(C)n2)=O)CCC2CCC(NC(=O)C(C)C3CCCO3)C1C2 Cc1nc2ccnn2c(C)c1C(=O)NC1CC(NC(=O)CC(C(C)C)C(C)C)C1 C1(c2nnnn2Cc2ccc(F)c(F)c2)(Nc2cc(C)sc2)CCCN(C)C1 C1(NC(c2c(C)nc(C(C)C)s2)=O)CC(F)CN(C(=O)CCN2CCCC2=O)C1 C(CCCCC(=O)N1CC(O)(CNC(c2cnc(C3CC3)o2)=O)C1)OCC c1(C(=O)NCCCN(C(=O)CCc2cccc(Cl)c2)CC)cc(C)cnc1F N1(C(C(CC)N(CC)CC)=O)CCC(O)(C(C)NC(C23CSC(C2)C3)=O)CC1 C1(CC(=O)N(CCOCCNC(Cc2cn(CCC)nn2)=O)C)CCCC(=O)C1 C1(C(=O)NC(C(=O)OC)C(C)C)CC(C)CN(C(=O)CC2COCC(C)O2)C1 c1(C(c2nnnn2C(C)C(=O)OC)NCCNC(C=C)=O)ccc2c(n1)OCCO2 C12(NC(c3[nH]cc(CC)n3)=O)CCCC1N(C(=O)C(c1ccc(Cl)cc1)O)CC2 N1(C(CCC)=O)CCCC(N(C(=O)CC2(C[SH2]CC)CC2)C(=O)C2CC2)C1 C1(NC(C2C(OC)CCC2)=O)C2CCCC1N(C(=O)CC(C)(C)NC(C)=O)C2 C1(C(=O)NC(CNC(c2coc(Cl)n2)=O)CO)CCCC2(CCCCC2)C1 CC1(C)CCC(C(=O)NC2CSC2)(NC(=O)Cc2cc(C(C)C)no2)C1 CC1Cc2c[nH]nc2C(C(=O)N2CC(C)(NC(c3cc4c(o3)CCCC4)=O)C2)C1 C1(C)(C(=O)NC2CC3(C(NC(c4ccnc(C(C)C)n4)=O)C3)C2)CCCNC1=O N1(C(C(COC)(C)C)=O)CCC2CN(C(=O)Cc3cn[nH]c3)CC2C1 c1(N2CCC(OC)C2)nnc(-c2ccc(C)s2)n1CC(N1CCOCC1)=O CC1(C)CN(C(=O)CCCCn2cc(C3(n4ccnn4)CC3)nn2)CCCO1 CCC(CC(=O)C(=O)C(F)C(CC)CC)C(F)F.N1CC(C)(N)C1 N1(C(C(C)=CC2CC2)=O)CCC2C(NC(c3ccc(OC(F)F)nc3)=O)CC12 C1(C(=O)OCC)CC(n2cc(C3(CC)CCC3)nn2)CN1C(=O)C(F)(F)N(C)C N1(C(c2cnc(CC)nc2O)=O)C2CCCC1CN(C(C1CCCOC1)=O)C2 c1(C(N2CCC(C(C)(C)NC(C(C)NC(CC)=O)=O)C2)=O)cc(O)nc(O)n1 c1(CC(=O)NC2CN(C(CC(OCC)OC)=O)CC(O)C2)n[nH]c2c1CCCC2 O(NC(=O)CCN(C(=O)CCc1ccco1)CCCO)CC(=C)C C1(C(=O)N(C)CC2CCN(C)CC2)(NC(c2c(C)csc2)=O)CCCC1C N1(C(C2CCC(C)O2)=O)CCCC2(C1)CN(C(=O)CN1CCOC1=O)C2 C1(C(=O)NCCCOCC)C(C2CC2)CCN1C(C)=O C=CC(C)(CCOC)C(=O)NCC(C1CC1)NC(C1(C2CCCO2)CC1)=O C1(NC(c2cc(C)nc(Cl)c2)=O)CCN(C(C2CCSCC2)=O)C12CCCC2 C#Cc1ccc(OC)c(C(N2CCC(C)C(NC(=O)Cn3ccc(C)n3)C2)=O)c1 CC(C)CCCCCC(=O)N1CCC1CC(=O)NCc1conc1C(C)C C#CCC(C(=O)OC)NC(C1CCN(C(C2CC(CC)C2)=O)C1)=O c1(OC2CN(C(c3c(C)cncc3)=O)CC2C)ccc(Br)cc1F C1(CC)CC(C(N2CCC(CN(C(=O)CSCC(F)(F)F)C)C2)=O)CCO1 c1(C(=O)NCCN(C(=O)C(c2ccccc2)C)CC)ncc(C)nc1OC N1(C(C(CC(C)C)C)=O)CC(C(=O)N(C2CCC2)C2CCC2)C2(CCC2)C1 N1(C(c2cnn(C)c2Cl)C(=O)NC)CC2(C(=O)OC)CCC1CC2 C1(NC(C(C)OCC#C)=O)CC2CC(NC(c3ccc(CC)cc3F)=O)CC12 C1(C(N2CCC(CC=C)(NC(=O)CNS(N)(=O)=O)C2)=O)COC(C)(C)CO1 c1(CC)ccc(C(N2C3CCC2CN(C(=O)CN(C2CCC2)C)C3)=O)cc1C#N N1(C(c2nc(CC)sc2)=O)CCC(C)(C)C1CC(=O)NCC1=NOC(C)C1 CC1(CNC(C2CC3C(C2)C3(F)F)=O)CCCN(C(C2CN3CCN2CC3)=O)C1 c1(C(=O)NC)ccc(OCC(N2CCOCC2NC(=O)CCl)=O)cc1F Cc1nc(CNC(c2n[nH]c(C)c2Cl)=O)oc1C(=O)NCC1(C)CCCO1 c1(NCCC(=C)C)cc(=NC(C)c2ccncn2)[nH]c(COC)n1 N1(C(CC2CCN(Cc3ncc(C)cc3F)CC2)=O)CCc2cc(F)ccc2C1 C1(CNC(c2cnn(CC)n2)=O)CCC(NC(=O)CCCc2n[nH]c(=N)s2)CC1 N1(C(c2c(C)c(C(F)(F)F)n[nH]2)=O)CCC(CNC(=O)CC(F)F)C(O)C1 CC1CN(C(=O)C=Cc2cc[nH]n2)CCC1NC(=O)C(c1ccccc1)C C1(F)(C(=O)NC2CCC(CCNC(c3ncn(C(C)C)n3)=O)C2)CCOCC1 C1(C(C(=O)NC(CNC(=O)Cc2ccoc2)CO)OC)CCCCC1 N1(C(c2cc(F)cc(F)c2)=O)CC2CCCCC2(CNC(C2CC(O)C2)=O)C1 c1(-c2ccc(C)cc2CO)cccc2c(C(N3CC(F)CC3C(N)=O)=O)[nH]nc12 N1(C(c2cc(CC)on2)=O)CCN(c2ncncc2Br)C(C(N)=O)C1 c1(C(N2CCCC(NC(Cc3n(C)ncc3)=O)CC2)=O)nc(F)ccc1Cl c1(NC(C2COCCN(Cc3cc(OC)cc(C)c3)C2)=O)cc(O)c(Cl)cc1F Cc1nn(C)c(S(=O)(=O)NCC(c2ccccc2)C)c1Cc1cnc[nH]1 Cc1cc(NC(=O)CC2C=CC(NC(=O)C(N3CCCCC3)C)C2)ccc1Cl c1(C(=O)NCC2(C)CC(NC(C3(c4ccsc4)CC3)=O)C2)ccc2nc(S)oc2c1 c1(-c2ccc(NC(c3c(C)nsc3)=O)nc2)ccc2c(c1)OCO2 C1(NC(C=CC)=O)CCN(C(=O)CNC(c2c(Cl)cccc2Cl)=O)CC1C CC(CC(=O)NCCCN(C)C(c1csc(C(F)(F)F)n1)=O)c1cccnc1 c1(NC(C2SCCN(C(c3ccc(C(=O)OC)cc3)=O)C2)=O)cc(Cl)cc(Br)n1 c1(OC)cscc1C(=O)NCCC1CN(C(c2cnc(S)[nH]2)=O)C1 c1(C(=O)NCC(CC)NC(=O)CC2CCOCC2)ccc(OC)c(S(N)(=O)=O)c1 C1(NC(C(CC)(C)CO)=O)CN(C(c2ccc(F)c(Cl)c2)=O)C2(CCOCC2)C1 O=S(=O)(c1ccc(NCCc2ccnc3ncnn23)cc1)N1CCCC1 C1(CN(C)C(C2COCC2(C)C)=O)CCCN(C(=O)C(Cl)=CCl)C1 Cc1cc(C#N)sc1NC(C1CC(NC2CCCC2CO)C1)=O.S(C)(=O)(=O)N c1(N2CC(NS(CCC)(=O)=O)C2)nccc(=NCCCCCN2CCCC2)[nH]1 C(=O)(CC(C)CC(C)C)NCC(CC)(CC)NC(c1cc2n(n1)CCC2)=O c1(C(N2CCC(NC(c3c(CCC)occ3)=O)C2)=O)cc(F)cc2nc(S)[nH]c12 c1(OC)cccc2c1OCCC2NCc1cc(S(=O)(=O)N(C)C)ccc1Cl c1(CC)cn2c(n1)CCC(C(=O)NCCC(C)NC(c1c(C)cnn1C)=O)C2 c1(OC)ccc2c(C)c(C(=O)NCC3CCC(NC(=O)CC(C)F)C3)oc2c1 c1(CNC(=O)OC(C)(C)C)cccc(C(=O)NCCC2CC3CCC3C2)c1 Cc1cccc(C)c1C(=O)NC(C)Cn1cc(-c2cc(F)ccc2N)nn1 C=C(C)CC(Cc1ccccc1)NC(C1CC1C1CC1C(=O)O)=O N1(C(c2ccc(C#C)cc2)=O)C(C)CC2CN(C(C3CC4C(C3)C4(F)F)=O)CC12 C(c1cocn1)=CC(=O)NCC(CNC(=O)C(C)C#N)OC C(CCCCN=[N+]=[N-])NC(CC1(C)CCN(C(CC(C)CN(C)C)=O)C1)=O C1(O)(CNC(C2C(C)(C)CO2)=O)CCCN(C(=O)CSc2n[nH]c(O)n2)C1 c1(C(N2C(C)(C(=O)NCc3ccc(Cl)cc3Cl)CC2)=O)cc2cccnc2s1 S(=O)(=O)(c1ccc(C)cc1)N(C(C(=O)NC(c1scc(C)n1)(C)C)=O)CCC#N c1(C(N2CC(CC(C)NC(c3nccn3C)=O)C2)=O)coc(-c2ccccc2)c1 C1(C(=O)NCCCn2cnnn2)COCCN(C(=O)C=Cc2nccs2)C1 CCCC(C)(C)CC(=O)N1CCC(CNC(C2CC3CCC2C3)=O)(OC)C1 Cc1cc(C)c(C(=O)N(CCCCCNC(C2CN3CCC2C3)=O)C)cn1 c1(C(CNC(=O)C2CC2)NC(C(C2CCC2)OC)=O)ccc(N(C)C)cc1 C1(CNC(CSCCCC)=O)C2CN(C(=O)C(CC3CC3)CC)CC12 N1(C(CC2(NC(c3nccc(CC)c3)=O)CC2)=O)CC(C#N)C2(CCC2)C1 Cc1nc(C2CC2)ncc1C(=O)NC1(CF)CN(C(c2cnn3c2OCC3)=O)C1 C1(NC(c2coc(CCNCCSC)n2)=O)CCCC(NC(=O)CS)C1.C(N)(=O)N C1(Sc2ccc(C(=O)OC)cn2)CCN(N2CC3(CC(=O)NCC3C(C)C)C2)C1 N1(C(C23CC(C)(C2)OC3(C)C)=O)CCC2(NC(C3CC(F)C3)=O)CCCCCC12 N1(C(C=Cc2c(C)cccn2)=O)CC2(CCN(CC3CC(C)CC(C)(C)C3)C2)C1 c1(C(=O)NC2C3CN(C(C4C(C(=O)OC)C4)=O)C2CC3)cc2nccc(Cl)c2s1 c1(C(=O)NCC2(C)N(C(CN(C3CC3)CC)=O)CCC2)ccc2nnnn2c1 C1(NC(c2cnn(-c3ccccc3)c2)=O)CCN(CC2CC(N3CC(F)C3)C2)C1 C1(SC(c2ccccc2)CNS(CCCC)(=O)=O)CCCS(=O)(=O)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])N1CCOCC(CNC(C(n2ccc(C)n2)C)=O)C1 c1(C(=O)NC2(CN(C)C(C34CCC3C4)=O)CC2)cccc(C2(C#N)CC2)c1 c1(NC(c2scnc2-c2ccc(CO)nc2)=O)cc(F)ncc1F C(=O)(C(C(C)(C)C)SC)N1C(CNC(C2(C)CNC(=O)O2)=O)CC(C(F)(F)F)C1 c1(C(N2CC(NC(c3cc(Br)co3)=O)(CO)C2)=O)cccnc1S C1(NC(COc2cc(C)on2)=O)CC2CCC1(NC(c1cc(F)ccc1F)=O)C2 C(=O)(CS(=O)(=O)CC(=O)NC1CN(C(=O)CC2CCCC2(F)F)CC1(C)C)OC N1(C(C(CC)OC)=O)CCC(F)CC1C(=O)NC(C)(C)COC(C)C c1(CC)ccc(C(=O)NC2CCN(C(c3ccc(-c4ccccn4)o3)=O)C2)nc1 C1(c2nnnn2CC2CC2)(Nc2cc(CC)c(Cl)cn2)CC2(COC(C)C2)C1 N1(C(C2(C)CCC(C)(C)C2)=O)Cc2nccn2CC(NC(c2ccco2)=O)C1 c1(C(=O)NCC#CC(=O)NCC2(CC)CCCO2)cc2n(n1)CCO2 CCC(C)(C(=O)N1CCCC1CNC(c1c(-c2cccnc2)noc1C)=O)OC c1(C(=O)NC2CCC(CNC(c3cc(C)n(C)n3)=O)C2)ccc2ocnc2c1 C1(OC)CC(C(=O)NCC(O)C(C)(C)C)N(C(=O)CC(C)(C)OC)C1 c1(OC)ccc(F)c(CN2CCN(S(=O)(=O)CC3CC(N)C3)CC2)c1OC N1(C(CCCOCC)=O)CC(NC(C2CC2c2ccc(Cl)cc2)=O)C(O)C1 N1(C(C(=O)Nc2cnc(CCCC)s2)=O)CCC2CC3(CCC3)C2C1 C(=O)(CC(=O)NCC1CC1)NCCC(C)NC(C1CCC=CO1)=O c1(C(=O)NCC(CNC(C2CNC(=O)N2)=O)OC)ccc(Cl)c(F)c1 C1(O)(CNC(C2CC(OC)C2)=O)CCN(C(=O)C(=O)NC2CCCCC2C)CC1 c1(C(=O)NCCC(CNC(C=C(C)C(C)C)=O)O)cn(C)nc1-c1cccs1 c1(C(=O)NCCC(C)NC(=O)C(O)C(F)(F)c2ccccc2)ccc(=O)n(C)n1 N1(C(C(c2cc(F)cc(F)c2)C)=O)CC(NC(=O)CO)CC(CC(N)=O)C1 N1(C(c2c(C)nccn2)=O)CC(C)(C)OCC1CNC(C1CSCCS1)=O c1(OC)ccnc(C(=O)NCC2CCCC2NC(C2(C)CCCO2)=O)c1 C1(OCCOCC)CCCN(C(C2(C)CNC(=O)N2)=O)CC1 C1(CC)(CC)CC(C(=O)NCCC2CC(NC(=O)C(C)C3CCC3)C2)C1 c1(CN(C2CCCCCC2)CCN(C)C)ccc(C2CC2C2CCC2)cn1 N1(C(=O)NCC2OCC(C)C2)CCN(C(C)CNC(=O)C(F)(F)F)CC1 C1(C)(C(N(CCC#C)C)=O)CCN(C(=O)C=CC2(C)COC2)C1 C1(CNC(C=CC(=O)OCC)=O)CC2CCCC2C1.C1(C2CCCC2)C(=O)N1 c1(C(=O)NCC(C)N(C(c2cnc(COC)s2)=O)C)c(C)csc1Cl C=CCCCCC(=O)N(C1(CC(=O)N(C)CC2(O)CCOC2)CC1)C CC1CN(C(c2ncc(Br)cn2)=O)CCCN1C(c1cnc(O)s1)=O C1(Cn2c(CN3CCOCC3)nc(-c3ccn(C)n3)n2)CCN(S(N)(=O)=O)CC1 C(=O)(CCCC(C)(F)F)NC(CNC(C(COC(C)=O)C)=O)C(C)C C1(CC(NOCC(=O)OC)=O)CN(C(c2cc(C(C)C)[nH]n2)=O)C(C)(C)C1 c1(OC)ccc2c(C(=O)NC3CCN(C(=O)CC(C)OC)C3C)n[nH]c2c1 C1(NC(CCCCC#C)=O)CCCC12CCN(C(c1cnc(CC)s1)=O)CC2 C=C(Cl)CC(C(=O)NC1CCCCC1(C)C)NC(C1C2CC3C(C2)C13)=O C1(CC)CC(CC(N2CCOC(CNC(=O)CCCCSC)C2)=O)CCO1 C1(CC)CN(C(=O)CN2CCN(C(=O)C=C(C)C)CC2)C(CC)CN1C(C)=O c1(CC(=O)NCC(CN(C(C2CC(O)(CC#C)C2)=O)C)O)ccc(OC)cc1F c1(C(=O)NCC2(NC(C(CC)NS(C)(=O)=O)=O)CCCC2)cc(F)c(F)cc1N N1(C(C2(COC)CCC(=O)N2)=O)CCCC(NC(C2CC=CC2)=O)C1C C1(CC)CCCC(NC(C2CN(C(=O)CCc3ccn(C)n3)C(C)(C)C2)=O)CC1 C1(NC(CCN(C)CC)=O)CCC(O)CN(C(C2(C)CCN(C)C2)=O)C1 C1(C(N2C3C(NC(CCCC)=O)CC(C3)C2)=O)CCC2(CCCCC2)C1 Cc1sc(C(N2CCCC2CNC(C2CCCS2(=O)=O)=O)=O)nc1C(F)(F)F C(=O)(C(=O)CC(C)C)N(C(C1CCOC1)CO)CC.C=C1CC2(C1)C(=O)NC2 c1(C(C)=O)ccc2nc(-c3cnc(NC(c4ccc(F)c(C)c4)=O)nc3)cn2c1 C1(NC(C2(C)CCSCC2)=O)CN(C(=O)Cc2cncs2)CC2(CCOCC2)C1 c1(OCC)cc(OC(F)(F)F)ccc1NC(c1cn(CC)cn1)=O C1(C(=O)NC2C(CNC(c3c(C)nns3)=O)CCC2)CCc2nnnn2CC1 C1(CC)CCC(C(=O)NCC2C=CC(NC(=O)CSc3ccccn3)C2)O1 C1(NC(CC2(C=C)CCCCC2)=O)CC1C1CCN(C(C2CCC(O)C2)=O)CC1 C1(NC(c2nn(CC)c(C)c2)=O)(CC)CCCN(C(=O)C(C)(CC)CC)C1 N1(C(CCCCOC)=O)CC2CCC1C(NC(c1ncccc1Cl)=O)C2 c1(C(=O)C2CC2)ccc2[nH]c3c(c2c1)CCCC3C(=O)N1CCc2cccc(F)c21 C1(CC)CN(C(C2CC3CCC2N3C(c2cnn3c2CCC3)=O)=O)CCCO1 N1(C(c2ccc(CC)c(N)c2)=O)CCCC2CN(C(=O)C(C)N3CCC3)CC12 C1(C(=O)NCC(C#C)OC)C2CC2CN1C(=O)CCc1ccccc1 c1(C(=O)NCCCC(C)NC(C2C(F)(C(=O)OC)C2)=O)cc(C(F)(F)F)cn1C c1(CC(=O)NC(CCCCNC(c2ccc(OC)s2)=O)C)cccc(F)c1Cl N(C(=NCCCC1CC1)N1CCC(Cc2ccccc2F)C1)CC(C)C C(C(C(=O)NCC(C1CCCCC1)F)NC(=O)C(=O)NC1CC1)N(C)C C1(NC(c2[nH]c(=NC)sc2)=O)CC2CC(NC(=O)C(F)C(C)C)CC2C1 c1(C(N2CC(OC(C3C(C(N(CCC)CC)=O)C3)=O)C2)=O)cc2scnc2[nH]1 c1(C(=O)NCC(C)N(C(=O)C=Cc2cccnc2)CC)ccc(Cl)cc1F Cc1ncc(CCC(=O)NC(CNC(c2ccsc2Cl)=O)C2CCC2)s1 CC1(C)CN(C2CCN(C3CCCC(F)(F)C3)C2=O)CCS1 C(C(C)C(C)(C)C)N(CCC#C)C.C1(=O)CN1C(C)CC c1(C(=O)NC(CCCNC(c2cn(CC=C)nc2)=O)C)ccc(OCCF)cc1 N1(c2cc(NCC3CC(C)(C)OC3)ncn2)CCN(Cc2cccnc2)C(=O)C1 N1(C(C2(CSC)CC2)=O)CCC(C2CCN(C(c3c(C)ncn3C)=O)CC2)CC1 c1(C(=O)NCC(CCOC)NC(c2ccc(Cl)c(C)c2)=O)cccc(Cl)c1N CC1CC=C(C(=O)N2CCC(F)(C(=O)NCC(CO)C(C)C)C2)CC1 C1(CNC(c2cccc(SCC)c2)=O)CC2CCCC2N1C(C1CC(CC)=NO1)=O C#Cc1cc(C(=O)NC2CCC(NC(=O)C(F)CC3CCC3)C2)cc(Br)c1 C(=O)(CCC(=O)N(CCCCCCNC(=O)C(F)(F)C1CCC1)C)N(C)C C1(NC(c2cnc(C)[nH]c2=N)=O)CN(C(C2CCC(C)O2)=O)Cc2nccn2C1 c1(C(=O)NC(CNC(C2(C(=O)OC)CCC2)=O)(C)C)ccnnc1NC(C)(C)C.CC C1(CNC(c2ncc(C)c(Cl)c2)=O)CC2(CCN(C(=O)Cn3cnnc3)C2)CO1 C(=O)(C#CC1(CC)COC1)N(CC=CC(=O)NC(c1nncn1C)CC)C C(=O)(C(C)S(N)(=O)=O)NCCCC1(CNC(Cn2c(C)ncc2)=O)CCCC1 C1(CNC(c2c(C)cn(C)n2)=O)CCN(C(c2ccc([N+](=O)[O-])o2)=O)C12CC2 C12(CNC(c3n(C(C)C)ccc3)=O)CC1CN(C(c1nnsc1CN(C)C)=O)C2 CC1C(=O)CC1C(=O)N(C)CC1CCN(C(=O)CCOC2CCCC2)C1 O=C(CCS(=O)(=O)C(F)(F)F)NC1CCC(CNC(C2(F)CC=CC2)=O)C1 c1(N(CC(=O)N(CC(C)NC(C(N2C(=O)CCC2=O)C)=O)C)C)ccc(Cl)cn1 C(C1COn2cc(nn2)C2N(C1=O)CCCC2)OC.C1(NC(C)=O)CC2CC2C1 C12(CNC(c3cc(C)no3)=O)CCCC1N(C(=O)CN1CC3C=CC1C3)CCC2 N1(C(c2nccc(N(C)C)c2)=O)CCC2CCN(C(=O)CC(C)(C)C)C2C1 C1(C(=O)NC(C2CCCO2)(C)C)CC2CCCC2N1C(=O)CC1NC(=O)NC1=O Cc1sc(C(=O)NC2CC(NC(=O)C(C)Cn3ccnc3)CC2O)nc1O C1(C(N(CC(C)NC(=O)CC2CNC(=O)O2)CC)=O)CCC2(CCCC2)C1 c1(C(N2CCC(N(C(C(CN(C)C)N(C)C)=O)C)C2)=O)cc(Cl)cc2c1CCC2 O=C1CNc2ncc(C(N3CC4CC3CN4C(=O)C(O)c3cnc[nH]3)=O)cc2N1 c1(C(=O)NCCCN(C(=O)CCOC2CCCCC2)CC)cc(C(F)F)cs1 N1(C(c2c(C)cc(F)cc2)=O)C2CCC1CN(C(=O)CSC(F)(F)F)C2 C(CCCC(=O)N1CC(F)(F)CC1C(N1CC(=O)NCC1C(N)=O)=O)(OC)OC C1(NC(c2n(C(C)C)ccn2)=O)CC2(CCC(CNC(=O)C(F)C(C)C)OC2)C1 C=CC(C)CCNC(=O)C(C)N(C(C1(CCF)CCC1)=O)C1CC1 CC1CN(C(C2CN(C)CCN2C(=O)CCc2cncs2)=O)CC(C)N1C C1(CNC(C=CC=CCC)=O)C2CN(C(c3cnn(C)c3C)=O)CC12 n1(C(C)C)cc(-c2cn(C(C)CNC(C3CCC3C#N)=O)nn2)cn1 c1(C(N2C(C(=O)Nc3c(OC)ccc(C)n3)CC(O)C2)=O)ccc(Br)c(F)c1F N1(C(c2cn(C)c(C(F)F)n2)=O)CCC(NC(=O)Cc2cc[nH]n2)C(O)C1 Cc1nc(N2CC(C(=O)NCc3ccncc3Cl)C(C)(C)C2)ccc1C#N CC(C(=O)NCCN(CC(=O)NCC1(CC2CC2)CC1)C)n1ccnn1 c1(C(=O)NCC(C)NC(COCC(C)C)=O)cn(C(C)C)nn1 C1(N(C(=O)CC2CC(C)(C)CO2)C)CN(C(C2CC3C(C2)C3(C)C)=O)CC1(C)C O=C1CC(C(=O)NC2CCCC2C(=O)Nc2ccc(C(F)(F)F)cc2I)NC(=O)N1 C1(NC(Cc2c(C)noc2C)=O)CC(O)CN(C(c2ccnc(N(C)C)c2)=O)C1 CN1CC2OCCN(C(C3CN(C(c4ccc(I)cc4Cl)=O)CCC3O)=O)C2C1 C(CCC(c1ccccc1)NC(=O)CC1CCCC1)N(C(C1(Br)CC1)=O)CCO Nc1cc(C(=O)NC2CC2NC(=O)COCCN(C)C)c(Br)cn1 N1(C(c2cc(C)ncn2)=O)CC(C2CCCN(C(=O)CCC3CCC(=O)N3)C2)C1 N1(C(CC(=O)N(C)C)=O)CCCN(C(c2cccc3c2CCO3)=O)C(CO)C1 CC(C)CC(F)C(=O)N(C)CCC1CCN(C(C2CCCC2)=O)CC1 C1(C(N2CCN(C(c3ccn(CCF)n3)=O)CC2CF)=O)CCc2cncn2C1 N1(C(CC(CNC(=O)CC2CCCNC2=O)C2CCC2)=O)CC2CC1C(F)(F)C2 c1(C(=O)NCC2(C(C)NC(C(C=C)O)=O)CC2)cc(Br)c(O)nc1C c1(NCC2C(C(=O)O)C2)cnc(CSc2ccc(C(F)(F)F)cc2O)c(F)c1 C1(NC(C(C)SCC)=O)CC2(C1)CC2NC(c1coc(C(F)F)n1)=O C1(C(=O)Nc2ccc(F)cc2)CC(O)CN1CC1CN(C(C(C)NC(C)=O)=O)C1 C1(O)(C(C)NC(CSCCCC)=O)CN(C(C2CCCC2c2ccccc2)=O)C1 c1(CNC(C(=O)NC2C(NC(C)=O)C2)=O)nccnc1C C1(CC)C(C(=O)OC)CCN1C(c1cncc(C(N)=O)c1)=O N1(C(c2ncc(C)c(Br)c2)=O)CCOC2(CCCN(C(=O)CCCCBr)C2)C1 C1(C(C)C)CN(C(=O)CCOCC(F)(F)C(F)F)CCC1NC.S(=O)(=O)(CCC)N c1(OC(CC)C)ccccc1C(=O)NC1CC1NC(C1(c2cn[nH]c2)CC1)=O C1(CC)CN(C(=O)C(C)CSC)CCC1CNC(=O)C(F)(F)CO C1(CNC(C(C)OCCOC)=O)CN(C(=O)CCC(=O)OC)CCCO1 C(=O)(C(C)(C)C)NCCO.C(C(=O)NCC1CC1CNC(=O)CN)SC N1(C(c2nnnn2C)C)CC2CC1CN2C(c1ccc(-n2ccnc2)cn1)=O C(=O)(C1CCOc2ccc(F)cc21)NCC1CCC(NC(c2cc(C)[nH]n2)=O)C1 C1(C)(Cn2cc(CN(C3CCN(C)CC3)C)nn2)CCCCC1(F)F N1(C(C(c2ccc(C)o2)C)=O)CCOCC(CNC(c2ncoc2C)=O)C1 N1(C(C2(OC)CCC2)=O)CCC2(CC1)CN(C(C1CC1C)=O)C2C(C)C O=C(C1CC(O)c2ccccc21)NCC1CC(NC(=O)CC2CCCO2)C1 C1(C(C)C(=O)NC2CCN(c3ccncc3)C2)CCN(C(=O)N(C)C)CC1 C1(CC)C(NC(=O)CC(O)CN(C)C)CCCN1C(C1CCOC(C)C1)=O C1(NC(CC2CCN(C(CCCCCC)=O)C2)=O)C2CCC(C2)C1(C)C c1(CNC23CC(C(=O)NCC4(C(=O)OC)CCC4)(C2)C3)c[nH]c2cccc(Cl)c12 Cc1c(CCN2CCCC(CCNC(C3CCC(=O)N3)=O)C2)cnn1C c1(C(c2ccccc2)NCNC(C2CCC(C3(c4[nH]c(=N)oc4)CCC3)O2)=O)cccc2nsnc12 C12(NC(C(C3CCOCC3)OC)=O)CCCC1CN(C(c1cnc(C3CC3)[nH]1)=O)C2 c1(C(N(CC(C)N(C(C(C)NC(COC)=O)=O)C)C)=O)cnc2[nH]c(=N)sc2c1 C1(NC(CN(C(=O)OC)C)=O)CC(C(=O)NCCC2CCCCO2)(CO)C1 C12(NC(c3nc(CCC)oc3)=O)COC(C1)C(NC(=O)CC1C=NN(C)C1=O)C2 C1(CC)CCN(C(C2CN3CCC2CC3)=O)C(C(N2CCC(C)(CCO)C2)=O)C1 Cn1cc(C2(NC(=O)C(=O)NCCC3CC3(Br)Br)CCC2)cn1 C1(=CC(=O)N(C(c2cn(CCC(C)C)nn2)=O)C(=O)OC(CC)C)CCN(C)CC1 C(=O)(C(C)(O)C(C)(O)C(=O)N1CC2C=CC2C1)OC C1(NCc2c(=N)cc[nH]c2)CC2(C1)CC(NC(c1n[nH]cc1[N+](=O)[O-])=O)C2 C(=O)(CC(F)(F)F)NCC(C)(CO)OC(C(C)OC1CCCC1)=O Cc1cc(=NC(C)c2cccc(N3CCCC3)c2)[nH]n1C(C)(C)C c1(C(=O)NC2(C(=O)OC)CCCOC2)cc2c(s1)CCC(C)(C)C2 N1(CC(=O)NCCC2CCCN(C(C3C(=C)C3)=O)C2)CC(=O)Nc2ccccc21 CC1(C)CN(C(C2CC2C23CC(CO2)C3)=O)CC1NC(c1cc(N)ccn1)=O Cc1c[nH]c(=NCCCCN(C(=O)CC2C(=O)N(C)N=C2C)C)nc1O CC1CCC(C)(C=CC(=O)N(C2CCCN(c3nnnn3C)CC2)C)C1(C)C c1(C(=O)NCCC2CCN(C(C3N(C)C(=O)CC3)=O)C2)nc2c(s1)COCC2 N1(C(C2OCC(C)C2)=O)CCC2(CCN(C(c3cnsc3)=O)CC2)C1 C(=O)(CC(CC)CCCC)NCC(CCC)C(=O)NCc1ccoc1C c1(-c2c(C(=O)NCCCN(C(CCCOC(C)C)=O)C)c[nH]n2)ccccc1Cl C=C1CC2(C1)CC(C(N1CCC1CNC(c1c(C)nn(C)c1C(F)(F)F)=O)=O)C2 C1(NS(CC(CC)C)=O)CC2OC(C)(C)OC2C1 C1(C(N2CCC(NC(=O)Cn3cnnc3)(CF)C2)=O)Cc2cc(F)ccc2O1 CN1C(=O)NC2(CCC(C(=O)NC3CC(NC(C4CCCCC4)=O)C3)CC2)C1 N1(C(CCCOCC)=O)CC(CNC(C2(CC(=O)OC)CCC2)=O)C2(CC2)C1 c1(C(=O)NCC(C2CCOC2)NC(CC(C)C)=O)ccccc1SC(F)F C(C)(CC(=O)N1CCC(NC(=O)C(C)=CC2CC2)CC1)(C1CCC1)N(C)C S(=O)(=O)(c1cccc(Cl)c1)NCCC(=O)NC(CN(C(=O)CCOC)CC)C c1(N(CCC#N)C)[nH]c(=NCCNC2(OCC)CCOCC2)nc2c1ncn2C C1(C(=O)NCC2CCCC(CNC(=O)COC(F)(F)F)C2)CCC2(CC1)CC2 c1(C(=O)NCC2N(C(C3C(C)CC(C)O3)=O)CC(C)(C)C2)[nH]nc([N+](=O)[O-])c1Cl N1(C(C2(F)C(C)C2)=O)CCCCC(CNC(=O)Cc2ccc(F)cc2F)C1 C#Cc1ccc(C(N2CCCC2CNC(c2occc2C(C)C)=O)=O)c(OC)c1 Cc1cc(C(N2CCC(NC(=O)C3CC3)C(O)C2)=O)c(C)n1C1CCCCC1 c1(C(=O)NC(C)CCN(C)C(C2CC(=C3CC3)C2)=O)cc2cc(Cl)cnc2[nH]1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(C1CN(C(C2CCCS2)=O)C1)C C1(C(=O)NC(c2ccc(-c3ccc(F)c(F)c3)s2)C)CCCN(C(=O)C(N)=O)CC1 Cc1ccc(C(=O)NCCC2CCN(C(=O)C(C)n3cccn3)CC2)cc1O N#CCCCC(=O)NCCN(C(c1cnn(C2CC2)c1)=O)CC1CC1 C1(C(=O)Nc2cccc(SCC(=O)OC)c2)CC2CCC(C1)S2 N1(CC)C(=O)CCC1C(=O)NC1CC(NC(c2ccnn2C2CCOCC2)=O)C1 Cc1cn(C)cc1C(N1CCC(N(C(=O)Cc2cncn2C)C)CC1)=O N1(C(=O)COc2cccnc2)CCC2C(CCCN2C(=O)CC2CC=CC2)C1 C(C)(C)(C(C)CC(=O)NC(CC1CC1)C1CCC1)NC(CN(C(=O)OCC)C)=O Cc1cc(N)cc(C(=O)NC(c2cn(-c3ccc(CO)cc3)nn2)(C)C)c1F C(=O)(C1=CNC2=NCCC2=C1)NCCN(C(C1N(CCCCC)CCCC1)=O)C c1(C(=O)NCC(C2CCCC2)NC(C(CC)=CC)=O)cnc(C#N)s1 c1(C(N2C3C(NC(=O)COCC4CCC4)C(CC3)C2)=O)ccc2sncc2c1 C(CCCCC(=O)NCC1CN(C)CC(C)O1)n1cc(-c2c(C)nsc2)nn1 c1(C(=O)NC2CN(C(C(C3CCCOC3)OCC)=O)C2)c[nH]nc1Cl C(CC(C)CC)(C(=O)N(CC(C)(F)F)C)NC(C(CCC)OCC)=O C1(O)(C(C(N2CCOC(CNC(C3CC4C=CC3C4)=O)C2)=O)F)CCCCCC1 Cc1cc(-c2cn(CCN(C(=O)NCCCC(N)=O)C3CC3)nn2)cc(F)c1 c1(CC)cc(C(=O)NC2CCCC2NC(C2(SC)CCC2)=O)ccc1Cl C1(CNC(CN2CCN(C)C(=O)C2)=O)CCCC2CN(C(=O)C(=O)N(C)C)CC12 C(=O)(C(C)C(C)C(C)(C)C)NCC1CC(NC(c2ccc(C(=O)OC)nc2)=O)C1 Cc1ccc(NCC(N2CCCC2CCNC(=O)NCC(N)=O)=O)cc1C C1(C(N)=O)(C(=O)N(CCOCC(=O)NCCF)CCO)CC1 Cc1noc(CCC(=O)N(CC(=O)NCCc2ncc(C)o2)C2CC2)n1 C1(CCC)(NC(C2CCCC23CCC3)=O)CCCN(C(=O)C(C)(C)CF)C1 C(CCCCC(=O)N(CCCNC(=O)C(C)c1ccco1)CCO)NC(=O)OC c1(C(N(C2CCC(NC(C3(CF)CC3(F)F)=O)C2)C)=O)ccc(-c2cccs2)o1 C1(C(=O)NC(C)(CN2CCOCC2)C2CC2)CCC(NC(c2ccsc2Cl)=O)C1 C(N=c1[nH]c(=NCCCOC2CC2)[nH]c2cc[nH]c12)C1(C)CCCCC1(F)F N1(C(C(C)Cc2ccc(Cl)cc2)=O)CC2CC(C1)CN(C(=O)C1=CCC1)C2 C1(OC)CN(C(=O)C(c2ccccc2)O)CC1CO.N1(CCC(=O)CO)CCCC1 c1(-n2c(C)cnn2)cc2c(cc1F)NCC2 C1(C(=O)NCC(C(C)(C)C)NC(CCSCCC)=O)CC(C(C)(C)C)=NO1 C12(NC(CC(C)(C)C3CC3)=O)CCCC1CN(C(=O)C(C)(C)S(C)(=O)=O)C2 Cc1cc(Cl)c(C(=O)NCC(C2CCC2)NC(=O)C(C)(C)N2CCOCC2)cn1 CCCCCCC(CC)C(=O)NC(C)CC(C)NC(=O)C(C(C)C)SC C1(CC(=O)N(C(C)C(=O)N2CC(n3cccn3)C2)CC)CCCCC1 N1(C(c2cn(CCC=C)nn2)=O)CCC2CN(C(=O)CCC(C)(C)C)CC2C1 c1(C(=O)NCC(CNC(C(C(C)C)OCC)=O)(C)O)cccc2nonc12 C1(CC(N2CC(N(C)CC)C2)=O)CCCC(NC(c2sccc2C#N)=O)C1 N1(C(CNC(=NCCCC(=O)OC)NC(C)C(C)SC)=O)CCC(C2(OC)CC2)C1 N1(C(c2c(C)snc2)=O)CC(=O)NCC1C(=O)NCCSCCO c1(C(=O)NC(C2(O)CCN(C(c3cnn(CCF)c3)=O)C2)C)cc(N)ccn1 C(C(CN=c1[nH]c2cccc(F)c2s1)C(F)(F)F)NC(C1CCc2nnc(O)n2C1)=O c1(-c2ccc(OC)cc2)n[nH]c(=NC(=O)NC(c2ncsc2C)C)s1 N1(C(c2ncn(C)c2)=O)CCC2(CC(C(=O)N3Cc4ccncc4C3)=NO2)C1 C12(C(=O)NC3(CC=C)CCC3)CCN(C(=O)CN3CCC(F)CC3)CCC1C2 n1(CCOC)nccc1C(=O)NC1CCCC1NC(=O)C(C)Cn1cccn1 C(=O)(C(C)(C)C1=CCSCC1)N(CCC(C)NC(C1CC1C(F)F)=O)C c1(C(=O)NCC(CCNC(CC=C)=O)O)cnc2c(c1)NCC2 C(N=c1[nH]c2c(c(=NC(C)c3c[nH]ccc3=N)[nH]1)CCC2)c1c(CC)nco1 Cc1cccnc1-c1cn(C2CN(C(C3CCC3C(=O)N(C)C)=O)C2)nn1 C12(C(=O)NC(C(C)NC(c3c(C(C)C)cco3)=O)C)CCC(CC1)C(C)O2 c1(OC)ccc(F)c(CC(=O)N(CCN(C)C(c2cc(C#N)on2)=O)C(C)C)c1 C(=O)(C1=CC2C=CC(C1)C2)NCC(CC=C)NC(=O)CC(C=C)CC Cc1ccc(Cl)c(C(=O)NC2CCCC2NC(C2CN3CCCC2C3)=O)c1 C1(O)(CNC(C=CC=CCC)=O)CCCN(C(=O)CCOC2CCC2)C1 c1(C(=O)NCC2(C)CCN(C(C3CCC3)=O)C2)nc2c(Br)cncc2[nH]1 N1(C(Cn2c(C(C)C)ncc2)=O)CC2C(CN(C)C(c3coc(O)n3)=O)C2C1 C(C)(CCCC(C)C)(c1n(CC)nnn1)NC12CCC(C(=O)NCC)(CC1)C2 O(N(C(=O)C1CCCC1N(C)C)C(C)C)CC.C1(=O)C(CC(C)C)N1 N1(C(c2cc(Br)nn2C)C(=O)NC)c2ccccc2CC1Cc1ccccc1 Cc1oc([N+](=O)[O-])cc1C(=O)NCCCOCCNC(c1ccc(N)cc1Cl)=O Cc1nn(C2CC2)c(Cl)c1C(=O)NC(C)C(CO)NC(=O)CC(=O)OC(C)(C)C C12(C(N3CCC(OCCNC(c4cccc(Cl)c4)=O)C3)=O)CCN(C1)S(=O)(=O)C2 Cc1ccc2c(C(=O)NC(C)CNC(=O)CCC3CC3C)ccnc2c1 c1(N(C)CC2(OC)CCCC2)nnc(Cc2ccccc2)n1C N1(C(C23CC(C)C2C3)=O)CC(NC(=O)CN(C2CCCC2)C)CC(C)C1 c1(CNc2c(F)ccc(Br)n2)cc2cc(Br)ccc2s1 N1(C(C(C)(Cl)Cl)=O)CC(CNC(c2sccc2-n2cnnn2)=O)C(O)C1 CCCCC(C)CC(=O)N1CCN(C(c2cc(C)no2)=O)C(CCO)C1 CC(C)CC(C(=O)NCC1(C(C)(C)C)CCN(C(=O)C2=COCCC2)C1)C(C)C N1(C(C(c2cncnc2)C)=O)CC2CCC1CN2C(=O)CCC(=O)N(C)C1CC1 c1(CC)cc(C(=O)NC2(CCNC(=O)C(C)(C)C3CCOCC3)CCC2)ncn1 C(=O)(CC(C)(C)C(=O)NCCNC(c1cn(C2CCN(C)C2)nn1)=O)OCC c1(OC)ccc(S(=O)(=O)NC(C)CCC(=O)NC(C)(C)C)c(F)n1 C1(NC(c2c(C)nc(C)s2)=O)CCCCCC1C(=O)NC1CC(O)C1OC C=CCCC(F)(F)C(=O)N1CC(C(=O)NC(c2ccnn2CC)C)(C(N)=O)C1 c1(C(N2CC3CC(NC(c4coc5c4COC5)=O)C3C2)=O)cccc2ncoc12 c1(CCC(N2C(C(C)NC(c3cc(C)ncc3)=O)CCC2)=O)ccc(O)c(Cl)c1 C(=O)(NNC(=O)CCCCCCBr)c1c(C)n(-c2ccc(C(C)(C)C)cc2)nc1 N1(C(c2c(OC)scc2)=O)CC(NC(c2c(F)cccc2Cl)=O)C(C2CC2)C1 CC12CC(C(=O)NCC(O)CNC(c3cc(C4CCC4)no3)=O)(C1)C1(CCC1)O2 c1(CNC(=O)N(C2CC2)Cc2ccccc2)cc2ccccc2s1 Cc1ncc(CCC(N2CC3CC2CN3C(=O)CN(C)C2CC2)=O)c(O)n1 c1(C(C(=O)NCCC)N(C)Cc2nnc(C3CC3)o2)cccc2c1nnn2C N1(C(C(C)OCC)=O)CCC(C(=O)NOc2ccc(CC)cc2)C12CC2 c1(CC2CCN(C(c3ccn(C(F)F)n3)C(=O)NC3(C)CC3)C2)ccc(Cl)cc1 C1(NC(C(=O)N(C)C)=O)COC2(CCCN(C(=O)CCc3cccnc3)C2)C1 N1(C(C(CC=C)(F)F)=O)CCC2(CC1)CN(C(=O)CCC(C)OCC)CC(C)O2 c1(NC(C2CN(Cc3cccc(OC(F)(F)F)c3)CCS2)=O)cccc(O)c1 N1(C(C(CN(C)C)NC(C2COCCN2C)=O)=O)CCN(C2(C)CC2)CC1 c1(OCC)ccc(CC2(c3nnnn3CC)CC3(CSC3)C2)cc1OCC C(=O)(CCCCSC)N1CC(CCCNC(c2ccc(CC)o2)=O)(COC)C1 CC(CC(=O)Nc1cncnc1O)C(C)(C)N1CCC(C)(N(C)C)C1 c1(C(=O)NC(C)CNC(c2cc(Br)cs2)=O)cn(C)[nH]c1=N c1(N2CC(CC)C(O)C2)ncc(C)cc1S(=O)(=O)NC1CC(OC(C)(C)C)C1 c1(CC)ccc(C(C)NC(c2nccnc2C)c2nnnn2C(C)C)c(C)c1 c1(NC)ccccc1C(=O)NC1CC(CCC(=O)N(CC(C)CC)C)C1 C1(NC(Cc2ccc(C)nc2)=O)CCC(C)N(C(c2csc(C)c2N)=O)C1 CN1CCN(C(=O)CCCCC2CC2)CC1C(=O)NC1CC(C(F)F)C1 C=C1CCC(C(N2CCC(C(C)NC(c3ncccc3NC(C)=O)=O)C2)=O)CC1 C1(=O)C(CCCCCC)CN1.C=C(C)CCC(C)NC(=O)OCC.C(C)(C)(C)O c1(NC(=O)NCCc2ccno2)coc(C2CCCN2c2ccncn2)n1 CS(=O)(=O)c1ccccc1NCC1CCC2(CN(C(=O)OC(C)(C)C)C2)O1 c1(OC)cc(C)c(C(N2CCC(O)C(NC(=O)CC(C)NC(N)=O)C2)=O)c(F)c1 C(C(C)(C)CC(=O)N(C1CCCN(C(=O)C(C)c2ccsc2)C1)CCO)OC CCCC(C)CC(=O)N1CCN(C(c2cnn(CC)c2)=O)CC1c1ncc[nH]1 Cc1nc2cnn(C)c2cc1C(N1C2CCCC1CN(C(=O)CSC(C)C)C2)=O N1(C(C2CC3CCC2O3)=O)CCN(C(c2nc[nH]n2)=O)C(CF)C1 C(=O)(C(O)C1=CCCCC1)NC1CC2CCCC(C1)N2C(C1CC2(CC2)CO1)=O C(N=c1[nH]c2c(c(=NCC(F)F)[nH]1)COC2)c1ncc(C(C)(C)C)s1 C1(CNC(C(C=C)(C)C)=O)CC2(CCC2)CN1C(C1CC=CCC1)=O Cc1c(Cl)c(C(=O)NCC(C)(C2CC2)NC(C2CC2C(C)C)=O)nn1C N1(C(CC=CCNC(C2(C)CCC(=O)NC2)=O)=O)CC2CCC(O)C2C1 c1(C(=O)NCC2(NC(Cc3ccc(C)o3)=O)CCC2)cnc2n1CC(C)CC2 c1(C(=O)NC(C(=O)OC)C2CCC2)cc(C)c2cc[nH]c2c1 C(=O)(C1CCCc2c[nH]nc21)N1C2C(NC(=O)C(F)C3CCOC3)(CCC2)CC1 C1(NC(=O)C=Cc2ccncn2)CC(O)CN(C(c2cnccc2Cl)=O)C1 CCC(CCOC)C(=O)N1CC(O)CC1CNC(c1ccc(C2CCCO2)[nH]1)=O N1(C(C(CC)C)=O)CCN(C2CCN(C(=O)Cc3c[nH]nc3O)CC2)CC1 c1(N(C(CNS(C)(=O)=O)=O)CCCC2CC3CC2CN3)c(F)cc(F)cc1F N1(C(C(CC)OCC)=O)CC2CC(C)C(C1)N2C(=O)C(C1(O)CCCC1)F c1(CC)cccc(C(=O)N(CC(O)CNC(=O)C(F)n2cccn2)C)n1 CC1(NC(c2ccc(Cl)c(O)c2)=O)CCN(C(=O)C=Cc2ccc(Cl)s2)CC1 C1(NC(CC(=O)NCC)=O)CCN(C(c2cccc(C(C)(F)F)c2)=O)C12CCC2 C1(C(=O)NC23CC(NC(=O)C(F)F)(C2)C3)CCC2C1C2(F)F Cc1ccc(-c2cn(CC(=O)NC(c3ccccc3)CN)nn2)cc1 Cc1ncccc1CC(N1CCCC(CCC(=O)NC(C(C)C)C2CCC2)C1)=O c1(OC)ccc(N(CC(=O)NCC(CC2CC2)CO)C)cc1 N1(C(C2C(=C)C2)=O)CCC2CCC(C1)N2C(=O)C=C1CCCCC1(C)C c1(C(N(C2CCCN(C(c3cnccc3Cl)=O)C2)CC)=O)ccc(C)cc1C C1(N(C(C(C)P(C)(C)=O)=O)C)CCN(C(c2ccn(C3CC3)n2)=O)CC12CC2 C#CC1(C(=O)NCC2CCC(=O)N2)CCN(C(=O)CCCn2ccnn2)C1 c1(C(N(CCCNC(c2ccc(Cl)[nH]2)=O)C)=O)c(C(F)(F)F)cccc1Cl c1(C(N2C(C(C)C)CN(C(=O)CSC3CC3)CC2)=O)cccc2c1CNC2=O C1(NC(CCC=C)=O)CCCCC12CCN(C(=O)C(OCC)OCC)C2 C(=O)(C1=C(C)OCCS1)N1CCC(C(N2CCCC(OCC)CC2)=O)(CF)C1 N1(C(C2CCC(C(C)=O)O2)=O)CCCC(N(CCO)C(c2oc(C)cc2C)=O)C1 c1(OC)ccc(CCC(=O)NC(C)CCNC(=O)C(C)C2CCCO2)cn1 c1(C(N2CCC(C3N(C(C(C)n4cncn4)=O)CCC3)C2)=O)ccnn1C C1(NC(C2(C(N(C)C)=O)CC2)=O)CCN(C(C2CC3CCC2C3)=O)CC1(C)C c1(CNC(C(=O)NC2(CSC)CCNCC2)=O)sc2[nH]cnc(=O)c2c1C N1(C(=O)C=Cc2cn3c(n2)CCCC3)CCc2nc[nH]c2C1c1ccncc1 C1(CNC(C(CCCC)O)=O)COC(C)(C)CN1C(=O)CCC(C)(F)F c1(CC(=O)NCCc2c(C(=O)OCC)c[nH]n2)cc(C)ccc1OC N1(C(C(CCC)N(C)C)=O)CCCC(CNC(c2c(C)n[nH]c2C)=O)CC1 N1(C(c2c(C)nsc2)=O)CC(CNC(=O)C=Cc2cnc[nH]2)CC12CCC2 C1(C(=O)NCCSCC(=O)OC)CC1C1CN(C(=O)CCC(=O)NC)C1 C(=O)(C(C)(C)CC(F)(F)F)NCC1N(C(C2(C=C)CC2)=O)CC1 C1(NC(c2csc(C(F)(F)F)c2)=O)CCC(NC(C2CC(CCO)C2)=O)C1 CS(=O)(=O)c1ccc(Cl)c(C(=O)NCCC2CN(C(C3CC3F)=O)CCO2)c1 c1(C(N2CCC(Cn3cc(C(C)OC)nn3)C2)=O)cc(Br)ccc1CNC c1(O)ccncc1.c1(C(C)(C2COC2)NC2(COC)CC2)nnnn1CC(F)F C1(CNC(C(CSC)O)=O)CCC(CNC(c2cnn(CC(F)(F)F)c2)=O)CC1 N1(C(CC2(CNC(C(C)SCC)=O)CCCC2)=O)CCC(C(N)=O)CC1 c1(CC)ncsc1C(=O)N(C)CCOCCC(=O)NCCCn1cncn1 N1(C(C(CC)N(C)C)=O)CC(OC)C(CNC(=O)Cc2cccc(F)c2)C1 C1(NC(c2ccc3nncn3c2)=O)CC(C2CCN(C(=O)C3CC3)C2)C1 n1(CCC=C)cc(C(=O)NCCC2(O)CN(C(c3cnc(C4CC4)o3)=O)C2)nn1 CCCC(CCC)CC(=O)N1CCC(NC(C2CN(C(=O)N(C)C)C2)=O)C1CC CC1CCCCN1NC(=O)C(F)=C1CC(OC)C1.n1(CC(=C)C)cncn1 C1(C(=O)NCC(C)OC(F)F)CCCCCN1C(c1ccsc1)=O Cc1cncc(NC(C2(CNC(C3(C)CCSCC3)=O)CC2)=O)c1 C(C)(CSC)(C(=O)NCc1ccnn1C)NC(CCC=CC)=O C1(NC(N(CCC)Cc2ccc(OCC)c(OC)c2)=O)CC2CCCCC2O1 C12(CN(c3ccc(NC(=NC)NCC(=O)NC)cc3)CC)CCC(CC1)C2(C)C C(=O)(C#CC1CCCO1)NC1CCN(C(c2ccnc(C)c2C)=O)CC1 C=CCC(C(=O)NCCN1CCN(c2nnc(C(=O)OCC)s2)CC1)NC(C)=O C1(NC(c2cc(C)nc(O)c2)=O)CCSC12CN(c1ncnc(C(C)(C)C)n1)C2 CCCC(CC)CC(=O)NCC1(C)CCN(C(=O)CCSc2ccccc2)CC1 c1(-c2cn(CCOCCC(=O)NC(C)C(C)(C)CO)nn2)cnn2c1NCC2 C(=O)(CC(C)(C)C(=O)c1ccccc1)N1CCN(CC(c2cccs2)OC)CC1 C1(C)(CNC(=O)Nc2sc(C(=O)OC)c(C)n2)CCC(C)C1(C)C C(C(=O)NC(C)C(=O)NC1CCOCC1)(C(C)CC1CCCC1)N1C(C#C)CCC1 CCCCCC(O)C(=O)N1CCCC(CCNC(c2c(C3CC3)cnn2C)=O)C1 CCC(CC)CC(=O)N(C1CC1)CC1CCN(C(C)=O)CC1O.NC N1(C(CCCC#N)=O)CCC2CC2(NC(=O)CSc2cc(Cl)ccc2Cl)CC1 C#CCCC(=O)NC(CNC(=O)C(C)(C)NC(=O)Nc1ccccc1)CC c1(CC)cc(C(=O)N(CC(C)(C)NC(c2sc(C3CC3)nc2C)=O)C)cc(O)n1 C1(=O)CCCCCOC(C)CO1.CC1CC2(C(=O)OC(C)(C)C)CC12 N1(C(C2N(C(c3ccc(C#N)[nH]3)=O)CCCC2)=O)CCCCCCCC1 C1(CNC(C(C=C)(C)O)=O)CN(C(c2ncoc2CC)=O)C2(CCC2)C1 c1(CC2(C(N(C)CC3CCN(C(c4cccs4)=O)C3)=O)CCC2)ccc(F)cc1 C12(C(=O)NCC3C(NC(CNC(CCNC(C)=O)=O)=O)C3)CC(C1)C(C)(C)O2 C#CCC(C)C(=O)NC(C1CCCC1)CNC(=O)CSCC(c1ccncc1)=O C1(C(N(C(C)C(=O)NCC2SCCS2)C)=O)CCCN1C=O c1(C(=O)NC(C2(CNC(=O)CC(C)NC(N)=O)CC2)C)cnc(Cl)c(N)c1 C1(NC(c2n(C)ncc2C(F)(F)F)=O)CC2(C1)CN(C(C1CC3(CC3)CO1)=O)C2 N#Cc1ccccc1N1CCCC(C(=O)NCC2CSCCO2)C1 Cc1cc(C(N2CC(F)(CNC(c3ccc(OCC(N)=O)cc3)=O)C2)=O)oc1C C1(=CC(=O)NCC2CCCC2NC(c2cc[nH]c2)=O)CCOc2ccccc21 C1(NC(C(C)CC2CCCC2)=O)CC12CCN(C(c1ccc(-c3ccco3)[nH]1)=O)C2 c1(CC(N2CC3(C(NC(C(C)C)=O)CCS3)C2)=O)ccc(Cl)cc1[N+](=O)[O-] C1(CNC(c2cscc2F)=O)CCCCN1C(c1conc1C(F)(F)F)=O c1(CC(N2CC3CN(C(C4(CO)CCCC4)=O)CC3C2)=O)ccc2n[nH]cc2c1 N1(C(c2n(C)cnc2)=O)CC2(CCCN(C(C3CC3c3ccccc3Cl)=O)C2)C1 N1(C(CCCOC(C)=O)=O)CCC(C2CC2)C1C(=O)NCCC1(C)N=N1 N1(C(c2nc(C(C)=O)sc2)=O)CCC(NC(c2cc(C)n(C)n2)=O)C1(C)C c1(NCCC2(CNC(c3cn(CC)nc3)=O)CC2)cnc(OC2CCCC2)nc1 C1(CNC(=O)COCCO)CCCN(C(=O)CN2CC3CC3C2)C1 c1(NC(C2C(CNC(C3CC3c3ccccc3)=O)C2)=O)cc(Cl)cc(Cl)n1 C=CCC(C)(C)CC(=O)NC12CCCC1N(C(c1ccn3nccc3c1)=O)CC2 N1(C(CCc2n(C)cnn2)=O)C(CC(=O)NCCn2cnccc2=O)C2CCCC12 Cc1ccncc1C(=O)NCCC1CC(C(=O)NCc2cnccn2)C1 CC(C)CCC(O)C(=O)N1C2CCC1CC(C(N1CC(O)C(O)C1CO)=O)C2 c1(C(N2CC(OCCNC(C3CC(C)(CC)C3)=O)C2)=O)ccc2c(c1)CCO2 C1(C2CCCN(C(=O)CCCN(C)C)C2)(NC(c2n(C)c(S)nc2)=O)CC1 c1(C(C(=O)NCCCOC)N(C(C)CC(C)(C)C)C)ncc(C)cc1Cl CC(CS(C)(=O)=O)C(=O)N1CCC(O)(CCNC(c2cncc(C(N)=O)c2)=O)C1 N1(C(C2C(C)CC(=O)N2)=O)CCN(C(c2ccc3[nH]ccc3n2)=O)CC12CC2 c1(C(C(=O)NCCCF)N(CCCC)C)ccc(OCCOC)cc1 C12(C(N3CC(O)(C(C)NC(=O)CN4CC(N(C)C)C4)C3)=O)CCCC1C2(F)F C(=O)(C(C)C(O)CC)NCC1(CNC(c2ccc(C(=O)NC)nc2)=O)CCC1 c1(CC(=O)NC2(C)CN(C(=O)CCC(F)(F)F)C2)cc(C(F)(F)F)cc(F)c1 C12(C(N3C(C(=O)NC)CC3)=O)CCCC1CCN2C(=O)C(n1cc(C)cn1)C N1(C(c2cc(C#N)[nH]c2)=O)CC2CCN(C(=O)CCc3cccc(F)c3F)CC12 N1(C(c2c(C)oc(Br)c2)=O)CCC(O)(CNC(=O)C=C2CCC(C)C2)CC1 C1(O)(CN(C)C(C2(C(N)=O)CC2)=O)CCN(C(=O)C(F)(F)C2(O)CCC2)CC1 C1(C(=O)NC(C)CCCNC(=O)CCN2CCOCC2)NC(=O)OC1C C(C(C(=O)NC1CC=CC1)NC(C1C=CCS1)=O)OCC C1(NC(c2cc(OC)ncc2)=O)CCN(C(c2ncc(C)cc2OC)=O)CC1C C=CCCCCCC(=O)NN1CCCC1C(=O)NCC1C(C)(C)C1(F)F C1(C2=CCOCC2)(CNc2cc(N3CCCC(CN4C(C)CCC4)C3)ncn2)CC1 N1(C(C2NCCN(C(c3c(OC)ccs3)=O)C2)=O)CC(O)C(O)C(O)C1CO c1(C(=O)Nc2ccccc2N2CC(C)NC(C)C2C)csc2c1CCOC2 CC1(CNC(=O)COCCF)CN(C(C2CCC3(CCC3)C2)=O)CCO1 C(CC(C(=O)N1CCOCC1C(C)O)NC(C1C=CC=CC=C1)=O)=CC N1(C(c2c(C)con2)=O)CCN(C(c2cc(Br)cnc2O)=O)C2CC12 C(=O)(C(F)C(=O)NC1CN(CC)CC1NS(=O)(=O)CCCOC)OCC.C(=O)(COC)N c1(NC2CC(OC)(OC)C2)ccc(S(=O)(=O)NCCOC(F)F)cc1F C(=O)(C1=CCC(C)(C)CC1)N1CCC(C)C(NC(=O)CCc2cnccn2)C1C C1(C(N2C(C)(C(=O)OC)CC2)=O)CCCC(NC(=O)CC(C)c2ccco2)CC1 C#CC1(OC)CCN(CCNC2CC2c2cc(Br)ccc2F)CC1 C1(C(C)C)CN(C(C2CC2C)=O)CCN1C(c1cc(Cl)no1)=O N1(C(C(CC)CCOC)=O)CCC2CC(NC(C3CC3(F)F)=O)CCC2C1 Cn1ncc2c1CN(C(c1csc(NC(c3ccc(O)cc3)=O)n1)=O)CC2 C1(C(N2CCCC(C3N(C(COC(C)=O)=O)CCCC3)C2)=O)C2CC(F)(F)CC12 C(=O)(C(C)(C)c1cncs1)N(CC(O)CN(C)C(C1CCCS1)=O)C N1(C(CCCCCCC)=O)CCCC2CN(C(C3(C)CCN(C)CC3)=O)CCC12 N1(C(c2c(C)cc(CC)o2)=O)CCC(CNC(c2sc(C)cc2OC)=O)C(C)C1 C1(NC(C2CCC(O)CC2)=O)CC12CCN(C(c1cc(Cl)ccc1O)=O)CC2 C1(NC(CCC#C)=O)CCCCCC1NC(=O)COc1ccc(F)cc1Br Cc1c(C(N2CC(O)CC2C(N2CCC3(CCOC3)C2)=O)=O)ccc2c1OCO2 c1(C(=O)OC)cc(NC(=O)C(=O)NC2CC(CS(C)(=O)=O)C2)ccc1Br C(N=c1nc2c(ncn2C)c(NCCC2SCCS2)[nH]1)c1cc(C)cc(C)n1 CN1CCOC(CNC(C2OCCC2NC(=O)CCCn2cncn2)=O)C1 CCCCCCCC(=O)NCc1cc[nH]c1C(=O)NCc1cc(C)ncn1 CCC(C(=O)NC(C(=O)N1CCC1C(C)(C)O)c1ccco1)C(C)C CCCCC(C)(CO)NC(C12CC(CN(C(c3cc(C)c[nH]3)=O)C1)C2)=O C(=O)(C(C)(C)CCCF)N1CC(C(N(OC)C)=O)C(COC)C1 C(CC(C(C)(C)C)NC(=O)CNc1ccc(Cl)cn1)NC(C(C)(C)O)=O c1(C(N(C)CC2CCN(C(C(C(C)C)OCC)=O)C2)=O)sc([N+](=O)[O-])cc1Cl CC(C)(C)CC(CNC(=O)CCNC(=O)NC1CC1)CO N1(C(C(C)(C)N(C)C)=O)CCC(C)(C)C(NC(C2CCCCC2(F)F)=O)C1 c12cc-1on2.O=C(NOCCC1CC1)NC1CC(n2ccnc2)C1 C1(NC(C2CCC(CCC)CC2)=O)CCN(C(c2ncccc2F)=O)CC1F C1(NC(Cc2nc(C(C)(C)C)sc2)=O)CN(C(C2CC23CC3)=O)CC12CCC2 CC1(C)COCC1C(=O)NC1CC1NC(c1ccc(-n2cnnc2)cc1)=O C(C)(C1=NOC2COCC12)NC(C(=O)Nc1ccc(OCCCOC)cc1C)=O C(=O)(C(CC)(CC)CC)N1CC(CCC)C(C(N2CCOC(COC)C2)=O)C1 n1(CCC)ncc(C(=O)N(C)CCN(C(=O)C(=O)NC2CC2)C(C)C)c1Cl C1(NC(C2CC(C)(O)C2)=O)CC(CNC(=O)CN2CCCC2=O)C12CCC2 C1(NC(CN(CC)CC)=O)CC2CCC1CN2C(=O)CCc1cccc(O)n1 C#CCCCC(=O)NCC(C1CC1)NC(=O)Cc1conc1C C1(NC(C2CCC(O)CC2)=O)CC2CC(C1)N(C(c1ccc3sncc3c1)=O)C2 c1(C(N2CCC(NC(C(C(C)C)CO)=O)(CO)CC2)=O)cccc2cncn12 c1(C(=O)NC(C(C)NC(=O)Cc2cc(Br)cs2)C)ccc(Cl)cc1N C12(NC(C3CC(C)(C)C3)=O)CC(C1)N(C(=O)C(=O)NCc1ccc(F)cc1)C2 S(=O)(=O)(c1cnccc1N1CCC(O)CC1(C)C)NCCNCC=C C1(NC(C(C)OCC)=O)CCCN(C(c2ccc(C3CC3)o2)=O)C1CC C1(NC(C2(OC)CCSC2)=O)CN(C(C2SCC=C2C)=O)CC1(C)C n1(CC(=O)NC2(CCNC(CC(C)C3CC3)=O)CC2)cnc2ccccc12 c1(C(N(C2CCN(C(C(C3CCCC3)OC)=O)C2)CCO)=O)cc(C)cnc1C CC(C1CCCc2ccccc21)NC(C1CC1CN)=O c1(-n2c(-c3c(C)ncn3C)nc(Cn3cccn3)n2)nc2ccccc2[nH]1 N1(C(C2CN(C)C(=O)C2)=O)CC(NC(C2(c3ccccc3F)CC2)=O)C(C)(C)C1 C1(C(=O)NC(CNC(c2scc(C)c2)=O)C2CCC2)Cc2c(C)cccc2O1 C(C)(C(=O)N1CCC(C(=O)N(C2CC(OC(C)=O)C2)C)O1)OC N1(C(c2cc(CC)c(C)s2)=O)CC(C)N(C(c2nc(OC)cc(C)n2)=O)CC1C c1(CC(=O)NCC2CCCC2C(F)(F)F)nnc(C(=O)O)s1 c1(NCC2N(C(C(C(C)C)C#N)=O)CCC2)ccnc(S(C)(=O)=O)n1 N1(C(CCSC)=O)CC2CCC2(N(C(=O)CCCCNC(=O)OC(C)(C)C)C)C1 C1(NC(Cn2cc(-c3c(Cl)ccc(OC)c3)nn2)=O)Cc2cccnc2NC1=O C(C1CCCN1C)=CC(=O)NC(C1CN(C(c2coc(C(F)F)c2)=O)CCO1)C Cc1cc(C(F)(F)F)nc(NC(C2CC(NC(=O)OC(C)(C)C)C2)C)n1 c1(OC(C)=O)ccc(Br)c(C(=O)OCCCCc2cccc(Cl)n2)c1 C1(NC(Cc2n[nH]c(=N)s2)=O)CC2(C1)CC(CNC(=O)CC1COCCO1)C2 Cc1oc(Cn2cc(Cc3ccc(OCO)cc3)nn2)cc1Br Cc1ccc([N+](=O)[O-])c(NC2CN(C(c3ccc(O)nc3Cl)=O)CCC2CO)c1 CC(F)(F)CCCC(=O)N1CC(c2ocnc2CNC(c2ccc(Cl)o2)=O)C1 c1(C(=O)NCC2(O)CCCN(C(CCCC(C)=O)=O)C2)c(Cl)nc2sc(C)cn12 c1(C(=O)NC(C2CN(C(C3(C)CC3F)=O)C2)C)nccc2cc[nH]c12 CC1C(NC(C2CCCC3(CC3)C2)=O)C(C)CCN1C(=O)CCc1cn(C)nn1 C1(C(=O)NCCCCNC(c2csc(CO)n2)=O)CCC12CCC2 N1(C(CC(CCCC)NC(=O)C=Cc2ccoc2)=O)Cc2ccc(O)cc2C1 C(c1ccc(F)cc1F)=CC(N1CC2C(NC(C3N(C)CCOC3)=O)(C2)C1)=O CCC(C)C(O)CC(=O)N(C(C)C=CC(=O)N(CC(F)(F)CC)C)C C1(C)(SCCNC(=NCCC)NCCN2CC=CCC2)CCC(F)(F)CC1 c1(C(=O)NCCCN(C(=O)C2=CCCC2)CC)cccc(C(N)=O)c1F n1(C(C(=O)NCCNC(CC2C(C)(C)OCC2)=O)(C)C)cc([N+](=O)[O-])cn1 c1(C(CC)NC(C2CCCO2)=O)cc(-c2cc(OC)ccc2OC)ccc1F C1(NC(c2cncc(CC)c2)=O)CCN(C(c2coc(Cl)n2)=O)CC12CCC2 O=C1NCC2(CN(C(=O)CCC3CC(NC(c4cc[n+]([O-])cc4)=O)C3)C2)N1 c1(CC(N2CC(O)CC(NC(c3cc(C)c(C)s3)=O)C2)=O)ccccc1[N+](=O)[O-] c1(C(N2C(CNC(C(C)=O)=O)COCC2)=O)cc([N+](=O)[O-])ccc1F C1(C(=O)NCCc2ccncn2)CCC(C2CC2)N1C(c1ccnc(O)c1)=O c1(C(=O)NC(CNC(CC(CC)C)=O)(C)CO)cc(C)cc2c1OCC2 Cc1ccnc2nc(C(=O)NC(C)C(C3CCCCC3)NC(=O)C(N)=O)nn12 C1(CNC(=O)C(Cl)=CCl)CCN(C(c2cnc(-c3cccnc3)s2)=O)C12CCC2 C1(CC)CN(N2CC(C)(c3cccs3)C2)CC1c1nccn1C C(=O)(CCCCC(C)=O)NC1CN(C(C=CC=CCC)=O)CC1(F)F N1(C(CC2(C)CCOCC2)=O)CCC2(C=C(C(=O)NCC3(C)CCOCC3)C2)C1 n1(CCC(=O)NCC2C=CCN2C(C2CC2F)=O)ncc(=O)c2ccccc12 c1(C(=O)NCC2CCC(NC(c3csc(Cl)n3)=O)C2)cnc(O)c2ccccc12 C(=O)(C1CCCc2ccccc21)N1CC(NC(c2nn[nH]c2Cl)=O)CC2(C1)CC2 CC1C(NC(=O)Cn2ccccc2=O)CCCN1C(=O)C(O)CN(C)C c1(CNC(C2(CC#C)CC2)=O)cccc(CNC(C2OCCC2C)=O)c1 c1(C(C)=O)ccc(C(=O)NC(C)C(C)NC(=O)CC2CC(N(C)C)C2)cc1F CC1CN(C(C2CCCCN2N=O)=O)CCCN1C(C1CC(S(C)(=O)=O)C1)=O c1(CC(=O)N(CC(CNC(C(C=CCCC)O)=O)C)C)cccnc1C c1(C(=O)Nc2cc(OCC=CC)c(C(C)(C)C)cc2)nc2c(Br)cccc2[nH]1 Cc1cc(=NC(=O)C(c2ccccc2)NCc2nnc3n2CCNC3)[nH]o1 CC1C(C(N2CCC(NC(c3cnn(Cc4ccccc4)c3)=O)C2)=O)CCN1C c1(C(=O)NC(CNC(C(c2ccccc2)NC(COC)=O)=O)C)nccnc1C c1(C(=O)OCC)[nH]c2ccc(Oc3cn(C)nc3C)cc2c1C c1(C(=O)NC2CN(C(CN(CCOC)C)=O)C(C)C2)ncc(OC)nc1OC c1(C(=O)NCC2N(C(CC(COC)O)=O)CCCCC2)ccnc2ncccc12 c1(NC(=O)NCc2ccc(C(C)=O)cc2)c[nH]c2ccc(F)cc12 N1(C(=O)CNCC2(c3ccccc3)CCC2)CCN(CCC2CCCO2)CC1 c1(C(=O)NCC2C3CN(C(c4c(C)cno4)=O)CC32)ccc(Cl)cc1F C(CCC(=O)N(C(C)C(=O)N(C)CCc1ncccn1)C)OC(C)C C1(COCCOCCCC)CCN(C(c2ncccc2C(F)F)=O)CC1C Cc1cc(C)c(C(=O)NC2CC(NC(C3CCC(C(F)F)CC3)=O)C2)cn1 n1(C2C(C)C2)nc(-c2ccc(N3CCCC3)cn2)nc1COC(C1CCCC1)=O C1(C(N2C(CC(=O)NC(c3ccccn3)C)CCC2)=O)CCCN1C=O C1(NC(CC(C)(C)OC)=O)C(C)(C)C(NC(=O)COC)C1(C)C N1(C(C2(CF)CC2)=O)CC2(CCCN(C(C3(CC)CCCO3)=O)C2)C1 Cc1ccc2c(c1)CC(C(=O)NCC1(NC(=O)C#CC3CCCC3)CCC1)S2 C(=O)(CS(=O)(=O)CCOC)NCC(CCCC)NC(=O)CC(C1CC1)C1CC1 CCC(C)C(O)C(=O)NC1CC2CC1N(C(c1cnc(C)s1)=O)C2 C1(CC)C(NC(=O)C(C)CC(N)=O)CCCN1C(=O)CC1CC(C)(C)CO1 C(CCCOC)(C(=O)N1CCOCC(O)C1)NC(C(C)OCC=C)=O C1(CNC2CN(CCOS(C)(=O)=O)C2)CCN(Cc2cccnc2)CC1 c1(C(=O)NCCOCCNC(C(C2CCOCC2)C)=O)cncc2nnn(C)c12 c1(C(N2CC(OCC(=O)NC3CCC(C)(CC)O3)C2)=O)cc([N+](=O)[O-])cn1C c1(C(=O)NCCCCNC(C2C3CCN2CC3)=O)ccc2c(c1)OCC2 C1(C(=O)NCCCCNC(c2c(C(=O)OC)cnn2C)=O)CC(=O)N(OC)C1 N1(CC(=O)NC)CCC2(CCCN(C(c3cnn(-c4ccccc4)c3Br)=O)C2)C1 N1(C(C2=CC(O)C(NC(C3(C)CCSCC3)=O)C2)=O)CCC(O)(C2CC2)CC1 C=C(C)C(CC(=O)NCC(CNC(C1CC(OC)C1)=O)OC)OCC C=CCCCC(C(=O)NCC1CC(C2CC2)=NO1)NC(=O)Cc1c[nH]nc1C c1(C(N2CCCC(C)C2CCNC(=O)CCCCCF)=O)ccc2c(c1)COC2 C(C(=O)NCC(C)C(C)O)(C(C)(C)O)NC(c1c(C)oc(CO)c1)=O c1(C(=O)NC2CC(C)N(C(c3cnsn3)=O)C2)cc(=O)cc(Cl)[nH]1 CC(C)C(CCC(=O)NC1C(O)CC1O)NC(=O)Cc1cncnc1O C1(C(=O)NC2CC(CC)OCC2)CCC2(CCN(C(C3(Cl)CC3)=O)C2)C1 C1(c2nnc(-c3cc(C#N)c[nH]3)o2)(C2CCCO2)CCN(C(=O)COC)CC1 c1(-c2ncn(C)n2)cccc(C(N2CC3(NC(=O)CCCF)CC2C3)=O)c1 C1(c2cn(CCCC(=C)C)nn2)(NC(=O)COC2CCCC(C)C2)CCOCC1 N1(C(CC2C(C)CCO2)=O)CC2CCCN(C(C34CCOC(C)(C3)C4)=O)C2C1 c1(CC(=O)N(CCNC(c2cnc(C(C)C)[nH]2)=O)C2CC2)nc(C)c(C(=O)OC)s1 C12(C(N3CC(NC(C4=C(C)CCC4)=O)C(CO)CC3)=O)CC3CC(CC(C3)C1)C2 CC(C)CC(O)C(=O)NCC1CC(CNC(=O)Cc2cccc(C(C)C)c2)C1 C1(CNC(CC2CCC(C)CC2)=O)CCN(c2cc(F)ncn2)CCC1(F)F C1(C(=O)NC(C)(CO)C2CC2)C2CCN(C(C3CC3(C)C(F)F)=O)CC12 N1(C(c2ccc(CCC=C)cc2)=O)CCC(NC(=O)COCCOC)CC1C c1(OCC(=O)NC(C(C2CC2)OC)C)ccccc1F c1(C(N(C2CN(C(C(CC)O)=O)C2)C)=O)ccc(Br)c(OC)c1 c1(NC(c2cc(C)nc(C)n2)=O)ccc([N+](=O)[O-])c(C)c1.C(=O)OC C(=O)(C1=NNC(C(F)(F)F)C1)N1C2(CCSCC2)C(=O)NCC1.CCOC c1(C(=O)NC23CC(CNC(c4ccoc4)=O)(C2)C3)cc2c(F)cc(F)cc2o1 n1(CC)nc(C(=O)NC2CCCC(CNC(=O)C=CCN(C)C)C2)cc1C1CC1 C1(N(C(c2c(C)nns2)=O)C)CN(C(=O)CCCOCCN(C)C)CC1O C(=O)(CCC(C)(C)NC(C1C(C)(C)C1(C)C)=O)NC(c1ccccc1)C C#CC1(C(=O)N(C)Cc2ccc(F)cc2)CCN(C(=O)C(C)Cn2cccn2)C1 C(c1cccc(F)c1)=CC(=O)NCC(C)CN(C)C(c1ccc(C(C)(C)C)s1)=O N1(C(C2C(C3C(C)C3)C2)=O)CC2CC1CN(C(=O)CN(C)C(c1cccs1)=O)C2 C1(C(C)C)COCCN(C(c2ccc(C(N)=O)o2)=O)C1.C12CN(CCO1)C2 N1(C(C2CC(n3cc(C(C(C)C)N(C)C)nn3)C2)=O)CCCS(=O)(=O)CC1 N1(C(c2cn(CC)nc2)=O)CC(C)C(NC(c2cnn(CCO)c2C)=O)C(C)C1 CN1C(=O)C(c2nc(C(F)F)nn2CCS(N)(=O)=O)Cc2ccccc21 c1(CC)nc(C(C)N(c2ccccc2)C(C2CC2Cl)=O)n[nH]1 C(=O)(CC(C)C(F)F)N1CCCC(N(C(CSC(C)C)=O)C)C1 CC(C)CC(Cc1ccc(F)cc1)N=c1[nH]nc(C2CCCN2)s1 c1(C(=O)NC2CC3CN(C(COCC(=O)NC)=O)C2C3)ccc2nonc2c1 c1(NC(C2CC3(CN(C(c4c(C)n[nH]c4)=O)C3)OC2)=O)ccc2ncccc2c1 C12(C(=O)NCC3N(C(C4CCOC4)=O)CCC3)COCC1CS(=O)(=O)C2 CCCCC(C)CCC(=O)N1CC=CC1(C)C(N1CCCC(C(C)(C)O)C1)=O C(C(C)C(F)C(=O)N1CC2CC2C2CC12)NC(c1ccc(OC)nc1)=O N1(C(C2N(C(C(C)=NOCC#N)=O)CC=CC2)=O)CCC(F)(F)C(O)C1 N1(C(C2CC(=O)NC2)=O)CCC(C2CN(C(C3COCCO3)=O)C2)CC1 C1(CNC(C(C2CC2)OC)=O)CN(C(C2CCCCS2)=O)CC1C(F)(F)F N1(C(C2N(C)CC2)=O)CC(CNC(C2CCC(NC(N)=O)CC2)=O)CC1(C)C C(C(=O)NOCCCNC(C(C)C1CCOC1)=O)OCCC(=O)N(C)C c1(CN2CC(C(=O)NC(COC)COC)OCC2)cc(C(C)(C)C)n(C)c1 c1(NCC2(F)CC(NC(C(C)=C3CC3)=O)C2)ncnc2cccc(C)c12 n1(CCC(=O)NCC(C)(C2CCC2)NC(Cn2c(C)ccn2)=O)ncn(C)c1=O Cc1noc(C)c1-c1cn(C2CC(C(=O)NCC(CCBr)CBr)C2)nn1 C1(CNC(C2N(CC)CCC2)=O)CC2CCC1CN2C(C1CCCO1)=O N1(C(Cc2cn(CC)nc2)=O)C2CCC1CC(CNC(C1C3COCC13)=O)C2 Cc1nc(Cl)c2c(n1)CN(Cc1cccc(-c3nn[nH]n3)c1)CC2 c1(NC(C(CNC(CC2C(C)(C)CCO2)=O)CC2CC2)=O)cccc2c1CCC2 CN(C)S(=O)(=O)N(C)CC(=O)NCCC1(O)CN(C(C2COC(=O)O2)=O)C1 C1(CCOC)CN(C(=O)C=C=C(C)C)CCN1C(=O)C(C1CCOCC1)F Brc1ccc2[nH]nc(N3CC(C4CNCCOC4)C3)c2c1 c1(C(C)C(N2CC3CC2C3NC(=O)CCc2cnccn2)=O)ccc(Cl)c(Cl)c1 C1(CNC(C2(C3CCCO3)CCCC2)=O)CN(C(=O)C=C(Cl)Cl)CC2(CCC2)O1 c1(N2CC(CC=C)(NC(=O)C=CS(C)(=O)=O)C2)cncc(C#N)n1 C=CCC(CNC(=O)CCCC1CC1C)C(=O)N1CC=CCC1COC N1(C(CC2(OC)CC2)=O)CCCC(NC(C2(c3nnc[nH]3)CCC2)=O)CC1 c1(C(N2CCC(CC)C2CNC(C2CCCCC2O)=O)=O)cccc(F)c1C c1(CC(=O)NC(CC(C)C)CNC(=O)CC2(CS(C)(=O)=O)CC2)cn2ccsc2n1 C1(NC(CCC(=O)NC)=O)COCCN(C(C2CC(C)=NO2)=O)C1 C1CC2COCC2C1.C1(C(=O)OCC)(C(=O)OCC)CC1C(=O)NCCOC c1(CC(=O)NC2CC3(C(NC(c4c(N)nccn4)=O)C3)C2)cc(F)cc(F)c1 c1(C(N2C(C3(NC(C(CC#C)(C)C)=O)CC3)CCCC2)=O)cc(F)c(C)cc1O CC(CC(C)(F)F)C(=O)NCC1(C)CCN(C(c2cnc(O)c(F)c2)=O)CC1 C1(C(C)C)(C(=O)NC(CO)c2ncc[nH]2)CCN(C(=O)C(O)CC2CC2)C1 C12(C(N(CCCNC(C3(C)C(CC)CCC3)=O)C)=O)CCOC(C)(C1)C2 CN1CCCCC12CCN(C(c1cccc(NC(C3CCCCC3)=O)c1)=O)CC2 c1(CNC(C(C)SC(C)C)=O)ccc(NC(C2(C(N)=O)CC2)=O)nc1 c1(OC)nccnc1C(=O)NCC(C)CC(=O)NC1(c2cc[nH]n2)CC1 C1(CNC(c2c(C)nn(C(C)C)c2)=O)CCN(C(=O)CC2CC(F)C2)C1(C)C C(=O)(CCCCCO)NC1CCC(CNC(CCOC)=O)C1.C1C(=O)O1 c1(NC(CCCc2c(C)cc(Br)cc2)=O)nc2ccncc2n1C N#Cc1ccc(C(N2CC3CC2CN3C(c2cc(Br)c(O)cc2F)=O)=O)c(Br)c1 c1(C(N2CCC(C3CC(CN)C3)CC(F)C2)=O)ccc(SC)cc1[N+](=O)[O-].C(=O)OC N1(C(CC(CC)OC)=O)CCC(C2CCN(C(C3CCOC3)=O)CC2)C1 c1(C(N2CCC(F)(CNC(CCC=C(C)C)=O)C2)=O)cc(F)cc2c1NCCC2 CS(=O)(=O)C1CCCN(Cc2cc(=NCc3cc(F)ccc3F)[nH]cn2)C1 N1(C(c2ncc(CC)s2)=O)CCOc2cc([N+](=O)[O-])ccc2C1 C1(F)(C(N(C)C)=O)CCN(C(c2cccc(-c3cccc(CO)c3)c2)=O)C1 c1(C(=O)NCC2OCCN(C(CCNC(=O)CO)=O)C2)cccc2c1COCC2 CCC(COC)C(=O)NC(CNC(C1(OC)CCSCC1)=O)CCOC C1(=O)CC(O)CN1.c1(C(N(CC)CC)=O)cn(C2CC2)nc1C(C)C.C(C)(C)(C)CO N1(C(C2(C)CCC2)=O)CCCC(C(=O)NCC2CC(O)C2(C)C)C1 CCCCC(CC)C(=O)NCC1(C)CCN(C(=O)C(C)(C)C2CCOCC2)C1 N1(CC)CCOCC1C(=O)NCCCCC(C)NC(c1ccc(C(F)F)o1)=O c1(C(=O)NCCCCCNC(C(COC)(C)OC)=O)cnc2nc(C)oc2c1 c1(C(C)C)nc(=NC2CC(CNC(=O)C3=CC4(CCOC4)C3)C2)s[nH]1 C1(c2nnnn2C(C)C(NCP(OCC)(C)=O)=O)(OC)CCN(C(C)=O)CC1 c1(CC)nccnc1C(=O)NC(CNC(=O)C(F)CC)Cc1ccccc1 N1(C(c2sc3ncn(C)c3c2)=O)CCC2CN(C(=O)CN3CCCCC3)CC2C1 Cc1cccc(N2CCC(OC(=O)CC3CC(C)OC3C)C2=O)c1 N1(C(CC2CC(NC(C=CC(C)(C)C)=O)C2)=O)CCC(CC2CCCCC2)C1 C1(CN=[N+]=[N-])CCCN(C(C2CCCCN2C(=O)C=CC2CCCC2)=O)C1 CN1CC(C(=O)NCCCCC2CN(C(c3cccn3C)=O)C2)NC1=O CON(CCCO)C(=O)C1(NC(=O)CN2CCCCC2)CC1(C)C c1(C(=O)OC)[nH]c(C)c(C(=O)NCCNC2(C)CCCC2O)c1C N1(C(c2c(C(C)C)con2)=O)CCC(C)N(C(c2conc2C)=O)CC1 Cc1cn2c(C(=O)N(C)CC3COCCN3C(c3cnn[nH]3)=O)cnc2s1 N1(C(Cc2c(C)ocn2)=O)CCCC12CCN(C(C13CCCC1C3)=O)CC2 C1(NC(C(=O)Nc2ccc(N(C)C)nc2)=O)CCC2(CC1)OCc1ccccc12 Cc1ccc(C)c(C(N2CC3(NC(C4CCCOC4)=O)CCC2C3)=O)c1O N1(C(C(c2ccccc2)OC)=O)CC(NC(c2ccoc2Br)=O)CC(O)C1 c1(C(=O)NC2CCC2CNC(=O)C(O)c2ccsc2)ccccc1N1CCCC1 N1(C(C(CCCC=C)NC(=O)CNC(=O)C(C)CC)=O)CCc2oc(C)nc2C1 Cn1cc(C(=O)NCC(CNC(=O)Cc2cccn2C)CO)nn1 c1(C(N2CC(C)(c3ccccc3F)OCC2)=O)ccc2cccc([N+](=O)[O-])c2n1 N1(C(C2C(C=C)C2)=O)CCCC(CCNC(=O)COCCOCC)C1 C(=O)(CCCCCC(C)O)NCC1(Cn2cc(C(CC)OC)nn2)CCOCC1 C1(C(=O)NCCCCSC)N(C(C2CCC(F)(F)C2)=O)CCC1(C)C CC1(C)CC(NC(C2CC2(C)C)=O)CN(C(c2ccc(CCN(C)C)cc2)=O)C1 N1(C(c2cn(CCC)nn2)=O)CCOC(C(=O)Nc2cnn(CC(N)=O)c2)CC1 N1(C(C(CC(=O)OC)NC(=O)COC(C)=O)=O)CC(CO)C2CCCC12 C(=O)(CCC(=O)Nc1cccs1)N1CC(n2cc(NCc3c(C)nsc3)nn2)C1 C(=O)(C1=CN=C2N=CNN2C1)NCC(C)NC(c1c[nH]c2nccc-2c1)=O c1(C(=O)NCC(CC)NC(C2(C#N)CC3CC3C2)=O)c(F)ccc(C)c1F c1(CC(C)NC(=O)C(=O)NCC23CCN(CC2)CC3)c(F)cccc1F c1(C(=O)NC(C)C(C)NC(=O)CNC(=O)Cc2cnns2)nnc(S)s1 CCC(CC)C(C(=O)N1CC(NC(c2nc(O)c(C)s2)=O)C(C)(C)C1)OC c1(C(C(C)NC(C(CC)O)=O)OC)cccc(Br)c1 c1(NC(C23CC(C(=O)OC)(C2)C3)=O)ccc(C)cc1SC.C12(C(=O)N)CC(C)(CO1)C2 CN1CCN(C(C2CCCC(C#N)C2)=O)CC1CNC(=O)Cc1cnc[nH]1 CCCCC(CC)CCCN(C)C(=O)NC(c1cccs1)CN1CCOCC1 N1(C(C2CCCN(CC=CC)C2)=O)CCCN(Cc2ccc(F)nc2F)CC1 c1(C(C)C)ccc(C(N2CC(NC(=O)Cc3nc[nH]n3)C2)=O)cc1Br c1(OC)cccc(C(N2CCC(C)(NC(=O)CC3(O)CCC3)C2)=O)c1 N1(C(C(C)(CO)OC)=O)CCOCC(C)(CNC(=O)C=Cc2ccnn2C)C1 c1(C(N2CCC(NC(C3C(=C)C3)=O)(CO)CC2)=O)occ2c1CCOC2 c1(C(=O)NCC(CC)NC(=O)CCc2nc(O)n[nH]2)cc2c(o1)CCCNC2=O c1(C(=O)NCCOCCNC(CC(=O)NCC#C)=O)ccc(C(F)F)cc1 N1(C(C2(COC)CCC2)=O)CCC(CC(C)NC(c2cc(Cl)ccn2)=O)CC1 c1(C(c2nnnn2C2CC2)NCC(C2CC2)SC)cccc(C2CC2)c1 c1(C(N2CCCC(NC(COCCOCC#C)=O)C2)=O)ccc([N+](=O)[O-])cc1 C1(C(N(CC(C)CNC(c2cnc(S)[nH]2)=O)C)=O)CC2(C1)CC(O)C2 C1(CC(=O)N(C)CC2CCCN(C(=O)CCS(C)=O)C2)CC2CCC(C1)C2 c1(OC(CC)C)ccc(C(=O)NCC2CN(Cc3c(C)noc3C)CCO2)cc1 C(=O)(C(CC(C)C)NC(=O)CC(C)N(C)C(c1cc(F)n(C)n1)=O)NC c1(C(N2CCN(C(=O)CCc3ccon3)C(C3CC3)C2)=O)cccn2cnnc12 C(=O)(CC(CC)CCC)NCC(CN(C(c1cnc(CCCC)s1)=O)C)C N1(C(c2c(OC)ccs2)=O)CCCN(C(=O)C(C)C(C)C)CCNC1 CCC(Cc1cccc(C)c1)C(=O)NC1(COC)CCN(C(=O)C(OC)OC)C1 c1(C(=O)NC2C(N(C(c3cc(OC)nn3C)=O)C)CCCC2)cnc2n1CCS2 CCC(CC)C(C(=O)NC)N1CCCC1CNC(c1sccc1C#N)=O N1(C(N2C(C)C(N3CCOCC3)CC2)=O)CCC(S(=O)(=O)c2ccccc2)C1 C1(CC)CCCCC1C(N1CCC(CO)(CNC(=O)C(C)SC(F)(F)F)C1)=O C(CC(CNC(C1C=C(C)CS1)=O)NC(=O)CSCCC#N)OC N1(C(C2N(c3c(Br)cnc(C)n3)CCC(O)C2)=O)CCC2COCC2C1 N1(C(C2C(C)CC2)=O)CCC2(CC1)CCN(C(c1cncc(N)c1)=O)C2 C1(F)(CNC(CCSCC(C)C)=O)CCCN(C(C2CC(C)(C)CO2)=O)C1 CCCCCCCC(=O)N(C)CCC1CCCCN1C(C1CC(=O)CCO1)=O c1(OCC)ccc2c(c1)CC(C(=O)NC1CCC1NC(=O)C(C)(CC)OC)CO2 C1(C(=O)COC(C2(Cl)CC2)=O)CCC(Cc2ccccc2)C1 c1(C(N2CC(OCC)C(CNC(C3CC=CC3)=O)C2)=O)ccc2nncn2c1 c1(CCNC(C(=O)NC(CC(=O)OC)c2ccccc2)=O)ccc2ncsc2c1 C(=O)(C#CC1CCCOC1)N1CCCC(CNC(C=C(C)Cl)=O)CC1 N1(C(CCc2n(C)ccc2)=O)CC(O)CCC1C(=O)NCC1OC(=O)CC1(C)C CC(c1cccnc1)=CC(N1CCC(CF)(NC(C2CC2C(N)=O)=O)C1)=O C1(NC(c2ccc(-n3cnnc3)cc2)=O)CCCC(NC(C23CCC2CC3)=O)C1 CC1(C)CC1(C#N)CNC(C1(n2cc(Br)nn2)CC1)=O C1(C(N2CCC(C(F)F)(CNC(CP(C)(C)=O)=O)C2)=O)CCCCC12OCCO2 c1(CCC)cc(C(=O)NC(C2CCCN2C(C2C=CCCC2)=O)C)n(C)n1 O=C1NCc2ccc(C(=O)NC3(CF)CCN(C(C4CC4F)=O)C3)cc2N1 CCC(CCO)C(C)NC(=O)NC1C2CC1(c1cccc(C(F)(F)F)c1)CO2 O=C(C#CC1CCCC1)NCC1CC1NC(C12CCN(CC1)C2)=O N1(C(C2C(C)CCCC2)=O)CCC(C)C(CNC(C2CCC3CC3C2)=O)C1 C#Cc1ccc(CC(N2CC(O)(CNC(C3(C)CC(O)CN3C)=O)C2)=O)cc1 c1(C(=O)NCC(CNC(C2CC(C)(F)C2)=O)OC)ccc(N(C)C)c(F)c1 c1(OC)ccc(Br)c(C(=O)NC2CCC(NCc3cnc(Cl)cc3Br)C2)c1F c1(C(=O)NCC2CC(NC)C2)cnc(C)cn1.C1C(F)C(=O)N1.N(CC)(CC)CC O=C(CC1CCOc2ccccc21)OCC1(c2ccccc2)CC1(F)F C1(CNC(C2N(CC)CC2)=O)CCC(C(=O)NCCCCC2CC2C)O1 CN1C2CCCC1CN(C(C(=O)NCC1CC3CC1C1CC31)=O)CC2 CC1=CCN(C(C2(NC(=O)CC3CCCC3C)CC(F)(F)C2)=O)CC1 C1(CN(C(c2ccc(Cl)cc2)CCC=C)C=O)CCOC(C)(C)C1 c1(CC)cc(OC(C)C)ccc1CNCc1ccc(C)n1C N1(C(=O)Cc2cnsc2)CC2=C(C1)CN(C(=O)Cc1ccc(Cl)cc1F)C2 N1(C(c2cn(CCC(C)C)nn2)=O)CCC(NC(c2sccc2F)=O)C12CC2 c1(NC)cnc(Cl)cc1C(N1CCN(C(=O)CCOCCOC)CC1C1CC1)=O c1(N2CCCC(C)(OC)C2)ncccc1S(=O)(=O)NCc1cc2sccc2n1C C1(CC)CCCN(C(C2CC(O)CN2C)=O)C1C(=O)NCC1CCN(C)C1 N1(C(C(F)=CCC)=O)CCN(C(=O)COC(c2cccc(OC)c2)=O)CC1CC C(=O)(C1CCCc2c1ncn2C)N1CC(CNC(C(C)=C(C)C)=O)CC12CCC2 c1(C(N(N(C(=O)CS)C)CCOC)=O)cnc(O)c(F)c1.C1(OCC)CC(N)C1 O=C1CSCC(C(=O)NC2CC2C(=O)NCCc2ccnc(O)c2)N1 c1(NCc2c(C(=O)OC)cccc2F)ccc2[nH]c(=O)c(=O)[nH]c2c1 c1(-n2cc(C3(O)CN(C(c4ccc(F)c(Cl)c4)=O)C3)nn2)ncnc2c1OCCO2 C1(C(N2CCC(CCC(=O)NCC3=NOC(C)C3)CC2)=O)CCC2(CCC2)C1 C1(C(=O)NC(C2CC(NC(C3CC3c3cccs3)=O)C2)C)C=CCC1 n1(C(C)C(=O)NCCC2(CNC(=O)C(=O)NCCC(N)=O)CC2)cnc(C#N)n1 CC(CCCNC(=O)CCNC(=O)CN(C1CCSC1)C)N(C)C N(C1CCOc2c(Cl)cc(Cl)cc21)C(C(=O)Nc1cccc(Br)c1)=O N1(C(C(C)=C(CC)C)=O)CCC2(CC1)CC(C)N(C(C1CC(C)(CC)C1)=O)C2 C1(C#N)(CC)CCN(C(=O)C(O)CNC(=O)CC2CC(C)C2)CC1 c1(CC)ccc(C(=O)NCC(CC)NC(c2nc(C)ncc2OC)=O)c(OC)c1 O=C(C(CN1C(=O)NC(C2CC2)C1=O)CCc1ccccc1)Nc1cc(CO)cc(F)c1 Cc1cc([N+](=O)[O-])nn1C(C)C(=O)N(CC(C)(C)O)C1CCOC1 N1(C(c2c(CC)c[nH]n2)=O)CCOCC(NC(c2oc(C3CCC3)nc2C)=O)C1 C(=O)(C(C)C(C)NC(=O)CCOC)N(CC=C)C c1(C(=O)NCC2C(C(=O)NC(CCC)C)OCC2)cc(CC)nn1C C1(c2nnnn2CC)(NCc2cn(CC)nc2)CCN(Cc2ccccc2)C(C)C1 C(=O)(C(O)(C(F)(F)F)c1ccccc1)N1CCN(C(c2n(C)ccc2)=O)CC1 C1(NC(COCC=C)=O)CC(NC(=O)C(C)Cc2ccnn2C)CC1O c1(C(N2CCC(N(C(C(C(C)O)N(C)C)=O)C)C2)=O)ccc(CO)c(F)c1 c1(C(N(C)CC2N(C(C(CCCC)O)=O)CCOC2)=O)c(F)ccc(C)c1Cl N1(C(C(CC(=C)Cl)NC(c2noc(CC)c2C)=O)=O)CCC2(CCC(O)C2)C1 C1(NC(c2c(CNC(C(C)CC#N)=O)nccc2)=O)CC12CCCCCC2 N1(C(CC2(OC)CCC2)=O)CCOCC(CNC(C2CC(C(C)C)=NO2)=O)C1 Cc1ccc(Br)c(C(=O)NC2CCCC2CNC(c2cc(Cl)no2)=O)c1 c1(C(N2C(C(=O)OCC)C=CC2)=O)ccc(Br)cc1Oc1ccccc1 Cc1nc(O)ccc1C(=O)NC(C)(C)CN(C(=O)CC1C=NN(C)C1=O)C c1(N2CC(c3ccc(C)s3)OCC2)nc(=NC(C)CCO)[nH]c2ncn(C)c12 Cc1cc(C(=O)Nc2cccc(NC(=O)C=C3CCN(C)C3)c2)c(Cl)cc1Cl C(N=C(NCC1(c2ccccc2F)CC1)NC1CCN(C(C)CC)CC1)CCC=C CCC(C)CCCCC(=O)N1CCCC(Cc2cn(Cc3cnns3)nn2)C1 CCC(CCOC1CCOC1)C(=O)N1C(C(=O)OOCBr)COc2ccccc2O1 c1(CCC(=O)NCC(CN(C)C(C2(C)CSC2)=O)O)ccc(Cl)cc1F N1(C(C2CCN(C(N)=O)CC2)=O)CCN(C(c2c[nH]nc2F)=O)C2COCC12 CC1CN(C(=O)C(c2ccc(Br)cc2)NC(=O)OC(C)(C)C)CC(C)(C)C1 N1(C(C2CN(C(C)=O)C2)=O)CCCC(C)(C)C1C(=O)NC1(C(=O)OC)CC(O)C1 C1(CNC(=O)CC2CC3(CC3)CO2)CN(C(=O)CC23CCC(CC2)C3)C2(CCC2)C1 c1(C(N(C2COC2)CC)=O)cnc2c(c1)CCN(Cc1cnc(OC)c(Cl)c1)C2 c1(CNC(COCC#C)=O)ncccc1C(=O)OC1(CCCC)CC1 c1(NC(C(N2CC3C(c4cc(C)[nH]n4)CC(C3)C2)=O)=O)n[nH]c2ccc(F)cc12 N1(C(c2cnn(CC)c2C)=O)CCN(C(=O)Cc2cc(OC)cc(F)c2)C(C)C1 c1(C(=O)NC(C2CCCCC2)C(C)NC(=O)CCF)sccc1Cl N1(C(c2c(C)nco2)=O)CC(NC(C2CC(=O)N(C)C2)=O)C2CC2C1 Cc1nccn1CC(C)CN1CCC1C(=O)NCCCc1nncn1C C(=O)(C(CNC(=O)CCc1cn[nH]c1)N(C)C)NC(C1CCOCC1)C#C c1(C(=O)NC2CC(NC(c3nc(C(C)(C)C)oc3)=O)C2)ncc(Br)cc1N Cc1cc(C)n2nc(C(=O)N(C)Cc3cn(CC4CCCCC4O)nn3)nc2n1 c1(C(N2CCCC2CCNC(C2CCC(O)C2)=O)=O)n[nH]c2cccnc12 c1(C(=O)NCC2CC(NC(=O)CC3CC3(Cl)Cl)C2)cccc2c1CCO2 N1(C(c2c(CC)cc[nH]2)=O)CCCCCCC1C(=O)N(C1COCC1OC)C C(=O)(CCCCCC(c1nnnn1C)NC(C(C)CC(=O)OC)C1CC1)OC N1(C(CNC(=O)C2CC2)=O)CC2CC(Nc3ncc(Cl)cn3)CC1C2 C#Cc1ccnc(NC(=O)C(C)OC(=O)C(COC)OC)c1 Cc1cc(CNC(C2C=CCS2)=O)oc1C(N1CCC(c2ccco2)C1)=O C12(C(=O)NC(C3CCN(c4ncc(C(=O)OC)nc4)C3)C)CCCC(C1)OC2 C1(CNC(C(CC)NC(C)=O)=O)CN(C(c2ccc(N)c(O)c2)=O)CCC1(C)C CCCC(C)(O)C(=O)N1CCC(C)(CNC(c2cc(F)ccc2C(F)F)=O)C1 C=Cc1cc(C(=O)N(C2CCCCN(C(=O)C3=CCCCC3C)C2)C)cc(F)c1 CC(C)CC(C(=O)C(=O)CC1CC2(CC2)CO1)NC(N)=O.C(CNC1CC1)N CC(C)C(O)CC(=O)NC(C)CC(=O)NCCCc1ncccn1 C1(C(=O)OC)C(C)OCCN1C(c1cn(-c2cccc(Cl)c2)nn1)=O C12(CNC(=O)CSCC3CCCCO3)CCC(CC1)N2C(C1CC1F)=O CCC(C)(F)C(=O)N1CCC(OCCn2cc(-c3cc(Br)cs3)nn2)C1 C1(CNC(CC(=C)C)=O)CC2CCC(C1)N2C(C1CC1c1ccc(C)cc1)=O Cc1[nH]c2cccnc2c1CNC1CCN(CCC(C)C)CC1 N1(C(C=Cc2c(C)nccc2)=O)CCC2(CC1)CN(C(C1CC3(CCC3)C1)=O)C2 N1(C(c2ncc(C)nc2)=O)CC(F)(F)CC1CNC(c1ncc(Br)cc1F)=O C(=O)(CCCCCN(C(=O)CC1(OCC)CC1)C)N1C(CCC)CCC1 Cc1cc(CC(C)NC(=O)C(C)CN(C)C(c2scnc2Cl)=O)n[nH]1 C12(NC(=O)CCOCC3CC3)CC(NC(=O)CCc3cscn3)(C1)C2 c1(C(=O)Nc2ccc(-c3cccc(O)c3)cn2)c[nH]c2cc(Cl)ccc12 c1(OC)ccc2c(c1)CCC(NC(=O)NCCNC(=O)NC1CCCC1O)C2 c1(C(=O)OC)ccc(COC(c2[nH]nnc2Cc2ccc(Br)cc2)=O)cc1Cl c1(CNC(C(CC)(C)C)=O)cc2n(n1)CCN(C(=O)C(=O)NCCNC(C)=O)C2 C=CC(C)C(=O)NCC=CC(=O)N(CCCC(C)O)C C1(C)(C(=O)NCCN(C)C(c2ccc(NC=O)cc2)=O)CC2CC2C1 N1(Cc2cn(CC)nc2)c2ccccc2CC1C(N1CCC(O)C(C(=O)OC)C1)=O C1C(C)(C)CNC(=O)C(=O)N1CC.c1(C(=O)NC)cnc(CC2CC2)s1 C(CC(C)(C)C(=O)N(CCCNC(c1cccc(-c2nc(O)n[nH]2)c1)=O)C)OC N1(C(CCCC(CCC)C2CCCCC2)=O)CC(=O)N2CCCC2C1 C12(CCNC(c3c(C)cnn3C)=O)CCC(CC1)N(C(=O)COC1CCC1)C2 N(C1COc2cc(Cl)ccc21)C(=O)NCC.C1(OCCl)CC2(CC2)C1 S(=O)(=O)(c1ccc(CBr)s1)N1CC(C(N(C)Cc2noc(C)n2)=O)C(O)CC1.CN C(=O)(N(C)OCc1ccccc1)C1(CNC(=O)CC2CC2(C)C)CCC1 CC1CC(CCNC(c2ccnnc2)=O)CCN1C(=O)CNc1ccc(Cl)nc1 N1(C(c2c(CC)cccc2)=O)CCC(F)CC1C(=O)NCCCP(C)(C)=O C1(C(N2CCCC(CNCc3cncc(-n4cccc4)c3)C2)=O)CCCC1(F)F N1(C(C=CC=CCC)=O)CC2(CCCC2NC(C2Cc3nnc(C)n3C2)=O)C1 C1(CCO)(N)CNC1.c1(C(C(=O)C=CC2CC2)=O)cnccn1 c1(C(=O)NC(c2cc(Cl)ccc2Cl)CC)ccc(C2CC2)nc1O N1(C(C2C(C)OC(C)C2)=O)CCCOC(CNC(=O)C=CCF)C1 c1(C(=O)NCCCC(F)F)cccc2cc(F)ccc12 C(=O)(C(C)CC(C)C(C)=O)NCCCOCCNC(C(CN(C)C)C(C)(C)C)=O c1(C(N(CC(C)NC(=O)C(O)Cc2ccccc2)C)=O)cccc2c1NCCC2 C1(NC(C2N(C(C)=O)CCOC2)=O)CCN(C(c2ccc(F)cn2)=O)C1(C)C c1(C2C(=O)N2)cc(Cl)c(OC)cc1Cl.C1(NC(COC)=O)CCNC(=O)C1 C1(NC(CCc2c(C)nn(C)c2)=O)CN(C(=O)CC2CCCC(=O)C2)CC1(C)C N1(C(C2C(CCOC)C2)=O)C2CCC1CC(NC(c1ccccc1S(C)=O)=O)C2 C1(C(=O)OC)CCN(C(=O)CC2CCN2C(C2CC3CCCC3C2)=O)O1 C(=O)(C(F)C(F)(F)F)N1C(CNC(C(C=C)C)=O)CCC1 C(=O)(C(COC)CC(C)C)N1CCC(O)(CCNC(CC(C=C)(C)C)=O)C1 N1(C(C=NOC)=O)CCC(F)(F)C(CNC(c2cc(C(N)=O)cn2C)=O)C1 Nc1cc(C(F)(F)F)ccc1C(=O)NCCCNC(=O)C(O)CF O=C(C1=CCCOCC1)NC1CC(NC(c2ccc3c[nH]nc3c2)=O)C12CCC2 c1(C(=O)NC)nc(C)oc1OC.c1(CCCCC)cc(CC)n[nH]1.C12CC1CC(=O)NC2.CC N1(C(C2CCC(C)O2)=O)CCCC(C2CC2NC(c2nnc(C(F)(F)F)s2)=O)C1 Cc1nnc2n1CCC(C(=O)NCC(C)NC(=O)CCN1CCCC1)C2 c1(C(N(C2CN(C(COc3ccc(C)cc3)=O)C2)C)=O)ccc([N+](=O)[O-])cc1F c1(OC)c(C(=O)NC2C3CC2N(C(c2ccc(C4CC4)cc2)=O)C3)cccc1Cl Cc1ccccc1C(C)(C)C(=O)NCC(O)CNC(C1CC1(C)Br)=O N1(C(C(CC)SC)=O)CCOC2CCN(C(=O)CNc3cccc[n+]3[O-])CC12 c1(OCC(=O)NC2CCN(Cc3cn(CC=C)nc3)C2)c(F)cccc1F Cc1cn2c(CC(N3CCOC(C(=O)NC4(c5cnn[nH]5)CC4)C3)=O)csc2n1 C(=O)(C(C)(C)CNC(c1cnnn1C)=O)N(C1CCCC1C(=O)O)C C(C1=NOCC1)(c1nnnn1C1CCOCC1)NCCCNC(=O)OC CCC(CC)CCCC(=O)NCC1CCCN1C(C1(c2ccncc2F)CC1)=O C1(C#N)(CC)CCN(C(=O)CC2(NC(C3CC4(CCO3)CC4)=O)CCC2)CC1 c1(C(=O)NC(CC)CNC(=O)CCC#N)ccc(C2CCC(=O)N2)cc1 CC(C)C(O)C(=O)NCC1CCCN1C(C12CC(CCO1)C2)=O c1(C(=O)NC2CCN(C(C3CC34CC4)=O)C2)nnn(C2CC2)c1C(F)(F)F C1(C(N(CCC(=O)NC(c2cnn(C)c2)CO)CC=C)=O)CC=C(C)CC1 C(=O)(CCCCCc1nn[nH]n1)NC1CCN(CCOC)C1 c1(C(=O)NCC2(C)CC(NC(c3nscc3Br)=O)C2)coc(C#N)c1 c1(C(=O)Nc2ccc(-c3cnc(C4CC4)nc3)nc2)ccc2c(c1)OCO2 CC1CCC(CC(N2CC(CC(F)C(=O)NC3CCN(C)C3)C2)=O)OC1 c1(C(N2C(C)(CNC(C(CC)NC(N)=O)=O)CCC2)=O)cnc2ncccn12 CC1CN(C(=O)CCc2cscn2)CC1CNC(c1cccc(C2CC2)c1)=O CC(CC(=O)NC(C)CC1CN(C(=O)COc2ccccc2O)C1)CC(F)(F)F c1(N2CC=C(C)C2)nc(=N)[nH]c(=NC2CC2CCn2ccnc2)[nH]1 c1(COC)cncc(C(=O)NC(C(=O)N2CC(N3CC(F)C3)C2)C2CC2)c1 C1(NC(c2n(C)cnc2)=O)CN(C(c2ccnn2C2CCOCC2)=O)C(C)(C)C1 C1(c2c(C)c(Br)ccc2)CCC2(CC1)CNC(=O)C2 N1(C(c2n(C)ncc2)=O)CCC(C)(C)C1CC(=O)NCC1CC12CCCCC2 N1(C(CN2CCC(C(N)=O)CC2)=O)CCC(NC(=O)CC2CC2(Cl)Cl)C(C)(C)C1 C1(CC(N2CC(C(C(=O)N(C(CN(C(C)=O)C)C)C)O)C2)=O)CC(C2CC2)C1 c1(-c2cccc(OC)c2C)ccc2cc(C(N3CCC(C)C3)=O)cn2c1 C1(C(N2CC3C(CNC(c4[nH]cc(CC)c4)=O)(C3)C2)=O)CS(=O)(=O)CCO1 C1(NC(C=CCN(C)CC)=O)CN(C(=O)CC(C)(C)CN(C)C)C2CCCC12 c1(OC)ccc2c(C(=O)NCCCN(C3CC3)CC34CCCC3C4)c[nH]c2c1 N1(C(C2=CC(C)(C)C2)=O)CCC2(CC2)CC1C(=O)NC(Cc1ccco1)CO CCCC(O)(CCC)CC(=O)N1CC2CCC(CNC(c3cc(C)co3)=O)C2C1 Cc1nc(C=CC(N2CCC(NC(C3(P(C)(C)=O)CC3)=O)C(F)C2)=O)[nH]c1C C1(C(N2C(CCNC(c3c(C(C)(C)C)ocn3)=O)CCC2)=O)CC2(C1)CC2(F)F C1(NC(C2C3CCCC23)=O)CCN(C(=O)Cc2ccco2)C12CCC2 c1(OC)c(C(=O)N(C)CC2CN(C(=O)CC(O)C(C)C)C2)cccc1Cl n1(CC(=O)NC)ccc2c(OC3CCC3)cccc12.c12ccc(cc1)[nH]c2=O O(P(C)(=O)CNC(=O)C(C)N(C(=O)CCn1cc(C)cn1)C(C)C)CC N1(C(C(C)(F)F)=O)Cc2ccccc2C(NC(C2CCC=CCCC2)=O)C1 N1(NC(C2(CC)CCN(C(CNC(=O)OCC)=O)C2)=O)CCc2ncncc2C1 n1(CC)nncc1C(=O)NC(C1CCN(C(=O)C(F)=CC2CC2)C1)(C)C C(=O)(CC(CN(C)C)C(F)(F)F)NC12CC(CO)(C1)C2.C12(CCC1)C(=O)N2.CCOC C1(C(=O)Nc2c(CC)cccc2)CCN(C(=O)CCCCCNC(C)=O)C(C)C1 N1(C(C2N(CCC)CCC2)=O)C2CCC1C(CNC(c1ccncc1F)=O)C2 CCC(C)(C)C(O)C(=O)N1CCC(F)(CNC(=O)CC23CC(C(=O)O)(C2)C3)CC1 CC(CN=C(NCC1CC1)NC1CC1)N(c1cc(OC(F)F)ccc1F)C CC1CNCCN(C(=O)CC2CC(F)CN2C(=O)CNC(C2CCCC2)=O)C1 N1(C(C2CC(OCC)C2)=O)CCCCC1C1CCOC1.C1(=O)CCCN1 C(CC(C)C(=O)NCc1cc(C(N2CCSC3CC23)=O)cs1)=CCC c1(C(N2CCCCC(NC(CCCCCC)=O)C2)=O)cc(F)c(O)c(F)c1 C(CNC(=O)CCOC1CC1)(C(C)C(C)C)NC(C1(SC)CC=CC1)=O c1(NC(C(CNC(CC2(CC)CCC2)=O)N(C)C)=O)ccc(O)cc1F C(=O)(CCCCCN(C(=O)C=CC1CCOCC1)C)NC(C=C)C(F)(F)F c1(C(N2C(CNC(C=CC(=O)OCCCC)=O)CCC2)=O)cccc(C#N)c1 S(=O)(=O)(c1cccc(Cl)c1F)N1CC(OC)C(NC(C2CCCC(C)C2)=O)CC1 N1(C2(N(C)C)CCC2)CCC(OCCn2cc(-c3cccc(Br)c3)nn2)C1=O C1(NC(=O)CNC(C2CCCC2)=O)CCCC1CNC(C1C=CCC1)=O Cc1c(CC(=O)NCC2CC2NC(c2ncn(C)n2)=O)ncn1C N1(C(c2c(C)scn2)=O)CCCCC(CNC(c2ccc(=N)[nH]n2)=O)C1 C1(C(=O)NC(C2CCCCC2)CNC(CC=C(C)C)=O)CCCC(=O)N1C C(=O)(C1=C(C#N)CCC1)NCCC(CNC(=O)CC1CC2CCC1C2)OC c1(C(=O)NC2CCC(OC)C2)cccc(NCc2ccccc2I)c1 CCC(CC)C(F)C(=O)N(C1(CC(=O)N(C2COCC2(C)C)C)CC1)C N1(c2c(C#N)ccc(C(F)F)n2)CCc2cc(F)ccc2C1 CC(CC(=O)NCC1(CNC(c2ocnc2C(F)F)=O)CCCC1)P(C)(C)=O CN1CC2CCC(C1)N2C(C12CC(C(=O)Nc3c(O)ccc(F)c3F)(C1)C2)=O C1(CC)(NC(C2CCCOCC2)=O)CCN(C(=O)CCC(=O)c2ccccc2)C1 N1(C(c2cc(C)ns2)=O)CC(NC(c2ccc3scnc3c2)=O)CC12CCOC2 N1(C(C2(C(C)NC(CCC=C)=O)CC2)=O)CCC(C)(O)C(O)C1 C12(NC(CC(C(C)C)OCC)=O)CC3CCC(C1C2)N3C(c1ccc(Cl)s1)=O Cc1ccc(NC(C2CCN(C(c3cnc(O)o3)=O)C23CC3)=O)cc1F C12(C(=O)NC3C(CC)N(C(=O)CCCCOC)CC3)CCC(C)(CC1)OC2 N1(C(C2CC(C(=O)OC)C2)=O)CCOC(OC)C1.N12CC3C(C3C1)C(OC)C2=O c1(C(=O)NC(C(=O)NCCOCCC)Cn2cccn2)cncnc1C C1(NC(C=CC(=O)NCc2cccc(C)c2O)(C)C)CCN2CCCC2C1 N1(C(C(C)Oc2ccccc2)=O)CC2CCC1(CNC(C1CC1F)=O)CC2 C(N=c1[nH]cnc(Cl)c1C#N)C1CCCC(NC(CC2N(C)C(=O)CC2)=O)C1 CP(C)(=O)c1cccc(NC(=O)C(=O)NC2CC3CCC2CC3)c1 N1(C(C(C)CC(F)(F)F)=O)CCC2CN(C(c3cc(O)cc(O)n3)=O)CC2C1 c1(C(=O)NC(C)CN(C(=O)CC2COCCO2)C)cc(Cl)c(F)c(Cl)c1 C1(c2cn(CC(=C)CC)nn2)CCCCCN1C(C1(C(=O)O)CCOC1)=O N1(CC(=O)NC2CC(O)(CNC(C3N(N=O)CCC3)=O)C2)CCCCCCC1=O N1(C(=O)Nc2c(OC)noc2C)CCC(O)C(NC(=O)CCCC(N)=O)C1 N12CCCC(CC1)OCC2C.c1(C(=O)CC)ccccc1OCC Cc1nc(CC(C)C)c(C(=O)NC2CC2CNC(c2ncn(C(C)(C)C)n2)=O)s1 c1(CC)cnc(N2CC3CC(NC(c4ccc(OCC)c(Cl)n4)=O)C3C2)c(C)c1 CC(CC(=O)N1CC(O)(CCNC(c2ccc(C3CC3)nc2O)=O)C1)C(F)(F)F C(=O)(C(C(CC)CC)OC)N1CCC(C(C)(C)NC(c2n(CCC)ccc2)=O)C1 c1(NC(C2C(CNC(C(C=C)C)=O)CCCC2)=O)cn(CC)nc1C#N C(=O)(CCCCCONC(C12CCN(CC1)C2)=O)N1C(COC(C)(C)C)C=CC1 C1(N)CC2(CCCN(C(C3CCCN3)=O)C2)C1.C(=O)(C(F)(F)F)C(=O)C1CC1 c1(C2C(C(=O)NCCOCCOCCON)C2)ccccc1F C1(O)(C(C(=O)NCc2ccon2)NC(C2CCS2(=O)=O)=O)CCCCC1 c1(C(N(C)Cc2cccc(CNC(c3ccc(F)cc3)=O)c2)=O)cc(O)ccc1Cl Cc1ccc(OCC(=O)NCC23CCC(C2)N(C(C2OCCO2)=O)C3)cc1C C(=O)(C(CC(C)C)NC(=O)C=Cc1ccnn1CC)N1C(CCC)CCCC1 N1(C(CC2ON=C(CC)C2)=O)CCCC(C(=O)NC2CCC(C)(O)CC2)CC1 c1(C(=O)NCCOCCNC(C(C(C)C)n2cnnn2)=O)cnc2[nH]c(O)nc2c1 N1(C(C(C)OC)=O)CCC(C2(O)CCN(C(C34CC(C(C)C)(CO3)C4)=O)C2)CC1 N1(C(C(C)(C)SC)=O)CC2(C1)CN(C(c1ccn3c(C)cnc3c1)=O)CC2CO C1(NC(c2cnn(CCO)c2N)=O)CN(C(=O)C2CC2)CC1c1scc(C)n1 C1(NC(C=Cc2ccc(C3C(C)C3)o2)=O)CCN(C(=O)CO)CC1(C)C C(CC(C)(C)CC(=O)NC1CN(C(C2CC(OC)C2)=O)CC12CC2)OC C1(CCC)(NC(CC(=O)NCC#C)=O)CCN(C(C2CCCSC2)=O)CC1 C1(CC(N2C(CC)COCC2)=O)CCCN(C(C2(COC)CC2)=O)CC1 N1(C(CCCCC)=O)CCN(C(c2c(C)nsc2NC(C)=O)=O)CC1CC Cc1nn(C(c2ccccc2)CCc2sccc2Br)c2sc(C(=O)N(C)C)cc12 C(=O)(CC(O)CN(C)C)NCC(C)N(C(=O)CN1CC2CC2C1)C Cc1nsc2ncc(C(N3CC(NC(=O)CC(F)F)CCC3C)=O)cc12 C1(NC(C2(COC)CC2)=O)CCCN(C(c2cnc(Cl)c(Cl)c2)=O)CC1 CCC(C)C(O)C(=O)NCC(C)(C)OCCNC(C1C(C)C1(F)F)=O N1(C(=O)COC2CCC2)CC2CC(C(N3CCOCC3CO)=O)(C2)C1 C(=O)(C(F)CC(C)(C)C)NCC1CC2(CN(C(C3C(CC)CCO3)=O)C2)C1 c1(C(=O)NCC(CC)NC(c2cncc(OC)c2C)=O)ccc2scnc2c1 C(=O)(CCC(C)(C)C#N)NCc1c(C(N2CC(C)S(=O)CC2)=O)n[nH]c1 N1(C(c2c(C)onc2)=O)CC2(CCCC(CNC(C3CC(=O)NC3(C)C)=O)O2)C1 c1(C(=O)NC(CN(C(C2COC(=O)C2)=O)CC)C)cccc(CF)c1 C1(CCC)CN(C(=O)C(C2CCCCC2)O)CC1C(N1C(C)CC1(C)C)=O C1(c2cn(C(C)C)nc2)CN(C(=O)CN2CCC(n3cccc3)C2)CCO1 C(c1ccc([N+](=O)[O-])cc1)=CC(C1(F)C(C(=O)OC(C)C)C1)=O NS(=O)(=O)CC(=O)N1CCC(C2OCCC2C(=O)O)CC1.C12(O)CN(C1)C(=O)C2 C1(C)(NC(C(C(C)C)NC(C(C)OCOC)=O)=O)CCC(C)(C)C1 c1(CNC(=O)NCCCC(C)(C)C(=O)O)cccc2ncccc12 c1(OC)ccc(C(=O)NCCC(O)CNC(c2nocc2Cl)=O)nn1 C(=O)(C#CC1CC1)N(C)CC1CCC(C(N2C(CN3CCCC3)CCC2)=O)O1 N1(C(C2C(c3c(C)ccs3)C2)=O)CCOC(C)(CNC(c2cccnc2)=O)C1 C#Cc1cccc(C(N2CC(COC)CC2CNC(C2(C)CC(F)C2)=O)=O)c1C N(C(=NCC1CCCN(C(C)=O)C1)N1CC=C(F)C1)C(C=C)C Cc1csc2ncnc(N3CCC(O)CC3C(=O)Nc3ccccc3)c12 O=C1CCOC(COC(=O)CCc2ccc(C(F)(F)F)cc2)C1 c1(SCNC(N(C)CC2CCCCC2)=O)cccc(Cl)c1Br Cc1cccc(Cl)c1C(=O)NC1CN(C(C23CC(C)(CO2)C3)=O)CCC1C c1(C(=O)NCC2CN(C(C(CCOC)OC)=O)C(C)C2)nc(Cl)ccc1F c1(CNC(=O)Nc2nc(Cl)ccc2Cl)c(O)cc(O)cc1O CCCCC(C)(F)C(=O)NCCCC(C)NC(c1nc(C)sc1C)=O N1(C(CNC(CCNC(=O)OC)=O)=O)CCC2(CC(NC(=O)C=C(C)C)CO2)C1 c1(OC)ccc(F)c(C(N2CCC(NC(=O)CC3(C)CCCO3)C(C)C2)=O)c1F c1(OC)cc(C(=O)NCC2(F)CN(C(C3(F)CCOC3C)=O)C2)c(F)cn1 n1(CC)nnc2c(N3CCC(NC(=O)Cn4c(O)nnc4O)C(C)C3)ncnc12 c1(C(N2CC(C)(NC(C=CC=CCC)=O)C2)=O)cnc(C2CC2)cn1 N1(C(C(CCC)=CCC)=O)CC2C3CCC(C2C1)N(C(c1cc(N)c(F)cn1)=O)C3 NC(=O)CCCCC(=O)N1CCCC(NC(C2CC(n3ccnn3)C2)=O)C1 C(=O)(C(F)(CNC(=O)C(C)n1cncn1)C(C)C)NCCc1c(C)cncc1 N1(C(CN(C2CCC2)C)=O)CC2CC(NC(C3CNC(=O)N3)=O)CC(C2)C1 c1(N(CCN(C(=O)C(C)Cc2cccnc2)CCOC)C)ccncc1 c1(CCC(=O)N(C)CC2(NC(C3CC(CC)OCC3)=O)CC2)cccc(F)c1Cl Cc1cnccc1C(C)C(=O)N1CC1CNC(=O)CCn1ccnc1 CCC1=C(C(=O)NC2CN(C(=O)C(Br)=C(C)C)CC2c2ccnn2C)CCCO1 c1(C(=O)NCCC(=O)NCC2(CC)CC2)cc[nH]c(=N)n1 Cc1c(NC(N2CCN(C(C3CCN(CC(C)C)C3)=O)C3CC23)=O)cccc1F C1(C(CNC(C2CC=CC2)=O)NC(c2ccn(C3CC3)n2)=O)CCCCCC1 N1(C(C2CN(C(C)=O)C2)=O)CCC2CCN(C(c3c[nH]cc3Br)=O)CC2C1 CN1C(=O)c2ccccc2C1Cc1nc(COC)nn1C1CCC2(COC2)O1 N1(C(c2c(C)nns2)=O)C2CCC1CC(NC(c1ccc(CN(C)C)cc1)=O)C2 c1(CC)nn(C)cc1C(=O)NCC(O)CNC(=O)COc1ccccc1O C1(C(N2CC(CNC(C(C#C)(C)C)=O)OCCC2)=O)CN2CCCN1CC2 c1(N(C)C)nc(C(N2CCC(C)C(CNS(C)(=O)=O)C2)C(=O)NCCCF)cc(O)n1 N1(C(CN(CC)CC)=O)CCC(C(=O)NCCC(C)N2CCCC2)C1 C1(CCOC)CN(C(=O)CC=C(C)C)CCN1C(=O)CCCc1ccnn1C c1(CC(=O)NC2CC3CC2N(c2ccncn2)C3)ccc(F)c(F)c1 C=CCCCCCC(=O)NC(C)(C(=O)NC(c1ccn(C)n1)C)C1CCC1 c1(OC)ccc2ncccc2c1C(N1CCCC(CCNC(=O)CC(C)O)C1)=O C1(NC(=O)C=Cc2cn[nH]c2)CCCCCN(C(C2CC(F)C2)=O)C1 C12CC(C(C)C)CC1OCSC1(CCC1)C2SCC.c1(C)cn(CCCCOC)nn1.OC c1(C(=O)NCc2cc(O)no2)ncn2cc(-c3cccc(F)c3O)sc12 c1(NC2CC(=O)NCC2)ccc(S(=O)(=O)NCc2nc(Cl)cs2)cc1F c1(C(=O)NC2(C(=O)NCCN3CCOC3=O)CSC2)conc1C1CC1 c1(C(=O)NCC2N(C(C3C(C)(C)C3)=O)CCC2)c(F)ccc([N+](=O)[O-])c1F c1(-c2cn(CCCC)nc2)ccc(C(=O)N(CC)Cc2cccnc2)c2[nH]ccc12 c1(C(N2CCC(C(C)NC(=O)C(F)=C3CCC3)C2)=O)cc(C(F)(F)F)cc(N)c1 c1(C(=O)NC(CNC(C2N(C(C)=O)CCOC2)=O)CO)c(CC)nn(C)c1CC C(c1cnn(C)c1)=C(C)C(=O)NC1(CNC(=O)CCn2ccnc2)CCC1 C(=O)(C1=NN(C)C(=O)CC1)NC1C(C)CN(C(=O)Cn2nnc(=O)[nH]2)C1 c1(C(=O)NCC2(CNC(C3(C)CC3(F)F)=O)CCCC2)cc2cnccc2[nH]1 C1(C(=O)NC(CC(C)C)C(N)=O)CC12CCN(C(=O)C(F)C(F)(F)F)CC2 C1(C(=O)NCC2(CNC(c3cn(CC)nc3)=O)CC2)CC1C1CCCC1 N1(C(c2c(CNC(CC3C(CC)C3)=O)ccs2)=O)CCCC12CCNC2=O c1(C(=O)NC(C2OCCN(C(COCCOC)=O)C2)C)ccc2nc(S)oc2c1 C1(CNC(c2c(CC)non2)=O)CN(C(=O)C(=Cc2cnn(C)c2)C)CCCO1 Cc1cnc(NCC(C)(C)CC2(NC(=O)C(O)CC(C)(C)C)CC2)nc1S(C)(=O)=O C1(O)(CN(C(C(C)NC(C2CCCC2)=O)=O)C)CN(C(C2CC(F)(F)C2)=O)C1 O=C(C1=CCC(F)(F)CC1)NC1CCCC1NC(c1cc(O)nc(C2CC2)n1)=O C1(C(=O)NC2CC(C)(NC(CC(CC)OC)=O)C2)OCC2CCCC12 c1(C(=O)OC)cc(C(=O)N(C2CN(C(c3ccc(OCF)cc3)=O)C2)C)c(C)s1 N1(C(C(C)S(C)(=O)=O)=O)CC=C(CC(=O)N(C2CCCN(C)C2)C)CC1 CC1(C)CN(CC2(C(=O)O)CC3(CCOC3)C2)CC2(CC3CCC2C3)O1 C1(CNC(C(=O)NCC)=O)CCC(C(N2CCCC2CC)=O)CC1 C1(C(N2CCCC(N(C(c3ccc(C)[nH]3)=O)CC)C2)=O)CCOC(C)(C)C1 C1(C(=O)NCC2CC(C(=O)NC3(C)CCSCC3)C2)Cc2nccn2C1 CC(C)(C)C(CNC(C1CCOC(=O)CC1)=O)C(=O)NCC1(CO)CCC1 c1(CN2C(CNC(c3ccc(CC)o3)C(=O)OC)CCC2)ccc(OC)cc1Br C1(C2CCCO2)(C(N)=O)CCC1.C(CCOCCNC=O)OCCNC=O C1(C)(C(=O)NCc2c(C(=O)NCCN(C)C3CC3)[nH]cc2)COC(=O)C1 N1(Cc2cnc(C)nc2C)CCC(F)(F)C(C(=O)Nc2cc(N(C)C)ncn2)C1 Cc1c(C(N2CC(F)(CNC(C3CCOC3)=O)C2)=O)sc2cc(F)ccc12 C1(NC(C(C(C)C)NC(=O)Cc2cn[nH]c2)=O)CCC2(CC1)N=N2 C1(CNC(C=COCC)=O)CC(C)(C)CCC1NC(=O)C(C)(C)n1cccn1 C1(CC(N2CC=CC(NC(Cc3ccc(C)nc3)=O)C2)=O)Cc2ccccc2N1 CC(C)(C(=O)NCC(O)CNC(C1CCCN(S(=O)(=O)C(F)F)C1)=O)C(N)=O N1(C(Cc2ccc(C)cc2Br)=O)CCc2ccc(Cl)c(F)c2C1C C(=O)(C1=CCC2CCC1N2C(=O)C(C)CC(C)C(C)=O)N(c1noc(C)n1)CC C1(CNC(C(CNC(c2cn[nH]c2)=O)OC)=O)NC(=O)CC1(C)C Cn1ccc2ccnc(C(=O)NC3CCN(C(c4snc(O)c4Cl)=O)C3(C)C)c12 c1(OC)ccc(C)cc1CC(=O)NC1CC(O)CN(C(c2csc(C)c2)=O)C1 C1(=O)C(CCCC(=O)OC)N1CCC(CC)OC.N(C)(C)CC C1(C(=O)NCC(CNC(c2n(CCC)ncc2)=O)(C)O)CN(CC)CCO1 c1(NC(C=CC(=O)N(CCCCCC)CC#C)(C)C)cc(C)c(C)nn1 N(C1CCc2cccnc21)C(C1C(CNC(CC2N(C)CCC2)=O)CCC1)=O Cc1cccc(F)c1C(N1CCC(CCNC(=O)CSc2n[nH]c(O)n2)CC1)=O C1(C(N2CCC(O)(CO)C2)=O)C=CCCN1C(=O)C=C1CCCCC1 C=CC(CCC)CC(=O)NCC1CCN(C(C2(n3ccnn3)CC2)=O)CC1(F)F c1(CC(=O)NCCOC2CCN(C(C3(O)CC(O)C3)=O)C2)cc(F)c(F)cc1F N1(c2nc(SC)nc(C)c2)CC(C2CCCN(C(c3nc(O)sc3C)=O)C2)C1 Cn1nc(C(=O)NCC=CCNC(C2CCCCN2C2CCCC2)=O)c(Br)n1 C(=O)(CC(C)F)NCC(C)NC(C1CC1(C)C)=O C(C(O)C(F)(F)F)N(C)C(C1(CN)CCCO1)=O C1(C2CC2)(C(N(CC(C)CNC(c2c[nH]nc2C(F)(F)F)=O)C)=O)CC1 C(=O)(C(CC)CC(C)C)NCC(CNC(COCCC=C)=O)OC c1(C(=O)O)cc(CN2CCCC(c3ccc(F)cc3F)C2)cnc1O c1(CC(=O)NC2CCC(N(C(C(C)C(C)O)=O)CCO)CC2)cc(O)nnc1O N1(C(C(C)OCC)=O)CCC2(CCN(C(c3cnns3)=O)C2)C1 CCC(CC)CCCC(=O)N1CCCCC1CCC(=O)NCC(C)(F)C(C)(C)F c1(C(=O)NCC(C(C)C)NC(C2CC2c2cscn2)=O)cnc2[nH]cnc2c1 C1(NC(CS(CCC)(=O)=O)=O)CC2(CCCCN2C(C2CSC(C)=N2)=O)C1 C1(NC(C2CCC(=O)N2)=O)CCC2CN(c3nnco3)CCC2C1 C1(NC(C=CC(C)(C)C)=O)CC2CC1N(C(=O)Cc1ccn(C)n1)C2 C1(CNC(C(C)N(C(C)=O)C)=O)CC2CCC1N2C(C1(O)CN2CCC1CC2)=O c1(NC2CCCN(S(c3c(C)noc3C)(=O)=O)C2)ncccc1S(C)(=O)=O N1(C(COCCOCCOC)=O)CCCC(O)(CN(C(=O)C2=CCCS2)C)C1 N#Cc1ccc2cc(C(N3CCN(C(c4csnn4)=O)C4CCC34)=O)ccc2c1 C1(NC(C(=O)NCCCc2ccc(C#N)cc2)=O)Cc2cccnc2C1 c1(N2CC(C(C)NC(C3(CCF)CC3)=O)OCC2)ccc([N+](=O)[O-])cc1Cl N1(C(COc2cccc(OC)c2)=O)CC2(CCCN(C(=O)CS(=O)(=O)CCl)C2)C1 Cc1cccnc1C=CC(N1CCCC(N(C(=O)C2=CCCCC2)C)CC1)=O Cc1ccc(C(C)NC(=O)C(CCN(C)C)NC(c2ccccc2C)=O)nc1 N1(C(c2cc(C)c(Br)s2)=O)CC(NC(c2n[nH]c(C)c2F)=O)CC(F)C1 C12(CNC(c3scc(C)c3C)=O)CCC(C1)N(C(=O)C(C1CC1)C1CC1)C2 C=CC1(C(=O)NC2CCN(C(=O)C(=O)CCc3ccsc3)C(C)C2)CCOCC1 C1(C(N2CCN(C(c3cnn(C)n3)=O)C(CO)C2)=O)CCCCCC1(F)F C1(C)(NC(c2nc(C(C)C)sc2)=O)CCN(CCO)CC1 Cc1cc(C)c(C(N2CCC(NC(=O)CC3CCC(C)(C)CO3)CC2)=O)c(=O)o1 c1(CCO)ccc2c(c1)CCO2.C(c1cccnc1)=CC(C(=O)CO)=O c1(NC(C2N(C(CCC=C)=O)CCSC2)=O)ccc(C(=O)OC)c(C#N)c1 C1(SCCC(=O)NC2C(NC(c3c(CC)c[nH]n3)=O)CCC2)CCS(=O)(=O)C1 N1(CC(=O)N(CCC(=O)NCCc2cc[nH]n2)CC=C)CCCNC1=O CCCC(CNOC)C(=O)NCC(C)C(=O)C(=O)C=Cc1cc[nH]n1 c1(C(=O)NC(c2cn(Cc3sc(C)nc3C)nn2)CCC)c(Cl)cc(C#N)cc1Cl C=CC1(C(N2CCC(C(C)NC(C3(C)CCCC3CC)=O)CC2)=O)CCOCC1 CCCCC(CC)CC(=O)NCc1ccc(C(C)NC(c2ccncn2)=O)cc1 c1(C(N2CCC(N(C)CC)C2)=O)ccc2c(c1)n(C)c(=O)n2C c1(CC)ccc(O)c(C(=O)NCCCCC(C)NC(c2ocnc2C)=O)c1 N1(C(CSCCC)=O)CC(NC(=O)CN=S(C)(C)=O)CC12CCCOC2 c1(CC(=O)NCC2C(CNC(C3(C#C)CCC3)=O)C2)nc(C)c(C)[nH]1 CCN(OC)C(=O)CNC(=O)CC(C1CC1)NC(c1ccsc1C)=O c1(C(=O)NCC(C(C)C)NC(=O)CCCS(C)(=O)=O)nnc(O)c2c1CCCC2 C1(C)(C(=O)NCC2C(OC)CN(C(c3c(COC)ncs3)=O)C2)CC2(CCC2)C1 Cc1ccc(O)c(CNC(=O)C(CO)NC(c2ccc(C(C)C)o2)=O)n1 n1(CC(=O)NC(C)CC(C)NC(=O)C(C)NS(C)(=O)=O)ccc(=O)n(C)c1=O C1(OC)CN(C(=O)CCc2cc(C)no2)CCC1NC(C1CC1C1(C)COC1)=O c1(C(N2CCC(C(=O)NC3COC3)(CF)C2)C(=O)OC)cncc2c1CCC2 C(CN=c1[nH]nc(C(N)=O)s1)C1N(C(CCC(=C)Cl)=O)CCCC1C CC(C)C1=NOC(C(N2CCC(CO)(NC(=O)CC3C(C)(C)C3(C)C)C2)=O)C1 C(=O)(C#CC1CCCO1)N1C(CCC)CN(C(=O)Cc2cn3ccsc3n2)CC1 N#Cc1ncc(N2CCN(C(=O)CCN3CCCCC3=O)CC2)nc1C#N C1(NC(C2(CC=C)CCCC2)=O)CN(C(c2cn(CC)nc2C)=O)CCC1C C1(NC(c2c(C)[nH]c(C(C)(C)C)c2)=O)CC12CCN(C(=O)CO)CC2 Cc1[nH]nc(C(=O)N(C(C)CC(=O)NCCC(C)N(C)C)C)c1O c1(C(=O)OC)ccc(C(C)=CC(=O)NC2CCCC(NC(=O)Cc3ccno3)C2)o1 CCCCC(CCC)NC(=O)CCN(C(=O)C(F)CC1CCOC1)CC N1(C(Cc2c(C)n[nH]c2)=O)CC(N(C)C(C2CCCS(=O)(=O)C2)=O)C(C)(C)C1 c1(C(=O)NC2CCN(S(C)(=O)=O)C2)cc(OC(F)F)ccn1 C1(CC(=O)N(C)CC2CCSC2)COCCN1C(=O)Cc1cc[nH]c1 Cc1cc(CO)oc1C(=O)NC(CNC(=O)C(O)CCc1ccccc1)CO C=CCC(C(=O)N(C)CC1(C#N)CCC1)NC(=O)CCN1CCOCC1 CC1(C)C=NN1C(=O)C(N=[N+]=[N-])c1ccccc1 c1(CN2C(C(=O)Nc3sncc3Cl)CC2)ccc(-n2ccnn2)cc1 C1(C(N2CCN(C(c3c(CC#N)cccn3)=O)CC2)=O)CC2C(C1)C2(F)F C#Cc1ccc(CNC(=O)C(CC(C)C)ONC(=O)C(CO)OCC)cc1 C(CC(C(C)(C)C)NC(c1cnc(Br)s1)=O)N(C(=O)C1=CC(C)(C)C1)C c1(C(N2CCC(C(C)NC(CN(C(COC)=O)C)=O)C2)=O)ncc(Cl)nc1Cl Cc1cn2nc(C(=O)NCCCC3CCNC3)cc(C)c2n1 N1(C(c2ccc(CC)[nH]2)=O)C2CCCC1CC(NC(c1c[nH]ccc1=O)=O)C2 C1(N(C(C=CC(C)C#N)=O)C)CC2CCC(C1)N2C.n12cnc(c1)C(=O)NCC2 C(=O)(C(C)CCCc1ccccc1)NCC(CC(C)C)NC(c1cnsc1)=O N1(C(C(C)n2ccnn2)=O)CC2CC1CC2CNC(=O)Cc1cc(Cl)ccc1O C(=O)(C(=O)C(C)(C)C)NC(C)CCCCNC(c1cccc(C2(O)COC2)c1)=O CC1(C)C(Cc2cc(O)cc(N)c2Cl)CCN1C(C=CC(=O)NCn1cnnc1)=O n1(CC(=O)NC2C(CNC(c3c(CCC)n[nH]c3)=O)C2)nc(C)n(C)c1=O N1(C(C(Cc2ccccc2Br)NC(CC(CC)OC)=O)=O)CCC(C)(F)CC1 c1(NC)ccccc1C(=O)NC.C1CCCC(=O)NCC2CCOCN12 CN1CC(C)(C(=O)NC23CCC(CNC(=O)CNC=O)(CC2)OC3)CCC1=O C1(C(=O)NC(C2CSC2)C)CCOCCN1C(=O)Cc1nc(=N)[nH][nH]1 Nc1c(C(N2CCC=C(CNC(=O)CC3CCCC3)C2)=O)cnc2ccnn12 c1(C(=O)NC2(C)CC(NC(C3CC34CC4)=O)C2)cc2c(cc1F)OCC(=O)N2 Cc1cccc2nc(N3CC(NC(=O)C=CC(C)(C)C)CC4(CC4)C3)sc12 C(=O)(C(F)(CNC(C1(CCC)CC(=O)C1)=O)C(C)C)NC(CCC)C c1(C(=O)NC(CNC(CC(C=C)C)=O)C2CCC2)ccc(C(F)(F)F)c(O)c1 C1(CCCC)CN(C(=O)C(C2CCC2)OC)CCN1C(C1CC1C(F)F)=O c1(C(C)=O)cccc(OCCCC(=O)N2CCC2CNC(c2cnc(O)s2)=O)c1 C1(C(=O)NCC2C(C)CCCN2C(c2cnc(Cl)cn2)=O)CCc2nncn2C1 N1(C(C23CC(C)C2C3)=O)CCC2(CC1)CN(C(=O)C(c1cc(F)cc(F)c1)O)C2 N1(C(c2nccc(C)c2)=O)CCCC(O)(CN(C(=O)CCC(C)(F)F)C)C1 c1(C(=O)NCC(C)N(C(CC2CCC(C)O2)=O)C)cc2c(=O)[nH]ccn2n1 c1(OC)ccc(=NC(=O)CCC(=O)NCC2CC2c2ccccc2)[nH]n1 c1(C(=O)NCCC(C)NC(C2CC3C=CC2CC3)=O)c(F)ccc(O)c1F c1(C(=O)NCCC2OCCN(C(C(CC)(F)F)=O)C2)c(N)cccc1[N+](=O)[O-] c1(C(N(C2C3CCCC23)C)=O)[nH]ccc1CNC(c1cc(CO)on1)=O C#CCCCCC(=O)NC1CC(C)N(C(=O)C(=O)NC(C)C)C1 c1(CCC(=O)NCCC(C)N(C)C(c2cc(C(F)F)n(C)n2)=O)cncc(F)c1 c1(C(=O)NCC2C(C)(C)C(=O)C2)ccc(F)c(F)c1F C#CC1CN(C(C2CC(O)C(F)C2)=O)CCN1C(=O)CCCSC(C)(C)C c1(C(C(=O)NCCCOC)N(c2ccc(C)cc2)C)ccc(F)c(I)c1 N1(C(c2c(C(=O)OC)con2)=O)CC(NC(C2CCN2S(C)(=O)=O)=O)C(C)(C)C1 N(C1CC2(CCCC2)c2ccccc21)C(c1n(C)c(Cl)cn1)c1nnnn1C1CC1 N1(C(C(C)(CC2CCC2)OC)=O)CC2CC(NC(=O)CC3C=CCCC3)C(C2)C1 Cc1cc(Cl)cnc1C(N1CC(C)CC1C(N1CCS(=O)CC1)=O)=O c1(CC)nc(C#N)cc(=NCCN2CCC(NC(C3NC(=O)CC3C)=O)C2)[nH]1 CCC(O)C(C)C(=O)NC12COC(NC(=O)C(C)Oc3ccc(F)cc3F)(C1)C2 C(=O)(CC1C(=O)Nc2cc(Cl)ccc21)NCC1C(NC(CN(C)CC)=O)CC1 N1(C(CCC(C)SC)=O)CC(NC(c2cnn(C)c2N)=O)CC12CCCC2 CCCCC(C(=O)NC)NC(=O)C(C(=O)NC(CC)C(C)(C)O)N(C)C C1(NC(COCCCC#C)=O)CCCC(CN(C(=O)CSCC2CCCO2)C)C1 N1(C(c2coc(C(F)F)c2)=O)CC(O)CC1C(=O)N(C1CCOCC1)CCO c1(C(N(CCN(C(=O)CCN2CCCCC2=O)CC)CC)=O)nn(C)c(N)c1C n1(CCC)nc(-c2cc(SC)ccn2)nc1Cc1cccc(C(C)C)c1 C(CC(O)C(C)(C)C)N(CC(N1CCC(C)(O)C1)=O)Cc1n(C)ncc1 c1(C(C(=O)NCC)N(CC(C)C)C2CC2)ccc(Br)c(F)c1 CCC(CCCC(=O)O)NCC(=O)Nc1cncc(C(F)(F)F)c1 C1(NC(c2scc(OC)c2)=O)CCN(C(=O)CC2(O)CCC2)CCC1(F)F c1(C(N2CCC(NC(C3CC3c3ccccn3)=O)CC2)=O)cc(Cl)nc(Cl)c1 C1(CN(CCN(C)C)C)CC2COCC2C1.c12ccc-1o2 C1(C(N2C(COC)CCCC2)=O)CCCCN(C(c2ccc(F)cc2C)=O)C1 C1(C(N2CC(N(CC=C)C)C2)=O)(CC)CCCN(C(=O)CCCCSC)C1 c1(C(=O)NC2CC(C(=O)NCc3cccc(COC)c3)C2)onc2ccccc12 c1(C(c2ccccc2)C)cnc(NC(C2CCC(C(C)(C)C)CC2)=O)nc1 N1(CCC(C)CCNC(N2CCCC2CCO)=O)CCCCC1C N1(CCC(=O)NC2C=CCN(C(COC(CC)C)=O)C2)CCSC(C)(C)C1 c1(C(N2C(C3(NC(CCSC(C)C)=O)CC3)CCCC2)=O)cnc2ccoc2c1 c1(C(=O)NCCC(C)N(C(c2ccn(CC(C)C)n2)=O)C)ccccc1S(C)=O C1(=CC(=O)NCC2CCC(NC(=O)C(F)(F)C3CCCC3)C2)CN2CCC1CC2 Cc1ccc(C(C)(C)C(=O)NCC=CCNC(=O)CC2CCCC(O)C2)cc1 C(=O)(C(F)C(C)(F)F)N1CC(CC(=O)NC(COC(C)C)C)C(C)C1 N1(C(C2(CC=C)CCC2)=O)CC2CCC2(CNC(=O)CN2CC(C)(C)C2)C1 N1(C(C2(COC)CCCC2)=O)CCN(C(C2CCCC(C)C2)=O)CC(C)(F)C1 C1(C(=O)NCC(NOC)=O)C(CC)CCN1C(c1cccs1)=O CC1CCN(C(C23CC2CN(C(c2cccc(OC(F)(F)F)c2)=O)C3)=O)CC1 C(=O)(C1=CS(=O)(=O)CCC1)N1C(CN(C(=O)C(C)(C)CCC#N)CC)CCCC1 CC1(CNC(C2(OC)CCCOC2)=O)CCCN(C(C2CC3CC3C2)=O)C1 c1(C(N2C(C(C)NC(c3csc(C4CC4)n3)=O)CCC2)=O)ccsc1S(N)(=O)=O O=C(CCN1C(=O)CCc2ccccc21)Nc1c[nH]ccc1=O c1(-c2nc(CSC)nn2CCCCO)cc(C)c(OCC(C)C)c(C)c1 C1(CC(=O)N(C2CCN(c3ncnc(C(C)(C)C)n3)CC2)C)CC=CCN1C C(=O)(CCCC(C)(C)CC)NCC1CCC(C(=O)NC2C(OCC)C2C)C1 C(=O)(C(C)(C)CCCNC(C1CCC(C)(C)OC1)=O)N(C)Cc1ncc[nH]1 c1(C(=O)NC(CN(C(C2(C(F)F)CC2(F)F)=O)CC)C)ccnc(Cl)c1OC C1(CC(=O)NCC2(C)CCN(C(c3ncc(Cl)cc3F)=O)C2)CN2CCN1CC2 C(=O)(C(F)(F)C(O)C1CC1)Nc1cccc(CNC(C=Cc2n(C)cnn2)=O)c1 c1(SCC(=O)NN(C(C2CC(NC(CCCC#C)=O)C2)=O)C)cc(O)ccc1C N1(C(CC2N(C(c3cc(C)nc(C)n3)=O)CCCC2)=O)CCn2ncc(O)c2C1 c1(C(=O)NC2CC(O)CN(C(=O)Cc3csnn3)C2)ccc2ccccc2c1 C12(NC(CS)=O)CCCN(C(=O)CSc3ccc(OC)cc3)CC1C2.CCCN(C)C C(=O)(C(C)CN1CCOCC1)NCCN(C(C(C1CC(F)(F)C1)OC)=O)C1CC1 C1(NC(C=Cc2cc(OC)c(F)cc2)=O)CN(C(=O)C2=CCOC2)CC1N=[N+]=[N-] c1(C(=O)NCCOC2CCN(C(CC(C)C(F)F)=O)C2)sccc1S(N)(=O)=O C1(O)(CN(C)C(C2CCC(=O)NC2)=O)CCN(C(=O)C(C)(Cl)Cl)C1 CC1=C(C(=O)N(C2CCN(C(=O)Cc3cn(C4CC4)cn3)C2)C)CCCC1 C1(NC(CS(=O)(=O)NCC)=O)(CNC(=O)C(C#N)(CC)CC)CCC(F)(F)CC1 N1(c2nc(N3CCC(c4ncc[nH]4)CC3)cc(C)n2)Cc2nn(C)c(N)c2C1 C1(C(=O)NCCN(C(=O)C(n2ccc(C3CC3)n2)C)CC)CCOC1=O CC1CC(C(=O)NCCC2CC(C(=O)NC34CC(C)(C3)C4)C2)=NO1 c1(NC(C(N2CCCC(Nc3cccc(C)c3)CC2)=O)=O)ccc(C)n(C)c1=O C(CCC(C)CC(=O)N1CCC2(CC1)CC2NC(=O)CC1CC1)=C(C)C C(=O)(N1CCCc2nccn21)OC(C1(C2(O)CCOC2)CCC1)=O c1(C(=O)NCC(C(C)C)NC(c2scc(C)c2Cl)=O)cc2cnccc2[nH]1 N1(C(C2C(C(=O)CCN3CCCCC3)C2)=O)C2CCC1CN(C(=O)C(=O)N)CC2.CO c1(N2CCN(C(N(C3CCOCC3)CCOC)=O)CC2)ccc(N)c(Cl)c1 Cc1nccc(C(=O)NCc2c[nH]nc2C(=O)NC2CC(Cl)(Cl)C2)n1 Cc1nc2sccn2c1C(N1CC2CCC1C(CNC(=O)CN=S(C)(C)=O)C2)=O Cn1cc(C(N2CCC(c3cn(CC4CC4)nn3)C2)=O)c2c(c1=O)CCCC2 C1(C(N(C2CCN(C(c3cn(C)nc3C)=O)C2)CCC)=O)CC(C)CC(C)(C)C1 c1(C(=O)NCCCCC2CCCN(C(C3C(CC)C3)=O)C2)cc(F)c(F)cc1F CCC(CC)(C(C)C)NC(c1ccc(CNC(=O)C(C)CC(C)C)s1)=O c1(C(=O)NCC2C3CN(C(CCC=CC)=O)C2C3)cnc(O)n(C2CC2)c1=O N1(C(Cc2c(C)ccs2)=O)CC2CCC2(CNC(C2CCS2(=O)=O)=O)C1 C1(=O)CC(=O)N(CCOC)CCCN1.C(=O)(CCC1CC1)Nc1nccs1 N1(C(C(CC#C)C2CC2)=O)C2CCC1CC(C(=O)NCC(CC=C)CC(C)C)C2 C1(NC(C2CCCC3(CC3)C2)=O)CCC2(CCN(C(c3ccncc3F)=O)C2)C1 N1(C(C(C(C)C)COC(C(C)C)=O)=O)CCCC(F)(C(F)(F)F)C1 N1(C(C#CC)=O)CC(NC(c2cnccc2C(=O)NN)=O)C(C#N)C1 Cc1cc(C(=O)NCCN(C(=O)Cc2cc(Cl)sc2Cl)C(C)C)c(C)o1 Cc1ccc(NCC(=O)NCC2CC(C)N(C(C3CC(O)C3)=O)C2)cc1C N1(C(CCCCOC)=O)CCC(NC(c2cn(C(F)F)cn2)=O)C12CCC2 c1(C(=O)NCC2=CCCN(C(C3C(C)(C)C3(C)C)=O)C2)cc(Cl)c(F)c(Cl)c1 C1(C2CC2)(C(N(C2CCC(NC(=O)Cc3cnn(C(F)F)c3)C2)C)=O)CC1 CCC(C(=O)NC1CCC(NC(c2cc(CC3CC3)[nH]n2)=O)C1)N(C)C CCCC(CNC(c1[nH]ccc1C1CC1)=O)C(=O)NC(C(C)C)C1CCC1 N1(C(C=CC=CCC)=O)CCN(C(C2CCCOC2)=O)C(c2cn[nH]c2)C1 S(=O)(=O)(c1ccccc1Cl)N1CC2CN(C(=O)CSc3ccc(F)cc3)CC21 CCCC(C)(O)C(=O)NC(Cc1ccco1)C(N1CC2CCC(C2)C1)=O CCC(CC(=O)NC1CCN(C(=O)CN2CCCNC2=O)CC1F)C(F)F C1(NC(C23CC2C3)=O)CCN(C(=O)CC2CCS(=O)(=O)CC2)CC1F C1(C(=O)NC(c2cccc(Br)c2)CC)CC(F)(F)CN1C(c1sccc1C)=O c1(OC)ccc(OC(C)C(=O)NC2CCCN(C(C3CCCC(=O)N3)=O)C2)cc1 O=C(C(O)CC(F)(F)F)N(CCCCN)C(c1ccnnc1Cl)=O.C12CCN1C2 c1(OC)ncc(C)cc1-c1cnn(C)c1.C1(=O)CCCO1 C1(C(N2CCC(NC(C3CN(CCOC)C(=O)C3)=O)C2)=O)CC12CCOCC2 N1(Cc2ccc(C)c(C)c2)Cc2ccccc2C1C(=O)NCc1cc(Br)ccn1 N1(CC2CCC(OC)CC2)CCC(=O)N(CC=C(Cl)Cl)C1=O C=CC(C)N=C(NC1CC(CS(N)(=O)=O)C1)N1CCc2cc(Cl)cc(Cl)c2C1 c1(NC(C2(O)CCN(C(C3(C(C)C)CCC3)=O)CC2)C)ccc(Br)cc1[N+](=O)[O-] CC1CCC=C1C(=O)N1CCC(CN(C(=O)C(O)Cc2ccccc2Cl)C)CC1 c1(C(N(C)CC2CCN(C(c3cn4c(n3)SCC4)=O)C2)=O)ccc2nccn2c1 C1(NC(C=CC)=O)CCCOC12CCN(C(C1CC(C)(F)C1)=O)CC2 C(CN=c1ccc(C)c[nH]1)NC(=O)NCC=CCCOC N1(C(c2cncnc2C2CC2)=O)CCC(c2cn(CC3CCCO3)nn2)C12CC2 c1(C(=O)NC(CCOC)CNC(=O)C(O)CC(C)C)cc(Cl)c(N)c([N+](=O)[O-])c1 c1(C(=O)NCC2(c3cc(F)cc(F)c3)CCC2)cc(=O)n2nccc2[nH]1 c1(C(C(N2CC(=C)C2)=O)Oc2ccco2)c[nH]c2ccccc12 c1(C(=O)NC2C(NC(c3c(C)cc(C)s3)=O)COC2)cc2c(cc1O)CCCC2 Cc1ccc(C(=O)NCCC2CCC(NC(=O)C(=O)NCC3CC3)C2)c(O)c1C CC1CN(C(=O)C(N)=O)CCC1CNC(=O)COc1cccc(C(F)(F)F)c1 N1(C(C2C(C)C2)=O)CCCC2(C1)CN(Cc1cc(C(=O)O)cc(Br)c1)C2 c1(C(N2CCC(C)(NC(C3CCC(=O)N3)=O)C2)=O)cc(F)cnc1O c1(OC)ccc(NC(c2ccccc2CNC2CNC2)=O)cc1 CN1CCN(C(c2cncc(Cl)c2)=O)C(CNC(=O)CC2(C(F)F)CC2)C1 c1(SC)cc(C(=O)NCC(C)CNC(c2noc(C)c2Br)=O)c(C)o1 C(=O)(C(F)(F)c1cncs1)NCC1C(NC(CCNC(COC)=O)=O)C1 c1(CC(=O)NC(CNC(C(C)OCCN(C)C)=O)(C)C)cc(F)ccc1Cl C1(C(N(C(C(=O)N(CCCc2ccco2)C)(C)C2CC2)C)=O)CCCCN1C C(CC(Cc1ccccc1)C1C(CS(C)(=O)=O)C1)NC(=O)C(N)=O N1(C(C(CC)(CC)OC)=O)CCC2(C1)CN(C(=O)CCCc1cnn[nH]1)CCO2 CC(CC(=O)N1CC(NC(C2(C#N)CC3CCC2CC3)=O)C(C)C1)CC(C)(C)C C1(C)(C)CCCC(=O)N1.CCC(C)C(C(=O)NCCC1CC1C(=O)OC)OC CN=c1cc(NC(C)C(=O)Nc2ccccc2N2C(=O)CCC2=O)cc[nH]1 c1(C(=O)NC2CC(CNC(=O)Cc3ccsn3)C2)cnn2c1OCC(F)C2 c1(C(N(CC(C)NC(C2CC3CCC2CC3)=O)C)=O)ccnc2[nH]cnc12 C1(CNC(Cc2ncc(C)s2)=O)CC2(CCC2)CN1C(=O)CCC1CCOC1 c1(NC(C2(OCC)CC2)=O)cn(C)nn1.C1(=O)CCC2CC(C2)CN1 C1(CC(=O)NCCOCCn2cc(C(CC)(C)O)nn2)CCN(C(C)=O)CC1 CC1(C(=O)NCC(CO)NC(c2cscc2Br)=O)COCCO1 C=CC(C)(CCOC)C(=O)NCCN(C)C(c1nc(C)oc1OCC)=O N1(C(C2CCN(C(=O)C=CCF)O2)=O)CCC(C2=NOCC2)C1 c1(CC)cc(N2CCCC(C(N3CCN(C(=O)CSC)CC3)=O)C2)n(CCO)n1 c1(NC(=O)CSC(C)(C)C)ccccc1O.C(=O)(CCC1CC1)NCCCOCC C12(CNC(CCCNC(c3c[nH]nc3Cl)=O)=O)CCC(C1)C(=O)N2 CC(C)CC(C(=O)NCC1(CNC(=O)CN2CCCCCC2=O)CCC1)C(N)=O C1(NC(c2c(C)cnnc2)=O)CN(C(c2c(C(C)C)cnn2C)=O)CCC1C N1(C(C(C)SC)=O)CCN(C(c2ccnc(N(C)C)c2)=O)CC1C(C)C.C1(N)CC1 Cc1ccnnc1C(=O)NC(C)CCCCNC(C1CC(=O)N(C(C)C)C1)=O N1(C(C(C)C(F)F)=O)CC2CCN(C(=O)CCC(c3ccc(F)c(F)c3)=O)C2C1 CC(CC#CCN(C)C)C(=O)N1CCOC(CN(C)C)C1 C(=O)(CC(C(C)OC)NC(=O)CCC(N)=O)N1CC(N(CCC)CC)C1 c1(OC)cc(F)c(C(=O)NC(C)CN(C)C(C2Cc3nncn3C2)=O)c(F)c1 CC(C)CC(C)CC(=O)N1CCOCCC1C(=O)NCc1cn(C)nn1 N1(C(c2ccn(CCOC)n2)=O)CCC2CN(Cc3cc(C#N)ccc3F)CC12 C(=O)(C(CC(C)C1CC1)N1CCC(C(=O)OC(C)=O)(OC)CC1)NCCCSC c1(N2CC(C)(C)C(NCc3cc(Cl)c(Cl)cc3O)C2)ncnc2c1CCCC2 C=CCC(C)C(=O)NCC(C)N(C(=O)C(C)Cc1ccccn1)C N1(C(CCN(S(C)(=O)=O)C)=O)CCN(C(C2(O)CC2(C)C)=O)CC1 CC1CC2(CC(C(N3CCCN(C(C4CCCC4CF)=O)CC3)=O)C2)C1 c1(OC(C)(C)C)c[nH]cc(Br)c1=O.Cc1cc2sc1-c1cccc(c1)C(=O)N2 c1(C(CC)CC)cc(C(=O)NCCC2(NC(c3sccc3C(C)C)=O)CC2)on1 c1(OC)csc(C(=O)NCCC2(NC(C3CCSCC3)=O)CC2)c1OC C(C(C)(O)C(=O)NCC1(CNC(C2CCN(CCF)CC2)=O)CC12CCC2)OC c1(NCCCC(C)NC(C2C(C)CC(=O)NC2)=O)cccc(F)c1[N+](=O)[O-] N1(C(C(C)c2ccsn2)=O)CCN(C(=O)C2=COCC2)CC1c1ccccc1Cl N1(C(Cc2cccc(C)c2)=O)CCCN(C(C2CCC2(F)F)=O)C(CO)C1 C1(NC(C(CC)F)=O)CN(C(c2ccc3c(c2)CCOC3)=O)Cc2nccn2C1 CCC(F)(F)C(=O)NCCC(C)NC(=O)CN1CCCC(N(C)C)C1 c1(CN(CC(F)F)C(C2C(=C)C2C(=O)OC)=O)ccncc1.C1C(=O)N1 C1(CNC(C2(OC)CC2)=O)CC(C)N(C(=O)CC=CCc2ccccc2)C1 N1(C(CS(CC)(=O)=O)=O)CC2CCC1CC2NC(C1CCC(C)C1)=O C(=O)(C1CCCc2nnn(C)c21)NC(C1CCCC1)CNC(CCCC#C)=O c1(NCC2ON=C(CC)C2)cc(N2CC=C(Br)CC2)nc(CC)n1 C(C(CN=c1cc(C)nc(N2CCCC(C)(CC)C2)[nH]1)C(C)C)N(CC)CC C1(CNC(C2(F)CN(C(CCc3cn(C)nn3)=O)C2)=O)CNC(=O)CO1 C=CC(C)CC(=O)NC1CCCN(C(=O)CCc2ccc(CO)cc2)C1 C1(NC(C(C)(C)NC(C=COC)=O)=O)CC2CC(NC(C3CCCSC3)=O)C1C2 c1(C(=O)NCC#CCNC(C(c2cccc(OC)c2)C)=O)ccc2c(c1)CCN2 N1(C(CCC=C)=O)CC(NC(c2ccc(NC(=O)NC)cc2)=O)CC(C)C1 C(=O)(C1=CCc2ccccc21)NC1CCCN(C(C(C(C)(F)F)(C)C)=O)C1 Cc1ncc(Br)c(C(=O)NC2COCC2CNC(=O)CNC(=O)C2CC2)n1 N1(C(C)=O)CCCCC1C(=O)NC(c1ccc(CN(C)C)cc1)C C1(C(=O)NCCc2cnc(C)s2)C2CCC(C2)N1C(=O)C(O)CC(N)=O CC1(C)CCCN(C(C2CCCC(O)C2)=O)C1C(=O)NCCCOC1CCCC1 c1(CC(=O)N(C(C)CCNC(C2CCCN2C)=O)C)ccnnc1O CCCCCC(O)CC(=O)NOCC(N1CCC2(CCSCC2)CC1)=O CC1CN(C(C2(C(F)F)CCCO2)=O)CC2(CCN(C(=O)C(C)(C)C(N)=O)CC2)O1 C=CCN=c1[nH]cc(C(=O)NCCCC(C)NC(c2cccnc2C)=O)s1 C1(CNC(CC=C)=O)CN(C(c2cnn[nH]2)=O)CCC1C(F)(F)F C1(C(=O)NC2CCN(c3ncn(C)c(=O)c3)C2)CC2(CCCC2)CO1 CC(C(=O)NCC1(NC(c2nnc(S)n2C)=O)CC(F)(F)C1)C(C)(C)C C(=O)(C(C(CC)CC)OC)N1CCCC(CC=C)(NC(=O)CC2CCC(=O)N2)C1 C=CC(CC)CC(=O)N1CCC(C(N2CCC3C(C(N)=O)C3C2)=O)(CC)C1 c1(CNC2(c3nnnn3C3(C)CC3)C(CCOC)CCC2)cc(C)ccc1OC c1(C(=O)NCC(CNC(c2ccccc2Cl)=O)CO)cncc2sccc12 N1(C(Cc2ccn(CC)n2)=O)CCCC(CC(=O)Nc2cnn(C(C)C)c2C)C1 c1(C(=O)NCCC(C)NC(C(C)OCCC#C)=O)c(C)noc1CCC c1(C(N2CCCC(CC=C)(NC(=O)CCF)C2)=O)cnc2nc(O)nc(O)c2c1 C(=O)(C(C)(C)CCC(=O)N1CCC(NC(C2C3CCCCC23)=O)CC1)OC CCC(CC(=O)NC1COCC1NC(=O)Cc1ccnn1C(C)C)C(F)F c1(C(N2CCC(N(C)C(c3ccncn3)=O)C2)=O)cc(=O)c2cc(Cl)ccc2o1 C(CC(C)C)(C(=O)NCCC(C)(C)C(=O)NC(C)CCOC)OC c1(C(=O)NC(C(c2ccccc2)NC(C2(SC)CCC2)=O)C)cc(O)cc(O)n1 c1(CCC)onc(C)c1C(=O)NCCC(C)NC(C1CCOC1=O)=O N1(N2C(CC=C)(C(=O)NC(CC=O)C)CCC2)CC23CCC2(COC3)C1 Cc1ccc(CCNC(=O)CC2(NC(C3CCCC34CC4)=O)CCCCC2)nc1 c1(C(N(CC(C)NC(CCC(C)N(C)C)=O)C)=O)cc2cc(Cl)ccc2[nH]1 Cc1cc(CSc2ccc(F)cc2)ccc1Cl.N12CCN(CC1)C(=O)N1CC2C1 C#CC1C(C(=O)NCCN(C(=O)CCCc2ccccn2)C(C)C)C1(C)C CCC(CNC(=O)CN1CCC(C(N)=O)CC1)(CC)NC(C1CCNC1=O)=O C(=O)(CS(=O)(=O)CC)NCC(c1cccnc1)NC(CCOCC#C)=O Cc1ccc(Br)c(C(N2C3CC2CN(c2ccncn2)C3)=O)c1 N1(C(C2C(c3cn(CC)nc3)C2)=O)CCC(C2CCN(C(C3CCC3)=O)CC2)C1 c1(OC)ccc2[nH]c(C(=O)NCCN(C(=O)CC3CCN(C)C3)C3CC3)cc2n1 N1(CC(C)(C)NC(C(=O)NC(C(c2cccc(Cl)c2)OC)C)=O)CCCCCC1 C1(CC)CN(C(=O)CO)CC12CC2.C(=O)(CCCOCc1ccccc1)N(C)C1CC1 C1(CC(NOCC=C(C)C)=O)CCCCN1C(=O)C(C1CC1)N(C)C C1(CC=C)(NC(=O)CCCC2CC2)CCN(C(=O)C(C)(C)Cc2cnn[nH]2)C1 c1(C(N(C)CC2(NC(C(C(C)O)C)=O)CC2)=O)c(F)cncc1Br N#Cc1ncc(C(=O)NC2CC23CC(NC(=O)C(O)C2CCCC2)C3)s1 C(=O)(CCC(C)(C)C(=O)NC1CCCCC1CNC(=O)CC(C)C(C)C)OC Cc1cn2ccnc(C(=O)NC(C)CNC(=O)CC3CSCCS3)c2n1 C1(C(=O)NC(CNC(c2[nH]cc(C)c2C)=O)C2CC2)CCn2nnnc2C1 C1(SCC2N(C(=O)OC(C)(C)C)CC2)SC(=Nc2ccccc2)NC1=O C(C(O)(CNC(=O)C(CCSC)NC(=O)Cc1ccsc1)CO)OC Cc1nn(C(C)C)cc1C(c1nnnn1C)NCCOCC1CC1 C12(C(N(C)Cc3cccc(O)c3)=O)CCCC1CCN2C(C1CCCC1O)=O O=C(C1CCc2c[nH]nc21)NCC1(O)CCCN(C(=O)C2=CCCC2)CC1 C1(C)(CC)CCN(C(=NCCN2CCCCC2)NCc2nc(-c3ccco3)cs2)C1 N1(C(CC2(OCCOC)CC2)=O)CCC(F)(CNC(C2CCOC2C2CC2)=O)C1 CCC(=O)CCC(=O)NOCC(N1CCCC12CCOCC2)=O N1(C(C2(CC#C)CC2)=O)CC(NC(C2CC(O)C2)=O)C(C2CC2)C1 c12nc(c(C)s1)C(=O)NCCCOCCN(C(C)C)C(=O)C2.CCC(=O)NC CC1(C(=O)NCC2CCCC2NC(c2cnn(CC3CC3)c2)=O)CCNC1=O CCC(C(=O)N1CCN(C(c2ccccc2I)=O)CC1)C(C)O C12(C(=O)NC3CCCCN(C(c4ccc(NC)cc4)=O)C3)CCCCC1C2(F)F N1(C(C2C(CCC)CCC2)=O)CC(NC(C2COC(=O)N2C)=O)CC(C)(C)C1 c1(C(C(=O)NCC(C(C)C)NC(C2(C)CCCN(C)C2)=O)O)cccc(Cl)c1Cl C(=O)(CCC(C)(C)C)NC(C1CCN(C(c2cccn2C)=O)C1)C c1(C(N2CCN(C(C(C3CCC3)OCC)=O)C(CF)C2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 Cc1nc(N2CCC(NCc3ccc(I)c(Cl)c3)C2)cc(C(F)(F)F)n1 C(=O)(C1=NNC(=O)CC1)NC(CC)CNC(c1csc(-c2ccncc2)n1)=O c1(CC(=O)NC(C(=O)NC(c2ncn(C)n2)C)C2CCCC2)ccc(O)nc1 c1(C(=O)NCCC(C)NC(c2cc(O)ccc2F)=O)cc2c(Cl)ccnc2s1 Cc1cccc(-c2cccc3sc(C(N4CCN(C(C)C)CC4)=O)cc23)c1C#N C1(C(=O)NC(c2ccsc2)CO)CC2(CC2)CN1C(c1ccc(F)cc1F)=O C12(CO)CC1CN(C(c1cc(CNC(C3(N4CCCC4)CC3)=O)on1)=O)C2 C(CC(C)C(=O)N(CC(=O)NCc1cnsc1C(N)=O)C)=CCC c1(C(N(C2CCC2c2ccc(F)cc2)CC(=O)NC)=O)ccc(OCCC#N)cc1 C1(CC(=O)N)C=CS(=O)(=O)C1.Cn1nncc1CC(N1CC(C(=O)NCCSCC)C1)=O N1(C(C(c2ccc(CC)s2)=O)=O)CCC2CN(C(C3CCCC(=O)N3)=O)CC12 C1(NC(C2(COC)CCCCC2)=O)CC2CC(C1)N(C(c1cc(Cl)no1)=O)C2 C=C1CC(C)(C(=O)NC(C2CCCCC2)CNC(c2cc(C(N)=O)[nH]n2)=O)C1 C(=O)(CC(C)CC(C)C)NCC(CC)NC(=O)C(CO)N(C)C C1(C(=O)Nc2ccc(O)nc2)C2CC1N(C(c1cc(-c3ccccc3)no1)=O)C2 Cc1nc2cccc(C(=O)N(C3CN(C(=O)C=Cc4ccsc4)C3)C)c2s1 c1(OC)ccc(Cl)cc1C(CO)NC(c1c[nH]nc1-c1cccc(Cl)c1)=O C(=O)(C1CCCc2ncc(C)n21)N1CCCC(C)(NC(C=CCC)=O)C1 N1(C(C(CC)(CO)OC)=O)CCC=C(C(=O)N2CCC(n3cncn3)C2)C1 N1(C(C(CC)c2ccccc2)=O)CCN(C(=O)C(C)CO)CC1CCO CCC(C)(C)CCNC(=O)CC=CCNC(C1COCC1C(N)=O)=O C(=O)(CCCCCN=[N+]=[N-])N1CC(C(=O)NCCCCC2C(C)C2)N(C)CC1 C1(CCC)C(O)C(=O)N1.c1(C(N(CCN(CC=C)C)CC)=O)c(C)cncc1F C1(C)(CC)C=C(C(=O)N2CCC(C)C(NC(=O)C(F)CC3CCOC3)C2)C1 CN1CC(C)(C(=O)NC2CCC(NC(=O)CCc3ccc(Cl)s3)CC2)CC1=O Cc1c(C(N2CCCC(NC(c3cnc(C#N)s3)=O)C2)=O)cncc1Br C1(NC(c2cc(OC)nc(F)c2)=O)CC2CC(NC(C3CC34CCC4)=O)CC2C1 C(=O)(CCC(=O)c1ccc(Cl)cc1)NCC(CNC(CC(C)C1CC1)=O)(C)O CCCCCCC(C)NC(=O)C(CCC)n1cccn1 c1(CC(C)NC(C(C)C)=O)ccc(CNC(c2scnc2C(C)(C)C)=O)cc1 C1(CNC(C(COC)(C)O)=O)CN(C(=O)C(F)=C(C)C2CC2)CC12CCC2 N1(C(c2n(CC)ccn2)=O)CC2(C1)CN(C(C1CC13CCCC3)=O)C2 CC1(NC(=O)Cn2nccn2)CCCCC1C(=O)NCc1ncsn1 CCC(C)(C)CCN=C(NC1CCOCC1)NC1CCCS(=O)(=O)C1 C=CCCC(C(=O)NCC(C)(C)C1CCCO1)NC(C1CC2(CCC2O)C1)=O N1(C(=O)CC2CC=CC2)CCC(C2CCN(C(=O)C3=C(Cl)CCOC3)C2)C1 CC(C)(C)C(O)CNC(C1CC1C(=O)NCC(=O)NCC1CC1C)=O CCC(C)(CO)C(=O)N1CCC(CCNC(c2cc(-c3ccco3)[nH]n2)=O)C1 C(=O)(C1Cc2ccc(C)cc21)NCc1c(C2CN(C(C(C=C)(C)C)=O)C2)ocn1 C(=O)(C1CCCc2cccnc21)NCC(C(C)C)NC(c1ccc(C)c(F)c1)=O C(C)(C(=O)NCCCCN(C(=O)COC1CCOC1)C)OCC=C c1(OC)cncc(C(=O)NC(C)(C)CC(=O)N2CCCC2CC2CC2)n1 C1(NC(CN(C(C(C)C)=O)C)=O)CC(F)CN(C(c2ccc(Cl)cc2)=O)C1 C(=O)(C(F)CC1CCCCC1)NC(=O)C=CC(=O)N(CCN(C)C)C.C1C=CC1 C1(CNC(C(CSC)OC)=O)CN(C(c2occc2Br)=O)CC(C)(C)C1 C1(C(N)=O)CCCCCN1C(=O)NCCc1nc(Cl)cs1.C(COCCS)NC=O C1(CCNC(C2C(COC)C2)=O)CC(F)(F)CN1C(c1cc(C2CC2)no1)=O c1(C(=O)NC2CCC(CCNC(=O)CCOC3CC3)C2)c(Cl)cccc1[N+](=O)[O-] NC1CC(CC(N2CCN(C(=O)C(=O)c3ccco3)CC2)=O)C(O)C1 C1(O)(CC)CCN(C(=O)C(CCSC)NC(c2cocn2)=O)C1 c1(C(=O)NC2(CC)CN(C(=O)CC(C)N(C)C)C2)ccc(C(C)C)c(C)c1 Cn1nnc(C(=O)NC2COCCC2NC(c2csnc2Cl)=O)c1N C1(CC)OCCC1C(=O)NCCOCCN(C)CCO.C(CCO)O CCCCCC(O)CC(=O)N1CCN(C)C(CNC(c2occ(C)c2C)=O)C1 C1(C(=O)NCCN(C(C2CCCC23CCC3)=O)CC)CC2(CCO1)CC2 N1(C(c2cc[nH]n2)=O)CCC2(CCOCC2C(N2CC(F)C(F)C2)=O)CC1 N1(C(c2cccc(CC)c2)=O)CCC(C)(C)C1CNC(c1cnc(CC)o1)=O c1(CNC(COCCC#C)=O)ccnc(C(=O)Nc2cnn(CCN(C)C)c2)c1 N1(C(C(=O)NCCCSC)=O)CCN(C2CCCN(C)C2)C(=O)C1 C1(CCOC)(NC(c2c(C)csc2Cl)=O)CCN(C(c2nc(O)c(C)s2)=O)C1 c1(C(=O)OCC)cc(CO)on1.C(=O)(COCCN(C)C=O)N.CCCSCCO Cc1nn(C)c(Cl)c1C(=O)NCCC1CCCN(c2ccnc(C3CC3)n2)C1 c1(OC(C)C)ccc(C(=O)NCC2C=CCN2C(=O)C(O)C(F)F)cc1 CC1OCCC1C(=O)NC(CC1CCCC1)C(=O)N(C)Cc1ccccn1 c1(NC(c2cc(-c3ccc(C(C)(C)C)nc3)c(F)nc2)=O)nccn2ccnc12 c1(CC)onc(C)c1C(=O)NCC(C1CN(C(=O)COC2CCC2)C1)F c1(C(=O)NC2CCN(CCNC(C3(C)COC(=O)N3)=O)CC2)ccc2c(c1)CC2 C12(C(N(C3CCCC3O)CC)=O)CCC(CC1NC(c1cn(C)c(=O)n1C)=O)C2 N#Cc1cc(F)c(CN2CCSCC2C(=O)NCC2CCCO2)c(Cl)c1 CCCCC(O)C(=O)NCCC1CN(C(=O)Cn2ccc(Br)cc2=O)C1 CCC1=NOC(C(=O)NC2CC(CNC(c3cnn(CCF)c3)=O)C2)C1 n1(CC(=O)N(CC(C)NC(c2nnc(C(C)(C)C)s2)=O)CC)nnc(=O)[nH]1 n1(CCC)ncc(C(=O)NCC2CC3CC3N2C(=O)C(C)C#N)c1C1CC1 C1(C(=O)NC2C=CC(C(=O)NC)C2)CC(F)(F)CN1C(C1CSCC(=O)N1)=O N1(C(CC(C(=C)C)OCC)=O)CC(C(=O)NC(CC2CC2)CC)C(C2CC2)C1 c1(C(=O)NC(C)C(C)(C)NC(C2CCC(=O)O2)=O)ncnc2c1OCCO2 c1(OCC)ncc(C(=O)NCCC(C)(C)NC(=O)CCc2ccncc2)s1 C12(NC(c3occ(C)c3C)=O)CCC1CN(C(=O)CN1CC(C)C1)C2 c1(C(N(CC(O)CNC(=O)CN2CCCC2=O)C)=O)c(F)cccc1Cl c1(C(C)C)cccc(C(N2CCC2CNC(=O)CCC2CCC(=O)NC2)=O)c1 N1(C(CCc2cc(C)[nH]n2)=O)CCCC(N2CCC2)C1 O=C1COC(c2ccc(NCCc3ccc(F)cc3)cc2)=N1 C1(NC(CCCC)=O)CCCCC1NC(C1CCOC1=O)=O CCC(CC)CCCC(=O)NC(CCC1CC1)C(=O)N(CC(C)C#N)C C(=O)(CCCCCCCC1CC1)NC(CNC(C1CN(CCC)C(=O)C1)=O)C c1(-n2c(C(c3scc(C)c3)C3CC3)nc(C3CCOC3)n2)ccc(F)cc1C C(CC(C)C)(C(=O)NCc1ccccc1CNC(c1nnc(Cl)cc1N)=O)OC N1(C(C2CCC(NC(C(C)OC(C)=O)=O)C2)=O)CCc2ncncc2C1 c1(COC2(CC(=O)NC3CN(C(c4sccc4Cl)=O)C3)CC2)ccccc1 Cc1cc(=NCCC2CCCC3(CCC3)C2)[nH]c(=NCc2cscc2C(N)=O)[nH]1 c1(OC)cc[n+]([O-])c(C(=O)NCC2(O)CC(NC(C3CCCCC(=O)N3)=O)C2)c1 C(=O)(CCCC(C)(C)C)NCCCN(C(=O)CCc1cncn1C)CC CCC(CC)CCC(=O)N(C)CCN(CC(C)C(C)C)C(=O)CCN(C)C N1(C(Cc2c(C)nc(S)s2)=O)CCCC(C)C1CNC(c1coc(C(N)=O)c1)=O CC1(C)CN(c2nc(Cl)c(C#N)s2)CCC1NC(=O)CC1CC=CCC1 CC(CN(C)C)CC(=O)N1CCC(F)(CNC(=O)Cc2cc(Cl)sc2Cl)C1 CC1Oc2ccc(C(=O)NC3CCCN(C(=O)CCc4ncc[nH]4)C3)cc2C1C C1(NC(Cc2c(OC)ccc(Br)c2)=O)CCCC2CN(C(C3CCCO3)=O)CC12 N1(C(C(C(C)O)NC(N)=O)=O)CCCC(NC(c2cc(C(F)F)[nH]n2)=O)CC1 N1(C(c2cccc(SCC#C)c2)=O)CCC(NC(=O)Cc2cscn2)C(C)C1 C1(C(=O)NCC2CC(OC)CN2C(c2ccn(CF)n2)=O)CC2(CCCC2)CO1 [N-]=[N+]=NC1CCN(C(=O)NCc2ccc(C(N)=O)cc2)CC1F Cc1cnc(C(=O)N(CCCNC(C2CCOC2C(F)(F)F)=O)CCO)c(C)c1 C1(CC)COC(C2(OC)CC2)CN1C(c1cc(C)nn1Cc1ccccc1)=O c1(C(=O)NCC2CC(O)CN2C(C2CC(O)CCO2)=O)ccn2ncnc2c1 c1(N2CCC(O)(C(C)NC(c3nc(F)ccc3Cl)=O)C2)nc2cc(F)ccc2o1 C1(NC(CN2C(C)CCC2)=O)CN(C(c2cc(Cl)sc2Cl)=O)CCC1F C1(C(=O)NC(C(=O)NC)C(C)C)C2CC3C(C2NC(=O)Cc2cn[nH]c2)C13 N1(C(CC2CC(CC)C2)=O)CC2(CCN(C(C3CSCCS3)=O)CC2)CC1C C1(C(=O)NC(C=C)CO)C(C2CC2)CCN1C(c1ccc(OC)nc1)=O c1(C(N2CCC(CNC(Cc3nc(N)sc3)=O)C2)=O)cnc(S)nc1 c1(C(N(CCC(C)NC(CCCCCC)=O)C)=O)cccc2sncc12 CC(C)CC(F)C(=O)N(C1CC(NC(C2(c3cccc(F)c3F)CC2)=O)C1)C Cc1cc(-c2nc(Cc3cccs3)n(CC3CC3c3cnccn3)n2)ccc1F N1(C(C2CCC(=O)NC2)=O)CCC2(CC1)CC(NC(C1COC1)=O)CCO2 C=CCC(CC=C)C(=O)NC1CCCC(C(=O)NCc2ccccc2F)CC1 CCC(C)C(C(=O)N1CC(NC(c2cnnn2-c2ccccc2Cl)=O)C(C)C1)OC C1(COC)CC(CNC(c2c[nH]c(=N)s2)=O)N(C(=O)C(C)n2cccn2)C1 CC(CCC(=O)N1CCC(C(C)C(=O)NC2(CO)CC(F)C2)CC1)N(C)C N1(C(CSSC)=O)CCC(N(C(=O)CCCC2CC2)CC)C1 C1(C(=O)NC2C(NC(CCC=C(C)C)=O)C2)Cc2ccc(Br)cc2C1 c1(C(N(C2CCN(C(C(COCC)C)=O)C2)CCO)=O)cc(C(F)F)ccc1F CCC(C)(C)C(O)C(=O)NCc1cc(C(N2CCOC(CF)C2)=O)co1 C(=O)(N=c1cc[nH]c2ccc(Br)cc12)C1N(Cc2cc(C#N)c(Br)cc2)CC1 C(C(C)(C)C(=O)N1CC(N(C(Cc2cn(CC)nc2)=O)C)C(F)C1)SC CC(C)CC(CNC(C1C=CC(NC(c2cccnc2Br)=O)C1)=O)N(C)C c1(C(N(C2C(C)CCN(C(=O)CO)C2)C)=O)cnc2[nH]cnc2c1 C1(N(C(C2CCC2CF)=O)CC)CCN(C(=O)CC(C)C2CCCCC2)CC1 c1(CC=C)cn(CC2CCC(NC(=O)CCSC)C2)nn1 Cc1ccnnc1C(=O)NC(C)C(c1ccccc1)NC(=O)CN1CCCC1 CN1CCCCC1CCC(=O)NC1CCOCC1NC(c1cncs1)=O C1(C)(CNC(c2c(CC(C)C)n[nH]c2)=O)CCC(NC(=O)Cc2nn[nH]n2)C1 C1(NC(Cc2cc(OC)ncc2)=O)CN(C(c2ccc(C)s2)=O)CCC12CCC2 c1(C(=O)Nc2cnc(C(=O)OC)s2)[nH]c(C)nc1C.C12CCC(C1)NC2 Cc1cc(C)c2c(Cl)c(C(N3CCC(CNC(C4CC(C)(O)C4)=O)C3)=O)sc2c1 c1(SCC)nccnc1C(N1CCC(O)(C(C)NC(C23CC(C)(C2)C3)=O)C1)=O C1(NC(C=Cc2ccc(SC)s2)=O)CN(C(=O)COC2CCCCC2)CC1(C)C c1(C(=O)NC(CCCNC(C2(C#C)CCCCC2)=O)C)cc(F)c(O)c(F)c1 CCCC(CCC)CC(=O)N1CCOCC1CN(C)C(c1c[nH]cc(F)c1=O)=O Cc1nsc(N)c1C(=O)NC1CCCC(NC(=O)COCCOCCO)C1 c1(C(=O)NCC(CO)NC(=O)CN2CC=CC2)ccc2nc(C(F)F)[nH]c2c1 CCC(CCC(=O)NCC(C)(CO)NC(c1ccc(C(=O)OC)cc1F)=O)OC C(CCC)(C(=O)N1CCC(OCC2CC(O)C(O)C2)C1)=CCC CC1CN(C(=O)Cc2cn(C)nn2)CC1CNC(C1CC1F)=O C1(NC(C)=O)CCN(C(c2csc(-c3ccco3)n2)=O)CC1.c12cn(nn1)C2 c1(C(N(CC(C)NC(C2C(OCC)C2)=O)C)=O)csc2ccc(C)cc12 C(=O)(CC(C)NC(C1CCN(CCCO)C1)=O)OC c1(C(=O)NC(C)C=CC(=O)NC2CC(C(N)=O)C2)ccc(N)c(F)n1 c1(CC)cc(C(=O)NCC(C2CC2)NC(C2CC2CF)=O)cc(O)n1 c1(C(N2CCN(CC(N)=O)CC2)=O)cn2cc(Cl)cc(Br)c2n1 c1(NC(C2CC(=O)OC2)=O)nc2c(s1)COCC2 Cc1ccc2cc(C(=O)NCC3CC3CNC(c3cccc(N)c3C)=O)[nH]c2c1 CC(C)CCC(=O)NC(C1CCCC1)CNC(c1cnn(CCF)c1)=O C1(Nc2ncc(-c3nc(C4(C=C)CCCCC4)on3)s2)CC2(CCCCC2)C1 C(=O)(CCCCCCNC(=O)CN1CCCC1)NC(C)COCC1CC1 C1(NC(CCCCC#C)=O)CN(C(C2CCN(OC)CC2)=O)CC(C)(C)C1 Cc1c(-c2cscc2C(=O)NCc2nnn(C)c2C(F)(F)F)cccc1O N1(C(CSCCOC)=O)CCOC(CNC(c2cc(CCCC#N)oc2C)=O)C1 C(=O)(C(C(C)C)NC(c1ccccc1)=O)NCC1CN(C(c2c(C)cco2)=O)C1 N1CCCC(O)CC1.C#CC1(CNC(=O)CN(C(=O)C(C)C)C)CCCC1 c1(C(N(C)CCOCCCNC(c2cnc(S)nc2)=O)=O)cc(F)cc(N)c1F Cc1ccnc(C(=O)NC2CC(NC(C3(F)CCCN(C)C3)=O)C2)c1F C(=O)(C#CC1CCCCC1)N1C(CNC(=O)Cc2ccno2)CC(COC)C1 C#Cc1cc(F)c(C(=O)NCCC(C)NC(c2cnnn2C)=O)c(F)c1 N1(c2[nH]c(=NCC3CC=CC3)cc(C)n2)CCc2c(ccc(Cl)c2F)C1 CC1C(C(=O)N(CCO)CC2CC2)CCN1C(c1csc(Cl)c1)=O N1(C(N(c2cccnc2Sc2ccccc2)C)=O)CCCC12CCCC2 C1(NC(C(CC)n2nccc2C)=O)CN(C(C2CC(C)=NO2)=O)CC2(CCC2)C1 C=CC(C)(C)CCNC(=O)C(C)(CSC)NC(=O)C=C1CCC1 Cc1ccc(C(N2C(=S)NC(c3nnn(C(C)C)n3)C2=O)=O)c(C2CC2)n1 Cc1noc(C(F)F)c1C(=O)NC1CCCN(C(=O)CC2CCCN2C)C1 c1(C(N2CC3(CN(C(C4CC4C4CCCC4)=O)C3)C2)=O)sc2sccc2c1Cl c1(OCC)cc(F)ccc1C(=O)NC1CCN(OCC)CC1 c1(C(N2C(C)CC(NC(c3c(C)cc(C)s3)=O)C2)=O)cc(C)c(Cl)cn1 Cc1nn(CC(N2CCCCC2CN(C)C(C23CCC2CC3)=O)=O)cc1Cl c1(C(C(=O)NC(C)(C)CCNC(=O)C2CC2)C2CC2)cccc2ccccc12 C(N=c1ccnc(NCc2cn(CCCF)nn2)[nH]1)c1ccc(CC(N)=O)nc1 C1(COC)(NC(=O)C(C2CC2)C2CC2)CCCN(C(C2(CO)CCSCC2)=O)C1 c1(OC)ccc(NC(=O)COC2CC(NC(c3n[nH]c4c3COC4)=O)C2)c(O)c1 c1(OCC)ncc(C(=O)NC2(CNC(=O)CCc3cc[nH]n3)CCCC2)cn1 C(C)(N=c1[nH]c2cc(F)ccc2o1)C1N(C(CC(=O)NC)=O)CCCC1 C(=O)(C(CCC)S(N)(=O)=O)NCC1CCCN1C(C1(CC#C)CC1)=O N1(C(C(COC)OC)=O)CCCCC1CNC(=O)CCCCN(C)C C(CC(=O)C1=C(c2cccc3cccc(CO)c23)OC1)OC C#Cc1ccc(C(=O)NCC(CCC)C(=O)NC2CCC(=O)NC2)cc1C c1(C(CNS(N(CCCOC)C(C)C)(=O)=O)O)cc(F)c(F)c(F)c1 Cc1nc2cccc(C(N3CCC(C)(C)C(NC(c4coc(Cl)c4)=O)C3)=O)c2[nH]1 N1(C(CCC2(C)CC2)=O)CC(NC(c2nnc(O)nc2O)=O)C2CCCC12 N1(C(C#CC(C)(C)O)=O)CC2(CCC2)CC1CNC(=O)CCCn1ccnc1 Cc1c[nH]nc1C(=O)NC(Cc1cn[nH]c1)C(=O)NC(c1cnn(C)c1)C C#Cc1ccc(C)c(NC(=O)C(CCOCC)NC(=O)C(C)CC=C)c1 c1(C(=O)NCC2N(C(C=CC(=O)OCC)=O)CC2)c(C)c(C)cc(C)c1C C(=O)(C1=NN(C)C(=O)CC1)N1CC(n2ncc(NC(c3noc(C)c3C)=O)c2)C1 N1(C(C23CC(OC)C2C3)=O)C2CCC1CN(C(=O)Cc1cc(Cl)cnc1C)C2 Cc1cnc(C=CC(=O)NCC=C2CCN(C(=O)C=Cc3ccccn3)CC2)[nH]1 Cc1c(C(=O)NCCCNC(=O)C(C)CC(N)=O)sc2[nH]cnc(=S)c12 C1(C(=O)NCC(CNC(c2c(CCC)[nH]cc2)=O)CO)C2CC3C(C2)C13 Nn1nc(C(=O)NC2CC3CCC2N3C(c2ccccn2)=O)c2ccccc12 c1(-c2cn(CC(CCNC(C3C(F)(F)C34CC4)=O)F)nn2)cccc(F)c1F Cc1cncc(C(=O)NC(C)CCN(C)C(C2CCC(F)(F)C2)=O)c1 CC1(C)CN(C(=O)CCC2CCCCN2C(=O)C#CC2CCC2)CCS1 c1(C(=O)NC2CC(CNC(C3(CC#C)CCOC3)=O)C2)cccc(N(C)C)c1 c1(C(C(=O)NCC(C2CCC2)NC(C(C)=CC)=O)(F)F)ccc(C)cc1 N1(C(CNS(N)(=O)=O)=O)CCN(C(=O)Cc2ccns2)C2(CCC2)C1 N#CC1(C(=O)NCC2CCCC(CNC(=O)Cc3cc[nH]n3)C2)CC2CC2C1 CC1(CNC(C2(C)CCCO2)=O)CCN(C(C2(C3CCCCO3)CC2)=O)C1 N1(C(CC2CCCN(C)C2)=O)CCC2C1CCN2C(c1cc[n+]([O-])cc1)=O CC1(C)CC(NC(=O)Cn2cnnc2)CCN(C(=O)Cc2cn(C3CC3)cn2)C1 c1(C(=O)NC2(CO)CN(C(c3ccsc3C(F)F)=O)C2)n[nH]c2c1CCSC2 N(C(=NCCN1CCCC1)NCc1cnc(-c2ccccc2)o1)C1CC(C)SC1 N1(C(c2c(CC)nc[nH]2)=O)CCCN(C(C2CS(=O)(=O)CC(=O)N2)=O)C(CO)C1 C12(C(N3C4CC(NC(Cc5c(C)cccc5)=O)C(C4)C3)=O)CC(C)(C1)OC2(C)C c1(OCC)ccc(NC(=O)C(C)C23CC(C2)C3)c2ccccc12 C1(=CC(=O)NC2C(CNC(C(C)(C3CC3)OC)=O)C2)CCN(C)CC1 CC(O)C(C(=O)NC(C)CN(C)C(=O)NC1CC12CCC2)NC(=O)C(C)(C)C CCCC(C#N)C(=O)NC1CC2(C1)CC(C(N(C)CC1(OC)CC1)=O)C2 C(CCC(O)C(=O)NCc1cccc(CO)c1)NC(c1cc[nH]c1)=O c1(CCC)cc(NC(=O)CSCC(F)F)ccc1Cl.N12CCCC(C1CC)C2=O N1(c2n(CC(C)OCC)nnn2)CCCC2(CCC(=O)NC2)C1 c1(C(N2CC(CCNC(C3C(CC)C3)=O)C2)=O)ccc(Br)cc1OC c1(C2(C(=O)NC3CCN(C(C4(C)CC4(F)Cl)=O)C3)CC2)ccc2nn[nH]c2c1 N1(C(=O)CCc2c(Cl)cncc2Cl)CC2CCCC(C1)N2C(C1CCCO1)=O N1(C(C(SC)SC)=O)CCC(NC(=O)C(C)CC2CCCC2)C1C c1(C(N2CCCC(C)(CNC(C(CC)(C)CO)=O)C2)=O)cc2c(cn1)OCCC2 C1(C(=O)NC2CCN(C(=O)C(Cl)=CCl)C2)CC2CCC(C1)C2O N1(C(C23CCC(OC)C2C3)=O)CC2(CC2)CC1C(=O)N(C)CC1CC(F)C1 C#Cc1ccccc1CN1CCC(C(=O)Nc2ccnc(C3CC3)c2)CC1 CCCC(CC)C(=O)NC(C)C(=O)NC1CCN(CCO)CC1 Cc1nc(NC(c2[nH]cnc2C#N)=O)ccc1-c1cncc(O)c1 N1(CC(C)C)CC(C(=O)NCC2CC3CC3N2C(C2CCOCC2)=O)CC1=O Cc1cc(CC(N2CC(N3CC(NC(C4CCCO4)=O)CC3=O)C2)=O)ccc1Cl c1(OC(CCC(C)OC(C2CCCCC2OC)=O)=O)cc(Cl)cc(Cl)c1 C(CN=c1ccnc(N2CCC(C3CCC3)C2)[nH]1)NC(c1ccccc1F)=O Cc1cc(NC(c2ccncc2Cl)c2nnnn2C(C)(C)C)ccc1F N1(C(c2ccnn2CCF)=O)CC2CCC1CN2C(C1CCn2nncc2C1)=O Cc1c(OCC(=O)NCC2CN(C(C3C=CCCC3)=O)CC2(C)C)cccc1Cl c1(C(=O)OC)cccc2sc(C(=O)OC(=O)C(c3cccc(Cl)c3Cl)OC)cc12 CCC(CCC(=O)NC(c1cscn1)CO)NC(c1ccc([N+](=O)[O-])o1)=O c1(C(=O)NC(CC)CNC(c2ccc(OC(C)(C)C)cc2)=O)ccc(F)cc1C N1(C)CC(NC(CC=C=C)=O)CC1(C)C.C(CCCC=O)C(=O)OC C=CC(C)(O)CC(=O)NCCC1CC(NC(=O)CCSCCC)C1 CC1CC(CNC(C2CCC23CCC3)=O)CCN1C(c1ccco1)=O C1(C(C)NC(=O)C=CC(=O)N(C)C)CN(C(=O)CSC2CCOC2=O)CCO1 c1(C(=O)NCCCNC(=O)Cc2cnccc2Cl)cc(Cl)cc([N+](=O)[O-])c1 N1(C(C(CC)c2ccccc2)=O)CC2CCOC2(CNC(=O)CC2CCCC2)C1 CC1CC2(CCN(C(c3ccc(Cl)[nH]3)=O)CC2)CN1C(=O)Cc1cocn1 C1(NC(CCOCC)=O)CCCCC12CCN(C(c1cnc(OCC)nc1)=O)C2 N1(C(C2CCC(C(=O)OC)CC2)=O)CC2CCC1(CNC(=O)C(C)N(C)C)CC2 CCC(O)C(C)C(=O)N1CC2CC(C1)C2NC(=O)CCCCCN(C)C c1(C(N2CC(C(C)NC(c3cnn(C4CC4(F)F)c3)=O)C2)=O)ccc(N)cc1O CC(C1COc2ccccc21)N(C(=O)NNC(=O)C(=O)Nc1ccccc1Cl)C CCCC(CCC)=CC(=O)NCC1C(C)CCN1C(c1cnoc1C)=O N1(C(C2(CC)COC2)=O)CCN(C)CC1CNC(=O)C=Cc1cnc[nH]1 c1(OC)ccc(C(F)(F)C(=O)NCC2CCN(C(c3cc(C)co3)=O)C2)nc1 CCCCCC(O)C(=O)N1CCCC1(C)CNC(c1cccc2ccoc12)=O N1(C(c2[nH]cc(C(N)=O)c2)=O)CCOCC(n2cc(C3(O)COC3)nn2)C1 c1(NC(C(C)N(CCC)C(c2ccc(C#N)cc2)C)=O)ccc2ccccc2c1 c1(C(=O)NCCC=C)cc2[nH]ccc2cc1-c1cc(SC)ccn1 O=C(CCN1CCC1)NOC1CCCCC1.C1(COCC(=O)O)CCCO1 CCN=C(NCC1(F)CCCCC1)N1CC2CCCC2C1 C1(N(C)C(c2ccccn2)=O)CCCN(C(=O)C(C2CCCCCC2)O)C1 CCCCC(CNC(C1CC(C)(C)CO1)=O)NC(=O)CCCn1c(C)csc1=O c1(COCC(=O)N(C2CCOC2)CCNC(C2CC(OCC)C2)=O)cccnc1 C1(CC(=O)NCCCOCCN(C(CN(C)CC)=O)C)CCCCO1 C(c1ccc(Cl)cc1F)=CC(=O)NC(CNC(CC12CCC(OC)(CC1)C2)=O)C C1(N(C(c2scc(CC)c2)=O)CC)CCCN(C(C2C(C)C2C)=O)CC1 C1(C(=O)NCCNC(=O)CO)(NC(C(c2ccn(C)c2)C)=O)CCCC1C c1(CC(=O)NCC2(NC(C3CCC3n3ccnc3)=O)CCC2)ccoc1 c1(C(=O)NCCC2N(C(C(CO)NC(N)=O)=O)CCCC2)nccc2n[nH]cc12 c1(C(=O)NC(CC)(C)CNC(=O)C(C2CC2)SC)cc2c(o1)CCCC2 N1(C(C(C(C)C)(C)O)=O)CCC2(CC1)CN(c1ncc3ccsc3n1)CCO2 c1(C(N(C2CCN(C(C3(CCOC)CC3)=O)C2)CCC)=O)n[nH]c(C2CC2)c1Cl C(N=C(NCC1CCCO1)N1CCCCC1)C1CC(=O)NCC1 c1(N2CC(=CCC)C2)nc(=NCCN(C)C2CC2)[nH]c2cc[nH]c12 N1(CC(=O)NC)C(=O)NC2(CC(c3ccc(CCCC(=O)O)cc3)C2)C1=O O=S(=O)(c1cccc(=NCCCc2cccs2)[nH]1)N1CC2CCC2(CO)C1 C1(NC(C2C(CCOC)C2)=O)CCN(C(c2cnn3c2OCCC3)=O)CC(O)C1 C1(N(C(c2cccc(C(C)=O)c2)=O)C)CCN(C(c2ocnc2C)=O)CC1C CC1=C(C(=O)NC2CN(C(C3C(C)C3C)=O)CC2F)CCS1(=O)=O C1(C2CC2)(C(=O)NCc2c(C)cccn2)CN(C(=O)C(=O)N(C)C)C1 Cc1cc(C(N2CCCC2CNC(C2CCCC(F)C2)=O)=O)c2c(c1)CCCN2 N1(C(C(C(CC)O)C)=O)CC(N=c2ccnc(-c3cccc(C)c3)[nH]2)C(C)(C)C1 c1(CC)nc(C)ncc1C(=O)NC1CN(C(=O)CC2CCCO2)CC1(C)C C1(NC(c2cc(C)c(C#N)cc2)=O)CCCOC12CCN(C(=O)C=C(Cl)Cl)CC2 CCCC(C)(C)CC(=O)N(C(C)CN(C)C(C1(C2CC2)CC=CC1)=O)C c1(C(=O)NCC(CC(C)C)NC(C2CCC(C)(C)OC2)=O)cc(Cl)c(Cl)cc1N c1(N(C2CC3CNC2C3)C(C2CC(O)C2)=O)ccc2c(c1)OCCO2 CCCC(C)(O)C(=O)N1CC(C(C)NC(c2ncncc2OC)=O)C1 C#CC1(O)CCN(C(C2CCN(C(c3c[nH]nc3CCC)=O)C2C)=O)C1 c1(CNC(COC)=O)nn(-c2ccccc2)cc1C.C1C(O)C(=O)N2CCC(C2)O1 C1(C(=O)NCC(F)(F)C(N)=O)(CNC(CC=CC)=O)CC12CCC2 Cc1ccc(C(N2CC(F)(F)CC2CNC(C2CCN(C)C2=O)=O)=O)c(N)n1 C#Cc1ccc(C(N2CCCC(C)(NC(=O)C(C)C(O)CC)C2)=O)cc1Cl c1(CCC(=O)NCCC(C)NC(C2CCN2C2CC2)=O)nnc(-c2ccsc2)o1 CC(C(=O)NC(C)(C)CCNC(c1cnn(C2CC2)c1)=O)C(F)(F)C(F)F Cc1nn(C)c(C(F)F)c1C(=O)NC(CNC(C1(CO)CCCO1)=O)CC(C)C C1(C(=O)NCC2C(C)CN(C(=O)CC3CC3(C)C)CC2)CCC2CCCCC2C1 c1(C(N2CCC(NC(COCCCC)=O)C(C)C2)=O)c(F)cc(C)cc1Cl C1(CNC(C2(C)COC2)=O)C(C2CC2)CCN1C(=O)C(O)Cc1cnc[nH]1 N#Cc1ccccc1OC1CCN(C(=O)CCc2cc(Br)ccc2F)CC1 Cc1ccc(F)cc1CC(=O)NCC1C=CC(NC(=O)CCOC2CCCC2)C1 c1(C(=O)NC(CCN(C(C(C)OCCC=C)=O)C)C)cc(C(C)C)nc(O)c1 CC1=C(CNC(=O)C(C)N(C(c2n[nH]nc2C)=O)C2CC2)COCC1 Cc1cc(C)c(C(N2CCCCC2CN(C(=O)CCNc2ccccn2)C)=O)s1 CCCC(C#N)C(=O)NC(C1CCN(C(=O)C=CCF)CC1)(C)C c1(C(=O)NC2C(NC(C3(SC)CCC3)=O)CCC2)cc(C#N)ccc1Br C(=O)(C(C)S(C)(=O)=O)NC(C(=O)N(C1CCCNC1=O)C)c1ccco1 c1(C(=O)NCC2(C)CN(C(c3cc4ccccn4n3)=O)C2)ccc2nc[nH]c2c1 C1(CNC(=O)CCn2ccnn2)CCCC1C(=O)NCC(N1CCCC1)C Cc1cc(N2CCCN3CCCC23)ncc1S(=O)(=O)NC1CC(C)n2ccnc21 O=C(NN=c1ccc2nncn2[nH]1)NC1CCC2(C(=O)O)CCC12 C(CCCC(C)(C)C(=O)NNC(=O)C1CCCS1)NC(CC1=NN(C)C(=O)C1)=O N1(C(C2C(CC(C)(C)C)C2)=O)CC2CCC(C1)N2C(C1(C)CSC1)=O Cn1c(CNC(=O)C(=O)NCc2conc2C(F)(F)F)cnc1[N+](=O)[O-] CC(C)C(C(=O)NC1C2CCC1CC2)C(C)NC(=O)CCc1cnn(C)c1 Cc1cc(=O)c(C(=O)NCC23CC(CO2)N(C(c2cnc(C#N)s2)=O)C3)cn1C c1(OC)nc(C(=O)N(C2CCCCC2NC(c2ccc(F)s2)=O)C)cc(O)n1 c1(COCC)nc(C(=O)NCC2CCCC2NC(=O)Cc2cc[nH]n2)cs1 N1(C(C2N(C(=O)OC(C)(C)C)CCC2)=O)CC2CC1CN2C(=O)CC1CC(F)C1 C1(F)(CNC(C(Cn2ccc(C)n2)C)=O)CCCN(C(c2ccc(Cl)s2)=O)C1 C#CC1(C(=O)NC2CCCC(NC(=O)CCc3cnn(C)n3)C2)CCCC1 N1(C(C(C)CN2CCOCC2)=O)CCC(C(=O)OC(C(=O)NC2CC2)=O)C1CO c1(CC)ccc2c(c1)COC2.N12CC(OCc3n(CC=C)cnn3)OC1C2.OC C1(n2cc(C(C)N(C)C(c3c[nH]c(Br)c3)=O)nn2)CCCN(C(=O)OC(C)(C)C)C1 c1(CC(=O)N(C2CCC(NC(C=NOC)=O)CC2)C)ccc2ccccc2c1 Cc1ccc(CN2CC3C(C2)N3C(C2CCC(=O)NC2)=O)c(F)c1F N1(C(c2c(OC)cncc2)=O)CCCN(C(c2ccc(F)cc2F)=O)C(CO)C1 C1(C(N2CC3C(CO)C3C2)=O)CCN(C(=O)C2COCC2O)O1 C1(C(=O)OCC)(C(=O)NC2CCCC2NC(c2ccc(OC)s2)=O)CCCCC1 Cc1cnc2c(C(N3CC4(CC(NC(C5CCNC5=O)=O)CO4)C3)=O)cccn12 N1(NCc2ccc(-c3c(C)cccc3)cc2)CC2(CCOCC2)CC1C(=O)O N1(C(C2CCCC(C)O2)=O)CCC2(CC1)CN(C(=O)CCCC(C)(C)C)C2 c1(C(=O)NCC(CO)NC(c2c(C)coc2Br)=O)c(C)nc(=N)[nH]c1C N1(C(C=CC=CC)=O)C(CC(=O)NC23COCC(C2)C3)C2CCCC12 N1(C(C2C(C)(C)C2)=O)CCC(N(C(=O)Cn2nccn2)CCO)C1 C1(NC(c2cn(CC)nn2)=O)CN(C(=O)C(F)(F)c2ccnn2C)CCC1F C12(C(=O)NC(CNC(c3c(C)cccc3)=O)CO)OCCCC1C2(F)F c1(OC)cc(N)ccc1C(=O)NC1CCC(CNC(C2CC=CCC2)=O)CC1 c1(C(C)C)nccc(C(N2CCOC(C(C)NC(=O)CC3(C)CCCC3)C2)=O)n1 c1(C(C)Nc2c(OCCOCC)cccc2)ccc(C)n(C)c1=O c1(C(N2C(C)(C)C(CO)C2)=O)cc(O)nc2c1CN(C(C1CC(F)C1)=O)CC2 Cn1cc(C(N2CCC(CC3CC(C(=O)OC4CCCC4)C3)C2)=O)nn1 O=S(=O)(c1ccnn1-c1ccccc1C(F)(F)F)NC1CCCC2CC12 CC1NC(=O)OC12CN(C(=O)CC(C(F)(F)F)NC(=O)CC(Cl)Cl)C2 c1(C(N(C(CNC(COCCC#C)=O)C2CC2)C)=O)cc(Cl)c(Cl)s1 C1(CNC(C(C)OCCN(C)C)=O)N(C(C2CCC(=O)N2C)=O)CCCC1(C)C Cc1c(N)ccc(C(=O)NC2CN(C(=O)C=Cc3ccoc3)C2)c1F Cc1nn(CCC(=O)NCC(O)CN(C)C(c2ocnc2C)=O)c(C)c1[N+](=O)[O-] c1(C(=O)NCCC2(NC(C(C3CCC(=O)N3)C)=O)CC2)ccc(Br)c(O)n1 C(C(CCC)C(=O)N1CC=CC1CN(C)C)NC(C1C(=C)C1)=O c1(C(=O)NC(CN(C(C(Cc2c(C)nc[nH]2)O)=O)C)(C)C)cc(F)cc(F)c1N c1(CC(=O)N(CCCNC(c2ccon2)=O)C)cc(Cl)cs1 N1(C(C2(C)CNC(=O)C2)=O)CCC(O)C(NC(c2cccc(C3CC3)c2)=O)C1 N1(CCN(C)Cc2ccc(OC3CC3)cc2C(=O)O)CC(=O)N(C)C1=O N1(C(C2CN(CC)C(=O)C2)=O)CCN(C(=O)Cc2cncn2C)C(C)C1 C#CC1(C(N2CCCOC(CC)C2)=O)CCN(C(=O)C=CC2CCCN2C)C1 C1(NC(c2ccc(C#C)cc2)=O)CN(C(C2(NC(N)=O)CC2)=O)CC2(CCC2)C1 Cc1ccc(C(=O)NC(C2CCN(C(c3nonc3C(C)C)=O)C2)C)nc1 c1(COC)nc(C)cc(=NC2CN(C(=O)CCn3cccnc3=O)CC2C)[nH]1 C1(C(N2CCC(F)(CNC(Cc3cncc(C)c3)=O)C2)=O)CC2(C1)CC(C)C2 N1(C(c2ncn(CCNC(C(c3ccccc3)C)=O)c2)=O)CCOC(C)CC1 N1(C(Cn2nnc(=N)[nH]2)=O)CCN(C(=O)CNC(=O)C=CBr)CC1 N1(C(C2(C=C)CCC2)=O)CCCCC2(CCN(C(=O)Cc3cnns3)C2)C1 C(C(CO)(CO)NC(=O)COCC(=O)OC)N(C(CCCOCC=C)=O)C N1(C(CSC(C)C)=O)CC2(C1)C(NC(C13CC(C)(CO1)C3)=O)CCS2(=O)=O C12(C(=O)NC(C3CCN(C(=O)CCc4cncn4C)C3)C)CCCC1C2(F)F N1(C(CCCC(=O)OCC)=O)CCC(NC(c2ccncc2)=O)C(CO)CC1 c1(C(=O)NCC(C)(C)NC(c2cn(CCOC)nc2C)=O)cc(O)nc(O)n1 N12CC(CC(O)C1)NC(=O)C(F)(F)C(F)OC2=O.C(C)(C)(C)OC(C)C CC1(O)CCN(C(c2cc3c(s2)CCC3)C(=O)NCC2CC2)CC1O C12(NC(CNC(CC)=O)=O)CN(C(=O)C=Cc3cocn3)CC1CS(=O)(=O)C2 N1(C(C(C)Cc2cnn(C)c2)=O)CCC(NC(=O)Cc2cnsc2)C12CC2 C(=O)(CCC(C)(F)F)N1CCC(C(N(CC(C)C)C)=O)(CF)C1 c1(CC(=O)N(CCN(C(=O)CC2CCC(C)O2)CC)CC)cnn2c1OCCC2 n1(C(C)OC)nc(C)cc1C(=O)NC(c1nc(-c2ccccc2C)no1)C c1(OC)ccc(CN2CCC(O)(C(=O)Nc3cccc(C)c3Cl)C2)cc1O c1(C(N2CC(CC(C)NC(c3cc(Cl)on3)=O)C2)=O)sccc1C(F)F C1(F)(C(=O)NCC2(OC)CCC2)CCCN(C(C2(C)CCCCO2)=O)C1 c1(-c2cn(CC3N(CC(N4CCC(N5CCC5)C4)=O)CCC3)nn2)cc(Cl)ccc1F c1(CC(=O)NCCC2(C)CCN(C(C3CC(C)C3)=O)C2)ccc2c(c1)OCO2 C(=O)(CC1=CCOCC1)N(C)CC1(CNC(c2ccn(C3CC3)n2)=O)CC1 C(=O)(CCCCC(C)(C)C)N1CC(C)(C(=O)NCCCC(C=C)(C)C)CC1(C)C CC1CCN(C(=O)CCCCN2CCOC2=O)C(C)C1CO.n12cc(nn1)C2 N1(C(C(c2cnn(C)c2)C)=O)CC(NC(=O)CCc2ncco2)CC12CCCC2 CCCC(CNC(=O)C=Cc1ccoc1)C(=O)NCCc1c(O)n[nH]c1C c1(CC)nc(NCC2CCC(NC(c3c(F)cccc3Cl)=O)C2)c2ccsc2n1 c1(C(=O)OCCc2ccc(CC)cc2)cc(I)c(Cl)cc1N N1(C(c2cc(=O)n3ccccc3n2)=O)CCc2ncc([N+](=O)[O-])cc2C1 c1(C(=O)OC)ccc(S(=O)(=O)Nc2cc(C(=O)OC)c(Br)c(C)c2)cc1 Cc1cc(=NC(=O)C2CC(C)CN2Cc2cccc(Br)n2)[nH]c(C)c1C#N N1(C(C(C)N2CCCC2)=O)CC=C(CC(=O)N2CCC(C)C(CO)C2)CC1 C12(CNC(=O)C3=CCSC3)CCC(NC(=O)Cc3csnn3)(CC1)CO2 c1(OC)ccc(CN=C(NCC(C)C)NCc2nnc(SC)s2)cc1.C(C)C C1(CNC(CC(C=C)C)=O)CN(C(=O)C(C2CCCCCCC2)O)CCCO1 C(=O)(CCCCC(F)F)NCCC(N1CC(C)C(O)C(C)C1)=O c1(C(=O)Nc2c(NC(C3CC3N)=O)cc(OC)nc2)cc(Cl)c(O)cc1F c1(C(C2CCCO2)C)cn(CC2CCCN2C(=O)COC2CC=CC2)nn1 Cc1ccc2c(=NCCN(C)C)[nH]c(=NC(C)c3nnc4n3CCCC4)[nH]c2c1 CC(c1cccnc1)=CC(=O)OC(C)C.N12CCCC1C=CCNC2=O N1(C(C2N(C)CC2)=O)C2CCC(C2)C1CC(=O)NCCC(O)CO c1(OC)ccc(CC#N)cc1NC(=O)NCC(c1ccn(C)n1)C CN1CC2OCCN(C(=O)CCCNC(c3ncn4ccccc34)=O)C2C1 c1(C2C(C(=O)NC3CCC(NC(COCCCC(C)C)=O)C3)C2)ccc(O)cc1 C1(NC(CNC=O)=O)CCN(C2CCN(C(C3CC(F)(CO)C3)=O)CC2)CC1 CC1=C(C(=O)NC2CCN(C(=O)CC3CCCC3O)C(C)C2)CCC1 N1(C(CCC)=O)CCCC1C(=O)N(C)CC1CCCN1C(C12CC(C1)C2)=O C(C)(C)(C(=O)NCCOCCO)OC.C12CCCN1C2=O c1(CC(=O)NC2CCC(NC(CN(C)C(=O)C3CC3)=O)CC2)c(Cl)cccc1Cl CCCCCC(C)CCNC(C)C(=O)NC1CCCCC1 C=CC(CC)C(=O)NCC(CC1CCCC1)C(=O)N(C)CCC1CCOCC1 C(C1=NOC2CCCC12)NC(C1C=CCN(C(c2n[nH]c(=N)[nH]2)=O)C1)=O N1(C(c2cn(CCOC)nc2)=O)CCOCC1CCNC(C1CCCC1(F)F)=O Cc1cnc(C=CC(=O)NC2COCC2CNC(=O)CC23CC(C2)C3)[nH]1 CC(C)CC(C(=O)N1CCN(C)C2CC12)ONC(=O)C1CC(n2ccnn2)C1 c1(C(N2CCC(C(=O)NCCCC(=O)NC)CC2C)=O)cccn2nccc12 N1(C(c2n(CC)nnc2)=O)CCCC(C)(NC(=O)CCc2cnco2)C1 C(=O)(C(C)(C)C(F)(F)F)N1CCN(C(c2cncc(OC)n2)=O)C(C2CC2)C1 c1(C(=O)NC2C3(CC(NC(C(C)SCCCC)=O)C3)C2)cn2c(n1)SCC2 N1(C(C2C(CC)OCC2)=O)CCCC2(CCN(C(c3n[nH]c(C)c3F)=O)C2)C1 C(CC)(CC)(CCNC(c1ccc(C(C)=O)cc1)=O)NC(C(CC=C)C)=O C(c1c(F)ccc(Cl)c1F)=CC(=O)NC1C(NC(C(C)c2cccs2)=O)CC1 Cc1nn(C)c2c(NCc3ccc(Cl)nc3)nc(=NCCCOC(C)(C)C)[nH]c12 c1(C(=O)NC2C(NC(C(COC)OC)=O)CCCC2)cccc2c1NCCC2 N1(C(C(C)OC)=O)CCC(CNC(c2ccccc2O)=O)C12CC2 N1(C(C(C)Cc2ccnn2C)=O)CCSCC1CCNC(=O)C=C1CCCC1 C(=O)(C(C)(C)CCCF)N1CC(C(C)NC(C=CC(CC)C)=O)OCC1 C1(NC(=O)NC(CN(CCCC)C)(C)C)CCCC(O)C1 C(CCO)(CC(C)C)NC(C1(NC(c2c(OC)nn(C)c2)=O)CC(O)C1)=O C1(C2CCCN(C(c3ccc(N)c(C)c3)=O)C2)(NC(C(CC)C(C)O)=O)CC1 c1(N2CCN(C(CCN(C)CCO)=O)CC2)nc(=N)[nH]c(=NCC2(Cl)CC2(F)F)[nH]1 CCC(O)C(C)(C)C(=O)N(C1CCN(C(C2CCCOC2)=O)CC1)CCOC C(=O)(CC(O)C(C)C)NC(CCN(C1CN(C2CCOCC2)C1)CC)(C)C N1(C(C2C(C)C2)=O)CC=CC(NCC(=O)OC(c2ccc(CC(N)=O)cc2)=O)C1 C1(CCNC(C2(n3cncn3)CC2)=O)CC2CC2C1.C12(CC1)C(=O)NC2 c1(C(N2C(CNC(C(C(C)C)OCC)=O)CCCC2)=O)cc(=O)n2ccsc2n1 C1(N(C)C)(C(=O)NC2CCC(NC(C3OCC3(C)C)=O)CC2)CCCOC1 c1(-c2ccc(C3(C(=O)OC)CC3)cc2)ccc(NC(=O)NCC(C)C)nc1C C(C)(CCCC(=O)O)NC(c1cnn(-c2c(OC)cccc2)c1N)C N1(C(=O)OC(C)(C)C)CCCC(NCC(C(F)(F)F)NC(=O)C(O)C2CC2)CC1 C(=O)(CCC(C)CN(C)C)NCC1(C(N(C)Cc2c(C)n(C)nc2)=O)CCCO1 c1(CNC(C2CSC3(CNC3)C2)=O)cn2c(Br)cccc2n1 N1(C(c2n(COC)ncc2)=O)CCCCC1CNC(=O)C(C)c1ccsn1 C1(C(N2CC=CC(C(N3CCC(F)CC3)=O)C2)=O)(CC)CCCCC1 c1(CNC(C(C(C)(C)C)c2nn[nH]n2)=O)cn2cc(Cl)cc(Cl)c2n1 c1(C(=O)NCC2C(NC(C3(CC=C)CCC3)=O)C2)ccc2ncnc(O)c2c1 C(CCC(N)=O)(C(=O)N1CCC(NC(c2cc(F)c(Br)cc2C)=O)C(F)C1)OC c1(C(=O)NCC2(C)CC(NC(C3CCC(CC)CC3)=O)C2)nc(C)c(C)nc1C c1(C(=O)NCC23C(CN(C(C(CCCC)OC)=O)C2)CC3)cncc([N+](=O)[O-])c1 c1(C(=O)NC2CC(NC(C(C)NS(CC)(=O)=O)=O)C2)cn2c(n1)CCC(C)C2 c1(C(C(=O)NCC(=C)C)N(C(C)Cc2ccccc2)C)cncc2ccccc12 c1(C(=O)NC2C(OC)CN(C(c3ccc(C#N)o3)=O)C2)cc(F)c(F)cc1Cl N1(C(C(C(=C)C)(C)C)=O)CC2CC(C(=O)N(C)C(c3ccncc3)C)CC2C1 n1(CC)ccc(=NC(C)(CCc2cc3ccccc3o2)c2nnnn2C(C)C)[nH]1 Cn1ccc2ccnc(C(=O)NCC3CCCN(C(C4(C)CC(F)C4)=O)C3)c12 N1(C(CSc2cccc(OC)c2)=O)CCN(C(=O)CC(F)F)C2CCC12 N1(C(c2c(C)snn2)=O)CC(CC(=O)N2CC2CN(C)C)C2(CC2)C1 N1(CC)CCOC(C(=O)NCC=CCNC(=O)CCc2ncc[nH]2)C1 C(CNC(C1CCN(c2ccccc2F)C1)=O)(C(F)(F)F)OC C1(F)(CNC(C2CC3CC3C2)=O)CN(C(=O)CCc2nc(-c3cccs3)no2)C1 c1(CNC2CCC(C(=O)NCc3cccc(C)c3F)OC2)c(Br)cc(F)cc1Br CC1CCN(CCC(=O)NC(C)C(C)NC(=O)Cc2cscn2)CC1 C1(NC(c2c(C)csn2)=O)CCOCC1NC(c1nnc(S)n1C)=O c1(C(=O)NCC(C)(O)CNC(=O)C=CC(=O)N(C)C)ccc(Cl)c([N+](=O)[O-])c1 C1(CC(=O)NC2(CNC(C(N)=O)=O)CCCC2)CCCC12CC2 Cc1ccc2ncc(NC(N3CC(C(O)CC(C)C)C3)=O)n2c1 c1(CC(=O)NCCCOCCNC(C2COC(=O)O2)=O)ccsc1Br C12(NC(C=C(C)Cl)=O)CCC(CNC(c3cc(F)cc(C)c3N)=O)(CC1)CC2 c1(C(C)C)c(C(N2CC(CO)(NC(=O)Cn3cc[n+](C)c3)C2)=O)cnn1C C1(CC(=O)N(CC(C)(C)CNC(=O)CC2C=CCCC2)C)Cc2ccccc2O1 C1(NC(C2(n3cccc3)CC2)=O)COCC1NC(C1CC1F)=O c1(C(N(CCNC(C2CC2(C)C)=O)CC)=O)cnc(C(F)(F)F)s1 c1(C2CCN(C(C(CCCC)NC)=O)CC2)nc2ccccc2[nH]1 N(C(=NCCSC1(C#N)CC1)NCC1CCOCC1)C(CC)C C(=O)(C1=C(CC)OCCC1)NCCCN(CCC)C(c1ncccc1Cl)=O c1(NC(C2C(C(=O)OC)CCCC2)=O)ccc2c(Cl)ncc(C)c2c1 C1(NC(C(C)(C)CF)=O)COC2(CCN(C(=O)CCc3cccnc3)CC2)C1 Cc1csc2ncc(C(=O)NC(C)CN(C(=O)C=Cc3ccoc3)C)n12 c1(C(N2CC(C)N(C(=O)C(=Cc3cccn3C)F)CC2)=O)cnc2cc[nH]c2c1 C1(C(N2CC(NC(CCc3ccc(C)s3)=O)C(O)C2)=O)CC12CCCCCC2 C1(NC(C=CCC2(NC(C(C)CN(C)C)=O)CCC2)=O)CN(C)C2(CCC2)C1 c1(C(N2C(C(=O)Nc3c(C)cc(F)nc3)C=CC2)=O)cc2cccnc2[nH]1 c1(OCCC(=O)N(C)CCNC(=O)CO)ccc(Cl)cc1.C(=O)(C(C)(O)C1CC1)N n1(CC)cc(C(=O)NC2(CCCNC(c3ccoc3C(C)C)=O)CC2)cn1 C1(C(=O)NC2CCCN(C(CC(C)C(F)F)=O)C2C)C2CCC1(C)C2(C)C c1(CC(=O)N(C(CC)C(=O)OC)CCC)csc2nccn12 C12(CNC(C3(OC)CCC3)=O)CCCN(C(=O)CCOCC(C)C)C1C2 N(C1CCc2cccnc21)C(C1C(O)CCN(Cc2ccc(C(=O)O)cc2)C1)=O C1(OC)CN(C(c2cc3n(n2)CCO3)=O)CC12CC2.C12CC(C1)CNC2=O C=CC1COCCN1C(C12CC1CCN2C(c1cc[nH]c1)=O)=O c1(CNC2(CC(N3CCC(CCCO)CC3)=O)CCC2)c(F)ccc(F)c1O N1(C(C2CCC(=O)C2)=O)CCCN(C(C2OCC3COCCC23)=O)CCC1 C1(O)(CNC(c2cc(Br)ncc2Br)=O)CCCN(Cc2cnc(Br)s2)C1 Cc1ccc(CNC(c2cc(CNC(=O)CCOCC(F)F)cs2)=O)cc1C n1(CCC(N2CC(O)(C(C)NC(C=C(C)C3CC3)=O)C2)=O)nc(C)cc1C CC1CCC(C2CCC2)CN1C(=O)CN1CC(C)(c2ccc(Br)cc2)C1=O C1(C(=O)NCCc2ccc(CNC(C3CC=CCC3)=O)cc2)C2CC3C(C2=O)C13 C(=O)(C(=O)N=S(C)(C)=O)NCC1(C)CCCN(C(C(CN(C)C)O)=O)C1 c1(CN2CC(NC(c3cc(O)ccc3Br)=O)C(O)C2)cc(F)cc(Br)c1 CCC(C)(C)C(=O)N1CC(NC(=O)CCc2ncco2)C(c2cncn2C)C1 c1(C(N(CC(=O)NC2CN(Cc3ccccc3)C2)C2CC2)=O)cc(F)cc(F)c1F CC1Cc2ccccc2C1Nc1cc(NC2CCN(CC3CC3)C2)ncn1 C(=O)(C(C)CCCC(C)C)N(CCOC)CCNC(C1CCCC(=O)CC1)=O c1(CNC(c2cc(OC)ncc2-c2ccn(C)n2)=O)cc(F)c2cc[nH]c2c1 C(=O)(C(C(C)C)n1cnnn1)NCC(CCC)NC(c1cc(Cl)n(C)n1)=O CC(F)(F)CCC(=O)NCCOCCNC(c1ncnn1C1CCOCC1)=O N1(C(C(CC=C)(C)C)=O)CCC(NC(=O)CC2CN3CCC2CC3)CC(C)(C)C1 c1(C(=O)NC)ccc(C(=O)NCCC(=O)NC2CC(F)(COC)C2)cc1 CCCCCCC(=O)N1CC(CNC(c2n[nH]cc2F)=O)OC(C(F)(F)F)C1 Cc1cc2c(cc1C)OC(COC(C1CC(=O)CO1)=O)C2 N1(C(c2c(O)cccc2Cl)=O)CCCC2C1CCN2Cc1cc(O)cc(F)c1 C1(C(N2CC(C(C)(C)C#N)C2)=O)CN(C(=O)CC2(O)CCCCC2)CCO1 c1(OC)ccc2c(c1)OC(C(=O)NC1(c3ccc(C#N)[nH]3)CC1)C2 C1(NC(c2ccc(OC)c(Br)c2)=O)CC2CC1CN(C(=O)CC(C)SC)C2 N1(C(c2nc(OCC)oc2)=O)CC(CNC(C2(c3ccno3)CCC2)=O)CC1C C(=O)(CS(=O)(=O)CC1CCCO1)N(C1CN(C(CNC(CC)=O)=O)CC1O)C O=C(C(Cc1cccc(Cl)c1)CCCO)NC1CC2OCCC12 C1(NC(=O)Nc2nc(COc3ccc(F)cc3)cs2)CC2(CCCCO2)C1 C1(NC(C(C)SC(C)C)=O)CN(C(c2ccc(CN(C)C)o2)=O)C2CCCCC12 C1(NC(C2CC(C)(C)OCC2)=O)CN(C(=O)CCC(N)=O)CC12CCCC2 C(=O)(CCCC(F)(F)C(F)(F)F)NC1C(NC(=O)CCCc2cnccn2)C1 C1(CNC(C2CCCN2C=O)=O)CN(C(c2ccnc(C(C)=O)c2)=O)CC(C)O1 C1(C(C)C)CC(N=c2nc3sccc3c(N3CCC(n4cccn4)C3)[nH]2)C1 c1(N2C(CCNC(C3CCC(OC)CC3)=O)CCC2)nc(Cl)nc2c1ncn2C Cc1cc(-c2cnc(C(=O)NCC3CNC(=O)C3)c(C(F)(F)F)c2)cnc1O Cc1cccc2[nH]cc(C(=O)NCCC(O)CNC(c3cncc(F)c3Cl)=O)c12 CS(=O)(=O)c1cccc(C(N2CCC(NC(C3CCSC3)=O)C(O)C2)=O)c1 N1(C(C(CCC)O)=O)CC2CCC(CNC(=O)Cn3cccnc3=O)(C2)C1 C#CCCCC(C)C(=O)NCC(C)N(C(=O)CCCN1C(=O)CN(C)C1=O)C Cc1cc(CCCC(=O)N(C)CCOCCNC(c2nnc(S)n2C)=O)c(C)s1 N1(C(C)C)C(=O)CCC1C(N1CC(NC(c2cnn(CCO)c2)=O)C(C)C1)=O CN1CC(C(=O)NC(C2CCN(C(C3CCSCC3)=O)CC2)CO)CC1=O Cc1ccc(F)c(C(=O)NC(C)CCCNC(C2CC2C(C)C)=O)c1F c1(C(N(CCCCNC(=O)CC2OCCC2(C)C)C)=O)cccn2[nH]c(=N)nc12 C1(C2(O)CN(C(=O)CCCCc3ccccc3)C2)(CNC(c2ccsn2)=O)CC1 c1(C(=O)NC(CC)CNC(C2CCCCN2C(N)=O)=O)cc(Cl)c(Cl)cc1N CC1CCCC=C1C(=O)NCC(C)(F)CNC(=O)C1=CC2C=CC1C2 C1(CN(C(=O)CCSCC(C)C)CC)CCCCN1C(c1cccnc1)=O C=CCC(C(=O)NCc1ncccc1C(N1CCC(N(C)C)C(C)C1)=O)C(C)C C1(CNC(C(CC)Cc2ccccc2C)=O)C(C)CCCN1C(=O)COCCO N1(CCOC)CCCC1C1CCCCN1C(C12CC(C)(C1)OC21CCC1)=O CC1(F)CCC(C(=O)N(O)Cc2cn(CC3(F)CCOC3)nn2)CC1 C1(NC(CC2(CNC(=O)CC3CC=CC3)CC2)=O)CC(Cl)(Cl)C1 c1(NC(C2CC3(CC(C(N(C(C4CCCO4)C)C)=O)C3)C2)=O)cc2cc[nH]c2cn1 C=CCCCCCC(=O)NCC1CC2(CC2)CN1C(c1ccc(C(C)(C)C)s1)=O c1(C(N2CCC(C)C2CNC(=O)C=Cc2cncn2C)=O)cc(Br)c(C#N)s1 c1(C(=O)NCC2(F)CC(NC(CS(CC)(=O)=O)=O)C2)cc2ccc(F)cc2o1 c1(CC)oncc1C(=O)NC(C)CCN(C)C(c1ccc(-c2ccco2)s1)=O N1(C(C)=O)CCOC(C(=O)NC2(C(=O)NC3CCCC3(C)C)CC(F)C2)C1 C12(C(=O)OC)CCCCC1CN(Cc1sccc1CO)C2 C1CC(=O)N1.CS(=O)(=O)N(C1(CNC(=O)CCOC(C)=O)CC1)C1CC1 C1(c2nnnn2C)(NCc2c(Cl)cc(C)s2)CCOC(C(F)(F)F)C1 C12(C(=O)Nc3c(C)cc(NC(C4CC(CF)C4)=O)cc3)CCC(CC1)C2(C)C C(=O)(C1=NOC2(CCOC2)C1)N1CC(C)(NC(c2c(Cl)cccc2[N+](=O)[O-])=O)C1 C1(NC(c2cscn2)=O)CCN(C(c2ccns2)=O)CC1O N1(C(C=Cc2ccc(C)cn2)=O)CCC(NC(=O)C(C)SC(C)C)C(C)(C)C1 C1(C(N(CCC(=O)NCC2(C)CC3CC3C2)CC2CC2)=O)CC2(CCC2)CO1 N1(C(C2CN(C(=O)COc3ccsn3)CC2F)=O)CCC12CCC(O)CC2 C1(NC(C(=O)NC)=O)C2CC1N(C(=O)C(C)Oc1ccccc1F)C2C C(CCC(C)C)(C(=O)NC(C1(CCOC)CCC1)=O)NC(C1CC(SCC)C1)=O C(C(C)(C)OC)NC(=O)NC.C1(C(=O)NCCNC(=O)CSC)CC1C1(C)CC1 c1(CNC2(c3ccc(-c4c(OCC)ccnc4)cc3)CC2)nccc2ccccc12 c1(CC(=O)NC2CN(C(C3(C)CC=CCC3)=O)CC23CC3)cnc2n1CCOC2 C(C)(N=c1cc[nH]c(=NCCC2CCC3CC23)[nH]1)NCc1cccc(OC)c1 N1(C(c2cc(C)on2)=O)CC2CC(CNC(=O)Cc3ccc(Cl)c(F)c3)C2C1 C(=O)(C1CCCc2nncn21)NC12CC(CNC(C(C)CC(N)=O)=O)(OC1)C2 c1(C(N2CCC(CN(CCC)C)C2)=O)c(C)nn(CC(F)F)c1C Cc1cc(F)c(COC(c2cocc2Br)=O)nc1Cl C1(CCC)CN(C(c2nc(C(F)(F)F)cn2C)=O)CCN1C(c1c[nH]nc1C)=O c1(C(=O)NCC2(F)CN(C(c3n(C(CC)C)ncc3)=O)C2)ccnn(C)c1=O CC1CCN(C(=O)CCN2C(=O)CCC2=O)CC1CNC(C1CC(F)C1)=O C1(CNC(CS(=O)(=O)N(C)C)=O)CCC2(CN(C(C3CCOCC3)=O)C2)O1 Cc1cnc(Cl)[nH]c1=NCCCCCCN(C)C(c1c(Cl)n[nH]c1C)=O C1(NC(C(C)CC#N)=O)CN(C(=O)CC2CCC2)C2(CCC2)C1 Cc1cc(C(N2CC3CC3(CNC(c3nnn(C)c3N)=O)C2)=O)cc(F)c1 C=CCCC(F)(F)C(=O)NC1CCC(CNC(c2ncc(Cl)cc2Cl)=O)C1 c1(C(=O)NC(CN(C(C2CC2F)=O)CC)C)ccc2c(n1)OCC(=O)N2 c1(C(=O)NCC(C2CC2)NC(C(c2ccc(OC)cc2)O)=O)cc2c(ncn2C)[nH]1 C1(CC)(CC)CC(NC(=O)C(C)=CC(C)(C)C)CN1C(=O)CSc1ccc(F)cc1 C1(C(=O)NCc2ccc(CC)o2)(CNC(c2cnc(O)o2)=O)CC12CCC2 C(C)(CC1=CCCCC1)NC(C(CC)NC(=O)CCc1nccs1)=O C1(C(=O)NCC2CCCC2NC(=O)CCNC(=O)NC)(CC)CCCCC1 N1(C(CC=CC=C)=O)CC2(C1)CN(C(=O)Cn1ccc(C3CC3)n1)CCO2 N1(C(C(CCC)F)=O)CCC(NC(c2ccc(OC)cc2F)=O)C(CO)C1 c1(OC)cc(C)cc(C(N2CC(NC(=O)C=CC3CC3)C3CC23)=O)c1C C1(C(N(CCNC(CCc2ccc(=N)[nH]c2)=O)C2CC2)=O)CCN2CCOCC12 N(C1CCC(NC(C2(CCF)CC2)=O)c2ccccc21)C(c1c(C)cns1)=O C(=O)(C=O)NCCC1(NC(=O)COCCOCCO)CC1.CC1CC1C(=O)N c1(C(c2n(CCCSC)nnn2)NCC2CCSC2)cc(Cl)cc(Br)c1F c1(NC(C2CCC(NC(COCCCC)=O)C2)=O)c(C)ccnc1OCC C1(CNc2ccc(NC(C(C=CC)O)=O)cc2)CCC2(CN(C(=O)COC)C2)O1 c1(C(N(C(CN(C(C2N(CC)C(=O)OC2)=O)C)C)C)=O)nn2ccccc2c1C C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CC(=O)NC(CC)(CC)CC)CC N1(C(C(=Cc2ccco2)C)=O)CCN(C(=O)Cc2csnn2)C2CCCC2(C)C1 C1(NC(CNC(=O)OCC=C)=O)CCCC(CC(=O)NCc2csc(C)c2C)C1 C1(CNC(C2CC3CCCC23)=O)CC2CCC1N2C(C1CC1(F)F)=O c1(-n2c(CC(=C)C)nc(CC(C)C)n2)ccc(=O)n(C(C)C)c1 Cc1ccc(C(=O)NCC2CC3CN(C(C4CC4(C)C)=O)CC23)cc1F C1(O)(C(=O)NCC2C(CNC(C(COC(C)=O)C)=O)C2)CN2CCC1CC2 CCC(C)(C)C(O)C(=O)N1CC2CN(C(=O)C(C)SC)CC2C1 C(=O)(C1=NOC2(CCC2)C1)NC1(C)CCN(C(C2C(C)N(C)CC2)=O)CC1 C1(Cc2ccccc2)COCC2(CCN(c3cnc(C)c(C(N)=O)c3)C2)O1 C12(NC(c3cc(C)[nH]n3)=O)CCCN(C(c3c(C)cc(F)cc3C)=O)CC1C2 N1(C(COC(C)=O)=O)CC2CCCN(C(=O)C(=Cc3ccc(Cl)cc3)C)C2C1 c1(OC)ncccc1CC(=O)NCC(C)NC(c1nocc1-c1ccccc1)=O Cc1nc(NC2(CNC(c3ccnn3CCF)=O)CCOCC2)ncc1Br c1(CN2CCCC(C(=O)Nc3nnc(Br)s3)CC2)ccc(F)c(Br)c1F N1(C(C2(CCCC)CC2)=O)CCC(NC(=O)Cc2ncoc2C)C(CC)C1 Cc1cc(C)c(-c2nc(Cc3ccccc3F)no2)cn1 c1(CC)noc(C)c1C(=O)NCC1CC(NC(c2ncncc2OC)=O)C1 O=C1CC(CC(=O)NC23CC(NC(C4CCCCC4(F)F)=O)(C2)C3)=NN1 C=C1CC2CC1CC2N(C(=O)C(=O)NCCC(=O)NCC)C c1(OC(C)C(=O)NCCCCNC(=O)CSc2ccccc2)ccccc1C#N C(=O)(C1=NOC2(CCC2)C1)NC1CCC(CNC(C2C(=C)C2)=O)C1 C(=O)(C(C)CC(N)=O)NC(C1(O)CN(C(CC2(OC)CC2)=O)C1)C CN1CCC(C)(C(=O)NC(CNC(c2ccn(CC(F)(F)F)n2)=O)CO)CC1 c1(C(N2CCC(C(C(=O)NCC(C)OCC#C)(C)C)C2)=O)ccc(CC#N)cc1 Cn1cc(C(c2cc(-c3ccccc3)nn2C(C)(C)C)=O)c2ccccc2c1=O c1(C(=O)NC(CNC(c2ccc(CCC)[nH]2)=O)C(C)C)ccc(C#N)c(F)c1 c1(CC(=O)NCC2CCC(NC(C(CC)(C)F)=O)C2)ccc([N+](=O)[O-])cc1 C1(NC(C2(CC=C)CC=CC2)=O)CN(C(c2ccccc2F)=O)C(C)(COC)C1 N1(C(C2CCC(=O)N2)=O)CCOC(CNC(c2cccc(C(F)(F)F)n2)=O)C1 c1(C(N2C(CNC(C(CC)OC3CCCCC3)=O)CC2)=O)ccnc(O)c1 Cc1c(C(=O)NCC(C2CCCC2)NC(=O)CCCc2nccs2)cncc1N C12(CNC(c3nc(C)sc3C)=O)CCC(CC1)N2C(=O)CC1CC12CC2 N1(C(CC(C(C)C)C)=O)CCC(CNC(c2cccs2)=O)C(F)(F)C1 c1(C(=O)NCCn2ncc(C(=O)NCC3ON=C(C)C3)c2)ncc(C)cc1C C1(C(N(C)CC2CCCN(C(COCC#C)=O)C2)=O)CN2CCN1CC2 C1(c2ccc(Oc3cccc(Cl)c3)s2)CN(N2CCC(CBr)CC2)C1 c1(C(=O)NC2(C)CCN(C(c3ccc(CC)[nH]3)=O)C2)cc(OC)c(OC)c(N)c1 S(=O)(=O)(c1cc(C(=O)NCC2CC3(CC3)CN2C(=O)C2=CCSC2)c(C)o1)NC C1(NC(Cn2c(C)ncc2)=O)CCCN(C(c2scnc2C(F)(F)F)=O)CC1F Cc1ccc(N)cc1C(=O)NCC(F)CNC(c1coc(C(F)F)c1)=O C12(NC(=O)C3CC3)CC1COC21CCC1.N12CCC(C(F)C1)C(=O)N(C)CC2=O N1(CCNC(c2c(C)c(Cl)ccc2)=O)C(C)CN(C(=O)C2CC2)CC1C C1(C(=O)NC2CC(CNC(=O)CCCc3ccsc3)OC2)COC2(CCC2)C1 CC1CC(C(=O)NCC2CCCCC2NC(C2(C(N)=O)CC2)=O)=NO1 C1(NC(C(C)S(N)(=O)=O)=O)CCN(C(c2n[nH]cc2Br)=O)CC1(C)C CC(CC(C)NC(c1ccn(CCF)n1)=O)NC(C1CC(F)(CO)C1)=O c1(C(C(=O)Nc2nc(C)co2)NC(Cc2scc(C)c2)=O)c(C)cccc1Br N1(C(CC(CC=C)(C)C)=O)CC2CC(C)N(C(C3CCCN3C3CC3)=O)C2C1 CCCC(CCCNC(=O)C=CCC1CC1)NC(c1ccc(CC(C)(C)C)cc1)=O N1(C(CCOCCC)=O)CCN(C(=O)CC2OC(C)(C)OC2=O)CC1C1CCC1 CC1CN(C(=O)CCCOc2cccnc2)CC1NC(C1CSCCS1)=O c12nnc(-c3cnc(C4CC4)[nH]3)n1CCN2CC.c1(CC)ccccn1 N1(C(C(C(C)C)n2cnnn2)=O)CCN(C(c2cc(=O)n(C)o2)=O)C(C)C1 C1(CC(=O)NCCCCn2cc(C(CC)OC)nn2)C(=O)NN=C1C CON1CCC(C(=O)NC2CC(O)C2CC(=O)NCC(F)C2CCC2)CC1 C1(O)(CC)CCCN(C(C2CCC(NC(c3cc(CO)n(C)n3)=O)C2)=O)C1 CC(C)C(C)C(C)CC(=O)NCc1ncccc1C(F)(F)F N1(CCNC(CNC(CO)=O)=O)CCCC1C(=O)OC.C1C(=O)N1.OC CN1CCCN(C(C2CNC(=O)CN2C(c2ccc(N)c(F)n2)=O)=O)CC1 C1(CC)(CC)CC(NC(=O)CCOCC(F)F)CN1C(c1cc(O)nn1C)=O C1(C(N(CCCNC(=O)C(O)c2ccsc2)C)=O)CCc2ncccc2C1 C(CN=c1[nH]ncn2ccc(Br)c12)(C1CCCC1)OC CC(C)C(F)(CNC(C1(C)CC(C#N)C1)=O)C(=O)N1CC2(CNC(=O)N2)C1 C=CCCC(F)(F)C(=O)N(CCCCCNC(c1cc(Cl)cs1)=O)C N1(C(C(=O)NCC2(OC)CCCC(C)(C)CC2)=O)CCc2c(ccnc2C)C1 Cn1cnc2c1C(C(=O)N1CCOC(CCCNC(=O)C(C)(C)C)C1)CC(=O)N2 N1(C(C(CC)NC(c2ccccc2)=O)=O)CC2CC(C)N(C(=O)CSC(F)F)C2C1 c1(C(N2CC(NC(=O)C=CC3CCCC3)C(F)C2)=O)cc(Cl)c(Cl)cn1 N1(C(C2=C(C)CC2)=O)CC2(CCCC2NC(=O)CN2CCOCC2=O)C1 C(=O)(CC(C(C)CC)NC(C1(C)CC(=O)C1)=O)N1CCC(CC#C)CC1 C(c1ccc(Cl)cc1F)=CC(=O)NC(C(C)C)C(=O)N1CCCC1 c1(C(=O)NCC2CC(OC)CN2C(c2cccs2)=O)csc(=NC2CC2)[nH]1 N1(C(COCC)=O)CC(CNC(c2oc3ccccc3c2CC)=O)N2CCC1C2 C12(C(=O)NCC(C)(CO)NC(=O)Cc3sccc3Br)CCCC1CC(=O)C2 c1(OC)ccc2c(n1)NC(C(=O)NCCC(C)NC(c1c[nH]nc1C(C)C)=O)C2 c1(SCC)ccc([N+](=O)[O-])cc1C(=O)N(C1CN(C(=O)C(C)N(C)C)CC1F)C Cc1ccc(OCC(=O)NCc2ccccc2F)cc1.C12COC(C1)NC(=O)N2 CC1CCCC(C(=O)NCc2ncccc2C(F)(F)F)O1 CCC(CC(=O)NC1(CCCF)CCCCC1)NC(=O)C(C)NC(C)=O c1(C(=O)NC(C)(CNC(c2ccnc(O)c2)=O)CO)cc2n(n1)CCCNC2=O C(=O)(C(C(C)C)Sc1nc(OCC)no1)N(CCn1cc(C2(O)CC2)nn1)CC N1(C(CCC(=O)OC)=O)CCCC(O)(CN(C(=O)CN(C)S(=O)(=O)N(C)C)C)C1 C12(CNC(C(c3cccc(O)c3)C)=O)CCCC1CN(C(=O)Cc1ccns1)C2 c1(NC(N(C)Cc2c(O)ccc(C)c2)=O)cccc2c1OCO2 C1(NC(CN(C2CCCNC2)C)=O)CCN(CCCO)CC1 c1(C(=O)NCC(C)NC(C=Cc2n(CC)ccn2)=O)coc(S(N)(=O)=O)c1 Cc1nc2ccnn2c(C)c1C(=O)NCC1COCCN1C(=O)COCCF C1(CC)CN(C(c2ccccc2Br)C(=O)NC2CCC2)CC(C)O1 N1(C(CN(C)CC)=O)CC(NC(C23CC(CF)(CO2)C3)=O)C(F)C1 N1(C(C2CC3(CC3)CO2)=O)C2COCC1C2.c12nocc1C(=O)NC2C c1(CN(CCNC(c2nc(CCC(C)C)oc2)=O)C2CC2)nc2ccccc2[nH]1 c1(C(N)=O)ccc(Br)cc1C(N1CCC(CN=c2[nH]nc(C3CC3)o2)C1)=O C1(c2n(C)cnc2)CN(C(=O)C2=CCC2)CC1NC(=O)CC(C)(C)OC1CCCC1 c1(OC)ccc(Cl)cc1C(F)(F)C(=O)NCC(CO)NC(C1CCSC1)=O C(=O)(N1CCCc2ccnn21)C1CCC(NC(CC(C)OC)=O)CC1 N1(C(c2ccn(CC)n2)=O)CCN(C(=O)CCC=C2CCCC2)CC1 N#Cc1nccc2cc(NC(C3CN(C(c4c(Cl)cccc4Cl)=O)C3)=O)ccc12 C(=O)(CC(F)(F)C(C)C)N(CCOC)CCNC(N1CCCC(C(N)=O)C1)=O C(C(C)(C)CC(=O)NC(C)CCNC(c1cnn(-c2ccccc2Cl)c1)=O)OC C1(C(=O)NCC(C2CCCCC2)C)CC2(CCN1C(=O)C(C)CO)CC2 N1(C(C2NCCC23CC3)=O)Cc2ccccc2CC12CCC2 N1(C(C(CC=C)OC)=O)CC(C)(C)CC1CC(=O)Nc1csnc1OC N1(C(C(CCC)NC(C)=O)=O)CCCN(C(c2cnc([N+](=O)[O-])n2C)=O)C(C)C1 C=CC(C)(CCOC)C(=O)NCC(C)(C)CN(C(=O)C(C)(C1CC1)OC)CC C(CCN=C(NCC(F)F)NC1CC(=O)N(C(C)C)C1)=CC c1(C(N2CCC3CCC(NC(CCS(C)(=O)=O)=O)C32)=O)ccc2c(n1)OCCO2 Nc1cc(C(=O)NC2CC(CO)N(C(c3cnsn3)=O)C2)cc(F)c1 Cc1ncncc1NC1(CO)CCN(C(=O)CCCc2cnccn2)C1 N1(C(C(CCC=C)(C)C)=O)CC2COCCC2(NC(C2CCCNC2=O)=O)C1 C1(C)(NC(CC=CCNC(c2nc(CC)oc2)=O)=O)CC=CCC1 C1(OC)(CO)CN(C(C2(CCNC(=O)C(C)CO)CCCC2)=O)C1 c1(CC)ccc(C(C)CC(=O)N(CCCNC(=O)C=CC2CCCN2C)C)cc1 N1(C(C(NOC)=O)=O)CCN(C(=O)CC2CN3CCN2CC3)CC1C1CC1 Cc1nc(C(=O)N(C(C)(C)CC(=O)N2CC(F)(C#N)C2)C)sc1C C1(S(N)(=O)=O)(C(=O)NC2C(CNC(C3(C)COC3)=O)COC2)CC1 N1(C(C(CCc2ccccc2)N(C(CC(CC)C)C)C)=O)CC2CN(C)CC2C1 c1(CC)cc(C(=O)NCCOC(C)(C)CNC(c2cscc2F)=O)ccc1C c1(C(N2C(C)CC(NC(C(CC)CC3CCCCC3)=O)C2)=O)c[nH]c(=N)cc1C C1(NC(C2C(C(C)C)C2)=O)CC2(C1)CC(C(=O)NOCCF)C2 c1(SC(C(C)c2nc(-c3nccn3C)cs2)(F)F)ccccc1Br Cc1cc(Cl)ccc1C(=O)NCC1CCCN1C(=O)C1=NOC(C2(O)COC2)C1 C1(OCC)CC2(C1)CC2NC(=O)Cc1cccc(C)c1.C1(=O)C(C(C)C)N1 Cc1ccc2c(c1)C(NC1CCCCN1CC#N)CCCO2 c1(CN2CCC(NC(c3c(C)nc(Br)cc3)=O)C(F)C2)ccc(Br)c2nsnc12 c1(CN(C(c2cc(CNC(=O)CC3CCCCO3)on2)=O)CC)ccncc1Cl c1(C(N2CCCC2C(N2CCC3CC23)=O)=O)ccc(Br)c(Cl)c1F N1(C(c2n(CC)ncn2)=O)CC23CCCC2(C1)CN(C(=O)CSCCOC)C3 C#CC(CNC(=O)C(C(C)C)NC(=O)C(C)N(C)C(C)=O)CC(C)(C)C C12(C)CCCN(C1)C2=O.C1(NC(C2(COC)CCC2)=O)CCCC1C#N CC(CCCNC(=O)C(C)(F)c1ccccc1)NC(C1CC1(C)Br)=O CCC(C)CCC(O)CC(=O)N(CCNC(=O)C1CC1)CCOC N1(CCCC)C2CCC1CN(C(c1oncc1C)=O)C2 c1(C(=O)NC(C)CNC(=O)CC2CCCC2C)cn2c(n1)CCC2 C(N=c1cc(NCC(C)(C)CC2CC2)nc[nH]1)c1c(C)sc(C)c1Br c1(NCC(C(=O)NC2(C(=O)OCCOCC)CC2)c2ccccc2)ccnc(S)c1 N1(C(c2ccc(C#N)[nH]2)=O)CCC2CC1CN(C(=O)CC1CCC3(CC1)CC3)C2 C1(N(C(C(C)SC(C)C)=O)C)CCN(C(C2CC(O)C(O)C2)=O)CC1 CC1CC2(CC2)CN1C(c1cc(CNC(c2cncs2)=O)on1)=O c1(C(N2CC(CCNC(C(C)C3CC3)=O)OCC2)=O)cc2n(n1)CCC2 C(C)(CCC(=O)N(CC(C)NC(=O)C(C)Cc1ccccc1)C)OCC C(C)(N=c1[nH]n(C)c(C(F)(F)F)c1[N+](=O)[O-])C1CCC(NC(COC)=O)C1 C(=O)(C1=C(Cl)CCC1)NCC1(C(N2CC(C)SCC2)=O)CCCC1 N1(C(CN2CCC(OC)C2)=O)CCCCC(CNC(=O)CCC2OCCO2)C1 Cc1c(N)cc(C(N2CCC(NC(C3CCS(=O)(=O)N3)=O)C(C)C2)=O)cc1N C1(NC(C2(COC)CCC2)=O)CC2CC(NC(c3cnccc3Cl)=O)C2C1 c1(C(N(C2CCCC(NC(c3c(C#C)c[nH]n3)=O)C2)C)=O)cccn2nccc12 Cc1sccc1CC(=O)NCC(C(C)C)NC(c1c[nH]cc1Br)=O c1(C(N(C2CC(OC)C2)C)=O)cc(CNC(c2cnc(O)o2)=O)ccn1 C1(NC(CC(C)F)=O)C2CC3CC(C2)CC1(CNC(=O)C(C)(C)C(C)C)C3 C1(NC(c2nc(C(C)C)oc2)=O)CN(C(=O)CCC#N)C2(CCC2)C1 N1(C(C(COC)O)=O)CCC2(CCCN2C(=O)C(C)Cc2cnc[nH]2)CC1 N1(C(C(C2(O)CCC2)NC(c2oc(CC)c(C)c2)=O)=O)CCC2(CNC(=O)N2)C1 C1(C)(CNC(c2ncc(C)nc2)=O)CCCN(C(C2CCS2(=O)=O)=O)C1 C1(OCC)CC2(C1)CC2C(=O)NCC(C)(C)CN(C)C(c1cncc(N)c1)=O c1(SCC)ccc(C(=O)N(C)CCN(C(C2CCC(CC)C2)=O)C(C)C)cn1 CC1CN(C(=O)C=Cc2ncco2)CC1NC(=O)C(c1ccc(Br)cc1)(C)C C(C(=O)NCC1(NC(c2cccc(C)c2)=O)COC1)(C(C)C)SCC C1(CC(=O)NCc2ccc(COC)o2)COCCN1C(=O)CC1CC(OC)C1 Nc1c(F)cc(C(=O)NC2CCC(NC(C3(CO)CCCCC3)=O)C2)cc1F C(CNC(C1CC2CC2N1C(=O)CCC(C)N(C)C)=O)(C(C)(C)C)OC C(=O)(CCC1=NNC(=O)CC1)N1CC(NC(c2nc(OCC)sn2)=O)C2C1C2 C=C=CC(C)C(=O)N1CCC(CC(=O)N(CC(C)CC)C)C1 N1(C(c2cc(COC)nn2C)=O)CC(C2CN(C(=O)C(F)CC3CCOC3)C2)C1 CC(C)C(C(=O)NC(CCC1CCC1)C(=O)NCCC1CCSC1)C(C)C C(CNC(=O)COCC1CCOC1)(CCNC(=O)Cc1nonc1C)OC C1(N(C)C)CN(C(C2CC(NC(=O)CCC(N)=O)C2(C)C)=O)CC1O C1(CC)(CO)CCCN1C(=O)C(C1CCCO1)NC(c1cc(CO)n(C)n1)=O c1(SCC=CC=CCOCCNC(c2cc(-c3cccs3)[nH]n2)=O)c[nH]nc1F c1(CC(N2CCN(C(c3cccc(=O)n3O)=O)CC2)=O)ccc(Cl)cc1[N+](=O)[O-] C(CCCC(=O)NC(C)CCCNC(C12CCCC1(C(N)=O)C2)=O)N(C(C)=O)C C(=O)(CC(C)CCC(=O)NCC1CC1CNC(C1(C)CC=CC1)=O)OC C=CC1(C(=O)NCCCCCNC(=O)Cc2cccn2C)CCC1 Cc1cc(C(=O)NCCCCNC(=O)CC2CCCC2O)ns1 C1(NC(=O)CC2C=CCC2)CC2CC(NC(c3csc4nnsc34)=O)C1C2 c1(C(N2CC(N(C)C(C3CCCOC3)=O)C2)=O)c(F)ccc(Cl)c1N c1(CCC(=O)N(C(CNC(c2c(CC)non2)=O)C)C)cccc(Cl)c1 C(=O)(C(CCC1CCC1)NC(=O)C=CC(F)(F)F)Nc1cn(CCOC)nc1 C1(=O)CCC(CC)OCCN1.C1(C(N(CC(=O)NC)CC#C)=O)CCCS1 N1(CCC#C)CC2CCN(C(c3csc(C(F)(F)F)n3)=O)C2C1 CC1(C)CCCCC1NCCC(C1CCCCCC1)O c1(CNC(c2ccc(OC)cn2)C)ccnc2cc[nH]c12 N1(C(C(C(C)C)OC)=O)CC23CCCC2(C1)CN(C(c1cccnc1S)=O)C3 CC(C)CC(O)C(=O)N1CCN(C(c2ccc(-c3nc[nH]n3)cc2)=O)C(CO)C1 C(=O)(C(C)(C(F)F)c1ccccc1)NCC(C)(C)NC(c1n(C(C)C)cnc1)=O c1(C(=O)OC(c2nc(C)[nH]n2)C2CCOCC2)cc2c(cn1)NC(=O)CO2 CC1CCN(C(c2cnccn2)=O)CCN1C(C1CC2(C1)CC(O)C2)=O c1(C(=O)NC(C(=O)NCC(=O)OCC=C)CCC)ccn2ccccc12 c1(C(=O)NC2C(C(=O)NC3CC(OC)C3)C2)cccc([N+](=O)[O-])c1Br C1(C(=O)NC2(CC)CN(C(C)=O)C2)CN(C(=O)CCCCSC)CC12CCC2 CC1(C(=O)NCC2(C)CCC(NC(c3cnc(C(F)(F)F)s3)=O)C2)CCOCC1 CC1CCN(C(=O)CC2CCSC2)CC1CC(=O)N(C)Cc1ncn(C)n1 N1(C(CC(CC)(F)F)=O)CCC2CCN(C(C3CC(N(C)CC)C3)=O)CC2C1 N1(C(CSCCC(C)C)=O)CCC2C(C(=O)NCC3CCC(C)(C)CO3)C2C1 C(=O)(C=C1SCC(=O)N1C)N1CC(CC)C(NC(=O)CCC2CC(F)(F)C2)CC1 CC1C(NC(c2cc(Cl)ccc2Cl)=O)CC2CCC1N2C(C1(CO)COC1)=O c1(C(=O)NC2C(NC(c3ccc(C)nc3C(C)C)=O)C2)cccc2c1OCC2C CON1CCC(C(=O)NCCN(C)C(c2nocc2CC(C)C)=O)CC1 N1(C(Cc2n(C)cnc2)=O)CC(C(=O)NC(c2cscn2)CO)C(F)(F)C1 c1(C(N2CCC(C)(CC)C2)C(=O)NC2CC2)cc2c(cc1C)OCO2 C(=O)(CCCC(F)(F)C(F)(F)F)N1CCCC(CNC(CC=CC)=O)C1 C(=O)(C(O)CC(N)=O)NCCC1N(C(c2c(OC)cccc2)=O)CCOC1 c1(COC)cccc2ccc(C(N3CCCC4(CCCC4)C3)=O)nc12 S(=O)(=O)(c1cccc(CC(=O)OCCc2nc3c(s2)COCC3)c1)NC C1(NC(=O)NCc2ccc(NCC)cc2)CC(=O)NC(C)C1 C1(C(NOCC2(C=C)CCC2)=O)(CC)CCCN1C(C1CC12CC2)=O c1(C(=O)NC(CC)CN(C)C(c2c[nH]c(Br)c2)=O)ccc2c(c1)CC2 n1(CC)ncnc1C(=O)NC1CCCC1NC(=O)CNC(=O)CNC(C)=O CC(C)(C(=O)NCC=CCC(=O)NCC12CCCC(CO1)C2)C(N)=O N1(C(C2(C(=O)OC(C)(C)C)CC2(C)C)=O)CCC(NC(=O)CCCCC)C(O)C1 c1(C(=O)NCC(CC)NC(=O)CC2(O)CCCOC2)cc2c(o1)CCCC2 C1(C(=O)NC)CCCCN1CCc1nnc(COC)o1 c1(C(N2CCC(NC(Cc3c(C)con3)=O)C(C)C2)=O)ccc2cncn2c1 c1(C(N2CC3C(NC(c4cccc(=O)n4O)=O)C3C2)=O)nccc2occc12 N1(C(C(C)NC(COC)=O)=O)CC2=C(C1)CN(C(=O)CN1CCCNS1(=O)=O)C2 c1(OC)cnc(F)c(C(N2CCCC2(C)CNC(c2ccc(O)nc2)=O)=O)c1 c1(C(=O)NCC2CC(SC)C2)oc(CNC(C2CC(C)=NO2)=O)cc1C Cc1c(F)ccc(C(N2CCCC(NC(c3cnn(C(C)(C)C)c3)=O)C2)=O)c1N c12ccc-1nn2.Cn1nccc1C(O)CNC(=O)CSC1(F)COC1 N1(C(C2C3(CN(C(c4ccc(CC(C)C)cc4)=O)C3)C2)=O)CCn2cccc2C1 c1(C(=O)NC(C)CCCCNC(C2CCSC2)=O)cnc2c(F)cccc2c1 c1(C(=O)OC)nccc2c1CCCN2C(=O)Cc1coc2ccccc12 c1(C(=O)NC2CC(C)(NC(CCOC)=O)C2)cnc(O)nc1O c1(NC(C23CCCN(C(CCC=C)=O)C2C3)=O)cc2c(C)cccn2n1 C1(C(N(CC)OC)=O)CN(C(C2CC(=O)CO2)=O)CC12CCC2 C1(NC(Cc2cc(C)[nH]n2)=O)CCC(CNC(C2CCOC2C(C)C)=O)CC1 CC1CCCC1(C)NC(c1[nH]ccc1CNC(C1(F)CCCCC1)=O)=O C1(C(N2CC(CC(=O)NC(C)CCO)OCC2)=O)Cc2nccn2C1 c1(C(=O)NC2C(C(=O)NCCN(CCC)CCO)C2)cc(F)cc(F)c1Br Cc1ccc(C2CC2C(=O)NCCCN(C)C(C2CCO2)=O)cc1C N1(C(N(C2CCCO2)C)=O)CCCN(Cc2cn(C3CC3)nn2)CC1 c1(C(=O)NC2C(CNC(=O)CCc3cnn[nH]3)CCCC2)cc2cscc2s1 c1(C(=O)NC2CC(CNC(CSC)=O)CC2O)cncc2c1CCC2 C=CCC(C(=O)N1CCC1CNC(c1cc(CCOC)nc(O)c1)=O)C(C)C c1(NC(C(C)N(C(=O)CC(C)N(C)C)C)=O)ccc(C(F)(F)F)cc1C#N CC#CCCCCNC(=O)C(C)N(C(c1cc(CCO)on1)=O)C1CC1 N1(C(C2(CCC=C)CC2)=O)CCCC(C(C)C(=O)NCCN2CCOCC2=O)C1 C1(SCC23OCC(C(F)(F)F)C(C2)C3)CCOC12CCCC2 C1(CCC)CN(C(c2c(C(F)(F)F)ncn2O)=O)CCN1C(C1CC12CC2)=O C12(NC(COCC(C)C)=O)CCCN(C(=O)CCN3CCCCCC3=O)CC1C2 c1(CC)cc(C(=O)N(C2CC(NC(c3nccc(Cl)c3F)=O)C2)C)cn(C)c1=O Cc1ccccc1S(=O)(=O)CC(=O)NC1CCCN(C(c2cncnc2)=O)CC1 c1(OCC(=O)NCCC2CSCCN2C(=O)CCF)ccc(Cl)nc1 c1(CC(=O)NCC2N(C(CC(C)(C)OC)=O)CC(OC)C2)ccc(F)c(F)c1 N1(C(Cc2nc(C)[nH]n2)=O)CC(NC(c2cc(C(N)=O)oc2C)=O)C2CC12 c1(CC)cccc(CC)c1CC(=O)N(CC(O)CNC(C1CCC(C)C1)=O)C C1(NC(Cc2ccc(OC)c(F)c2)=O)CN(C(C2CC23CC3)=O)C2(CCCC2)C1 c1(C(=O)NCC2N(C(C(CCC)CC)=O)CC=C2)ccc(F)c2c1OCC2 C1(CC)(CC)CC(NC(c2cc(Cl)ccc2N)=O)CN1C(C1CC1(C)C)=O N1(C(c2ccnc(N(C(C)C)C)c2F)=O)CCC(F)(F)C(C(N)=O)C1 C(=O)(C1=CCc2ccccc21)NCCCCCN(C(=O)CCc1cncnc1)C c1(CC(N2C(C(C)NC(=O)C=CCO)CCC2)=O)cc(F)ccc1O c1(C(N2CC(C)C(C)C2)C(=O)NCCC)ccc(C)cc1F N1(C(C2CCN(C(CC(C)(F)F)=O)C2(C)C)=O)Cc2cccc(F)c2C1 C1(C(=O)NCC(CC)NC(c2cn(C)nc2C(F)F)=O)COc2ccccc2C1 C(C(C)C(=O)NC(C(=O)NCC12CC(C(N)=O)(C1)C2)C1CCCO1)OC(C)C c1(C(=O)NC(CCSC)C(=O)N2CCCC(OCCO)C2)cn(C)c(=O)n1C c1(C(=O)NC(C2CCN(C(C3(C)CC3)=O)CC2)CO)cccc2c1CCO2 CC(C)C(C(=O)NCCOC(C)(C)CNC(=O)CCC(=O)N(C)C)NC(N)=O C(=O)(CC(CC)OC)NCC(C)(C1CC1)NC(c1cnc(CCCC)s1)=O N1(C(COCC(C)C)=O)CC(F)CC1CNC(c1csc(-c2cnc[nH]2)n1)=O N1(C(c2ccc(N)cn2)=O)CCC2CCN(C(c3cc4n(c3)CCOC4)=O)C2C1 C(=O)(C1CCCc2sc(=N)[nH]c21)N(CCN(C(=O)C1CCCc2ncnn21)C)C S(=O)(=O)(c1ccc2c(c1)CCCC2)N1CCN(C(=O)C=CS(F)(F)(F)(F)F)CC1 C1(NC(CCC2N(C)CCCC2)=O)CCN(C(=O)CN=S(C)(C)=O)CC1F N1(C(c2cnc3nncn3c2)C(=O)NCCOC)CCSC2COCCC12 C(C)(C)(CCCCNC(C1CC1(C)C(C)C)=O)NC(C1C(C=C)C1)=O Cc1cc(C(N2CCC(O)(C(=O)Nc3ccccc3CO)C2)=O)cc([N+](=O)[O-])c1 C1(NC(=O)CC2CC3(CC3)CO2)CCCC(C(=O)NCCC2(SCC)CC2)C1.CO c1(C(=O)NC(C(=O)NCCCC)Cc2ccccc2)ccc(CO)cc1F N1(C(c2cc(OC)ns2)=O)CCN(C(=O)COc2cc(C)on2)C(C2CC2)C1 C1(C(N2CC3(CC(NC(COC4(C)CCC4)=O)C3)C2)=O)CC2CC(O)CC(C1)C2 c1(OCC)cccnc1C(=O)NOCc1cn(-c2ccc(CO)nc2)nn1 C12C3CCCC3N1C2=O.N1(C(C(C)N(C)C)=O)CCCC1(C)C(C)(C)C Cc1cc(C(N2CC=CC2CNC(=O)CC(F)(F)Br)=O)c(F)cc1F N1(CC(=O)NCC(CNC(C2(C(F)(F)F)CCCC2)=O)CO)CC(=O)NC1=O C1(c2ccn(C3C(C)C3)n2)CCS(=O)(=O)CN1.C1(=O)CN1 N1(C(C(CC)(C)C)=O)CCC2(CC1)CC2c1cn(CC2CCC2OC)nn1 N1(C(C=CCN(C(=O)CCC2CC2)C)=O)CC2(CC2)C1 C1(O)(CN(C(=O)CC2C=CCCC2)C)CCCN(C(=O)COCC(F)(F)F)C1 N1(C(Cn2c(=N)[nH]nc2)=O)CCCC2(NC(=O)Cn3ccsc3=N)CC2C1 Cc1cc(CC(=O)NCCCN(C(=O)CCOCC2CCC2)C(C)C)cc(F)c1 C(C(CC1CC1)CO)NC(C(C)N(C(=O)CCc1ccnn1C)CCC)=O C(N=c1[nH]c(=NCCNS(=O)(=O)NC)[nH]c2c1SCC2)C1CCCC(SCC)C1 CCCCC(CC)CC(=O)NC1CN(C(c2sccc2-c2cc[nH]n2)=O)CC1C S(=O)(=O)(c1cccc(NC(C(=O)N2CCCC2)=O)c1)NC.N1(C(C)O)CCCS1(=O)=O c1(CC(=O)N(CC(C)NC(c2ccncc2O)=O)CC)cc2ccccc2s1 C12(NC(C)=O)CCOCC1CN(C(C1CCOC1c1ccncc1)=O)C2 CC(CCC(=O)NC1COCCC1NC(=O)C(C)(C)O)c1ccc(Br)cc1 N1(C(C2CN(CC)C(=O)C2)=O)CCCC2C1CCN2C(c1ccncc1)=O c1(C(=O)NCC(CNC(c2c(O)ncc(CC)c2)=O)F)cccc2c1CC(=O)N2 Cc1cccc2c1CC(C(=O)NC1COCC1NC(c1cc(CO)[nH]n1)=O)O2 N1(C(C23C(CN(C(c4c(C)ccc(F)c4)=O)C2)CC3)=O)CC2(C)CCC2(C)C1 O=C(CCCCC(F)(F)F)NCC1CC1NC(C1CC(n2ccnc2)C1)=O C(CC(C(F)(F)F)N1CCOCC1)NC(c1cccc(-c2ccc(O)cc2)c1)=O C1(C)(NC(CC2(C=C)CC2)=O)CCN(C(=O)Cc2csc(NC(=O)C3CC3)n2)C1 c1(C(=O)NC(CC)CNC(C2CSCN2C)=O)c(C)ccnc1C N1(C(CCC#C)=O)C2CCC1C(CNC(c1cncc(OC(F)F)c1)=O)C2 C(=O)(C1=NOC(CC2(O)COC2)C1)NC1CC(NC(=O)COC2CC2)C1 CCCC(O)C(CO)NC(=O)CCC1CCCN(C(=O)Cc2ncccc2F)C1 Cc1nc(N2CCCC(CN(C)C(C3CCCCO3)=O)C2)c2c(C)csc2n1 N1(C(C2C(CNC(CC3CC(CC)C3)=O)C2)=O)CCCC2(CC2)C1 CC1(C)CC(n2ccnc2-c2cc(-c3ccc(F)cc3)no2)CS1 N1(C(C2CC(CC(=O)OC)C2)=O)CC(C)(NC(=O)C=CC2CCOC2)C1 C(c1cc(Cl)ccc1OC)=CC(=O)NCCC(CCNC(C=CCOC)=O)C C1(NC(CSCC=C)=O)CC2CC(NC(c3cnn(CC(F)F)n3)=O)C1C2 C1(NC(C2(C)CN(C(=O)Cn3ccnc3)C2)=O)CCOCC12CCC2 c1(CC(=O)N(C(C)C(=O)NCC(c2ccco2)O)CC)cc(C)on1 N1(C(C(CCC)CNC(c2c[nH]c3cccnc23)=O)=O)C2CCC1CC(CO)C2 CC1CON(Cc2cccc(Cl)c2)C1 c1(CC(C(=O)NCCC(=C)CNC(C2(n3cncn3)CC2)=O)C)cccc(F)c1 N1(C(CNC(CCC)=O)=O)CC2ON=C(CNC(=O)CCn3ccc(C)n3)C2C1 C(=O)(C(C)(C)CC(C)(C)C)NCC12C(CN(C(C(CC(C(C)=O)C)C)=O)C1)C2 C1(NC(CC(=O)OC)=O)CCCN(C(=O)C(C)C2CC2)C1C c1(C(N2CC(C)(NC(c3onc(C(C)C)n3)=O)C2)=O)cc(C#N)c[nH]1 C1(NC(CCNC(COC)=O)=O)CN(C(=O)C(C)C(C)(F)F)CCC12CCOCC2 C(CO)(CCCCNC(=O)CCC1CCC(O)CC1)NC(CCC)=O c1(C(C)C(=O)NCCC(O)CNC(c2cnn[nH]2)=O)cn(C)c2ccccc12 C1(CC(=O)NCC2(O)CC(NC(=O)CN3CCC(O)CC3)C2)CCC2(CCC2)CC1 C1(CC)CN(C(C23CCC(CO)(CC2)C3)=O)CCN1C(c1ccncc1)=O N1(C(=O)NCc2c(Br)nc(N(C)C)s2)CCOCC12CCS(=O)(=O)C2 C1(C(=O)OC)CN(C(=O)Nc2cccc(C(=O)N(C)C(C)C)c2)CCS(=O)(=O)C1 N1(C(c2n(C=C)nnc2)=O)CCOCC1(C)C CC1=C(C)CN(C(C2(CNC(C34CCCC3C4)=O)CC2)=O)CC1 c1(C2(C(N3CCC(C)(c4onc(C)n4)C3)=O)CC2)ccc(Cl)c(Cl)c1 CC(C)(C)C#CCCN(C(=O)CNC(=O)C=CC(=O)NCCF)C C1(NC(c2n(C)ncc2)=O)CCC(F)(CNC(=O)CNC(c2cccs2)=O)C1 c1(C(=O)OCC=CC)cc2c(cnn2C)nc1C Cc1cnc(C(N2CC=CC2(C)C(N2CCC(CC(C)(C)C)C2)=O)=O)c(C)c1 c1(CNC(=O)NC2CCN(CC(=O)OCC)CC2)cnc(C#N)c(Cl)c1 n1(CCC)ncc(C(=O)NCC2CCCC(NC(C3(SC)CC3)=O)C2)c1Cl c1(C(=O)NC2CC(NC(C(CCCC)CC)=O)C2)ccnc2c(C(N)=O)cnn12 c1(CN2CCC(NC(c3cc(C)nn3C(F)F)=O)C2)ccc(F)c(C#N)c1 c1(C(=O)NC(CCCNC(C(C)NC(=O)NC)=O)C)nnccc1C c1(C(=O)NC(C(C)C)C(=O)NC2CC=CC2)ccc(=O)n(C)c1 c1(SCC(N2CC(O)(CNC(C3CCC(OC)C3)=O)C2)=O)ccc(C)cc1 C(=O)(CC(=O)NCC(C)(C)OCC(=O)NCCCC1CCOC1)N(C)C N1(C(c2nc(CC)oc2)=O)CCC2(CNC(=O)CNC(=O)C3CC3)CCCCC12 c1(C2CN(C(C(n3cc(C4(COC)CCCC4)nn3)C)=O)C2)ccnc(Cl)c1 c1(C(N2CCC3C(C(N4CC(CC(C#C)C)C4)=O)C3C2)=O)ccc2cc[nH]c2c1 C1(C(=O)NCC2(NC(C3CC(CN(C)C)C3)=O)CCC2)CCCOCC1 N1(C(=O)NCC2(C(=O)NC)CC2)CCC(CO)c2ccc(F)cc21 N1(C(=O)CCc2ccc(O)nc2)CCC12CN(C(=O)CN1CCCS1(=O)=O)C2 CCC(C)CC(C(=O)NCC12CCC(CC1O)C2)NC(=O)CCCN(C)C(C)C CCCC(C(=O)NCC1CC1CC(=O)NCC1C(C)(C)C1(F)F)OC CCCCC(CNC(=O)C(c1cnn(C)c1)O)NC(=O)C(COC)COC C(CCCCC(=O)NC1CCCN(C(=O)COCCCF)C1)OC C(CCCCCC1CC1)NC(CCC1(NC(C2N(CCC)CCC2)=O)CCC1)=O Cc1nc(C)c(C(=O)N(CCCNC(=O)CC2CCOC2)CCO)c(C)n1 c1(C(=O)NC2C(NC(c3cccc(Br)c3F)=O)C2)cc(Cl)ccc1F N1(C(CC(=O)NCC#C)=O)CC2CCCC(NC(=O)C(C#N)C(C)C)C2C1 N1(C(CC2(C)CCN(C(C(C=CC)O)=O)C2)=O)CCc2nc[nH]c2C1 N1(C(c2cnc(CNC(CC3CC(SC)C3)=O)nc2)=O)C2CCC1CC(CO)C2 C(=O)(C1=CCC(C)CC1)N1C(C(C)NC(c2conc2C2CC2)=O)CCCC1 c1(C(N2CCCC(N3CCCCC3)C2)C(=O)NC(C)C)ccc2c(c1)CCCO2 Cc1ccc(C(N2CC(NC(=O)CN(c3ncccn3)C)C3CC23)=O)cc1F O=C(C1=CCCCC1)NC(c1ccccc1)CNC(c1ccsc1)=O c1(C(=O)NCC(C)CNC(C2CSCCS2)=O)cc(CC2CCC2)c[nH]1 CC(N=c1[nH]c(=NCCC2CCCS2(=O)=O)[nH]c2c1COCC2)c1snnc1CO N1(C(c2c(C)ccc(C)c2)=O)CCC2CCC(C1)N2C(C1CCS1(=O)=O)=O c1(C(=O)NC2CC(CNC(C3C(c4n(C)ncc4)C3)=O)C2)cc(OCCO)n(C)n1 CC1CN(C(c2cc(CNC(=O)CCCn3cncn3)on2)=O)CCN(C)C1 C(=O)(C(COC)COC)NCCC1(C(N(CC#C)CCF)=O)CCCC1 Nc1ccc(Cl)nc1NCCn1cc(CNC(c2snc(O)c2Cl)=O)nn1 c1(OC(C)C)ccc(C(N2CCC(C(C)NC(=O)CNC=O)C2)=O)c(Cl)c1 c1(C(=O)NCC(CNC(CC(C=C)C)=O)F)ccc(OC)c2occc12 c1(N(C)C)ncccc1CCC(=O)NC1(CCNC(C2CC3CCC2C3)=O)CC1 c1(C(=O)NCCCN(C(C2(C)CCOC(C)C2)=O)CC)ccc2cnc(C)n2c1 C1(CNC(C2C(C)OC(=O)N2)=O)(NC(=O)CCCN=[N+]=[N-])CCC(C)(C)CC1 C(CCCC(C)NC(C1(C(C)NC(=O)Cc2cccc(F)c2)CC1)=O)OC C1(CC(=O)NCCn2cc(CNC(C(COC)C)=O)nn2)Cc2ccccc2O1 C1(NC)CC2(C1)CN(C(c1[nH]c(COC(C)=O)nc1C)=O)C2.C12(CC1)CC(=O)N2 O=C1NCCC1C(=O)NCC1(NC(c2csc(C(F)(F)F)c2)=O)CCOC1 C1(CN(C(C(C2CC2)OC)=O)C)CN(C(=O)CN(CC(C)(C)C)C)CCO1 c1(OC)ccc(C(=O)NCC2CC2CNc2sccc2CO)c(Cl)n1 N1(C(C(c2ccccc2Cl)N(C)C)=O)CC(NC(=O)C2CC2)C2(CCC2)C1 c1(C(N2CC3C(NC(CCC=CCC=C)=O)(C3)C2)=O)cccc2[nH]cc(Cl)c12 S(=O)(=O)(c1cccc(Cl)c1C)CN1CC(OC)C(c2c(Cl)cc(F)cc2Cl)CC1 N1(C(CCC=CC(C)C)=O)CCC(F)C(NC(=O)CC2CC2C(F)(F)F)C1 N1(C(CSC(C)C)=O)CCN(C(c2ccc(O)cn2)=O)CC1 c1(OCC(=O)NCC2(C)CCN(C(C(CCC)OC)=O)C2)cc(C)c(Cl)c(C)c1 c1(CNC(=O)NC(C)Cc2nn[nH]n2)nn(C)c2ccccc12 c1(SC)onc(C)c1CC(=O)N(CC(=O)OC(C)(C)C)C(C)C N1(C(c2ccc(C#C)nc2)=O)CCC2(CCC2)C(NC(=O)CCNS(C)(=O)=O)C1 C(=O)(C(C(C)(C)C)n1ccnn1)NC1CC(Cn2cc(C(C=C)=O)nn2)C1 Cc1nsc(C(=O)NC2CCC(N(C(=O)C=Cc3ccc(C(N)=O)o3)C)C2)c1N c1(C(=O)NC2C(CCC)CN(C(=O)C=C(C)C(C)C)C2)cncc2[nH]ccc12 C(=O)(C(F)(F)C(O)C(C)C)NC1(CO)CN(C(C(CCOC)C)=O)C1 C1(OC)CC(NC(c2ccnnc2O)=O)CN(C(c2c(C)[nH]c(C)c2C)=O)C1 Cc1cnc2nc(C(N3CC(NC(c4cncc(F)c4)=O)CC(O)C3)=O)nn2c1 c1(C(=O)NCC(C)NC(C(C)P(C)(C)=O)=O)cccc2c1COCC2 C1(NC(c2cc(COC)sc2)=O)CCCN(C(c2ccc(C(N)=O)s2)=O)CCC1 N1(C(c2ncc(OCC)nc2)=O)CC2CCCC2(NC(=O)CCC(C)(C)F)C1 N1(CC)CCOCC1CC(=O)NC1CN(C(C23CC(F)(C2)C3)=O)CC1C(F)F N1(C(c2cn(CCC=C)nn2)=O)CCOCC1CN(C)C(C1CSC1)=O N1(C(CN(C(C(c2cn(CC)nc2)=O)=O)C(C)C)=O)CC(C)(C)C1C(C)C C1(NC(C(C)NC(N)=O)=O)CN(C(c2csc3cccnc23)=O)C2(CCCC2)C1 N1(C(Cc2c(C)occ2)=O)CCCC(NC(c2cc(C(F)(F)F)ccn2)=O)C1C C(=O)(C(C)CC(C)(F)F)N1CC(CN(C(c2nccc(C)n2)=O)C)C1 c1(CC(CO)N(C(C2C(C(=O)ON)C2)=O)C2CC2)cccc(Br)c1 CC(N=c1[nH]c(N(C)Cc2nc[nH]n2)nc2c1CCCCC2)C(C)CO c1(C(=O)NCC(CC)NC(=O)CCSc2ccccn2)c(C)cc(C)oc1=O C(=O)(C1=NNC(=O)C1)NCC(C)N(C)C(C1CCOC1)=O n12nnc(c1N)C(=O)OC(=O)COC2.c1(OC)ccc(C(F)(F)F)cc1 N1(C(CCCOC)=O)CC2(CCOCC2)CC1CNC(=O)C(F)(F)c1nccs1 N1(C(c2ncc(OC)cn2)=O)CCC(NC(=O)C=CCN2CCCC2)C(C)C1 c1(CC)noc(C)c1C(=O)NC1CCC(N(C(=O)Cc2ccc(Cl)cc2)C)C1 c1(C(c2nnnn2C2CC2)NC(c2cc(Cl)cc(Cl)c2F)C)ccccc1[N+](=O)[O-] N1(C(c2c(CC)nn[nH]2)=O)C2COCC1CC(NC(c1cc(C)[nH]n1)=O)C2 N1(C(C2(CCCC)CCC2)=O)CCC(NC(=O)CCC2CCCN2C)C(C)C1 C=CCC(CC)C(=O)NC(CNC(C1CC2CCC(C1)S2)=O)(CC)CC c1(C(c2n(CCOC)nnn2)NCCOCCCS(N)(=O)=O)c(F)cc(F)cc1F C1(C(=O)NCC2(NC(c3ccc(C)cc3F)=O)CC(OC)C2)CC2(C1)CC(C)C2 Cc1ccc(C=CC(N2CC(F)(C(=O)NCCC(C3CC3)C3CC3)C2)=O)o1 CS(=O)(=O)c1ccc(C(N2CC3CCC2CC3NC(C2CC23CCC3)=O)=O)s1 C1(C(=O)NC2CC(C(=O)NCC(C)C(F)F)C2)CC(=O)C12CCC2 c1(C(N(C)CC2N(C(c3ccc(CCC)[nH]3)=O)CCC2)=O)cc2[nH]ccc2s1 C(=O)(C(O)CC(C)C)N(CCNC(=O)C(CSC)c1ccccc1)CC N1(CC(=O)NC(C)C)CCN(C(=NCCF)NCC(C)(C)C(F)F)CC1 c1(OC)ccc(F)c(C(N2CCC(NC(c3sccc3OC)=O)C(F)C2)=O)c1 CCS(=O)CC(=O)N(C)CC1CCCN(C(C2(C(=O)N(C)C)CC2)=O)C1 C1(NC(C(CC)C)=O)CCN(C(c2cccc(Cl)c2N)=O)C1(C)C N1(C(Cc2n[nH]c(=NC)s2)=O)CCN(C)CC1CNC(=O)C(C)(C)NS(C)(=O)=O C1(C(=O)NCC2=NOC(C)C2)(CC)CCCN(C(c2cc(C)nc(O)c2)=O)C1 N(C1c2ccccc2CCC1F)C(=O)Nc1cc2ccn(CC)c2cc1 N1(C(C(CC)(C)O)=O)CCOC2(CCC(NC(C3CCCC3C)=O)CC2)C1 c1(C(=O)NCC2C3CN(C(CC(CC)C4CC4)=O)C2C3)cccc2nc[nH]c12 N1(C(C(C(C)C)SCC)=O)CCC(C2(O)CN(C(C3CC3(F)F)=O)C2)CC1 Cc1ccc(C(C)C(=O)NCC2CCCC2NC(=O)CCN2CCC2)s1 N1(C(C2(CC)COC2)=O)CC2CCCC2(C(=O)NC2CNC(=O)C2)C1 C1(COC)(CNC(C2(Sc3nnc(C(C)(C)C)o3)CCCC2)=O)CCCN1C(C)=O c1(NC)ncccc1C(=O)N(C1CCN(C(C23CCC2C3)=O)CC1)C CCCCC(C(=O)NCC1CCN(CC)C1)NC(=O)CC(CC)C1CCC1 C(=O)(C1Cc2ccc(F)cc21)NCC(C(C)C)NC(=O)CNC=O C(C)(C(F)(F)C(F)(F)F)=CC(=O)NCC1(O)CC(CNC(C(CC)N(C)C)=O)C1 c1(C(C)NC(=O)CC(CC2CC2)NC(=O)C(N)=O)cn(C)nc1C(F)(F)F c12ccc(cc1Br)CNC1CC(C1)C(=O)O2.c1(CNCC)ccc(Br)cc1Cl c1(C(=O)NCC2(OC)CN(C(C(CC#C)C)=O)C2)cccc([N+](=O)[O-])c1C CC1(C)CN(C(=O)CN2C(=O)CNC2=O)CC(CNC(c2cc(Cl)ccn2)=O)O1 c1(CN(CC=C)CC=C)ccncc1.C(=O)(CC(c1ccccc1)OC)NC CCC(CC(=O)NCC1(CCO)CN(C)C1)NC(c1cn(C)nc1C)=O N1(CCCOC(C(CC)NS(C)(=O)=O)=O)CCc2ccccc21 c1(NC(c2n[nH]cc2NN2CCC2)=O)ncc(F)c(-c2ccco2)n1 C1(NC(C=C(C)C(C)C)=O)CCC(C)(CNC(c2ccc(F)cc2)=O)C1 CCC(C)(C)CC(=O)NC(C)(CNC(c1cc(C(F)(F)F)cs1)=O)C1CC1 CC1CN(C(C2(N(C)C)CCN(C(=O)CCN(C)C)C2)=O)CCC1CO N1(C(C2(CN(C)C)CC2)=O)CC2CCN(C(C3CC34CCC4)=O)CCC2C1 C1(SCC(=O)NCC2(COC)CN(C(c3cccs3)=O)C2)CCOC1(C)C C1(C(=O)OC)(OC)CCCN(C(=O)C(c2cccc(Cl)c2F)NC(C)=O)C1 N1(C(CC2(C#N)CCCCC2)=O)CCC2(CCC(NC(c3cn[nH]c3)=O)CC2)CC1 c1(NC(C2OCCN(C(c3n(CC)ccc3)=O)C2)=O)ccc2c(c1)CCO2 N1(C(C(CC)C(F)(F)F)=O)CCN(C(c2cc3n(n2)CCC3)=O)C2(CCC2)C1 C=CC(C)(CC)C(=O)NCC12CC(C1)C(NC(=O)C(C1(O)CCCC1)F)CO2 C1(N(C(=O)CO)C)CN(C(=O)CS(C)(=O)=O)CCC1O C1(NC(c2n(CC(C)C)ncc2)=O)CC(C)CN(C(c2cncn2C2CC2)=O)C1 c1(C(=O)NC2CCC(NC(C(N3CCOCC3)C)=O)C2)cc([N+](=O)[O-])n[nH]1 CC1CN(C(=O)CSCC2CCCO2)CCC1CNC(c1ccnc(Cl)c1)=O C1(NC(C2CC(OC)C2)=O)(CNC(c2csc(C)c2)=O)CCCCC1C Nc1cnc(Br)c(C(=O)NCCNC(C2CCCS(=O)(=O)N2)=O)c1 CC1C(NC(C2(CO)CC2)=O)CCCN1C(=O)COc1cccc(F)n1 c1(CC(N2CC(O)(CNC(C3CCC(C)S3)=O)C2)=O)csc2c(F)cccc12 C1(CNC(C=CC(=O)OCC)=O)CC(C)(C)CN1C(=O)CC1CC(C)C1 n1(CC(=O)NC2CCCCC2NC(C2(CCF)CCC2)=O)ncc2cccnc12 C12(C(=O)NC(C(CCC)C)C)CCC(CC1)N(C(=O)Cc1nonc1C)C2 C(=O)(CC(C)n1cc(Br)cn1)NCC(C)(C)NC(C(C1CCC1)OCC)=O C1(C(=O)NCCCC(C)NC(C2COCCN2C)=O)CC2C=CC1C2 c1(CS(C)(=O)=O)cccc(-c2cnc(N3CCCCC3)nc2)c1.C12(CC1)C(=O)N2 c1(C(=O)NCC2N(C(C(C)CC3CCC3)=O)CC(O)C2)cccc([N+](=O)[O-])c1O Cc1ccc(-c2cn(CCC3CC(NC(=O)Cn4nc(C)oc4=O)C3)nn2)cn1 O=S1(=O)C2=CC=CC(=NCC3(CCC3)N1)N2.C1(CO)C=CCC1 c1(C(CC)(C)C)ccc(C(=O)NC2(C)CN(C(=O)C(C3CC3)C3CC3)C2)cc1 c1(CCCC)nc(C)c(CC(=O)NC2CN(C(C3CC(C)N(C)C3)=O)CC2O)s1 C(=O)(CCCC(F)(F)CO)N1C(C)C(NC(=O)CN(C2CCSC2)C)CCC1 C(=O)(C(O)C(F)(F)F)NC(C(=O)NCC1(C)CCOCC1)CCC1CCC1 c1(OC)c(C(=O)NCC(c2ccccc2Cl)O)ccnc1F c1(C(N2C(CC(=O)Nc3nccc(Cl)c3Cl)CCC2)=O)c(Br)cncc1F Cc1nc(O)[nH]c1C(=O)NC1CC12CC(NC(=O)C(F)(F)C1(O)CCC1)C2 c1(C(C)C)c[nH]nc1C(=O)NCC1CCC(N(C)C)C1.C12CC(C1)OCC(=O)N2 CC1CCC(C(=O)NC2CCSCC2)N(C(C2CC2C2CC2)=O)C1 C(C(C)(C)C(F)(F)F)NC(C(c1ccnn1C)NC(c1nc(CC)oc1)=O)=O S(=O)(=O)(c1ccc(NCCC2(c3ccccc3)CC2)c(Cl)c1)Nc1c(C)cco1 C12(C(NOCC(=O)OC)=O)CC(CO)(CN1C(=O)CCN1CCOCC1)C2 C1(NC(COCCOC)=O)CCCC(C(=O)Nc2ccc(CCF)cc2)CC1 C1(C(=O)NC2C3CN(C(c4cc(OC)ncn4)=O)CC2C3)CCCC(C)(C)CC1 Cn1cc(C(=O)NCCC2CCCN2C(=O)COC2CC=CC2)c(O)n1 C1(NC(c2n(C)ncc2Cl)=O)CCN(C(=O)CC2CN3CCN2CC3)CC12CC2 C1(CCC(=O)NCCC#CCC)CCCCN1C(c1cc(C)nn1CC)=O N1(C(CCNC(COC)=O)=O)CCC(CO)(NC(c2ccc(=O)n(O)c2)=O)CC1 N1(C(CC2(OC)CC2)=O)C2CCCC1CC(NC(c1ccnn1C(C)C)=O)C2 C1(CC)(NC(c2nnn3c2CCC3)=O)CCCN(C(=O)CCOC2CC2)C1 N1(c2ncc(C(=O)OC)s2)CCCC2(NC(C3CC(C)CC(C)(C)C3)=O)CC2C1 N1(C(COCCCC)=O)CCCC(O)(CNC(=O)C(O)(CC)c2ccccc2)C1 c1(C(=O)O)ccccc1-c1csc(-c2nnc(-c3cccc(CCF)c3)o2)n1 C1(NC(=O)CCCn2ccnc2)CN(C(C2CC2C(F)F)=O)CC1C1CC1 c1(C(=O)NC(c2cccs2)C)c[nH]c2ccc(-c3scc4c3OCCO4)cc12 N1(C(C(C)C#N)=O)CC(CNC(=O)C=Cc2cc[nH]c2)CC(C)(C)C1 CC(C)C(O)CN1C(C(=O)NC(C)CCF)C(C)C1 C12(C(=O)NCc3ccnc(OC)n3)CC1CCN2C(C1CC(O)C(F)C1)=O CS(=O)c1ccccc1CC(N1CCC2(NC(c3ccncc3)=O)CCCC12)=O c1(CC)ccccc1CC(N1CCC(C(C)NC(c2ccc(CC)nc2)=O)C1)=O C1(NC(CCNC(=O)OCC)=O)COCCC1NC(C1CC1F)=O C1(NC(c2c(C)ccs2)=O)CN(C(=O)C(N)=O)C2(CCOC2)C1 CCC(C(=O)NC(Cc1cn(C2CCOC2)nn1)C(=O)O)Sc1ccccc1 CCC(C)C(O)C(=O)NC1CCCN(C(c2ccnc(OC(C)C)c2)=O)C1 c1(CNC2C(C(=O)Nc3cc(O)nc(CO)n3)CCCC2)n[nH]c2ccc(Cl)cc12 C1(O)(C(C)CNC(c2cncnc2)=O)CCN(C(=O)CCCC2(C)N=N2)C1 N1(C(=O)CO)CCC2CN(c3cc4ncnn4cn3)CCC12 C(N=c1[nH]cnc(Cl)c1F)C1CCC(NC(c2c(C)nc(CC)o2)=O)CC1 C=C(Cl)C(C)(C)C(=O)NCC1CN(C)CCN1C(c1ccn(CC(F)(F)F)n1)=O c1(C(N(CCCNC(=O)COC2CCCC2)C(C)C)=O)cc(F)cc(F)c1 C1(C(=O)NCC(CC)NC(c2cc(O)ccc2OC)=O)Cc2cc(F)ccc2O1 C#CC1(O)CC(C(=O)NC2CCN(C(=O)C(C)=C3CCC3)C2)C1 c1(C(C(=O)NC(CN(C(C=CC=CCC)=O)CC)C)CC)c(C)noc1C C1(NC(=O)CN2CCCC2)(CO)CCCN(C(C2CCCCC2(F)F)=O)C1 C1(CC)CC(CC(=O)NCCC(C)(C)CNC(=O)Cc2ccsc2)CCO1 C1(C(=O)NC2CN(C(C)C(=O)NCC3CC3)CC2C)CCC2(C1)CC2(F)F N1(Cc2c(F)ccc(C)c2)CC(C)Cc2cccc(O)c21 CCCCC(CNC(=O)CC1(C)CCCO1)NC(=O)CC1CN(C)C1 c1(OC)cccc(N(CC(=O)NCC2CCCCC2)C)c1Cl c1(C(=O)NCC(C)NC(c2ccc(CNC(C)=O)o2)=O)cc2c(Cl)cncc2s1 CC1CCC(C(N2CC(CNC(C3CC34CC4)=O)C2)=O)C1 c1(C(=O)NCC2C(CNC(Cc3scc(C)c3)=O)C2(F)F)cnc(O)cc1C C=Cn1ncc(C(=O)N(C(CC(F)F)C(=O)NCCC(O)C(C)C)C)c1N C1(CCNC(COC(C)(C)C)=O)CN(C(C2(C)CC=CCC2)=O)CCS1(=O)=O N1(C(C2N(C(CN(C(=O)OCC)C)=O)CCC2)=O)CCC(OC2CCOC2)CC1 c1(CNC(=NCC(C)C)NCC(O)COCC(C)C)ccc2c(c1)C(=O)NCC2 c1(C(=O)NC(C(C)NC(CC(CC)SC)=O)(C)C)nnn(Cc2ccsc2)c1C c1(OCC(=O)NCC(C)CNC(c2ncoc2CN)=O)ccc2c(c1)CCCC2 N1(C(=O)Cn2cc(C3CCC3)nn2)CCCC1C1(O)COC1 N1(CC)CCCC1C1CCCN1C(=O)Cc1cccnc1Cl CC1CCN(C(=O)CCc2nncn2C)C(C(=O)NCC2CC2(C)C)C1 Cc1cc(C(=O)N(C2CCCC2)CC(N2CC3C(CO)C3C2)=O)c2cc[nH]c2c1 c1(C(N(C2CCC(NC(=O)C(C)(C)F)C2)C)=O)cn(C)c(O)n1 C(C(C(=O)NC)N(C)C)NC(C)=O.C(C#CCCO)NC(C=CCOC)=O c1(OC)ccc(-c2cnccc2NCCC(=O)NCCC(C)C)cc1F C1(C(C)C(N2CC=CCC2)=O)CCCN(C(=O)CC2COCC2(C)C)C1 C(=O)(CCCCC#N)NCC(C1N(C(CCc2cnc(C)s2)=O)CCCC1)(C)C N#Cc1cscc1C(=O)NCC1(CNC(=O)CCOc2ccccc2Cl)CC1 C(=O)(C#CC1(C)COC1)NC(CC#CC)C(=O)NCc1ccc(F)c(F)c1 C1(C(=O)OC)CCCCCCN1C(C12CC(CN1C(=O)C(C)CO)C2)=O CC(CN(C)C)C(=O)NC1CCC1CNC(C1CC=CCC1)=O CCC(CC(=O)N1CCCC1C(=O)NCc1cc(OC)ncn1)C1CCC1 CC1(C(=O)NC(C2CCOC2)CNC(=O)C2=NNC(=O)C2)CCS(=O)(=O)CC1 c1(C(C(=O)NC(C)CCNC(=O)CN2CCCCC2)C)ccc(F)cc1 CCCCC(C)C(=O)N(C(C)C(=O)Nc1cncc(F)c1)CCC c1(C(N(CCN(C(CCC(=C)Cl)=O)C(C)C)C)=O)nsc2ccc(C)cc12 C1(CNC(C(C(C)C)NC(C)=O)=O)CCC2(CCNCC2)CO1 Cc1cc(CNC(=O)CCN(C(C2COCC(C)O2)=O)C(C)C)oc1C C1(C(N2CCCC(CC=C)C2)=O)CCC2CCC1N2C(c1cn2c(n1)CCC2)=O Cc1oc(C)c(C(=O)NC2CCC(CNC(=O)CNC(N)=O)C2)c1C N1(C(C(CC)OC2CCCCC2)=O)CC(NC(=O)CCCCO)CC2(CC2)C1 c1(C(C)NC(=O)NC2(CO)CCOCC2)ccc(OC(F)(F)F)c(Cl)c1 C1(CNC(C(CC)(C)O)=O)(CO)CCCN(C(c2ccc(C)cn2)=O)C1 C1(CC#C)(C(=O)NC(CNC(C2CC(n3ccnc3)C2)=O)C2CC2)CCCC1 Cc1cc(NC2CCCOC23CCC3)ncc1S(=O)(=O)N1CCCC1CF C1(NC(c2scc(C)c2)=O)CN(C(C2COCCC2(F)F)=O)C2CCCC12 CC(C)(CCNC(=O)CCc1cc(-c2ccccc2)on1)C(F)(F)F c1(C(=O)NC2CC3CC(NC(=O)CC4CC=CCC4)C2C3)cc2sccc2cn1 CC1CCCN(C(=O)Cn2ccnn2)C1CNC(c1ncc(F)cn1)=O C1(NC(c2ccc(C=C)cc2)=O)CN(C(=O)CCc2nc[nH]n2)CC(C)(C)C1 CC1CN(C(=O)Cn2cccn2)CC(C)N(C(=O)Cn2ccnc2CCC#N)C1 CCC(C)CCCCC(=O)N(CCNC(c1ccco1)=O)C(C)C Cc1nn(CC(=O)NCC2CC(NC(C3SCCCS3)=O)C23CCC3)c(C)c1C N1(C(C(C2CC2)OC)=O)CC(NC(c2cnc(O)cc2C)=O)CC(O)C1 Cn1c(CNc2ccc3[nH]nc(CO)c3n2)nc2cc(Cl)ccc12 N1(C(C2(C(=O)NC)CCC2)=O)CCC(F)(F)C(CNC(C2CC23CCC3)=O)C1 C1(C(=O)NCNC2CC2)CN(Cc2nccc(CO)n2)CCO1.n12cc(cn1)C2.CC c1(C(C)C)cccc(NC(CC2CN(C(c3cccc(C(C)(F)F)c3)=O)C2)=O)n1 c1(CN2C(C(=O)NCc3cccnc3)CC(O)C2)ccc2ncccc2c1 C=C(C)CCCC(=O)N1CC(OC)CC1CNC(c1cc(C(N)=O)cs1)=O c1(CNC2C(F)(F)CCN(C(c3cnc(C)[nH]3)=O)C2)c[nH]c2nccc(Cl)c12 N1(C(c2nccc(C)n2)=O)CCC(CNC(=O)C(C)N(CC(F)(F)F)C)C1(C)C Cc1nc(C(=O)NC(C2CCN(C(C3(O)CCSCC3)=O)C2)C)c(C)o1 c1(CC)nn(C)cc1C(=O)NC1CCCCC1CNC(=O)OC1CCC1 C1(C(N2CCC(CNC(C3CC(SC)C3)=O)C2)=O)CCCC(C)(C)C1 C(=O)(C1CC(=O)c2ccccc21)N1CC(CC)C(NC(=O)CCC(F)F)C1 c1(C(N2C(CCC)CCCC2)C(=O)NCCCSCC)cc(F)c(F)cc1F c1(C(N2CCC(N(C(C3C(OCC)C3)=O)C)C2)=O)ccc(N)nc1 N1(C(COCCCCC)=O)CCOCC(NC(=O)C(=O)NCCNC(C)=O)C1 C(=O)(C(C)(CC)CC=CCN1CCOC(C)(CC)C1)NCC c1(C(N2C(C(=O)NC(c3c(OC)cccc3)C)CCC2)=O)ncc(F)cc1C C1(C)(NC(CNC(CNC(C)=O)=O)=O)CCN(C(C2C3COCC23)=O)C1 N1(C(C(CC)C)=O)CCC2(CC1)CC(NC(c1ccnc(OCC(F)F)c1)=O)C2 Cn1cc(Cl)cc1CC(=O)NC1C2CC(NC(C3CC(C)(F)C3)=O)CC12 C1(CC)(CO)CCCN(CC(=O)N(C)C)C1.C(C)(C)(C)N(C)C(=O)O Cc1c(C(N2CC(NC(C34CC(CCO3)C4)=O)C2)=O)sc2ccc(Cl)cc12 c1(C(C(=O)N(CCN=[N+]=[N-])CC)NC(=O)C(C2CCCC2)OC)cn(C)nn1 N1(C(c2c(C)scc2)=O)CCC2CN(C(=O)CCC3CCCCN3C)CCC12 C12(C(N(C)CCOCCNC(=O)CC34COCC(C3)C4)=O)CC1COC21CCC1 C1(C(N2CCOCC(NC(c3c(C)ocn3)=O)C2)=O)CCC(S(N)(=O)=O)CC1 CC1CCc2nc(SC3(C#N)CCN(C(=O)OC(C)(C)C)CC3)cn2C1 c1(C(=O)NCC2OCCN(Cc3scc(C)n3)C2)cc2n[nH]cc2cc1Cl CC(C)C(C(=O)N(CC(C)(C)C#N)C)C(C)NC(=O)CCCn1cccc1 C(=O)(CC(C)(CN)C(F)(F)F)NCC(=O)NC(CC#C)CCOC C1(CNC(Cc2nc(C)oc2)=O)CCC(F)(NC(c2nn(C(F)F)cc2Cl)=O)C1 c12cccc(c1)C(=O)N(C)CC(C)CCO2.C(=O)(C=C(Cl)Cl)OCCCC N1(C=O)CC(S(C)=O)C1.C1(CNC(=O)OC(C)(C)C)(CO)CC1(F)F C(=O)(CCC(C)N(C)C)N1C(C(N2CC(CCO)(CC)C2)=O)C=CC1 CC(C)CC(CNC(=O)CC1CCCOC1)NC(=O)C(C)CO c1(CC(=O)N(C2CCN(C(c3ccc(C(F)F)cc3)=O)CC2)C)ccc(Cl)cn1 CC12CCC(CC1)CN2C(=O)CO.c1(C(=O)NCCSCC)ccc(F)cc1Cl CC1(C)C(CNC(=O)Cc2ccncc2Cl)CCN1C(C1Cc2nncn2C1)=O c1(NC(CC)(CNC(=O)CC2CC3CC3C2)CC)ccc([N+](=O)[O-])cc1C CCC(C)CCC(O)CC(=O)N(CCCCCCNC(=O)C1=CCCS1)C C1(CNC(C23CCC(OC)C2C3)=O)CCCCN(C(=O)CN2CCNC(=O)C2)C1 c1(C(=O)NCC2(F)CC(NC(C(C)O)=O)C2)cnc(OCC(F)F)c(Cl)c1.C1(C)CC1 Cc1cc(F)ccc1C(O)C(=O)NCCCC1(NC(c2cnc(S)[nH]2)=O)CC1 c1(C(=O)Nc2c(OCC)cc(C)cc2)ccc2c(c1)C=CS2(=O)=O CC1(C(=O)NC2CC(NC(=O)C(O)Cc3ccccn3)CC2O)CCCCO1 C(=O)(CC(C)(C)CNC(C1OCCCC1(C)C)=O)NC(CC=C)C C=C(Cl)CCC(=O)N1CCC(CCNC(=O)C(C2CCC2)OC)CC1 C1(C(=O)NC2(C3CCN(C(C4CCCCC4)=O)C3)CC2)CCC2(CC1)CC(O)C2 c1(OC)ccc(Cl)cc1S(=O)(=O)NC(=O)CCC1CCC(=O)N1 CC(C)CC(CN=c1cc(C(C)C)nc[nH]1)NC(C1CCCCN1C)=O CC1C(NC(c2cccc(Br)c2)=O)CC2CCC1N2C(=O)Cn1ccnn1 C1(C(=O)Oc2cccc(CC)c2)CCC(N=c2cc[nH]cc2OC)CC1 N1(C(=O)COc2ccc(F)nc2)CCC2(C1)CN(C(C1OCCO1)=O)C2 C#CCCC(=O)NC(c1cn(CC(C)NC(=O)C(C)(C)C)nn1)CC Cc1c(CNC(=O)C(=O)NC(c2cccc(F)c2)C)cccc1N(C)C Cc1cc(C)c(C(=O)NCCCN(C(C2CC2c2ccc(F)nc2)=O)CC)cn1 N1(C(C2C(C)(C)CO2)=O)CCC(CN(C(c2cccnc2O)=O)C2CC2)CC1 C(=O)(CCCCCCC(C)C)NCCOC(CNC(C(CC(=C)C)C)=O)(C)C c1(CCN2CC(CNC(C(CN(C)C)O)=O)OCC2)nnc2ccccn12 n1(CC(=O)NCC(C)NC(C(C2CCC2)OC)=O)ncc2ncccc12 N1(CCOC)CCC(OCCCS(=O)(=O)NCC)CC1C C(C)(C(=O)NC1CC(NC(=O)CC2(O)CCC2)C1)NC(C)=O c1(C(=O)NCCC(C(C)C)NC(C2CC3C=CC2O3)=O)ccn2ccnc2n1 CCCCCC(C)(C)C(=O)NCC(O)C(=O)NC1(C)CCC(C)(C)C1 C1(C(=O)NC(CNC(C=C(COC)C)=O)CO)(CC2CC2)CC=CC1 S(=O)(=O)(c1cc(F)ccc1C)NC(CC)C(=O)Nc1ccccc1[N+](=O)[O-] c1(C(=O)NC(C(C)NC(c2cn(CC)nn2)=O)C(C)C)cccc2nccn12 C1(NC(COCc2nnc(C)s2)=O)CCN(C(C2(CO)CCCCC2)=O)CC1(C)C C1(NC(C(=O)NC(CC)COCc2ccc(C(C)=O)cc2)=O)CCCCS1(=O)=O c12cccc3oc(nc13)c(=O)[nH]2.CC(C(CO)c1ccccc1)c1ccccc1 CCC(CC(=O)Nn1ccccc1=O)N(C(=O)CC1CCOC1(C)C)C CN1C(=NC(=O)N(C)Cc2cnc3ccccn23)NCC1c1ccccc1 CCCC(CNC(c1cc(C)sn1)=O)C(=O)NC(C)(C)CC(C)(C)C C1(CNC(C2(OC(C)C)CCC2)=O)CCCCN(C(c2cccc(CF)c2)=O)C1 N1(C(C(c2ccnn2C)C)=O)C2CCC1CC(NC(C1C(C)C1C)=O)C2 C1(NC(C(c2ccccc2)SC)=O)CN(C(=O)CC2CC=CC2)C2(CCC2)C1 c1(C(=O)NCCN(C(CC2(CC)CCC2)=O)CCOC)cc2cnccc2[nH]1 CCC(C)C(C(=O)NCc1nc(C)c(C(=O)N(C)CCN(C)CCO)o1)OC Cc1cc(C2CCC2)ncc1C(N1CCCN(C(=O)CSCCN(C)C)CC1)=O C1(C)(NC(C(C)CC2CCCC2)=O)CCCC1NC(=O)CN1CSCC1=O C(=O)(C(=O)NNC(=O)c1sccc1C(N)=O)N(C(C)Cc1ccc(C)cc1)CC N(C1CCCc2ccoc21)C(C1(NC(c2ncn(C(C)C)n2)=O)CC(CO)C1)=O c1(C(C(=O)NC(CCNC(c2c(CC)n(CC)nc2)=O)C)O)cc(F)cc(F)c1 c1(-c2cn(CC3CC(CNC(C(C=C)(F)F)=O)C3)nn2)ncc(Cl)cc1F S(=O)(=O)(CC(=O)NCC1C(C)CCN1c1ncc(O)cn1)NC Cc1nc(Cl)c(NCC2(c3ccc(-c4cc(F)c(F)c(F)c4)cc3)CC2)cc1Br CC(F)(F)C(C)(C)C(=O)NC(CNC(c1ccc(SC2CC2)cc1)=O)CO N1(C(c2c(OC)scc2)=O)CCC(C(F)(F)F)C(CNC(=O)CC(C)SC)C1 C(=O)(CC(CN(C)C)C(F)F)N1CCC(CNC(C=C(CC)CC)=O)C1 N1(C(Cc2ccc(C)c(C)c2)=O)CCN(C(=O)CCP(C)(C)=O)CCC1C.C(CC1CCC(C)C1)O CC(C)(CCC(=O)N1CCC(NC(=O)C(O)C2CCCC2)C(C)(C)C1)[N+](=O)[O-] C(CS(=O)(=O)CC(=O)N(N1CCCN(C(=O)CSCC(N)=O)CC1)C)OC N1(CC(=O)Nc2cc(CCCCC)[nH]n2)C(C)(C)CC(=O)CC1(C)C C1(C(=O)NC(c2cn(CCC=C)nn2)CC(N)=O)CCCC(C2CC2)O1 O=C1CCCCC1CC(N1CCC(C(=O)NCC2CC3CCC3C2)C1)=O N1(C(CC2N(C(c3cc(C)ncn3)=O)CCC2)=O)CCC(C)C(CO)C1 C(c1c(F)cccc1F)=CC(=O)NCCCn1cc(CO)nn1.C1(OCCO)COC1 c1(NC(=O)NC(c2ccc(CO)cc2)C)ccn(O)c(=O)c1 CC12CCC(CN3CCC(CC(N)=O)CC3)(CO1)C2 c1(N(C)C)ccc(NC(=O)CC2CCCC2NC(C2CC(=O)CCO2)=O)cc1 C1(CN(C(=O)COC2(C)CCC2)C)CCCN1C(=O)C(c1ccccc1)SC1CC1 C1CCCCCN=C2C=CC(=CN2)S(=O)(=O)N1.C1(CSC)(OC(C)C)CCC1 C1(C(=O)NCC(C(C)(C)C)O)CC2CC1CC2NC(C1CC2CCCC2C1)=O C1(NC2CC(=C)C2)CCN(C(=O)COC(F)(F)F)CC1C c1(C(N2CCC(CC(=O)NCc3cnc(C)s3)C2)=O)cnc2[nH]cncc1-2 C1(C(C)NC(C2(C)CC(C)C2)=O)CN(C(c2nn(C)cc2N)=O)CCO1 C1(NC(CNC=O)=O)(CO)CCCN(C(=O)CCC2CCCC(=O)N2)C1 C1(NC(c2c(C(C)C)ncs2)=O)CC(NC(C2CCCC(C)C2)=O)C(O)C1 Cc1cccc(Br)c1C(C(=O)NCc1nc(C2CC2)n[nH]1)NC(=O)COC(C)C c1(NC(=O)C2=CCC2)cccc(NC(C2C3CCCOC23)=O)c1 C1(O)(C(=O)NC(C)C(=O)Nc2ccc(Cl)cc2Cl)CCN(C)CC1 N1(C(CSCC)=O)CCC2(CCC(CNC(c3ocnc3C)=O)OC2)CC1 C=CC1(C(=O)NCC(C)OC(F)F)CCN(C(C2CC23CCC3)=O)CC1 c1(C(N(C(c2c(COC)noc2)C(=O)NC)C)C)ccc(S(C)(=O)=O)cc1 C=CCC(C(=O)NCCC1(NC(=O)C(O)C(C)C)CC1)C(C)C C(=O)(CC1OCc2ccccc21)NC1CC(NC(CCC=C)=O)C1 C1(C(N(C2CCN(C(=O)C=Cc3ccncc3)C2)CC)=O)CCC2(C1)CC2(F)F CN1CCOCC1C(N1CCC(N(C)C(c2ccccc2)C2CC(C)(O)C2)C1)=O Cc1cnn(C(C)C(=O)NCC2CC2NC(C2CC2c2ccc(Cl)s2)=O)c1 c1(C(=O)NC(C2CC(C(=O)NCC(F)(F)F)C2)C)cccc(=O)n1C c1(NC(C23CC(CNC(c4ccc(OC)cn4)=O)(C2)C3)=O)cc2n(n1)CCC2 c1(C(=O)NC(CCNC(C2CC(CCC)C2)=O)(C)C)ncc2ccccn12 Clc1ccc(-c2nc(C3CC3c3cn[nH]c3)n(CCCO)n2)cc1 C(=O)(C1=NOC2COCC12)N1CCOCC(CNC(CC(C=C)(C)C)=O)C1 C1(NC(C2(C)CCCOC2)=O)CC2CC1N(C(c1c[nH]nc1C1CC1)=O)C2 C1(NC(C(C(CC)O)C)=O)CC2CCCC(C1)N2C(=O)CCSc1ccccn1 C(=O)(C1=CCC2CCC1N2C(c1cncc(Cl)c1)=O)N(CC(CC)O)C C1(C)(CC(=O)NCC(CC=C)NC(c2cnccn2)=O)CCCCC1 C(=O)(NNC(=O)CCCN)NC(c1ncc(CC)s1)C c1(C(N2CC(O)(CNC(c3nc(CC)oc3)=O)C2)=O)n[nH]c2cc(OC)ccc12 C1(C(N(C)Cc2ccc(CC)o2)=O)CN(C(c2cnn(C)c2N)=O)C(C)(C)C1 C(C)(C(C(=O)N(CC(=O)NCC1COCC(C)O1)CC1CC1)N(C)C)OC n1(CC(=O)NCC(CC)NC(C2(COC)CCCO2)=O)c(O)nnc1O C1(C(=O)NC2CCN(C(c3cncc(OCC)c3)=O)C2)CCc2cnnn2C1 C1(NC(C(C)(C)OC)=O)CCCN(C(C2OC(C)(C)OC2=O)=O)CC1 C1(NC(C2C(C(=O)OC)C2)=O)CC(F)(CNC(c2sncc2C)=O)C1 C=C(C)CC(C(=O)NCC(C)(C)CC1CC1)NC(C1CC(=C2CC2)C1)=O.COC C1(NC(c2c(CC)occ2)=O)(CNC(=O)C(F)OC(F)(F)F)CC(F)(F)C1 N1(C(N(c2ccc(F)cc2)CC)=O)CC2(CC2)c2ncccc21 CN1C(=O)CC(N)C1c1cccs1.N12CCN(CC1)C(=O)NNC(=O)C(=O)C2 N1(C(=O)CN2CCN(C(c3cccs3)=O)CC2)CC2CCC(C1)C2O N1(C(c2nc(-c3ccc(C(F)(F)F)cc3)no2)C)CCc2cc3c(cc2C1)CCCC3 N1(C(C(C)(C)C2CCCC2)=O)CCCC(CNC(=O)CN2CC3C=CC2C3)C1 C1(CNC(=O)CN2CC3CC3C2)CCC(C(N2CCC3CC23)=O)CC1 C(=O)(C(Cc1ccccc1)C12CCCC1C2)NCC(C1CCC1)OC N1(C(=O)CCC2CCCCO2)CCN(CCCNC(C2CC(O)C2)=O)CC1 C1(CC)(CC)CC(O)CN1C(=O)C(CNC(C1OCCC1C)=O)N(C)C C1(C(=O)NC2CC(CNC(COCC(=C)C)=O)C2)CCCCC(C)(C)C1 c1(C(=O)NCCC(F)Cn2cc(C3(C(=O)O)CC3)nn2)cnc(O)c2ccsc12 N1(C(CC(CCC)(C)C)=O)CCC2(CC1)CCN(C(C1(O)CCCC1)=O)C2 C1(C(=O)NCC(C2N(C(COCC(C)C)=O)CCC2)(C)C)C(F)(F)C12CC2 c1(C(=O)NC2C(CNC(C3(C(C)C)CC3)=O)C2)cc2ccc(F)cc2nc1O Cc1cc2ccc1C(=O)N1CCOC(C1)N2.C1(CN(C)C)CCCCCC1 C1(C(=O)NC2C(C)CCC2)CC2OCCC2N(C(=O)Cc2ccsc2)C1 c1(C(N2CC(NC(C(C(=C)Cl)(C)C)=O)CC3(C2)CC3)=O)ccc2c(cnn2C)c1 CC1CC(N(C(=O)CC2CC(N(C)C)C2)C(c2ccc(F)c(F)c2)=O)CN(CC)C1 c1(C(=O)NCC2C(NC(C3CC(N=[N+]=[N-])C3)=O)CCC2)cnn2c1OCCC2 CC1CC(C(=O)NCC(F)(F)Cl)CN(C(=O)CC=CC(C)(C)C)C1 N1(C(c2ccc(Cl)[nH]2)=O)CCC2OCCN(C(=O)CC3CC=CCC3)C2C1 c1(C(=O)NC(CNC(C2CC3(C2)CC(F)C3)=O)CO)cc2cccc(Cl)c2s1 C(c1ccoc1)=CCNC(C12CC(CO1)C2)C.C(CO)S C12(C(N3C(CN(C)C)C=CC3)=O)CCC(CN(C(=O)CCC3CCCC3)C1)C2 c1(C(=O)NCCCCCCN(C(C(C)CC(N)=O)=O)C)cccc2[nH]ncc12 C1(CNC(c2cc(CC)oc2C)=O)CC2(CC2)CN1C(=O)CC1OCCCO1 N1(C(C(CSC)(C)C)=O)CC2(CC(CNC(=O)Cc3cc(F)ccc3C)C2)C1 C(CC(C(=O)NCC(C)C1CCC1)NC(c1ccc(OC)o1)=O)OCC C(CCNC(c1ccc(CC(N)=O)cc1)=O)(C(C)(C)C)NC(C(C)SC(C)C)=O N1(C(CN(CCOC)C)=O)CCC2(NC(=O)C=Cc3ccsc3)CCCCC12 c1(N(C(CC)=O)C)ccc(NC(=O)NC2(CO)CC(F)C2)cc1 c1(CC)cccc(C(N2CC(O)CC2CC(N2CCCOCC2)=O)=O)c1 Cc1cccc(CC(=O)NCC2(O)CC(NC(=O)C(c3ccccc3)F)C2)c1 O=S(=O)(c1c[nH]ccc1=NCC1(S(=O)(=O)c2ccccc2)CC1)N1CCCC1CO c12ccc(cc1)NCc1nnnn1-2.c1(CCCC)cn(Cc2ccc[nH]2)nn1.OC c1(C(N(C2CN(C(C3CC(O)C3)=O)CC23CC3)C)=O)cc(Br)cnc1F C1(NC(=O)CC2COCCO2)(CO)CCCN(C(C2CCNC2=O)=O)C1 C1(C(N2C(C(N(C(CC(C)C)C)C)=O)C(C)C2)=O)COCCN1C C1(OC)CCC(O)CN(C(C23CC(C=O)C2C3)=O)C1.c1(SC)nccc(C)n1 c1(C(CNC(c2cc(C)[nH]n2)=O)NC(C2(NC(N)=O)CC2)=O)cccc(Cl)c1 c1(C(CC(=O)OC)NC(=O)NCC(C)(C)OCC(=O)O)ccccc1F Cc1cc(Cl)ccc1C(=O)NCC1CCN1C(c1cnc(S)n1C)=O C1(NC(=O)CCc2cc(Cl)cs2)CCC2CC1CN2C(=O)CCc1cnc[nH]1 n1(CC(C)C)[nH]c(C2CC2)cc1=O.c12cnc(s1)NC(=O)C2.C(C(=O)NCC)SCCl N1(C(c2cccc(SCC)c2)=O)CC2CCC(NC(=O)C(COC)OC(C)=O)(C2)C1 CC(C)(C)CC(C)(C)C(=O)N1CSCC1C(N1CCc2c(nnn2C)C1)=O c1(CCC(=O)C(=O)ONC(CN(C2COC2)C(=O)OC)=O)ccc(Cl)cc1F.O CC(C)(O)C(F)C(=O)N1CC2CC1C2NC(=O)CC1=CCCC1 N1(C(c2cc(C)nc(C)n2)=O)CC(NC(C2(C(F)F)CCCC2)=O)CC(C)(C)C1 c1(OC)c(C(N2CCSCC2C(=O)Nc2cc(C)c(F)cn2)=O)cccc1Br N1(c2ncnc(CC)n2)CC2CC(NC(=O)C(O)C(C)CC)CC2C1 C1(c2cccs2)(C(=O)NC(c2cccc(F)c2)CO)CCOCC1 C12(NC(CC(=O)OC)=O)CCCC1CN(C(c1nccc3occc13)=O)C2 C1(NC(C(C)(C)OC(C)C)=O)CCC(C(=O)NC(C(C)(C)O)C2CC2)CC1 c1(C(=O)NC2CC(C(C(=O)NCC=CC)F)C2)cc(OC)n[nH]1 C(=O)(CS(=O)Cc1cccc(Br)c1)N(CC=C)CCOC N1(C(c2ncc(C)cc2C)=O)CCC(NC(c2cnn3c2OCC3)=O)C12CCC2 N1(C(C=C(CCC)C)=O)CCCC(C)(CC(=O)NC2C3COCC23)C1 c1(NC(C23C(CN(Cc4c(O)ccc(OC)c4)C2)C3)=O)cccc(C#N)c1F CN1C(=O)CSC1=CC(=O)NCC1(F)CCC(NC(=O)CC2CCCC23CC3)C1 C1(CCOC)(NC(=O)Cc2ccc(Cl)cc2F)CCN(C(=O)C(O)C2CC2)CC1 N1(C(c2cc3c(Cl)cccn3n2)=O)CCC2OCCN(C(C3C=CCC3)=O)C2C1 C1(C(=O)NCC2CCCC(NC(=O)C(c3ccnn3C)O)C2)(OC)CS(=O)(=O)C1 C1(NC(c2nc(OCC)sn2)=O)CCCC(NC(c2cncc(SC)c2)=O)C1 c1(C(=O)NC2(COC)CN(C(C3CCCCC3(C)C)=O)C2)ccc(C#N)cc1C CC1(NC(c2cc(=O)cc[nH]2)=O)CCN(C(C2(C)CC3CC3C2)=O)CC1 C(=O)(CC(C(C)C)c1ccccc1)NC(CCNC(C1C(C)(CC)C1)=O)C CCC(CC(=O)N1CCC2(C1)CN(C(c1ccc(O)c(N)n1)=O)C2)C(F)F c1(C(=O)NCCCC2N(C(C#CC(C)(C)C)=O)CCC2)cccc2c1C(=O)NC2 C1(C)(C(=O)NCC(C)(C)CNC(=O)Cc2ccc(NCC#N)cc2)CCCN1C c1(CC(=O)NC2(CC)CN(C(=O)C(C)CCCOC)C2)cncc(C#N)c1 C1(NC(C2(OC(=O)C(F)C(=O)NCC)CC2)=O)CCOCC1(C)C N1(C(c2c(C)nc(C)s2)=O)CC2C=CC1C(C(=O)NCCN1CC(CF)C1)C2 C(=O)(CC(C)C(F)(F)F)C(C)C(N1C(C)COCC1(C)C)=O CCC(C)C(O)C(C)C(=O)N1CC(NC(=O)C(C)C(C)C)CC(C)C1 c1(NC2CC(C)(CC)C2)nccc(N(C)CC2CC2)n1 C(=O)(C1=CCC2CCC1N2C(=O)C(C)(C)C(N)=O)NCC(C)C#N CC1(C)CC(NC(=O)Cc2cc[nH]c(=N)c2)CN(C(c2ccc(Cl)s2)=O)C1 c1(C(=O)NC2CN(C(C3(C=C)CCCC3)=O)C2)cc(OC)ccc1F c1(OC)c(NC(=O)C(=O)Nc2ccc(OC(C)C(C)C)cc2)c(C)nn1C Cc1cc(=NC2CCN(C(c3cccc4cc[nH]c34)=O)CC2)[nH]cc1C#N c1(OC)nc(Cl)ccc1C(=O)N(CCC(C(C)C)NC(=O)CC(O)C(C)C)C c1(OC)cccc(CC(=O)NCCC2CSCCN2C(=O)COC2CCC2)c1F N1(C(CC(C)CN(C)C)=O)CCC(NC(C2CC(C)(C)C2)=O)C(F)(F)CC1 c1(C(N2CCCC(CCNC(Cc3cc(C)ns3)=O)C2)=O)c(C)cc(C)oc1=O Fc1cc(-c2cccc(C(F)(F)F)c2)ccc1SCC1COC1 C1(CNC(C2CC(C#C)(O)C2)=O)CC12CCN(C(=O)C=C(C)Cl)CC2 CC1(C)CN(C(=O)C(CNC(C2(C)CNC(=O)N2)=O)CC2CCCC2)CCS1 N1(C(C2C(C=C)C2)=O)CCCC12CCC(NC(=O)C=C(C)CCC)CC2 Cc1cccc(F)c1C(N1CCCC(CCCCNC(c2cnn[nH]2)=O)C1)=O C1(C(=O)NC(CNC(c2cc(OCC)no2)=O)(C)C)CCC2CC1C2(C)C Cc1ccc(CC(N2CC3CN(C(c4cnon4)=O)C3C2)=O)c(C)c1 C1(NC(C(C)N(C)C)=O)CCCC12CN(C(=O)Cn1cc3ccccc3n1)C2 n1(CC)nccc1-c1cn(C(C)(C(=O)NC)NCCCSC(F)(F)F)nn1 N1(C(C(C)SCCCC)=O)CCC(O)(C(C)NC(c2[nH]ccc2C(C)=O)=O)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CC)CNC(C1(COC)CC=CC1)=O C(=O)(C#CC1CCOC1)NCCC(=C)CNC(C1CC(C(C)C)=NO1)=O n1(C(CC)C)nnnc1C(c1ncoc1COC)NC1CCSC1 N1(C(C(C2CCOC2)OCC)=O)CCCCC1CNC(=O)CCCCF c1(CC)cc(N)ccc1C(=O)NCC(O)CNC(C1CC1F)=O C(=O)(C1CCCc2cccnc21)NCCCCNC(c1nc(CCC)sc1)=O c1(C(N2CCCC2c2cccc(O)c2)C(=O)NC)nc2c(s1)CCCC2 c1(CCC(=O)NC2(C(=O)NC(C)C(F)(F)F)CCCC2)cc(F)ccc1F c1(C(C(N2CCC(NC(C3C4C=CC3CC4)=O)CC2)=O)=O)ccc(Cl)cc1O Cc1cnc(C(N2CC3C(CNC(C4(n5ccnn5)CC4)=O)C3C2)=O)cc1Cl c1(C(=O)NC2CCCC23CC3)ccccc1-n1cc(CCO)nn1 c12cccc(c1)OC1(CCCCNC(=O)C2)CC1.C=CC(O)C(=O)NC(C)C C1(NC(C2C(=O)NCC2)=O)(CNC(C2(C3CC3)CCCO2)=O)CCCCC1 CC1CN(C(C2C(C)CN2C(=O)C(C)CC(F)(F)F)=O)c2ccccc21 c1(C(N(C(C)C(N2CCCCC2CO)=O)C)=O)cccc(F)c1 c1(C(N(CC(O)CN(C)C(C2(c3cc[nH]n3)CC2)=O)C)=O)cc(Cl)cc(Cl)c1F c1(C(N2C(CC)CN(C(=O)CNC(C)=O)CC2)=O)nc2c(s1)COCC2.C(=O)(CC)N c1(C(C)NC(N2CCC(C(N3CC4CC4C3)=O)C2C(F)F)=O)ccc(Cl)cc1 c1(CCC)cccc(C)c1C(c1nnnn1-c1ccccc1)NCC1(OC)CC1 CCCC(CCC)=CC(=O)NC1(CO)CCN(C(C2CCCO2)=O)C1 C(=O)(CCCCCCC)NCC1(C(=O)NCCCC)CCCO1 C(=O)(CCC(C)C)NCC1N(C(C2N=C(C)SC2)=O)CC1 Cc1cc(CC(N2CCCC2C(C)CNC(C2(C)CCNC2=O)=O)=O)cc(C)c1 Cc1ccc2c(c1)C(NC(=O)C(C(C)C1CC1)NC(=O)OC(C)(C)C)CO2.OCN C(=O)(C1=CCC2CCC1N2C(c1n[nH]cc1Cl)=O)NC(C1CCCC1)CC C1(CC(=O)N(CC2CN(C(C3CN(CC(C)C)C3)=O)C2)CC)CCCCC1(C)C Cc1noc2cc(C(=O)NC3CCC34CN(C(=O)CN3CCCC3=O)C4)ccc12 Cc1cc(C(N)=O)ncc1NC(=O)NCCCCN1CCS(=O)(=O)CC1 c1(C(=O)NCC(CCNC(C(C=CCCC)O)=O)O)sc(C)c(C)c1C N1(C(C2C(OC)CCCC2)=O)CCC(CNC(c2cnc(Cl)[nH]2)=O)C(C)C1 N1(C(CS(CC)=O)=O)CC(C)(C)CCC1CNC(=O)C(C(C)O)N(C)C c1(NC2C(c3ccc(C)s3)CCC2)ccncc1S(=O)(=O)NCc1ccon1 C1(NC(C(C(=O)OCC)(C)C)=O)CC2(CCN(C(=O)C=Cc3ccc[nH]3)C2)C1 C1(NC(C2(C)CCC2)=O)(CO)CCCN(C(C2(CO)CCCO2)=O)C1 C(=O)(CS(=O)(=O)CCO)NCC1C(C)CN1C(N)=O.C1(C(C)C)C(=O)N1 C(=O)(CCCC(F)(F)C(F)(F)F)N1C(C)(COC)CC(NC(=O)CC=C(C)C)C1 C(=O)(C1=CC2(CCN(C(c3csc(C#N)c3)=O)C2)C1)N1CC2C(C)(CSC2)C1 n1(C(N(CCN(C(=O)CCOC2CCCC2)CC)CC)=O)nc(C)c(C)c1C N1(C(COCCCC)=O)CC(CCNC(=O)C(C2CC(F)(F)C2)O)C(C)C1 CC1CCC2(CC2)N(C(C2CCC(C)(C)N(C(c3c(F)cccc3F)=O)C2)=O)C1 C12(CCNC(=O)Cc3cnc[nH]3)CCC1CN(C(c1ccc(C3CC3)nc1)=O)C2 Cc1cc(C(=O)NCC2CC2CNC(c2ccoc2)=O)nn1-c1cccc(F)c1 N1(C(c2c(CCC)[nH]cc2)=O)CCN(C(c2nc(C)ccc2F)=O)C(C)CC1C N1(C(C2(C=C)CC2)=O)CC(CNC(c2cc(O)nc(OCC)n2)=O)C(F)(F)C1 c1(C(N2CC(=C(CNC(C(CCCC)O)=O)F)C2)=O)ccc2c(c1)NC(=O)C2 N1(C(=O)OC(C)(C)C)CC2CCN(C(=O)C=CC3=C4C(C)(CN=C3)N=N4)CC2C1 c1(C(N2CC3C(C2)N3C(c2cccc(Cl)c2)=O)=O)ccc(Br)cc1I C1(NC(C2CCS(=O)(=O)C2)=O)CC2CCC(C1)N2C(=O)CCC1CCCC(O)C1 c1(C(N(C2CN(C(=O)Cc3cc[nH]n3)C2)C)=O)ccc(Cl)nc1N C#Cc1ccc(OC)c(C(=O)NC(C)(CNC(=O)Cc2ccc(F)cc2)CC)c1 Cc1ccc(C2(C(=O)NC3CCN(c4nc(C)ns4)CC3)CC2)c(Cl)c1 Cc1cccc(C)c1CC(N1CC(C)(C)CC1CNC(=O)Cc1cccnc1)=O C=C(C)CCCC(=O)NCC1CCC(NC(=O)CCCC2CCCO2)C1 C1(CNC(Cc2c(C)con2)=O)CC(C(=O)NCCC2(C)CCCO2)=NO1 C1(O)(CNC(C2C3CCC(=O)C23)=O)CCN(C(c2ccnn2C2CCC2)=O)CC1 C=CCCCCCCCC(=O)NCC(O)CCNC(=O)Cc1ccccc1OC CCC(C(=O)NC(CNC(C1CC(c2ccccc2)C1)=O)CCOC)N(C)C CC1(C(=O)OC(CCOCCNNC2CC3(CCC3)C2)=O)CC2C=CC1C2 C1(C(=O)O)(CC)CCCN(Cc2ccc(C(N)=O)cc2)C1 C(C(C)N=c1[nH]c2ccccc2nc1C#N)(c1ccccc1)NC(CCC(=C)Cl)=O O=C(CCCC(=O)N1CCCN(C(C23CCCC2C3(F)F)=O)CC1)C1CC1 C(=O)(C(C)CC1CC1)NCCC(C)N(C(C(C)NC(C1CCCC1)=O)=O)C c1(C(=O)NC2CN(C(CC3(C=C)CCC3)=O)C(C)C2)cn2ccnc2s1 c1(C(N2C(CNC(CCC3N(C)CCC3)=O)CC2)=O)cnc2cccnn12 C(CCC)(C(O)C(=O)N1CC2CCC2(COC)C1)NC(CNC(=O)OCC=C)=O c1(C(=O)NC(C2N(C(c3ccc(C)o3)=O)CCC2)C)cc(C)c(F)c(C)c1 C1(CNC(CC(=C)C)=O)CN(C)CCN1C(=O)CCS(C)(=O)=O c1(C(=O)NC(CN(C(CCCC(CC)C)=O)C)C)cc(F)c2ncccc2c1 c1(CCC(=O)NC2CCN(C(CCC#C)=O)C2)cncc(F)c1 CC1(C)CC(NC(=O)COCCF)CN1C(c1coc(-c2ccsc2)c1)=O C1(CNC(C2(CCN=[N+]=[N-])CC2)=O)CN(C(=O)C2=COCC2)CC1c1ccccc1 C(=O)(C1=CCC2(CC1)CC2(F)F)N(CCCNC(=O)C(F)C1CCOC1)C N(C(=NCc1ccc(C(=O)NC)cc1)N1CCC(C(C)C)C1)C(C=C)C N1(C(CC2N(C)CCC2)=O)CCCC(NC(=O)Cc2cc[nH]c2)CC1 c1(NC(C2CCOC2)=O)cccc2[nH]c(-c3cccnc3C(F)(F)F)cc12 Cc1cc(C)cc(C=CC(=O)NC2CCN(C(c3ccoc3)=O)CC2(C)C)c1 c1(CN2CCCC(C(N(CC=C)CC3CC3)=O)C2)c(OC)cccc1F N1(C(c2occ(C)c2)=O)C2CCC1CN(C(c1cnc(Cl)cn1)=O)CC2 N1(C(c2c(C)nccn2)=O)CC(NC(=O)C(c2ccc(Cl)c(Cl)c2)C)C(C)(C)C1 C(=O)(CC1=CCCC1)N(CC(=O)N(C1CCCC1C#N)C)C1CC1 N1(C(COC2(CNC(C3COCCO3)=O)CC2)=O)CCC(SCCCC(N)=O)C1 c1(CNC(C2C(C)C2)=O)ccccc1NC(C1CC1COC1CCCCC1C)=O c1(C(=O)OCC)cc(-c2ccc(CN(C)Cc3ncc(Cl)s3)cc2)cn1C C1(NC(c2n(CCOC)ncc2)=O)CCCN(C(=O)C(n2nc(C)cc2C)C)C1 c1(C(c2nnnn2CCO)C2CC2)cn(C)c2ccc(F)cc12.C(C(C)N)NC(=O)OC C(=O)(CCCCC#N)NC(c1ccc(C)cc1)CNC(C1(Cl)CC12CCC2)=O C=CC(C)(O)C(=O)NCCN(C(C1CCN(CC(F)(F)F)C1)=O)C(C)C C1(C(=O)NCCS(CC)=O)CCC2CCC1N2C(c1ccoc1C1CC1)=O CC(C)CC(C)(O)C(=O)N1CCC(F)(C(=O)NC(C)(C)CC2CCOC2)C1 c1(C(=O)NC2CCC3(C(NC(CCCOC)=O)C3)CC2)cnn2c1CN(C)CC2 N1(C(C(C)OCC(F)(F)F)=O)CC2(CCC(NC(=O)C(F)C3CCCC3)CC2)C1 Cc1cnncc1C(=O)NC(CC1CCCC1)C(=O)N1CCC1C1CCCC1 CN(C)S(=O)(=O)N1CC2(CC(c3ccccc3)=NO2)C1 CCC(CC)C(C(=O)NC1(COC)CCN(C(c2cc(CO)[nH]n2)=O)CC1)OC CC1=C(C(=O)NC2CN(C(c3onc(C)c3C)=O)CC2O)CCS1(=O)=O N1(C(C(C)OCC)=O)CC(CNC(c2csc(C(F)F)n2)=O)C(O)C1 CC(O)C(C(=O)NC1COCCC1O)N(C)C.C1(NC(=O)CN(C)C)CC(N)C1 C(=O)(C(C)(C)CC1CCOC1)NCCOCCOCCNC(C1CCC(CC)C1)=O c1(C(N2CC(NC(CCC(=O)NC)=O)C2)=O)nc(Br)n2c1COCC2 C(C)(C)(CCC(=O)NCC1CC(OC)C1(C)C)NC(C(COC)COC)=O C1(C(=O)NCC2N(C(c3ccc(OC)cc3C)=O)CC2)CN2CCCN1CC2 N1(C(C(N2CCC(O)CC2)C)=O)CC2CC(C1)CN(C(c1csnn1)=O)C2 C=CCC(CC=C)C(=O)NCC(c1cccc(C)c1)NC(c1cc(OC)n[nH]1)=O Cc1ccnc(O)c1C(=O)NC1CCCC(N(C(=O)CC2CSC2)C)C1 C1(C(=O)OC(C)(C)C)CCN(C(=O)C(F)=CCOC(C(C)SC(F)F)C)CC1 C1(NC(=O)C(=Cc2c[nH]cn2)F)CCOCC1NC(=O)CC1CCCC12CC2 c1(C(=O)NCC=CCNC(C(C)N2CCC2)=O)ccc(=O)n2c1CCCC2 C(=O)(CC(P(C)(C)=O)P(C)(C)=O)NCC1(C)CCN(C(C(COC)(C)C)=O)C1 Cc1cnc(Cl)c(CN2CC(C(=O)Nc3c(F)cccc3Br)CC(F)C2)c1 C(=O)(C(CNC(=O)C(F)C(C)(C)O)C(C)(C)C)NCCN(C(C)C)CCF CCC(C)(C#N)C(=O)NCC1CN(C(c2cc(Cl)c[nH]2)=O)CCCO1 C1(C(=O)NCCC)CN(C(=O)CNC(C2CC2C(=O)OC)=O)CC1CC c1(C(N2CC(F)CC(C(=O)Nc3cc(O)ccn3)C2)=O)ccc(F)c(F)c1O C1(NC(c2cc(OC)cc(Cl)c2)=O)CN(C(C2CC(O)C2)=O)CC2(CC2)C1 c1(OCC=C(C)C)ccc(C(C(C)C)N(CCC(=O)NC2OCCCO2)C)cc1 N1(C(CCC(C)N(C)C)=O)CCn2nc(CNC(=O)CC(C)(F)F)cc2C1 N1(C(C(C(CC)(C)C)O)=O)CC2CCCC(Nc3ncnc(Cl)c3C)C2C1 C1(CC)(CC)CN(C(C2(NC(=O)C=Cc3cocn3)CC2(C)C)=O)CCO1 C1(OC)CCC2(C(=O)NC3(C4CN(C(=O)C(C)S(C)(=O)=O)C4)CC3)CCC12 c1(OC)cc(C(=O)NCC2CCC(C)N(C(=O)CCCSC)C2)cc(Cl)c1 N1(C(c2nc(C)oc2)=O)CCC2(CC1)CC(NC(=O)C(C)c1cccs1)CO2 C(N=c1[nH]nc(C(C)(C)C)o1)C1C(NC(c2cc(CC)no2)=O)CCCC1 C1(NC(=O)C=Cc2cc[nH]n2)C2CCN(C(=O)CCc3cccc(O)n3)CC12 c1(OC)cccc2c(C(N3CCCC(NC(=O)CCC(F)(F)F)C3)=O)c(C)[nH]c12 C1(NC(c2c(CC)oc(C)c2)=O)CN(C(c2cc(CSC)c(C)o2)=O)C2(CCC2)C1 C1(C(=O)NC2(CN(C(=O)CC(C)C(C)(C)C)C)CC2)CCc2c(nnn2C)C1 c1(C(=O)OCC)cnn2c1N(C(c1ccnc(OC)c1)=O)C(C)CC2 CCS(=O)(=O)c1ccc(NC(=O)CCCNC(=O)NC(C)(C)C)cc1 C(=O)(C(O)C(CCC)NC(=O)C(C)C(O)C(C)C)N(CC#CC)CC#C C1(NC(=O)CC(C2CCC2)C2CCC2)Cc2cc(F)ccc2NC1=O N1(C(COCC=C)=O)CCC2(CC1)CC(NC(c1cccc(C)c1)=O)CCO2 C(C#CC(=O)NC(C1CCCN(C(c2cccnn2)=O)C1)C)(OCC)OCC C1(CC(=O)NCc2cn(CC=CC)nn2)CCCN(c2ccc(OC)cc2)C1 c1(C(N2CC(F)(CNC(c3c(C(C)C)onc3)=O)C2)=O)cccc2c1NCCC2 N1(C(C2N(C(c3c(C)nsc3)=O)CC(=O)NC2)=O)CCCN(C)C(=O)C1 c1(C(N(C2CCN(Cc3ccccc3)CC2)C)=O)nn(C)c2ncccc12 N1(CCCNC(=O)CC2C=CCC2)CCN(C(=O)C2=CSCS2)CC1 Cc1nc(C(N2CCC(NC(=O)Cc3cc[nH]n3)C2C(C)(C)C)=O)cn1C c1(C(=O)NCC2N(C(Cc3nc(C)sc3)=O)CCC2)nc2sccn2c1C c1(OC)cc(F)c(C(=O)NCC(Cc2ccccc2)NC(=O)CO)cc1Br c1(C(C)C)ncsc1C(=O)NCCC(C)N(C(=O)C(C)Oc1ccccc1)C C1(CC)C(C(=O)NC2(C(=O)N(C)CCc3ncon3)CCOCC2)CCN1C C1(NC(CC(C)(C)O)=O)CN(C(=O)Cc2ccnc(O)c2)CC2(CCC2)C1 N1(C(Cc2cnc(C)[nH]2)=O)CC2(C1)CN(C(=O)CN1C(=O)CCC1=O)C2 Cc1cc2c(C(N3CC(CNC(C4CNC(=O)N4)=O)C4(CC4)C3)=O)cccc2o1 c1(C(=O)NC2CCC(NC(CCCCC#N)=O)C2)cc2cc([N+](=O)[O-])ccc2s1 C1(C(N(C2CCCC2)CCNC(C(N2CCCCCC2)C)=O)=O)CCC(C)(C)O1 c1(C(=O)NC(CNC(C(=O)NCCOC)=O)C(C)(C)C)ccn2c1CCC2 C(c1cccnc1)=C(C)C(=O)N(C)CC1CCCN1C(=O)C(c1cnn(C)c1)C C1(C)(NC(c2cc(CC)[nH]n2)=O)CCN(C(=O)CCc2ccc(Cl)s2)CC1 CC1(C(=O)Nc2cnn(CCF)c2)CCN(C(=O)CC(O)C2CCCC2)C1 c1(CC)ccc(C(=O)NCCCCC2(NC(c3oncc3CC)=O)CC2)cn1 c1(C(=O)NC(CCN(C(C(CCOC)C)=O)C)C)cc(OC)ccc1OC(C)C C1(NC(C2CCCC(C)C2)=O)(CO)CCCN(C(=O)COC(F)F)C1 c1(NC(C23C(CN(C(C4(C)CC5CCC4O5)=O)C2)C3)=O)cc2nc[nH]c2cn1 n1(CC(=O)N(C2CCN(c3ncc(C#N)cc3Br)C2)CC)cc2ncccc2n1 c1(C(=O)NCC2(O)CCCN(C(C=C(C)C)=O)C2)ccc(Cl)c(Cl)c1N N1(C(CN(c2ncccn2)C)=O)CC(NC(c2cccnc2O)=O)CC2(CC2)C1 Cc1nc(SCCC(=O)NCCC(O)CNC(=O)CCc2cccnc2)n[nH]1 C(C1CN(C(=O)CC2(CC(C)C)CC2)CC1C(N1CCC1)=O)=CC.C1(C)CC1 N1(C(C2CN(C(C)C)C2)=O)CCC(NC(C2C3CCC2CC3)=O)C(O)C1 C(CCC(C)C)(C(=O)N1CCC(CSC)C1)NC(C(COC)OC)=O N1(C(c2c(C)cccc2F)=O)CCOC2(CCN(C(=O)Cc3nc(=N)[nH][nH]3)C2)C1 c1(OC)cc(CNC2CCCC2C(=O)NC2CCCOC2)cc([N+](=O)[O-])c1 Cc1ccc(C2CCN(C(c3nc(C(C)C)n[nH]3)C(=O)NC3COC3)C2)c(C)c1 C1(C)(NC(C=C(C)C(F)F)=O)CCC(NC(c2cccc(C3CCC3)c2)=O)CC1 N1(C(C(CC)F)=O)CCC2(CCC(NC(=O)CCOc3ccccc3Cl)C2)CC1 C1(C(N2CC(C(C)NC(C(c3ccccc3F)OC)=O)C2)=O)(CF)CCOCC1 CC1CN2CCN1C(C(=O)NC1CCCN(C(C3(N(C)C)CCC3)=O)CC1)C2 C12(NC(c3scc(C(C)=O)c3)=O)CC3CCC(C1C2)N3CCn1nc(C)cc1C C(=O)(C#CC1CCOCC1)N1CC(CC(=O)NC2CCC(CO)C2)C1 c1(C(=O)NC(CCNC(C2C(CCOC)C2)=O)(C)C)c[nH]c2ccc(Cl)cc12 c1(CCC(=O)NCC2CN(C(c3c(C)nns3)=O)C2)ccc(Br)cc1 C(=O)(C(C(F)(F)F)C(F)(F)F)N1C(C)CCN(C(=O)CCc2ncccn2)CC1 C1(C(=O)NCC(CNC(=O)CNS(=O)(=O)N(C)C)OC)CCC(=O)N1C(C)C N1(C(CCNc2ncoc2C2CC2)=O)CCC(C(C)(C)Cc2cn(C)nc2)CC1 c1(C(=O)NCC(C)N(C(c2cccc(C)n2)=O)C)ccc2c(c1)NC(=O)C(C)O2 C1(SCC(=O)NC2C(NC(CCCN(C(=O)OCC)C)=O)CC2)CC(=O)N(C)C1 c1(C(=O)NC2CN(C(c3cnc(CC)[nH]3)=O)CC(O)C2)c(C)sc2ccccc12 C1(CC=C)(NC(=O)CC2(C)CC2)CC2CCC(C1)N2C(c1cc(C(F)F)on1)=O N1(C(C(C)CO)=O)CC(CNC(=O)C=C2CCOCC2)CC1(C)C c1(OC)cccc(F)c1C(=O)NCCCC(C)NC(=O)C=Cc1ncc(C)[nH]1 CN1CCc2cc(C(N3CC4C(C(N5CCC6(CCC6)C5)=O)C4C3)=O)ccc21 c1(C(N2C(COC)(CNC(C3CC(OC)C3)=O)CCC2)=O)cc(N)cc(O)n1 N1(C(c2c(C)n(C)nc2)=O)CCN(C(=O)Cc2nn(C)cc2Cl)C(CC(F)F)C1 C1(C(=O)NCCCN(C(=O)C(C)=CC2CC2)CC)CCCN1c1nccs1 S(=O)(=O)(c1ccc(NC2CCC(F)(F)CC2)c(F)c1)N1CC(C)OC(C)C1 c1(C(N2CCC(C(F)(F)F)C2)C(=O)NCC(C)C)cnc(C(F)(F)F)c(F)c1 Cn1ccnc1CNC(C1CC(O)(CNC(c2cocn2)=O)C1)=O N1(c2nc(C)cc(C)n2)CCN(N2CCc3cc(F)ccc3C2)CC1 c1(CC)oc(C)cc1C(N1CCC(C(=O)Nc2cccc(SC)c2)(CF)C1)=O c1(C(N2CC(C)C(NC(c3ccc4n[nH]cc4c3)=O)C2)=O)nccc2ccn(C)c12 c1(C(=O)NCC2CN(C(C(CCC)(C)O)=O)CC2C)ccc2c[nH]nc2c1 C(=O)(CCS(=O)(=O)c1ccccc1)Nc1ccc(OCC)c(OC)c1 c1(C(=O)NC2CC(C)N(C(=O)C(O)CCS(C)=O)CC2)cccc2c1NCC2 c1(OC)cc(C(=O)NCC2CCN(C(c3cncc(F)c3)=O)C2)ncn1 C(=O)(C1COc2ccccc21)N.C1(N(CC)CC)CCN(C(C2CC2C(=O)OC)=O)C1 N1(C(CCSc2ccc(C)cc2)=O)CCN(C(=O)C(O)C(C)(C)C)CC12CCC2 N1(C(c2coc(C(F)F)n2)=O)CCN(C(c2ccc(F)c(F)c2)=O)C(CF)C1 c1(C(N2CCC(OCCNC(C(C)C)=O)C2)=O)cc(N)ccc1Br N1(C(CC2C(=O)OCC2)=O)CCC(N(C(c2cnn[nH]2)=O)CC2CC2)CC1 N1(C(C2=CCC(NC(c3ccoc3)=O)C2)=O)CCCC(C2CC2)CC1 CCN=c1[nH]cnc2cc(C(=O)NC(C)CCNC(c3cncnc3)=O)ccc12 C#CCCC(C(=O)NCc1ncnn1CC)NC(c1cc(O)cc(F)c1)=O C(=O)(CC1COCc2ccccc21)NCC1CC(OC)CN1C(C1CCC1)=O c1(OC)nc(Cl)c(C(N2C(CNC(C34CCCCC3C4)=O)CC3CC23)=O)s1 N1(C(C(C(C)C)O)=O)CC(CNC(c2cc(C(F)F)ccc2F)=O)C(C)(C)C1 c1(C(=O)NCC2CCCN(C(C3CC(=C)C3)=O)C2)ccc(Cl)c(C)c1 CS(=O)CCC(=O)NCC1CCCCC1NC(=O)C(C1CCOCC1)F c1(COC)cc(C(N2CCC(N(C)C(c3cnn(CCN(C)C)c3)=O)C2)=O)no1 C1(OC)CCCC(CNC(=O)C(CNC(c2sccc2CO)=O)N(C)C)C1 Cc1ccc(CC(=O)NC(C)CCCNC(c2ccc(Cl)nc2O)=O)cc1Cl C1(CNC(C2(C)CNC(=O)C2)=O)CN(C(=O)C#CC2CC2)CC2(CCC2)O1 C1(C(=O)NC2CCN(C(=O)CSc3ccncc3)C2)CC2C=CC1CCC2 C12(NC(=O)COC3CC3)CC1CN(C(=O)CCc1cncs1)C2 C1(NC(CC)=O)CCN(C(=O)CCc2scnc2C)CC12CCC2 C1(NC(CC)=O)C(C)(C)C(NC(c2ccc(-c3nc(CC)cs3)cc2)=O)C1(C)C N1(C(=O)Nc2cnc(C(C)OC)s2)CC(=O)Nc2ccccc21 C1(NC(CCCCOC)=O)CN(C(C2SCCCS2)=O)C2CCCCC12 N1(C(C2(C)CCCN2)=O)CCOCC(C)(C(=O)NCC(c2ccccc2)O)C1 N1(C(CC(=O)OC)=O)C2CCCC1CN(C(c1ccc(N)c(C(F)(F)F)n1)=O)C2 Cc1ncc(C(N2CC(CCNC(C3CC3F)=O)C2)=O)c(C)n1 CC1CC(C)(C(=O)NC2CC(CNC(c3nc(Cl)c(=O)[nH]c3N)=O)C2)CC(C)O1 C1(CC)CCN(C(=O)C=CC(=O)N(C)C)C(C(=O)NC(C)CS(N)(=O)=O)C1 c1(C(=O)NC2CCCC(C(=O)OC)C2)c(C)n(C)c2ccccc12 Cc1cccc2c1CCOC2C(=O)NCC(CNC(=O)C=C1CCCCC1)CO c1(OC)cnc(F)c(-c2cnccc2C(=O)NCCOc2ccc(Cl)cc2)c1 c1(NC(=O)NC2CCC(C(C)(C)C)C2)ccccc1C(F)(F)C(F)(F)F C#CC1(O)CCCN(C(=O)C(c2ccc(Cl)cc2)OC)C1 C(=O)(C(C)(C)CC(F)F)NCCC1CCN(C(c2scc(C)c2C)=O)C1 c1(NC(c2nnnn2C(C)C)(CC)C2CCOC2)cc(F)ccc1C C1(NC(C2(C3N(C(C4OC5CCC4C5)=O)CCC3)CC2)=O)COC2(CCC2)C1 C1(C(=O)NC(CNC(C(C)(C)OC(C)C)=O)C(C)C)CCC(C)C(C)C1 c1(C(N(C(C)CNC(=O)C(c2ccc(Cl)cc2)N(C)C)C)=O)ncnc(O)c1F N1(C(C(C)CC2CCCO2)=O)CC2(C1)CN(C(=O)CC1CC(F)(F)C1)C2 O(NC(=O)C(C1CCOCC1)NC(=O)CC1CCC(=O)C1C)CC(=C)Cl c1(C(=O)NCC2N(C(CCC=C=C)=O)CC(OC)C2)ccc(Br)c(F)c1C N1(C(C=C(C)CNC(c2cc(=O)cc[nH]2)=O)=O)CC(CO)CC(C)(C)C1 CC(C)(CC(=O)NCC1(NC(C23CC2C3)=O)CC(F)(F)C1)c1cccs1 N1(C(c2c(C(C)(C)C)c[nH]c2)=O)CC(CNC(C2CS(=O)(=O)C2)=O)C(O)C1 C1(CC(N2CC(C3CCCO3)C2)=O)(NC(C(CC)SC)=O)CCCCC1 N1(C(c2ccn(CC)c2C)=O)CC2(CNC(C3CC3C(F)F)=O)CCC1CC2 C(=O)(Nn1cnnc1C)C1N(C)CCN(C(C(C(C)C)OC)=O)C1 N1(C(C2(CCOC)CCC2)=O)CC(C2(NC(=O)CCCc3ccc(C)s3)CC2)C1 C1(N(C(CSCCCC)=O)CC2CC2)CCN(C(=O)C(C)C=C=C)CC1 S(=O)(=O)(c1c[nH]c(=NCC(C)C(C)(F)F)cc1C)N(C(CC)CO)C C1(NC(C=CC=CC)=O)CC(CNC(=O)Cc2ccc(O)cc2C)C12CCC2 Cc1ccnnc1C(=O)NC1CN(C(c2cc[n+]([O-])cc2)=O)CC1C(F)F C12(NC(COCCCCC)=O)CC1CN(C(=O)C=CC1CCOCC1)C2 c1(OCC)cc(Cl)ccc1NC(C=CC(=O)NC(C)Cc1cncs1)=O c1(CCC(=O)NC2CCC(N(C)C(c3ccnnc3)=O)C2)ccc(CO)cc1 C1(C(=O)NCCC(C)NC(C2CS(=O)(=O)C2)=O)CCS(=O)(=O)C(C)C1 c1(-c2cn(C3C(NC(C4C(=C)C4(F)F)=O)COC3)nn2)ccc(C)cc1C C1(C(N(CCCNC(=O)CC(C)(O)C2CC2)C)=O)Nc2ccccc2C1(C)C CC(O)C(C)C(=O)N1CC(CCCCNC(=O)C(=Cc2cccnc2)F)C1 CC(CC1CC1)C(=O)NCCC1(NC(=O)CCc2ncno2)CC1.c1ncc[nH]1 CC1=C(C(=O)NC(CNC(C2CCCCN2C(C)C)=O)C2CCC2)CC1 N(S(=O)(=O)N(C)C)CC(N1C(C2CCN(C(CCOCC#C)=O)C2)CCC1)=O C(=O)(C(C)(Cc1ccccc1)C(C)C)NCC(CNC(CN(C1CC1)CC)=O)O C(CCCCC(=O)Nc1ccc(F)cc1OC)N1CCCC(N(C(C)=O)C)C1 c1(C(=O)NCC(C)OC)ccc2c(n1)CN(C(=O)C1=NOC(C)C1)CC2 c1(C(=O)NCC(CNC(CC2C(C)(C)C2)=O)O)cc(Cl)cc(Cl)c1O C1(N(C(c2cnn(C3CC3(F)F)c2)C(=O)NCCC2CC2)C)CCCCC1 C1(NC(CSCCC)=O)CCC(NC(C2(COC)C=CCC2)=O)C1 N1(C(C2(F)C(C)(C)C2(C)C)=O)CCCC(C2CN(C(=O)COC(F)(F)F)C2)C1 N1(C(C2N(C(C)=O)CCC2)=O)CCCC(C)(C(C)NCc2nnnn2C(C)C)C1 CC1CCN(C(=O)C2=COCCC2)CC1CCNC(c1cccc(F)c1F)=O C(C(CC(C)C)NC(c1cnnc(O)c1)=O)NC(Cc1cnc(C)[nH]1)=O C(=O)(C(CCC(N)=O)N(C)C)N1CC(N(C(=O)CC2CCC3CC3C2)C)C1 c1(COC)ccc(C(=O)NCC(C)(F)CNC(c2n[nH]cc2C)=O)o1 S1(=O)(=O)c2ccc(c(Cl)c2)N2CCC(C2)N1.C(C(C)C#N)N(CC)CC c1(OC)cc(C(=O)N(CCC(=O)NCc2cc(C(C)C)[nH]n2)CCCO)ncn1 c1(C(N2CCOCC(NC(CCC(=C)C)=O)C2)=O)cc(O)cc([N+](=O)[O-])c1 CS(=O)(=O)CCC(=O)N1CCC(OCCCNC(C2OCC3CCCC23)=O)CC1 c1(CC(=O)NCCCCCCNC(=O)Cn2nnc(=O)[nH]2)ncn2c1CCC2 c1(NC(CN(CCCNC(c2c[nH]c(=NCC)s2)=O)C)=O)cccc2c1CCC2 C12(NC(=O)CCc3cccnc3Cl)CCC1CN(C(c1cn3ccnc3s1)=O)C2 N1(C(c2ccc(CNC(C(C)CCN(C)C)=O)nc2)=O)CCC(N(C)C)CC1C C(=O)(CCCCCCNC(C1CCS1(=O)=O)=O)NC(C)CCCO C(=O)(C(O)CCN(C)C)NCC(C)NC(=O)CCCNC(N)=O N1(C(=O)NC(C)C(CO)N(C)C)CC(c2cnn(C)c2)C(C)(C)C1 C=CC1(C(N2CCCC2CC(=O)NCC(C)(O)CSCC)=O)CCOCC1 C1(C2CCC2)(C(N2CC(O)(C(C)NC(C3CCC(F)C3)=O)C2)=O)CC1(F)F N1(C(C(C)N(C)C)=O)CCC(NC(c2ccccc2F)=O)C1c1cccs1 Cc1ncc2cc(C(=O)N(C)CCN(C(=O)C(F)(F)c3nccs3)C)ccn12 Cc1ccc(N)c(C)c1C(=O)NCC1CC(NC(c2sc(Br)nc2C)=O)C1 c1(CC2N(C(C3CC3Nc3ncc(Br)cn3)=O)CCC2)ccnc2ccccc12 c1(OC)ccc(F)c(C(=O)NCCC2CCCCN2C(=O)CN(C)C)c1OC C(C(C)(C)CCNC(c1ccco1)=O)NC(C(C)OCCC#C)=O Cc1c(CNC(C23CCC2CN(C(c2cc(Cl)no2)=O)C3)=O)cccc1F Cc1ccc(C(C)NC(=O)NC(C2CCC3(CCC3)O2)C2CC2)c(F)c1 c1(C(=O)N(CCNC(=O)C(O)CF)C2CC2)cncc(F)c1C(F)(F)F c1(NC2CCCN(C(N3CCCC4C(O)CC34)=O)C2)ncnc2ccccc12 N1(C(CC(COC)C)=O)CCC(NC(c2cccc(O)n2)=O)C2(CCC2)C1 c1(OC)cc(CC(N2CC(NC(=O)Cn3ncn(C)c3=O)C3CC23)=O)ccc1C N1(C(C=C(C)C(C)C)=O)CC(O)(CCNC(C2(Cc3cnn[nH]3)CCC2)=O)C1 C1(C(=O)NCC(C)CNC(c2ccnc(C(F)(F)F)c2)=O)CCc2nncn2C1 CCCCC(O)C(=O)NCC(C)(C)NC(=O)CCC(=O)NC1CC1 CCC(C)(CCO)NC(=O)C(CO)NC(=O)CC1CC(F)(F)C1 n1(C(COC)C)nc(-c2ccnn2C)nc1-c1ccnn1Cc1ccncc1 c1(CC(C)C)n[nH]c(=NC(CNC(c2ccc(F)nc2F)=O)C(C)C)s1 N#CC1CN(Cc2ccc(SC(F)(F)F)cc2)CCN1C(c1cc([N+](=O)[O-])cs1)=O c1(NC(C2(C3N(C(C(CCC)N(C)C)=O)CCC3)CC2)=O)c(OC)ncnc1C c1(C(N2CCC(C#N)(NC(c3cncc(Br)c3)=O)C2)=O)c(O)cccc1[N+](=O)[O-] C(=O)(C1=C(NC(C2CCN2Cc2cc(C(F)(F)F)nn2C)=O)CCC1)OCC C12(C(=O)OCCC3(C)CCN3)CCOCC1C2(F)F C1(C(=O)NCCCN2CCN(C(C(C(=C)C)(C)C)=O)CC2)C2CCCCCCC12 c1(C(=O)NC2CN(C(CCc3onc(C)n3)=O)CC2C)c(C)cc[nH]c1=N C1(C(C(=O)OCC2CC2)N(CCCCNC(C)(C)C)C)(C(=O)OC)CCCCC1 Cc1cncc(C(N2CCCC(N(C(=O)C=CC3CCCO3)C)C2)=O)c1 C(=O)(C(C(=O)N1CCC(CN(C(=O)C(F)CC2CCOC2)C)CC1)OC)OC C1(CCC(N2CC(C(C(=O)NCC(C#C)OC)O)C2)=O)CCC(=O)C1 n1(CC)nc(C(=O)NCC(C)(F)CNC(=O)C(C(C)C)n2ccnc2)c(C)n1 N1(C(COC2(C)CCC2)=O)Cc2ccccc2C(NC(=O)Cc2nc[nH]n2)C1 C1(C(=O)NC2C(NC(Cc3c(C)nsc3)=O)COC2)C2CCCCC12 C(C(C(=O)NC1CC(CC(N)=O)C1)NC(c1coc(C(N)=O)c1)=O)OCC CCC(CN=c1cc(N(C)Cc2ccoc2)nc[nH]1)OC Cc1ccc(C(N2C(c3c(Cl)cccc3Cl)CCC2C(=O)O)=O)c(F)c1C N#Cc1cnn(CC(N2CCC(CNC(C3CCC(F)(F)C3)=O)C2)=O)c1N CC1CN(C(C23C(NC(=O)CCC4CCOCC4)C4CC2C3C4)=O)CC2(CC2)C1 C1(CC)CC(C)CN1C(=O)CC1CCC(NC(=O)CC2CCCC2C)CC1 C1(NC(C2(COC)CN(C(c3cnnc(O)c3)=O)C2)=O)CC2CCCC2C1 O=C(C1Cc2ccccc21)NC1CC2(C1)CC(NC(C13COCC1C3(F)F)=O)C2 CC1OCCC1CC(=O)NCC(C1CCCC1)NC(=O)C(=O)NCC(F)(F)F c1(NC(=O)N)ccc2c(cnn2C(F)F)c1.c1(C(C)C)cc(C)n(C)n1 c1(COC)nc(N2CCCC(CNC(=O)CC3CCCCC3O)CC2)cc(C)n1 O=S(=O)(c1cnc(N2CCCC2c2c(F)cccc2Cl)c(Cl)c1)N1CCC12CCCC2 CN1CC(NC(=O)C(Cc2cn[nH]c2)NC(=O)CNC=O)C(C)(C)C1 c1(CCC(N2CCN(C(CN(C(C)=O)C)=O)CC2)=O)c[nH]c2ncccc12 Cc1cc(C(=O)NCC2CC(C)N(C(c3cccn3C)=O)C2)c(C)n1CC1CC1 Cc1cc(CC(=O)NC2CCC(C)N(C(=O)C(=Cc3cnc[nH]3)F)C2)cc(O)c1 c1(C(C)C)ccc(C(=O)N(CCCN(C)C(C2(c3ccccc3)CC2C)=O)C)s1 C(=O)(C(N)CCC1CCCCC1)NC(CC(=O)NC)C C1(N(C(Cn2c(C)nnn2)=O)C)CN(C(C2CC2Br)=O)CC1(C)C Cc1ccc(C(=O)Nc2ccc(NC(c3cccc(C)c3I)=O)cc2F)c(C)c1 N1(C(C2CCN(C(C)=O)CC2)=O)CCN(C(c2csc(C#N)c2)=O)C(CO)C1 C1(C)(C(=O)NCc2occ(C(N)=O)c2)CN(C(=O)CC2CCCSC2)C1 C1(NC(c2cn(CCC)nn2)=O)CC(C(=O)NCCn2cnnc2C)C1(C)C CC1(C)Cc2cc(CNC(=O)NCc3ccccc3I)ccc2O1 c1(C(=O)NC2CCN(C(C3CC(C)(CC)C3)=O)CC2O)nn2c(c1C)OCCC2 n1(Cc2nc(CCSCC)n(-c3ccc(C)c(F)c3)n2)cc(Br)ccc1=O c1(C(N2C(C(C)NC(C(CC#C)C)=O)CCC2)=O)occ2c1CCCC2 c1(C(=O)NCC(CNC(c2cc(Cl)c[nH]2)=O)OC)c(F)cncc1Cl c1(C(=O)NCCOCC(C)C)cccnc1Sc1ccccc1 N(C1CCc2ccc(Cl)cc21)C(CS(=O)(=O)C(C)C)CC(C)C Cc1nnc(CN(C(=O)CN(C2CC(C#N)C2)C(=O)C(F)C2CCOC2)C)o1 c1(CS(=O)(=O)NC2C(C(=O)OC)CCC2)ccc(F)cc1F CC1=CCC(C(N2CC3CC2(CNC(=O)CCC(C)C)C3)=O)CC1 c1(NCN2CCN(C(C3C(=C)C3C(=O)OCC)=O)CC2=O)cccc2nonc12 CC1CN(C(=O)Cn2cc([N+](=O)[O-])cn2)CCCN1C(=O)CCC1CNC(=O)N1 c1(C(=O)NC)cccc(S(=O)(=O)NC2CC(OCc3ccc(F)cc3)C2)c1 C1(CC(N2CC(N(C)C(c3ccc(F)cn3)=O)C2)=O)CCCC(C)(C)O1 CCCC(C)CC(=O)N(CC(C)NC(=O)C(=O)Cc1ccccc1)CC CCC(C)(O)C(=O)NCCN1CCN(C(=O)Cc2ccc(Cl)s2)CC1 CCS(=O)(=O)c1ccccc1C(=O)NC1CC2CCC1N(C(C1(F)CC1)=O)C2 N1(C(CC2C(C)CCC2)=O)CCC2CN(C(c3csnc3Cl)=O)C2C1 C12CC(O)CN1C2=O.C(=O)(CC(=O)OC(C)(C)C)NCC(C)N(C)C c1(C(N2CCC3(NC(CCCCNC(C)=O)=O)C(C2)C3)=O)cc(C#N)ccc1Cl C(CC(C(=O)N(CC(C)O)C)NC(=O)C(C)=C1CC1)OC CCCC(C)CC(=O)NCC(O)CNC(=O)C(F)CC1CCCC1 n1(CC)cc(Cl)c(C(=O)NC(CO)C(C)NC(=O)CCCOC(C)=O)n1 N1(Cc2cc(C(=O)OC)c(Cl)s2)CC(C)c2ccc(OC)cc21 C1(C(=O)O)CN(C(=O)C(Cc2cccc(C(=O)O)c2)c2ccccc2)CC2CC12 N1(C(C2(c3nc(C)[nH]n3)CC2)=O)CCC(n2cc(CC3CCCOC3)nn2)CC1 c1(C(=O)NC2CC(n3cc(-c4n(CC)ncc4)nn3)C2)cc(Cl)c(Cl)c(Cl)c1 C(=O)(C(C)CC(F)(F)F)N1CCN(CC(N2C(C(=O)OC)CC2C)=O)CC1 C12(CS(=O)(=O)C1)C(=O)N2.C12(NC(=O)Nc3ccccc3)COC(CO)(C1)C2 C1(CC(=O)N)SC2=NCCN2C1=O.C1(NC(N)=O)CCC(C(=O)NC2(CF)CC2)CC1 N1(C(CCC)=O)CCC2(CC1)CC2NC(c1ccnc(C2CCNCC2)n1)=O C12(CCCC1)NC(=O)NC2.C(CC(=O)NCC(C)(C)OC)C(C1(CCF)CC1)=O c1(C(=O)NCCN(C(=O)CC2(C#N)CC2)CC)cccc(C2CC2(F)F)c1 C(=O)(C(Cc1cccnn1)OC(=O)NC(C)(C)C)C(N1CCC(OC)C1)=O.C(C)(C)(C)O N1(C(C=CC)=O)CCN(C(=O)C(C)N(C)C)CC1CS(C)(=O)=O O=C(C1=NOCC1)NC1CCN(C(=O)COc2ccc(Cl)nc2)C1 c1(NC(C)CCNC(c2ncccc2Br)=O)cc(C(C)(C)C)ncn1 N1(C(C2C(C)OCC2)=O)CC=C(CC(=O)N2CC3CC(C2)CN(C)C3)CC1 c1(COCC(=O)NCC(C2CCCC2)NC(C2CC(CC)C2)=O)nnc(S)n1C CN1CCC2CCC(C1)N2C(c1coc(CNC(=O)CNC(=O)CN(C)C)n1)=O c1(C(=O)NC2CCCN(C(C(C)(O)C3CC3)=O)C2)c(F)cc(N)cc1F C1(NC(CC(CC)CC)=O)CCN(C(c2cnc(C)c(N)c2)=O)CCC1CO c1(CC(=O)N(C(C)CNC(=O)CCc2cnc(C)o2)CC)ccc(F)cc1F N1(C(c2c(C(C)C)con2)=O)CC2C(NC(=O)C(C)CC3CC3)CS(=O)(=O)C2C1 N1(C(c2c(C)n(-c3ccccc3Cl)nc2)=O)CCNC(=O)CCCC1 N1(C(C2(O)CCC2)=O)CCCC(NC(C2CCCC2F)=O)C(F)C1 c1(C(N2CCN(C(C)=O)C(C)C2)C(=O)NCCOCC)ccnc(Cl)c1F C#CCCCCCCC(=O)N1CCC2CC12C(=O)NC1CCC(C)(C)C1 C(C)(C)(CCCC(=O)NCC1(O)CC=CC1)NC(CC=CC=C)=O C1(CNC(C(CC)n2cncn2)=O)CN(C(=O)CC23COCC(C2)C3)CC1NC Cc1cc(C(=O)NCC2CCC2NC(C2COCCO2)=O)c(N)c(C)c1 CSC=CC(=O)NCCCNC(=O)C=CC=C(Cl)Cl Clc1ccc2c(c1)C(NCc1cn(C3CCCC3)nn1)CO2 CN1CCC(C)(C(=O)NCc2ccc(C(N3CCC(CC(F)F)C3)=O)o2)CC1 N1(CCC)CCN(C(=O)C(c2ccnn2C)NC(=O)CN2CCCCC2=O)CC1 Cc1ccc2cc(C(=O)Nc3cc(F)c4cn[nH]c4c3)ccc2c1 CCCCCC(C)(C)C(=O)NCc1cc(C)c(C(=O)NCCCn2nccn2)o1 C1(C(=O)NC23CCN(CC2)C3)(CNC(=O)CC2(C3CC3)CC2)CC12CCC2 C(=O)(CCC(C)(C)C)N1CC(C)C(C(=O)N(CC(=O)NC2CC2)C)C1 N1(C(c2cc(C(F)F)no2)=O)CCC2CC12C(=O)NCc1ccncc1Cl Cc1ccc(NC(=O)C(=O)Nc2ccc(S(C)=O)cc2)c(Cl)c1C c1(C(C2CC=CCC2)(C)NCC2CC3(CC3)C2)nnnn1-c1ccccc1 c1(C(=O)NCC2OCCN(c3nccc(CC#N)n3)C2)ccc2cnsc2c1 CCC(C)(C)C(O)C(=O)NCC(=O)NCC1CCN(C2CC2)C1 N1(C(C(CC)F)=O)CCN(CC2CCCN(C(=O)COC)C2)CC1 CC(C)CC(C)(C)C(c1nnnn1CC(F)F)NCc1ccccc1F N1(C(CCN(C(Cc2c(C)occ2)=O)C2CC2)=O)CCC(O)C(C)C1 Clc1ccc2c(c1)CCC21CCN(Cn2cc(CCOC3CCCCC3)nn2)C1 CCCC(C(=O)N1CCC(C)(NC(=O)CC2C(=O)ON=C2C)CC1)C(C)C C1(C(=O)NC(CNC(C(C)NC(=O)OC)=O)CO)CCC(NC(C)=O)CC1 N1(C(c2cc(NC3CC3)no2)=O)CCC(CNC(C2(F)CCCC2)=O)C12CC2 C1(CCOC)(NC(c2ncn(CC)c2)=O)CCN(C(=O)C(n2nccc2C)C)C1 CCCCC(CNC(c1ccn(-c2ccncc2)n1)=O)NC(=O)C(C(C)C)SC c1(NC(C2N(C(c3ccn(C)c3)=O)CC=C2)=O)cc(F)c(Cl)nc1Cl c1(C(=O)NCCCCCNC(CCc2ncc(C)[nH]2)=O)ccccc1OCCF Cn1ncc2c(-n3cc(C4CCCN4CC(=O)NCC4CC4)nn3)nc(Cl)nc12 CCC(C)C(O)C(C)C(=O)N1CC(C)(C(=O)NCC2(C3CC3)CC2)CC1(C)C CC(C)S(=O)(=O)C(C)C(=O)NCC(C)(C1CC1)NC(=O)CCn1cccn1 c1(C(N2CCC(N(CCC)C(C3CC=CCO3)=O)C2)=O)cc2c(s1)CCC2=O C1(CN=C(NC(c2cccs2)C)NCc2cccs2)CCc2cnn(C)c2C1 c1(C(=O)NC(C(=O)NC(c2ncc[nH]2)CC)Cn2cncn2)nc(O)sc1C N1(C(C2CCN(S(CCC)(=O)=O)CC2)=O)CCC(NC(=O)CS(=O)(=O)NC)C1(C)C c1(C(=O)NCC(CC)NC(C2CC2C)=O)nn(C)nc1Br Cc1cc(C(=O)NCC2CCCN2C(=O)Cc2cccc(Br)c2)c(C)cn1 Cc1cc(=NCc2cc(Cl)ccc2F)[nH]cc1S(=O)(=O)NCC(Cl)Cl C(=O)(CC1=CCOCC1)NCc1c(C(=O)NCc2occ(C)c2)c[nH]n1 N1(C(C(C)OCCOCC)=O)CCCN2CCCC2C1.c12cc(on1)C(=O)NC2 CC(C)CC(C)CC(=O)N1CCCCC1C1(NC(=O)C(C)(C)N2CCCC2)CC1 c1(C(=O)NC(CN(C(c2ccc(Br)o2)=O)CC)C)cc2c(cc1N)OCO2 N1(C(C2(COC)CC2(F)F)=O)CCC12CCCOC2 c1(C(=O)NCC2CC(NC(C3(CC#C)CCCOC3)=O)C2)cnc(O)cc1C C1(C(=O)NC(C)C(C)NC(=O)C(c2cccc(C(F)(F)F)c2)O)C2CC3C(C2)C13 C1(CNC(c2sc(CCC)c(CC)c2)=O)CCN(C(=O)C(C#N)CC)C12CC2 Cc1ccc(O)cc1NC(=O)CNC(=O)C(C)(C)N1CCCC1 C1(NC(C2ON=C(CC)C2)=O)CC(NC(c2[nH]cnc2C)=O)C12CCC2 C12(CNC(C3(O)CC(C)(C)C3)=O)CCCC1CN(C(C1CC3CC1CC3O)=O)C2 CCC(CC)(CCNC(c1cccc(C(C)(F)F)n1)=O)NC(C1(N(C)C)CC1)=O Cc1ccc(Br)c(S(=O)(=O)NCC2CN(C(C3CCN(C4CCCC4)C3)=O)C2)c1 N1(C(C(N(C(CCOCCOC)=O)C)C2CC2)=O)CC2CCC(C1)C2C#N CC1CC(C(=O)NCc2cccc(Cl)c2)CN(C(=O)C(c2ccc(O)cc2)C)C1 C=CCC(CC(=O)Nc1cc(CC)ccc1C)NC(=O)C(COC)OC C(=O)(CN=c1ccc(Cl)n[nH]1)N1CC2C(NC(CC(C)N(C)C)=O)(CC2)C1 c1(C(=O)NC(CCNC(CC2CC(=C)C2)=O)C)cc(C(F)(F)F)[nH]c1C c1(C(=O)OC)ccc2c(c1)CCCC2NC(=O)NC1CCc2nc[nH]c2C1 CCC(C)CC(=O)C(=O)N1CCC(CNC(C2CCCS(=O)(=O)C2)=O)C(O)C1 c1(C(=O)OC)cc(C(F)(F)F)nn1C.c1(C(N(C(=O)CSN)CCN)=O)ccncc1 c1(C(=O)NCCCN(C(C2(C(C)C)C(C(=O)OC)C2)=O)C)c(Cl)cncc1Cl CC(O)CCCCCC(=O)NCC1CC2(CO1)CN(C(c1ncccc1N)=O)C2 C12(CNC(C(C)OCC)=O)CC(CO1)N(C(c1ccccc1CC(C)(C)C)=O)C2 C1(C(=O)NCCCCC=C)(NC(=O)CSC)CCC(C)(C)C1 c1(C(=O)NCC2CC(NC(C(C(C)O)(F)F)=O)C2)cc2cc([N+](=O)[O-])ccc2o1 C(=O)(C(C)(CC#C)NC(=O)C=Cc1ccco1)NCCCCCC#C O=C(CCC(CF)CF)NC1(C(=O)NCC2CC23CCOC3)CC(O)C1 C1(C(=O)OC(C)(C)C)CC(C(=O)O)CCO1.C12CCN(CC1)Cc1cc2no1 FC(F)CCCCCN1CCCC1c1nocc1Br CC12CN(C(=O)C=CCF)CC1(C)CN(C(c1ccc3oc(O)nc3n1)=O)C2 CS(=O)(=O)c1ccsc1C(=O)NCC1CCCCN(C(=O)C(F)F)C1 C(=O)(CC(C)CC(=O)N1CCC(C(N2CCc3n[nH]cc3C2)=O)O1)OC c1(C(=O)NCC(C)(O)CNC(C2CC(C)(O)C2)=O)ccc2c(c1)NC(=O)CCS2 O=C1COc2ccc(C(N3CC4CC3CN4c3cc4nncn4cn3)=O)cc2N1 C(=O)(CCCC(=O)NC(C)(CO)C(=O)NCCC1CC=CC1)OC c1(CNC(CN(CC)CC)=O)ccc(C(=O)N)s1.c1(CO)cc(C(N)=O)co1 c1(C(N)=O)ccc(C(=O)NCC2(CN=c3[nH]nco3)CCC2)cc1 c1(C(=O)NC2C(NC(C3N(CCC)CCC3)=O)COC2)ccccc1SC C1(C#N)(C(=O)NCCN(C(c2n(CCC)nc(C)c2)=O)CC)CC12CCCC2 Cc1cc(Br)ccc1-n1nc(COCC(C)C)nc1C12CCC(C)(C1)OC2 Cc1cccc(C(C)NC(C2(CCNC(c3ccnn3CCF)=O)CC2)=O)n1 c1(OC)cccc(C(=O)NCC2CC2NC(=O)CCc2cnco2)c1O C1(O)(CCNC(=O)CC2CCOC2)CCCN(C(C2CCC3(CC2)CC3)=O)C1 CC1CC2(CC(C(=O)NC3(C(=O)NCCC(O)C(C)C)CCOCC3)C2)C1 CC1CC=C(C(=O)NC2CC=CCC2C(=O)NCCS(C)(=N)=O)CC1 c1(OC)cccc(Cl)c1CC(=O)NC1CCC1NC(C1(C)CCC(OC)CC1)=O c1(CCC)ccc(C(=O)NCC2CC(CNC(=O)C=CCO)CO2)[nH]1 C(=O)(C#CC1CCOCC1)N1CC2=C(CN(C(C3C(C)NC(=O)CC3)=O)C2)C1 C1(CNC(COc2cccc(OC)c2)=O)C(C)CCCN1C(=O)CCC(C)OC C(=O)(CC(C)C(=O)N(CC(C)CNC(=O)C(C)(C)c1csc(C)c1)C)OCC CC1CCC(NC(c2ccnc(F)c2N)=O)CN1C(c1ccon1)=O C1(NC(CC)=O)CCN(C(c2nc(-c3ccccc3C)oc2C)=O)C1C N1(C(C2(O)CCN(C(=O)CCC3CCC3)CCC2F)=O)CCc2c(O)n[nH]c2C1 C12(NC(C=Cc3c(C)ccs3)=O)CCN(C(=O)C(=Cc3cccnc3)F)CC1C2 c1(CNc2cc(OC)ncn2)ncc(C(=O)NC2CC3(C2)CN(C)C3)c(C)n1 Nc1ccc(F)c(F)c1C(N1CCN(C(C2CCCS2)=O)C(C2CC2)C1)=O N1(C(c2c(C)n(C)cn2)=O)CCC2(CC2)CC1C(=O)N(CCC(C)(C)C)C N1(CC(=O)N(CC=C)CC=C)CCC2(CCC(NC(c3csc(C)c3)=O)CC2)CC1 N1(C(c2c(CCC)n[nH]c2)=O)CCN(C(C2CCCC(C)(C)C2)=O)C(CC)C1 CN1CCC(C(=O)Nc2cccc(NC=O)c2)(NC(C2CC2(C)C)=O)C1 C(CC(C(C)C)NC(C1C=CCC1)=O)NC(C(CC)N(CC)CC)=O CON(CCC(=O)c1ccncc1N)C(=O)C1CN(S(=O)(=O)C(C)C)C1 N1(C(C(C)O)=O)CC2CCC1C(CNC(c1csc(C(F)(F)F)c1)=O)C2 C12(Cn3c(-c4[nH]nc(-c5ccco5)n4)ncc3)C3C4C5C3C1C5C24.CCC(C)NC=O C1(NC(C)=O)CN(c2nccc(-c3ccccc3F)n2)CC1(F)F C1(NC(C2(C(C)NC(c3cc4ccccn4n3)=O)CC2)=O)CN(C)CCN(C)C1 C(CC(C(=O)NCc1cccnn1)NC(=O)C=CC1CCCN1C)OC N1(C(C2CC(=C)C2)=O)CC(NC(=O)Cc2cc(F)ccc2Br)CC(O)C1 c1(C(N2CCC(O)(CNC(CN(C)C)=O)C2)=O)n[nH]c2c1COC2 C1(C(N2CCC(C(C)(C)C)(CNC(CCC=C=C)=O)C2)=O)CCC2(CC1)CC2 Cc1ncnc(C(=O)NCC(C2CCN(C(C3C(C)(C)C3(F)F)=O)CC2)O)c1C CC(C)(CC(=O)N1CCCC(C)(NC(=O)COCCO)C1)C(F)F N1(C(CC(CNC(Cc2cn(CC)nc2)=O)C)=O)CCC2CCN(C)CC12 CCC(C)CC(C(=O)NC1COCC1OC)NC(=O)C1=C(Cl)CCC1 N1(C(c2ccc(CC(F)(F)F)cc2)=O)CCC12CN(Cc1c(Cl)cccc1I)C2 CCC(CC(=O)N1CCN(C(=O)CCc2ccc(C)o2)CC12CC2)C(C)(C)C C1(NC(CSCC=C)=O)CCS(=O)(=O)C12CN(C(C1COC(=O)N1)=O)C2 Cc1ncc2ccccc2c1C(=O)NCC1CC(C)N(C(=O)CCC(C)(C)C)C1 c1(CCCC(=O)NCCCNC(C(C)C(F)F)=O)nc2ccccc2[nH]1 N1(C(CN(S(C)(=O)=O)C(C)C)=O)CC(NC(=O)CN(C)C)C(S(C)(=O)=O)C1 c1(C(C)NC(C2CCC(C)S2)=O)ccncc1NC(=O)OC(C)(C)C C(CC(C)C)(C(=O)NCC(F)CNC(c1cccc(F)c1Cl)=O)NC(C)=O C(C)(C)(C(C)NC(c1cn(C2CCCC2)nn1)=O)NC(C(C)O)=O c1ccc(OCC(=O)NC(C2CC(C(=O)NC3CN(C(C)C)C3)C2)C)cc1.CC c1(C(C)=O)ccc(C(=O)NC(C)CNC(=O)C(C2CCC(=O)N2)C)o1 C1(NC2(c3n(CC(=C)C)nnn3)COC2)CC(C(=O)OC)C12CCC2 C1(CC(C)C)CN(C(=O)C#CCc2cn(CCC(=O)OC(=N)O)nn2)CCO1 c1(OC)ccc(OC)c(C(=O)NC2CCC(CNC(=O)Cc3csc(C)c3)C2)c1 c1(C(=O)NC2CCCC(CC(=O)NCc3ccnc(F)c3)C2)c(O)cccc1F C(CN=c1[nH]cnc2c(S(C)(=O)=O)cccc12)C1CCC(NC(C(CC)C)=O)C1 c1(N2C(C)C(NC(c3cc(Cl)c[nH]3)=O)CCC2)nc2c(cc1C#N)C(=O)CCC2 Cc1cc(C2C(CN3CCC(NC(=O)Cc4ccccc4)CC3)C2)cc(Br)c1 N1(C(CC2CCC(NC(c3cccc(C#N)c3)=O)C2)=O)CCC2(CC1)CSC2 N(C1CCCn2ccnc21)C(c1c(CNC(C(CO)OC)=O)nccc1)=O c1(C(N2CC(NC(C3CC(O)C3)=O)C(C(F)F)C2)=O)c(F)cc(F)cc1Cl c1(CNC(c2c(OC)csc2)=O)ccnc(Br)c1 C1(CNC(c2ccc[nH]2)=O)C2CN(C(c3ccc(Br)o3)=O)CC12 C(=O)(CC(C)(C)CC(=O)OC)NC(CN(C(c1ccc(C#C)cc1F)=O)C)C CC(F)(F)CCC(=O)NC1CS(=O)(=O)CC1NC(=O)COC1CCCOC1 c1(OCC)ncc(C(=O)NCC2CC(NC(C3CC3[N+](=O)[O-])=O)C2)cn1 Cc1cc(C(=O)NCC(C)NC(C2CC2c2ccccc2)=O)nnc1C C(CC(C)(C)CC(=O)N1CCC(C)(NC(=O)C(C)(C)C(F)(F)F)C1)OC CC1(C(N2CCC(O)(C(C)CNC(=O)COCC3CCCC3)C2)=O)CC2(CC2)C1 CC(C)C(C(=O)Nc1cncc(Cl)c1)N(S(C)(=O)=O)C1CC1.C12(F)CC(C1)CNC2=O CCCCC(O)C(=O)NC1CC2C1CCN2C(c1cnc(COC)s1)=O C1(NC(=O)CC2CC(F)(F)C2)CC2CC(C1)N(C(C13CCOC1CCOC3)=O)C2 CN1CCN(c2ccccn2)CC1.C12CN(C1)C(=O)NC1CC1C(=O)NC2 Cc1c(C(N2CCCC(C)(CNC(=O)C(=O)NCC3CC3)C2)=O)nn(C)c1N N1(C(CCCC(=O)OC)=O)CCCC1C1CCCN1C(=O)Cn1ccnc1C c1(C(=O)NCC(CC)NC(c2cnc(C(F)F)s2)=O)coc(Cl)c1 Cc1noc(Cl)c1CCC(=O)NC(C1CN(C(c2cnn(C(F)F)c2)=O)C1)C C(C1=CCCN(C(=O)CC2CCCC3CC23)C1)C(=O)C1CC1.C1(OC)CC(C(=O)O)C1 c1(NC(C)=O)ccc(-c2nc(C(=O)NC(c3ccccc3)C(=O)O)cs2)cc1 Cn1cc(Cl)cc1C(=O)NCCn1ccc(C(N2CCN(CCF)CC2)=O)c1 c1(-c2cccc(C#C)c2)ccc2[nH]cc(C(=O)Nc3ccc(OC)c(F)c3)c2c1 Cc1cc(C(=O)NC(C)CC2CN(C(=O)CCN3CCC(F)C3)C2)cn(C)c1=O c1(C(=O)NCCC(C(=O)N(CCCCC)CCO)O)ccc2cc[nH]c2c1 CC1CN2CCCC2CN1C(C12CC(NC(c3cnc(N(C)C)nc3)=O)(C1)C2)=O C1(NC(C2C(c3ccc(C)o3)C2)=O)CCCC(NC(c2cnn(C)n2)=O)C1 c1(C(=O)NC2C(NC(=O)Cc3cscn3)CCCC2)cc2cccnn2c1 CCC1C(=O)Nc2ccc(C(=O)NCC(C3CCC3)NC(=O)CC#N)cc21 N1(C(C(C)C(C)(C)C)=O)CC(C)(C)OCC1CNC(=O)CCC1CCCCCC1 C1(C(=O)NC2CN(C(=O)C(C)(C)COC(C)C)CC2C)(OC)CCC(F)(F)CC1 Cc1cnn(C)c1C(=O)NCC1CCCC(CNC(C2CC2c2nc[nH]n2)=O)C1 C1(CCNC(C(C2CCOC2)OCC)=O)CCN(C(=O)Cc2ncc(C)s2)CC1 N1(C(c2cc(CC)no2)=O)CC(CNC(=O)C=NOC)C(F)(F)C1 CC1CC(NC(=O)CC2CSCCO2)CN(C(c2nn(C)cc2Cl)=O)C1 c1(C(=O)NC2CCC2)nc2ccccn2c1F.CC1(CC(=O)NC)CC1F Cc1nc(O)[nH]c1C(=O)N(CCNC(c1ccc(C(C)C)cn1)=O)C(C)C c1(C(=O)NC2C3CN(C(=O)CCC4CCOC4)CC23)cccnc1N1CCCC1 C1(NC(C2CC(C)(CNC(CNC(C(C)N(C)C)=O)=O)C2)=O)CC2CC(=O)C1O2 CC1CCN(C(=O)Cc2ccsc2)C1CNC(c1cc(Br)n(C)n1)=O c1(C(C)NCc2nc(C(C)N(C)C)[nH]n2)cccc(C#N)c1 CC1CN(c2ccc(C(F)(F)F)cn2)CCN1C(=O)CN1CCOC1=O C=CC1OCCC1C(=O)NCc1occc1C(=O)NC(CCC)CCO C(C(C)(C)CC(=O)NC1CCC(C)(CNC(=O)C(C2CCCCCC2)C)C1)OC C12(NC(=O)Cc3cccc(C(F)F)c3)CCN(C(c3cocn3)=O)CC1C2 c1(C(=O)NC(C2CCCN(C(c3onc(C)n3)=O)C2)C)ccnc(O)c1F c1(C(N2C(CNC(C(C)OCCN(C)C)=O)CCC2)=O)cc(N)cc(O)n1 c1(CC)cc(C(=O)NC2CCC(C)N(C(=O)CC(=O)NC3CC3)C2)ccc1O CCC(C)(O)C(=O)N1CCC(NC(c2ccnc(N3CCOCC3)n2)=O)C1 C1(C2CCN(C(c3cn(C)[nH]c3=N)=O)CC2)(NC(CC(CC)O)=O)CC1 C1(C#N)(C(=O)NCC(CNC(c2n(CC(C)C)ncc2)=O)O)CC2(CC2)C1 C1(SC(C)(C)C(=O)O)CCN(C(=O)NCc2cncc(Cl)c2)C1c1ccccc1 c1(C(C)C(=O)NCC2CC3CC2CN3C(=O)CSC(F)F)ccc2c(c1)OCO2 CC(C)C(F)(F)CC(=O)NCC1CN(C(=O)CCCCN(C)C(N)=O)C1 c1(-c2n(C(C)C)ccn2)ccc(F)cc1-c1cccc(C2(C(F)F)CC2)c1F C(=O)(C1=C(C)S(=O)(=O)CC1)NCC1(C)CCC(NC(C=CCC)=O)CC1 N1(C(Cc2ccn(CC)n2)=O)CC2CCN(C(c3ccc(C)cc3C)=O)CC2C1 c1(C(N2CCN(C(=O)COCC3CC3)CC2CC2CC2)=O)ccc2occc2c1 C1(CC=C)(NC(C2CCCCN2S(C)(=O)=O)=O)CCN(C(=O)C(F)=CC2CC2)C1 C1(C)(CC)CC(NC(C23CC(F)(C2)C3)=O)CN1C(c1ccc(C#N)cc1)=O c1(Sc2ccccc2)ccncc1S.CC(C)C(=O)Cc1csc(CN)n1 Cc1cc(Br)c(NC(C2CN(S(=O)(=O)CCCl)CCC2O)=O)cc1[N+](=O)[O-] c1(C(N2CCC(CC(N3CCCC(C(=O)OC)C3)=O)CC2)=O)c(I)ccnc1Cl CC1(C)CCCCC(C(=O)NC2CCCN(C(c3csc4nnsc34)=O)CC2)C1 C(CCC(F)(F)F)N(C(C1(NC(c2c(CC)ocn2)=O)CCCC1C)=O)C Cc1ccc(CC(=O)NCCCN(C(C2CCN(C)C2)=O)C2CC2)c(Cl)c1 Cc1ccc(F)c2oc(N(CC(O)COc3cccc(C(F)(F)F)c3)C)cc12 CC(C)CCC(=O)N(C1(CCC(=O)NCCC2CC2C2CC2)CCC1)C1CC1 C1(C(=O)NCCC2CCN(c3nc(CC)cc(CC)n3)C2)CC12CCOC(C)C2 CC1CN(C(C2(CF)CCN(C(C34CCCC3C4(F)F)=O)C2)=O)C=CCCC1 C1(OC)CC2CC(N)CC12.C1(=O)CC(C)C(=O)NC(C)(C)C=CC1=O.C1(N)CC1 n1(-c2c(C#N)ccc(Br)c2)ccc(=NC(=O)CC(Cl)(Cl)Cl)[nH]1.N1CCCCS1(=O)=O C1(C(=O)NCCCC(C)NC(=O)CCOc2ccccc2)CCC(N(C)C)CC1 CCC(CC(=O)NCCc1ccsc1)N(C(=O)CC1CCCC2CC12)C N1(C(=O)NC)CC(C)OC2(CCN(CC(=O)NCc3ccccc3)C2)C1 C=C(F)C1(CC(=O)NC2COCC2CSc2cc(C(=O)NC3CC3)no2)CCC1 C1(C(=O)NCC2N(C(c3c(C)nc(C(C)C)o3)=O)CC(F)C2)CCCC(F)(F)C1 N1(C(C(C=C)OC)=O)CCOCC(NC(C2(CO)CCN(C)C2)=O)C1 c1(C(=O)NCC2N(C(CC(CC)OC)=O)C3C(C2)C3)cc2c(Cl)cncc2s1 C12C(CC1O)CN(C)C(=O)C2.c1(C(=O)NC(=O)OC(C)(C)C)ncc(Cl)s1 c1(C(=O)OCc2cnc3sccn23)ncn2cccnc12 CS(=O)(=O)c1sccc1C(=O)NCC1(NC(=O)CC2CCOC2=O)CCC1 Nc1c(Cl)cnc(C(=O)NCCCCc2nccs2)c1Cl N1(Cc2ccc(OCC)cc2)CCC(O)C(C(=O)Nc2cnn(C)c2)C1 c1(C(N2CCC(NC(c3c(C)nc(CO)s3)=O)C(F)C2)=O)cnc2cc[nH]c2c1 N1(C(CCN(C(=O)CCc2ccccn2)CC)=O)CCCC2NC(=O)CC12 CCCCCCCCCCCC(=O)NC1CC1CNC(C1CC2CC2C1)=O c1(SCCn2cc(CCCNC(C3CC3(F)F)=O)nn2)cc(Cl)sc1Cl Cc1ccc(C=CC(=O)NCC(C)(CO)NC(c2cscn2)=O)c(C)c1 CC(C)(CS(N)(=O)=O)C(=O)NC1CCCN(C(c2ccc(C(F)F)s2)=O)CC1 CCCC(CNC(c1ccnc(C)c1)=O)C(=O)N(CCN=[N+]=[N-])CC c12ccc(cc1F)C(=O)N1CC(CC1(C)C)CNC2.c1(CC)ccc(CC)o1 CC1CN(C(=O)Cn2cc(C3CCC3)nn2)CC1NC(=O)Cc1sccc1Cl C(=O)(C1=CCCCO1)NCc1occ(C(=O)NC2CC(CCC)C2)n1 Cc1ncnc(O)c1C(N1CCCN(C(C2COC(C)C2)c2ccccc2)CC1)=O C(=O)(CCC(N)=O)NCC1CC(NC(C2CCN(C)C2)=O)C1 C1(NC(C(CNC(CSC)=O)CC2CC2)=O)CC2CC3C(C2)C13 CCCC(C#N)C(=O)NC(C)(CO)C(=O)N(C(C(N)=O)C1CC1)C N1(C(C2(C)N(C(c3ncc(C)nc3)=O)CCC2)=O)Cc2cccc([N+](=O)[O-])c2C1 C1(C(CNC(=O)CCSc2ccccc2)C2CC2)COCCN1C(c1cnc[nH]1)=O C12(C(N3CC(CC)OCCC3)=O)CCC(CC1)N(C(=O)C(C)(O)C1CC1)C2 C(CN=c1[nH]c(=NCCCN2CCCCCC2)[nH]c2c1SCC2)(C(C)(C)C)OC Cc1c(CCNC(C2CCN(C(c3ccoc3)=O)C2C)=O)cnn1C N1(C(C(c2ccoc2)OC)=O)CCOCC1CC(=O)NCCc1ccc(F)nc1 C#CCC(C)(C)C(=O)N1CC(CCNC(=O)CC2(CC(=O)OC)CC2)C(C)C1 N1(C(c2c(C)cnn2C)C(=O)NCCC)CCC2CCCC12C(=O)OC C1(NC(CCSC)=O)CCCC(CC(=O)N(CCO)Cc2cccc(F)c2)C1.NCO c1(CC(=O)NC(C2CN(Cc3ccc(OC)cc3)C2)C)ccc(F)cc1F c1(OC(C)C)cncc(C(=O)NC2CCCCC2N(C(=O)C(C)CO)C)c1 c1(CC)nn(C)cc1C(=O)NC1(CN(C(=O)Cc2ccc(SC)nc2)C)CC1.C1(SC)CC1 C=CCCC(F)(F)C(=O)NC(C)CCCC(=O)NC1C(=O)OCC1CO C1(CNC(C(C)NC(=O)NC)=O)CN(C)CCN1C(C1CC1C(C)O)=O C12(NC(CCCC=C)=O)CCCCCC1N(C(c1nnc(S)n1C)=O)CC2 C1(NCc2nn(C)c(=O)o2)CN(Cc2ccccc2)CCC12CCC2 C1(NC(c2ccc(C)s2)=O)CCC(C)N(Cc2snnc2C)C1 N1(C(C2CCCOC2)=O)CCC(C)N(C(Cc2c(OC)ccc(F)c2)=O)CC1 N1(C(C23OC(C)C(C2)C3)=O)CCC2(C1)CN(c1ccc([N+](=O)[O-])cc1Br)CCO2 C1(NC(CN(C)C)=O)CN(C(C2CCN(c3ccncc3)C2)=O)CC12CCC2 N1(C(c2ccc(OC)c(F)c2)=O)CC2(CC1CNC(=O)CCC(N)=O)CC2(F)F C#Cc1ccc(CC(=O)NOC(CC(C)C)C(=O)NC(C)CCSC)cc1 c1(C(=O)NCC2C(C)CCN2C(c2ccccc2Cl)=O)cc2ccnn2cn1 c1(NC(=O)CCC2CCCN2C(c2sccc2I)=O)cc(Br)cc(Cl)c1O C#Cc1cnn(C)c1CNC(=O)NC(c1ccc(F)cc1F)C1(CC)CCC1 C1(CC(=O)NC(c2ncn(C)n2)C)C2CN(C(c3cc(Cl)cn3C)=O)CC12 CCC(C)C(C(=O)NC)N.C1(C(C(=O)OC(C)(C)C)=O)CCN(C(n2cnnn2)=O)C1 C1(NC(c2cn(CC(C)C)nc2)=O)CC2CC(NC(=O)Cn3ccnn3)C2C1 N12CCC(CC1)n1cc(nn1)C2=O.c1(OC)cncc(Br)c1.C1CC1 CON1CCC(C(=O)NC2CCC(N(C(=O)C=CC(C)(C)C)C)CC2)CC1 N(C1CCCc2c1[nH]c1ccc(Cl)cc21)S(Cc1ccc(C(=O)OC)cc1)(=O)=O N1(C(c2cnn(C(C)C)c2N)=O)CCCN(C(=O)Cn2cc(CO)nn2)C(C)C1 N1(C(c2c(C)occ2)=O)CC(C(=O)NCC(C)(O)C(C)C)CCC1C CS(=O)(=O)C1CCCC1C(=O)NCC1CN(C(=O)CCc2ccc(F)cc2)C1 c1(C(=O)NCC(CC)NC(c2c(C(F)(F)F)n[nH]c2C)=O)cncc(SC)c1 c1(OC)cc(CNC2CCCC(C(=O)Nc3cc(C)cnc3O)C2)cc(O)c1 C(C1CCCCC1)=CONC(Cn1cc(CNC(C(CSC)O)=O)nn1)=O Cc1cc(CN(C)CCOCCNC(=O)CN2CC(C)(C)C2)ccc1F C1(C(N(C2CCC2)C(=O)OC(C(C)C)C2CC2)=O)CCCC2CCCCC12 CCCC(C#N)C(=O)NC1(CNC(c2ccc(-c3sccc3C)s2)=O)CC1 C12(C(N3CCCC(F)(CNC(c4cscn4)=O)C3)=O)CCC(C(F)F)(CC1)CC2 c1(NS(Cn2ncc(COC)c2)(=O)=O)cnn(-c2cccc(C3CC3)c2)c1C C(C)(CC(=O)NC(COC(C)=O)C1CC1)N(C(C(C)SCCCC)=O)C c1(NC(c2n(CCSC)nnn2)c2nccs2)cccc(S(=O)(=O)C(F)(F)F)c1 c1(C(N2C(C)CCN(C(C3CCCC3(C)C)=O)CC2)=O)cnn2c(N)ccnc12 c1(CN=c2scc(CC(=O)NC(C(=O)OC)CCO)[nH]2)ccc(Cl)c(Cl)c1Cl N1(C(c2nc(C(F)(F)F)ccc2Br)=O)CC2CCCC2(C(=O)OCCO)C1 C=CCC(C(=O)N(C)CC1CN(c2ccccc2)C(=O)O1)Nc1ccco1 CC(C)C(C(=O)N(C)CC1CCCN(C)C1)NC(c1ccncc1Cl)=O c1(NC(C=CC(C)NC(C2(SC)CC2)=O)=O)cc(C#N)ccc1O c1(C(=O)NCC2C(CNC(CC3ON=C(CC)C3)=O)C2)cc2cc(F)ccc2o1 c1(C(=O)NCC(CN(C(c2cc(C)no2)=O)C)(C)C)cc(C)n(C2CC2)n1 C1(NCc2scc(C(=O)NC(COC)C)n2)CCCC(C)C1 c1(CN=C(NC(C=C)C)NCC2(O)CCCC(C)(C)C2)n[nH]c2c1CCCCC2 Fc1cccnc1C1CCN(c2cnnc(Br)c2)CC1 N1(C(CCCOC(C(C)C)=O)=O)CCC2C1CCCN2C(C1C=CCCC1)=O c1(C(=O)NCCNC(=O)Cc2cnc[nH]2)cc(C(F)(F)F)c[nH]1 N1(CC(=O)NCC2C3CN(C(=O)CC4CCCCC4O)CC23)CCCCCC1=O c1(C(=O)NCC2N(C(c3cncc(C)c3)=O)CCC2)ccc(N)c2ccncc12 c1(-c2scc(NC(=O)C(O)c3ccco3)n2)ccnc(-c2ccco2)c1 Cc1ccc(C)c(CN2CCC(NC(c3c(Cl)cncc3Cl)=O)C(O)C2)c1O C1(NC(C2C(CC)C2)=O)CCCC(C(=O)NCCc2cccs2)CC1 N1(C(Cc2c(C)nccc2)=O)CCC(C2CC2)(CNC(=O)CS(N)(=O)=O)C1 C(=O)(CCN=C(NC1CN2CCC1(C)CC2)N1CCCC(C)C1)NC CC1(C)CN(C(=O)CC23COCC(C2)C3)CC1NC(c1ccc(Cl)c(O)c1)=O N1(ONC(CCCn2cc(SC)nn2)=O)CC2(CCC(=O)N2)C1.Cc1cc(F)ccc1O c1(C(C)SC2(C#N)CC(Nc3cccc(COC(C)(C)C)c3)C2)ccnc(Cl)c1F O(S(=O)(=O)c1ccc(Cl)c(Br)c1)c1c(C)ccc(NC(=O)C(C)C)c1 C1(N(C(=O)Cc2nocc2C)CC)CC(=O)C12CCCC2.C1(C)CCN(C=O)CC1 Cc1nnc(CCC(=O)NC2CN(C(C3CN(CC(F)(F)F)CCO3)=O)C2)n1C c1(NCCC(C)F)cc(Br)ccc1S(=O)(=O)N1CC2CSCC(C2)C1 c1(N2CCC(C3C(C(=O)OC)C3)C2)ncnc2c1CCC2 C=CC(C)(C)CC(=O)NC1CCN(C(c2cccc(N3CCCC3)n2)=O)CC1 c1(C(N2CCC(CC#C)C2)C(=O)NC2CCOCC2)ccc(C)c(OC)c1 c1(C(=O)NC(CCOC)CNC(=O)C(C)(O)C2CCC2)ccc(C#N)c(F)c1 C1(C(=O)NC2CN(C(=O)CS(=O)(=O)NC)CCC2F)(COC)CCCNS1(=O)=O CC(C)CC(C)(O)C(=O)N1CC2(CC(NC(c3cc4ccoc4s3)=O)CO2)C1 CC1CC(C)N(C(=NCCc2ccc3c(c2)CCO3)NC(c2ccnn2C)C)C1 C1(CNC(=O)CCn2cc(Br)cn2)COC2(COCCN(C(=O)CCBr)C2)C1 CC1CCCCC1(CNC(c1cnc(S)n1C)=O)NC(c1ccccn1)=O S(=O)(=O)(c1ccccc1)NC(C(=O)N(C1CC(O)C1)CC(C)C)C c1(N2CCC(NC(c3c(C(C)C)onc3)=O)C(F)C2)ncnc2ccc(Cl)cc12 c1(C(=O)NC2C(N(C)C(c3nn(C)cc3Br)=O)CCCC2)cc([N+](=O)[O-])c[nH]1 c1(C(N2CC3N(C(CC(=O)OC)=O)CC(C3)C2)=O)cn2ccc(CO)cc2n1 CC1(CO)CCN(C(c2cc(-c3c[nH]nc3-c3cccs3)ccn2)=O)C1 c1(OC)ccc(C=CC(N2CC3CC2CN3C(=O)C=C(C)C(C)C)=O)c(OC)c1 CC(C)(C)CC(O)CC(=O)NC(C(=O)Nc1ccc(F)c(C#N)c1)C1CCOC1 C1(n2cc(-c3n(C)c(S)nn3)nn2)CC2(CCCCC2)CO1 CC(C)C(C)CNC(C1CCCN1C(=O)C=CC1CCC1)=O C1(C(=O)NCC(CNC(CN(c2ccccc2)C)=O)(C)C)CCC2(CCC2)O1 Cn1nc(-c2ccco2)cc1NC(c1sc(Br)cc1Cl)=O C(=O)(C1=COCCO1)NC1(c2ccccc2)CCN(C(C2(CF)CCC2)=O)C1.C=CC N1(C(C=C(C)Cl)=O)CC(CNC(c2ccc(NS(=O)(=O)NC)cc2)=O)C2(CC2)C1 CC1CCc2ccccc2N1C(=O)CS(=O)(=O)Cc1ccc(I)cc1 C1(NC(C2(CNC(CN(C3CCC3)C)=O)CC(C)(C)C2)=O)C=CC(C)(C)CC1 C(CCC)(C(=O)NCC(=O)NCC1CCN(Cc2ncon2)CC1)=CCC C#CCC(CC#C)C(=O)NC(CN(C(=O)C=C1CCOCC1)CC)CC Cn1ccc(C(=O)NCCOCCNC(c2csc(CO)n2)=O)c1 C12(NC(CCCC(=O)NCC)=O)CCCCC1N(C(C1SCCS1)=O)CC2 CCC(CCC(=O)N(CCCNC(=O)C=C1CCOCC1)CC)OC CC1CCCC(C(N2CCCC3(CNC(=O)C=CCO)CC23)=O)CC1 c1(OC)[nH]c(=NCC2CCCCCC2NC(=O)CC2CC2C)ccc1[N+](=O)[O-] C1(NC(c2c(C)sc(CC(C)C)n2)=O)C2CCC1N(C(=O)Cc1cnoc1)C2 c1(NC(c2cnn(C3CC3)c2)=O)cnc(C2CCC2)o1 CCCC(CC1CCCC1)C(=O)NCC1CCN1C(c1cc(OC(C)=O)c(Cl)s1)=O S(=O)(=O)(c1ccc(C(=O)N(C(C)C(=O)O)C2CC2n2ccc(C)n2)o1)NCC CC(CCC(=O)NC12CCN(CC1)C2)NC(C1CC(=C2CCC2)C1)=O c1(NCC(=O)NC)nc(NCC(CC(F)F)c2ccccc2)c2ncn(C)c2n1 C(C)(CCN=c1[nH]cc([N+](=O)[O-])cc1C#N)NC(c1ccc(C#C)cn1)=O N1(C(c2c(CC)cns2)=O)CCCC(C)(C)C1CNC(c1ccc(O)cn1)=O Cc1cc(C(=O)N(CC(O)CN(C)C(C23CSCC2C3)=O)C)cc(O)n1 N1(C(CC(C)OC)=O)CCC(CF)(NC(c2cc(C)cnn2)=O)C1 C1(NC(=O)COCC2CC2)CCN(C(C2(C3CCC3)CC2)=O)CC12CCC2 c1(C(=O)NC(C2CCN(C(C(c3ccccc3)C)=O)C2)C)cnnc(O)c1 c1(C(N2C(C)CC(NC(C3CCCN3CC(F)(F)F)=O)C2)=O)ccn2ccccc12 N1(C(C2CCC(N(C)C)C2)=O)CCCC(C2OCCO2)C1 c1(Nc2c(CCC(=O)OC)cccc2)cc(C)c2cc(C(=O)OC)[nH]c2c1 C(=O)(CC(C(F)(F)F)n1cccn1)NCC=CCNC(CCC1(C)CC1)=O C1(NC(c2scc(C)c2Cl)=O)CN(C(c2ccc(C#N)[nH]2)=O)CC12CCOCC2 c1(C(=O)NCCN(C(=O)CCS(=O)(=O)NC)CC)cn(CC#N)c2ccccc12 CCC(C)N(OC)C(=O)C(F)C1CCN(C(=O)CC2CCCCN2C)C1 c1(C(=O)NCCCCCN(C)C(C2CCOC2(C)C)=O)ccc2cnn(C)c2c1 C=CCC(CC)C(=O)N1CCCC1C(C)(C)CNC(c1ccccc1)=O C1(c2cn(C(CC)C)nn2)CCCN(C(=O)Cn2ccnc2C)C1 c1(OCC)c(CCC(=O)Oc2ccc(C(C)OC)cc2)[nH]c2ccccc2c1=O CCCCC(F)C(=O)NCCC1CSCCN1C(=O)Cn1cnc(=N)[nH]1 c1(-n2c(C)cnn2)ccc(C(N2CC(NC(=O)Cc3ccc(O)cc3)C2)=O)cc1 c1(C(N2C(C)CC(NC(c3c(CC)n[nH]c3)=O)C2)=O)cc(C)cc(Br)c1F c1(C(=O)NC2CC(NC(C3(C(=O)OC)CC3C)=O)C2)cc(O)nc2cnccc12 N1(C(C2C(C)CCOC2)=O)CCC(C(=O)N(C)CC2CCCC3CC23)C(C)(C)C1 C1(C(N(CCCC)CCO)=O)(OC)CCN(Cc2cnc(N3CCCC3)nc2)CC1 C1(NC(C2OCCC(NC(=O)CC(C3CC3)C3CC3)C2)=O)CCn2nccc2C1 c1(OC)ccc(O)cc1C(N1CCC(O)(C(=O)NCc2ncccc2F)C1)=O C1(CCC)CCCN1C(=O)C(=O)NCCCN(CCOC)CC N1(C(C(CC)C#N)=O)CC(OC)CC(NC(=O)Cc2ccn(C3CCCC3)n2)C1 C1(CNC(c2cc(Cl)cs2)=O)CN(C(=O)CN2CCS(=O)(=O)CC2)CC12CC2 N1(C(C2C(=C)C2C(=O)OCC)=O)CCCC(CCC(=O)NCc2cn(C)nn2)C1 c1(C(CCC(F)Cn2cc(-c3ccccc3)nn2)=O)cccc(F)c1.N(CC)CC c1(-c2nnc(OCCC(C(OCCOC3C4(CC(=O)NC3)CC4)CC[N+](=O)[O-])=O)s2)cc2cccnc2s1.OCC Cc1ccc(C(N2CC=CCC2C(N2CCCC(CC3CC3)C2)=O)=O)cc1F C(=O)(C(O)CC(F)(F)F)NCCC1(NC(C(C2CCC2)OC)=O)CCCC1 c1(SCC(N2CC3C(NC(C=NOC)=O)C3C2)=O)nnc2ccccn12 c1(OC)ccc(C(=O)NCCCN(C)C(c2cocc2C)=O)nn1 c1(CC(=O)N(C2CCN(C(=O)C(C#N)C(C)(C)C)C2)C)c(F)c(F)cc(F)c1F C1(n2ccnn2)CCC(N=c2ccnc(N3CCCC4(CCC4)C3)[nH]2)CC1 N1(C(=O)OCC)CSCC1C(=O)NC1CCN(C(c2cc(C3CC3)[nH]n2)=O)C1 C1(CCC(=O)NCCOCCC(C)(C)NC(CCCSC)=O)CCC(=O)NC1=O C1(OCC)CCN(C(C2CC=CC(NC(c3[nH]ccc3C)=O)C2)=O)C1C C1(N(C(c2c(C)[nH]c(C(C)(C)C)c2)=O)C)CC2CC1N(C(c1cc(Cl)no1)=O)C2 N1(C(C(C)SC(C)C)=O)CC(CNC(=O)C=Cc2cocn2)CC1(C)C N1(C(C2CC23CCCC3)=O)CCOC(c2cn(C3(C(=O)O)CC3)nn2)C1 Cn1ccc2nc(N3CC(CC)C3)ncc12.C(=O)(C=CCOC(C)(C)C)OCC CC1COCC(C(=O)NCc2n[nH]cc2C(=O)N(c2ccccc2)C)O1 CC(C)CC(C)(O)C(=O)N1CC2C(C(=O)Nc3ccc(C(C)C)nc3)C2C1 N1(C(C(C=C)(C)CC)=O)CCC(C(=O)NCCN2CCCCCC2=O)C(C)(C)C1 C(=O)(C(Cc1ccncn1)NC1CCCC1)OC1CCN(C(C)(C)C)C1 c1(C(N2C(C(N3CC(=O)NCCC3)=O)CC(O)C2)=O)c(F)cc(Cl)cc1Br c1(C(=O)NCC2(OC)CCN(C(=O)CN3CC4CC4C3)C2)noc2c1COCC2 CCC(CCN(C)C)CCOC.C1(C)CN1C c1(C(=O)NC2CC(NC(c3c(C)c(=O)cc[nH]3)=O)CC2O)cc2n(c1)CCCC2 CCC(C)(CNC(c1nc(C)ccc1F)=O)C(=O)N1CCC12CC(O)C2 c1(C(=O)NC2C(NC(c3ccc(C(C)=O)o3)=O)CCCC2)ccnc2c1CCC2 c1(CC(=O)OCC)cccc(C(F)(F)F)c1F.C(CCC(=O)OC(C)(C)CN)OCCO c1(C2C(F)(F)C2)ccc(CSc2ccccc2)cc1.N12CCC(C1)OCC2 n1(CC)nnc(C(N2CCCC2C(C)(C)NC(=O)CC2CC(F)(F)C2)=O)c1C C(CC(=O)NCc1ccc(O)nc1)(C(F)F)NC(c1ccc(C)cc1)=O c1(C(N2CC(CNC(CCC3CCC(C)O3)=O)C2)=O)cnc2ccccn2c1=O Cc1nnc(C(=O)N(C(C)CNC(=O)C=CI)C)s1 C1(CNC(C=C(C)C(C)C)=O)CCN(C(c2ccc(-c3cccs3)o2)=O)CC1C CCC(CC(=O)OC(c1ccc(OC)cc1)CN(C)C)c1ccc(C)cc1 c1(C(=O)NC(c2ccccc2F)C(=C)C)cc(CC)cc(C(F)F)c1 CC1CC2C(CC(C(=O)OC(=O)OC(C)(C)C)N2CCC(C)(C)C(O)C(F)(F)F)O1 N1(C(c2c(CC)c[nH]c2)=O)CCCC1(C)C(=O)NCC(C)(C)OC Cc1cc(C(N2CCSCC2CCNC(C2CC2C(F)F)=O)=O)sc1C C(C)(CO)(CN=c1ccc(NC(C)(C)C)c[nH]1)OC.N12CCCC(C3CN1C3)C2 C(=O)(CCC1=NNC(=O)CC1)NC1C(C)CN(C(c2ncoc2C2CC2)=O)CC1 N1(C(c2c(CC)n[nH]c2)=O)CC2(CC(NC(=O)C(c3ccccc3)F)CO2)C1 N1(C(C2(OCC)CCCC2)=O)CCOC(C(C)NC(c2cncc(F)c2)=O)C1 C1(C(=O)OC(C)(C)C)CCCCN1C(C1CCCN1Cc1ncc(Br)s1)=O C1(C(=O)OC)CC2C(CCC(C)N2CC2Cc3cc(Br)ccc3C2COC)O1 CC1=NN(C)C(=O)C1CC(N1CCN(C(c2[nH]cnc2C)=O)C(C2CCC2)C1)=O N1(C(CC(=O)NCC#C)=O)CCCC(NC(c2cncc(C)n2)=O)C1CC c1(CCC)ccc(S(=O)(=O)N2CC3C(NCc4nc[nH]c4C(C)(C)C)C3C2)cc1 C1(C(=O)NCC=CCC(=O)NCC(C)CC=C)CCCC(=O)C1 c1(C(N(CC(CO)(CO)NC(=O)C=Cc2cnc[nH]2)C)=O)csc([N+](=O)[O-])c1 CC1(CNC(c2ccncn2)=O)CC(F)(F)CN1C(c1cscc1Cl)=O N1(C(CCC=C(C)C)=O)CCN(C)C(CNC(c2ccncc2)=O)C1 c1(CCNC(=O)NCc2ccc(O)nn2)cccc(F)n1 C1(C2CCCNC2)(NC(c2ccc(CSC)cc2)=O)CCOCC1 C1(C)(CNC(CCN(C(CCOC)=O)C2CC2)=O)C=CCCC1 C1(CNC(C(C(C)C)SC)=O)CC2(CCCCN2C(=O)C=CC(=O)N(C)C)C1 c12cccc(c1[N+](=O)[O-])N2.CCCC=CC(=O)NCCOCCNC(C)=O C1(C(N2CC(C(C)NC(C(CCCC)NC(N)=O)=O)C2)=O)Cc2nnc(C)n2C1 Cc1ccc(F)c(CNC(c2c(I)cnn2C)c2nnnn2C2(C)CC2)c1 Cc1cc(C(=O)N(C2CCCC2)CCCNC(=O)C(C)C(C)C)cn1C C(=O)(CC(C(=O)N1CCC(NC(=O)CC(=O)N(C)C)C1C)N(C)C)OC c1(C(=O)NCC2(NC(C=C(C)Cl)=O)CC2)cccc(Br)c1CO C1(NC(COc2ccc(C(CC)C)cc2)=O)CCCCN(C(=O)CC(F)F)C1 CCC(C)(C#N)C(=O)NC(CC(=O)NCC1(CC)CCCO1)C(C)C c1(C(=O)NC(CNC(C(Cc2c(C)noc2C)C)=O)C)ccc(F)c2occc12 CN=c1[nH]nc(CC(N2CCC(C)C2CNC(c2cnn(C)c2Cl)=O)=O)s1 c1(C(N(C(C#C)C2CCC2)C)=O)cc(CNC(=O)C(C2CC2)C2CC2)on1 N1(C(CCNC(CC(C)C)=O)=O)CCCN(C(c2ncccc2Cl)=O)CC1C CC1CC2(CC(C(=O)NCC3CCCCC3NC(C34CC(CO)(C3)C4)=O)C2)C1 CC(C)CCCC(=O)N1CCC(NC(c2cn(CCO)nn2)=O)C1 CCC1=NOC(C(=O)NC(CNC(=O)Cc2cncn2C)CC(C)C)C1 Cc1nn(CCO)c(C)c1C(=O)NCCCN(C)C(C1COC(C)CO1)=O Cc1cc(C(=O)NC2CC(F)(CNC(c3cc(C(C)C)on3)=O)C2)c(N)cc1F N1(C(C2C(C)(CC)C2)=O)CC(C2CN(C(c3ccc(Cl)c(NC(C)=O)c3)=O)C2)C1 C1(C(=O)NC2(C3CN(C(c4occc4C4CC4)=O)C3)CC2)CCCCC12CCC2 C1(C(=O)NC23CC(CNC(c4cnccc4Cl)=O)(C2)C3)CCCC1C1CC1 c1(NC(N(CC(c2ccccc2)CC)CC)=O)nc2ccc(I)cc2s1 c1(C(C#C)OC(c2cc(C3CC3)ns2)=O)ccccc1F C(=O)(CC1=CCCCC1)NCC(C)(C1CC1)NC(C(C(COC)C)C)=O N1(C(CCOCC)=O)CC(C)C(C)(CNC(c2c(N)cccc2Cl)=O)C1 c1(NCC(C)Oc2c(C)cccc2)ccc(S(=O)(=O)NCC=CC2CC2)c(Cl)c1 c1(CC2C(NC(=O)NC(C)CCF)CCC2)cc(N2CCCC2)ccn1 N1(C(c2n(C=C)ncc2)=O)CCC2(NC(=O)C=C3CCSCC3)CCCC12 c1(CCC(=O)N(C(C)CN(C(=O)CSc2n[nH]c(O)n2)C)C)cncc(F)c1 c1(C(=O)NC2C3N(C(C=CC=CC)=O)C(CC3)C2)cc(Br)cc([N+](=O)[O-])c1 N1(C(c2nn(CC)nc2C)C(=O)NC2CCC2)CCc2ncc(C)n2CC1 c1(C(N2CCC(OCCNC(=O)Cc3cncs3)C2)=O)cncc(C(F)F)c1 c1(C(=O)NCC(CC)NC(=O)CC2(C)CCCC2)cc(O)c2cnn(C)c2c1 N1(C(c2cc(C)c(Cl)cn2)=O)CCC(C)N(C(c2ncn3c2COCC3)=O)CC1 Cc1ccc(O)c(C(=O)NCCC2CN(C(=O)C3=NOC(C)C3)CC(C)O2)c1 c1(OCC)cncc(NC(C2CCCN2C(c2ncccc2Cl)=O)=O)c1 C(=O)(C(CNC(c1c[nH]nc1C(F)F)=O)C(C)C)N1C(C)(C(C)C)CC1 C1(C(=O)Nc2cc(OCC)c(COC)cc2)CCOc2ccccc2N1 C1(C)(C(N2CCCC(CC(=O)NC(C(=O)OCC)COC)C2)=O)CC2(CCC2)C1 Cc1nc(CCNC(C2(NC(=O)CCc3ccsc3)CCOCC2)=O)c(C)o1 C(=O)(C1=COCCO1)NC1C(C#N)CN(Cc2nc(SCC(C)(C)C)[nH]n2)C1 C(=O)(C1=COCCC1)NCC1(F)CCC(NC(CC2(OC)CCC2)=O)C1 N1(C(C2CCN(C(C)=O)CC2)=O)CCN(C(=O)Cc2cnn(C)c2C)CC(O)C1 C12(C(N3C4C(N(C(=O)C(O)C5CC5)C)CC(C4)C3)=O)CCC(CO)(CC1)CC2 CCCCCCC(C)(CC)C(=O)NC(CNC(C1(C(N)=O)CCC1)=O)CC CC1Cc2cccc(-c3nc(CS(C)(=O)=O)nn3-c3cccc4c3OCO4)c2O1 N1(C(C2(C)COC(=O)C2)=O)CCCC(C)(C)C1CNC(=O)CCCC1CC1 c1(C(C(=O)NCCCN(CCCC)CCCC)N)cccnc1 C(=O)(C1CCCc2n[nH]cc21)N1CCC(CNC(C(C)(F)F)=O)(CO)C1 c12ccc(cc1)c(=O)[nH]2.C1(CCN(CCNC(C2(C#C)CC2)=O)C)CCOCC1 N1(C(C(=Cc2cn[nH]c2)C)=O)CCC(C)(C)C1C(=O)N(C)CCN(C)CCO C(=O)(C#CC1CCCOC1)NC(C)(C)CNC(=O)C(C)(C)C(C)(C)C C1(CCCNC(C(CC)N(CC)CC)=O)CCCN(C(c2ccccc2Cl)=O)C1 N1(C(C2C(=C)CC2)=O)CCC(CN(C(C2CC(=O)N(C)C2)=O)CC)CC1 Nc1ccnc(C(N2CCC(F)(CNC(c3nsnc3O)=O)C2)=O)c1 c1(C(C)C(=O)N(C)Cc2cn(CCCCCF)nn2)ccc(O)cc1 C1(C(N(C(CCNC(c2n[nH]c(C)c2N)=O)C)C)=O)CC1C1CCCCC1 c1(CC)nc(=N)[nH]cc1C(=O)NC(CNC(=O)C1=COCCC1)CC(F)(F)F c1(C(=O)NCCOC2CN(C(C3CCC4CC34)=O)C2)cc2c(=O)[nH]ccn2n1 N1(C(C2CC=CCC2)C(=O)NCCCF)CCCC2(CC(O)C2)C1 N1(C(C2CCCC(C)(C)C2)=O)CCC2(CC1)CN(C(=O)Cc1ccccc1Cl)C2 CC1(C)CN(C(C2CC(NC(=O)C=Cc3cc[nH]n3)C2)=O)CCO1 CCCC(CC)CC(=O)NCC(C)(C)CN(C(c1cc(Cl)cn1C)=O)CC c1(OC)cccc2ccnc(NCCNC(=O)CCCCNC(=O)OC)c12 C1(C(N2CC(C(=O)Nc3cccc(F)c3)C2)=O)C2CC3C(C2)C13 C1(C(N(CCCN(C(C(COC)COC)=O)C)C)=O)CCC(C2CC2)C1 CCC(CC(=O)N1CCCC(C)(CNC(c2snc(C)c2N)=O)C1)C(C)(C)C Cc1c(NC(=O)C(CCC2(C#N)CC2)N(C2CC(F)(F)C2)C2CC2)cccc1Cl C(=O)(C(O)CC(C)(C)C)NCC(CNC(c1n(CC)nc(C2CC2)c1)=O)F c1(C(N(CC(=O)OC)Cc2ccccc2)=O)cc(Cl)c(Br)c([N+](=O)[O-])c1 C1(NC(CCN2CCN(C(C)C)CC2)=O)CC(F)CN(C(c2cnns2)=O)C1 N1(C(CC(CC)c2ccc(C)cc2)=O)CC2(CC(NC(=O)C(C)NC(C)=O)C2)C1 C1(NC(=O)CCC2CCN(C(C3CC4(CCC4)C3)=O)C2)CCCCCCC1O c1(C(=O)NCCC2CCC(NC(CC3(C=C)CC3)=O)C2)cc2cc(O)ccc2[nH]1 c1(CC)cc(C(=O)NC2CN(C(c3nn(C)cc3C)=O)CCC2C)cc(F)c1 C(=O)(C(CC)C(=O)OC)N(C)Cc1ccc(CNC(C2CC(CCC)C2)=O)cc1 c1(C(N2CCC(C)(CNC(c3ccncn3)=O)C2)=O)ccnc(Br)c1F CCC(C)(C)C(C)CC(=O)N1CC(NC(c2c(Cl)ccc(F)c2F)=O)CC(C)C1 c1(CNC(c2cnc(CC)o2)=O)ccc(C(=O)N(C2CCCC2C)C)nc1 c1(C(N(C)CC2CCN(C(=O)CC3CCC(C)(C)C3)C2)=O)cc(S(N)(=O)=O)c[nH]1 c1(C(N2C3(CN(C(c4c(C)ncn4O)=O)C3)CC2)=O)cc(C#N)c(N)cc1O CC(C)CC(O)C(=O)NC1(C)CCN(C(=O)C(C)C(F)F)CC1 N1(C(C2OCCC(=O)C2)=O)CCC(NC(=O)C=Cc2ccco2)C(F)C1 c1(C(N2CCCC(N3CCOCC(=C)C3)C2)=O)cc(CC)nc(Cl)c1C#N CC1(CNC(c2n[nH]cc2F)=O)CN(C(=O)CC(c2ccc(F)cc2)O)CCO1 c1(C(N2CC(O)(CNC(C3C4COCC34)=O)C2)=O)ccccc1Br c1(OCC)cccc(N(C(C(=O)NC2CC2c2ccco2)=O)C(C)C#N)c1 C(=O)(CCCC(=O)NC1CC1)NCC1N(C(C(CCC)F)=O)CC(O)C1 N1(CC)CCOCC1CC(=O)NCCc1ncoc1C.c12nc(co1)C(=O)N2 Cc1cc(NC(=O)CC2CN(C(c3cc(Br)ccc3Cl)=O)C2)ncc1F C1(CNC(C(c2ccc(C(F)F)cc2)C)=O)CCC(NC(=O)C(F)(F)CF)CC1 N1(C(C(c2c(C)noc2C)CC)=O)CCCCC12CN(C(c1ccn(C)n1)=O)C2 N1(C(C(CC(C)C)ONC(CC2ON=C(C)C2)=O)=O)CCCC(C)(C#N)C1 C(C(C)(C)C(c1ccccc1)NCC(=O)O)NC(=O)OC(C)(C)C.C(=O)(CCC=CBr)N Cc1sc(C(=O)NC2CCN(C(c3ccoc3Cl)=O)C2C)nc1Br CCC(C)(C(=O)N1CC(O)(CCNC(=O)CC2CC3(CCC3)CO2)C1)C(N)=O N1(C(c2c(F)ccc(C#C)c2)=O)CC2CN(C(=O)Cc3ccsc3)CC2(C)C1 C1(C(N2CCC(N(C)C(c3nccnc3Cl)=O)C2)=O)CC2CCC(C1)S2 c1(NC(C23C(CN(Cc4cncc(C#N)c4)C2)C3)=O)cccc2c(Cl)ccnc12 c1(C(=O)NC23CN(C(CCC(C)C)=O)C(CC2)CC3)c[nH]c2cc(F)ccc12 Cc1cn(C)cc1C(N1CC(NC(=O)CC2CSC2)CC1C)=O C(CCC(C)C(=O)N1CCN(C(c2cccc(N)c2OC)=O)C(C)C1)OC CN1CCC(C)(C(N2CCCC2(C)CCC(=O)NCC(CO)C2CC2)=O)C1 N1(C(c2csc(O)n2)C(=O)Nc2ccccc2)CCC(COC(CC)(C)C)CC1 c1(OC)ncc(Br)cc1NC(C1CC1C(=O)Nc1cccc(C2CC2)n1)=O N1(C(C(C(=O)OC)SC)=O)CCOCC(C(=O)N(C)CC2CC(F)(F)C2)C1 c1(C(=O)NC(C)(CNC(C2CCC(O)C2)=O)CO)nnc(Cl)cc1N CCCCCCCC(=O)NC(C)(CNC(c1ccnc(O)c1F)=O)CC C=C(C)CCCC(=O)NC1CN(C(c2ccc(OC)cc2C(F)F)=O)CC1C N1(C(c2nc(C)[nH]n2)=O)CCCC2CC(NC(c3ncn4c3CCC4)=O)CCC12 c1(C(=O)NCC(C)N(C)C(C2C=CCCC2)=O)cc(C(F)(F)F)cnc1O N1(C(C2C(c3cc(C)no3)C2)=O)CC2(CCN(C(C3(C)COC(=O)OC3)=O)C2)C1 C(C)(C)(CC(=O)Nc1ccc(C(N)=O)cn1)N(C(CSC)=O)C c1(C(=O)NCC2CCCC(NC(CSCC)=O)C2)c[nH]c2c(F)cccc12 c1(C(N2CCC(NC(c3c(C)nccc3)=O)CC2C)=O)cc2ccccc2cn1 CN1CC(O)CC1C(N1CCC(C(C)(C)NC(=O)CCc2ccc(O)cc2)C1)=O CC(C)CCCCC(=O)NCC(C)(C)CN(C(=O)CC12CCCC1C2)C C1(CCN(C)C(C2(O)CCCC2)=O)CCN(C(=O)CCS(C)=O)CC1 N1(C(C(c2ccccc2)OC)=O)CC2CC1CN2C(=O)C(N1CCCC(O)C1)C N1(C(C)=O)CCC(C(N2CC(NC(C3(C)CSC3)=O)C2)=O)CC1 NS(=O)(=O)c1ccsc1C(=O)NC1CC(NC(C2CCCO2)=O)C1 c1(C(=O)OC)ccc(C(=O)N(CC(O)CN(C(=O)CN2CCC2C)C)C)c(F)c1 c1(CCC(=O)NCCC2CC(NC(C3CC3(F)F)=O)C2)cccc(F)c1 C1(C(=O)NC2C=CCC(C(N3CC=CCC3)=O)C2)CC2C(C1)C2(F)F Cc1ccc(C(C)C)cc1OCC(=O)NCC1CCC1NC(c1cccnn1)=O N1(C(C2ON=C(C)C2)=O)CCC2(CC1)CN(c1nccc(C(C)C)n1)CCO2 N1(C(c2cnccn2)=O)CCC2(CC1)CN(C(c1ccc(Cl)s1)=O)CC2CO N1(C(c2cccc(OC)c2Cl)=O)CC2CN(Cc3cc(F)c(Cl)c(Cl)c3)CC2C1 C=CC(CC)CC(=O)N1CCC2C(C(=O)NCc3cccc(O)c3)C2C1 C(=O)(C1=CSCCO1)N(CCCCCNC(CCC)=O)C.C1C(=O)N1 c1(C(=O)NCC(CNC(c2n(C(C)C)ccc2)=O)CO)cccc(N)c1O Cc1ncc(C(N2CCCC2(C(N2CCC(CC3CCC3)C2)=O)CO)=O)cc1Cl c1(C(C(=O)NC2CC(CCNC(=O)CNC(=O)C(F)(F)F)C2)O)cccc(Cl)c1 Cn1c(=O)cc(C(=O)NC2CCCC2NC(=O)C=CC2CCC2)c2ccccc12 n1(CC(=O)NC2CCC(C#N)CC2)cc(-c2cccs2)cc(C(F)(F)F)c1=O N1(C(c2cc(OCC)no2)=O)CCN(C(=O)C(C)N2CCCC2)C2(CCC2)C1 c12cc(sc1C)C(=O)N2.c1(C2(C(N(CC)CC)=O)CC2)ncccc1O C(=O)(CCCCO)NC.C#CC1(C(=O)NCC2(C(=O)NC3CC3)CC2(F)F)CCC1 c1(OCC)c(Cl)ccc(C(N2CCC(F)C(NS(=O)(=O)CC3CCC3)C2)=O)c1F N1(Cc2ccc(N(C(C)C)C(=O)C3CC3)cc2)CC(C(=O)O)CC1(C)C c1(C(=O)NC2CCCC(NC(c3nc(CC)oc3)=O)C2)ncnc(OC)c1F c1(OC)cccc2c(C(N3CCC(N(C(=O)C(C)=C4CC4)CCO)C3)=O)coc12 C1(C(=O)NCCC2CC(C)C2)CCN(C(=O)C2=COCC2)CC1(C)C c1(C(N2C(C)CCC2C)C(=O)NC2CCOC2)cccc2c1ccn2C C1(C(C)C(=O)NC2(CCO)CN(C(=O)C(C)C3CCC3)C2)CCC(=O)N1C CC1(C)C2CCC1(CC(=O)NC1CCCC(NC(c3cc(F)n[nH]3)=O)C1)CC2 N1(C(c2cc(OC)ncc2)=O)CCN(C(C2CCN2C2CCCC2)=O)CC1C C1(C(N(CCCN(C)C)CCSCCCNC(=O)CN2CCC2)=O)CCOC1C C(CC(N)C(=O)N1CCOC(CN2CCNCC2)C1)=CC N1(C(c2ncc(OCC)nc2)=O)CCN(C(=O)C=CSC)CC1CC(F)F C1(NC(C2COCCO2)=O)(CO)CCN(C(c2sccc2-n2cccc2)=O)CC1 N1(C(c2sc(CC)c(C)c2)=O)CCC(NC(c2cncc(C(C)C)c2)=O)C(C)C1 O=C(C(F)C(F)(F)F)N1CC2(CNC(C3(Oc4ccccc4)CC3)=O)CCC1C2 c1(NC(C2CCN(C(C(C)(C)C)=O)CC2O)=O)cc(Br)cnc1[N+](=O)[O-] C1(CC=C)(NC(c2coc(Cl)n2)=O)CCN(C(=O)C(N2CCNC2=O)C)C1 C1(NC(CCC(=O)N(C(C)C)C)=O)CCC2CN(C(C3C4CCCC34)=O)CC2C1 C1(NC(c2cc3ccccn3c2)=O)CCCCC12CCN(C(=O)CCCF)C2 N1(C(C2C(C)OCC2)=O)CC2(CCN(C(=O)COCC3CCCC3)C2)C1 c1(C(N2CCC(N(C(=O)COCC(F)F)CCO)C2)=O)cc2ccccc2o1 Cc1cc(C(=O)NC2CCCC(N(C(=O)CC3CCOCC3)C)C2)ncc1F c1(NC(=O)NCC2(NCC)CCSCC2)cc(OC)c(C(F)F)cc1F C(=O)(C1=COCC1)NCCN(C(=O)CSCCc1ccccc1)CCC C1(CNC(c2cnc(OC)s2)=O)(NC(=O)CCC2CC2(C)C)CCOCC1 C1(CCNC(c2c(OCC)ccs2)=O)CC(OC)CN1C(c1ccsc1C)=O c1(C(C(=O)NCc2ccc(COC)o2)NC(C(CC=C)C)=O)c(C)cccc1Br CC(C)(C(=O)NCC1(CC(=O)NCC2CCC(F)C2)CC1)C1CCOC1 c1(OC)cccc(CN2CCC(NC(c3ccc(OC)cc3I)=O)C2)c1O c1(C(N2CC(C)N(c3cncc(Cl)n3)CC2)=O)nnn2ccccc12 c1(C(=O)NC(C)(C)CNC(c2coc(Cl)c2)=O)ccc2c(c1)CC(C)(C)C2 C1(CO)C2CCC(C2)N1CCn1cnnc1.O=C1CCn2nc(OC(F)F)nc21 C1(OC)CN(C(=O)C=Cc2ccn(C)c2)CC1NC(=O)Cc1ccc(C)cn1 C1(OCC)CCN(C(=O)C=CCOCCNC(C2CCC(F)(F)C2)=O)C1CSC C1(CN(C(=O)C(F)(F)CO)C)C2CN(C(=O)C(c3ccc(Br)s3)=O)CC12 c1(C(=O)NC2C(CC)N(C(c3cscc3OC)=O)CC2)cc(Cl)ccc1C(C)C n1(CCC(N2CCC(N(C(=O)CSC3CC3)C)C2)=O)sc2ccccc2c1=O c1(N2C3C(NC(=O)CN4CCCC4=O)(CCC3)CC2)nc2ncc(Cl)cc2s1 C1(C)(C(=O)NCC(CC)n2cccn2)CC(NC(c2csc(O)n2)=O)C1 CC12CCCCC1CN2c1nc2c(F)cccc2o1 c1(C(=O)NCCCCn2cc(CS(CC)(=O)=O)nn2)ccc(F)c(Cl)c1F C(=O)(C#CC(C)(C)C)NC(CNC(C(n1cc(C)nc1)(C)C)=O)(C)CO C1(c2n(C)ccn2)CN(C(c2ccoc2Cl)=O)CC1NC(c1cc(O)no1)=O CC(C)CCC(O)C(=O)N1CCOC(CN(C(=O)COc2cccc(F)c2)C)C1 C(=O)(C(C(=O)N1CC(C)C(C)(CNC(=O)C2CC2)C1)C(C)(C)C)OC(C)(C)C Cc1cccc(CN)c1Cl.N12CC(C3(CC3)C1)CNC2=O.C(C)(C)(C)OC(=O)NCC c1(C(N2CCN(C(c3ccc(SC)cc3)=O)CC2C)=O)cc2cccc(C)n2n1 N1(C(c2c(Cl)ccc(C)c2)=O)CCN(C(C2CC(C)(O)C2)=O)C2CS(=O)(=O)CC12 C1(C(C)N(C(=O)CCCc2ccccn2)C2CC2)CCCN(CCCCCF)C1 C1(C(N(CCOC)CCO)=O)CCC(CNC(C2CCCCC2C)=O)CC1 c1(C(=O)NCC2(NC(CCc3ncc(C)[nH]3)=O)CCCC2)c[nH]ccc1=N C1(C(N(C(C)C)C)=O)CN(C(=O)CCC2CCCC2)CC1F Cc1cc(N)cnc1C(=O)NCC1CC(C)N(C(=O)CN2CCCCC2=O)C1 c1(CCC(=O)N(CC(=O)NC2(CC3CCC3)CC2)C)cncnc1 Cc1cccc(CC(N2CC(CNC(c3ncc(Cl)n3C)=O)CC2C)=O)c1 C1(C(N2C(CN(C(c3ccccc3Cl)=O)CC)CCC2)=O)CC(=O)CC12CCC2 N1(C(c2c(CC)ocn2)=O)CCOC2(CCCN(c3ccnc(C4CC4)n3)C2)C1 C1(C(=O)NCC(C)NC(c2n(CC)cnn2)=O)CN(C(C)=O)CCO1 CC(C)(CC#N)C(=O)N1CCCC(CCNC(C2CC3(CCC3=O)C2)=O)C1 c1(CN(C)C(C2CCCSC2)=O)ccccc1CNC(=O)C(CO)N(C)C n1(CCCOC)nnnc1C(c1ccn(CC(F)(F)F)n1)NCC1CC1(C)C c1(NCc2c(C(C)O)n[nH]c2)cccc(OC(C)(C)C)c1 CCC(O)C(C)C(=O)N1CCCC1C=CC(=O)NCc1cccc(Cl)c1 CC(C)CC(C(=O)NC1CCCC(O)CC1)N(C)C(c1cnn(C2CC2)c1)=O c1(C(=O)NCC(CO)NC(c2c[nH]nc2C2CC2)=O)c([N+](=O)[O-])cnn1CCO c1(C(=O)NC2CN(C(c3nc(C)oc3)=O)CC2C)c(Cl)cncc1Cl C1(C(=O)NC2CC(O)C2CC(=O)NCCC2C=CCC2)(CC)CCCC1O N1(C(C(CC)Sc2ccccc2)=O)CCC(C)(NC(c2nn(C)cc2N)=O)C1 c1(OC)ccc(C(C)C(N2CC(NC(=O)CC#N)C(C)(C)C2)=O)c(C)c1 c1(OC)cc(C(C(=O)NC2CCS(=O)(=O)C2)N(C)C(c2ccco2)C)ccc1Cl C(=O)(C1=CNC2=NCCCN12)NCCN(C(C)C)C(C1C=CCCC1)=O N1(C(C(C)NC(=O)NC)=O)CC(O)(C2(CCNC(=O)C3=C(C)CCC3)CC2)C1 C12(CC(=O)N(CCCNC(C3CN(C(C)=O)C3)=O)C)COC(CF)(C1)C2 C(=O)(C(C)(C)C(O)C(C)C)NCC(CC(=O)NC(C1CCOC1)C#C)(C)C C1(NC(C(C2CCC(=O)NC2)C)=O)CCCCC1(C)C.c12ccc(o1)n(C)c2=O c1(C(N2CCC(CC3C(C)(C)C3)C2=O)NC(=O)C(F)(F)F)cccc(Cl)c1 C12(C(=O)NC(CC)CNC(=O)CC3(O)CCCOC3)CCCN(CC1)C2 C(=O)(C#CC1CCCCC1)NC1CCCC1OCC(N1CCC(C)(CCO)C1)=O c1(NC(N2CCCC(NC(c3nc(OC)sn3)=O)C2)=O)cc(Cl)cc(Br)c1F C1(CNC(c2cccc(C(C)C)c2)=O)CCN(C(=O)Cc2cncn2C)C1(C)C C(=O)(C1=CC(O)C(NC(=O)CC(C)(C)O)C1)NCc1nc(C)oc1 Cc1ccnc(C)c1C(=O)NCC1(F)CCC(NC(=O)C(C)CC2CCCC2)C1 C1(CCC(=O)NC2(C)CCCS2)CCCCN(Cc2ccccc2)C1 N1(C(C2(CCNC(C3CC4(CCO3)CC4)=O)CCCC2)=O)CC2CC1CS2=O C(=O)(CCCC(C)(C)C)NCC1(C(N2CCCCC(CO)C2)=O)CC(=C)C1 C1(C(=O)NCCN(C(c2ccc(OCCOCCO)cn2)=O)CC)CCOC1(C)C N1(C(=O)OC)CCCC(C(=O)NCC(CO)NC(c2onc(OC)c2Br)=O)C1 c1(C(=O)NC2CN(CC)C2)c[nH]c2ncc(Cl)cc12.c12ccc(cc1)CNC2=O Cc1nc2c(s1)CCCC2C(=O)N1CC2(CCCC(CNC(=O)C3=CCC3)O2)C1 C1(NC(c2nc(OCC)oc2)=O)CN(C(c2coc3c2COC3)=O)CC1(C)C.OCC S(=O)(=O)(CC(C)c1ccccc1)NCCC=C.O1NC1=O c1(OCC(N2C(C)C(NC(=O)Cc3csnn3)CC2)=O)nc(O)nc(O)n1 C=C1CCN(c2ccc(NC(c3ccc(CSc4cnn(C)c4)o3)=O)cc2)CC1 N1(C(c2c(C)coc2)=O)CC2CCC(C1)N(C(c1csnc1Cl)=O)C2 CCCC(O)CC(=O)N1CC2CC2(CNC(c2ccc(C)cc2Cl)=O)C1 CC1CC=C(C(=O)NC2CN(C(c3cccc(F)c3C(F)F)=O)CC2F)CC1 c1(C(=O)NC2(C)CCN(C(C3C(C)C3(F)F)=O)C2)ncc(C(F)(F)F)cc1N C1(NC(C(C)=CC2CC2)=O)CC2(C1)CC2NC(c1cc(CS(C)(=O)=O)on1)=O C(C(O)C(=O)N(C)CCOCCC(=O)NC(C)(CO)C1CCC1)=CC c1(C(N(CC)CC)=O)ccc2c(c1)CN(C(=O)CCc1ccc(C)nc1)CC2 C1(OC)CCN(C(=O)C2=CCN(C(=O)CC3=CCCC3)C2)CC1C c1(C(=O)NCC=CCNC(c2cn(C3CC3)cn2)=O)cc(F)cc(Br)c1O Cc1ccnn1CC(=O)N(CCC(=O)NCCCn1cncn1)C(C)C CCC1=NOC(CC(=O)NCC2CN(C(=O)CC(C)CN(C)C)CCO2)C1 CON1CCC(C(=O)NC(CNC(=O)CSC(F)F)CO)CC1 c1(OC)cccc(C(N2CCOCC(NC(=O)CC3C=CS(=O)(=O)C3)C2)=O)c1O N1(C(C=C(CC)CC)=O)CC2(CCC2)CC1CNC(c1nnn2c1CSCC2)=O c1(CNC)cnccc1-c1csc(C(=O)NCC(O)COc2ccccc2C)c1 c1(C(C(=O)NCC(C)N(C(C(CC)O)=O)C)O)ccc(O)c(OC)c1 c1(C(=O)NCC(CNC(=O)C=Cc2ccc(Cl)nc2)O)cc2cccn2c(O)n1 C1(NC(C2(F)C(C)C2)=O)CN(C(=O)CCCCN2CCCC2)CC1F c1(C(=O)NC(C)CN(C)C(c2cnn(C)c2)=O)cc(C2CC2)n(C)n1 N1(C(c2c(C)sc(Cl)n2)=O)CC2COCCC2(NC(c2csc3nnsc23)=O)C1 C(=O)(CCCCCSCCC(C)C)NCCN(C(CCCOCCC)=O)C C1(C(C)(C)C)(C(N2CC(NC(=O)CCc3ccsn3)C2)=O)CCCCC1 O=C(C1OCCn2ccnc21)NCCC1CC(F)(F)CN1C(=O)CC1CC1 Cc1ccncc1NC(c1ccc(CNC(=O)C(O)CC2CCCC2)s1)=O c1(OC)cc(C(N2CCCC(NC(=O)C(C)C(C)C)C2)=O)cc(Cl)n1 C1(NC(C(C)C2CC2)=O)CCC2(CC1)CN(C(c1ccnnc1S)=O)CCO2 c1(CCCC)nc(-c2cn(C3CNC3)nn2)n(C2CCCOC2)n1 Cc1cccc(C=CC(=O)N(C2CCN(C(=O)Cn3cc(Br)cn3)C2)C)c1 c1(OC)ccc2c(c1)CC(NC(c1c[nH]c3cccc([N+](=O)[O-])c13)=O)CCC2 c1(OCC)ccc(NC(=O)CC2C(N)CC2O)c(OC)c1 CCC(COC)C(=O)N1CCCC1(C)C(=O)NCc1ncn(C2CC2)n1 Cc1[nH]c(C)c(C(=O)NC(C)CCNC(=O)CC2NC(=O)NC2=O)c1C O=C1COc2cc(C(=O)N=c3cc(CCO)o[nH]3)cnc2N1 N1(C(C(C(C)(C)C)O)=O)CC=C(CC(=O)NC2CC3(COCCO3)C2)CC1 C(=O)(N=c1nc[nH]n2cc(Br)cc12)Nc1c(-c2c(C)ccc(F)c2)cncn1 N1(C(c2c(C)nccc2Cl)=O)CC2CC1CN(C(=O)Cc1cncn1C)C2 C1(COC)(NC(c2ccc(C(=O)OC)o2)=O)CCN(C(=O)Cc2cn(C)nn2)C1 N1(CC(=O)N(C(CCNC(Cc2ccc(C(C)=O)s2)=O)C)C)CSCCSC1 Cc1csc(C)c1C(=O)NC1C2CN(C(=O)CCCc3cnn[nH]3)CC12 C1(O)(CC(=O)NC2C(OC)CN(C(=O)CCCSC(C)(C)C)C2)CCCN(C)C1 Cc1c(OC(F)F)cc(C(=O)NC2CCC(C)(C)CC2)cc1F O=C(CC1CCc2ccc(O)cc21)NC1(Cc2ccccc2)CCCC1 CC1(O)CC(CNC(C2CCN(C(=O)CC3CCOC3=O)C2)=O)C1 Cc1cc(C(=O)N(C)CC2(O)CCN(C(C34CC(C)(C3)C4)=O)C2)cc(Cl)c1 C(=O)(C(O)P(C)(C)=O)N1CCCC(N(C(=O)COCCF)C)C1 N1(C(CC=C)=O)CC(NC(c2ccc(=O)n(CCOC)n2)=O)CC12CCOC2 C1(C(=O)NC(c2nnnn2C)C)CCN(C(C2CC2[N+](=O)[O-])=O)C(C)(C)C1 CC1CCCN(C(=O)COC(C)(C)C)C1.C1(C)CCNC(=O)OC1 c1(CC)ocnc1C(N1CC(C(O)C(=O)NCC2CC3(CC3)C2)C1)=O C(=O)(C(F)C(C)C(F)(F)F)N(C(C)CNC(=O)CC(C)n1ccnc1)C CC1(C)CC(C(=O)NC2CC(O)C(O)C2)CCN1C(=O)C(=O)NCC1CC1 CC1=C(CNC(CCCOc2ccccc2C#N)=O)C(C)(C)CCC1 N1(C(c2ccc(COC)[nH]2)=O)CC(C)(C)CC1CNC(c1cccc(OC)n1)=O N1(CC(=O)NCCCN(C(C2C(C)CC2)=O)C)CCn2nccc21 Cn1ccc2nc(N3CCC3(C)C(=O)Nc3ccc([N+](=O)[O-])c(Cl)c3Cl)ncc12 CC1(C)CC(NC(c2ccc(C#N)cc2)=O)CN1C(=O)C=CI C(=O)(C(C)CC(=O)c1ccc(F)cc1)NCCC(C)NC(c1ccnn1C)=O c1(NC(C2CCC(C)N2Cc2cnc(Cl)s2)=O)cccc2c1C(=O)CC2 C12(NC(c3c(COC)scc3)=O)CCOCC1CN(C(=O)C(C)=CCO)C2 c1(SC)cccnc1C(=O)N(CC(C)N(C(=O)CC1CCCN1CC1CC1)C)C Cc1sc(S(=O)(=O)Nc2ccc(OC3CCCCC3)nc2)cc1[N+](=O)[O-] C=CCC(CNC(=O)COCCCN(C)C)NC(=O)CCC1CCC(C)O1 c1(OC)ccc(CN2CC=CC2C(=O)Nc2cc(Cl)cnc2Cl)cc1I c1(C(=O)NCCOCCC(=O)N(C)CC2(C)CCC2)cccc(=O)o1 CC(C)CC(C(=O)N1CCCC(C)(NC(=O)Cc2coc(C(F)F)n2)C1)N(C)C C=CCCC(C(=O)NC1(C(=O)OC)CC1)NC(C1CCCC(CF)C1)=O c1(OCC(=O)NCC2OCCN(C(c3c(CC)ncs3)=O)C2)cc(Cl)ccc1Cl c1(CC(N2CC(NC(C3(CCF)CCC3)=O)C(O)C2)=O)noc2ccccc12 C1(C)(C(=O)NCCCCN(C(C2(CCC)CCC2)=O)C)CC(C2CC2)=NO1 N1(C(c2c(C)nc(COC)s2)=O)CCN(C(c2cnn(CC(F)F)n2)=O)C(C)C1 C1(CC(=O)NCC(CC)NC(=O)Cc2cc(C)sc2C)CCCC2(CC2)C1 N1(C(C2C(C)OC(C)C2)=O)CCOCC(NC(=O)C(c2cc(F)cc(Cl)c2)=O)C1 C(=O)(C1CN(C(c2ccc(C)c3c2CCC3)=O)Cc2ccccc21)OCC c1(OCC2CC(NC(C(c3ccc(C(C)(C)C)cc3)CC)=O)C2)ccc(Cl)cc1 C1(C(=O)NC2CN(C(C3(C(F)(F)F)CC(F)C3)=O)C2)C=CC=CC=C1 N1(NC(C(CC2CC2)NC2C(NC(C)=O)C2)=O)C(=O)NC(C)(C2CC2)C1=O O(NC(=O)C(c1ccoc1)NC(C1CCO1)=O)CC(CC)C C#Cc1cccc(C(=O)NC(C2CN(C(=O)CNS(=O)(=O)NC)CCC2F)=O)c1 C(C(N=[N+]=[N-])C(=O)N1C(C(N2CC3(CCCO3)C2)=O)CCC12CC2)OCC C(=O)(CC(C)(C)CN(C)C)NC(C)CCNC(c1cncc(Cl)c1)=O Cc1nn(C)cc1C(N1CCC(O)(CCNC(=O)C(O)C(C)C)C1)=O C1(C(N(C(CC)C(=O)OC)C)=O)C=CCN(C(=O)CCc2nc(C)no2)C1 Cc1nc(C(C2CC2)NCC2CC(NC(=O)C=CC3(C)COC3)C2)c(C)o1 Cc1cnc2n1CCC(C(=O)NCC=CCNC(c1cc3n(n1)CCCN3)=O)C2 C=CC1(C(=O)NCCC(=O)N(C)CC)CCN(C(C2CC(N(C)C)C2)=O)C1 S(=O)(=O)(c1ccc(NCCS(=O)(=O)NC)cc1Cl)NC1C(CC)CN(C)C1 Cc1cccc(NC(C2CC23CCN(C(c2ccccc2Br)=O)C3)=O)c1[N+](=O)[O-] Cc1cc(C(=O)N(C)CC2(NC(C3CNC(=O)CC3C)=O)CC2)c2c(c1)CCO2 c1(CC(N2CC(N(C(=O)CC34CCCC3C4)C)C2)=O)ccc(Cl)c(C(F)(F)F)c1 CC1CCN(C(=O)C(O)Cc2cnc[nH]2)CC1NC(c1n[nH]cc1Cl)=O CC(C)(F)C(=O)NCCOC(C)(C)CNC(=O)CCc1cccnc1 c1(C(N(CCCNC(=O)C(C)(F)CC2CCCC2)C)=O)cc(Cl)c(F)cc1F c1(C(C(=O)NCC2CC(NC(=O)C=CCOC(C)(C)C)C2)SC)ccccc1 c1(CC(=O)NCCCN(C(=O)CC2CC23CC3)CCO)ccccc1O c1(C(N(CC)CC2CCN(C(c3ncoc3C)=O)CC2)=O)cccc(=S)n1O c1(CN(C(C2CCCO2)C)C2CC2)noc(-c2ccn(CC(F)(F)F)n2)n1 N1(C(C(N2CCSCC2)C)=O)CCC12CN(C(C1COCC(C)(C)O1)=O)C2 CC(CC(Cl)Cl)NC(C1CCC1CN=[N+]=[N-])=O C(=O)(C(F)(F)CCCC)N1CCC(N(CC#C)C(C2(C)CCC(C)CC2)=O)CC1 n1(CC(=O)N(CC(C)N(C(c2cc(C)ncc2C)=O)C)C)cnc2ccccc12 C#CCCCCCC(=O)NCC(C1CCCC1)NC(=O)CC1COCC(C)(C)O1 CC(C(C)(C)C)N(C(=O)CN(C(=O)CC1(C)CC1)C1CC1)C c1(CC(=O)NC2C3(CC(NC(C4(C)CCCO4)=O)C3)C2)c(F)cccc1F Nc1ccc(C(=O)N(CC(N2CCS(=O)(=O)CC2)=O)CC2CCCO2)nc1N Cc1ccc2c(C(=O)N(C3CCCN(C(c4cnsn4)=O)C3)C)coc2c1 N1(C(CCN(C2CCCCC2)C)=O)CCC(NC(C2(F)CCOCC2)=O)C(F)C1 CC1=CCC(C)(C(=O)NC(C2CN(C(=O)C(C)N3CCCC3)C2)C)CC1 CC1COc2ccc(C(N3CC4CCN(C(=O)CCc5cnco5)CC34)=O)cc21 C(c1cnn(C)c1C)=CC(=O)NC(CCCCNC(C=Cc1scc(C)n1)=O)C CC1(CNC(C2C3CC4C(C3NC(=O)Cc3ccccc3)C24)=O)CC2CCC1C2 C(C1=NOC2CN(C(=O)C3=CCCCCC3)CC12)NC(c1cc(C)nc(O)c1)=O n1(CC(=O)NC(C(=O)NCC(C)(O)C2CC2)C2CCC2)cccn1 N1(C(c2ccc(Cl)c(F)c2)C(=O)NC(C)C)CCCC(C2CCCC2)C1 C(=O)(CC(CNC(C1CCOC1C)=O)C1CCC1)NCC(c1ccsc1)C N1(C(C(CC)C(C)O)=O)CCCN(C(c2cc(C)cs2)=O)CCC1 N1(c2ncc(OCC)cn2)C2CCC1CC(CC(N1CCC(O)C1C)=O)C2 C#CCC(O)C(=O)NC1CCC(CC=CC(=O)NCCC2(OC)CCC2)C1 C(=O)(C(C)(O)C(C)(C)C)NC1CCN(C(c2cnc(CCCC)s2)=O)CC1 CCCCC(O)C(C)C(=O)NCc1ccc(C(=O)N(C)Cc2cnccn2)cn1 c1(C(N(CC(CNC(c2cnc(C)s2)=O)C)C)=O)c[nH]c(=N)c(C)c1 C=C(Cl)CCC(=O)NCC(CCNC(c1ncccc1C(F)F)=O)OC c1(CNC(c2ccc3cccnn23)=O)cnn2c1CN(c1ncc(Cl)cn1)CC2 c1(C(=O)NC(C(C)NC(=O)CSCCN(C)C)C)cn(C)c(=O)n(C)c1=O c1(-c2c(C)csc2)ccc2oc(=O)c(C(=O)N(c3n[nH]c4nccnc34)C3CC3)cc2c1 C1(N(C(=O)C(c2cnn(C)c2)=O)C)CN(C(=O)Cn2cc(Br)c(=N)[nH]2)CC1O C1(CC)CCCN(C(C2C(C)CN2C(=O)CC2CCC(=O)C2)=O)C1 CC(C)(F)CCC(=O)NCC1C2CN(C(c3cnc(N)c(CO)c3)=O)CC12 Cc1nn(C)c2nc(O)cc(C(=O)NC(C)CNC(c3snc(O)c3Cl)=O)c12 N(C(=NCCCF)NCC1CC(N(C)C)C1)C(c1ccccc1F)C C(=O)(C(=O)C(C)(C)C)NCCn1ccnc1C(C)CC(N1CC(CO)CC1C)=O c1(OC(C)=O)ccc(F)cc1C(=O)NC1CC1CNC(=O)CCc1cn(C)cn1 C1(N(C)C)CCCN(CC(=O)NC(CNC(=O)Cn2cc(Cl)cn2)C2CC2)C1 c1(CCNC(C2C(NC(=O)COCCF)CCOC2)=O)ccc2ccccc2n1 c1(C(N(CCOC)CCNC(C2CC3CC3C2)=O)=O)ccc(-c2cnn(C)c2)cc1 CC(C(=O)NCc1cc(C(N2CC(C)OCC2C)=O)co1)C(C)(C)C c1(OC)c(NN2CC(NCc3cc(OC)ncn3)C2)cccc1C#N N1(C(C(CC)(C)C)=O)CC2CCC1CN2C(=O)C(=O)NC1CC1 N1(C(c2c(C)snc2)=O)CCCCC1C(C)NC(c1csc(-c2nc[nH]n2)n1)=O C12(NC(C3N(Cc4ccc(C)cc4)CCOC3)=O)CCC(N)(CC1)CC2.C(N)=O CCCN=C(NCCc1cc[nH]n1)NCc1nnc(C(C)(C)C)s1 C(C1=CCCOC1)N(C(C1CC(C)N1C(c1cn(CCO)nn1)=O)=O)C c1(C(=O)Nc2cccc(NC(C(C)n3cncn3)=O)c2)n[nH]c2c1COCC2 N1(CC(C(=O)CC2(C)CCCC2)=O)CCC(O)CC1.CC(CCC)Nn1cncn1 CC1CN(C(c2ccnc(F)c2)=O)CCN1Cc1ccc(-c2nn[nH]n2)cc1 CCCC(C(O)C(=O)NCCCCN(C)C1CC1)NC(c1ncc(CC)s1)=O Cn1nnc(Br)c1C(=O)NCC1CC(NC(c2cccc(C3CC3)c2)=O)C1 N1(C(=O)Nc2cn(CCCC#C)nc2)CCC(C(=O)OC)c2cc(Br)ccc21 C(N=c1ccnc(NCC2(C)CCOCC2)[nH]1)C1(C)CCCC1(F)F Cc1ccc2c(c1)S(=O)(=O)OC2=O.c1(-c2cc(CNCCF)sn2)ccc(F)cc1 C1(C(N2CC(NC(c3ccc(O)c(C(F)F)c3)=O)C(F)C2)=O)CC2(CCC2O)C1 c1(C(=O)NC(CC)CNC(c2cccc(CO)n2)=O)cc(NC)ccc1F C(=O)(C1CCCc2scnc21)N(C)CC1CN(C(=O)Cn2nccn2)CCO1 N1(C(c2cccc(Cl)n2)C(=O)Nc2ccc(OC)cc2C)CCS(=O)CC(C)C1 N1(C(C23C(CN(C(C(C4CC4)OCC)=O)C2)C3)=O)CCn2nc(C)cc2C1 C(C(C(=O)N1CC(c2nncs2)C1)C(C)(C)C)NC(Cc1c(C)ocn1)=O N1(C(C(Cc2ccc(C)cc2)C)=O)CCC2CCC(NC(=O)CC3CC3)C12 C=CCC(CC(C)C)C(=O)NC1CN(C(c2cc[n+]([O-])cc2)=O)C2(CCCC2)C1 Cc1cc2cccc(NCC3CCCC(C4CC4)O3)c2cn1 C1(=O)CCCN1.C1(CCNS(N)(=O)=O)CCN(C(=O)CC(O)c2ccsc2)C1 N1(C(C(C)(C)CO)=O)CC2CCC1C(NC(=O)CC1CC(=O)NC1=O)C2 C(=O)(C1CC(=O)Nc2ccccc21)N1CC(OCCNC(c2c(C)cnn2C)=O)C1 c1(C(N2CCC2CNC(c2cc(CO)[nH]n2)=O)=O)cc2ccccn2c1C1CC1 CCC(C(=O)NCCn1cc(CNC2CCCOC2)nn1)SC1CCCC1 C(N=c1[nH]c(Cl)ncc1[N+](=O)[O-])C1CCN(C(C2CC(C)OC2C)=O)C1 c1(OC)cccc(COC(=O)NC2CC2c2ccc(Br)cc2F)c1C Cc1nc(Cn2cc(CCC(=O)NOCC(C)C)nn2)c(C#N)c(C)c1C.C(COC)S N1(C(C2CCC(CNC(=O)CCCC3CC3)O2)=O)CCCC2CC12 c1(C(=O)NCCN(CCC)C(c2csc(CC(F)F)n2)=O)cccc([N+](=O)[O-])c1 c1(NC2(CNC(C(CC)C)=O)CCOCC2)nccnc1C#N C1(NC(CC(C)C(F)(F)F)=O)CN(C(=O)OC(C)(C)C)CCC12CCOCC2 CCC(C)C(O)C(=O)N(CCNC(C1CC2CCC1CC2)=O)CCOCCO N1(C(C(C=CC)O)=O)CC(CCNC(c2ccnn2-c2ccncc2)=O)C(C)C1 c1(NCCc2nccc(C)n2)ccc(C(F)(F)F)cc1S(=O)(=O)NCC(C)(C)C C1(=O)CCCOCCN1.C(=O)(C(C)NC(=O)CCC1CC1)NCCC c1(C(N2C(C(=O)NCCOCCC)CCC2)=O)cccc2c(Cl)cccc12 c1(C(N(C(C)CNC(=O)C(c2cnccn2)C)CC)=O)c[nH]c2c(F)cccc12 CC#CCCCC(=O)N1CC(OC2CCN(C(=O)C(C)(C(C)C)OC)CC2)C1 CCCC(O)CC(=O)N1CCC(CN(C)C(C2(C#N)CC3CC3C2)=O)CC1 C1(CNC(C(CN(C)C)NC(Cc2c(CC)con2)=O)=O)COCC1(C)C N1(C(Cn2ccc(C)n2)=O)CC2C(CN(C(=O)CCC3CC3(Cl)Cl)C)C2C1 C(=O)(C(O)CC(C)(C)C)NC1CC(CC(=O)NC2CN(C)CC2(C)C)C1 c1(C(=O)NCC2(NC(c3csc(Cl)c3)=O)CCC2)cnc(C2CCOCC2)nc1 c1(CC(=O)NC(C2CCCN2C(=O)Cc2ccnn2CC)C)nnn(C(C)(C)C)n1 N1(C(c2cc(SCC)ncc2)=O)C(C)C2CC1C2NC(c1cc(Br)co1)=O c1(N2C(CO)CC(C)C2)cc(Br)ccc1S(=O)(=O)NCC12CCC(CC1)OC2 C1(C(=O)NCC(CC)OC)CCCCCN1C(c1cc(C)cc(C)n1)=O c1(OC)cc(C(=O)NC2CC(CCNC(C3(C(C)(F)F)CC3)=O)C2)ccc1C C(=O)(C(CCC1CC1)NC(C1CC12CC2)=O)NCC1CC(C(N)=O)C1 c1(CNC(C2N(C(N)=O)CC2)=O)cn(-c2ncc(C(=O)O)s2)nn1 N1(c2cc(C)nc(CO)n2)CCC(C2CC2)(CNC(C2CC(N(C)C)C2)=O)C1 C1(CCNC(c2c(C)nsc2)=O)CN(C(C2CC3CC2C3)=O)CCO1 N1(C(C2(CCC=C)CC2)=O)CC(NC(=O)CCc2nc(C)c(C)[nH]2)C2(CCC2)C1 c1(C(=O)NCCN(C(C(COC)(C)OC)=O)C)cccc2cn(C)nc12 N1(C(=O)CC2CCSCC2)CCC2(C1)c1[nH]cnc1CCN2C(c1nncs1)=O C1(C(=O)NC(C(CC)C)CN(C)C)CCN(C(=O)Cn2ncnn2)C(C)(C)C1 Cc1ncc(C(=O)NCC(C2CC2)NC(=O)Cc2cccc(O)c2)n1C(F)F c1(C(N(CCN(C)C(=O)OC(C)(C)C)C2CC2)=O)cn(-c2ccccc2)cn1 C(=O)(C1CCCc2nncn21)NCCCCCNC(=O)C(F)C(F)(F)F c1(C(=O)NC(C)C(C)NC(C2CCC(=C(F)F)CC2)=O)n[nH]c2cccnc12 C(=O)(CCC(C)(C)F)N1CC(OC2CCN(C(C3C(C=C)C3)=O)CC2)C1 C(C(=O)N(C)Cc1cnco1)(C(C)(C)O)NC(CNC(C1C(C)C1)=O)=O C(=O)(C(C)(C)CNC(C1C(C)C1C)=O)NC(c1snnc1C)C c1(C(=O)NCC(C)NC(C(CC)N(C)C)=O)cnn(-c2ccccc2)c1Cl N1(C(c2c(C)nc[nH]2)=O)CCC(CNC(C2(O)CC(C)(C)C2)=O)C(F)(F)C1 N1(C(C(c2ccc(F)cc2)C)=O)CCCC1(C)C(N1CCC(NC(=O)N(C)C)C1)=O C1(NC(CCN(CC)CC)=O)CC(O)CN(C(c2nc(OC)cc(OC)n2)=O)C1 C1(C(N2CCC(N(C(=O)Cn3cnc(C(N)=O)n3)C)CC2)=O)CC(C2CC2)=NO1 n1(NC(C(N)=O)Cc2ccc(F)cc2F)ncc2ccc(Br)cc2c1=O CCC(CC(=O)NC(C)CN(C(=O)CCNC(c1ccccn1)=O)CC)C1CC1 CN1CCN(C(=O)C=CC2CCC2)CC1C(N1CCN(C)C2CC12)=O n1(CC)nc(COC(C2CCN(c3ccc(Br)cc3)C2=O)=O)c(Br)n1 C1(CN(C(CC)C)Cc2ccc(Cl)cc2)CC(F)CN(C(C2CCCC2)CC)C1 N1(C(C2C(C(C)NC(=O)CC(C)C(F)F)C2)=O)CCN(C)CC(C)C1 N1(C(C2CCCN(CCC)C2)=O)CCC(C2(NC(c3nccn3C)=O)CC2)CC1 C1(C(=O)NCCNS(CC)(=O)=O)CCCCCC1NC(C12CCCC1C2(F)F)=O N1(C(C2CC(OCC)C2)=O)CCCN(C(c2ccc([N+](=O)[O-])cc2)=O)CC1C c1(C(=O)N(CCC(=O)NC(C2CCCC2)CO)CCO)n[nH]c2ccccc12 c1(C(=O)NCC(N(C(CC=C)=O)C)C2CC2)c[nH]c2nc(Cl)ccc12 N1(C(CC(C)n2cccn2)=O)CCN(C(c2cc(N)cnc2Cl)=O)CC(C)C1 CC1(CNC(=O)C(C2(O)CN(C(C3(Cl)CC3)=O)C2)F)CCCC(=O)N1 Cc1cc(C)c(C(N2CC3CCC2CN3)CNc2csc3nccn23)c(=O)o1 N1(C(C2(C)CC(=C)C2)=O)CC2CC2(CNC(C2COCCN2C2CCCC2)=O)C1 CC1(C(N2CCCCC2CNC(=O)CCN2CCNC(=O)C2)=O)CC=CCC1 C1(C(=O)NC(CC)C)CCCCCC1N C1(CNC(=O)CC2CC3(CCC3)C2)COCCN(C(C2CC3CCC(C2)O3)=O)C1 c1(C(N2C(C)CC(CNC(c3cncc(N)n3)=O)C2)=O)coc2ccc(Cl)cc12 C1(CNC(C(C)OCC(C)C)=O)CN(C)CCN1C(c1cn2c(n1)CCC2)=O C(=O)(CCC(C)(C)C#N)N1CC(CC(=O)NC(C2CCOC2)C#C)C(C)CC1 c1(NCC(=O)NC2(C)CCN(C(CC3(OC)CCC3)=O)C2)cnc(O)n(C)c1=O C1(C(CO)NC(c2ccccn2)=O)CCN(C(=O)C(F)n2ccnc2)CC1 O=C(CCCCCF)NC1CCN(C(C2Cc3nccn3C2)=O)CC1F N1(C(c2cccc(F)c2Cl)=O)CC2CCN(Cc3cc(Cl)ccc3O)C2C1 C#CCCCC(C)C(=O)N1CC=CCC1C(=O)NCC1CCCO1 C(=O)(C(O)Cc1ccccn1)N(C1CC(NC(=O)C=CC(=O)NC2CC2)C1)C C1(C(N(C)CCc2cnccn2)=O)CN(C(c2ncncc2N)=O)CC12CCC2 C(CCC(C)(C)C(=O)NCC1(C)CC2(CC2)C1)NC(c1c(CC)cc[nH]1)=O C=CC(C(=O)N1CC(O)(C(F)C(=O)NC(CC)C2CC2)C1)OC CC(C)CCCCCC(=O)N1CCC(C)C(CNC(=O)CCc2ccncc2)C1 C1(C(=O)NCC2CCN(C(CCn3c(C)ncc3)=O)C2)CCCC(=O)N1C C1(C#N)(CNC(C2C(NC(C(C3CCC3)OCC)=O)CCCC2)=O)CC(C)(C)C1 N1(C(c2nc(C)sc2)=O)CCC(NC(c2coc(C(F)F)n2)=O)C(F)(F)CC1 c1(C(N2C(CNC(c3cc(COC)cn3C)=O)CCC2)=O)cn2cccnc2n1 c1(N(C)C)ccc2cc(C(N3CCCC(C(=O)NC4CCOC4)C3)=O)ccc2c1 N1(C(CC2CC(CC)C2)=O)CCC(C)(NC(c2sc(C3CC3)nc2C)=O)CC1 Cn1ccc(C(C)(C)C(=O)NCC(C)(C)CNC(c2ccc(Cl)[nH]2)=O)n1 C=C(C)C(CC(=O)NOC(CC(C)C)C(N1CCCC(C)(C)CC1)=O)OC c1(OC)cc(CNC(C2CCN2C(c2ccc(OC)c(N)n2)=O)=O)ccc1O C1CCC2(CC1)CC2.c1(CC)cncc(C(=O)NCC2CC2CNC(=O)C2CC2)c1 Cc1ccc(C(=O)NC2CCC(C)N(C(c3ccc(F)s3)=O)C2)nc1C C1(CNC(c2ccc(Cl)s2)=O)CCN(C(=O)CCCCCF)CC1O c1(C(=O)NCC(CNC(c2cccc(OC)n2)=O)OC)nc2c(s1)CCCC2 C(=O)(CCP(C)(C)=O)N1CC(C)C(CC(=O)NCC(O)C(C)O)C1 N1(C(CSCC)=O)CC(CNC(c2cn(CC(O)CC)nn2)=O)CC1C N1(C(C2C(C(C)C)N(C(=O)CN3CCCC3=O)CC2)=O)CC(N(C)C)C2(CC2)C1 CC1=C(C(=O)N2CCCCC2CCNC(=O)Cc2cn[nH]c2)CCC1 c1(C(=O)NCCN(C(CCOC)=O)C2CC2)cc2c(n1C)CCOC2 c1(C(=O)NCCCOC2CCN(C(CC(C)F)=O)CC2)cnc2sccn12 C(C(CC(C)C)NC(C1(C)CCN(C)C1)=O)NC(CCCOC(C)=O)=O C1(=O)CC(C)N(C)N1CCCN(C)CC(C)(C)C.CC(C)NC CCCC(C#N)C(=O)NCCn1cc(C(=O)N(C2CS(=O)(=O)C23CC3)C)nn1 C1(CC=C)(C(=O)NC(C)C2CC2)CCN(C(c2c[nH]c(C)c2)=O)CC1 c1(C(N2CC3C(NC(C(CCCC)(C)F)=O)C3C2)=O)cc([N+](=O)[O-])ccc1NC CC(C)S(=O)(=O)C(C)C(=O)NC1COC2C(NC(=O)C(O)C(F)(F)F)COC12 C(C(CNC(=O)C=Cc1cn[nH]c1)C(F)(F)F)NC(c1c(C#N)csc1)=O N1(C(CCC(C)(C)OC)=O)CCCC(F)(C(N2CC3C(C)C3C2)=O)C1 c12cn3c(n1)COCC3C(C)=CSC=CC(=O)N(CC(C)O)CCNC2=O C#Cc1ccnc(C(=O)NCC2(NC(=O)C=CC3CCCC3)CCCCC2C)c1 C#CCCCC(C)C(=O)N1CCCC(F)(CNC(C)=O)C1 c1(C(=O)NC2(C)CCN(C(C(CCCC)C)=O)C2)cc(F)cc(C)c1N N1(C(C2(CC)CCN(C(=O)CCc3ccncc3)C2)=O)CC2CSCC2(C)C1 N1(C(CS(=O)(=O)N(CC)CC)=O)CCC(C)(C)C(NC(c2ccnn2C)=O)C1 N1(CCCC)CCOCC1C(=O)NCCCC(C)NC(c1cnoc1C(C)C)=O c1(C2CC(NC(C)=O)C2)cn(CC(N2CC(C)(C(F)F)C2)=O)nn1 C1(CCNC(C2CCCO2)=O)CCCN(C(c2ccc(C(F)(F)F)o2)=O)CC1 c1(OCC2(O)CCN(C(=O)NCc3c(C)cccc3)C2)ccc(F)c(F)c1 Cc1nccc(CNC(C2(CNC(=O)CCCF)CC(C)(C)C2)=O)n1 N1(C(C2N(C(c3c(O)ccc(C)c3)=O)C3C(C2)C3)=O)CC2CCCC(C1)N2C C1(C(=O)NC2CCCN(C(c3cc(C)c(Cl)s3)=O)C2)CCC(C)(F)CC1 C(=O)(C(C)CC(C)C(C)=O)NCc1c(C(=O)NCC(CCCC)O)n(C)nn1 C1(NC(CN(C(C(C)C)=O)C)=O)CCCC(CNC(=O)C(=Cc2cccs2)F)C1 c1(CC)oc(C(N2CCCC2CN(C(=O)C(O)C2CCCC2)C)=O)cc1C N#Cc1c(F)c(NCC2CCCN2CC(F)F)nc(F)c1F CC(C)CC(O)C(=O)N1CC(NC(c2cccc(O)c2Cl)=O)C1 C1(COC)(CNC(C2CC3(CC3)CO2)=O)CCCN1C(=O)C=Cc1cc(C)no1 C#CCCCC(C)C(=O)NC(Cc1cn[nH]c1)C(=O)NCC12COC(C1)C(O)C2 N1(C(c2cncc(C)n2)=O)CCCN(C(C2CC2c2ccncc2)=O)C(C)C1 N1(C(CC(C)OC)=O)CCC2CCCC(C1)N2C(c1ccnn1C)=O N1(C(C2=C(C)OCC2)=O)CCC2(CC1)CN(C(C1CCCC(C)CC1)=O)C2 c1(C(=O)NC(CC(=O)NC)(C)C)cc(C)nc(S(C)(=O)=O)n1 c1(C(N2C(c3c(C)cncc3)CCCC2)=O)nncc2ccccc12 N#Cc1cc(NC(C2CC(F)CN(C(c3cc(I)ccc3Br)=O)C2)=O)ncn1 Cc1nc(N(c2cn(CC3CCN(C(C45CC(C)C4C5)=O)C3)nn2)C)nc(O)c1C CN1CCC2CCN(C(=O)CC(O)CNC(C3CCC4(CCC4)C3)=O)C2C1 Cc1cc(Br)ccc1CN1CCN(CC(=O)Nc2ccnc(Cl)c2C)CC1 N1(C(c2nc(COC)oc2)=O)CCC(C)(NC(C2CCCN2C=O)=O)C1 C(=O)(CCCC(=O)NCCOCCCNC(c1ccc(C2CC2)[nH]1)=O)OCC C(CC(C)(C)C)(C(=O)N(CCCCCC(=O)NCc1cc(C)cc(C)n1)C)OC C(=O)(CC(C)(C)CN(C)C)N1CC(COC)(CNC(=O)C(C)CCOC)C1 C(=O)(C(F)CC(C)(C)NC(C1CCC(=O)CC1)=O)Nc1c(OC)ccc(C)c1 CCCCCC(O)C(=O)NC(CCC(=O)NC1CCC1)C(C)C N1(C(C(C)CC(N)=O)=O)CCC2C(C1)CN2C(c1cc(Cl)cnc1O)=O Cc1cc2occ(C(=O)N(C3CN(C(C4CCNC(=O)C4)=O)C3)C)c2cc1C N1(C(Cc2nnc(C)s2)=O)CC2CN(C(=O)Cc3cc(Cl)ccc3O)CCC12 N1(C(CC2(C=C)CC2)=O)CCCC(C(N2CC(C(C)(O)C(C)C)C2)=O)C1 C1(N(CCC(=O)NCCC2(CC(C)C)CC2)CCOC)CCCC1 C1(CNC(c2ccc(OC)o2)=O)(NC(=O)Cc2ccc(OC)cn2)CCCCCC1 c1(C(C(C)C)C(=O)OCCN(C2CC2)CC2CC2)ncnc2cccc(F)c12 Cc1c(CCC(=O)NC(C)CNC(=O)CC2CCCC2)cccc1Br C1(C(=O)NC2(CCC)CCN(C(C3CCCO3)=O)CC2)CC2(CCOCC2)CO1 C(C(C)(CC(C)C)NC(=O)Cc1cccc(Cl)c1)NC(C(CC)=CC)=O N1(C(c2cnn(C)c2C2CC2)=O)CCN(C(=O)CCOC2CC2)C(C(C)(C)C)C1 N1(C(CC=CCCCCC)=O)CC2CCC(CNC(c3cscc3C)=O)C2C1 C1(C(=O)OC)CN(C(=O)Cn2cc(OC3CCCS3)cn2)CCCN1C(C)=O CC(C)CC(CNC(C1CC12CC2)=O)C(=O)NC1CCn2ncnc2C1 c1(C(=O)NC(C(C)(C)C)c2cccs2)ccc(-n2cccn2)c(F)c1 CC1CC1C1CC1NC(=O)CC(C)(C)NC(=O)C(F)n1ccnc1 c1(C(=O)NCC(CC)NC(C(C)OCCC#C)=O)coc2cc(F)cc(F)c12 CN1CC(C)(C(=O)NCCCCNC(C2C(C(F)F)C2(C)C)=O)CCC1=O C(=O)(CC(C(C)C)NC(=O)Cc1ccoc1)NC(CCC)CCC C1(C(N(CCCC)CCOC)=O)COCC1NC(=O)CSCC(N)=O C1(C2CCN(C(C3CNc4ccnn4C3)=O)C2)(NC(c2n(C)ccc2)=O)CC1 c1(C(N(CCCNC(=O)C(F)CC2CC2)CC)=O)[nH]c2c(C)cccc2c1C c1(CCC)[nH]ccc1C(N1CC(C)(OCC(N2CCC(CC)C2)=O)C1)=O C1(NC(c2ccc(C3CC3)cc2F)=O)CCN(C(=O)C=CCO)CCC1(F)F c1(C(N2C(C)CC(NC(C3(C)C(CC)CCC3)=O)C2)=O)cc(C)ccc1C c1(N(C)CC2N(C(c3c(CC)c(C)sc3)=O)CCC2)ccc(C#N)cn1 c1(C(=O)NCCN(C(=O)C(C)SC)CC)nn(C)cc1Sc1ccccc1 c1(CC(=O)NCC2C(NC(C(C)OCC(F)(F)F)=O)CC2)cn(C)nn1 n1(CC=C)cc(C(=O)NCC(O)C(=O)NCCCC(N)=O)cn1 CC#CCC(C(=O)Nc1csnc1OCC1CC1)NC(=O)Cc1cn(C)nc1C Cc1cc(C)c(C(N2C3CC2CN(C(=O)CC2CCC(F)(F)CO2)C3)=O)cc1C N1(C(CCc2onc(CC)n2)=O)CCCN(C(c2coc3c2COC3)=O)CC1C C1(NC(Cc2c(C)n[nH]c2)=O)CC2CCC1N2C(c1ccc(N)cc1F)=O c1(C(N(CCCOC(=O)COC2(C)COC2)C)=O)cc(O)nc(O)n1 C1(OCC(C)C)CN(C(=O)C(C2CCCCC2)F)CC(C)(C)C1.C12CC1NC2=O N1(C(C(C(C)CNC(C2CC23CCOCC3)=O)F)=O)CC=C(C(C)(C)C)CC1 CC(C)C(C(=O)NCCOCCNC(=O)C(C)c1cccs1)c1cccc(Cl)c1 C1(CNC(C(=Cc2cccnc2)C)=O)CCCCCN1C(C1(F)CCOC1)=O N1(C(CCC(C)O)=O)CCCC12CCN(C(c1cc3ncccc3s1)=O)C2 CCC(C)CCCC(=O)NCC(C)(O)CNC(c1csc(COC)n1)=O C12(NC(Cc3c(C)nc[nH]3)=O)CCN(C(=O)C=Cc3ccn(C)c3)CCC1C2 N1(C(C=C=C(C)C)=O)C2CCC(C2)C1CNC(C1CC(C)(O)C1)=O C1(C(C(=O)N(CC(C)C(=O)NCCc2cncnc2)C)C)CCC(C)(C)O1 c1(C(N2CC(C)C(NC(c3cc(C4CC4)nc(Cl)c3)=O)C2)=O)c[nH]nc1S(N)(=O)=O c1(OC)ccc2cc(CC(=O)NC(CNC(C3CC(C)(C)C3)=O)CO)ccc2c1 CC1(C2CN(C(C3(NC(=O)CC4CCCC5CC45)CC(F)C3)=O)CCO2)N=N1 c1(C(=O)NCCC2(O)CCN(C(c3ccc(OC)nc3)=O)C2)c[nH]cc(C)c1=O c1(C(=O)NCC2(C)CC(NC(c3n(C)ccn3)=O)C2)cnc(O)c(Br)c1 Cc1cccn2nc(C(N3CCCC(C)(NC(c4ncncc4Cl)=O)C3)=O)cc12 c1(CN2CC(C)(C(N3CCOCC3COCCF)=O)C2)cn2ccccc2n1 c1(SC)cc(F)ccc1C(N1CCC(C)(NC(c2csc(CC(F)F)n2)=O)C1)=O CC1Cn2nc(C(N3CCCC(NC(=O)CC4CC=CC4)CC3)=O)cc2C(=O)N1 CN1CCN(C(=O)CCCN=[N+]=[N-])CC1C(=O)NCC1(O)CCCCC1 c1(C(=O)OCC(=O)NCCCC(F)(F)F)ccc2c(n1)COCC2 c1(N2CC(CNC(C=CC=CCC)=O)C2)nnc(Br)s1 c1(C(N2C(C)CCC2C(=O)N(CC(F)(F)CO)C)=O)cncn(C)c1=O C(=O)(C1CCCc2scnc21)NCCCNC(C1N(C)S(=O)(=O)CC1)=O CCC(CC(=O)NCCCOCCC(=O)NCC(=O)NCC(F)F)SC c1(CC)c(C(=O)NCC2CC(C)CCN2C(=O)C=CC(C)C)sc2ccccc12 N1(C(CNC(CC)=O)=O)CC=C(C(=O)NCC2CCOC(CC)C2)C1 N1(C(c2c(CC)nccc2)=O)CCC(NC(c2c(C)ncn2O)=O)C(O)C1 C(=O)(C1=CCCCO1)N1C(C2C3CN(C(C4C5CC(=O)CC54)=O)CC32)CCC1 c1(C(c2nnnn2C2CC2)NC(c2cncn2C)C)ccccc1OC(F)F CC(c1ccccc1)=CC(=O)NC1CCC1CNC(=O)C(C)(C)C Oc1cccc(SCC=Cc2ccc(N3CCOCC3)cc2)c1Br N1(C(c2[nH]cc(C)c2)=O)CC(CO)C2(C1)CN(C(C13CCC(CF)(C1)OC3)=O)C2 C1(NC(C(C=C)O)=O)CN(C(c2cnn(-c3ccncc3)c2)=O)C2CCCCC12 N1(C(CCCc2cn(CC(C)Cc3nc(C)on3)nn2)=O)CCS(=O)CC1C C1(C(N(CC(C)O)CCNC(C2(F)CCOC2)=O)=O)CCCCCCC1 n1(C(C)C)ncc(F)c1C(N1CCC(N(C(=O)CCN2CCCCC2)C)C1)=O N(C(=NCCC(C(F)(F)F)N1CCOCC1)NC1CCCC1)CC(CC)(C)CO c1(C(N2CCC(C)(NC(CN3C(=O)CC(C)(C)O3)=O)C2)=O)cn2ncccc2n1 C1(C(=O)NC2CCC(NC(C3CC=CCO3)=O)C2)(OC)CCCCCC1 N1(C(c2ncn(CC)n2)=O)CC2(CC2)CC1CNC(=O)Cc1c(F)cccc1F C1(CNC(CNC(N)=O)=O)CCCN(C(=O)CCCOc2cccc(Cl)c2)C1 C(=O)(C1CCCc2ccnn21)NC1CN(C(c2n[nH]c(C)c2F)=O)CC1O C(=O)(C(C)S(=O)(=O)C(C)C)NCC(C1CCC1)NC(Cn1ccc(C)cc1=O)=O N1(C(C(CC)CCOC)=O)CC(C)C(NC(C2CCC(C)C2)=O)C(C)C1 C1(CC(=O)NCC2CC23CC3)CCCC1NC(C1(O)CCC1)=O.C(CS)N c1(OC)ccc(F)cc1S(=O)(=O)N1CCC2(CC2C(N2CCC(CO)C2)=O)C1 c1(C(=O)NC(C2CCCN(C(C(C)O)=O)C2)C)cc(F)c(C(F)(F)F)cc1F C=C(C)CCCC(=O)NCCCOCCN(CC)CC.C(COC)O Cc1csc(=O)n1CCC(=O)NCC1CN(C(c2c[nH]nc2C2CC2)=O)CC1C CN1CC(CC(=O)NC(Cc2ccccc2)CCNC(=O)C(C)(C)F)CCC1=O C1(OC)CCC(C)N(N2CCn3ncc(C(=O)N(C4CCCC4)C4CC4)c3C2)C1 N1(C(C(=O)NCC)=O)CC(OC)CC(NC(=O)C=CS(C)=O)C1 C1(OC)CC2CC(NC(C3CCCCC3CNC(=O)C(C)CC#N)=O)CC12 C1(O)(CNC(C2C(C)C2)=O)CCCN(C2CCc3c(F)c(F)c(F)cc32)C1 c1(C(=O)NC2CN(C(C(C)(C)CC#N)=O)CC2(C)C)nc2ccccn2c1F C=CC(C)CC(=O)NC(=O)NC(c1ccccc1)CCC.C1C(=O)OS1 CN1CC(O)CC1C(N1CCC(C)(CNC(=O)CCNS(C)(=O)=O)C1)=O C1(N(C(=O)CC(C)C)CCO)CCN(C(=O)CNCCCCSC)CC1 CC(C)C(C(=O)N1CC(CNC(c2ccoc2)=O)C(O)C1)c1ccccc1 C(C(C)(CC)C(N)=O)C1c2ccc(cc2)-n2nnnc21.C(CC(F)(F)F)N.CC N1(C(c2nc(C)n(C)c2)=O)CC2CC1CN2C(=O)Cn1cccc(O)c1=O N1(C(c2c(C)scc2)=O)CC=CC(C(=O)NCc2ncccn2)C1 c1(C2(NC(=O)NCC(CNS(CC)(=O)=O)C)CCC2)cccnc1 N1(C(C(NC(C(CC=C)NC(C)=O)=O)SC)=O)CC(C(N)=O)C2(CC2)C1 CC(C)C(CO)CCNC(C1(NC(c2ccc(Cl)cc2)=O)CCC1)=O Cc1cccc(C)c1C(=O)NCC1CCCCN1C(c1cc(O)nn1C)=O C(C(=O)N1CCC(C)(NC(c2cnn(CCO)c2)=O)CC1)(C(C)(C)C)N(C)C C1(NC(Cc2occ(C)c2)=O)(CO)CCCN(C(c2ccc(O)c(Cl)n2)=O)C1 C#CCCCCCCC(=O)N1CCN(C(=O)C#CC2CCCOC2)C(C(C)C)C1 Cc1c(C(N2CC=CC2C(=O)N(C)CC2CCC2)=O)ccn1C c1(C(=O)NCCCN(C(=O)CC2CC=CCC2)C)ccsc1Br c1(C(=O)NCC2CN(C(C3CC3(F)F)=O)CCCO2)cc2n(n1)CCCO2 c1(NCCCCCCOC(=O)NC2CC=CC(C)CC2)ccc2c(c1)CCC2 N1(C(CCCCC#C)=O)CC2ON=C(CNC(=O)CN3CCOCC3=O)C2C1 c1(NC(C2N(C(CCSC)=O)CC=C2)=O)cccc(-c2cncnc2)c1 C1(CC)CCN(C(=O)CC#N)C1CNC(=O)CCc1cc(C)[nH]n1 N#Cc1cccc(NC(C2CN(C(c3c(I)ccnc3Cl)=O)CCN2)=O)c1Cl c12sccc1NC2=O.C1(C(N(C(C)C2CC2)C2CC2)=O)CCC1C(N)=O c1(CN2C3CN(C(c4coc(CO)c4)=O)C(C3)C2)cccc2nccnc12 O=C(C1=NOC2COCC12)NC1C=CCN(C(c2ccncc2F)=O)C1 CC(c1ccco1)=CC(=O)Nc1ccc(-c2nnc(Br)o2)cc1 C(=O)(C(C)CC(C)C(C)=O)N1CCC(C(=O)NC(CC(=O)NC)C)CC1C C1(C(=O)NC(C(=O)N(C)CC2CCSCC2)Cc2ccoc2)C(C)(C)C1(C)C CCCC(C)C(=O)NCCCN(C(=O)CC1CCCCC1C)C(C)C C=CC(C)C(=O)N(C)CCN(C(=O)CC1CC(F)C1)C c1(C(=O)NCC(CC)NC(=O)CN2CCCC2CO)cccc(N)c1 S(=O)(=O)(c1ccc(F)cc1)N1C(CC(=O)Nc2[nH]nc(SC)c2C#N)CCC1 N1(C(C2CN(C)CC(C)O2)=O)CCC(C(=O)NC2(CF)CCC2)C(C)(C)C1 n1(CCC)cc(C(=O)N(C)CCN(C)C(c2coc(C)c2)=O)c(C)n1 c1(CSC)cc(C(=O)N(C2CN(C(c3cc(O)nn3C)=O)C2)C)ccc1F N1(C(c2ccc(SC)o2)=O)CC2(CCCCN2C(c2nccn2C)=O)C1 C1(O)(CN(C(C(C=CCCC)O)=O)C)CCN(C(=O)CCc2cn[nH]c2)C1 c1(CC)ccnc(C(=O)NCC2CCCC(CNC(c3nnsc3C)=O)C2)c1 CCCCC(O)CC(=O)NC(C)C(C)(C)C(=O)NCC1(C)CC1(C)C C1(C(=O)NC2C=CC(CNC(c3c(C)csc3)=O)C2)CCCC(=O)N1 c1(C(N2CCC(C3(NC(=O)C(F)(F)CO)CC3)CC2)=O)ncn2cc(Cl)ccc12 c1(CC)c(Cl)nc(C)[nH]c1=NCCCN(C(=O)C(F)(F)c1cnn(C)c1)CC C=CCCCC(C(=O)NCc1ncccc1Cl)NC(c1cc(C)c(C)o1)=O C12(C(N3CC(O)(CN(C)C(C45CC4C5)=O)C3)=O)CCC(=O)N1CCS2 C1(NC(c2cc(C)n(C(C)C)n2)=O)CCN(C(c2cc3[nH]ccc3s2)=O)C(C)C1 N1(C(COCC(=O)OC)=O)CC(CNC(c2cccc(O)n2)=O)OC(C)(C)C1 C1(CN(C(C2C(C)C2)=O)C)CN(C(c2ccnc(NCCO)c2)=O)CCO1 c1(C(=O)NCCC2CCCCC2)sc(Br)cc1F C1(CNC(CCc2ncc(C)[nH]2)=O)CN(C(=O)C(C)NC=O)CC(C)(C)C1 C12(NC(c3cnn(CC)n3)=O)CCCC1N(C(=O)C=Cc1ccccn1)CC2 C1(O)(C(C)NC(C2CCSC2)=O)CN(C(=O)Cc2ccnn2-c2ccccc2)C1 C=C(C)CCCC(=O)NCCC1COCCN1C(c1cn2c(n1)CCC2)=O CC(CC(=O)NC1(C(=O)NCC(C2CC2)N(C)C)CSC1)n1cccc1 c1(-c2cc(CNC(=O)NCCC34CCCC3C4)no2)ccc(Cl)cc1 C1(CNC(C2CCC(C(C)C)CC2)=O)CN(C)CCN1C(C1C2CNC(=O)C12)=O C(=O)(CC(C)CC(=O)NC1CC(NC(=O)CC(F)(F)C(C)C)CC1O)OC c1(C(=O)NCCCC(C)NC(=O)C=Cc2nc[nH]n2)cnc(C(F)F)nc1 Cc1c(Cl)ccnc1C(N1CCC(CNC(C23CCC2C3)=O)CC1)=O N1(C(COC2(C)CCC2)=O)CCN(C(c2cccn3cnnc23)=O)C(CCO)C1 c1(C(=O)NCC(C(C)(C)C)NC(C2CCC3CC2CO3)=O)ncn2c1CCC2 N1(C(c2c(CNC(C3OCCC(C)C3)=O)ocn2)=O)CC2(CCC(=O)N2)C1 c1(C(=O)NC2CCCN(C(C3CC3C3CC3)=O)C2)ccc2c(=O)ccoc2c1 N1(C(C=CCCC(C)C)=O)CCN(C(c2ccc(=N)[nH]c2)=O)C(C2CCC2)C1 Cc1cc(C(=O)NC2CN(C(c3ccc(O)c(Cl)n3)=O)CCC2F)cc(=O)n1C c1(NCC2CCN(C)CC2)ccc(S(=O)(=O)NCCCCC(F)F)cc1C#N N1(C(CNC(C)=O)=O)CCCC(CNC(=O)Cc2sc(C)cc2Br)C1 c1(N2CCC(O)(C)CC2)ncnc2c1ncn2CCC1CCCOC1.FC(F)(F)O Cc1cc2ncn(CC(=O)NC3CC(C)(NC(C4CC4F)=O)C3)c2cc1C C#CCCCC(C)C(=O)NOCC(N1CCC(O)CC1C(=O)OC)=O C(=O)(C(CO)NC(C1(C(=O)CCOCCSC)CC1)=O)OCC.OCC C(=O)(NNC(=O)c1ccnn1C)NC1C(Cc2nc(CC)sc2)COC1 C1(C(C(=O)NCC2(C(=O)OCC)CC2)N(C)CC)CCC(C)CC1.c1cscn1 C1(CN(C(CCc2onc(C(C)C)n2)=O)C)CC(F)CN1C(C1CCOC1C)=O C1(CC=C)(NC(c2cnc(C)nc2C)=O)CCN(C(=O)CCn2cnnn2)CC1 N1(C(Cc2nc(C(C)C)sc2)=O)CC(C)C(C)(CN(C)C)C1 N1(CC(=O)NC(CN(C(c2cnc(C)[nH]2)=O)C)(C)C)C(=O)NC(C)(C2CC2)C1=O C(=O)(CCCCC(=O)NCC1(O)CCCN(C(=O)C(C)NC(C)=O)C1)OC C1(C(C)C)C(=O)NCCN1C(=O)CC1C=CC(NC(C2CCOC2(C)C)=O)C1 c1(NC(C2CC=CCC2)C)ccc(S(=O)(=O)NCCn2cnnn2)cc1Br C1(CCNC(C2(OC)CCCC2)=O)CCN(C(C2CCCOC2C)=O)CC1 C#CCCCC(C)C(=O)NC(C)CC1CCN(C(c2[nH]cc(C)c2C)=O)CC1 c1(C(N2C(CNC(C(N3CC(C)C3)C)=O)CCC2)=O)ccc(SC(F)(F)F)cc1 C(CCNC(=O)CC(C)(F)F)(C(=O)NCC1COCC(C)O1)OC Cc1cc(CN(C(=O)C(c2ccnn2C)N)C2CC2)ccc1Cl N1(C(C(C=C)(F)F)=O)CC(O)(C2(CNC(=O)CN3CCC(OC)C3)CC2)C1 C1(C(=O)NC2(C)CN(C(C(C)(C)c3ncco3)=O)C2)CCCC2(CCCCC2)C1 Cc1scnc1C(=O)NCCOCCCNC(c1cnn(C2CCC2)c1)=O N1(C(C2N(CC)CCC2)=O)CC(CC(N2CC(n3cc(C)cn3)C2)=O)C(C)C1 CC(C)C(C#N)C(=O)N1CCOCC(NC(=O)CCCOc2cccnc2)C1 c1(OCC)ccc(OCc2nc(-c3cncs3)n(CC(F)(F)F)n2)cc1 c1(C(=O)NCC(CCCC)NC(=O)COCC)cc2c(cnn2C)nc1C N1(C(CN(C)C)=O)CCN(C(C2CN(C3CCC3)C2)=O)CC(C)(F)C1 C1(CNC(c2c(C)cc(F)s2)=O)CC(C)(C)CN1C(C1CCC(F)(F)CC1)=O c1(C(=O)NC2(CC)CCN(C(C3CC3CF)=O)CC2)cnc2scc(C)n12 C1(c2ccccc2)(C(=O)NC2CC(NC(CP(C)(C)=O)=O)C2)CC2CCC1C2 C1(CNC(c2c(C)ocn2)=O)CCC(Cn2cc(CC(O)C3CC3)nn2)CC1 N1(C(C#CC(C)C)=O)CC(CO)C2(C1)CN(C(=O)CCCc1cccnc1)C2 CC(C)C(O)C(C)C(=O)NCC1(F)CCCN(C(=O)COCCCF)C1 c1(C(=O)NCC(C)(C2CC2)NC(C2CC(C)(F)C2)=O)cscc1-c1ccccc1 c1(C(C(=O)NC2CCOCC2)N(CC(F)F)CCC)cnc(-c2ccccc2)s1 c1(CCO)nnc(Cc2onc(C(C)C)n2)o1.C1(COC2CC2)CC1.OCO C123CCC1CN(C2)C(=O)C(O)CNCCNC(=O)C3.C(CF)OC(=O)C1CC1 c1(CSC)cc(C(=O)NCC(C)CN(C)C(C2(C#N)CC23CCC3)=O)ccc1F c1(C(=O)NCC(C2CCC2)NC(c2cc(Cl)ccc2F)=O)ccccc1[N+](=O)[O-] N1(C(CCN(C2CCOCC2NC)c2ccccn2)=O)CCc2sccc2C1.CO N1(C(CCC)=O)CC2(C1)CN(C(c1ccc(N3CCCC3)nc1)=O)CC2CO N1(C(C)=O)CCCC(C2CN(C(c3cc(C)c(Br)cc3Cl)=O)C2)C1 C1(CCNC(=O)CNC(N)=O)(OC)CCN(C(C2CN(C)CCO2)=O)C1 CN1CC(O)CCC1C(=O)NCC1CCC(C(=O)NCC2C=CCC2)CC1 N1(C(C(C)OCCN(C)C)=O)CCCC1c1cn(CCN(C)C2CC2)nn1 N1(C(C(C)CC2CCCCC2)=O)CCC(F)(F)CC(C)C1 c1(C(=O)NC2C=CC(C(=O)Nc3onc(C)c3C)C2)cc(Br)ccc1C#N C(=O)(C(CC)C(=O)NCCC(O)CNC(c1ccc(CF)cc1)=O)OCC C(=O)(CN=C(NCC(C)(C)C(F)(F)F)NCC1(N(C)C)CCC1)N(C)C C1(CCNC(c2nnn(CC)c2C)=O)CCN(C(c2ccccc2F)=O)C(C)C1 N1(C(C2SCC(=O)C2)=O)CCC(C(=O)NCc2ccc[n+]([O-])c2)C(O)C1 C(=O)(C1CCCc2nccn21)NCCN(C(c1cc(-c2cccs2)on1)=O)CC C(=O)(CCCn1cc(C(=O)NC(c2ccccn2)C)nn1)OC(C)=O C1(C(=O)N(CC(C)NC(=O)C(c2ccc(Cl)s2)=O)C)(OC)CCSCC1 N1(C(C2CCC(=O)O2)=O)CCCC2(NC(C3CC4CC3C3CC43)=O)CC2C1 Cc1cc(F)ncc1-c1cn(CCN(C(=O)C(C)OCCN(C)C)C2CC2)nn1 C1(NC(C(Cc2c(C)nc[nH]2)O)=O)CCN(C(C2CN(C(N)=O)C2)=O)CC1C C12(CN3CCN(c4nc(SC)nc(C(F)(F)F)c4)CC3)CCCCCC1OCC2 c1(C(N(C2CN(C(CC3(C=C)CCC3)=O)C2)C)=O)cc2c(F)cc(Cl)cc2[nH]1 c1(CN2CCC(CNC(=O)CCC(F)(F)F)CC2)ccc2ccsc2c1 C(=O)(N=c1ccn(Cc2ccccc2)[nH]1)N(CC)Cc1ccc(C)cc1C N1(C(c2c(C)nc(CC)o2)=O)CC2CC(NC(c3ccnc(F)c3N)=O)C(C2)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])N1CC(CC)N(C(c2ccn(C3CCC3)n2)=O)CC1 C1(NC(CCC(C)C)c2nnnn2Cc2cccs2)COC2(CCC2)C1 CS(=O)CCC(O)C(=O)NCC1(F)CC(CNC(=O)C=CBr)C1 C1(NC(C2OCCN(C(C)C)C2)=O)CCC2(CC1)CN(C(=O)C(C)CF)CCO2 C(=O)(C(C)C(F)F)NCCOCCC(=O)NCCCOCC=C c1(NC(C(=O)NC2CCC(CCNC)C2)=O)ccc(OC)c(OC)c1 N1(C(C2CC3(C2)CC3CC)=O)CC(C(N2CCOCC3(CC3)C2)=O)C2(CCC2)C1 N(C1CCc2ccccc21)C(C1(C)N(Cc2c(C)nc(C)s2)CCC1)=O c1(CN(C(Cc2cccs2)CO)C=O)cc(C2CCCCC2)cc(Cl)c1O N1(C(CSCCCC)=O)CCC(F)(CNC(c2sccc2CNC(C)=O)=O)CC1 Cc1cc(Cl)cc(C(N2CCN(C(=O)CC34COCC(C3)C4)CC2C)=O)c1O C(c1c(Cl)cccc1Cl)=C(C(N1CCC(NC(C(COC)COC)=O)C1)=O)C C12(C(N3CC(CO)C3)=O)CCC(CO)(CC1)CC2.c12cccc(c1)Cn1cc-2nn1 N1(C(C(C)NS(CC)(=O)=O)=O)CCC(CNC(=O)CN(C)CCO)C1(C)C c1(CNC(CCN(CC#C)C(C2CCC(C)(CC)O2)=O)=O)ccc(Cl)cc1 N1(C(c2c(CC)noc2)=O)CCCC2(CCC(NC(C34CC5CC3C4C5)=O)C2)C1 C1(CNC(CCC(=O)NCCC)=O)CC2CCC1N(C(c1cc(C)c(C)s1)=O)C2 c1(C(=O)NCC2(O)CCN(C(C3(C)CCCS3)=O)C2)ccc(Br)c(F)c1 c1(CCC(=O)NCC(=O)NCc2cn(CCN)nn2)nc2ccccc2s1 c1(NC(C(CCC=C)NC(c2ccoc2)=O)=O)cc(C)c(F)cc1F N1(C(C2(OC)CCCC2)=O)CC(N(C(=O)Cn2cc(C(C)O)nn2)C)C(O)C1 c1(CC)cc(CC(=O)NCC2CC(O)CN2C(=O)C=CC(C)(C)C)n(C)n1 C1(C(N2Cc3ccccc3C2)=O)C2CC(CC2F)N1C(c1cnnc(O)c1)=O C(=O)(C(F)C(F)(F)F)N1CCC(NC(C2CC(C)(F)C2)=O)C1 N(C1c2cc(C)ccc2CC1C)C(=O)NCc1nnc(COC)s1 C(=O)(CC(C(C)C)C(C)C)NCCC1OCCN(C(C(F)OC)=O)C1 N1(C(CNS(C)(=O)=O)=O)CCC2(CCCCN(C(=O)CNC(N)=O)C2)C1 C=CC(C)C(C)C(=O)N(C1CCCC1)CCNC(=O)C=Cc1sccc1C c1(CC(=O)NC2CC3CC(NC(C(C=CC)O)=O)C2C3)c[nH]c2cccc(C)c12 N1(C(Cc2nc(C)sc2C)=O)CC2CCC1C1CN(C(=O)C#CC3CC3)CC21 c1(C(c2nnnn2C2CC2)OC)cc(OC)n[nH]1.C1CN1C(C)C.CO C1(C)(C(=O)NC(CNC(c2c(C(C)C)occ2)=O)C2CCC2)CCCOC1 CC(C)C(C)C(=O)N1CCC1C(=O)NCCCC(O)CO N#Cc1ccc(N2CCC(CNC(=O)CCC3CC3)C2)cn1 c1(OCC)ccnc(N(C2CNCC2C#N)Cc2ccc(OC(F)F)cc2)n1 CC1CCC(CCN(C(=O)Cn2cccnc2=O)C)CC1.N12CCCC1CC2 c1(CNc2c(C)c(NC3CCC(C)CC3C)ncn2)n[nH]c2c1CCCC2 N1(C(C(C(C)C)N(C)C)=O)CCC2C1CCCN2C(=O)CS(N)(=O)=O n1(CC(=O)NC2CCC(CNC(C3OCC(C)(C)C3)=O)C2)cnc([N+](=O)[O-])c1 c1(CNC(N(C(C(F)(F)F)C(F)(F)F)C)=O)c(F)cc(Cl)cc1F N1(C(C2CCCC2)=O)CC(=O)NC2CN(C=O)CCC12.CCC(CC)C1CCC1 N1(C(Cc2cc(C)nn2C)=O)CCC(NC(=O)C=CC2CCCO2)C12CC2 CC(C)(C)CC(O)CC(=O)NCC(O)CNC(=O)Cc1ccc(C(N)=O)cc1 C1(CNC(C2(CC=C)CN(C(=O)CC(C)C)C2)=O)CCCN1C(=O)CN.C#CCO C(C(C)(C(=O)NC1CN(C(=O)CCF)CC1C(F)(F)F)OC)OC S(=O)(=O)(c1cccc(Br)c1F)N1CCC2CN(C(C=CC)=O)CC2C1 c1(C(=O)NCC(C)CNC(C2CN(C)C2)=O)nc(C2CC2)n2ccccc12 c1(C(N(C2CCN(C(COCC)=O)CC2)CC2CC2)=O)cc2ccccn2c1 C1(CC(=O)Nc2ccc(Cl)s2)CC2(C1)CN(C(c1ccnc(OCCO)c1)=O)C2 N1(C(C(CC)SC)=O)CCC(CNC(=O)C=CC(N)=O)(OC)C1 c1(OC)ccc(C(N2CCCC(c3cn(C4CCOC4)nn3)C2)=O)cc1 C1(C(N2CCC(NC(c3ccc(O)nc3Cl)=O)C(F)C2)=O)Cc2cccnc2C1 N1(C(C(=O)N(CC(C)C)CC2ON=C(C)C2)=O)CCCC2N(CCOC2)C1 c1(C(N2CCN(C(CCSCC)=O)CC23CC3)=O)c[nH]c2ccc(O)cc12 C(=O)(CCCOC)NCCN(C1CS(=O)(=O)C1)CCC C(C(=O)N1CC(O)CC1C(=O)NCCC1CC2CC2C1)(C(C)C)N(CC)CC CC(O)CC(=O)NCC(O)CCNC(=O)CC1CCSC1 c1(CC(=O)OC)ccc(NC(C2CSCCN2C(=O)C=Cc2ccsc2)=O)cc1 C=Cc1nc(NC(c2nc(C(C)(C)C)ns2)=O)n(C)n1 c1(NC)c(C(=O)NC2CC(NC(C3CCCS3(=O)=O)=O)C2)sc2nccnc12 c1(C(=O)NCC(C)CN(C(=O)C(C)(C)C)C)nccc2ccccc12 CCC(C)(CNC(c1cccc(F)c1Br)CO)C(C)O CN1CCCCN(C(=O)C(C2CC2)N(C)C(C2CC23CCC3)=O)CC1 c1(NC)cnc(C(C)C)nc1C(=O)NCCCN(c1ncn(C)n1)C C(c1ccccc1)=C(C(=O)N(CCCNC(CCC=C(C)C)=O)C1CC1)C C1(C(=O)NC2(C)CN(C(C3CC4(CSC4)C3)=O)C2)CC(c2ccccc2)=NO1 c1(CC(=O)NC2C(NC(CCC3CC(OC)C3)=O)COC2)cn2cc(C)sc2n1 CC(C)CC(CNC(=O)Cn1cccn1)NC(C1C(C=C(C)C)C1(C)C)=O N1(C(CCCN(C(C)=O)C)=O)CCN(C(C2CS(=O)(=O)C2)=O)CC1C C1(C(N)=O)CC(F)CN1C(c1cc(CC2CC2)on1)=O C1(CCOC)(NC(=O)CCC(F)F)CCN(C(c2cc(C(C)=O)cs2)=O)C1 C(=O)(C1CCCc2ccnn21)NCCOC(CNC(CC)=O)(C)C C#Cc1cccc(C(=O)NC(C(=O)NCc2cccnc2)c2ccco2)c1C C(=O)(CCS(N)(=O)=O)N1CC(CCC)C(NC2CCCCC2c2cn(C)nn2)C1 N1(C(C)CNC(C23CC(n4cc(C5CC5CO)nn4)C2C3)=O)C(=O)CCC1=O N1(CC)CCC(C(=O)NCC(O)CNC(=O)CCc2nc(C(C)C)no2)CC1 C1(NC(CCC2CC(CNC(CCc3n(C)ncn3)=O)OC2)=O)CCCC12CC2 C(CCCCC(=O)NC(C1(O)CN(C(c2scnc2CC)=O)C1)C)=CC CC(C(=O)NCC1(F)CCCN(C(=O)Cc2cccc(CO)c2)C1)C1=CCCC1 CCCC(O)(CCC)CC(=O)N1CCCC1Cc1ccc(F)cc1 c1(NC(CC2N(Cc3cc(C)nn3C)CCC2)=O)cc(F)cc(Br)c1 S(=O)(=O)(c1ccc(NCCCC2CCC2)c(F)c1)NCC(CCCCC)O CC1=C(C(=O)N2CCC(O)(c3cn(Cc4ncon4)nn3)CC2)CCCO1 N1(C(C(C)OCC#C)=O)CCC(C)CC1CNC(=O)CCCOCC C1(CC(N2CC(OCC)(CN)C2)=O)CC2(C1)CC1(CC(F)(F)C1)C2 C1(CNC(C2(C=C)CC2)=O)CC12CCN(C(c1cnn(CC)c1C)=O)CC2 C1(CNC(=O)CN2CCCC2=O)CCN(C(c2nnc(O)cc2O)=O)CC1(F)F c1(-c2c(C(N3CC(C)NC(=O)C3)=O)sc3c2CCC3)ccc2nc(O)[nH]c2c1 c1(CC=C)cccc(NC(C(=O)NCC)C2CC2)c1.C(=O)(C=C(C)C)N C(CC(=O)N1CCC(N2CCC2)C1)(C(F)F)NC(C=NOC)=O C(=O)(C(O)CCC(C)C)N1C(C(=O)NC(CC)C)C(C)(C)CC1 C1(NC(=O)CCC2CC2)CC2CN(C(c3cccc(CO)n3)=O)CC2C1 C(=O)(CCCCC(C)(C)C#N)NCC1C(NC(CC2N(CC)CCOC2)=O)CC1 C12(NC(=O)CSC(F)F)COCCC1CN(C(c1cc3c(s1)CCSC3)=O)C2 c1(NC(C2N(Cc3cc(C)c(F)cc3)CCNC2)=O)cc([N+](=O)[O-])cnc1C N1(C(c2n(C)ncc2)=O)CCCC(NC(c2ccnc(C3CCCC3)n2)=O)CC1 C1(NC(Cc2nc(=N)[nH][nH]2)=O)CC2CCC(C1)N2C(C1CC1(F)F)=O N1(C(C(C)=C2CC2)=O)CC(CNC(=O)CS(N)(=O)=O)C(F)(F)C1 C(CNC(C1(C)CCCS1)=O)(CC(C)C)NC(c1c(CC)non1)=O CC1C(C)CCC1C(=O)N(CCC(O)c1cccs1)C C(C(COC)CC(=O)NC(C)CN(C(c1ncccc1OC)=O)CC)OC C1(C(=O)NCc2cn(CC(=O)N(C)CC3CC(O)C3)nn2)COCC1(C)C C#CC1(C(N2CCCCC(NC(c3ncc(N)cc3C)=O)C2)=O)CCOCC1 C#CC(C)(C)C(=O)N1CCC(NC(=O)CNC(C)=O)C1 c1(CS(N2CCC3(C(C(N(C4CCC4)C)=O)C3)C2)(=O)=O)cc2ccccc2[nH]1 C1(C(N(C(C(=O)NCC(n2cccn2)C)C)C)=O)CN2CCC1C2 Cc1ccc(C(=O)NCCN2CCC(CN(C)C)CC2)c(OCC(C)C)c1 N1(C(C(=O)NC(CC)(C)C)C)CCC(NC(c2cc(C3CC3)no2)=O)C(C)(C)C1 c1(C(N2C(C(=O)Nc3cccc(C(C)F)c3)CC(C)C2)=O)ccc(Br)cc1I C(=O)(C1CCCn2ccnc21)N1CCOCC(NC(C(NOC)=O)=O)C1 N1(C(Cc2cc(COC)on2)=O)CCC(C)(CNC(c2ccnn2C(F)F)=O)C1 c1(C(N(C2CCCN(C(C3CCSC3)=O)C2)C)=O)c[nH]c2nc(Cl)ccc12 c1(CNC(c2cccc(CS(=O)(=O)CC)c2)=O)noc2c1CCC2 c1(C(=O)NCC2(CO)CCN(C(c3c(CC)ncs3)=O)C2)c(F)cc(O)cc1F N1(C(c2cc(C)n(C)c2)=O)CC2CCN(C(c3cc[nH]c(=N)c3Cl)=O)C2C1 Cc1cc(C(=O)NC2COCC2NC(C2CC(=O)N(C)C(=O)N2)=O)c(N)c(F)c1 C#CC1CCCC(CNC(=O)C(CC2CCCC2)NC(c2cc(Cl)ns2)=O)C1 c1(N(C)Cc2ccc(CC(=O)OC)cc2)c(Cl)cnc2[nH]nnc12 N1(C(c2c(N)non2)=O)CC2(C1)CN(C(C1CC1(Br)Br)=O)C2 N1(C(CSCCC)=O)CCN(C(=O)Cc2cocn2)C(C)C1C CC1(C(=O)Nc2cc3ccc(Br)cc3o2)CC12CCN(C(C1C3CCC13)=O)CC2 CCCC(O)C(=O)NCC(C1CC1)NC(c1[nH]ccc1-c1ccccc1)=O C=CCC(CCCCC)C(=O)N(CCCNC(=O)CCNC(=O)NCCC)C Cc1cc(C)c(CN2CC3CC2C3C(=O)N(C)OC)[nH]1 N1(C(CC2N(C(C3=NOC(C)C3)=O)CC2)=O)CCCC(F)(F)CC1 c1(C(=O)NC2CC(NC(=O)CCC(F)F)CC2O)cc(Br)cn2ccnc12 C(=O)(CC1=Cc2ccccc2C1)OCCC(CCC)CCC C(=O)(C(C)CC(C)(C)C)NC1C(C)CCN(C(c2cncc(Cl)c2Cl)=O)C1 C1(CC(=O)N(CC(=O)NC(CC=C)CO)CCOC)CCCC(=O)C1 Cc1cc(C(N2CCCC2C2CCN(C(=O)CSc3nc[nH]n3)C2)=O)cc(O)n1 C(=O)(C(C)(C)C(=O)N1CC(N2CCN(C(C)=O)CC2)C1)OCC.C(=O)N C(c1ccc(F)c(F)c1)=CC(=O)NC1C2CCN(C(CNC(N)=O)=O)C21 C(=O)(CC(CN(C)C)C(F)(F)F)NCC(C)(C)NC(COCCCCC)=O C1(c2cccc(F)c2)(NC(=O)NC(c2cccnc2)C2CCC2)CCOCC1 C1(C(N(CCCOCCN(C)C(C2(C)CCC(=O)N2)=O)C)=O)CCC(C)(F)CC1 Cc1cc(C)n(CC(N2CCC(CNC(c3cc(Br)c(C)s3)=O)C2)=O)n1 c1(C(=O)NCC(CNC(CCN(CCC)C)=O)C)cnc[nH]c1=N Cc1cc(C(N2CCC(OCC(=O)NCC3(O)CCN(C)C3)C2)=O)nn1C c1(C(=O)NCC(C)CNC(c2c[nH]nc2C(F)(F)F)=O)cc(Cl)ccn1 N1(C(C2C(=C)C2)=O)CCN(C)CC1CN(C(=O)CNC(=O)CCC)CC c1(C(=O)NC2(COC)CN(C(=O)CC3OCCC3C)C2)cccn2c(C)nnc12 N1(C(CSc2c(C)n[nH]c2C)=O)CCC(C)CC1CNC(=O)C(F)CC1CCC1 C1(CNC(COCCOCC#C)=O)COCCN1C(=O)C(C)SC CCC(C)C(O)CC(=O)N(C)CC1CCN(C(C2CCCN(CC)C2)=O)C1 c1(C(=O)NC(C(C)NC(C2ON=C(C)C2)=O)CO)cc(OC(F)F)cc(F)c1 C(C)(CC(F)(F)F)NC(c1n(CC=C)nnn1)c1ccncc1 C1(CC=C)(NC(C2(c3nocc3C)CC2)=O)CCN(C(=O)CCC2CCCO2)C1 C(=O)(CCC1=NNC(=O)CC1)N1CC2(OCC(NC(C3(OCC)CC3)=O)C2)C1 C(CCCCC(=O)NCc1cn(C2CN(C(=O)C(C)CF)C2)nn1)=CCCC c1(C(=O)NC2CCC(NC(C3(F)CC=CCC3)=O)C2)cc2c(cn1)OCCO2 c1(C(N2CC(C(=O)OC)C(O)C2)=O)cc(C)c(I)cc1C Cc1cc(Cl)ncc1CC(=O)NC1CCC(NC(=O)CC(C)(F)F)CC1 C1(C(=O)NCC2(NC(=O)CCC(=O)Nc3nccs3)CCCC2)CCCS1(=O)=O C1(C(=O)NCCC(C)(C)O)CN(C(=O)C(F)C(C)(F)F)CC12CC2 Cc1nn(C)cc1C(C)NC(=O)C(c1ccccc1)N(C)C C(=O)(CS(=O)(=O)CC(=O)N1CCCC1CCNC(C1COC2(CCC2)C1)=O)OC N1(C(CC(C)OC)=O)CC(Nc2ncc([N+](=O)[O-])cc2Cl)C2(CSCC2)C1 C1(C(C)(C)C)(CNC(CN2C(C)CCC2)=O)CCN(C(C2(F)CCCC2)=O)C1 Cc1ncnc(C)c1C(=O)NCC12CC(NC(c3snc(O)c3Cl)=O)(CO1)C2 C#CCC(C(=O)Nc1cnn(CC(C)C)c1)NC(=O)CCc1cscn1 C1(CNC(C2C(C=C)C2)=O)C(O)C(O)CN1C(c1sc(C)cc1Br)=O C(C(=O)Nn1cccn1)C1(C)CN(C(CC2C(C)CCC2)=O)C1 C(CCC(=O)NC(C)C(C)=O)OCCN.n12cc(nn1)C2 c1(C(N(C2CCCC2)CCNC(=O)CC23CCCC2C3)=O)ccc(CO)cc1F c1(OC)cc([N+](=O)[O-])ccc1C(=O)NCC(C)CNC(C1CC(C(F)F)C1)=O C(=O)(C(CCC)NC(=O)CC1CCC(C)(C)O1)N(CCOCC#C)C c1(C(C(=O)NCC(C(C)C)NC(C2CCC3CC3CC2)=O)C)ccc(F)cc1F c1(C(=O)NCCNC(CC2CC(C)(C)OC2)=O)ccc(OC(F)F)cc1F c1(C(=O)NCC2CCCC2NC(C2(O)CC(F)(F)C2)=O)ncc[nH]c1=O C(=O)(C1(C)CCc2ccccc21)NCC1N(C(CCCOCCC)=O)CCC1 Cc1cc(C(=O)NC(C)CCCNC(c2nsnc2O)=O)ccc1O N1(C(=O)C=NOC2CCCCO2)CC2(C1)CN(C(c1ccnn1C(F)F)=O)C2 Cc1ncccc1CC(=O)NCC1CC1CNC(=O)CCCCN(C)C C1(C(=O)NCC(C(C)C)NC(=O)CCc2cnccn2)CCn2c(O)nnc2C1 N1(C(CC(CC)N(C(=O)COc2ccccc2)C)=O)CCCC(C)(O)C1 c1(CC)nc(C)c(C(=O)N(C2CCN(C(c3cc(Cl)c(Cl)s3)=O)C2)C)o1 N1(C(C(C)(C)NC(=O)OC(C)(C)C)=O)C=COCC1c1ccccn1 CC(C)(C)CCCC(=O)NC1CC(NC(C2CCOC(=O)N2)=O)C1 C1(CNC(C(C)O)=O)CCC(CN(C)C(C2(Cc3cnn[nH]3)CCC2)=O)CC1 CCCC(C)(CCC)C(=O)NCCC1(O)CCN(C(C2CC2c2cccs2)=O)C1 C(=O)(C(C)(C)CCC(=O)OC)N1CCCC(CNC(CCSCCCC)=O)C1 N1(C(=O)C=CI)CCC(C2CCCN(C(C3Cc4c[nH]cc4S3(=O)=O)=O)C2)C1 c1(CC(=O)NCC(CN(C)C(c2cc[nH]c(=N)c2)=O)O)ccc(Cl)c([N+](=O)[O-])c1 c1(CNC(C(=O)Nc2ccc(CCC)cc2)=O)cccc(F)c1F CCCC(C(=O)N1CCOCC(C(=O)NCc2cnc(CC)[nH]2)C1)C(C)C CCCCCCCC(=O)NCC(CC(=O)Nc1cc(C)cc(C)c1)C1CCC1 C1(F)(CNC(c2c(C(C)C)occ2)=O)CCN(C(C2CC2C)=O)C1 CCC(C)(C(=O)NCC(C(=O)NCCCCCOC)N(C)C)OC C1(O)(CNC(CN2CCN(C)CC2)=O)CCN(C(C2CCCC(C)CC2)=O)CC1 C1(C(N2C(CN(C(C(CC)SC)=O)C3CC3)CCC2)=O)CC(O)(C#N)C1 CCCCC(CC)C(=O)N1CCCN(C(c2cnc(OC)s2)=O)CC1 CC(CCNC(C1CCCCN1C(c1ccn(C)c1)=O)=O)C(F)F C(C(F)(C(=O)N1CCN(CC(=O)NC)CC1C)C(C)C)NC(CC)=O C(=O)(C1CCc2c(Cl)cccc21)NCC(CC)NC(=O)CCC12CCC(CC1)C2 n1(CC(=O)NC2CC(C)(CNC(C3CCN(CC)CC3)=O)C2)cccc(O)c1=O c1(OC)cccc2c(CNC3CCC(CN=c4cc(CO)nc[nH]4)C3)n[nH]c12 c1(C(=O)NCC2OCCC(NC(C3C(C)(C(F)F)C3)=O)C2)ccc2c(n1)CCC2 c1(CNC(c2ccc(C(F)F)cc2)=O)ccc(OC2CCOC2)c(Cl)c1 c1(NC(C2CCN(C(c3cc(C4CC4)on3)=O)CC2O)=O)cccc2occc12 c1(COC)csc(CNCc2ncoc2C2CC2)c1 CN(CCCC(=O)NC(C1CCOC1)CNC(c1n[nH]c2c1COCC2)=O)N=O C1(C(=O)NC(CC#C)C(N)=O)CCCCCN1C(=O)CC1(O)CCC1 Cc1sc(O)nc1C(=O)NC(C)CN(C)C(c1cncc(-n2cccn2)n1)=O c1(C(N2CCC(n3cc(C4C5COCC45)nn3)C2)=O)nnc2n1CCCCC2 c1(CC)cc(OC)ccc1C(N1CCCC1C(C)NC(=O)C1=CCC1)=O CC1CN(C(=O)C(c2cn[nH]c2)N(C(c2nccs2)=O)CCO)CCC1N(C)C CC1(C)CCCCC1C(=O)NC1CC(C(=O)NOCC2CCC2)C1 c1(CCCC)ccccc1Cc1nc(CCC2CCCC2)nn1-c1ccnn1C N1(C(C2C(C)CC(=O)N2)=O)CC2(CC(NC(=O)C(c3ccccc3)F)CO2)C1 N1(C(=O)C2=COCCO2)CCCC12CCN(C(C1(C(F)F)CC1(F)F)=O)C2 c1(C(=O)NCC2C(C)CCCN2C(=O)CCCC2CCC2)ccc(C#N)cc1F C1(C(=O)NCCS(=O)(=O)NC)CCCN(C(=O)CCCC2CC2)CC1 CC(=O)CCN=C(NCc1ccc(C)cc1C)NCc1cccc(S(C)(=O)=O)c1 c1(C(=O)NCC(c2cccc(F)c2)OC)cccc(C2(F)CC2(F)F)c1 N1(C(C2(C)CC(=C)C2)=O)CCCC(NC(=O)CCN(CC(F)(F)F)C)C(F)C1 c1(NC(c2nnnn2C2CCOC2)C2(COC)COC2)c(SC)cccc1OC.C1CC1 N1(C(C2C(C#N)C2)=O)Cc2ccnn2CC(NC(c2cc(C(F)(F)F)c[nH]2)=O)C1 N1(C(Cc2cc(C)cc(F)c2)=O)CCC(NC(c2cnsc2)=O)CC(C)(C)C1 c1(-n2c(C)ncc2)ncccc1C(=O)NC1(C)CC(NC(=O)C=C2CCC2)C1 C(=O)(CS(=O)(=O)CC(C)C)NCCCNC(C1(C)N(CC)CCC1)=O C(CC1CCCCN1C(=O)C(N)=O)(C(F)(F)F)NC(CC1(C)OCCO1)=O.C(CSC)O C#Cc1ccc(C(=O)NC2CC(CC(N3CC=CC3(C)COC)=O)C2(C)C)cn1 N1(C(C2CC(NC(=O)CC3CCCC(O)C3)C2)=O)CCC2OCCC2C1 c1(C(N2CCC(C(C#C)C)CC2)C(=O)NCC)cc(C)c(OC)c(C)c1 C1(NC(CN2CC(C)C2)=O)CN(C(c2cc3c(F)cccc3[nH]2)=O)C2(CCCC2)C1 C1(C)(C(N(C)CC2CCCC(NC(COC(C)C)=O)C2)=O)CC2CCC1O2 C1(CC(=O)NCC2C(NC(C3(C(C)(F)F)CCC3)=O)C2)C2CC3C(C2)C13 CS(=O)(=O)C(CNC(C1C2CC3C(C2)C13)=O)CNC(C1(C(F)F)CCCCC1)=O c1(CCC(=O)N(CC(=O)NCC(C=C)O)CC)cc(C)[nH]n1 N1(C(C2(CC#C)CCCC2)=O)CCN(C(C2OCC2(C)C)=O)C(C2CC2)C1 N1(C(C2CCOC2)=O)CC2(CCN(Cc3cccnc3Cl)C2)C1 C12CC(CCO1)NC2.c1(N(c2ccccc2)C(C(F)F)C2CC2)ccccc1S C(C(C)C(=O)N1CCC(CCNC(c2csc(C(F)(F)C(F)(F)F)c2)=O)C1)SC CON1CC(C(N2CCC(C)(CSc3ccccc3OCC)C2)=O)CC1=O CCCCC(C)C(=O)NCC(C)(C)CN(C(c1cn(C)c(C)n1)=O)CC CCC(C)(CCNC(=O)C=CBr)NC(=O)C=Cc1cn(C)cn1 C1(CC#C)CN(C(=O)NCc2cc(C(=O)OC)c(C)s2)CCO1 c1(CC(=O)OC)ccc(C(=O)NCC2CCN(C(C3CSCCS3)=O)C2)c(OC)c1 N1(C(C2CN(C(CCCCC(C)C)=O)CC2C2CC2)=O)CCCC2NC(=O)CC12 N1(C(c2nn(CC)nc2C)=O)CC(C)OC2(CCN(C(=O)CCS(C)(=O)=O)C2)C1 N1(C(C(CC)C)=O)CC2(CC(C(=O)Nc3csc(C)c3C)CO2)C1 C1(NC(c2cc(CC)[nH]n2)=O)CCCC(CN(C)C(C2(C3CC3)CC2)=O)C1 c1(OC)c(Cl)cc(C(=O)N(CC(C)N(C)C(c2cnc(C)cn2)=O)C)cc1Cl CCC(CCCC(=O)N1CCS(=O)C(C)C1)NC(=O)Cc1n[nH]c(C)n1 N1(C(C=C(CC)CC)=O)CCCN(C(c2cc(C(N)=O)cn2C)=O)C(C)C1 c1(C(N2CC(NC(c3ccnc(F)c3)=O)C3(C2)CC3)=O)cc(F)c(F)cc1Cl N1(C(=O)NCC2CCC(C)CC2)CC=CCC2(CCOCC2)C1 N1(C(C)=O)CCC(C(=O)NC2(CNC(c3coc(C4CCCC4)n3)=O)CCC2)C1 C=C(C)CCC(C(=O)NC1CC1)N1CCCN(CC(O)CO)CC1 N1(C(CN(CCC)C)=O)CCCCCC1C(N1CC(O)C(O)C1)=O N1(c2ccnc(N(CCC(C(C)C)C)C3CCCC3)n2)CCC(O)C(F)C1 C(=O)(N1CCC(C(=O)Nc2ccccc2Cl)O1)C1C(C)SCCC1 C1(C(C2CC(C)CN(C(=O)COC3CCCCC3)C2)=O)COc2ccccc2O1 c1(C(N2C(CCNC(C3(OC)CC3)=O)CC(OC)C2)=O)cncc(S(C)(=O)=O)c1 C(C(CC(C)C)NC(C1CCC(C(C)(C)O)CC1)=O)NC(C(F)OC)=O Cc1cc(F)ncc1C(N1CC2CC(NC(C3CCC4(CCC4)O3)=O)C2C1)=O C1(C(=O)OCC(C)CN(C)C)(NC(=O)OC(C)(C)C)CCSC1 C(=O)(CCC(=O)NCC1(CCNC(c2ccncc2N(C)C)=O)CC1)NC C1(c2ccccc2)(NC(=O)C(C)CSC)CCN(C(C2(SC)CC2)=O)C1.C=CC N1(C(c2scc(C(=O)Nc3c(OC)cc(Br)cn3)n2)=O)CCC2(CCCO2)C1 CCC(CCC(=O)N(CCC(N)=O)C)NC(c1cccc(C)c1)=O C1(NC(c2cn(CC=C)nc2)=O)(CF)CCN(C(C2CC2c2ccsc2)=O)C1 c1(C(=O)NCC#N)cc2cc(-c3ccn4cnnc4c3)ccc2o1 CC(C)C(CNC(c1cc(Cl)n(C)n1)=O)C(=O)NCC1CC(O)CN1C CC1CCC(=CC(=O)N(C)CC2C3CN(C(c4ccsn4)=O)CC23)CC1 c1(C(N(CC(N2C(CC(=O)OC)CC2)=O)C)=O)occ(C)c1C.C12(CC1)C(=O)N2 N1(C(C(C2(O)CCCCC2)CC)=O)CCC(C)(NC(=O)C(C)C(C)O)C1 C1(CC)C(=O)N(C)CCN1C(=O)C(CNC(=O)C(CO)OC)N(C)C C#Cc1cnc(C(=O)NCC2CC(F)CN2C(=O)CC=C(Cl)Cl)c(C)c1 c1(C(C)NC(=O)CCOCCN(CCO)C2CC2)nnc(C(F)(F)F)s1 CC1C(NC(=O)CNC(C2CCC2)=O)CC2CCC1N2C(c1ccncc1F)=O NC1(c2cccc(F)c2)CCN(c2cc(C(N)=O)ncn2)C1 c1(N2CC(CCOC)OCCC2)nccc2cc(Br)sc12 CC(C)C(C(=O)N1CCCC(CNC(C2(n3cccn3)CC2)=O)C1)C1CCC1 Cc1cccc(C(=O)NC2CC(NC(c3cccc(Br)c3C(F)(F)F)=O)C2)c1C CC1CN(C(C2CC23CC(O)C3)=O)CC1(C)CNC(c1ccc(F)cc1)=O N1(C(C(C(C)C)C#N)=O)CCCC(C)(C)C1C(N1CCCC1CN(C)C)=O N1(C(c2cc(C)sc2)=O)CC(C(=O)N(CC(C)O)C(C)C)C(C)(C)C1 n1(CC)c(N2CCCC(C(=O)Nc3cccs3)C2)nnc1-c1ccc(Cl)nc1 c1(C(NNC(c2cccn(C)c2=O)=O)=O)cnn2ccc(O)nc12 C1(NC(c2ccc(C)o2)=O)CC2CC1CN(C(=O)C(C)(C)C1CCCCO1)C2 Cc1nc(NCc2nc3ccccc3s2)cc(=NCC(C)CC(F)(F)F)[nH]1 N1(C(C2(NC(C3CC(C(=O)OC)C3)=O)CC2C)=O)CC(C(=O)OC)C2(CC2)C1 c1(C(N2CCOC(C3CC3)C2)C(=O)NCCOCC)ccc2cccc(Br)c2n1 Cc1cc(O)ccc1CNC(=O)C(C)N(C)C(c1cc[nH]c1)=O c1(C(=O)NCc2nccc(C(=O)NC(CCC)CCC)c2)cc(N)cc(F)c1 c1(C(N2CCC(N(C(C3CC(=C)C3)=O)CC)C2)=O)cc(N)c(CC)o1 C1(NC(CCCOC(C)=O)=O)CCCN(C(=O)CC2CCNC(=O)C2)C1 N1(C(C(CCC)CC(C)C)=O)CCCC2CN(c3nnc(C(F)F)o3)CCC12 CC(C)C(O)C(=O)NCCOC1CCN(C(C2CC(N(C)C)C2)=O)CC1 C1(C)(NC(CN(C2CCC2)C(c2cnc(CC)nc2)=O)=O)CC(C)(C)OC1=O Cc1nn(C)c(Cl)c1CC(=O)N(C)CC1CN(C(C2CCC(O)C2)=O)C1 C1(NC(=O)CN(C)CCO)CC2(CCCN(C(=O)CSCc3cccs3)C2)C1 CC(C)CC1C(=O)N2C3C(CC)N1C(CCC3C(=O)OC)CCC(CC)C2 CC1CCCN(C(=O)C2=NOC(C)C2)C1CNC(c1ccc(N)c(Cl)n1)=O C1(NC(CCC2COC(C)(C)O2)=O)COCCN(C(C2CC(CC3CC3)C2)=O)C1 Cc1cn2c(n1)C(C(=O)NC1CCN(C(=O)C3=CCCCC3)C1)CCC2 c1(OC)nc(Br)ccc1CCCNC(N1CCCCCC1CCOC)=O N1(C(c2nnn(CC)c2C)=O)CC(F)(F)CC1CNC(=O)CS(=O)(=O)CC C1(C(=O)NCc2cnn(CC)c2C)CC2CC1CN(C(=O)CC(F)(F)F)C2 C(=O)(C(C)(CC)CCC(C)C)NC1CC2(CC(CNC(C(C=C)O)=O)C2)C1 c1(C(=O)NC2C(C)CCN(C(CCCC#CC)=O)C2)nc2ncccn2n1 C1(NC(C2ON=C(C)C2)=O)CCN(C(=O)COc2ccccc2)CC1C c1(OC)ccccc1C=CC(=O)NC(C)CCCCNC(C1CCCOCC1)=O c1(C(N2CCC(C)(CNC(C3(C)CC=CCC3)=O)C2)=O)ccc2c(c1)COC2 c1(C(N2CC(CNC(CSC(C)C)=O)C3C2C3)=O)cc(Cl)cc(Cl)c1N C1(NC(c2nnc(C(C)(C)C)s2)=O)CCC2CCN(C(C3CSCCS3)=O)C1C2 C(=O)(C(=O)N=S(C)(C)=O)NCCC1N(C(C2(N(C)C)CCCCC2)=O)CCCC1 c1(C(=O)OCC)cnc(=NC(C)CCCC(=O)NC(=O)CC(C)(F)F)[nH]c1 C(=O)(CC(CC)C(C)C)NC(CCCCNC(C=CCOC)=O)(C)C C1(C(=O)NCC2(CNC(CC=C(C)C)=O)CCCCC2)CC(=O)CC12CCC2 CCC(C)C(C(=O)N1CCC(C)C(NC(C2CCNC2=O)=O)C1)NC(C)=O Cc1nc(CC(F)(F)F)sc1C(=O)NC(C)COc1cccc(F)c1 c1(CCC(=O)NCCC(C)NC(c2cccc(C3(C)CC3)c2)=O)cncc(F)c1 C1(C(=O)NC2(CO)CN(C(C3(OC)CCC3)=O)C2)CCCCC12CC2(F)F c1(C(N2C(CNC(Cc3ccc(C)nc3)=O)CC2)=O)c[nH]c2nccc-2c1 Cc1nn(C)c(C(=O)NCC2CCN(C(c3cc(C)n(C)n3)=O)C2(C)C)c1Cl C(=O)(C1CCCc2ncccc21)OCC1CC=C(C)CC1 N(C(=NCC(C)C)NCC(c1ccc(O)cc1)O)CC(NOCC)=O c1(C(=O)NC2C(CC)CN(C(=O)C(Cl)=CCl)CC2)cc2cc(OC)ccc2[nH]1 Cc1cccc2c(C(=O)NCCCCC(C)NC(=O)Cc3cnns3)coc12 c12nnc(N3CCSCC3)n1C2.c1(C(C2CCCOC2)O)ncccn1 C1(F)(CNC(=O)Cc2ccc(F)cc2)CCN(C(C2C3CCOCC23)=O)CC1 c1(C(=O)NC2(CN(C(COCC(=O)NC)=O)C)CC2)cc(S(C)(=O)=O)oc1C CC1CN2CCCC2CN1C(c1ccc2c(c1)CCC2)C(=O)NC1CC(F)(F)C1 C1(C(C)CNC(c2cc(O)ncn2)=O)CCN(C(=O)CC2CCCC2(F)F)CC1 c1(C(=O)NCC(C)NC(c2ncc(Br)cn2)=O)cccc2c1NCCNC2=O N1(CC)CCCC2(CCN2C(=O)Nc2cc(F)ccc2OC)C1 n1(C(COC)C)nc(-c2cccc(F)c2)nc1CC(C)SC c1(COCCNC(c2n(CC(=C)C)nnn2)(C2CCOC2)C)cccc(C)n1 Cc1cc(C)c(C(=O)NC2(C)CCN(C(=O)CCC3CCCCO3)C2)s1 C(=O)(CS(N)(=O)=O)NC(C1CN(C(=O)CC2(C)CC2(F)Cl)CCO1)C c1(C(N2CC(CNC(C(C)(C(C)C)NC(C)=O)=O)C2)=O)cnc2c(F)cccn12 C1(C(=O)NCC(c2ccccc2F)NC(c2cnnn2C2CC2)=O)CCCNC1=O c1(C(C)=O)ccc(C(N2CC3(CCC3NC(=O)CC3(N(C)C)CC3)C2)=O)c(C)c1 c1(C(N(C2CCCC(N(C)C(C3CCC=CCC3)=O)C2)C)=O)cc2n(n1)CCO2 c1(C(N2CC(CNC(C=C(C)C)=O)C(C)C2)=O)ccn2nccc2n1 N1(CCC(=O)NCC2C(OC)COC2)C(=O)C2CCCCC2C1=O c1(OCC(=O)OC)cccc(C(N2CCOC(C(C)NC(=O)C(C)(C)C)C2)=O)c1 c1(C(=O)NCC(CN(C(c2[nH]cc(CC)c2)=O)C)C)cc(C)c2occc2c1 C(=O)(C1CN(C(=O)CNc2ccccc2C(N)=O)Cc2ccccc21)OC c1(C(=O)NCC(C)NC(C(C(C)C)NC(=O)OCC)=O)noc2c1COCC2 C1(NC(C(C)Cn2cncn2)=O)CC2CN(C(C3(F)CCCC=C3F)=O)CC2C1 C12(C(N3CCC(N4CCC(NC(C5CCCC5)=O)CC4)C3)=O)CCC(CC1)OC2 c1(N2CC(CC)OC3(C2)CCOC3)nc2cccnc2c(=NC2CN(C)C2)[nH]1 C=CCC(C(=O)N(C1CCCN(C(c2ccc(CO)cc2)=O)C1)CC)OC N1(C(CC2N(C(c3cncc(OC)c3)=O)CCC2O)=O)CC(OC)C2(CC2)C1 CCC(CC(=O)NC1CC(CC(N2CC(OC)CC(C)C2)=O)C1)CC(C)C c1(C(N2CC(C)C(NC(c3ccn(C)c3)=O)C2)=O)csc2nnsc12 Cc1cc(C(N2CC3(CCN3C(=O)C(C)n3ccnc3)C2)=O)nnc1C N1(C(CCC(C)(F)F)=O)CCC2(CC1)C(NC(=O)C=Cc1ccsc1)CS2(=O)=O C1(C(=O)NCC(CC(C)C)NC(=O)CC2(O)CCCOC2)CCCCCCC1 N1(C(C2(COC)CCCO2)=O)CC(NC(=O)C(O)Cc2ccccc2)C(C)(C)C1 C12(C(=O)NCC3(OC)CN(C(C4CC45CCOC5)=O)C3)CCCC(C)(C1)OC2 c1(C(=O)NC2C(NC(C(CC)NC(C)=O)=O)CCCC2)c[nH]c2c(Cl)cccc12 c1(C(C)C(N2C(CNC(C3(C#N)CC3(C)C)=O)CC3CC23)=O)cc(F)cc(F)c1 C1(CC(=O)NC(c2nc(CC)on2)C)CCCN(C(=O)CNC(N)=O)C1 C1(NCCc2cc(OC)cc(OC)c2)CCC2(CCNCC2)CO1 c1(C(=O)NCC2C(C)(C)N(C(=O)CCC3(O)CCC3)CC2)ccc2ocnc2c1 Cc1c([N+](=O)[O-])c(C(=O)NC2CC3CN(C(=O)CSC(F)F)CC3C2)nn1C N12CCN(CC1)C(=O)C(F)NC2=O.C(C)(C)(C)OCCN(C)C N1(C(c2c(OC)ccc(Cl)c2)C(=O)NCCOC)CCCCC2CCCCC12 C(=O)(C#CC1CCOCC1)N(C1CCC(NC(c2cc(C)n(C)c(=O)c2)=O)C1)C C(=O)(C(C)(O)CNC(c1cccc(OC(C)(C)C)c1)=O)OC c1(CC(=O)N(C)CCN(C2CCO2)C)ccccc1OC(F)F C1(CC(=O)NCC2(O)CN(C(C34COC(C3)C4)=O)C2)CC(=O)NC1=O.C1CO1 CCCC(C(=O)NCC1(C)CCCN1C(C1CC(N2CC(O)C2)C1)=O)OC C=CCCN=C(NCC(c1ccoc1)O)NC1CSC1(C)C c1(C(=O)NCC(CCNC(C(C)O)=O)(C)C)cc2c(s1)C(C)(C)CCC2 C1(NC(C(COC)C)=O)CCOC12CCN(c1ncc(C)cc1[N+](=O)[O-])CC2 c1(C(=O)NCCCOCCNC(CC2CC(=C)C2)=O)ccc(OC(F)(F)Cl)cc1 N1(C(C2C(CC(=O)N(C)CC)C2)=O)CCOC(Cc2cn(CCF)nn2)C1 Cc1ccc2[nH]nc(C(=O)NCCC3CN(C(=O)CC(C)P(C)(C)=O)C3)c2c1 Cc1ccc(CO)cc1NC(=O)C(F)CC1CN(C(C2CCCCCN2C)=O)C1 CCCCCCCCC(=O)NC1CCN(C(C23CSCC2C3)=O)CC(O)C1 C(=O)(CC(C)(C)NC(c1ccc(C(N)=O)[nH]1)=O)NC(CCC=C)C1CC1 O=C1CC(C(N2CCN(C(=O)Cc3ccco3)CC2C2CC2)=O)NC(=O)N1 c1(C(N2CC(CNC(c3cc(CCOC)on3)=O)C2)=O)cccc(Cl)c1[N+](=O)[O-] N1(C(C2C(CNC(CC(C)(C)C3CC3)=O)OCC2)=O)CCC(C2=NOCC2)C1 N(C(=NCC(F)(F)F)NCC1(N(C)C)CC1)Cc1ccc(SC)c(OC)c1.N(C)(C)C c1(NC(Cc2n(C)nnc2)=O)cc(C#N)ccc1Br C(=O)(C(O)CC(N)=O)NC(CSC)(C)C(=O)NCc1csc(C)n1 C1(C(N2CC(C(F)(F)F)C(O)C2)=O)CC2CCC1N(Cc1ccc(Cl)s1)C2 C(C(O)CC(=O)N1CC(C)(C#N)C1)NC(Cn1ccc(C)n1)=O c1(OC)cc(C)c(C(N2CCCN(C(=O)C=C(C)C(C)C)C(C)C2)=O)cc1Cl C1(C(=O)Nc2cccc(C3(N)CC(C)(C)C3)c2)NC(=O)OC1(C)C c1(OC)ccc(C(=O)NC2CC(F)CN(C(=O)C=C(C)c3ccsc3)C2)nc1N C(c1scnc1C)=CC(=O)NCC(CNC(C=CCN(CC)CC)=O)CO C(=O)(C(C)(C)S(C)(=O)=O)NCCCCN(CCNC(c1cccc2c1NCC2)=O)C C1(C(C)C)CCCC(NC(=O)Cc2cc(Cl)n(C)n2)CC1 C1(NC(c2cc(Cl)sc2Cl)=O)CC(C(=O)NC2COCCO2)CC1O C1(C(=O)NC2(C)CC(NC(c3cc4ncccc4[nH]3)=O)C2)CCC2CC1C2(C)C N1(C(C(CC#C)C)=O)CCC(NC(=O)CCCCn2ccnn2)CC1C CC1CN(C(C2CC(=O)C23CCC3)=O)CCN(C(=O)C=C2CCC(C)(C)CC2)C1 C(N=c1[nH]c2ccc(Br)cc2o1)C1C(C)CCN(C(C2CC(C(F)(F)F)C2)=O)C1 Cc1nc(C(N2CCC(NC(=O)Cn3ncccc3=O)C(C)C2)=O)ccc1C#N C(=O)(CCCCCCN=[N+]=[N-])Nc1cc(C)c(NC(C2(C3CC3)CCC2)=O)cc1 C1(C)(CNC(C2(C)N(C)CCC2)=O)CCCN(c2cc(O)ncn2)C1 C(=O)(C(F)CC(C)(C)NC(=O)C(C)CC=CC)NCCOCC=C.C=O C#Cc1cncc(C(N2CCC(CNC(=O)CCC3CC3(Cl)Cl)(OC)CC2)=O)c1 CC1(C)CC=C(C(=O)N2CC(CNC(=O)CNc3ccccc3Br)C2)CC1 C#CC1(C(=O)NCCC2(OC)CCC2)CCN(C(=O)C(CC)C(C)C)C1 N1(C(C(=O)NC(C)C)=O)CC2(C=C(C(=O)NC3CCCC(O)C3)CO2)C1 N1(C(CCCN(C(C)=O)C)=O)CC(N(C(=O)C=Cc2ccsc2)C)C(F)C1 c1(CNC(=O)NC(COC)C2CC2)sc2ccsc2c1CO Cc1ccc(NC(c2cc(C(=O)NC3CC(NS(C)(=O)=O)C3)cs2)=O)c(C)c1 C(=O)(C(C)(O)CSc1ccccc1)N1C(NC(CN(CCC#C)C)=O)CCC1 CCC(C)CC(C(=O)O)NC(=O)C(c1ncccc1Br)(F)F C1(CNC(Cc2c(SCC(=O)NC3(CF)CC3)cccc2)=O)CC2CC1CC2O CC1(C)CCCC(CNC(=NCCc2cccs2)NCC2CCC=CO2)O1 C(=O)(CC(F)(F)C(C)C)NC1CCN(C(C=C(C)c2ccco2)=O)C12CC2 CCCC(C#N)C(=O)NCCC(C)NC(c1cccc(-c2ccc(F)cc2)n1)=O c1(C(N2C(CC)CN(C(c3csc(=NC)[nH]3)=O)CC2)=O)cc(C)c(=O)n(C)c1 c1(C(N(C2CCN(C(c3n(CC)ncc3)=O)CC2)C)=O)c[nH]c2cccc(F)c12 N1(C(COCCCC(C)C)=O)CCC2CC2(C(=O)NC2(C)CCCC2)CC1 C(C)(C(=O)NC1CC(CCNC(=O)CCC2(C)CC2)C1)OCCCC CCC(CNC(=O)CC(=O)NCC)(CC)NC(c1ccnc(-c2ncc[nH]2)c1)=O C(=O)(C(C)CC(C)C)N(CC(CC)NC(c1cc(OC)ncc1Cl)=O)CC C1(n2cc(CCCC#N)nn2)(C(=O)OC)CN(C(c2cnn(C3CC3)c2)=O)C1 N1(C(C(=O)NCc2cnc(-c3n(C)ncc3)nc2)=O)CC(C2CCCC2)C1 N1(C(CC(C(C)C)OCC)=O)CCN(C(=O)C(C)CC(C)(F)F)CC12CCC2 C12(C(N(C)CC3CCN(C(C4CN5CCN4CC5)=O)C3)=O)CCC(N=[N+]=[N-])C1C2 Cc1nnc2n1CCC(C(=O)N(c1ccccc1F)C1CCNCC1)C2 C1(C(N2CC(SC)C(NC(C3CCOC3)=O)C2)=O)CCN(CP(C)(C)=O)CC1 N1(C(C2(COCC)CC2)=O)CCC(C)C(C(=O)Nc2cccc(CCSC)c2)C1 C(=O)(C1=C(Cl)CCOC1)NC(CNC(C(c1ccc(OC)cc1)CC)=O)CO c1(CC)cccnc1C(=O)NC1CCCCC1CNC(=O)C(O)C1CCC1 C1(C(=O)NC(C)Cc2nn[nH]n2)CN(C)CCN1C(C1CC1[N+](=O)[O-])=O C1(C(=O)NC2C(NC(C3N(CC)C(=O)CC3)=O)CCC2)C2CCC3(COC(=O)C13)O2 c1(C(=O)NC(C)Cn2cc(-c3csc(C(=O)O)c3)nn2)cc(S(N)(=O)=O)ccn1 C1(NC(=O)NC2CCCCN2c2cn[nH]c2)CCC12CCCC2 N1(C(C(CC)NC(C)=O)=O)CC2(CC(NC(=O)CC3CC3)C2)C1 C=CCC(CC)C(=O)NC1CCN(C(c2snc(Cl)c2Cl)=O)C1CC N1(C(COCC(=C)C)=O)CCC(C2CCN(C(c3cc(CC)[nH]n3)=O)CC2)CC1 c1(C(N(CCCNC(C#CC(C)C)=O)C2CC2)=O)cc(=O)c2ccccc2o1 C#Cc1c[nH]nc1C(=O)NC(c1ccc(CC)cc1)CNC(=O)C(CCC)OC Cc1cc(C(N2CCCC2C(=O)Nc2cccc(C)n2)=O)cc(Cl)n1 C1(C(C)C(=O)NCCN(CC(F)F)C)CCN(C(c2ccc(CO)s2)=O)C1 N1(C(C(CC)F)=O)CCCC(CCCCNC(=O)C(=O)NCCOC)C1 c1(-c2scc(C)n2)nc(C(N2CCCC2)C)n(CCC(F)(F)F)n1 CN1CCCC(C(=O)NCC2(NC(=O)CCOC3CC3)CCCC2)C1 S(=O)(=O)(c1ccc(F)c(Cl)c1)C(N(CCCNC(C1C2CC2C2CC12)=O)C)=O S(=O)(=O)(c1c[nH]c(=NCCc2cccs2)cc1C)NCc1ccc([N+](=O)[O-])cc1 C1(N(C(c2c(C)[nH]c(-c3nn[nH]n3)c2)=O)C2CC2)CCC2(CCCCC2)CC1 c1(CN(CCCn2cc(C(C)O)nn2)NS(=O)(=O)C2CC2)ccc(Br)nc1 C(=O)(N=c1[nH][nH]c2ncc(Br)cc12)C1(O)CCN(C(c2cccc(Cl)c2Cl)=O)C1 c1(C(=O)OC)c(C)c(S(=O)(=O)NCCc2cn3cccnc3n2)c(C)n1C Cc1nn(C)c(C)c1C(=O)NCC1(F)CN(C(=O)COC2CCOC2)C1 N1(C(C=CC(=C)C)=O)CCC(NC(=O)C(C(C)C)NC(N)=O)C(C(N)=O)C1 C1(NC(c2c(CC)cccc2)=O)C2COCC1CN(C(=O)Cc1cc(C)no1)C2 N1(C(C(C)SC)=O)CC2(COC(CNC(=O)CS(N)(=O)=O)C2)C1 c1(C(N2CCCC(NC(c3c(C)cns3)=O)C2C)=O)ccnc2c(F)cccc12 C1(CNC(C2(CC)CC2(F)F)=O)CN(C)CCN1C(=O)COC(C)C CC(O)C(F)(F)C(=O)NCC1CN(C(=O)C(N)=O)CCCO1 N1(C(c2cn(CC(=O)OCC)nn2)=O)CC2(CCCC2NC(C2CC2(F)F)=O)C1 c1(C(=O)OC)cc(C(=O)N(C)CC2CCN(C(=O)CC3CC(C)=NO3)C2)c(C)[nH]1 c1(NCN2C(=O)CC(OC(C)C)C2)nc2c(c(=NCCC(C)N(C)C)[nH]1)CCC2 S(=O)(=O)(c1ccccc1Cl)N1C(C(=O)Nc2ccc(C(N)=O)nc2)CC(O)C1 Cc1cnc2cc(C(N3CCC4C(NC(C5CCC(C)(C)OC5)=O)C34)=O)ccn12 CC1CC(C(N2CC(C(C)NC(=O)C(F)(F)c3cncs3)C2)=O)CC(C)O1 c1(C(=O)NC2(CCNC(C(C)NC(=O)NC)=O)CCOCC2)c(C)nn(C)c1C Cn1nc([N+](=O)[O-])c(Cl)c1C(=O)NCC(C1CCOC1)NC(=O)C(F)=CCCF c1(CS(=O)(=O)NCC(COC)O)ccccc1C c1(-c2cn(CC3N(C(Cc4cc(CC)no4)=O)CC3)nn2)cccc(OC)c1Cl C=CCC(C)(C)C(=O)N(C)CC1CCN(C(C2(N3CCOC3=O)CC2)=O)C1 Cn1ccc(S(=O)(=O)N2CC(O)CC2C(N2CCSCC2)=O)n1 C1(C(N2CCC(NC(C#CC3(CC)CC3)=O)CC2C)=O)CCCC2C1C2(F)F c1(NC(=O)NCC2(C(=O)OC)CCCO2)cccnc1C(C)(C)C C1(C(=O)NCCn2ccc(C(=O)NC(c3onc(C)n3)CO)c2)NC(=O)OC1(C)C C1(C(=O)NC(CNC(c2c(O)nc(C)c(C)n2)=O)CO)CCc2cnn(C)c2C1 c1(N2CCCC(CC=C)(NC(=O)COC(F)F)C2)ncnc2c(OC)cccc12 C1(CN(C(=O)CC2CC(OC)C2)CC)CCCCN1C(=O)CCCN(C)C1CC1 Cc1nc(CCC(=O)NCC2(O)CN(C(c3cc(C(F)F)[nH]n3)=O)C2)oc1C c1(C(=O)NCC(CCNC(c2c(C)cc(CO)o2)=O)(C)C)cccc(C)c1Cl FC1COc2ccccc2C1NCc1csc(I)n1 c1(CNC(C2(NC)CC(F)(F)C2)=O)ccc(C(F)(F)F)cc1C C1(CCNC(C2(C(F)(F)F)CCCC2)=O)(CNC(CCOC)=O)CCCC1 C1(CNC(C(C)C)=O)CC(F)(F)CN1C(=O)C=Cc1ccnn1C C(=O)(CCC(C)(F)F)N1CC(NC(c2nc(-c3ccc(C)o3)sc2)=O)C(O)C1 C1(NC(=O)NCCC(C2CCCCC2)C)CC(=O)N(C)C1c1cccc(F)c1 C(=O)(C(C)(C)C(C)(F)F)N1C2C(CNC(CN3C(C)CCC3)=O)C(C2)C1 c1(C(=O)NCC23CC2CN(C(c2csc(O)n2)=O)C3)cnc2[nH]ccc2n1 c1(NC(N2C(C)COCC2)=O)ccc(Br)c2cccnc12 S(=O)(=O)(CCC(=O)NCC1=CCCN(C(c2[nH]cnc2C)=O)C1)NC C(=O)(C(C)(C)CC(=O)OCC)N1CCC(CC#C)(C(=O)N(C2CC2C2CC2)C)C1 c1(C(N2CC(NC(C(c3ccccc3)C)=O)C(C)C2)=O)cc(Cl)nc(Cl)c1 c1(C(N2CCC(CCNC(C(C)c3cccs3)=O)C2)=O)ccc2nsnc2c1 C1(NC(CCP(C)(C)=O)=O)CCSC12CN(C(=O)CCc1ccc(N)cn1)C2 c1(C(=O)NC2CC(C)(NC(=O)CCCN3CCCC3)C2)cc(F)ccc1Cl Cc1cc(C(=O)NCC2(C)CN(C(=O)C(N)=O)C(C)(C)C2)c2c(O)nn(C)c2n1 c1(OC)ccc(O)cc1C(=O)NCCOC1CN(C(C2CCN(C)C(C)C2)=O)C1 c1(C(N(C2CCN(C(CC=CC)=O)CC2C)C)=O)ccn2cc(C)nc2c1 c1(C(N(C)CC2CCCN(C(c3ccccc3)=O)C2)=O)sc2ncccc2c1Cl Cc1cnccc1-n1nc(CCCN(C)C)nc1C1COCC1(C)C C1(C(=O)NCC2C(NC(c3c(CCC)n[nH]c3)=O)C2)CCOC2(CCC2)C1 CC(C)CC(O)CC(=O)NC1CCCCC1C(=O)NC1CCCC1(C)C C=CC1CN(C(=O)NCC(C)(O)CO)CCO1 N1(C(CC(C)OC)=O)CCN(C2CCN(C(c3ccc(C(N)=O)[nH]3)=O)CC2)CC1 C1(C(=O)O)(NC(CC)Cc2ccc(F)cc2)CCc2nc(C)ccc21 C1(NC(C(Cn2cccn2)NC(C2(COC)CCC2)=O)=O)C2CCC(C2)C1CO N1(C(C(=Cc2ccco2)C)=O)CCC(C2(NC(=O)CC34CC(C3)C4)CC2)C1 C12CC(C1(C)C)CC(=O)N2.C1(CNC(c2c(CC)ocn2)=O)CC(F)C(=O)N1 N1(C(C(C2CCCCC2)C)=O)C(C(=O)NC2C3CCCOC23)CCC12CC2 c1(C(N(C2CCN(C(COCCOCC)=O)C2)C)=O)ccc2sccc2c1 C=Cn1ncc(C(=O)NCC(C)C(=O)NC(C(C)C)C2CCC2)c1N c1(NC(=O)CCCn2cncn2)ccc(C(F)F)s1.C12CC(C1)C(=O)N2C CC1CCCC=C1C(=O)N1CCCC1(C)CNC(C1(O)CCCC1)=O CC1CC(NC(=O)Cc2cncs2)CCN1C(=O)C(C)N1CC(C)C1 C1(C(=O)OC(c2cccc(C)n2)C)COCC12CCC2 C(=O)(CCC(C)S(C)(=O)=O)NC(C=CC(=O)NC(CC)(CC)CC)C Cc1cc(C(=O)NCC(C)N(C)C(c2cn(C)nc2C2CCOC2)=O)cnn1 Nc1ccnc(C(=O)NCC2CC(CNC(c3ncsc3Br)=O)CO2)c1 C1(NC2c3ccc(OC)cc3CC2)CCN(S(=O)(=O)N2CCCCC2C)CC1 C1(C(=O)NCCCOCCCNC(c2c(C)c[nH]c2)=O)CCN(C)S1(=O)=O C1(C(=O)NC(C(=O)NC2(CC#C)CCC2)CC#C)CN2CCC1CC2 N(C1CCCc2nc(=N)[nH]cc21)C(=O)NC1CCN(C(C)C)CC1 c1(C(N2CC(C)C(NC(c3cccn3C)=O)C2)=O)ccc2c(c1)CN(C)C2 c1(C(=O)NC2C(C)CN(C(=O)CS(N)(=O)=O)C2)cccc(N)c1Br c1(OC)cccc2c1OCC(C(N1CCN(C(=O)CC#N)CC1C(C)(C)C)=O)C2 C(=O)(C1=NOC2(CCC2)C1)NCC1(C)CCCN(C(C2(C(N)=O)CCC2)=O)C1 Cc1cc(C)cc(C=CC(N2CCC(NC(C3CCC(C)O3)=O)C(F)C2)=O)c1 Cc1nsc(N)c1C(N1CCC(O)(CNC(C2CCSC(C)C2)=O)C1)=O N1(C(c2c(C)[nH]cc2)=O)CCC(CNC(c2cc(O)nc(O)c2)=O)C(F)(F)C1 C1(C)(CNC(CSCC)=O)CCN(C(c2cc(-c3ccccc3)sn2)=O)C1 C1(c2nnnn2CC(F)F)(NC(c2c(C)ccnc2)C)CCCC(C2CC2)C1 C(=O)(C(C)(C)C(F)(F)F)NC1CC(CNC(C(C(C)C)CN(C)C)=O)C1 C1(OCC(=O)NC)CCN(C(=NCCC2CS(=O)(=O)C2)NCC2CCCC2)CC1 c1(NC(=O)NC(C2CCCCC2)C2CCC2)cc2cc(Br)cnc2s1 C1(C(=O)NC2CC(CC(=O)N(C)CC3CC3(F)F)C2)(OC)CCCCC1 C1(NC(CCC2(C)CN(C(c3cc(Cl)c[nH]3)=O)C2)=O)CCCCCC1(C)C C1(CC(=O)NCCC2N(C(C3CC(C)(C)C3)=O)CCC2)CCC2(CCC2)O1 C1(C(N(C2CCN(C)CC2)CC)=O)C(C)CCCN1C(c1ccc(Cl)cc1)=O c1(C(C)N(C)C(=O)NC(C2CCCO2)COc2ccccc2F)ccc(F)cc1 C(=O)(C(C)C(C)NC(C1(C)CCCCO1)=O)NCc1ccn(C(C)C)n1 Cc1cc(C#N)cc(C)c1COCC(=O)NCC(C)(CO)CC(=O)O C(=O)(C1=CCC(NC(=O)CCc2cnco2)C1)NC(CC#C)CC C1(N=c2ccn(C(C)C(=O)OC)[nH]2)(c2n(CCOC)nnn2)CCC1C1CC1 Cc1ccc(C(=O)NCC2COC(CNC(=O)C#CC3(C)COC3)C2)c(=O)n1C C#CCCCC(C)C(=O)N1CC2CC2(C(=O)NCCN2CC=CCC2)C1 c1(C(N2C(C)C(NC(=O)C=C3CCN(C)C3)CCC2)=O)cccc2c1CNC2=O C1(CN(C)C(CC(C)(C)C)=O)CC(O)C(O)CC1CNC(=O)CC1CCCC1 C1(CC(=O)NCCn2ncc(SCC)c2)CC(C)(C)CN1C(=O)C(C)O C1(C(=O)NC(c2nc(C)on2)C)CCCCN(C(=O)Cn2ncn(C)c2=O)C1 c1(C(=O)NC2CCN(C(c3cccc(Br)n3)=O)CC2)ccc(O)c(C(F)(F)F)c1 N1(C(Cc2cc(CC)no2)=O)CCC(C=CC(=O)NC2CCC3(CCC3)C2)CC1 N1(C(=O)C=Cc2ccncc2)CC2CCC(C1)N2C(=O)CC12CCCN1CCC2 C1(CNC(c2c(C)con2)=O)CCN(C(=O)C(C)(C)N2CCCCC2)CC1C c1(OC)cc(C)c(C(N2CCCC2CNC(=O)C#CC(C)(C)O)=O)c(C)c1 Cc1ccc(C(=O)C=CC(=O)NCC2(F)CCC(CNC(=O)CC3CC3)C2)cc1 C12(NC(=O)CC3CCCCC3(F)F)CCC(CNC(c3ccc[nH]3)=O)(CC1)OC2 CCC(CC)(CC)NC(=O)C(C)NC(=O)C(C)(C)COCc1ccccc1 C1(C(N(CC(C)CNC(c2ccc(C(F)F)o2)=O)C)=O)CC(=O)CC12CCC2 c1(CC(N2CC(C(N(CC(C)CNC(=O)CN(C)C)C)=O)C2)=O)cncn1C C1(CC(N2CC3C(CNC(=O)Cn4ccc(CO)n4)C3C2)=O)CCCS(=O)(=O)C1 Cc1cccc(Br)c1C(C(=O)NC(C)C(C)F)NC(c1cc(C(N)=O)[nH]n1)=O CCC(C)(C#N)C(=O)N1CCC(CN(C(=O)C=Cc2nc(C)c(C)[nH]2)C)CC1 N1(C(c2nnc(C)s2)=O)CCCC(C)C1CCNC(c1cc(C2CCC2)no1)=O CC(C)(C)CCCC(=O)N1CSCC1C(=O)NC1(C)CCCC1(C)C c1(CNC2CCC(NC(c3c(F)cc(Cl)cc3F)=O)C2)cccc2occc12 CCC(C)CCCC(=O)N(CCC(=O)NC(C)CN(C)C)CC C1(NC(CCCC=C)=O)CN(C(c2ccc(-c3ncon3)cc2)=O)CC2(CC2)C1 c1(NC(c2n(C)ncc2)=O)cnc2[nH]cc(-c3cnn(C4CCC4)c3)c2c1 c1(C(C(=O)N(CCN(C(C(F)=CC)=O)C)C)N(C(=O)COC)C)ccccc1 C1(NC(c2c(CCN(C)C)cccc2)=O)CCOC12CCS(=O)(=O)CC2 c1(OC)cc(N)c(C(=O)NC2CCN(C(C3(OC)CCCC3)=O)C2)cc1Br Cc1cccn2ncc(C(=O)OC34CCC3CN(C(=O)OC(C)(C)C)C4)c12 c1(NC(C(=O)NCCC(COC)OC)=O)cnc2ccccn12 N1(Cc2cn(CC(=O)OC)nn2)CC(C)(C)OC2COCC12 C=CC1CN(C(=O)CCc2ncc[nH]2)CC1NC(=O)CCCNC(N)=O c1(C(=O)NC2(CNC(C(CC)NC(C)=O)=O)CCC2)ccc(OC)c2ccsc12 S(=O)(=O)(c1ccc(Br)c(Cl)c1)N1C(C(=O)NC(C)(C)CO)CCCCC1 C1(CN(C(=O)CC2CCCCC2)CC)CCN(C(C2COCOC2)=O)CC1 C1(C(=O)NCCC2(CNC(c3c(C)cn(C)c3)=O)CC2)CC2CCC1CC2 c1(CC(=O)NC2CCN(CC3(OC(C)C)CC3)CC2)ccc(C(F)F)cc1 C=CC(C)(C)CC(=O)NCCCN(C(=O)C=CCF)Cc1ccccc1 C(=O)(C1=C(C(C)F)N(C)C(=O)NC1c1csc2cncn12)OCC c1(C(=O)NC(CN(C(=O)C(C)(F)CC2CCCC2)CC)C)coc2c1COC2 c1(C(CC(=O)NC2C(CNC(Cc3cnc(C)[nH]3)=O)C2)O)ccc(Cl)cc1 CC(C)CC(C(=O)NCCCC1CCCN1C(=O)CCCF)c1ccccc1 N(C1CN(C(C2CCC2CF)=O)CCc2ccccc21)C(C1CCC(C)(C)CC1)=O c1(C(N2C(CN(C(COC(CC)C)=O)C)CCC2)=O)cc2ncccc2cc1Cl c1(CC)c(Cl)nc(C2CCC2)[nH]c1=NCCN(C)C(C1CN(C)CCO1)=O c1(C(C(N2CC(C)(NC(CCCC3C(C)C3)=O)C2)=O)C)cnn(C)c1C(F)(F)F C1(NC(c2c(C)csc2)=O)CCCCC1C(N1CCC1(C)C(=O)OC)=O N1(C(c2c(C)cn(C)n2)=O)CCOC2(CCCN(C(c3cnc(S)[nH]3)=O)C2)C1 c1(N(C)CC2CCN(c3ccc(Cl)c(Cl)c3)C2)ccc2nnc(C(C)(C)C)n2n1 C12(NC(CSC)=O)CCC1CN(C(=O)CC1(N(C)C)CCCC1)C2 c1(C(=O)NC2C(NC(Cc3c(C)non3)=O)CCOC2)cc2c(cn1)OCCO2 Cc1ccnc(CNC(=O)CCN(CCO)C(C2CN(C3CCC3)C2)=O)n1 CCC(C)C(O)C(C)C(=O)N1CC(CC(=O)N(CCN=[N+]=[N-])C)(OC)C1 N1(C(Cn2nc(C)c(C(=O)OCSc3ccccc3)c2)=O)CC2(CC(C(F)(F)F)C2)C1 C1(C(F)(F)F)(C(=O)NCCN(CC(C)O)C(c2ncc(F)cn2)=O)CCN(C)C1 c1(C(N(CCCNC(C2CCC(OC)C2)=O)C(C)C)=O)cccc(Cl)c1Cl N1(C(C(CC)n2ccnc2)=O)CC2CC1C2NC(=O)CCCc1cccnc1 N1(C(C(F)=CCC)=O)CC2CCC1C2NC(=O)CC1CCCCC1(C)C c1(SCC(=O)NC2C(CC)N(C(c3cccc(=O)o3)=O)CC2)cc(F)ccc1F N1(C(c2cccnc2NC)=O)CC2CC(CNC(=O)CCCC3CC3)C2C1.CO N1(C(C2C3CN(C(c4c[nH]c(=NC)o4)=O)C2C3)=O)CCCC12CCOC2 N1(C(C2CC(=C3CC3)C2)=O)CC2(C(=O)Nc3ccccc3)CC1CO2 c1(OCCOC)ncccc1C(=O)N(c1cc[nH]n1)Cc1ccc(F)cc1 c1(-n2c(-c3c[nH]c(C(F)(F)F)c3)nc(-c3ccn(C)n3)n2)ccc(F)c(F)c1 CC(C)CCCCC(=O)N(C1CC(NC(=O)COCC2CCCO2)C1)C c1(C(=O)NCC(CNC(c2c(SC)csc2)=O)F)cnc(C)c(C)c1 c1(C(=O)NCC2(NC(C(CSCC)C)=O)CCCC2)cc(OCC(F)F)ccn1 Cc1cc2ncn(CC(=O)NCCC(C)NC(c3cccc(O)n3)=O)c2cc1C CCCC(CCC)CC(=O)NCC1CCCCC1NC(C1C2CC(=O)CC12)=O CN=c1[nH]c(SC)ncc1CN1CC2CC1CC2NC(=O)CCC(N)=O C(=O)(C(F)(F)CC1CCCO1)NC(C1CC(NC(C2CCOC2(C)C)=O)C1)C c1(C(N2CC(C(C)Nc3ncc(C)cn3)OCC2)=O)cnc([N+](=O)[O-])cc1C c1(CN2CCOCC(NC(c3c(C)ncn3C)=O)C2)c(Cl)ccc(Cl)c1Cl c1(OCC)ccc(N)c(C(=O)NCC2C3CN(C(=O)C(C)C(C)C)CC23)c1 C1(CNC(c2ncc(C)cn2)=O)C(C)CCCN1C(c1n[nH]cc1C)=O c1(NC(CCC2N(Cc3c(C)n(C)nc3)CCC2)=O)cccn2nccc12 n1(C(C)C(=O)NC2CCCC2NC(c2cc(O)cs2)=O)cnc2ccccc12 C(=O)(CC1=CCN(C(=O)CC(C)(C)CN(C)C)CC1)N(CC)Cc1occc1C C1(CCCCC)(C(=O)NCC(CCNC(c2ccsc2)=O)OC)CCCO1 C(=O)(CC1=CCCCC1)Nc1cc(C)c(NC(=O)CC(O)CN(C)C)cc1 c1(CCC(=O)NC(C2CCCC2)CNC(C(CCC)C)=O)ccc(F)cc1F C(=O)(CC(C)(C)C#N)NCCOCCC(=O)NCC(CC)COC(C)(C)C.CC C1(NC(c2cc(C)ncc2)=O)CCN(C(C2(n3cccn3)CC2)=O)C(C)C1 N1(C(=O)CC2CCCCN2C(C2CCCCC2C(N)=O)=O)C2C=CCC1CC2 S(=O)(=O)(c1ccc(Br)cc1NC1CCN2CCCC12)NCC(CSC)OC C(CCC(O)C(=O)N(C1(CO)CCCC1)C)NC(C(C)SC)=O C(C)(CO)(C(=O)NCCS(C)(=O)=O)NC(CSC)=O c1(NC(C(=O)N(CCc2cnc[nH]2)CC)=O)nsc2ccccc12 c1(C(N2CCC(CNC(=O)C=CBr)C2)=O)c(F)cncc1Br C(=O)(C(=O)N=S(C)(C)=O)NCC1(COC)CN(C(=O)CCc2csc(C)n2)C1 c1(C(N2C(CN(C(c3ccnc(O)c3)=O)CC)CCC2)=O)ccc(Br)cc1C c1(C(=O)NCC2C(NC(C(C=C)(C)O)=O)CC2)cc2cc(Cl)ccc2[nH]1 N1(C(C2CC=C(C)CC2)=O)CC(NC(=O)CC2CC(C)C2)C2CC2C1 c1(C(C(=O)N(C)CC2CN(C(=O)C3=CSCS3)CCO2)O)ccc(F)c(Cl)c1 C1(CC(=O)NCCc2ccc(Br)cc2)COCCN1C(C1CCCC(O)C1)=O C1(NC(C2CCN(C(C=C(CC)CC)=O)C2C)=O)CN(C)C(=O)C12CC2 C1(NC(=O)CC=C(Cl)Cl)CC2(CCN(C(=O)CC3CC4(CCCC4)CO3)CC2)C1 N1(C(c2c(C)onc2)=O)CC2CCCC2(CNC(=O)COc2ccsc2Cl)C1 c1(C(=O)NC2C(NC(C(Cn3ccc(C)n3)C)=O)C2)ccc(F)c(F)c1F N1(C(c2nnn(C)n2)=O)CC2CN(C(c3cnc(CC(C)(C)C)[nH]3)=O)CC2(C)C1 c1(CC(N2CC(CNC(=O)C(O)C3CC3)OCC2)=O)ccc(F)cc1C(F)(F)F C(C(CC)CC(CC)CC)NC(c1n(CCCC)nnn1)c1ncc(C(C)C)s1 Cc1cc(N)c(C(=O)NC23CCN(C(C4OCCOC4(C)C)=O)CC2C3)cc1C N1(C(C)C)CC(CN(C2CC(CC(=O)NC(=O)CCC3CC3C)C2)CC)CC1=O c1(C(=O)NC(CC(C)NC(c2[nH]cc(C(=O)OC)c2)=O)C)c(F)cc(C)cc1F C1(NC(COC(C)(C)CNC(C2CC2C2CCC2)=O)=O)CCCCC1(C)C c1(C(=O)OC)cc(CN2CCC(N3CCCS3(=O)=O)CC2)oc1C n1(C2CCN(C(COc3nccc(C)c3)=O)CC2)cnc2c1CCCC2 C1(C(=O)NCC2(COC)CCCN2C(=O)CC(=O)OC)CCCCN1N=O.OC c1(C(=O)NCC(C(C)C(C)C)NC(C2(C(C)C)CC2)=O)cnc2n(c1=O)CCS2 S(=O)(=O)(c1c(C)coc1C)N(C(c1cc(C)n(C)n1)C)C N1(C(=O)NCC2(OC)CCCC(C)C2)CC23CCCC2(C1)CN(C)C3 c1(C(=O)NCC(C)NC(c2c(OCC)nccc2)=O)nc(C)ccc1O OC1CCCCCC1Nc1nc(CSc2cccc(Cl)c2)cs1 Cc1cccc(CCNC(C23CC2CN(C(C2(CO)CCOC2)=O)C3)=O)n1 c1(OC)cc(C(=O)NCCCC(C)NC(=O)CNC(C)=O)cc(N)c1OC c1(C(=O)NC(CNC(c2n(CC)ncc2)=O)C(C)(C)C)cc(O)ncc1F c1(-n2cc(C3CCNC3)nn2)ccc(Cl)cc1Cl.Cc1cc(-c2cccs2)ncn1 C#CC1CCCN(C(=NCCCCN2CCCC2)NCc2ccccc2)C1 C=CCCCCCC(=O)NCC1COCCN(C(C2C(C)(C)C2(F)F)=O)C1 c1(SCCC(=O)NC2(CC)CC2)ccccc1.C12CN(C1)CC(=O)N2 C(=O)(C1=CC2CCCC12)NC1(CNC(C=Cc2cncc(C)c2)=O)CCOCC1 c1(C(C)C)ccccc1C(=O)N(C1CN(C(C2CC2c2ccco2)=O)C1)C C(=O)(CCCCCN=[N+]=[N-])N1CCC2(CC(NC(C3C(C)(C)COCC3)=O)C2)C1 C(=O)(C(CCN(C)C)NC(=O)CCNC(=O)CO)N.CC(CN(C)C)N(C)C c1(C(=O)NC(C(=O)NCc2cn(CC)nc2C)c2ccco2)cc(C)nc(O)c1 C1(C(=O)Nc2c(CC)nsc2)CN(C)CCN1C(c1cc(C2CC2)on1)=O c1(N2CCC(S(=O)(=O)NCC)C2)nc(=NCc2ncoc2C)[nH]c2ncn(C)c12 N12CCN(CC(C)C1)C(=O)C1C(C1)C2=O.C1(COC)(SC)CCC1 C1(NC(C(CC)N(CC)CC)=O)CC1C1CCCN(C(c2cc(SC)oc2C)=O)C1 Cc1nc(CCCNC(=O)CC2CCN(C(=O)Cc3sccc3C)C2)n[nH]1 Cc1cc(C(C)(C)C)ccc1C(=O)NCCCCCNC(=O)Cc1ccno1 N1(C(Cc2c(C)n[nH]c2)=O)CCCC2CCCN(C(=O)CCCCCC(C)O)C12 C(=O)(C(C)(C)C(=O)N(C)C)NC1CC(C(N2C(COC)CC2)=O)CC1O N1(C(C2CN(C)C2)=O)CCCC(C(=O)NCc2nccn2C)C1 c1(C(=O)NCc2scc(C(N(CC(C)CO)C)=O)c2)c[nH]c2nccc-2c1 C(c1ccc(F)c(Cl)c1)=CC(=O)NC(C1CCCC1)CNC(C(C)OCC#C)=O c1(C(c2nnnn2C2COC2)NCCC=CCCOC)ccccc1Br c1(SC)cccc(N)c1.C(CC(C(C)C)N)NC(N1CCCC(C)C1)=O C1(N(C(C(=O)CCCSC)C(C)C2CCC2)N)CC2CC3CC(C2)CC1C3.C1CC1 c1(CC(C)C)cn(C2CN(C(=O)CC3CC(NS(C)(=O)=O)C3)C2)nn1 N1(C(CC2C(C)(C)C2)=O)CCC=C(C(=O)N(c2ccccc2O)CC2CC2)C1 Cn1nc(C(F)(F)F)cc1C1CC1.c12cc(on1)CC(=O)NCC#CCNC2=O c1(C(N2C3C(NC(=O)COCCCF)C(C3)C2)=O)ccc2ncccc2n1 N1(C(c2c(C)c(Br)sc2)=O)CCC(NC(=O)CN2CCC2C)C12CCC2 c1(CC)ocnc1C(=O)N(CC(C)NC(=O)C(C)C1CC1)CC c1(C(N2C(C(C)O)CC2)=O)cccc(C(C)C(F)(F)F)c1 N#Cc1ccc(F)c(-c2ccc(-n3cc(Br)cn3)cc2)c1 C1(NC(COCCCC#C)=O)CN(C(c2ccc(N)c(SC)c2)=O)CCC1CO N12CCC(CC1)C(=O)N(CCOSC)C(C)C2=O.c1(C2(SC)CC2)ccncc1 C1(NC(c2ncccc2O)=O)CN(C(C2CC3CCC(C2)C3)=O)CC12CCCC2 c1(NC(C2(c3cccc(F)c3)CC2)=O)nnc2n1CCNC2 C1(CC)CCCCC1NC(=NC)NC1CCN(c2cccc(N(C)C)c2)C1 c1(C(=O)NC(C2CCN(C(c3ncc(OC)nc3)=O)C2)C)cccc(C#N)c1 C1(CC(=O)NC2C(C=C)CN(C(c3ccccc3O)=O)C2)COCC2(CCC2)O1 C1(C(F)(F)F)(OC)CC(N)(C(=O)Nc2cccc(C3(O)CCCC3)n2)C1 Cc1nncn1NC(=O)C(C)N(C(=O)CC1CC=CC1)C C1(C(N2C(C)CC(CC(=O)NCC(=C3CCCCC3)F)C2)=O)CC2(CCC2O)C1 c1(C(=O)NC(C)(C)C)c(Cl)cccc1Cl.N12CCC(O)C1C(=O)NC(C)CC2=O CC1CC2CC(C(=O)OCc3cc(C(F)(F)F)ccc3Cl)(C2)O1 C#Cc1ccc(C(=O)NCC(O)CCNC(=O)Cc2cc(C)ccc2O)cc1C c1(C(=O)NCC2C3CCCC23)oc(C(=O)NCC2(CC)CCC2)cc1C c1(C(N2CC(C)(NC(CN(C)Cc3ccccn3)=O)C2)=O)cc(F)c(O)c(F)c1 CC1(C)CCOC(C(N2CC=CC2CNC(C2(CO)CCCC2)=O)=O)C1 c1(OC(C(c2n(C(COC)OC)nnn2)NCCF)(C)C)ccc(Cl)cc1Cl Nc1c(C(=O)NC2CCC(NC(c3ccnc4[nH]ncc34)=O)C2)cc(F)cc1F c1(C(N2CC(N(C(CCNC(=O)NC)=O)C)C2)=O)ccc(CSC)cc1F C(CC1=CCN(C(c2cc(Br)cc(F)c2F)=O)CC1)NC(C(C(C)O)C)=O C1(C(=O)NCC2C(NC(=O)CCCC(F)(F)F)CC2)CCc2nnc(O)cc2C1 C1(C(=O)NC(CCC)CCO)CC(C)CN(C(=O)CCCC(=O)C2CC2)C1 Cc1nc2cc(C(=O)NC3CC4CC3CN4C(C3CC3(C)C)=O)ccc2o1 C1(C(C(=O)NCCN(C(C)C)C(CC(F)(F)F)=O)O)CCC(C(C)(C)C)CC1 c1(C(N2CCC(N(C(C3N(C)CCC3)=O)C)CC2)=O)c(N)cccc1Cl C1(NC(=O)C(F)C2CCC2)CC2CN(C(C3CC3C3CCCO3)=O)CC2C1 C1(C2CC2)(CNC(=O)CC2OCCO2)CCN(C(C2CC2c2ccncc2Cl)=O)C1 C1(C(=O)NCCC2(NC(CCC=C=C)=O)CCCC2)CNC(=O)C(C)(C)C1 CN1C(=O)CCC1CC(=O)NC(C)(C)CNC(=O)CCN1CCCCC1=O C12(C(=O)NC(C(C)(C)OC)C)CCC(C1)C2(C)C.C12CCC(C1)NC(=O)C2 c1(OCC(N)=O)ccc(C(=O)NC2CC(NC(c3ncccc3O)=O)C2)cc1 c1(C(C(=O)NCCC#N)N(CCCN)CC)cccc(F)c1C C1(NC(C(C)N2CCC2)=O)CN(C(=O)Cc2ccnc(Br)c2)C(C)(C)C1 c1(ON)ccc2c(n1)CN(C(=O)C(C)(C)n1cccn1)CC2 c1(C(C)CC(=O)NCC(O)COC(F)(F)F)cccc2ccccc12 c1(CCC)nnc(S)n1CC(=O)N(C)CC1(O)CN(C(=O)Cn2nnnc2C)C1 C1(NC(NC(CC)CC)=NCCN2CCCC2)COc2c(C)cccc2C1 C12(CNC(C(C)(C3CCC3)NC(=O)COCCCF)=O)CCC(CC1O)C2 c1(OC)cc(N2CCC(C(C)NC(c3ccc(C(N)=O)cc3)=O)C2)ncn1 Cc1ccc(C2(C(N3CC(C)(NC(c4sccc4F)=O)C3)=O)CC2)cc1 CCCCCCN=c1ccn2nccc2[nH]1.C(=O)CC1CC1 C1(CNC(CC(C)(C)OC)=O)CC2CCC1N(C(C1CC=CCO1)=O)C2 C1(CC(=O)NCCNC(c2cccc(CC3CCC3)c2)=O)CCC2CC2C1 C1(C(N2CC(NC(c3cc(C4CCOCC4)on3)=O)C2)=O)(COC)CCNC1=O c1(NC(N(C2CCCCCC2(C)C)C)=O)nccn2c(I)cnc12 C(=O)(C1=NN(C)C(=O)CC1)NC1CCCC(CN(C(C2(CC#C)CCC2)=O)C)C1 CN1CCC(O)(CNC(=O)CC2CC(NC(c3ccncc3O)=O)C2(C)C)CC1 Cc1ccn(C(C)C(=O)NC(C)C(=O)N2CCCC2)n1 Cc1cc(Br)cc(F)c1CN1CCOC(C(F)(F)F)CC1.CC(C)SC c1(C(N(C2CCN(C(=O)C#CC3CC3)C2)CCC)=O)cn2c(n1)CC(C)CC2 N1(C(=O)CC2CNCCO2)CCC(CCF)(C(=O)O)CC1 c1(CN=C(NC(C#C)CCC)NCC(C)(O)c2cccs2)c(C)cc(F)cc1C c1(Nc2ccc(CCCNC(C(CC)CC)=O)cc2)ccc(S(=O)(=O)NC)cn1 C1(NC(c2ccc(C(C)C)cn2)=O)CC2CN(C(c3cc(Cl)no3)=O)CC2C1 c1(C(N(C)CC2N(C(C(CSC)C)=O)CCCC2)=O)cc(C)cc(N)c1 C(=O)(CCCC(=O)N1CC(NC(=O)Cc2ccccc2)C2CC12)OCC N1(C(C(C)Oc2ccccn2)=O)C2CCCC1CN(C(c1ccsc1C#N)=O)C2 N1(C(C2C(c3n(C)cnc3)C2)=O)CCN(C(C2C=CCCC2)=O)C(CCO)C1 C#CCC(CC(F)F)OCC(=O)NC1CC(NC(C2CCC(O)CN2C)=O)C1 C1(CC)CCN(C(=O)C(C)N2CC(C)C2)C1C(=O)NC(CO)C(F)(F)F CC1(C)CN(C(C2(F)CCCN(C(=O)COCP(C)(C)=O)C2)=O)CC1CO c1(C(N2CC(NC(c3[nH]cc(CC)c3)=O)C2)=O)ccc(S(=O)(=O)CC2CC2)cc1 N1(C(C(C)C(C)(C)C)=O)CCN(C(=O)COc2ccc(O)cc2)CC(C)(F)C1 CCC(CC)CC(F)C(=O)N1CC2(CCCC2NC(c2cc[nH]c(=N)n2)=O)C1 N1(C(c2nc(NC)c([N+](=O)[O-])cc2)=O)CCOCC1C1CCCO1 n1(CC#C)c(C)cc(C(=O)NCCCC(C)NC(=O)CCS(N)(=O)=O)c1C C(=O)(C1=CCCOCC1)N1CCC2(C)C1CN(C(c1cn3cccnc3n1)=O)C2 C(=O)(C1=COCCC1)N1C(C)CC(CNC(c2ccc(OCC(F)F)cn2)=O)C1 N1(C(COC)=O)CC2CCC2(CCNC(=O)CCP(C)(C)=O)C1 C(=O)(C(C(C)(C)C)C1CCC1)NC(CC)CNC(=O)CC(C)CN(C)C C12(NC(C(CC=C)(C)CC)=O)CCCC1N(C(c1cc3sccc3[nH]1)=O)CCC2 C(C)(C(C(=O)NC1CC(SC)C1)C(C)C)NC(c1c(CC)ccs1)=O c1(CC(C)Nc2nc(CS(C)(=O)=O)cs2)cscc1Br N1(C(C(C)(C)OCC)=O)CCCN(C(=O)CC2CC2Cc2cccs2)C(C)C1 C1(NC(C(CCC)C)=O)CCCC12CCN(C(=O)C(F)C(F)(F)F)CC2 C1(CNC(C(C2CCOC2)OC)=O)CN(C(=O)CC(C)C(C)C)CC(C)(C)O1 C1(C(N(C2(C(N3CCOCC3CCO)=O)CC2)C)=O)CCC(F)(F)C1 N1(C(C(c2cc(C)sc2)(C)C)=O)CCC(CNC(c2ccc(N)cn2)=O)C(O)C1 C(=O)(C(C)(CNC(c1cc(F)ccc1F)=O)CC)NC(CC)CN(C)C C(=O)(C1CC=Cc2ccccc21)NC(C1CCCN(C(=O)CN(C)CCO)C1)C CCC(C)CC(=O)NCCN(C(=O)CCCc1ccccc1)CCCN(C)C N1(C(C(F)=C(C)C)=O)CCOCC(NC(=O)CC2(C#N)CCOCC2)C1 C1(CNC(c2ccn(C(C)(C)C)n2)=O)CCCCC1NC(=O)C(F)CC1CC1 c1(C(=O)NC23C(n4cc(CC(C)(C)O)nn4)CC(CC2)C3)cnc2ncccn12 C(C(=O)N1CCC(C(N2CC(N(C)C)C(C)C2)=O)O1)c1c(CC)cccn1 c1(N(CCC2CCN(C(c3c(C)cns3)=O)CC2)C)cc(=O)n2ccccc2n1 C1(CC(=O)NC(CN(C(C(CC)OC)=O)C)(C)C)CC2CCC(C1)N2C c1(C(C)NC(C(N2C(CC(=O)OC)CCCCC2)=O)=O)ccc2c(c1)OCCO2 C(C1CCCc2cccnc21)NC(CCn1cc(-c2c(OC)scc2)nn1)=O.C(C)(=O)O CC(C)(CNC(=O)Nc1ncc(-c2ccc(F)cc2)cn1)C1=CCOCC1 Cc1cc(C(=O)OCc2ccn(C3CCCC3)n2)nn1C(C)(C)C C1(OC)(Nc2ccc(CC(=O)N3CCC3)cc2)CCN(C)C1 N1(C(C2(CC#C)CCOC2)=O)CC2(NC(=O)CCc3cc(OC)no3)CC1C2 c1(C(=O)NCCCN(C(CC2CC(=C)C2)=O)C2CC2)cccc(C2CC2(F)F)c1 N1(C(CCC2CCN(C(c3c(C)nn[nH]3)=O)C2)=O)CCC2(CNC(=O)O2)C1 c1(C2CCN(C(c3[nH]nnc3C)C(=O)NCCOC)CC2)nc2ccccc2s1 Nc1c(C(=O)NCC2CC(NC(C3(F)CC4(CCC4)C3)=O)C2)cccc1[N+](=O)[O-] c1(CC)cnc(Cl)nc1N1CCC(NC(C2CC(OC)(OC)C2)=O)C(F)C1 N1(C(CCC=C)=O)CC(C)C(C)(C(N2CCC(C=C)C2)=O)C1 CC(C)C(C)C(CNC(=O)CCNC(=O)C(C)(C)C)NC(c1nc(Cl)cs1)=O C(=O)(CCCN=[N+]=[N-])NCC1C(CNC(C2N(C)CCC2)=O)C1 c1(C(=O)NCC2CCN(C(C(CN(CC)CC)F)=O)CC2)cccn2cncc12 C1(NC(C(C2CCC2)OCC)=O)CC2C(NC(c3cc[nH]n3)=O)C2C1 C1(CNC(C(COC)(C)O)=O)CC2CCC(C1)N2C(c1c[nH]c(C(N)=O)c1)=O c1(C(N2C(C(=O)OC)CCC2)=O)cccc(C(F)(F)F)n1.Cc1nnc(N(C)CCO)o1 C1(C(N2CCCCC(NC(Cc3nc(C)[nH]n3)=O)C2)=O)CCc2ncncc2C1 c1(N)nc[nH]c(=NCC2(OCCN(CCCOC(C)C)C)CCCOC2)c1C N1(C(c2c(C)nc(C3CC3)o2)=O)CCC(F)(CNC(=O)Cn2cnnn2)CC1 c1(C(N2CC(C3(C)N(C(CCC)=O)CC3)C2)=O)ccc(C)nc1 N1(C(C2CCC(NC(c3c(C)cc(F)s3)=O)CC2)=O)CCC2(C1)CN(C)C2 c1(C2CCN(C(COc3c(C)cccc3)=O)CC2)cccc2c1OCCO2 N1(C(CC(CC)NC(c2cnn(C)c2Cl)=O)=O)CC(C)(C)OC(C)(C)C1 c1(OC)cc(Br)c(Cl)cc1NC(N1CC2(CCCN2c2ncc(I)cn2)C1)=O CCC(CNC(C1OC2CCC1C2)=O)(CC)C(=O)NC1CCCCCC1C c1(CNc2ccccc2)ccc(Br)cc1.CC(CC(=O)N1CCCCC1)N1CCOCC1 CC1COC(C(=O)NC(C)CN(C)C(c2cn(CC(F)(F)F)cn2)=O)C1 c1(N(CCOCC)C)nccc(-c2ccccc2F)n1 c1(OC(C(=O)NC(CN(CC)Cc2cnn(C)c2)C)C)ccc2c(c1)CCC2 c1(C(N(C(C)C)CCNc2ncnc3sccc23)=O)cnc(O)c2ncccc12 C(=O)(CCCC(C)O)NCC1C(NC(c2c(C)nc(CC)o2)=O)CCC1 Cc1ccc(C(=O)NCC2(O)CCN(C(=O)C(n3cc(C)cn3)C)CC2)c(C)c1 N1(C(=O)CCC2CCCN(C(C3CC3C3CC3)=O)C2)C2CCC1COC2 c12ccc3nc(C)c(n3n1)OCCNC2.C(CC(=O)OCC)NC(C(=O)NCC)=O C(N=c1[nH]cnc2c1CCC2)C1CN(C(C(C)NS(C)(=O)=O)=O)C1 C1(C(N(C2(CC(=O)NCC3(C)CC4(CC4)C3)CC2)C)=O)CC12CCOCC2 CN1CCC(CC(N2CCOC(CNC(=O)Cc3cn(C)nc3Cl)C2)=O)C1=O c1(C(=O)NC(C)CN(C(=O)CC2CCC2(F)F)C)ccc2c(c1)CCCCN2 c1(C(=O)NCC2N(C(C(CCC)(C)CC)=O)CCC2)c(OC)c(Cl)cc(O)c1Cl N1(C(C2(F)CCN(C(CN(C(C)C)C)=O)C2)=O)CCCC2CN(C)CC12 Cc1cc(O)nc(C)c1C(=O)NC1COC2(C1)CN(C(C1CC(C)(C)CO1)=O)C2 C1(NC(=O)C(Cl)=CCl)CN(C(=O)CSCc2ccc(F)cc2)C2(CCCC2)C1 C(CNC(c1cscc1C)=O)(CCOC)NC(COCCCC)=O c1(C(=O)NCC=CCNC(C(C)(C)COCC(F)F)=O)cc2n(n1)CCCC2O C1(CCNC(c2ccc(C3CC3)s2)=O)CC(F)(F)CN1C(C1C2CCCOC12)=O N1(C(c2c(C)cn(C)n2)=O)CCN(C(=O)CNC(c2cccc(F)c2)=O)C(C)C1 c1(NC(C2CN(C(c3cc(Br)nc(Br)c3)=O)CCO2)=O)cccc(F)c1F O(NC(=O)CC(C(F)F)NC(C1(C)CC2C=CC1C2)=O)CC(=O)N(C)C c1(OC)ncc(CN2CCCC(C(C)NC(=O)C(C)c3cccs3)C2)cn1 c1(N2C(C(C)(C)C)CCC2)cc(CN(C(C(C)NC(N)=O)=O)C)ncn1 c1(C(=O)NC2(C)CC(NC(C(C)O)=O)C2)cc2sc(F)cc2[nH]1 c1(C(CC)NCCC2CCCO2)ccc(I)cc1 c1(C(N2CCC(C3CCCN3C(c3ccc(O)nn3)=O)C2)=O)ncc(F)cn1 c1(CCC(=O)N(C2CC(NC(CCc3ccc(C)s3)=O)C2)C)ccccc1CO C(=O)(C(C)C(O)C(C)C)N1CC(CC=C)(NC(c2c[nH]nc2[N+](=O)[O-])=O)C1 C=C(C)C(CC(=O)Nc1cccc(NC(=O)NC(C)(C)C)c1)OCC C1(COC)CN(C(=O)C(O)P(C)(C)=O)CCN1C(=O)C1=CCCSC1 c1(C(=O)NCCCN2CCN(C(C3(C)CC3(F)Cl)=O)CC2)cccc(N)c1O c1(CN(C(=O)C(C)c2ccsn2)CC(C)C)cn(CC(=O)O)nn1 c1(C(=O)OC)nc(N2CC3CN(C(c4cc(Cl)ccn4)=O)CC3C2)c(F)c(Cl)n1 C1(NC(C(=O)NCC)=O)CN(C(=O)C(n2nnnc2CC)C)CC12CCOCC2 N12CCc3cc(ccc31)CNC2=O.C1(c2nn[nH]n2)(C(C)(F)F)CC(F)(F)C1 n1(CC)nc(C)cc1C(N1CCCC1C(=O)NC1CC1(C)C(F)F)=O CCC(C)(C)C(C)CC(=O)NCC1(OC)CCN(C(c2cnc(N)c(Cl)c2)=O)C1 Cc1cc(C(=O)NCC=CCNC(=O)C(C(C)O)NC(=O)C2CC2)ncc1CO c1(CC)ccc(C(=O)NC(CNC(=O)CCCc2ncco2)C(C)C)c(O)c1 CCC(CC(F)F)C(=O)N1CC2(CC2)CC1CNC(=O)COc1cc(C)on1 c1(NC2(CNC(C3CC(CCC)OCC3)=O)COC2)nccc2occc12 Cn1cc(Cl)cc1C(=O)NC1(CC(N2CC(O)C(O)C2)=O)CCCCC1 c1(C(N)=O)ccc(CNC(=O)Nc2ccc(C3CCC3)nc2)cc1 C(=O)(CC(CC)SC1(O)CC(C(=O)NC2CC2)C1)Nc1csc(C(=O)OCC)c1 CN1CCN(C(=O)Cc2ccns2)C(CNC(=O)COC2CCCOC2)C1 C1(C(=O)NCC(CCC)C)COc2ccccc2CN1 C1(NC(C2CC(OCC)C2)=O)CN(C(c2cc(C)n(C)c2)=O)CC1N=[N+]=[N-] C(C)(C)(C(=O)NC(C)CCNC(=O)C(O)CSC)OCC CC(C)C(C(=O)OC(C)(C)C)C(=O)NCC(C)NC(c1cc2n(c1)CCCC2)=O C1(C(=O)NC2C(CNC(CSS(C)(=O)=O)=O)CC2)CCCCC1 C(C(C)(C)CC(=O)NC)NC(C(CC1CN(C(C(C)OCCC)=O)C1)F)=O CC(C(F)C(=O)NC1CCN(C(=O)CCc2cnn(C)c2)C1(C)C)C(F)(F)F c1(OC)ncc(C(N2CCOC(C(=O)NCC(C)C(=O)OC)C2)=O)cc1F c1(C(=O)NC(CC=C)CNC(=O)CCCn2ccnc2)cnn(CCC)c1Cl c1(C(N2CCN(C(c3cc(Cl)cs3)=O)CC2CCO)=O)ccc2c(c1)CCCS2 C(CCCCC(=O)NCC1CC12CCOCC2)N(C(C1C(C(C)C)OCC1)=O)C N1(Cc2c(C)cc(F)cc2)CCC2CC(C(=O)NCC(O)CO)C2C1 c1(C(=O)NCC2(OC)CCN(C(C(C)N(C)CC)=O)C2)nc2ccccc2s1 c1(C(=O)NCC(C(C)C)NC(C(CC)OC)=O)cc2ncc(C)cn2n1 c12n[nH]c3c1CN(CC3)C(=O)CC2.C(C(=O)OC)(=CC)OC N1(Cc2cn(C(C)C)nc2)CCC(NC(=O)Cn2ccsc2=N)CC1C N1(C(C2CC(CCC)C2)=O)CC2CCCCC2(CNC(c2cncc(C)c2)=O)C1 Cc1cccc(-n2cc(C(C(C)C)NC(N)=O)nn2)c1Br.C1C(=O)N1 C(=O)(C(C)(F)C(C)(C)F)NCC(C)C(=O)NC1(C)CCCCCC1 N1(CC(C)(C)SC(F)(F)F)CCN(C(=O)CO)C(CCO)C1 N1(C(CC(=O)NCC#C)=O)C2CCCC1CC(CNC(=O)C1=NOC(C)(C)C1)C2 c1(CC(=O)N(C2CCN(C(=O)C(C)NC(C)=O)C2)CC)ccc2c(c1)CC2 C1(c2ccc(CC)o2)CCCCCN1CCc1cscc1Br CCC(C)C(O)C(C)C(=O)NCCc1cc(C(N2CC(C)CCC23CC3)=O)no1 c1(NC(c2c(C(=O)N(C)C)ccc(C)c2)=O)cc(C#N)ccc1C CC1C=C(C(=O)N(C(C)CN(C)C(c2csc(C3CCCC3)n2)=O)C)CC1 C1(COC)CN(C(c2ccnn2CC(F)(F)F)=O)CCN1C(=O)CN(C)C(C)=O CC(CN(C)C)C(=O)NCCSCc1cn(C2CCCC2)nn1 CC(C)C(C)(C(N)=O)NC(=O)C(CN(C)C)NC(=O)CN=[N+]=[N-] C(=O)(C(CCC1CC1)N(CCC=CCO)C)ON(C(C)(C)C)CCC N1(C(C2=CC(C)(C)C2)=O)CCN(C(c2cc(Cl)cc3c2CCC3)=O)C2COCC12 N1(C(C(C)CC2CCCCC2)=O)CCN(C(=O)Cc2cncnc2)CC12CC2 c1(OC)nccc(C(=O)NC(CCN(C)C)C(=O)NCC2CC(OC)C2(C)C)n1 c1(C(=O)NC2(C)CC(NC(=O)CCc3cncnc3)C2)ncn(O)c1Br c1(N2CCC(C)C(NC(=O)CCC(F)F)C2C)nc2ncc(Cl)cc2o1 N1(CC(C)C2CC2)CC2(CCOCC2)C1C1CC(NS(N)(=O)=O)C1 C1(CCNC(=O)C=CCO)COCCN1C(c1ccnc(-c2ccncc2)c1)=O C(CN=[N+]=[N-])(C(=O)NC(C)C(C)F)NC(c1c(Cl)cc(C)s1)=O c1(C(N2CC(N(C)C(c3cccc(F)c3N)=O)C(F)C2)=O)cc2cccnc2s1 CC1CC(NC(C2(O)COC2)=O)CCN1C(c1ccc(C(F)(F)F)c(O)c1)=O C(C)(C(=O)N1CCCCO1)n1cc(CNC(COC)=O)nn1 N1(C(c2cc(C)c(O)nc2)=O)CCC(C)N(C(C2CC3CC3C2)=O)CC1 C1(CNC(C2(CF)CN(C(c3n(C)ccn3)=O)C2)=O)CCCC(F)C1 CCCCC(C(=O)NC(C)(C)C)NC(c1c[nH]nc1OC)=O.C1(N)CCN(C(C)=O)C1 N1(C(c2cc(CC)nn2C)=O)CCCN(CCNC(C2(CO)CCCO2)=O)CC1 c1(C(=O)NC2CCN(C(CC(=O)Nc3nccs3)=O)CC2)n[nH]c2c1CCC2 c1(C(=O)NCCN2CCN(C(c3nc(C)oc3C)=O)CC2)ccc2oncc2c1 C1(C(=O)NC)(OC(C2C(C(=O)OCC)CC2)=O)CCOCC1 c1(CCC(=O)NC(C)C(C)NC(c2cc(C#N)c[nH]2)=O)nnc(S)nc1O c1(CC(=O)NCC(CC=C)NC(=O)C=NOC)cccc2cnccc12 C(=O)(C(C)(C)c1nncn1C)NCCC(C)N(C(=O)CCCN(C)C(C)C)C Cc1nsc(C(N2CCC(C(=O)NC3CCC4CCC34)C2)=O)c1N N1(C(CCC=C=C)=O)CCCC2CN(C(c3cc(C(N)=O)cn3C)=O)CC12 C(C)(CCC(=O)N1CCCC1CNC(c1cnc(C2CC2)o1)=O)OC Clc1cccc2c1OCC2NC1CC1.c12ccc(nc1)N1CCN(CC1)C2 C1(CNC(C(n2c(C)ncc2)C)=O)CCCCC1NC(c1cnc(O)o1)=O c1(C(N(CCn2cc(C(N3CCOC3=O)C)nn2)CC)=O)cnc2[nH]cncc1-2 c1(C(=O)NCC(CCCC)NC(C2(C(C)(C)O)CCC2)=O)c[nH]c(C)c(Cl)c1=O C1(C2CCC2)(C(=O)NCC(C2CC2)NC(c2cc(O)cs2)=O)CC1(F)F N1(C(C(C)OCCC=C)=O)CCN(C(=O)C2CCc3c[nH]nc32)CC(C)(C)C1 CC1(NC(=O)Cc2ccns2)CCN(C(C2(C)CC(C#N)C2)=O)C1 N1(C(COCCC(C)C)=O)CCC2CN(C(c3ccc4c(c3)CCN4)=O)C2C1 C1(NC(C(COC)C)=O)CCN(C(C2CC2c2ccc(C)cc2)=O)CC1 N1(C(CC(C(C)C)C)=O)CC2(CCC(CNC(C34CC(CO)(C3)C4)=O)O2)C1 c1(NC(C2CCCCN2C(=O)NC2CN(C(=O)C3CC3)C2)=O)cccc(Cl)c1 C1(NC(C(=Cc2ccncc2)C)=O)CC12CCN(C(c1cc(F)c[nH]1)=O)C2 c1(C(=O)NC2(CNC(=O)CC3(O)CCC3)CC3CCC2C3)ccn2nccc2n1 N1(C(CCCCOCC)=O)CCCCC12CN(C(=O)Cc1cc(C)on1)C2 Cn1c(C(=O)NCC(C2CC2)NC(=O)CNC(C2CCOCC2)=O)cnc1[N+](=O)[O-] N1(C(C2CCCC(NC(COCCC=C)=O)CC2)=O)CCCC(OC)CC1 N1(C(c2cc(C)c(C)s2)C(=O)NCC2CCOCC2)CC(C)(C)C2COCC12 C1(N=[N+]=[N-])(C(N(CCC)CCO)=O)CCN(C(=O)C(F)CC2CCOC2)C1 c1(C(=O)NCC(CNC(c2c(C)cc[nH]c2=N)=O)F)ccnc2ccc(F)cc12 S(=O)(=O)(c1cn(CC(C)C)nc1CC)Nc1c(C(=O)OCC)ncs1 N1(C(C2C(C(C)C)C2)=O)CC(CNC(=O)Cn2cc(Br)cn2)C2(CC2)C1 c1(OC)ncc(Br)c(C)c1C(N1CC2(CCC(NC(=O)Cc3cc[nH]n3)C2)C1)=O c1(CNC(C2COCC2NC(=O)CCCF)=O)ccncc1 c1(OC)cc(C(=O)O)ccc1OCCNC(=O)C(c1ccc(F)cc1C)(C)N N1(C(C=CCCNC(CCOCCOCC)=O)=O)CCC(OC)CC1C C1(C)(CNC(c2cnc(OC)nc2)=O)CCC(NC(=O)CC2CC23CC3)CC1 c1(N(C2C=CCN(C(COC)=O)C2)CC(O)COC)cc(F)cc(F)c1 Cc1cc(=NC2C(C)CN(C(c3ccnc(CO)c3)=O)CC2C)[nH]c(C2CC2)n1 CC(C)CS(=O)(=O)CC(=O)NC1CC1NC(c1ccc(=O)n(C)c1)=O N1(C(c2cc(COC)on2)=O)CCC2(NC(=O)C(F)CC(C)C)CCCCCC12 N1(C(c2nc(CCOC)oc2)=O)CCCCC1C1CCN(C(=O)C(C)=C(C)C)C1 N1(C(CC2(OCC)CC2)=O)CC(C(N2CC(O)(COC)C2)=O)C(F)(F)C1 C(=O)(C(F)(CNC(=O)CN1C(=O)CN(C)C1=O)C(C)C)NCCOCC(=C)C C1(NC(c2ccc(OC)s2)=O)CC(O)CN(C(c2nocc2C)=O)C1 c1(C(=O)NCC(C)C(=O)NCc2ccc(=N)[nH]c2)cccc(O)c1 C=CCC(C)(C)C(=O)NCc1ncc(C(=O)O)s1 Cc1cc(C)c(C(=O)N(CC(C)NC(c2ccc(C#N)cc2F)=O)C2CC2)c(=O)o1 C1(CCNC(c2nnc(C)s2)=O)CC(F)(F)CN1C(c1cccc(C(F)F)n1)=O CC1=C(C(=O)NC(CC(N)=O)C(=O)NC(c2nc(C)ns2)(C)C)CCO1 Cc1nc(N2C3CN(S(=O)(=O)Cc4ccccc4)CC23)c2c[nH]nc2n1 C1(CNC(CC(=O)NCC)=O)CN(C(c2c(Br)noc2C)=O)CCO1 Cc1nc(C(N2CCCCC2CCNC(=O)C(C2CCCCC2)O)=O)c(C)s1 C1(CC(=O)N(C2CCN(C(c3ccon3)=O)CC2)CC)CC2(CCC2)CCO1 c1(C(=O)NCC2(O)CC(CNC(c3c(C)occ3)=O)C2)cncn(C)c1=O c1(C(=O)NCCCNC(CC2CC(CC)OCC2)=O)c(C)nn(C2CC2)c1Cl c1(OC)nn(C)cc1C(N1CCCC(CC(=O)N(C2CCOC2)C(C)C)C1)=O CC1CC2CCC(C1)N2C(C1C=CCCC1CNC(c1occ2c1CCC2)=O)=O N1(C(c2cn(CCNC(Cc3ncn(C)c3)=O)nc2)=O)CCCC(CCO)CC1 c1(C(=O)NCC2C(N(C)C)CN(C(c3cnc[nH]3)=O)C2)nc2ncccn2n1 Cc1cc(C(=O)NC2CCN(C(=O)CCOc3ccc(F)c(Cl)c3)C2)nc(C)c1 c1(C(=O)NC2CN(C(=O)CCOC)CC2F)ccc2cncc(Br)c2c1 C1(C(N(CCCNC(C2CCOC2C(C)C)=O)CCC)=O)CCCC2(CC2)C1 CC(C)CC(C)CC(=O)NCCCCCNC(c1ccc2c(c1)CCC2)=O N1(C(CC=C=C)=O)CC(C(=O)NCC(C)CC(C)C)C2(CC2)C1 C1(C(N2C(C(C)NC(C(C)NC(COC)=O)=O)CCC2)=O)C(C)(C)C1(C)C C#Cc1cnc(C(N2CCC(C3CC3)C2C(=O)NOCC2CC2)=O)c(C)c1 CC(CC(C)(C)C)C(=O)NCCCO.C1(N2CCC2=O)CCN(CC2CC2)C1 C(=O)(CCCC(C)(C)NC(C12CCCCC1C2)=O)NCCC(C)(C)OC N1(C(C#CCNC(c2ccn(CCC)n2)=O)=O)CCC(C2CCC2)C1 C1(C(=O)NCCC(C)(C)C)(CNC(C(C)OCCC=C)=O)CC=CC1 C(=O)(C1=NNC(=O)CC1)NC(C1N(C(c2cc(C)nc(C)n2)=O)CCC1)C N1(C(C2(C(N(C)C)=O)CC2)=O)CCCCC2(C1)CN(C(=O)Cc1ccn(C)n1)C2 c1(COC)ccc(C=CC(=O)N(C(C)CN(C)C(C2CC2CF)=O)C)cc1OC c1(CN(C(C2CCCN2C(=O)C=Cc2cccs2)=O)C2CC2)ccccc1 Cc1csc(C(C)C(N2CCCC2CN(C)C)=O)n1.C1CCNC(=O)C12CC2 Cc1ccc(C(=O)CN2CCCC(NC(C)(C)C)C2)cc1C.N12CCCC1C2 CC1CCN(C(C2(C(C)(C)C)CCC2)=O)CC1CNC(c1nccc(N)c1Cl)=O c1(C2(C)C(NC(C3(c4c(C)cccc4)CCCC3)=O)C2)cc(Cl)ccc1Cl N1(C(CSc2onc(C)n2)=O)CCN(C2CCCN(C(=O)OC(C)(C)C)C2)CC1 CC(C)(C)CC(F)C(=O)NCC1(C(N2CC(CC3CC3)C2)=O)CCCCC1 N1(C(c2cc(OC)ns2)=O)C2CCC1CN(C(=O)C(C)(O)C1CC1)C2 O=C1CCC(C(=O)NCC23CC2CN(C(=O)CC2CC2)C3)n2cccc21 Cc1nc2ccc(C(=O)NC3CN(C(C4CCN(C)CC4)=O)CC3F)cc2n1C C1(C(=O)NCCCC(C)C)CCCC(NC(=O)C=CC2CCCN2C)CC1 N1(C(C2C(COC)C2)=O)CCN(C(=O)C=Cc2cncc(O)c2)C(CCO)C1 Cc1sc(=O)n(CC(N2CCC(NC(C3CCN(C)C3=O)=O)C(O)C2)=O)c1C CC(C)C(CN(C)C)C(=O)NC(C)CC(=O)N1C(CO)CC1CO c1(NC(C2(NC(C3=CC(=O)CC3)=O)CC2)=O)cncc2ccccc12 N1(C2CC3N(C(c4ccc(C)c(Br)c4)=O)C(CC3)C2)CCCC12CCNC2=O C(CCOCCO)(C(=O)NCCSCCO)NC(C1C(CCC)C1)=O C#CC1(O)CC(C(N2CCC(CN(C(C(=O)NCC)C)C)(CO)C2)=O)C1 CC1=C(C(=O)NC2CN(C(=O)C3COc4ccccc43)C2)Cn2ncnc2N1C C(=O)(CCCCN=[N+]=[N-])NC1(C)CCN(C(=O)C#CC2CC2)C1 C12(CNC(C3(CNC(C4COC(=O)N4C)=O)CC(=C)C3)=O)CCCN(CC1)C2 n1(C(CC)CC)nc(-c2ccc(Cl)o2)nc1Cc1ncc(C)o1 Cc1ccc(NC(C2CC3CCN(C2)C3)=O)c(-n2cc(C3(C)CC3)nn2)c1 CS(=O)(=O)c1ccc(Cl)c(C(=O)NCC2CN(C(C3(F)CC3)=O)CCO2)c1 C(=O)(C(CC(C)C)C(N)=O)N1CC(NC(C2CC3(CC(=C)C3)C2)=O)(CO)C1 C(=O)(C#CC1CCCCC1)NC(CN(C)C)C(N1CCC2(CCOC2=O)C1)=O C1(NC(CSCC=C)=O)CN(C(=O)CC(C)C2CCCCC2)CC2(CCC2)C1 C(=O)(C1=CC2CCCCCC12)N1CC(CNC(=O)CC2CC3(CCC3)C2)C1 c1(NCC(C)(CO)NC(CNC(C(CC)C)=O)=O)nccc(OC)n1 N1(C(COC)=O)CC2(NC(=O)C(C3CCCN(CCOC)C3)=O)CC1C2 N1(CC)CC(C(=O)NC2CC(NC(=O)C=CC(=O)N(C)C)C2)NC1=O c1(N(C)CC2CC(C)C2)nc2cc[nH]c2c(=NC2CC2c2ccccc2S(C)=O)[nH]1 CC(C)C(C(=O)NCC1CC(F)(CNC(=O)CCn2cc(Cl)cn2)C1)N(C)C C(=O)(C#CC1(C)CCCO1)N(C1CCC(NC(C(n2c(C)ncc2)C)=O)CC1)C C1(NC(CC=CCC)=O)CN(C(=O)CC2CCC(F)(F)CO2)CCC1O CCC(C(=O)OC)C(=O)NCc1csc(C(=O)NC2CC2c2cnn(C)c2)c1 N1(C(C(C(C)(C)C)OC)=O)CC2CCC1C1CN(C(=O)Cc3ccoc3C)CC21 Cc1cnncc1C(=O)NC(CNC(=O)CCCNC(=O)C1CC1)CC(C)C CCCCCCCN(C(=O)CCN(C(=O)CCc1conc1C)C(C)C)C N1(C(CCCCOC)=O)CCN(C(c2ccc(=N)[nH]n2)=O)C2CCCCC2C1 CCC(C(C)(C)C(=O)OC)NC(=O)CCCCCn1cc(C(O)C(C)C)nn1 O=C(CCCCC(F)(F)F)NCCC1CCN(C(=O)C(F)OC(F)(F)F)C1 CSC=CC(=O)N1CCC(OCCNC(C2(F)CCOC2)=O)C1 CCC(O)C(C)C(=O)NCC(O)CNC(=O)C=CC(c1ccccc1)=O CC1(NC(=O)CCC2CCCCN(C(=O)CCCC3CC3)C2)CCCC1(F)F n1(CC(=O)N(CCN(C(C=C(CC)C)=O)C(C)C)C)ccc2c(C)cccc12 Cc1cc2cc(CNC(c3cc(Cl)ccc3OCc3ccccc3)C)ccc2[nH]1 C1(NC(Cn2cc(-c3c(N)cc(F)cc3)nn2)=O)CCC2CCCC1O2 c1(C(N2CCCC3(CC3)C2)C(=O)NCCCCCC)ncc(Cl)cc1F N1(CC(N2CCC(C)C(CNC)C2)=O)CCc2sccc2C1.C(=O)(CNC=O)N c1(C(=O)NC2CN(C(c3cc(C)on3)=O)C(C)C2)cc(=O)c2ccc(Cl)cc2o1 CCC1=NOC(C(=O)N(CCC(N2CCC(COC(C)=O)C2)=O)C)C1.CCO C(CCCN=[N+]=[N-])NCCNC(CNCCOCCOCC#C)=O Cc1ccc2ncc(C(=O)NC3CC4CCC3(NC(=O)C(F)C3CCC3)C4)n2c1 Cc1cc(=NCC2CN(C(c3ncc(F)cc3F)=O)CC23COC3)[nH]c(Cl)n1 C(CN=c1[nH]c(N2CC3CCC3(C)C2)nc2c1CCC2)SC c1(SC)cc(N2CCCC(CNC(=O)CCc3cnc[nH]3)CC2)nc(SC)n1 C1(C(=O)NC(C)CCCNC(=O)CCCc2n[nH]c(=N)s2)CN2CCC1(C)CC2 C(CC(=O)NC1CCN(C)CC1C)(C(C)OC)NC(c1cc(CC)nn1C)=O c1(C(=O)OC)ccc2c(c1)CC(C)N2C(c1ccc2cnc(C)cc2c1)=O Cc1cnc2c(cnn2CC(=O)NC2CN(C(C34CSC(C3)C4)=O)CC2C)c1 Cc1c(C(=O)NCCCNC(C2CCCO2)=O)cc(CC)n1C.C1(C(N)=O)CC1CS c1(OC)cnc(C)cc1C(=O)NCCCc1ccc(-c2scc(O)c2C#N)cc1 CCC(O)(CC(=O)Nc1cccc(NC(c2nsnc2O)=O)c1)c1ccccc1 c1(CC)c(C(=O)NCC2(CO)CCN(C(C3CC3F)=O)CC2)cccc1F C=CC(F)(F)C(=O)NCCC1CC(NC(=O)CCNc2ccccc2)C1 C=CCC(CC)NC(=O)C(F)C1CC(NC(=O)C(C)(C2(C)CC2)OC)C1 Cn1ccnc1CC(=O)NCC(C)(C)CNC(=O)CCc1ccsc1 c1(C(N(C)CC2N(C(C(CCC)(C)C)=O)CCCC2)=O)c2c(nn1C)CCSC2 NC1CCC12CCC(C(=O)Nc1cnc(C3CCC3)o1)CC2 Cc1nc2cc(C(=O)Nc3ccc4c(c3)CCCC4)c(F)cc2[nH]1 c1(OC)cc2cnccc2cc1C(=O)NCC1CCC2(CCCCC2)O1.O C1(NC(c2ccc(NC)cc2)=O)CN(C(c2c[nH]nc2C(F)(F)F)=O)CCC1C c1(OCC(=O)N(CC(C)O)CCNC(=O)C(O)C2CC2)nc(Cl)c(Cl)cc1Cl c1(C(=O)NC(CNC(c2cc(C)cc(O)n2)=O)CC(C)C)ccnc2[nH]nnc12 Cc1ccnc(C2CCN(C(=O)C(N3CCCC(CNS(C)(=O)=O)C3)=O)C2)c1 c1(C(N2CC(C)(C(=O)NC(C)CCO)C2)=O)ccc(F)cc1Br N1(C(C2OCCN(C)C2)=O)CCCC2(C1)CN(C(c1nn(C)cc1N)=O)CCO2 C(=O)(CCS(C)(=O)=O)NC(CCOCC)C(=O)NCC(O)C(F)(F)F N1(C(CC2CC(C)C2)=O)CCN(C(=O)C(F)(F)CCn2cccn2)CC2(CC2)C1 c1(C(=O)OC)cncc(C(N2CCCC2CNC(c2c(Br)cnn2C)=O)=O)c1 c1(OC)nccc(C(=O)NC2CC(C(=O)NC3C=C(C)CCC3)C2(C)C)n1 C#CC(C)(C)C(=O)NC1CC(NC(c2n[nH]c(COC)c2C)=O)C1 c1(OCC)c(C(C)NC2CCN(c3ccc(Cl)cc3)C2)c(C)nn1C c1(C(C(=O)NC2CCC(NC(C3CC=CC3)=O)CC2)O)ccc(Cl)c(F)c1 c1(Cn2cc(Cn3ncc(C)c3)nn2)ccc(CNCc2cccc(F)n2)cc1 Cn1cnc2cccc(C(N3CC4CCC3CN4C(=O)CC3CNC(=O)O3)=O)c12 C=C(Cl)C(C)(C)C(=O)N1CC(CC(C)NC(=O)COCc2ccccc2F)C1 CN1CCOC(C(N2CCC(C)(CCNC(c3c[nH]c(=N)s3)=O)C2)=O)C1 c1(CNC(CCCC#C)c2nnnn2C2CCOC2)c(F)cccc1Br C1(CC(=O)NC2CCC(F)(F)C2)CC2(CC2)CN1C(=O)CCc1ccco1 c1(C(N(CC(=O)NCC(=O)NCCO)CCC)=O)sc(C)cc1C Cc1ccc(NC(=O)C(CNC(C2CCCC(C#N)C2)=O)N(C)C)cc1F c1(C(=O)NCCCCN(C)C(c2ccnc(CO)c2)=O)ccc([N+](=O)[O-])nc1 n1(CC(=O)NCC(C)NC(C(C)N(C)C)=O)cccnc1=O CCCC(CCCS(C)(=O)=O)C(=O)N(C1CCS(=O)CC1)CC(=O)OC N1(C(COc2ccn(C)n2)=O)CCC(O)(CNC(C2COC3(CCC3)C2)=O)CC1 CN1CCCC(C(C)(C)C(=O)OC(C2(CS(N)(=O)=O)CC(F)(F)C2)=O)C1 N1(C(Cc2c(C)cnn2C)=O)C2CCC1CC(NC(c1cc(O)nc(Cl)c1)=O)C2 c1(C(N(CCNC(c2c(C)n(CCN(C)C)nc2)=O)C)=O)cccc(F)c1C C12(C(=O)NCCC3(O)CN(C(C(CC)C)=O)C3)CCC(F)(CNC1=O)C2 C1(CCC)CN(C(=O)C(C)NC(=O)NC)CCN1C(c1cnn(C)c1Cl)=O Cc1ccc(CN2CCC(C(=O)Nc3ccc(I)c(C)c3)C(O)C2)c(Br)c1 C1(C(N(CC(C)NC(CCc2cc(C)[nH]n2)=O)C)=O)CCC(=O)N1C N1(C(C=C(CC)C)=O)CC(F)CC1CNC(=O)CCC1(C)CCC(=O)N1 Fc1cccc(-c2ncc(-c3nccn3CCOc3ccc(Br)cn3)s2)c1 Cc1nc(CNC(=O)CC2CCC2)oc1C(=O)N(C1CCC1)C1CC1 C(C(C)(C)CC(F)F)NC(C(c1ccccn1)NC(c1cc(OC)ns1)=O)=O C(CC(C)CCNC(C1(CF)CCC1)=O)NC(c1nc(C)[nH]n1)=O N1(C(C2CCN(C(C)=O)CC2)=O)CCC2(CC1)CCN(C(c1sncc1C)=O)C2 C=CC(CC)CC(=O)N1CC(CNC(c2cc(Cl)n[nH]2)=O)C(F)(F)C1 C1(CNC(c2c(CC)non2)=O)CCCN(C(c2cc(COC)cn2C)=O)CC1 c1(CN2CCCC2c2ccc(F)cc2)ccnc(O)c1.N12CCCCC1NC2=O C(=O)(C(=O)N=c1ccn(CC(=O)NC)[nH]1)NCCOc1c(C(CC)(C)C)cccc1 S(=O)(=O)(c1ccc(Cl)c(C(=O)O)c1)NCCNS(c1n(C)ncc1)(=O)=O C#CC1(C(=O)Nc2cncc(Cl)c2)CCN(C(=O)C(CN(C)C)CC)C1 C1(C(N2C(CC(N)=O)CCCC2)=O)C2CN(C(C3CCCC(=O)N3)=O)CC12 CCC(CCC(=O)NCCN1C(=O)CNC1=O)NC(c1ccc(Cl)cc1)=O c1(C(=O)NCCCCNC(C2CCC(c3cc[nH]n3)O2)=O)cc(CCCO)on1 C1(C(=O)NCCCN(C(=O)CS)C(N)=O)CCCN1C1CCC1.N1(C(C)C)CC=CC1 c1(N(C2CN(C(=O)Cc3ccccc3O)C2)C)ncc(F)c(C2CC2)n1 C#CCCCCC(=O)NCc1ccc(CCNC(=O)CC2CCC(C#N)C2)cc1 N1(C(COC(C)(C)C)=O)CCCC(CCNC(C2CC(C(N)=O)C2)=O)CC1 C#CCC(C)(C(=O)N(C)CCc1nccs1)NC(=O)CC1CC(CC)=NO1 c1(OC)ccc(C)c(C(=O)NCC2C(C)CCN2C(=O)Cc2cccc(Cl)c2)c1 c1(C(=O)NC(c2ccccc2Cl)C)cc(C2=CCC(C)(C)CC2)c2cn[nH]c2c1 C=CC(F)(F)C(=O)NC(C1CCCN(C(c2cc(F)n(C)n2)=O)C1)C N1(C(c2cn(CCCC)nn2)=O)CCC2CN(C(c3cocn3)=O)CCC2C1 c1(NC(N2CCOC(CC3CCCN(c4ccncc4)C3)C2)=O)ccc(F)cn1 N1(C(CC=CC)=O)CCC2(CC1)CC2(CO)CNC(=O)C(C(C)C)n1cncn1 c1(C(N2CCC(CC)C2C(=O)NCC2(CF)CCC2)=O)cc(O)cc(F)c1 C(=O)(C1CCCn2ncnc21)NCC1(OC)CN(C(c2cc(C)sn2)=O)C1 CC1=NOC(=O)C1CC(=O)NCC=C1CCN(C(c2cc(Cl)ccn2)=O)CC1 C1(C2CN(C(C3(c4cc[nH]n4)CC3)=O)C2)(NC(C(c2cccnc2)C)=O)CC1 N1(C(c2ccc(C)cn2)=O)CCN(C(=O)CN2C(=O)CCC2=O)CC1CCCCl c1(C(=O)NC2C(NC(c3c(C)nc(COC)s3)=O)C2)cc(SC)ccc1O c1(CNC(C2CNC(=O)N2)=O)ccc(C(N2CCC(N3CC(O)C3)C2)=O)cn1 C1(C(=O)NC(C)CN(C)C(C2(c3cc[nH]n3)CC2)=O)COC(=O)N1 N1(CCC)CC(C(N2CCN(C3CCN(C(=O)C(C)CC)C3)CC2)=O)CC1=O C12(C(N3CCC(NC(CC4CCN(C)C4)=O)C(O)C3)=O)C3C4C1C1C2C3C41C#N N1(C(CC(C)C(C)(C)C)=O)CCC2(CC1)CC(NC(=O)CCC1OCCO1)C2 n1(CCC)cc(C(=O)NCC(C)(C2CC2)NC(=O)CC2CC(CC)C2)nn1 C12(C(=O)NC(CCCC)CNC(c3sccc3C(C)C)=O)CC(C)(C1)OC2(C)C c1(C(=O)NCCCOCCNC(C(C2CCC(=O)N2)C)=O)cnn2c1NCCC2 CCCCC(F)C(=O)NCc1ccc(C(=O)NCC2COC(=O)N2)cn1 N1(C(c2nc(C)c(C)s2)=O)CCC(C(=O)Oc2c(Br)cnn2C(C)C)CCC1=O N1(CCNCCNC(C)=O)CCC(CCc2ccccn2)C1 C(=O)(C1CCCc2ccccc21)NCCC1CC(NC(c2cc(C#N)oc2)=O)C1 CCC(CC(=O)NCC1(NC(=O)Cc2ccn(C(C)C)n2)CC1)CC(F)(F)F N#Cc1ccc(OCC(=O)NCCC2CCCCN2C(=O)Cc2ccsc2)cc1 n1(CC(C)C(=O)NC2CC(NC(c3ccccc3)=O)C2)cnc2ccccc12 CC1CN(C(=O)Cc2cncnc2)CCC1NC(C1C2(CC2)C12CC2)=O C1(C(N(CC(C)N(C(=O)C=CC(=O)NC2CC2)C)C)=O)CCCCS1(=O)=O C(=O)(CCCN(C(=O)C(F)CC1CCOC1)C)N(CC)Cc1occc1C C1(O)(CCNC(CCC(=O)NCCC)=O)CCCN(C(=O)C(CC)NC(C)=O)C1 Cc1ccccc1C(=O)NCC(O)CNC(c1ocnc1C)=O C1(C(C)C(C2CCC(C)O2)=O)CN(C(=O)C(C)O)CCO1.NC N1(C(CCNC(C#CC(C)(C)C)=O)=O)CCC2CCC(C1)N2C CC1CCN(C(=O)C=Cc2ccnn2C)CCN1C(C1CCCNS1(=O)=O)=O N1(C(c2cc(Cl)ccn2)C(=O)NCCCC)CC(CF)C2(CCCC2)C1 N1(C(C2(C(F)F)CC(=C)C2)=O)CCOC2(CCCN(C(C3(C)CCSCC3)=O)C2)C1 c1(C(=O)NCCN(C(=O)Cc2cccc(Br)c2)CC)c(C)cc[nH]c1=N Cc1cc(-c2cccc(C3(NC(=O)CN4CCOCC4)CC3)c2)cnn1 N1(C(CC=C)=O)CCC2C(NC(c3ccc(F)c(F)c3C)=O)C2CC1 N1(C(CCNC(C)=O)=O)CCC2(CCCC2C(=O)Nc2cnc(Cl)nc2)C1 C1(NC(CCc2onc(CC)n2)=O)CCCCC1CNC(c1c(Cl)n[nH]c1C)=O c1(CC)ccc(C(=O)NC(CCN(C)C(C2(F)CCOC2)=O)C(C)(C)C)c(C)n1 CCC(O)C(F)(F)C(=O)NC1CC2(C1)CC(C(=O)NCCCc1ccccc1)C2 N1(C(C2C(C)=CCC=C2)=O)CC2CN(C(c3ccc(C(F)(F)F)c(O)n3)=O)CC12 c1(C(=O)C(C=CO)=O)ccc(C)n1C.N1(C(C2C(CCC)C2)=O)CC(C(C)N)C1 N1(C(c2c(F)ccc(C)c2)=O)CCC2C(NC(C3C4CC5C(C4)C35)=O)C(C)(C)C12 C1(NC(c2cc(CC)oc2C)=O)CN(C(=O)C(c2ccc(F)cc2)O)CCC1F C1(CC#C)(C(=O)NC(CNC(=O)CCn2cncn2)C2CCC2)CCCCO1 C(CC#CC)(C(=O)Nc1cnn(CC=C)c1)NC(c1n(CC#C)cnn1)=O C1(CC(C)(C)C)CN(C(C2(Cl)CC2(F)F)=O)CCN1C(c1cc(Cl)no1)=O N1(CC)CC(C(N2CC(OC)C(NC(c3ccoc3Br)=O)C2)=O)CC1=O C1(CC(C)NC(c2c(NCC)scn2)=O)CCN(C(=O)Cc2ccns2)CC1 c1(C(=O)[N+](CCOCCNC(CC2(CSC)CC2)=O)([O-])CC)ncccc1N=[N+]=[N-] c1(OC)cc(CN2CC(CNC(c3ccc4ccoc4c3)=O)C2)cc(O)c1O C#CCC(CC(F)F)C(=O)NC(CCC(C)C)C(=O)NCCCNC(=O)C(C)(C)C C1(C(=O)NC)CC2(CCC2)CN1C(c1nc(CNC(=O)OC(C)(C)C)ns1)=O C#Cc1ccc(OC)c(NC(C2CCN(C(=O)CSC)CC2NC(=O)C2CC2)=O)c1 n1(CC)nncc1C(=O)NC1CCC(CNC(=O)C(c2ccncc2)c2ccccc2)C1 C(=O)(C1=COCCO1)NC(C1CN(C(=O)C(O)CCN(C)C)C1)C C12(CNC(c3cc(CCCO)on3)=O)CC1CN(C(C1C=CC=CC=C1)=O)C2 c1(CN(C(C2(F)C(C(=O)O)C2)=O)Cc2cccs2)cnn(C2CCCC2)c1 Cc1ncc([N+](=O)[O-])cc1C(=O)NCC1CC2CC1CN2C(=O)CCC(C)C c1(C(=O)NC(C2N(C(COCCCC#C)=O)CCC2)C)cc(C)c(C)o1 Cc1ccc(C)c(C(N2CCC(O)(C(C)CNC(=O)CN(S(C)(=O)=O)C)C2)=O)c1 N1(C(CCSCCC)=O)CCCC1C1CCCN1C(=O)C=C(C)C1CC1 C1(C(=O)NCC(COC)(F)F)C(C)CCN1C(c1ccc(C#N)[nH]1)=O C1(O)(CC(=O)NCC(CC)NC(c2cc(C)ccc2Br)=O)CCCN(C)C1 c1(C(N2C(CN(C(=O)CCNC(=O)C3CC3)C)CCC2)=O)cccnc1O C(=O)(CCCNC(c1cn(CCNC(c2[nH]nnc2C)=O)nn1)=O)NC C1(CCN(C(=O)CC2CCCCC2)C)CCCCN1C(=O)C(c1ccnn1C)O C1(O)(CCNC(c2csc(Cl)c2)=O)CCN(C(C2CC(C(F)F)C2)=O)C1 c1(C(=O)NCCCC(CCC)NC(=O)CC2CC=CCC2)n[nH]c2c1CCSC2 c1(OC)ccc(CC(C)C(=O)N(CC(C)(C)CNC(C2C=CCC2)=O)C)cc1F c1(C(=O)NC(C)CN(C(=O)C=CCCc2ccccc2)C)ccn(C)c(=O)c1O CCCCC(=O)C(=O)N1CCC2C(C(=O)NCC3CC4OC3C3CC43)C2C1 c1(C(N(C2CC(C(N)=O)C2)C)=O)coc2c1CN(C(=O)C(C)(C)F)C2 C#CCC(CC#C)C(=O)NC12CC1CN(C(=O)C(COC(C)(C)C)NC(C)=O)C2 N1(C(c2c(C)[nH]cc2)=O)CC2(CNC(C34CCC(CC3)C(C)O4)=O)CCC1CC2 C1(NC(C2(COC)CCC2)=O)(NC(=O)C(=O)NC2CC2)CC(O)C1 C1(NC(CC(C(C)C)NC(CCCOCC)=O)=O)CCn2nccc2C1 c1(C(N(CCN(C(C2C(CC)C2)=O)C)C(C)C)=O)cccc(F)c1OC C1(CNC(c2nc(C)sc2C)=O)CN(C(C2CC2C(F)F)=O)C2(CCOCC2)C1 Cc1ccc2cc(C(=O)NC3CCCCN(C(=O)CC(C)F)C3)ccc2c1 N1(C(CCNC(CCCC(CC)C)=O)=O)CCc2nncn2CC1 CCCC(C(=O)OC)C(=O)NCC1CN(C(c2scnc2C)=O)CC1O N1(C(c2c(OC)ccc(O)c2)=O)CCN(C(=O)C(C)=C(C)CC)CC(C)(F)C1 c1(OCC)cc(C(=O)N(C(C)CNC(C2COC(C3CC3)C2)=O)C)ccn1 C1(O)(c2c(C(N3CC(N(C(C=CC(C)(C)SC)=O)C)C3)=O)c[nH]n2)CCOCC1 N1(C(C(=O)NCCOC)=O)CCCC2CN(C(C3(C)CC4(CCC4)C3)=O)CC12 CC1CN(C(C2CCSCC2)=O)CCC1CNC(c1cc(CO)[nH]n1)=O C(=O)(CCC(C)CN(C)C)NCC1(C)N(C(C(C(=O)OC)C)=O)CCC1 C(CC(=O)N1CC2(CNC(=O)CC3CCC3C)CCC1CC2)(C(F)(F)F)OC N1(CC(COCC(=O)N(C)C)O)CC=CC(NC(=O)CCN2CCCS2(=O)=O)C1 CN1CCc2ccc(C(=O)NCCC3CN(C(C4CC4(C)C)=O)CCO3)cc21 N1(C(C(CC)CC)=O)C2CCC1CC(NC(=O)C(O)Cn1cncn1)C2 CC(N=c1ccnc(N2CCC(NC3CC3)C2)[nH]1)N1CCC(CN)C1 C(=O)(C1CCCc2nc[nH]c21)NC1CN(C(C(CC)(F)F)=O)CC1C C1(C(=O)NC2C(CNC(CCCC#C)=O)CC2)CC2(C1)CC(F)(F)C2 c1(C(C)(C)C)nc(CNC(=O)C(=O)NC2(C3CCCO3)CCC2)c(Br)s1 N1(C(c2c(-c3c(OC)cccc3)onc2)=O)CC2(CCCCC2)CCC1C C1(C(=O)OC)CCC2C1C2(F)F.c12ccc(cc1)C1(CC1)NC(=O)NC21COC1 C12(C(N(CCCCC(=O)NC(CCOC)C)C)=O)CCC(C1)OC2C C1(CNC(C(C2CCCC2)OCC)=O)(NC(C2CCCO2)=O)CCCCC1 O=C(C1=CC2CCCCC12)NCC#CCNC(=O)C1Cc2ccccc21 Cc1ccnc(O)c1C(N1CC2CC(C1)N2C(c1ccsn1)=O)=O C1(NC(c2nc(OC)oc2)=O)CCCCN(CC2CC23CCC3)C1 c1(C(=O)NCCC2CCN(C(C(C)(C)CCF)=O)C2)nc2ncccn2n1 Cc1cc(C(F)F)oc1C(=O)NCC(C)CNC(c1ncc(C(F)(F)F)n1C)=O C1(C(N(CC(C)(C)C(=O)NC2CC3CCCC3C2)C)=O)Cc2ccccc2C1 c1(N(C(COC)C)C)nnc(-c2ccccc2F)n1CC(=O)Nc1ccccn1 c1(C(=O)NCCC(C)(C)NC(C(C)OC)=O)c[nH]c2cc(F)c(F)cc2c1=O Cc1nc(C)n(O)c1C(=O)NCCCC1CCCN1C(=O)Cc1cccc(F)c1 CON(C)S(=O)(=O)c1ccc(C(N2CCN(C(c3cc(F)c[nH]3)=O)CC2)=O)cc1 c1(NC(C(C)N(C(=O)CCCn2ccnc2)C2CC2)=O)ccc2cnccc2c1 N1(C(C(C)n2cccn2)=O)CCCC(C(=O)N(CC)Cc2ccc(F)cc2)CC1 c1(CN2CCN(Cc3nc(C(=O)OCC)on3)CC2)nccc(I)c1C N1(C(C(C)(N(C(Cc2ccc(C)nc2)=O)C)C2CC2)=O)CCCC(C)C1CO N1(CC(=O)NCC=C)CCSCC1NC(=O)CN1CCSCC1 C1(C(N(CC(CN(C(=O)CCC2CCC(C(N)=O)O2)C)O)C)=O)CCNC(=O)C1 C(CCC(c1nnnn1C1CCC1)NCc1nc(CC2CC2)cs1)OC C1(NC(CCOC)=O)CCN(C(=O)CC2(CO)CCOCC2)CC1CO N1(C(CC(=C)C)=O)CC2(CC(NC(c3cn(CC)nc3C)=O)CO2)C1 C1(C(=O)NCCN(CC)CC)CCN2CCCCC2C1.c1(-c2c[nH]nn2)cnn(C)c1 C1(CNC(c2csc(C(F)F)n2)=O)CCCN1c1nc(C2CC2)ns1 C1(CC)CC(CC(=O)NC2CCN(c3nc(SC)ns3)C2)CCO1 N1(C(=O)C(O)c2ccco2)CC2CCC(C1)N2C(C1CN2CCCC1C2)=O C#Cc1cccc(C(=O)NCC23CC(NC(c4ccc(CCC)[nH]4)=O)(C2)C3)c1Cl C(=O)(C1=CCN(C(c2ccc(C)c(C)c2)=O)CC1)NC(C1CCOC1)C#C Cc1cc(C(=O)NC2CC(C(=O)NC(CO)CCO)C2(C)C)n(C)n1 C(CS(=O)c1ccccc1)SCCC(=O)Nc1c(CC)cccc1 Cc1nc(C(C)(C)C)ncc1C(=O)NC1CC1NC(C1CC(=O)N(C)C1)=O C1(C(N2CCC(CO)C2)C(=O)NCC=C)Cc2ccccc2OC1CC.N(C)(C)CC c1(CC)ccccc1S(=O)(=O)N1CCCC(CCN)C1 N1(CC(=O)N(CC=CC(=O)NC2CCC(OC)C2)C)CCC(C)CC1 C1(=O)C(C(C)C)NC(=O)C2CCN1C2.C1(NC(CC)=O)CCCC1 C12(C(=O)NCC3C=CC(NC(C4(CC=C)CCCCC4)=O)C3)CCC(F)(CC1)CC2 c1(OC)nc(C2=NOC3(CCN(Cc4cncc5nc[nH]c45)C3)C2)nc(OC)n1 CC1(C)CC2(CC(C(N3CCN(C(C45CC6CC4C5C6O)=O)CC(O)C3)=O)C2)C1 C12(C(=O)NC(C)CNC(=O)C=CC=CC=CCO)CCOC1CCOC2.C(C(F)(F)F)N CC(C(=O)N(CC(=O)NC(C(N)=O)c1ccco1)C1CCC1)S(N)(=O)=O c1(-n2ncc(NC(C=CC3C(C)C3(Cl)Cl)=O)c2)ccc(Cl)c(F)c1 C1(CNC(c2nc(C)oc2)=O)CC12CCN(C(=O)C(F)CCN(C)C)CC2 C(CCC(C)(C)C(=O)N1CCCCC1)NC(=NCC1C(C(=C)C)OCC1)NCC c1(OC)ccc(Cl)cc1CC(=O)NCC1CN(C(=O)C(C)CN(C)C)CCO1 Cc1c(O)ccc(C(N2CCC(CNC(=O)C3=NOCC3)C2(C)C)=O)c1C N1(C2(CNC(=O)CSc3cncs3)COC2)c2ccccc2Sc2ccccc21 c1(C(=O)NC2CC3CC(C2)CS(=O)(=O)C3)cc2c(c([N+](=O)[O-])c1)OCO2 c1(-c2cn(CC(=O)NCC(c3ccc(Cl)cc3)C)nn2)cnccc1OCCO c1(C(=O)NCC2N(C(C(C)=CC)=O)CCC2)ccc(Br)cc1C#N CC(C)(C)CC(C(=O)N(CCN1CCOCC1)C1CC1)N1CCC1c1cccs1 c1(CC)c(C(=O)N(C)CC2CCCC(NC(c3cc(C)co3)=O)C2)nnn1CC N1(CC)N=C(C(=O)N2CC(N(C(=O)C=CCCC(C)C)C)C(F)C2)CCC1=O CN1CCN(CC(C)(C)C(=O)N2CC(O)(CN(C(=O)C(=O)N(C)C)C)C2)CC1 C1(NC(C(CC2CC2)NC(c2c(C)cccn2)=O)=O)CCC(O)C(O)C1 c1(C(N2CCN(C(COCC=C)=O)C(C3CCCC3)C2)=O)cc(Cl)c(F)cc1N Cc1cc(CCC(=O)NC2(C)CC(C(N3CC(O)(CO)C3)=O)C2)nn1C CC1(C)CC(C(=O)NCCCCCC2CC2)CN(C(=O)C=CC2CCCC2)C1 Cn1cc(C(=O)NC2CN(C(c3cnc(N(C)C)o3)=O)CC2F)c2ccccc12 C(=O)(CC(C(F)(F)F)NC(=O)CC1(C#N)CC1)NCC(CN(C)C)O C1(CNC(CC(=O)N(C)C)=O)Cc2ccccc2CN1C(c1c[nH]c(C#N)c1)=O CCC(CCCC(=O)N1CCS(=O)C(C)C1)NC(C1(C)CCCCCC1)=O Cc1cccc(OCC(=O)NCC2(NC(=O)CC(C)C3CC3)CCOCC2)c1 N1(C(CCC#CC)=O)CC(NC(c2cc(OC)cc(Br)c2)=O)CC(C)C1 N1(C(C2CCCCN(C(C(C3CCC(=O)N3)C)=O)C2)=O)CCC2(C=CCO2)CC1 c1(C(N2C(C)CC(NC(C3(OC(C)C)CCC3)=O)C2)=O)cncc(Br)c1C N1(C(C(CCCC)C)=O)CCCC2(CCN(C(=O)C(c3c(C)noc3C)C)C2)C1 N1(C(C(C)NC(CC)=O)=O)CCCC(C2CCCN(C(c3cccs3)=O)C2)C1 c1(SC)ccc(Cl)c(C(N2CC3CC(NC(C4CCCOC4)=O)C2C3)=O)c1 C1(C(=O)NC(c2ccc(C)cc2)C)CC2CC1CC2NC(C1CC(N(C)C)C1)=O N#Cc1cc(F)ccc1C(=O)NCC1(F)CC(CNC(C2(C3CC3)CCC2)=O)C1 Cc1n[nH]c2cnc(C(=O)NC3CN(C(=O)CCSC(F)(F)F)C4CC34)cc12 C1(N(C(=O)CCn2cnnn2)CC)CCN(C(=O)CN2CCOCC2)C1 C(C(=O)Nc1cn(C)nc1OC)(C(C)C)NC(C(C=C)C)=O C(=O)(CCCCC(=O)NCC1CCN(C(c2cc(C)ccc2Cl)=O)C1)NC c1(C(=O)NC2(CNC(C3C4CCC34)=O)CCC2)ncsc1Br C1(CC)CN(C(=O)CCc2nccn2C)CCC1NC(=O)C(CC1CC1)OC C1(NC(c2ccc(C)c(C)c2)=O)CCC12CCN(C(C1CCCCN1C)=O)CC2 C1(NC(C(=C)CO)=O)C2CN(C(=O)COC3CCC(C)CC3)CC12 N1(C(C2OCCC(C)C2)=O)CC2CCCC(C1)N2C(=O)CCCc1ccccc1 CCC(F)(F)C(=O)NC1CCCCC1CNC(=O)CN1CCCC1=O C(=O)(C(C)(C)CS(N)(=O)=O)N(CCCCN(C)C(c1cc(F)cc(Cl)c1N)=O)C c1(C(=O)NC2C(NC(C(C)OCC#C)=O)CCOC2)ccc2c(=O)ccoc2c1 C1(C)(CC)CCN(S(=O)(=O)Cc2ncoc2CN)C1 O=C1OC(C(=O)NC2CCN(C(=O)CC3CC(F)C3)CC2)Cc2ccc(F)cc21 c1(CC)cc(C(N2CCC(CCN(C)C(c3ncc(C)o3)=O)CC2)=O)c(C)nn1 C(CCC(C(=O)NCCc1cccc(O)c1)NC(=O)Cn1nc(C)oc1=O)OC C(CC(C(=O)NCCc1cnn(C)c1)NC(c1ncsc1C)=O)=CC c1(C(=O)NC(C2OCCN(C(C=CCCC)=O)C2)C)ccc(Cl)c(C(=O)OC)c1 N1(C(CNC(=O)NC)=O)CCC(C2CCCN(C(C3CC4(C3)CC4F)=O)C2)C1 N#Cc1cccnc1NC(C1CCN(Cc2cc(-c3cnco3)ccc2F)C1)=O C(=O)(CC1OC(=O)c2ccccc21)NS(c1c(C)cccc1C)(=O)=O C(=O)(C1=NOC2COCC12)NC1(C)CCN(C(c2cccc(CC(=O)OC)c2)=O)C1 c1(C(=O)NC2C(C)CN(C(c3cn(CC(F)(F)F)cn3)=O)C2)cc2[nH]ccc2s1 N1(CC(=O)NC(C(C)NC(=O)C(O)Cc2cnn(C)c2)CO)C(=O)CNC1=O c1(C(C)NC(=O)C(=O)NCCc2ccnc(C3CC3)n2)ccc(O)c(F)c1 c1(C(C)(C)F)cc(C(=O)NCC2C=CCN2C(c2cncc(F)c2)=O)ccc1F O=S(=O)(c1ccc(NCCCCO)c2cnccc12)NC1CCCC12CC2 C(=O)(C(C)C(C)S(C)(=O)=O)N1CCOCC(NC(C2C(C)CC(C)O2)=O)C1 CC(F)(F)C(C)(C)C(=O)NC1(C2CN(C(=O)CSC3CCOC3=O)C2)CC1 C(CCN=C(NCc1cn2cccc(C(N)=O)c2n1)N1CCC(O)C1)OC C(=O)(C1=NOC2(CCC2)C1)NC(C(C)(C)C)CNC(=O)COCc1cccnc1 C(CC1=CCN(C(=O)CN(C2CCCC2)C)CC1)NC(C(C)OCC)=O c1(CC)sc(C(=O)NCCN(C(=O)CC2OCCCO2)CC)cc1Br C(=O)(CCCCN=C(NCCC(F)(F)CO)NCC(C)(C)C)N(C)C CC12CCC(CN1Cc1ccc(-c3ccccc3C#N)o1)C2 CCC(C)CC(=O)C(=O)NCCCN(C(=O)Cc1cnsc1)CC C(CCCN=[N+]=[N-])NC(COC1CC(N(C(CC(C)C2CC2)=O)C)C1)=O c1(-c2n(C)ccc2)ccc(C(N2CC3CC2C3CNC(c2ccc[nH]2)=O)=O)cc1 CCC(C(=O)NCC1CC1NC(=O)C(N1CCOCC1)C1CC1)OC c1(C(N2CC(O)(CCNC(=O)C(F)C3CC3)C2)=O)cc(O)nc(O)n1 N1(C(C(Cn2cncn2)NC(c2cncs2)=O)=O)CC2CC2(CO)C1 C1(C)(CNC(C2CC(C)OCC2)=O)CCN(C(=O)CCN(C)CCO)CC1 N1(C(c2n(C)ccn2)=O)CCCCC(CCC(=O)NCC(O)CC(=O)OC)C1 N1(C(c2c(CC)cccc2)=O)CCCC(NC(=O)C=CC(C)CC)CCC1 C(=O)(CC(C)CN1CC(C2CCN(S(=O)(=O)C(F)F)C2)C1)OC c1(C(=O)NC(C(=O)NCCCCOC)(C)C)ccnnc1C C(=O)(C(C)(C)C1=CCSCC1)NC1C2CC(NC(CC(C)OC)=O)C(C2)C1 c1(CCC(=O)NC2CCN(C(c3coc(Br)c3)=O)C2)ccsc1Br C(=O)(C(CNC(=O)CNC=O)CC1CCCC1)N(CCN(CC)CC)C Cc1cccc2sc(C(=O)N(CC(C)NC(c3cc(CO)on3)=O)C)c(Cl)c12 C1(F)(CNC(CCCOCC)=O)COCCN(C(=O)CC(O)CC)C1 C(=O)(CC1=CCCC1)N1CC2C(NC(C(F)(F)C3(OC)CCC3)=O)C2C1 N1(C(CCC2N(C(C3CCC(=O)C3)=O)CCCC2)=O)CCC2(CCO2)C1 N1(C(Cc2n(C)ncn2)=O)CCCC(C(O)CO)C1 N1(C(c2onc(CC)n2)=O)CC2CC(NC(C3CCCS3)=O)C2C1 Cc1c[nH]c(C(=O)NC(C)CCC(=O)NC(C2CCCC2O)C)c1C CCC(C)C(O)C(=O)N1CC(O)(CN(C)C(c2nc(Cl)c(Cl)s2)=O)C1 N1(C=CC(=O)C(F)(F)F)CC1=O.c1(NC(CSC(C)C)=O)cnc(O)c(Br)c1O Cc1nn(C)c(C)c1OCC(=O)N(C)CC1CCN(C(=O)CCn2ccnn2)C1 C(N=c1[nH]c(N2CC3CC2CN3CCC)nc2c1SCC2)C1CCN(C)C1 C(=O)(C(C)(C)C(=O)NCC(CNC(=O)C(CC1CC1)CC1CC1)CO)NC CS(=O)(=O)C1(C(N2CCCC(F)(CNC(C3CC3Cl)=O)C2)=O)CCC1 c1(C(=O)NCCCNC(COC)C(C)C)cc(C)c(OC)cc1C C(=O)(CC(C)(C)CNC(c1cncn(C)c1=O)=O)NCC(=C)Cl C(=O)(CCCCCCC(=O)N1CCC(NC(C2CC3CCC2C3)=O)C(F)C1)OC CCCCC(O)C(C)C(=O)NCC1N(C(c2cc(OC)cnn2)=O)CCC1(C)C C1(C(N2CCC(NC(CC3CC(OCC)C3)=O)(CF)C2)=O)CCn2ncnc2C1 c1(NC(CC2(C)N(C(C(COC)COC)=O)CC2)=O)cnc(O)cc1C C1(C(=O)OC)CC2(CC(NC(=O)N(CC(C)OC)C)CCO2)C1 N1(C(c2ccc(C(C)(C)C)s2)=O)CC2CCC2(NCC2Cc3nccn3C2)C1 c1(C(N2C(C(=O)NCc3cnc[nH]3)CC(O)C2)=O)ccc2nc(Br)sc2c1 N1(C(CNC(=O)OC)=O)CCN(C)C(CNC(C2(F)CCC(C)CC2)=O)C1 N1(C(C)=O)CCCC2(NC(c3cc4cc(Br)ccc4[nH]3)=O)CCCC12 c1(NC(c2ccc(OC3CCCC3)cc2)COC)ncnc2[nH]c(C)nc12 C1CCC2C(CC1)C2(F)F.c12ccc(cc1)C(=O)NCc1cn-2nn1.CC1CC1 c1(CCC)cc(N(c2ccnc(C)n2)C(=O)Cc2ccc(Br)cc2I)nc(Cl)c1 Nc1nonc1C(=O)NC(c1cccnc1)C(N1CCC(CNC=O)C1)=O c1(C(N2CCC(C)(CC)CC2)=O)cc2cnccc2nc1C C(=O)(CC(C)(C)CNC(C1(F)CCCCCC1)=O)NC1CCCC(C(C)C)C1 C(C(C)(C)CCNC(c1cnc(SC)o1)=O)NC(Cc1c(C(=O)OC)csc1)=O C1(NC(c2nc(C)sc2C)=O)CN(C(c2ccnc(C)c2C)=O)CCC1CO CN1C(=O)NCC1CO.C(CCCCCF)N1C2(c3cn(nn3)CC1=O)CCC2 C(C1CN(C(C2CCCC(=O)N2)=O)CC1C(=O)N(C(C)C(=O)NC)CC)=CC C(CCCC(=O)NCC1CCC1NC(c1cncn1C1CC1)=O)SC C#CCC(CC#C)C(=O)N1CC(CCCCNC(C2CC2(Cl)Cl)=O)C1 c1(C(=O)NCC(CC)NC(=O)COc2ccsc2)ccc2ccoc2c1 C(=O)(C(O)CSC)NCCC(C)N(C(=O)CSC)C.N1(C(N)=O)CCCC1 N1(C(C2CCN(C)C2=O)=O)CC(CNC(C2(C)CC2(F)Cl)=O)OC(C)(C)C1 C(c1ccc(O)cc1)=CC(N1C(C(C)(C)NC(c2ncc[nH]2)=O)CCC1)=O c1(CC)cccc(C(=O)NCCCC(CO)NC(C2CCC(N(C)C)C2)=O)n1 c1(C(N2CCOC(CNC(N)=O)C2)C(=O)NCC(=C)C)cccc(Cl)n1 Cc1c(C(=O)NC2CN(C(=O)CC3(CO)CC3)C3(CCC3)C2)c[nH]c2nccc1-2 C1(NC(CCN(C(C)=O)C)=O)CCCC(NC(=O)C(C)C(=O)OC(C)(C)C)C1 N1(C(C2CC(O)(C(F)(F)F)C2)=O)CCC2(CCCN2C2CC2)C1 C(CC(C)(C)C(=O)N1CC(NC(C2CC=CCC2)=O)C(C(F)F)C1)SC c1(CN2CCCC2)cc(Cl)c(Cl)cc1Cl.C12CCCCC1CNC2=O C=CC1(C(=O)NCC(C)(C)CN=[N+]=[N-])CCN(C(=O)C(CC)n2cncn2)C1 Cc1[nH]nc2c(C(=O)NC(C)CCCCNC(=O)CC(C)C(F)(F)F)cccc12 Cc1cc(C(=O)N(C2CC2)CC2CC2)c(C(F)(F)F)o1.C12CCCCN1C2 CN(C)NC(=O)CCC(=O)NCC#CC(=O)NCc1cc(O)ccc1F Cc1noc(C(N2CCC(N(C(=O)C(F)CNC(=O)OC(C)(C)C)C)C2)=O)c1C C(C1OCc2ccccc21)N1CCN(CC(=O)NCC2C(N=[N+]=[N-])OCCC2)CC1 N1(C(CSCC)=O)CC(NC(=O)CCCc2sccc2C)CC(O)C1 C=CCC(C(=O)N1CCC(C(=O)Nc2cnccc2N(C)C)(COC)C1)N(C)C N1(C(C2CN(C)C(=O)CC2)=O)CC2CCC(NC(=O)C=CC3CCOCC3)C2C1 C1(C(N(CCN(C(=O)CCCC(F)F)C(C)C)C)=O)CCc2ncccc2C1 C1(C(=O)NCC2CCCN(C(C3CC4(CSC4)C3)=O)C2)CNc2ccnn2C1 C1(CC(=O)N(CC(C)NC(=O)C(C)(C)C#N)C)CCC(F)(F)CC1 Cc1cc[nH]c1C(=O)N(CC(C)O)CCNC(=O)C(c1cscn1)OC Cn1cnc2[nH]c(C(=O)NCC3CCC(NC(c4cccc(F)c4F)=O)C3)cc12 c1(C(N(CC(C)N(C)C(c2ccnc(S)c2)=O)C)=O)csc([N+](=O)[O-])c1 CCC(CNC(=O)C=C(C)CNC(=O)C=C1CC1)(CC)OCCOCC CCCCC(C)CCC(=O)NCCC(C)(C)C(=O)N(C(C)C(=O)OC)C c1(C(=O)NCC2CC(CNC(c3ccoc3)=O)OC2)c[nH]c2cc(F)ccc12 C1(NC(C2CC(=C)C2)=O)(CO)CCN(C(c2cnn(CCOCC)c2)=O)C1 c1(CC(=O)NC2(C)CCCN(C(C3CC(SC)C3)=O)C2)ccc2c(c1)CCC2 C(CN=c1cc(NC(c2nc(C(F)(F)F)cs2)c2ccccn2)nc(C)[nH]1)OC N1(C(C(C)SC)=O)CCC1(C)CC(=O)N(CC(C)COC)C N1(c2c(C)ccc(C)n2)CCC(C(N2CCCCC2)=O)CC(C)(C)C1 CC(CC(F)(F)F)C(=O)NC1CCCCN(C(C2(C)CC2C(F)(F)F)=O)C1 C1(C(N2CCCC(C)(CNC(c3sccc3Cl)=O)C2)=O)CC2(C1)CC21CCC1 C1(NC(=O)CCSCc2ccccn2)C2CN(C(C34CC3C4)=O)CC12 c1(OC)ccccc1N1CCC(NC(=O)CN(C)CC2(C)CC2(F)F)C1 N1(C(CC2C(CC)C2)=O)CCCCC1CC1CC1NC(C1(CO)CC(F)(F)C1)=O N1(C(C2(C#C)CCCC2)=O)CC(NC(c2ccccn2)=O)CC(O)C1 c1(C(=O)NC(CNC(CN(CC)CC)=O)CO)cnn(-c2ccccc2)c(=O)c1 N1(C(CC(COC)C)=O)CCN(C(=O)Cc2ccsc2C)CCC1C N1(C(Cc2cc(C)sc2)=O)CCC(C(=O)NC(c2c(C)noc2C)C)CC1C c1(CNC(=O)CNC(=O)NCC2CC2)c[nH]nc1Br c1(C(=O)NCCN(C(C2C3C4CCC(C4)C23)=O)CC)cc2cnccc2[nH]1 CC1CC(NC(C2(CC(F)F)CCC2)=O)CN(C(=O)OC(C)(C)C)C1 C12(C(N3CC(OCC)CC3(C)CNC(=O)CSC(C)C)=O)CCCC(C)(C1)OC2 C1(NC(CCC(C)NC(CCNC(=O)OCC)=O)=O)C2CCCCCC12 C1(C(N2CC(N(C(=O)C3=CCOC3)C)C(O)C2)=O)CC2CCC(C1)C2 C1(CNC(c2onc(CC)n2)=O)CC2CCC(C1)N2C(C1CCC=CO1)=O c1(N(C(=O)CCCCCBr)Cc2cn(CC)nc2)cccc2cc(O)ccc12 CC1(NC(=O)NC2CCC(C(N)=O)C2)CCCN(C(c2c[nH]nc2F)=O)C1 C(=O)(C(C)(F)C(C)(C)F)N1CCOCC(NC(C(c2ccccc2F)OC)=O)C1 CC1CCCc2ncc(C(=O)NC3CCCCN(C(c4ccncc4F)=O)C3)n21 c1(C(=O)NC2CN(C(=O)NC)C2)sc2ccccc2c1Br.N12CC(O)(C1)C2=O C(=O)(C(CCS(C)=O)N(C)C)N1CCC(CN(C(C=Cc2ncc(C)[nH]2)=O)C)C1 c1(OCC(=O)NC(C)CCCNC(=O)CCNC(=O)CO)nn(C)cc1[N+](=O)[O-] C1(CNC(c2c(C(C)C)occ2)=O)CN(C(=O)COC2CCCC2)CC(C)(C)C1 c1(C(N2CCCN(c3ncc(CC)s3)CC2)=O)c(F)cc(Cl)cc1Cl c1(C(=O)OC)ccc(NC(C2CC23CN(C(c2c[nH]nc2C)=O)C3)=O)cn1 CS(=O)(=O)c1ccc(C(=O)NCC(C2CC2)NC(=O)Cc2cncnc2)s1 c1(OC)ccc(Cl)cc1C(=O)NC(C)CNC(c1nnc(O)nc1O)=O C1(CC)CCC(C(=O)N(CC(C)C(=O)N(C(C)C(C)(C)C)C)CC)CC1 CCCCC(O)C(C)C(=O)N1CCC1C(=O)Nc1ccc(C2CC2)nc1 N1(C(C2CCN(C(c3cnn[nH]3)=O)C2)=O)CCCCCC1CCO N1(c2cc(SC)ncn2)CCCC(CNC(c2ccc(C)cc2)=O)CC1 C(=O)(CCC(=O)NCC1CCC(NCC=C(C)C)C1)OC C=CC(C)C(=O)N1CC=CC1C(=O)NC(C)Cc1nncn1C c1(C(N2CCN(C(C=CCOC)=O)C(C)C2C)=O)ccnc2cc(C)ccc12 N1(c2ncc(C)cn2)CCN(C(c2ccc(OC(C)C)cn2)=O)CCC1C Cc1cc(NC(=O)CC(C(F)F)NC(c2cc([N+](=O)[O-])n[nH]2)=O)cc(C)c1 CC(C)(C(=O)N(C1CCCS1)Cc1ccccc1)c1nccs1 C(=O)(CCCCC#N)NCC(C)CNC(C1CCCCCC1)=O N1(C(COCCOCC#C)=O)CCCC(CC(C)NC(C2(C)CCCCC2)=O)C1 c1(C(N(C)CC2(O)CN(C(c3c(CC)ccs3)=O)C2)=O)ccc2c(c1)OCC2 N1(C(c2cncc(C)n2)=O)CCCC(C)C1CCNC(=O)C(F)(F)CC1CC1 c1(CC)nn(C)c(Cl)c1C(=O)NCC(O)CCNC(c1coc(OC)n1)=O CC(C)C(O)C(=O)N1CCCCC1CNC(=O)CCC=CBr N1(C(c2cccc(SC)c2)=O)CC2CCN(C(=O)C(C(C)O)N(C)C)C2C1 C1(C)(CC)CC(NC(=O)C2CC2)CN1C(C1(c2cccnc2Cl)CC1)=O C#CCCCCCCC(=O)NCC(C)(C(C)C)NC(=O)CN(C)C(C)=O c1(C(=O)NCC2(O)CC(NC(C(CC)F)=O)C2)ccc2c(c1)C(=O)N(C)C2=O c1(CN2CCCC(CC(=O)Nc3cc(Br)c(F)cc3Cl)C2)ccc([N+](=O)[O-])cc1 c1(C(=O)OC)c(C)noc1S(=O)(=O)NC1CCN(C(C)=O)C2(CC2)C1 C12(C(N3CC(O)(CN(C)C(c4ccc(N)cc4O)=O)C3)=O)CCCCC1CCC2 C1(CC(=O)N(CCCN(C)C)CCNC(C(C)n2ccnc2)=O)CCCC1(F)F c1(C(N2C(C)CC(NC(c3ccsc3)=O)CC2)=O)cc2ccc(F)cc2o1 C1(C(=O)NC(C2CCC2)C)CCC(C2CC2)N1C(c1cccc(=O)o1)=O C1(C)(C(N(CCCNC(c2ccc(C)s2)=O)C)=O)CCc2ccccc2C1 O=C1OC2CN(C(=O)C(=O)NCC34CCC3CCN4)CC2O1 c1(C(C(=O)NCCOC)N(CC(C)C)Cc2ccccc2)ccc(F)c(I)c1.C N1(C(CCC(C)OCC)=O)CC(NC(C2CCC(C)(C)CC2)=O)C2CC2C1 Cc1cc(NC(=O)NCC(c2ccco2)O)c(Br)nc1C C(=O)(C1=CCS(=O)(=O)C1)NCC1OCCN(C(c2cc(C#N)sc2)=O)C1 CC(C(=O)N(CC(C)NC(=O)C(C)(C)c1cncs1)C)C1=CCCC1 c1(OC)ccc(C(N2CCN(CCN3CCCCC3)CC2)C)cc1C(C)C N1(C(C2(COC)CC(=O)C2)=O)CC2(C(=O)NCCCS(C)(=O)=O)CC1CO2 C1(C(C)NC(c2cc(CCCO)on2)=O)CCCN(C(=O)COC2(C)CCC2)C1 N1(C(CS(CC)=O)=O)CCC2(CCCCN(C(c3ccn4cncc4c3)=O)C2)C1 N1(C(CC2CCCN(C(=O)Cn3ccc(O)n3)C2)=O)CC2CCCC(C2)C1 C1(NC(=O)CC2(CO)CC2)CCN(C(=O)CNCc2ccccc2)C(C2CC2)C1 CC1CN(C(c2ccsn2)=O)CCN1C(C1CC2C=CC1C2)=O c1(NC(CCC=C(C)C)C)ncnc(NCCSC2CCC(C)(C)O2)c1C C1(NC(C2(CS(N)(=O)=O)COC2)=O)CCCCN(C(C2CC23CCOC3)=O)C1 C(=O)(CCCCCC#N)NCCC1(O)CN(C(c2c(CC)nc(C)o2)=O)C1 C(=O)(C(O)CC(C)(C)C)NCCC(C)NC(c1csnc1Br)=O N(C(=S)N1CCC(C(=O)OC)CC1)c1ccc(OC(CC)CC)cc1 c1(C(=O)NCC2(CNC(CC3(C(=O)OC)CCC3)=O)CC2)n[nH]cc1Cl c1(CC)cccc(C(N2CCC(C)(CC(=O)NCCC3CC(=O)N(C)C3)C2)=O)n1 C(=O)(C1=CCCC1C)N1C(CN(C(C)C(=O)NCc2ccc(Cl)cn2)C)C=CC1 C(=O)(CC(C)(C)CC(F)F)N1CCC(C)(NC(C(CCCCC)O)=O)C1 N1(C(c2ccc(CC)o2)=O)CC(CNC(c2ccnc(S)c2)=O)N2CCC1C2 N1(C(c2ncc(OC)nc2)=O)CC(O)CCC1C(=O)NCC1=NOCC1 Cc1c(C(=O)NCC(C)(C)CN(C)C(C2CCS(=O)(=O)N2)=O)ccn1C(C)C C1(C(N2C(C(=O)OC)CC(F)C2)=O)CC2(C1)CN(C(c1cccc(F)c1C)=O)C2 C(=O)(C(C)(C)CC1CC1)N1CCC(CNC(CCOCCN(C)C)=O)C1 CCC(CC)CC(F)C(=O)N1CCC(CNC(C23CCC(C(F)F)(CC2)C3)=O)C1 CCC(CC(=O)NOCCC(F)F)NC(=O)CNc1cnn(C)c1 c1(C(N(C(CNC(c2c(CCC)occ2)=O)C)CC)=O)ccc(OCCF)cn1 CC1C(C)N(C(c2coc(Br)n2)C(=O)NCC2CCC(F)(F)CC2)CCS1=O CCC(C)CCCC(=O)NCCCNC(=O)CC1CC2CCC(C1)N2C C1(NC(C(C)Cn2cccn2)=O)CCN(Cc2ccc(Cl)cn2)CC1F c1(C(N2CCCC(NC(C(C=C=C)C)=O)C2)=O)cc(S(=O)(=O)C(C)C)ccc1Cl c1(CC(=O)N(C(C)CNC(=O)CCC2CCCC(=O)N2)CC)c(C)n[nH]c1C N1(C(CCS(CC)=O)=O)CCC(C2CC(NC(C3CCCC(OC)C3)=O)C2)CC1 c1(Nc2cncc(NC(c3cc(OC)cc(C)c3)=O)c2)cc(F)c(F)c(F)c1 c1(C(N2CC(NC(c3n(CC)ccc3)=O)C3C2C3)=O)ccc2nc[nH]c2n1 c1(C(N2CC(OCCNC(=O)CCCC3CC3)C2)=O)cccc2c1CCOC2 c1(CCCC(=O)NC(C)C=C2CC(C(=O)OC(C)(C)C)C2)ccccc1Cl CC1(F)CN(C(=O)CCOC2COC2)CCN(C(C2(C3CC3)CCOCC2)=O)C1 N1(C(C(=O)NC(c2cnsc2)C)=O)CCCC2OCCC12 N1(C(C2=NOC(C)C2)=O)CC2CC(NC(c3cc(C(N)=O)ccn3)=O)CC(C2)C1 C(=O)(CCCC(CC)CC)N1CCC(C(=O)NC(CC=C)(C)C)(CC=C)C1 C1(C(N(CCCN(C(=O)CCCc2ccsc2)C)C)=O)CCc2nnnn2C1 N1(C(c2ccc(C)cn2)=O)CCC2CN(C(=O)Cn3cnnc3O)CC12 C(=O)(C1OCCn2ccnc21)NCC1N(C(c2cc(C)nc(C)n2)=O)CC1 c1(C(=O)NC(C(=O)N(C)Cc2cncnc2)c2ccco2)ccc2nccn2c1 C1(N2CCCC(C)CC2)CC2(CCN(C(c3ccc([N+](=O)[O-])[nH]3)=O)CC2)C1 c1(C(=O)OCC)cnc(NC(=O)CC(c2cccc(Cl)c2)O)nc1 C(=O)(CCCc1cnn[nH]1)NCCCCNC(CCC1(C)CC1)=O c1(C(=O)NCC2(O)CN(C(c3coc(C(N)=O)c3)=O)C2)ccc(C(N)=O)cc1F CC1(C)CC(CNC(C2CCC(=O)C2)=O)CN1C(=O)CC1CC(=O)NC(=O)C1 C#Cc1ccc(F)c(C(=O)N(C(C)CNC(c2c(C(F)(F)Cl)n[nH]c2C)=O)C)c1 Cc1c(CN2CC(c3cccc(C(F)(F)F)c3)C2)nnn1C1CCCCC1 Cc1sc(C(=O)NC2CCN(CCCNC(C3CCN(C)CC3)=O)C2)c(C)c1C c1(C(=O)NCC(C)(C)NC(CC2(C(=O)OC)CC2)=O)ccc(=N)[nH]c1Cl n1(CC)cc(Br)c(C(=O)NCCN(C(=O)CN2CCC(C)CC2)C2CC2)n1 C(=O)(C1c2ccccc2CN1Cc1c(C)scc1)Nc1cc2ccccc2n1C c1(OC)cc(C)c(C(=O)NCC#CCNC(c2nc(C)sc2Br)=O)cn1 C1(CC(N2C(CNC(c3c(C#N)scc3)=O)CC(F)C2)=O)CN2CCN1CC2 N1(C(CCc2nnc(C)o2)=O)CCN(C(=O)C(C)C(O)CC)CC(C)(F)C1 C1(C(=O)NCCCNC(C(c2cccc(Cl)c2)OC)=O)Cc2cc(F)ccc2O1 c1(NC(=O)NC2CC(C(=O)OC)(CC)C2)[nH]c2ccc(C(=O)C(C)C)cc2c1C N1(C(C(CCOC)NC(=O)C(C)Cn2ccnc2)=O)CCn2nc(C)cc2C1 N1(C(c2ccc(COC)[nH]2)=O)CC(NC(=O)C(CC)(CO)OC)C2(CC2)C1 N1(C(C2CN(C)C(=O)C2)=O)CCCC2(CCN(C(=O)C(C)(C)CC(F)F)C2)C1 Cc1ccc(CSCC(=O)NCC2(C)CCN(C(=O)CC3COC(=O)C3)C2)cc1 N1(C(CCC2CCCN(C(c3c(C)snc3)=O)C2)=O)CCCC2(CC1)CC2 Cc1cc(Cl)c(C(=O)NCC2C=CCN2C(C2CCCNC2=O)=O)c(Cl)c1 N1(C(Cc2n(C)cnc2)=O)CC2CC(NC(C3(C)CCC(F)(F)CC3)=O)C1C2 c1(C(=O)NCCCN(C(C2CCCO2)=O)CC)cc(C)cc(OC)c1C CCCCCC(=O)NC(c1ccccc1F)CNC(c1nc(C(C)C)oc1C)=O N1(C(C(CC)C(C)C)=O)CCCN(C(c2cccc(NC(C)=O)c2)=O)C(CO)C1 Cc1cc(C(N2CCN(C(c3sccc3Cl)=O)CC(C)C2)=O)c(F)cc1F N1(C(CCNC(=O)OCC)=O)CCC(C(C)NC(C2(C)CNC(=O)C2)=O)CC1 Cc1nn(C)c(Cl)c1CC(=O)NC1CN(C(C2CC2F)=O)CCC1CO N1(CC(C2CCOCC2)=O)CCCCC1CCN1CCSCC1 CCC(CC(=O)N(C1CC(NC(=O)CN2CCC(C)CC2)C1)C)c1ccccc1 c1(OCC(C)=CCC)cc(Br)cc(NC(C2CCOC(C3CCCN3)C2)=O)c1I N1(C(C(C(=O)OCC)OC)=O)CC2(CC(C(=O)N(CC(O)C(F)(F)F)C)CO2)C1 C(C(=O)NCc1ocnc1C(=O)N(C)Cc1n[nH]c(C)n1)(C(C)C)SC CC(C)(O)C(C)(C)C(=O)NC1CCCC(NC(c2n[nH]c3c2CSCC3)=O)CC1 C(=O)(C1=CCCC1(C)C)N1CCN(C(CCCC(=C)C)=O)C(COC)C1 Cc1cc([N+](=O)[O-])cc(C(=O)NC2CCCN(C(c3csnc3C)=O)C2)n1 C1(NC(=O)CCC(=O)N2CCC(O)CC2)CCC2CC2C1.C12CN(C1)C(=O)N2C n1(C(CC)CC)nccc1C(=O)NCC(C1CCOC1)NC(=O)CCSC CCC(CC(=O)NCC1(OC)CCN(C(=O)CC2(O)CC2)C1)C(C)(C)C C(=O)(CC(C)C(F)F)NCC1(C(N2C(COC)CCC2C)=O)CC(=C)C1 C=C(C)CCC(=O)NCC1CCCC(NC(=O)CC2(CSC)CC2)C1 C1(NC(C2C(CC)N(C(c3cnc(C)n3C)=O)CC2)=O)CCCC1C1CC1 N1(C(C2(CC)CCC2)=O)CC(NC(C2CCC(=O)O2)=O)C(CC2CC2)C1 C1(CN(C(C(C)OCCC=C)=O)CC)CCN(C(c2cccc(C)c2)=O)CC1 C1(NC(=O)NCC2(O)CCN(C(C)(C)C)C2)CCS(=O)(=O)C1(C)C.C1CCCS1 c1(NCc2c(CC)onc2C)cc(OC)c(C)c(OC)c1 CN1C(=O)NCC1C(=O)NC1CCC(CNC(=O)CN2CCNC(=O)C2)C1 c1(CCCNC(=O)Nc2c(CC)n(C(C)(C)C)nc2)ccc(F)c(F)c1F C(=O)(CCN(OC)C(=O)C(C)c1ccn(C)n1)NCC(=O)OC N1(C(C(C)NC(C)=O)=O)CC2(CCN2C(c2cnc(O)c(F)c2)=O)C1.N Cc1c(CC(N2CCC(c3cc(Br)no3)CC2)=O)ccc(Cl)c1Cl N1(C(C23CCC(OC)(CC2)C3)=O)CCC2(CCN(C(=O)C(F)C3CCC3)CC2)C1 C(C)(c1cn[nH]c1)=C(C(=O)NCC(CNC(=O)CN1CCCC1=O)OC)C c1(C(N2C3CCC2CC2(CC2)C3)C(=O)NCCSC)ccc2c(c1)C=CC(C)(C)O2 c1(C(=O)Nc2c(C(F)(F)F)cc(OCC)nc2)cc2ccccn2n1 c1(OC)ccccc1OCC(N1CC(N(C)C(C2CCCSC2)=O)C1)=O Cc1cncc(CC(=O)NCC(C)(C)CNC(c2ccc(C(N)=O)cc2)=O)c1 N1(C(C2CC(C#C)(O)C2)=O)CCCC2CN(c3nc(CC)nc(Cl)c3F)CCC12 C#Cc1ccc(CC(N2CCC(NC(c3nn(C)c(C)c3Cl)=O)C(C)C2)=O)cc1 N1(C(C(CC=C)C)=O)CC2CCC1C(NC(=O)CNC(c1cscn1)=O)C2 c1(OC)cc(C(=O)NC2CN(C(=O)CCCCCO)C2)cc(Br)c1Cl C(=O)(C1CCCn2ccnc21)N(CCC(c1cccs1)NC(=O)C=CCO)C N1(C(C(CC)NC(N)=O)=O)CCN(C(C2(CC(C)C)COC2)=O)CC1C c1(OC(C(=O)N(CCC(C)NC(=O)C=C(Cl)Cl)C)C)ccc(C(F)(F)F)cc1 C1(NC(c2ccc(CNC(C)=O)s2)=O)(CO)CCCN(C(=O)CC(O)C(C)C)C1 N1(C(c2c(CC)occ2)=O)CCC2CN(C(c3cc(F)c(Cl)cc3F)=O)CC2C1 CCC(C)C(O)CC(=O)N1CC(C(N2CC3CCCC2C3)=O)(SC)C1 N1(CCS(CC)(=O)=O)C(=O)CCN(Cc2ccc(CN3CCOC3=O)cc2)C1=O C(=O)(C(C)CC(=O)NCC(C)CNC(C1(C)C=CCCC1)=O)OC C1(C(N2CC(CC(C)NC(c3ccc(COC)o3)=O)C2)=O)CN(C)CC(C)O1 C(C)(C)(CC(F)C(=O)NCC(c1cnn(C)c1)C)NC(Cc1c(C)ccs1)=O c1(N2CCCC(NC(Cn3nnc(C)n3)=O)C2C)c(C#N)cccc1[N+](=O)[O-] CC(C)C(C)C(C)CN1CCN(C2CCS(=O)(=O)C2)CC1 Cc1c(Br)ccc(C(=O)N=c2ccn(-c3cccc(Cl)c3)[nH]2)c1F.C123CC(C1)(C2)N3 N1(C(C(C)=CC)=O)CCCCC(CNC(C23CC(CO)(C2)C3)=O)C1 c1(C(=O)NCc2ccc(C(C)=O)s2)cc2n(n1)CCCC2 N1(C(c2ccc(CSCCC)o2)=O)CCCCCC(NC(=O)CCS(C)=O)C1 C1(C(=O)NCC2CC(CNC(=O)C(F)F)C2)CCC2CC12 CC1C(C)N(C(c2nncn2C)C(=O)NC(C)(C)C)CCS1(=O)=O C1(C(=O)NC(CC)C(C)O)C2CN(C(c3sccc3OC)=O)CC12 C12(CNC(CCc3nc(C)sc3)=O)CCC1CCN2C(=O)CCn1cccn1 N12CCN(CC1C)C2=O.c1(CCOCC)cc(Cl)sc1Cl c1(CC)onc(C(=O)NCC(CC(=O)N2CCSC(C)C2)OC)c1C CC1(C)CCCC(CCN=C(NCC2CC(=O)NC2=O)NCc2ccccc2)O1 Cc1cccc(N2CCC(C(=O)NC(CO)C3COC3)CC2)c1 C(CCCC(=O)NC(CCC1CCCC1)C(=O)N(C(C)CCC(C)C)C)OC N(C(=NCc1ccccc1I)NCC(C)(O)CC)CC(Br)=C(C)C c1(OC)ccc(C(=O)C(=O)NCC(C)NC(c2cscc2F)=O)cc1 C1(O)(CCNC(c2c(CC(C)C)onc2)=O)CCN(C(c2csc(Cl)n2)=O)CC1 c1(CNC(C2N(C(C(n3ccc(C)n3)(C)C)=O)CC=C2)=O)cccc(C(N)=O)c1 C=CCC(C)(C)C(=O)NC1CC(CNC(c2c(C)ccnc2O)=O)C1 Cc1oc([N+](=O)[O-])cc1C(=O)NC12CC1CN(C(C1CCC(=O)N1)=O)C2 c1(C(N2CC(C(C)NC(c3cn(C4CC4)nn3)=O)C2)=O)ccc(C#N)nc1C c1(CC(=O)NC2CCN(C(C3CSC3)=O)CC2F)ccc2ncsc2c1 C1(NC(COCCC(C)C)=O)CC(CNC(c2cc(F)ccc2Cl)=O)C12CCC2 c1(C(N2CCC(NC(CCOCCOC)=O)(CO)C2)=O)nncc2c1CCCC2 N1(C(C2N(CC)CC2)=O)CCCCC2(C1)CN(C(c1cc(F)ccc1CC)=O)C2 C1(C)(NC(C(C)NC(=O)Cn2cnnn2)=O)CCCN(C(c2occc2Cl)=O)C1 N1(C(C(CCC)N(C)C)=O)CCC2C(CCN2C(c2cc[nH]n2)=O)C1 n1(CC)cc(CC(=O)NCC(C)CNC(C2(NC(=O)NC)CC2)=O)cn1 C1(CNC(C(C)(O)C2CC2)=O)CC2(CCN(C(C3CC(C#N)C3)=O)CC2)CO1 N1(C(C2(C)C(C)C2)=O)CCC(F)(F)C(CNC(=O)C(C2CC2)C2CC2)C1 C(=O)(C(O)CSC)NCC(COCCOC)N(CCNC(C)=O)CC.N C(=O)(C(F)CC(C)(C)NC(=O)CC1OCCCO1)N(C(C)CS(C)=O)C c1(C(N2CCC3(C(C(=O)NCc4nnn(CC)n4)C3)C2)=O)cccn2cncc12 N1(C(C(C(C)(C)O)NC(COCC=C)=O)=O)CC(C)N(C)C(C)C1 C1(C(N(C)Cc2cncn2C)=O)(C(C)C)CCCN1C(=O)C=CC(C)(C)C CCCC(C(=O)N1CCCC1CN(C(=O)C=Cc1ccc(CC)o1)C)NC(C)=O CC1CCC(=CC(=O)N(C(C)(C)CC(=O)NC2CC2c2cnn(C)c2)C)CC1 c1(NC(CC2CC(NC(c3cc(F)cnc3O)=O)C2)=O)ncc(Cl)cc1Cl C1(NC(c2c(C)n(C(C)C)cc2)=O)CCC(C)N(C(c2c[nH]cc(Cl)c2=O)=O)C1 C(=O)(CC(C)(C)C(=O)NCC1CN(C(c2cnc(S)n2C)=O)CCN1C)OCC CCCC(C)(O)C(=O)NC(C)CC1CCN(C(C2CCNC2=O)=O)CC1 C1(CNC(C2CN(C(C)=O)C2)=O)CN(C(=O)COC2CCCCO2)CCN1C C12(CNC(C3C(C)OC(C)C3)=O)CC(CO1)N(C(C1C3CCC(=O)C13)=O)C2 N1(C(C(C(=O)OC)OC)=O)CCOC(C(=O)N(C(C)C(C)C)CC)CC1 C1(C(N2CCC(CN(C(C34CCCC3C4)=O)CC)CC2)=O)CC(=O)NC(=O)N1 c1(NC(C2N(Cc3cccc(C)c3F)CCNC2)=O)cc(Cl)cc(Cl)c1Br C1(C(=O)OC(C)C(=O)OC2CCCC2)CC(F)(F)CN1C(=O)OC(C)(C)C CN1CCN(C(=O)C=CC2CC2)C(CNC(c2csc(-c3cnccn3)n2)=O)C1 C1(C(=O)NCc2nccc(OC)n2)COC2(C1)CN(C(=O)C(C)(C)C(=O)NC)C2 C1(NC(CCCCC)=O)CC(C2CCN(C(c3c(C)cc(F)cc3C)=O)C2)C1 c1(C(=O)NC(C2CCCC2)CNC(c2c(C)n(C)nc2)=O)ccc(F)cc1Cl c1(CNC(c2ccccn2)CCO)cc(Br)cc2[nH]ncc12 c1(C(=O)NC(C(=O)NCC#CCOC)Cn2ccnn2)c[nH]c(=O)cn1 N1(C(C2CCC(C)C2)=O)CC2CCCC(NC(c3ncc(Cl)n3C)=O)C2C1 C1(CCNC(C(CC)=CC)=O)CCCCN1C(=O)CC(F)F c1(CNC(C2C(C)(C)C2)=O)nnc2n1CCN(C(=O)Cc1cc[nH]c(=N)c1)C2 N1(C(c2c(OC)ccs2)=O)CCCC(C)(NC(c2ncc(C)cc2F)=O)C1 N1(C(C(Cc2cnc[nH]2)NC(C(C=C)OC)=O)=O)CCOC(C(C)C)C1 C1(C(=O)NCC=CCNC(C2N(C)C(=O)CCC2)=O)CN2CCCCC2CO1 c1(C(=O)OC)nc(=NCCN(C(c2cc3sccc3cn2)=O)C(C)C)c(C)c(C)[nH]1 N1(C(C2(CO)CCC2)=O)CC2CCC(C1)N(C(=O)Cc1ccsn1)C2 c1(N(C(=O)NCCNC(C2(CCN(C)C)CCOC2)=O)C)cccc([N+](=O)[O-])c1 c1(CC(=O)NC2CCCN(Cc3sccc3Cl)C2)c(Cl)cccc1Cl c1(CNC(c2occ(C)c2)=O)ccc2c(c1)CCN(C(C1(C)CC=CC1)=O)C2 N1(C(=O)CCc2ccccc2)CCN(C(C2CCCN2CC(F)F)=O)CC1CF N(C1CCOc2c(C)cccc21)C(c1n(CC=C)nnn1)CCC Cc1cc(C(=O)NCC(C)(C)CNC(c2cc(O)n(C)n2)=O)cnn1 c1(OC(C2CCC2)C)ccccc1CN1CC2C(C(=O)NC3CCCOC3)C2C1 c1(CNC2(c3nc(CC)on3)CC2)c(-c2ccc(F)cc2)nc2ccc(C)cn12 C=CCCCC(C(=O)NC1CC(NC(=O)CCC(=O)NC)C(O)C1)N(C)C C1(NC(C(CC=CC)CC)=O)CCN(C(=O)Cc2c[nH]nc2O)CC12CCC2 O=C1NCc2c(C(=O)NC3(CNC(C4CC(CF)C4)=O)CC3)cccc2N1 c1(NCC2CCN(CC)C2)[nH]c(=NCc2ccc(C)o2)nc2sccc12 CC1CCN(C(C2CCCCC2(C)C)=O)CCN1c1[nH]cnc2nc(Cl)cc1-2 c1(C(C(=O)OC)N(C2CCC(C)(C)C2)C)cc(Cl)cc(Cl)c1 CC1CCC(NC(c2cnoc2C2CC2)=O)CN1C(=O)CSCc1cccs1 CC1CC(NC(=O)CC(C)(O)c2ccccc2)CN1C(C1(c2ccncc2)CC1)=O C=CC1(CNC(=O)CC=CCNC(C2(Cl)CC2C(C)=O)=O)CCOCC1 C1(=CC(N2C(CNC(C3N(CC)C(=O)CC3)=O)CCC2)=O)CC2CCC(C1)N2C CC(C)CC(C(=O)NC1C=CC(CNC(C2CCCC2C)=O)C1)C(N)=O c12ncnc(c1F)NC1CC(C1)NC2=O.c1(CC)ccc(Cl)cc1C(C)C c1(C(=O)NCC(C)(CC)NC(C(C)OCC)=O)cc(-c2ccccc2)ccc1O CC(CN=c1[nH]c(=N)[nH]c(=NCc2cccc(Cl)c2Br)[nH]1)C(C)(F)F O=S(=O)(Cc1ccc(C(F)F)o1)c1ccc(CO)nc1 n1(CC(=O)NCCC(C)N(C(c2n(CC)ncc2)=O)C)ccc2ccc(Cl)cc12 O=S(=O)(C=Cc1ccc(F)cc1)NCC1(F)CCCC1 c1(OC)cc(Cl)cc(CNC2CN(c3cc(C#N)ncn3)CC2(F)F)c1O c1(OC(C)C(=O)NCC2C3CC2N(C(C2(N(C)C)CC2)=O)C3)ccccc1Cl O=C(C1=Cc2ccccc2C1)N1CC2CC1CCC2NC(C1CC(O)C1)=O c1(C(N2CC(C(=O)OC)C(C)(C)C2)C(=O)NCC(F)F)cc(Cl)c(F)c(Cl)c1 C1(CNC(COC)=O)CN(C(=O)CC2CN(C(C)=O)CCO2)CCN1C c1(C(=O)NC2CC(CCNC(C3OCCN(CC)C3)=O)C2)csc2c1CCCC2 c1(C(N2CCC(CNC(=O)Cn3ccnn3)C2)=O)ccc(C(O)CF)cc1 c1(N2CCCC(CNC(CCOCCN(C)C)=O)CC2)ccc([N+](=O)[O-])cn1 CC1(C2CCCN(C(C34CCCC3CCN4C(=O)OC(C)(C)C)=O)C2)CC1 S(=O)(=O)(c1ccc(N2CCOCC(CO)C2)cc1Br)NC(c1nc(C)sc1)C C1(NC(C2(OC)CCOC2)=O)CCN(C(c2cnc(CC3CC3)s2)=O)CC(C)(C)C1 N1(C(C2CC(OCC)C2)C(=O)NC(C)CC)CCOCC1 Cc1sc(Cl)nc1C(=O)NC(CNC(=O)CCCc1cc[nH]n1)CO CC(C(=O)NCC1(CNC(=O)CC2CCC(F)(F)C2)CC1)C(=O)N1CCOCC1 c1(OC)cc(CC(=O)N(CCCCN(C(=O)C#CC(C)C)C)C)cc(OC)c1O CCC(C)(C)C(C)CC(=O)N1CCCC1CNC(=O)C(C)=CC1CC1 c1(C(N2CCCCC(NC(C(CC)=CC)=O)C2)=O)cnc(O)c2cncn12 C1(C(N2CC(NC(COCCSC)=O)C3(C2)CC3)=O)COc2cc(Cl)ccc2O1 c1(C(N(CCNC(CC(C(F)(F)F)OC)=O)CC)=O)cc2c(F)c(F)ccc2[nH]1 C1(NC(CC(C)C)=O)(CF)CCN(C(c2ccc(C(N)=O)cn2)=O)C1 CC(CCO)C(=O)NC(CNC(=O)Cc1nncn1C)CO C1(C(=O)Nc2ccc(C(C)=O)cn2)CN(C(c2ccc(O)cc2F)=O)CCC1O N1(C(C=C(CCC)C)=O)CCC2(CC1)CC2NC(c1ccc(F)cc1CC)=O C(=O)(C1=CCCCC1C)N1CCCC(C(=O)NCCn2cccnc2=O)(CC)C1 C12(NC(C(CC)CC)=O)CCN(C(=O)Cn3nc(C)n(C)c3=O)CC1C2 c1(C(N2CCC(NC(C(=O)NCC)=O)C2)=O)cc(Br)cc2cccnc12 c1(NC)cc(Cl)ccc1C(=O)N(C)C.N12CC(C(C)C1)n1cc(nn1)COC2=O c1(NC(=O)CC2CCC(NC(=O)C(F)C3CCCC3)CC2)cc(Cl)ccc1O N1(C(C(n2ncc(C)c2)C)=O)CCCN(C(=O)CC(C)C)CCC1 c1(C(=O)NCC(CNC(c2c(CC)nns2)=O)F)cnc2c(ccn2C)c1 C(=O)(C(C#N)CC1CC1)N(CCCOCCC(=O)NCCC(C)OC)C1CC1 c1(C(C)OCC)nc(-c2cc(C(F)F)n(C)n2)n(Cc2cccc(OC(C)C)c2)n1 C(=O)(C(F)C(F)(F)F)NCC(CNC(C1C(CN(C)C)C1)=O)(C)C c1(C(=O)NCC2N(C(C=C3CCC(C)C3)=O)CC2)ccc(S(=O)(=O)CCO)cc1 C1(CNC(C2(CCC=C)CN(C(c3c[nH]cc3C3CC3)=O)C2)=O)CCCCN1C CC1(C)COCCC1C(N1CCOC(c2cn(CCCCO)nn2)C1)=O N1(C(Cc2c(C)nc(CC)nc2C)=O)CCN(C(=O)Cc2cnsc2)CCC1C CC1(C)C(=O)NCC1NC(C1C2CC3C(C2NC(c2ccc(O)cc2)=O)C13)=O c1(C(N2C(C(N(C)CC3(F)CCC3)=O)C(C)(C)CCC2)=O)ccc2cc[nH]c2n1 C(=O)(C1COc2ccc(F)cc21)NCC1(F)CCN(C(C2C(C#N)C2)=O)CC1 Cc1cc(C(=O)NCCN(C2CCCCCC2)C(C2CC2Cl)=O)[nH]c1C c1(C(N2CC3C(C(=O)NC(c4cncs4)C)(CC3)C2)=O)cc2cc(F)ccc2s1 C(=O)(C(C)(C)CNC(c1cc(C2CC2)no1)=O)NCCCC C1(NC(c2cn(CC)nc2)=O)CC(O)CN(C(=O)C(c2cncn2C)O)C1 C(=O)(CC(C)C(F)F)NC1CC(N(c2ccc(F)cc2C(F)(F)F)C(C)=O)C1 C(=O)(C1=CC2CCCCC12)N1CC(CNC(=O)C=Cc2ccco2)C1 C12(CNC(c3cnc(CC)s3)=O)CCC(CN(C(C3(OC)CCC3)=O)C1)C2 CC1C(NC(=O)C(CO)c2ccccc2)CCN1C(=O)CCC1CCCCO1 C(C(C)(COC)C(=O)NC1C2CC3C1C3C2C(=O)NCCCc1nc[nH]n1)OC C1(C(N2CC(NC(c3cc(-c4ccccc4)co3)=O)(CO)C2)=O)CCCC(=O)N1 C1(OC2CCC2)CCOCC1.N12CCCC1C1(CC1)C(=O)OCC2=O Cc1ccc2cc(C(=O)NC(C3CCN(C(=O)C(C)(C)C(C)C)C3)C)oc2c1 C1(C(N(C(C)CNC(=O)C(C)CCOC)CC)=O)CCC(N(C)C)CC1 c1(C2(C)CC2)cccc(C(=O)NC2CCCC2CNC(C2(C)CCCC2)=O)c1 Cc1cc(C#N)sc1C(N1CCCN(C(=O)C(F)C(F)(F)F)CC1)=O C(=O)(C#CC1CCOCC1)N1C(C)CCC(NC(c2c(O)nnc(C)c2C)=O)C1 c1(C(=O)NCC2N(C(CS(CC)=O)=O)CCC2)ccc2cnnc(O)c2c1 N#Cc1cc(C(=O)NCC2(CO)CCCCCC2)ccc1Br N1(C(C2CC3CC3N2Cc2ccccc2N2CCCC2)=O)CN2CCC1CC2 Cc1cc(N(C2CCNCC2F)C(C2(C)COC2)=O)nc(C)n1 C1(C(=O)NCC(C)(C)NC(C2CC=CCO2)=O)Cc2cc(F)cc(F)c2O1 CN1CC(C(=O)NCC2CCCC2NC(c2cnc(S)n2C2CC2)=O)NC1=O C#Cc1ccc(CC(N2CC(NC(=O)C(C)(C)CCCOC)C(C)C2)=O)c(F)c1 CCC(CCC(=O)NC1CC12CC(NC(=O)Cc1ccc(OC)c(Cl)c1)C2)OC c1(CN2C(c3cccs3)CCC(C)C2)n[nH]c2ccccc12 C1(C(=O)NCC(CC(=O)OCC)C)CCN(C(=O)C(C)N(C)C(C)=O)C(C)C1 C1(C(=O)NC(CC)CNC(=O)CCCn2cncn2)CCC(CO)CC1 Cc1nc(C(=O)NC2CC(NC(=O)COC3CCCC(C)C3)C2)c(=O)[nH]c1C N1(C(c2cnc(-c3ccccc3F)s2)=O)CCC12CCSCC2 C(=O)(CC(C)(C)C(C)=O)NC1CC(O)(CNC(Cc2c(OC)ccc(F)c2)=O)C1 c1(OC)cc(CN=c2ccnc(NC(C)CC#N)[nH]2)cc(OC)c1C C1(NC(=O)COCC(F)F)(CF)CCN(C(=O)CCc2cccnc2)C1 c1(OC)ccc(C=C2CCN(c3cccc(C(C)=O)n3)CC2)c(C)c1 CCC(C)C(=O)C(=O)N1CCC(C(N2CC(C=C)(CC)C2)=O)O1 N1(C(C(C(C)C)O)=O)CCC2CCC(NC(=O)CSc3ccc(Cl)cc3)C12 C1(CNC(C2N(C)C(=O)CC2)=O)CCN(C(=O)Cc2cn(C)nn2)C12CCC2 c1(C(N(C2CCC(NC(CC3C(C)CCO3)=O)CC2)C)=O)cc(F)cc(Cl)c1 CCCCCCC(CC)C(=O)NC1COCCN(C(c2ccns2)=O)C1 N(C1CN(C(c2cccc(O)n2)=O)Cc2ccccc21)C(C(C)(O)C(F)(F)F)=O C1(NC(C(CC)CC)=O)COC2C(NC(c3nc(C)n(C)c3C)=O)COC12 C1(OC)CN(C(=O)C(C(C)C)NC(=O)C2=NOCC2)CC1(C)C C1(CC(N)=O)(NC(=O)C(=O)NCC2CCC3(CC3)C2)CCCCCC1 Cc1nnsc1C(=O)N(C(C)(C(=O)NC(CO)C1CC1)C1CC1)C C1(NC(C2(C)CCC(C)C2)=O)COC2(C1)CN(C(=O)Cc1c(Cl)cnn1C)C2 c1(C(=O)NC(CC)C(C)CN(C)C)cc(NC(C)=O)c(S(N)(=O)=O)s1 C(=O)(CC(C)(C)C1CC1)N1CC(CC(C)NC(CC(C)F)=O)C1 C1(C(=O)OC)CCC(CNC(C2CN(C(=O)Cc3ccc(C)o3)C2)=O)C1 C12(C(=O)NCC(C)ONC=O)CC(CNC(=O)OC(C)(C)C)(C1)OC2C.CC(F)F N1(C(CN(C(CC(C)(C)C2CC2)=O)C2CC2)=O)CCOC2C(O)CC12 CC(C)CC(C)(CO)NC(C1CC(NC(C2OCCCC2(C)C)=O)C1)=O C1(CN(C)C(N)=O)CCCCN1C(=O)C(Cc1ccc(F)cc1)NC(=O)C1CC1 c1(CC)nccnc1C(=O)NCCC1(C(=O)NC(COC)CCO)CC1 c1(C(=O)NC2CCN(C(=O)CSCc3ncc[nH]3)C2)cc(Cl)cc2ccncc12 C(CCCCCNC(c1ncccn1)=O)N(C1CCS(=O)(=O)C1)CCC N1(c2n(CCC#C)c(Cc3ccc(CC)cc3)nn2)CC2CCCCC2C1C c1(C(=O)NC2CCN(C(=O)C=CCN3CCCCC3)C2)ccc(Cl)c(F)c1 c1(NC)cnc(C(=O)NCC(=C2CN(C(=O)CC3CC=CCC3)C2)F)cn1 CCCCC(F)C(=O)NCc1cn(C2CCN(C(=O)C(O)CSC)CC2)nn1 C1(NC(C(F)=CCC)=O)CCCN(C(c2cccc(C(N)=O)c2O)=O)C1C c1(OC)nccc(C(=O)NC(C)C(C)NC(=O)C(c2cnccc2C)(C)C)c1F CC(C)(C)C(O)C(=O)NCC12CC1CN(C(=O)Cc1nc[nH]n1)C2 C(CCCC(C)C)(C(=O)NCC)N(C(CC)CN1CCOCC1)C Cc1nc(CCC(N2CC(CNC(=O)CN3CCCCC3=O)C(O)C2)=O)oc1C c1(C(=O)NC2C=CCN(C(CCCNC(N)=O)=O)C2)cc2cccc(Cl)c2[nH]1 c1(C(=O)NCC2C(NC(c3nc(Br)c[nH]3)=O)C2)c(Cl)ccc2ncccc12 c1(CNC2C(C(N3CC(=O)OCC3)=O)CCCC2)ccc2nccnc2c1 Cc1cc(N2CCC(N3CCOC3=O)C2)nc(N(C)C)n1.N12CCOC(C1)C2 N1(C(c2c(C)cn(C)c2)=O)CCCC(C)(C)C1CNC(=O)CC(C)c1ccco1 c1(CC(N2CCN(C(C(CCC)(C)C)=O)C(C)C2)=O)ccc2c(c1)CCOC2 C1(F)(CNC(=O)COCC2CCCO2)CN(C(c2ncoc2C2CC2)=O)C1 c1(N(c2ccc(C(F)(F)F)cn2)C(C2CNCC2F)=O)ncnc2c1CCCC2 N1(C(CC(C(CC)(C)C)C)=O)CC(NC(=O)CCCC)C2(CCS(=O)(=O)CC2)C1 c1(C(=O)NCC(C)(C)OCC(=O)NCC(C)(O)C2CC2)c[nH]c2nccc-2c1 C1(CCNC(c2n(CCCOC)nnn2)c2sccc2C)CCCCCC1 C1(C(=O)NCCC(O)C(=O)NC23CC(F)(C2)C3)CCCC2(CC2)C1 N1(C(CN(C(C)=O)C)=O)CCC(C)C(N(C(=O)CC(C)n2cccc2)C)C1 N1(C(c2nc(C(C)NC(C3CCCCC3C)=O)oc2)=O)CC(C)CCCC1C CN1C(=O)CCCC1C(N1CC2(CC(CNC(c3cc(Cl)ncc3N)=O)C2)C1)=O n1(CC)ncc(Cl)c1C(N1CCCC(C(C)(O)CNC(=O)Cc2ccno2)C1)=O c1(NC(N2CCCC2)=O)ccccc1C(C)NC(C)CN(CC(=O)OC)C(C)C C1(NC(Cc2ccc(OC)cc2OC)=O)CN(C(=O)C=CS(C)=O)C2(CCC2)C1 c1(CC)cccc(Cl)c1.C12CCCN1C(=O)N(CC(C)CN(C)C)C2 N1(C(C2(COC)CC2)=O)CCC2(C=C(C(=O)NC(CO)C3(C)CC3)C2)C1 c1(C(=O)NC(c2ccccn2)CC)nc(CNC(C2C(C)(C)C2(F)F)=O)oc1C N1(C(CCCOCC=C)=O)CC(O)CC1(C)C(N1CCC(N2CCC2)C1)=O C1(C(=O)NCC2N(C(C(CC)NC(N)=O)=O)CCC2)CN(CP(C)(C)=O)C1 c1(NC(C2C(C)CN(C(C3CCCCO3)=O)C2)=O)cncc([N+](=O)[O-])c1 c1(C(=O)NCC2CC(CNC(CCCOC)=O)OC2)cc(Cl)cc(Cl)c1 c1(OC)cc(C(=O)NC(C2CCCN2C(C2OCC2(C)C)=O)C)ccc1C(N)=O N1(C(c2cc(Br)nn2C)C(=O)NCCCOC)CCC(S(C)(=O)=O)C1 CC1(C)CN(C(=O)CCc2ccccn2)CCN(C(C2CCC(F)CC2)=O)C1 N1(C(CC(C)(F)F)=O)CCN2C(=O)C(NC(c3cnc4n3CCCC4)=O)CC2C1 n1(CCCC)nc(C)c(C(=O)NCC=CCNC(=O)CC2CCC(C)(C)C2)c1Cl c1(CC(=O)NC(C2CN(C(=O)Cn3ccnn3)CCO2)C)cc(F)c(F)cc1F C1(C(N2CC3CC2C3)C(=O)NCCSC)CCC(CCC(C)C)CC1 C1(NC(c2sccc2C2CC2)=O)(CNC(=O)CC2CCC2)CCCC1 CC1OCCC1(C)C(=O)NC1CC(N(C)C(c2cc(C(N)=O)[nH]n2)=O)C1 CC(C)C(C(=O)N1CC2CCN(C(C3CC4CC3CC4(F)F)=O)C2C1)C(C)C CCC(CC)C(C(=O)N1CC(CCCCNC(c2c[nH]nc2Cl)=O)C1)OC c1(SC)csc(C(=O)N(C)CCN(C)C(C2(c3cnn(C)c3)CCCO2)=O)c1 C1(CC(=O)N(C2CC(NC(c3c(CCC)nco3)=O)C2)C)SC2=NCCN2C1=O N1(C(c2c(OC)cccc2)=O)CC(CNC(=O)C(C)N(C)C(C)=O)C2(CC2)C1 c1(C(N2C3CN(C(=O)Cc4sc(O)nc4O)C(C3)C2)=O)nncc2c1CCCC2 Cn1cc(C(N2CCN(CCNC34CCCCC3NC(=O)C4)CC2)=O)c(=O)n(C)c1=O C1(CS(=O)(=O)NCC(C)CN2CCOCC2)CCC(C2CC2)O1 C1(CNC(C2N(C)CCC2)=O)CN(CCCC2CC=CCC2)CCC1(F)F c1(C(=O)NCC2CCCCN(C(c3ccon3)=O)C2)c[nH]c2cccnc12 C1(C)(C(c2n[nH]c(O)n2)N2CCC(C3N(C(C)=O)CCC3)C2)CCCCCC1 C(C)(C)(CCC(=O)NC(C(=O)NCCCCS(C)=O)C(C)O)OC n1(C(F)(F)F)cncc1-c1nc(C23CCCC2C3)no1 c1(C(=O)OCC2(COC)COC2)cc(-c2ccncc2)[nH]n1 N1(C(=O)CCc2ccccc2)CCC2CN(C(C3CCCC(F)(F)C3)=O)CC2C1 Cc1cc(NC(=O)Cc2ccccc2O)ccc1NC(C1CCS1(=O)=O)=O c1(C(=O)NCC2CC(NC(C3CCCCC3)=O)C2)cnc2ccc(Cl)cn2c1=O C1(CCCC)CN(C(C2CCS2(=O)=O)=O)CCN1C(=O)CCCc1ccc(C)s1 Cc1cc(C(=O)NC(C(=O)NC2CC3(CCC3)C2O)c2ccoc2)c(O)nn1 C=CCC(C)(CC)C(=O)N1CCC(C(=O)NCCc2cnco2)O1 Cc1cccc(C(N2CC(N(C(=O)CC=CCc3ccccc3)CC)C(C)C2)=O)c1 c1(CC)c(C(N2CCOC(CCNC(=O)Cc3nncn3C)C2)=O)cnn1C C1(OCCOC(COc2c(C)occc2=O)=O)CC(C)CC(C)(C)C1 C1(C(N2CCC(CC(=O)NCCS(C)(=N)=O)C2)=O)CC2(CC2)CO1 Nc1cnc(C(=O)NCCCCC(=O)NCCC2(O)CCC2)cn1 CC1(NC(=O)Cc2ccc(O)nc2)CCN(C(C2CC(C(F)(F)F)C2)=O)CC1 C1(CCNC(CC=CC=C)=O)CCN(C(c2scc(OC)c2OC)=O)C(C)C1 C(=O)(C(C)C(C)(C)C)N1C(C(=O)NCc2c(C)ccs2)C=CCC1 N1(C(C(C2CCOCC2)C)=O)CCc2ccccc2C1CNC(=O)C=CCF N1(C(COC2CC(NC(c3c(CC)cncc3)=O)C2)=O)CCOC(C)(C)C1 Cc1cc(NC(c2ccc(Cl)cc2Cl)=O)ccc1NC(=O)C1=COCC1 C(=O)(N=c1cc[nH]cc1C)c1c(C)nc(-c2cc(O)nc(O)n2)cc1 c1(C(N2CCC(C(C)NC(c3nn(C)cc3Cl)=O)C2)=O)ncncc1F N1(C(c2n(CC#C)ccc2)=O)CC2CCC2(CC(N2CCC2C(N)=O)=O)C1 N1(C(c2c(C#C)c[nH]n2)=O)CCC2CCC12CNC(c1cccc(CC)c1)=O c1(C(N2C(C)C(C(=O)NOCC(O)C(C)(C)C)CC2)=O)cc2cccnn2c1 CN1CCC12CC(CNC(=NCCc1ccc(O)c(Cl)c1)NCCCF)C2 C1(C(N2CCC(F)(F)C2)=O)CN(C(=O)CCc2nncs2)C2(CCC2)C1 Cc1cc(C(=O)NCC(F)CNC(=O)CC=Cc2cccc(F)c2)c(N)c(C)c1 Cc1nc2c([nH]1)CC(C(N1CCC(CCNC(c3coc(Cl)n3)=O)C1)=O)CC2 c1(C(=O)NCC(CNC(c2cc(Cl)ns2)=O)O)cn2c(n1)CCCC2 CN(C1CS(=O)(=O)c2ccccc21)S(=O)(=O)c1ccc(NCC2CC2)c(F)c1 c1(OC)c(Cl)nc[nH]c1=NCCC(C)NC(c1ncccc1Cl)=O N1(C(C(COC)(C)C)=O)CCC(C(=O)NCC(C)(F)F)CC1(C)C Cc1cc(=NCC2CCC2NC(c2cc(Cl)c[nH]2)=O)[nH]c(C(C)(C)C)n1 Cc1cc(C(N2CCC(O)(C(C)NC(c3ccc(Cl)o3)=O)C2)=O)ccc1C(C)C c1(CC(=O)NCC(C2CC2)NC(C2(OC)CC2)=O)c(Cl)cccc1Br C(CC(C(=O)N1CC2CC1CS2)NC(=O)CC1COCCO1)N(C)C N1(CC(=O)NCCOC)CC2(CN(C(c3n[nH]cc3C(C)C)=O)CCO2)C1 C(=O)(C1=CNC2=NCCC2=C1)N1CCC(CNC(=O)C(F)C(F)(F)F)(CO)CC1 c1(CC(C)C)ncc(C(=O)NCC(C)(CO)NC(=O)C(=O)NC2CC2)[nH]1 c1(C(N2C3(CCN(c4ncc(C)cn4)CC3)CC2)=O)n[nH]c2ccc(C#N)cc12 C(C(=O)Nc1cccc(Cl)c1C)(C1=NOC2CC12)N1CCCC(C)(CO)C1 C1(CC(=O)NCCOC)CN(C(=O)CCCCc2cccs2)C12CCC2 N1(C(C(CC(C)C)NC(=O)C2=CCCC2C)=O)CCC(F)(F)C(O)C1 c1(C(N2CCCC(NC(C3CC4C(C)(C)C4C3)=O)C2)=O)ccc(Cl)c(Cl)c1N CC1CN(C(=O)CC2(CN)CC2)C2(COC2)CO1 C1(C(=O)NCC2N(C(C(CC)=CC)=O)C3C(C2)C3)CCn2c(Br)cnc2C1 C1(NC(C(C)OCCCC)=O)C2CCN(C(=O)C(n3cnc(C#N)n3)C)CC12 c1(SC)ncc(C(=O)NC2CC2CNC(C2(C)CC2(Cl)Cl)=O)s1 C1(C(N(C2CC(NC(c3nc(OCC)oc3)=O)C2)C)=O)CCC(C)CC1 CC1(C(=O)NCCNC(C2CCOC3(CCC3)C2)=O)CCCC(F)(F)C1 C1(OC(=O)CC2CCC23CCC3)CCOC2(CCC2)C1 C1(C(=O)NCCC2CCN(C(C3(NC(N)=O)CC3)=O)C2)CCc2[nH]nc(O)c2C1 C1(CNC(CCC2CCC(NC(=O)CCCC3CCCO3)C2)=O)CC2C=CC1C2 C(CCC(=O)NCc1ocnc1C(=O)NC1C(C)C1(C)C)=CCC=C N1(C(C(CC(=O)OC)(C)C)=O)CC2COCCC2(NC(c2ccc(Cl)s2)=O)C1 CCC(CN(C)C)CC(=O)N1CC2CC1(CNC(c1nc(Cl)ccc1F)=O)C2 N1(C(C(C2CCN(C(c3ncon3)=O)CC2)C)=O)CC2CCCCCCC12 N1(C(C2(COC)CC2)=O)CC2CCC2(CNC(c2ccc(C3CC3)cc2)=O)C1 CC1CCN(C(c2cnc(C(C)(C)C)nc2)=O)CCN1C(=O)Cn1nccn1 c1(OC)cccc2cc(C(N3CCCC(N(C)C(C4CCS4(=O)=O)=O)C3)=O)oc12 C12(C(=O)NCC3(OC)CN(C(=O)CC(F)F)C3)CCCCC1C2(F)F C1(NC(C2C(=C)C2)=O)CN(C(C2=CC(Br)(C(=O)OC)C=N2)=O)C2CCCCC12 c1(C(N2C3CCC2CN(C(=O)C(F)(F)F)C3)=O)cc(Br)c2occc2c1 C(C(=O)N(C)CC1CN(C(=O)C(=O)NC2CC2)CC1C)(C(C)C)OCC(C)OC N1(C(C2(C(=O)NC)CC2)=O)CCC(F)(C(=O)NC2CN(C)C(=O)C2C)CC1 N1(C(c2scc(Cl)c2Cl)C(=O)NC2CCCC2)CCN(Cc2cccnc2)CC1 c1(C(N(CCOCCCNC(C2OCC(C)C2)=O)C)=O)c(F)ccc(F)c1O N1(C(Cc2cc(OC)ncc2)=O)CC=C(CNC(c2ccc(C)cc2)=O)CC1 N1(C(C(COC)COC)=O)CC2CC1CN(C(c1ccn(C3CCCC3)n1)=O)C2 c1(C(N2CCC(N(C)C(c3ccccc3O)=O)C2)=O)[nH]nc2ncc(Br)cc12 c1(C(CC)(C)C)ccc(N2CCCC2c2cccn2C)cc1 N1(C(c2ccc(C)cc2C)C(=O)NCC2CCCO2)CC2(CCCCC2)CC1C c1(N(CC)CC)nc(C)cc(=NCCn2cc(C3CCOC3)cn2)[nH]1 N1(C(C2CCC2(F)F)=O)CCN(C(c2ccnc(N(C)C)c2)=O)C(CC)C1 c12cc[nH]c1C(=O)NC2.N1(OC(COCCC)=O)CCC(C(F)F)C1 c1(C(N(CCNC(C2(C)CC(=C)C2)=O)C)=O)c(C)ccc(F)c1Br C=CC(CC)CC(=O)N1CCCC1CN(C(=O)CC1(N(C)C)CCCCC1)C C1(CC)CC(C(=O)NCc2ccccc2CNC(c2csc(Cl)c2)=O)CCC1=O c1(C(=O)NC(C2CN(C(c3ccc(SC)s3)=O)C2)C)ccc(OCCF)cn1 c1(C(=O)NC2(CC=C)CC2)cnn(C(N2CC(OC(=O)N)C2)=O)c1.C(C)C N1(C(C2CCCN(C(C)=O)C2)=O)CCCC(F)(C(=O)NCC(C(C)C)C(C)C)C1 C12(C(N3CCCC(NC(=O)Cc4cccc(F)c4)C3)=O)CCN(C1)S(=O)(=O)C2 C1(COC)(OC(c2ccc(C(=O)OC)nc2)=O)CCN(C)C1 C1(CN(C(CSCCOC)=O)C)CCCCN1C(=O)C(c1ccccc1)C C1(CNC(=O)CCc2ccc(O)nn2)CCN(C(C2(F)CC2)=O)CCC1(F)F Cc1nc2c(C(=O)NC3CCCCC3CNC(C3CCC(C)C3)=O)cccc2o1 c1(NC(C2CCC(NCc3ccc(C(F)F)nc3)CC2)=O)onc2ccccc12 CC(C)CC(CN(CC(c1ccccc1)O)C)CC(=O)O C(=O)(C(C)(F)C(C)(C)F)NCc1ccc(CC(C)NC(=O)C2CC2)cc1 N1(C(CCC2C(C)C2)=O)CCC(CF)(NC(c2cc(=N)[nH]n2C)=O)C1 CC#CCCC(=O)NCCCC1CN(C(C2(CN(C)C)CCCC2)=O)CCO1 c1(OC)c(C(=O)NCC2CC(CNC(c3nsnc3O)=O)CO2)ccc(Cl)c1Cl c1(C(CC)C(=O)N(CCCn2cc(-c3cc(OC)ns3)nn2)CC)ccc(F)cc1 CC1(C)CC(NC(=O)CSC2CC2)CN1C(=O)CCC1CCCC1(F)F C(CO)(CCCC)NC(COCC(=O)NC(C#C)CC1CCCC1)=O N1(C(C(C)NC(N)=O)=O)C(C(=O)NC23CC(C)(C2)OC3(C)C)CC2CCCCC12 Cc1cc(C(N2CCNC(C(N3CCC(C(F)F)CC3)=O)C2)=O)nc(C)c1 C(=O)(CCC(=O)NN(C)C)NCc1c(C(=O)NCC(CC(=O)OC)C)scc1 c1(C(=O)NC2CCC(NC(=O)OC(C)(C)C)C2)ccc2cc(F)c(F)cc2n1 CCCCC(O)C(=O)NCCCC(C)(C)NC(=O)C(CN(C)C)C(C)C Cc1cc(CCC(=O)NC(C)(CNC(C2(C3(C)CC3)CC2)=O)C2CC2)cc(C)n1 CC1=C(c2ccc(NC(c3cccc(N(C)C)c3)=O)nc2)CCCC1 Cc1cccc(CN(C(=O)C(CCC2CC2)NC(=O)CCC=CC(C)C)C)n1 c1(NC(=O)NC2(c3ccccc3)CCC2)ccc(=NCc2ccc(Br)cc2)[nH]c1 C1(c2onc(-c3cnc(C)[nH]3)n2)C2CCCOC12 Cc1ccc(NC(=O)NC2C=CCC2)nc1 CC(CCCC(=O)N(C)CCN(C)C(C1(C#N)CC1(C)C)=O)c1ccccc1 [N-]=[N+]=NCCCCCCC(=O)N1CC(c2nn[nH]n2)(Cc2ccccn2)C1 c1(N(C)C(=O)NC2CC(c3ccc(F)cc3)C2)c[nH]ccc1=N C(=O)(CCC(CNC(=O)NCC1CCC(Br)C1)OC(C)(C)C)OCC N1(C(C(CC)C(=O)OC)=O)CC2CC(C1)CN(C(C1C3CN(C)CC13)=O)C2 C12(C(=O)NCCNC(C3N(C)CCC3)=O)CCC(C)(CC1)OC2 N1(C(c2ccccc2F)=O)CCN(C(c2cscc2Cl)=O)C(C2CCC2)C1 C(=O)(C(C)P(C)(C)=O)NCC1CC(NC(c2scc(COC)c2)=O)C1(C)C C1(NC(COCCCC#C)=O)CCN(C(=O)CSc2ccc(C)c(C)c2)CC1O C1(C)(C(N2CC(CNC(C(CCSC)(C)C)=O)C(C)C2)=O)CC(C(C)(C)C)=NO1 C1(C(C)=O)CCC(C)CN1C(c1ccc(C(=O)N(C2CC2(C)C)C)[nH]1)=O Cn1c(Cl)cnc1C(F)(F)C(=O)NCC1(NC(c2ccccn2)=O)CCCC1 C1(CC(=O)NC2C(CC=C)COC2)CC2(CC2)CN1C(=O)CC1CCCCCC1 C1(OC)CC(CCNC(c2c(C)ccn2C)=O)N(C(c2cnn(C(F)F)c2)=O)C1 N1(C(CCN(C(C2(C)C(C)C2)=O)CC2CC2)=O)CC(CO)CC(C)(C)C1 c1(CC(=O)NC(C(CC)C)CC(=O)NC(C)C)c(C)nc2cc(O)nn2c1C c1(SCC)c(CC(=O)NCCO)cnn1C.C12CCN(C1)CCNC2=O.SC c1(-c2nn(C)c(-c3ccccc3OCC(F)F)n2)cc(F)cc(F)c1 C(=O)(C(=O)C(C)(C)C)NCC1(C)CC(NC(C2OCCN(CC)C2)=O)C1 C(=O)(C1c2ccccc2C2CC1C2)NC1C(CNC(C(C)=CC)=O)C1 CCC(C)(C)C(O)CNC(=O)CCNC(=O)C(C1(O)CCCC1)F C#CCC(C)(C(=O)N1CC(O)(CO)C1)NC(c1sc(O)nc1C)=O N1(C(C(CC=C)NC(C)=O)=O)CCN(C(=O)C=C2CCC(C)C2)CC1CCO C1(NC(C#CC(C)(C)C)=O)COC2C(NC(=O)CCc3n[nH]c(=N)s3)COC12 N1(C(C2(C(=O)OCC)CC2)=O)C(CNC(=O)CC2CC2C)CC2COCC12 C(=O)(C1OC(C)Cc2ccccc21)O.Cc1cccc2cc(CN(C)C)[nH]c12 c1(CC)ccc(C(=O)NC2CC23CC(NC(=O)CN2CCOCC2)C3)cc1Cl N1(C(C(CCCC)NC(N)=O)=O)CCC(NC(C2CCCSC2)=O)C(CO)CC1 Cc1cc2n[nH]cc2cc1C(=O)NC1CCC1NC(C1CC1F)=O C12(NC(C3C(c4cn(C)nn4)CCOC3)=O)CCC(CC1NC(=O)CCCF)C2 C1(C(=O)NCC(C)NC(c2cn(CCC)nc2)=O)CCC2(CC2)C1 C1(CNC(C(C)(Cl)Cl)=O)CN(C(=O)CCNC(c2ccco2)=O)CC12CCC2 C(CC(=O)N1CCC1CC(=O)OC1(C)CCC1)N(CCC)C.C1CN1CC C(=O)(C1=Cc2ccccc2OC=C1)N1C(CNC(CCC=CC)=O)CCCCC1 c1(C(N2CCC(CCF)C2)=O)cc2scc(Br)c2[nH]1 C1(C(N(C)CCNC(C2CC3(C2)CC3(F)F)=O)=O)CN(C)C(=O)CCO1 c1(C(N2CCC(NC(C(COC)N(C)C)=O)C2(C)C)=O)nccn2nccc12 N1(C(CC2ON=C(C)C2)=O)CCC(CNC(c2occc2F)=O)CC1 C(=O)(CCC(=O)NC1CCN(C(c2cc(O)nn2C)=O)C1)NCCCOC Cc1cc(C(N2CC3(CCN3C(=O)C(C)SC(F)(F)F)C2)=O)c(S(N)(=O)=O)s1 C1(C(=O)NCCCCCNC(C(c2cncc(F)c2)C)=O)CCC(CO)CC1 C1(N(C)C2CC2)CCC2(CCc3ccccc32)CC1.c1(C=O)cccc(F)c1F N1(C(C(C)(O)CC2CC2)=O)CC2(CCCN(C(=O)C(O)Cc3cnc[nH]3)C2)C1 Cc1c(C(=O)NCCOCCN(C)C(C2CCCC2O)=O)cccc1Br c1(CCNC(C(C2CCOC2)NC(C(C=CC)O)=O)=O)cccnc1F C1(NC(=O)NCCCl)CC12CCN(c1nccc(Br)n1)CC2 C1(NC(C(C)OCCOC)=O)CC2C(NC(c3cc(SC)c(C)o3)=O)C2C1 N1(C(c2cnn(CC)c2Cl)=O)CC2C3CCC(C2C1)N(C(C1(C)CCC1)=O)C3 CN1CCc2[nH]nc(C(=O)NCC34CCC(CC3)N4C(=O)C=CBr)c2C1 N1(C(CC2CC(=C)C2)=O)CCC(CCOC)(C(=O)NC(C)COC(F)(F)F)C1 CC(C)CC(C(=O)NC1CN(C(=O)C2=CCSC2)C2(CCCC2)C1)C(C)C S(=O)(=O)(c1cccnc1OC(F)F)NC(C(C(=O)OCC)C)C CCCCCCCC(=O)NC(CC)CCCC(=O)NC(CC)C(C)C c1(C(=O)NC2CN(C(COCC)=O)CC3(C2)CC3)ccc2c(c1)nnn2C Cc1n[nH]c(C)c1COCCCC(=O)N1CC(CC(C)NC(=O)CC(C)(F)F)C1 N1(C(C2N(CC3CN(C)C3)CC3(CC3)C2)=O)CCC2(CC1)CC(C)(O)C2 CC1(C(=O)NCC(CO)NC(c2ccccc2OC(F)F)=O)CCC(=O)N1 S(=O)(=O)(c1cnn2ccc(=NCc3cc(Cl)ncc3Cl)[nH]c12)NC(CCC)C C1(CNC(COCCCC)=O)CCCCN1C(c1cccc(C2CCCC2)c1)=O C1(NC(c2cc(CCC)on2)=O)CCCCCC1C(N1CCCCCC1)=O c1(C(=O)NC2CC(N(C)C(c3cncc(N)c3)=O)C2)ccc(Br)c(F)c1F c1(NC(C2(C)N(C(CC(C)O)=O)CC2)=O)c(F)cc(Br)cc1[N+](=O)[O-] c1(N(C)C)ccc(C(N2CC(n3cc(CCO)nn3)C(O)C2)=O)cc1F N1(CC(c2cccc(SC(C)C)c2)OC)CCC2CCN(CCCN(C)C)CC12 N1(C(CC(C)(F)F)=O)CCCC(C2CCCN(C(=O)CCc3cncs3)C2)C1 c1(C(=O)NC23CN(C(c4cccc(OC)c4)=O)C(C2)C3)c[nH]c2nccc-2c1 C1(NC(C(CCC)(C)C)=O)CN(C)CCN(C(C2CCN2S(C)(=O)=O)=O)C1 Cc1cc2cc(C(=O)NC3CCCN(Cc4ccc(CO)cc4)C3)ccc2cn1 c1(COC)ccc(CC(=O)NC2CCC(Nc3nccc(OC)n3)C2)cc1 C(CCCCCC(=O)N(C1CC1)Cc1cnn[nH]1)NC(C(C)OCCC=C)=O N1(CCNC(C2(C(F)(F)F)CC(=C)C2)=O)CCN(C(C2CC3CCC3C2)=O)CC1 C1(NC(C2CCN(CC)C2)=O)CC2CC(NC(C3(C(F)F)CCCC3)=O)C2C1 N1(C(c2c(C)cc(F)c(Cl)c2)=O)CCC2(CC1)CCN(C(C13CC(C)C1C3)=O)C2 N#Cc1c(C(N2CCC2CNC(=O)CCCCC2CCSS2)=O)cc(Br)cc1F C1(OC)CCn2cc(C(=O)NCC(n3cc(C4CC4)nn3)C)nc2C1 N1(C(C(C(C)(C)C)=O)=O)CC2CC(C(=O)Nc3cc(Cl)cnc3O)C(C2)C1 C=CC1(O)CN(C(=O)CCOCCNC(=O)C=CC2(C)COC2)C1 c1(C(C(=O)NCC2CC(O)(CNC(c3coc(Br)n3)=O)C2)F)ccc(F)cc1 CC1OCCCC1C(=O)N(CCNC(c1cc(N2CCCC2)ncn1)=O)C1CC1 c1(C(=O)NC2CN(C(C3CCN(S(CC)(=O)=O)CC3)=O)C2)nn(C)c(Cl)c1Br c1(C(N2C(CN(C(C(C)=CC3CC3)=O)C)CC(F)C2)=O)ccc2n[nH]c(C)c2c1 CCC(C(=O)N1CCC1C(c1ccccc1)NC1(CO)CCSC1)C1CCCC1 C(=O)(C1=NN(C)C(=O)CC1)NCC(CNC(c1ccc2scc(C)c2c1)=O)OC c1(OC(CCC)=O)ccc(C(=O)NC(c2cn(CC3CCOC3)nn2)CC)cc1 c1(C(C)N(C)Cc2cn(C(C)CN3CCCC3)nn2)cn(C)nc1Cl CCC(C(=O)NC1(CNC(=O)C(O)CC2CCCC2)CCC1)C(C)O CCC(CC)CCC(=O)N(C(C)CCNC(c1cc(C(F)F)ccn1)=O)C c1(CC(=O)NCCCCN(C)C(C2(C)CC(F)C2)=O)cc(F)ccc1F C1(CNC(=NCCC)NC(C)COC)CCc2nncn2C1 CCC(C)CCCCC(=O)NCC1(C)CC(F)(F)CN1C(c1sccc1NC)=O C(=O)(C(CC)C(C)(F)F)NCC(=C)CCNC(c1cc(C)n(C(C)C2CC2)n1)=O c1(CC(=O)NCC2CC2NC(C2CCO2)=O)ccsc1Cl CCC(C)C(O)CC(=O)NCc1ccccc1CNC(c1ccccc1)=O N1(C(C2(C(=O)NOCc3ccccc3F)CC(C)C2)=O)CCc2ncsc2C1 N1(C(c2c(F)cc(OC)c(F)c2)=O)CCC2(CC(NC(=O)C3CC3)CO2)C1 c1(CC(N2C3CC(NC(=O)CCOC4CC4)C2CC3)=O)ccc2nc[nH]c2c1 c1(C(OC(C)C)C2CC2)nc(-c2ccc(Br)cc2)nn1C(C)C1CC1 C(=O)(C(O)CCN(C)C)N(CC(=O)NC(c1cc(C)[nH]n1)(C)C)C(C)C C1(c2nnnn2CCCF)(NCc2cnc(C(=O)OC)s2)CCSC1C c1(CC(=O)N(C2CN(C(C34CCC3C4)=O)C2)C)ccc(F)cn1 C1(CC(=O)NCC(CC)NC(=O)CC2(O)CCCCC2)CCN(C)C1=O N(C(=NCCCCl)NCc1c(F)cc(F)cc1F)C(C)CCc1ccccc1 N1(C(c2cc(CC)on2)=O)CCCC(CC(=O)NC2(CC3CCC3)CC2)C1 c1(C(N2CC(NC(C(CC)Cc3ccccc3C)=O)C2)=O)cn2cccnc2n1 N1(C(CC(C=C)(C)O)=O)CCC2(CC1)CN(C(C1(CN(C)C)CC1)=O)CC(C)O2 N1(C(C=CC(=O)N(C2CCCC2)C)=O)CCN(C(=O)CO)C(CCO)C1 C1(C(C(=O)NC2CCOCC2)N(C2CCCC2)CCN(C)C)CCCOCC1 C1(C)(CNC(C2(COC)CCOCC2)=O)CN(C(C2CCCO2)=O)C(C)(C)C1 C1(C(N(CCC(C)C)C)=O)(CNC(C2CCCN2C(C)C)=O)CCCO1 C1(NC(CC(c2ccccc2F)C)=O)CC2CN(C(=O)C(C)(C)CF)CC2C1 N1(C(C(CC)OC)=O)CCC(C(C)NC(=O)C(c2cccnc2)O)CC1 O=C(CCCF)NCc1cc[nH]c1C(=O)NC(C(F)(F)F)C1CC1 C#CCC(C(=O)Nc1ccc(CCC)nc1)NC(c1csc(C)n1)=O C(c1nc2ccccc2o1)=CC(=O)N(O)C(=O)c1cc(Cl)c[nH]1 N1(C(C(CNC(C2CC(C(=O)OC)C2)=O)(C)OC)=O)CCOC(COC)C1 N1(C(C(CC)C#N)=O)CC2(CCN2C(c2ccc(C(C)(C)C)cc2)=O)C1 C1(C(=O)NCCCC2(C)CC2)(NC(c2cc(CO)on2)=O)CCC(C)(C)C1 c1(C(C(=O)NCC(COC)C(C)C)NC(=O)CC(C)O)c(C)cccc1Br N1(CC(C)C(N2C(C)CCC2C)=O)CCCCCCC1=O C1(N(C2CCN(Cc3ccc(Cl)cc3)C2)C)C2CCC1(C)C2(C)C CCCC(C(=O)N(CC(=O)NC(C)C(=O)N1CCCC1)CC1CC1)C(C)C C(CCCOC)(C(=O)N1CCSCCC1C)NC(c1n(CC)ccc1)=O C12(C(=O)NCC(C)N(C)C(C3(O)CC(C)(C)C3)=O)CCC(C)(C(=O)O1)C2(C)C CCC(C)CC(C)C(=O)NCC(C)(C)CNC(c1ccc2ccnn2c1)=O N1(C(C)C(=O)NC(C)(C)C)CCCOC(C2CCN(C(=O)N(C)C)CC2)C1 C1(OC)CC(NC(=O)C(F)C(C)C)CN(C(=O)CN(C)C(C)=O)C1 N1(CCNC(C2(CCC=C)CN(C(=O)CCC(=O)N(C)C)C2)=O)CCCCC1C N1(C(c2cc(C)c(Cl)s2)C(=O)NC)CCCC(N2CCOCC2)CC1 c1(C(=O)NCCN(CC(C)O)C(c2ccc(Cl)s2)=O)ccc(C(C)(F)F)cn1 Cc1ncc(C(=O)NCCCCNC(=O)CC2(C=C(C)C)CC2)cc1N N1(C(C(N2CC(C)(C)SCC2)=O)=O)CCc2ccccc2C1.c1(C2NC2)cccc(Cl)c1 c1(N(C)CC2CCCN2C(=O)CC2COCC(C)(C)O2)cc(C(N)=O)nc(Cl)n1 N1(C(c2c(S(CC)=O)cccc2)=O)CCC2C(CCCN2C(c2ccc[nH]2)=O)C1 C(N=c1nc2c(cnn2C)c(NCC2(CO)CCOC2)[nH]1)c1cc(CC)on1 n1(CC)nc(C(C)C)cc1C(=O)NCCNC(C1C2CCC(=O)C12)=O C(=O)(C(C)(C)CS(C)(=O)=O)NC(C)C(C)NC(c1ccc(Cl)s1)=O N1(C(C(=O)NCC)=O)CCCN(C(C2C(c3ccccc3)C2(C)C)=O)CC1 C1(NC(C2(C)CCCO2)=O)CN(C(c2ccc[n+]([O-])c2)=O)C2(CCOCC2)C1 c1(C(N2C(C)CCC(NC(C3CC3(F)F)=O)C2)=O)cccc(N=[N+]=[N-])c1 C(=O)(CC1=NN(C)C(=O)C1)N1C(CN(C)C(C2CC(C)(F)C2)=O)CC1 C(C)(CCC#N)(c1nnnn1C1(C)CC1)NCCNC(COC)=O C1(C(=O)Nc2c(C(=O)OC)sc(C)c2)CC(F)CN(c2ncncc2C)C1 C1(C2CC2)(CNC(=O)C2CC2)COC1.C1C(N(C)C(N)=O)N(C)C(=O)C(C)O1 c1(C(=O)NCCC(CNC(C(COC)C)=O)O)cc(C)c(C)cn1 Cc1ccc(OCCn2ccnc2-c2cc(CO)c(C)n2C)cc1-c1ncco1 C12(C(=O)OC)CCC(C(N3CC(CC(C)(C)C)C3)=O)(CC1)C2 Cc1ccc(C(N2CCCC2(C)C(N2CCOC(C#N)C2)=O)=O)cc1[N+](=O)[O-] c1(N2CCCC(CSC)C2)ncc(S(=O)(=O)NC2CCSCC2)cc1Cl CCCC(C)C(=O)N1CC(O)CC1NC(=O)CNc1ccc(C(C)=O)cn1 Cc1c(NCc2ccc(CCC#N)cc2)ncnc1NC1CCOC1C C1(C(=O)NCCOCCCN(C(COCC=C)=O)C)OC2CCC1CC2 N1(C(CC(CC2CC2)NC(c2c(C)oc(C)c2C)=O)=O)CC[Si](C)(C)CC1 N1(C(C)=O)CCC2(CCN(C(C3CN(C(=O)OC(C)(C)C)C3)=O)CC2)C(C)C1 c1(CC(=O)NCCCCCNC(CC2C(C)CCC2)=O)ccc2oc(O)nc2c1 C(=O)(C(C)CC(C)(C)C)N(C)CC1OCCN(C(CCc2c(C)noc2Cl)=O)C1 O=C1NC2CCN(C(C3CSC4(CNC4)C3)=O)CCC2O1 CC1(C)CCCN(C(c2cc3ccccn3c2)=O)C1C(N1CC(F)(CO)C1)=O N#Cc1cc(C(=O)NC2(CNC(c3ccc(CO)nc3)=O)CCOCC2)on1 C=CCCCCCC(c1nnnn1C1CCC(F)(F)CC1)NC1COC(CO)C1 N1(C(c2nc(Br)c[nH]2)=O)CCN(C2CCN(C(C3CCOC3)=O)C2)CC1 C(=O)(CCC(C)C)NC1(CC=C)CN(C(c2cncc(C)c2)=O)C1 c1(CC2C(NC(C3CC(n4cc(C(C)(C)OC)nn4)C3)=O)C2)cccc(F)c1 N1(C(C2C(C(CC)=O)C2)=O)CCC(C(N2CC(OC(C)=O)C2)=O)(CC)C1 C1(NC(c2ccncc2O)=O)CC2CCC(C1)N2C(C1CC2CCC(C1)C2F)=O Cc1cc(CC(N2CCN(C(C3CCO3)=O)CC2CF)=O)ccc1CO C(=O)(CCCC(C)(F)F)NCCC1CCN(C(CC(=C)Br)=O)C1 C=C(CNC(=O)C(F)OC(F)(F)F)CCNC(=O)C(C)SCc1ccccn1 Cc1ccnc(C)c1C(N1CCC(CNC(c2ccc(C3CC3)cn2)=O)CC1)=O N1(C(c2c(Br)ccc(C)c2)=O)CCC2CN(c3ncncc3Br)CCC12 c1(C(=O)OC(C)(C)C2CC2)csc(C)c1.c1(CC2CN(C)C(=O)N2)ccccc1 c1(CC(N2CCCN(C(C(CCSC)OC)=O)CC2)=O)c(F)cc(F)cc1F C(CCNC(c1cc(CSC)on1)=O)(C(C)C)N(C(CC1N(CC)CCC1)=O)C C(C)(c1ccc(F)cc1F)=CC(=O)NC1(C)CC(NC(CCCC#C)=O)C1 c1(Nc2c(C)c(NC(C)CS(C)(=O)=O)ncn2)cnn2c1OCCC2 C(C(O)CC(=O)Nc1cccc(CSC)c1)NC(C1(OCC)CCCC1)=O c1(OC)cccc(C)c1C(N1CC(CNC(C2(F)CC2)=O)C(O)C1)=O CC(C)CC(C)(CNC(=O)CC1CC12CC2)NC(c1ccnc(CN(C)C)c1)=O N1(C(COCc2nnc(C)s2)=O)CCOC2(CCN(C(=O)CCC3CC3)C2)C1 CC1OCCN(C(C2CCCCN(C(C3CC4(CCC4)C3)=O)C2)=O)C1CO C1(N(C)C)CCN(C(=O)C(CNC(c2ccc(O)nn2)=O)CC2CC2)CC1(C)C C12(COC)CCC(C(N3CCCN(C(=O)CNS(C)(=O)=O)CC3)=O)(CC1)CO2 c1(C(N(CCC)CCNC(=O)CCC(=O)N(C)C(C)C)=O)cc(Cl)cc(Cl)c1 N1(C(C(C(C)C)CN(C)C)=O)CCC(CNC(=O)CS(=O)(=O)CCO)C(F)(F)C1 NS(=O)(=O)c1cc(C(N2CCCC(Cn3cc(-c4cn[nH]c4)nn3)C2)=O)cc(Br)c1 Cc1ccn(C(C)C(=O)NC2C3CC2N(C(=O)CC2CC(F)C2)C3)c(=O)c1 N1(C(C(CN(C)C)O)=O)CCCC(n2cc(CSc3nccs3)nn2)C1 CCC(C)CCCCC(=O)NCC1CC1C(=O)NCc1cccc(OC)c1 C1(C(=O)NCC(C)CN2CCCC2)CC(C)N1C(c1cncn1C1CC1)=O c1(C(N2CC3C(CNC(=O)CCCn4ccnc4)(C3)C2)=O)n[nH]c2c1CCOC2 c1(N2C(C)C(NC(C3CC34CCSCC4)=O)CCC2)ccc([N+](=O)[O-])cc1 Cn1oc(C(N2CCC(C(F)F)(CNC(C3(c4ccno4)CC3)=O)C2)=O)cc1=O c1(C(c2nc(C)c(C)[nH]2)(c2n(C(CC)C)nnn2)NC)cnc(N(C)C)c(F)c1 C1(C(=O)Nc2ccccc2OCc2ccccc2Br)C2CCN(CC2)S1(=O)=O CCC(C)(COC)C(=O)NCCC1(O)CCCN(C(=O)CCc2ccon2)C1 c1(C(N2CCC(C(O)C(F)F)CC2)C(=O)NCCOC)ccc2nc(C)[nH]c2c1 N1(C(c2ccn(CCCC)n2)=O)CC2CCC(CNC(=O)CCSCC)C2C1 CC(C)C(C(=O)N1CC(CN(C)C(C2CCS2(=O)=O)=O)C1)n1cccc1 N1(C(C(C)C)=O)CCOC(C(=O)NCCc2cccc(C(F)(F)F)c2)C1 C12(CNC(C=CC(C)C)=O)CCC(CN(C(=O)COCc3cccnc3)C1)C2 C12CC13CCN(CC3)C(=O)COC2=O.c1(C2C(C(C)(C)O)C2)ccccc1 c1(C(=O)NCC(C)(C)NC(c2cnc(NC(C)=O)o2)=O)ccc2cnccc2n1 C1(CCNC(CCC=C)=O)CN(C(c2ccc(O)c(Br)c2)=O)CC(C)O1 CC(C)CC(CNC(c1c[nH]nc1CNC(C1CC(C)CC(=O)N1)=O)=O)CO C(=O)(C(C)(C)C(N)=O)NC(CCN(C(c1c(C(C)C)ncs1)=O)C)C N1(C(CCC=C)=O)CCCC(CC)(NC(c2cnccc2N2CCOCC2)=O)C1 C1(NC(c2scc(C)c2)=O)CC2CC(C1)N(C(c1cnsn1)=O)C2 C1(C(=O)NCC(C)NC(C2(C)CSC2)=O)CCc2nncn2CC1 c1(C(N2C(C)CCC(NC(=O)C=C(Cl)Cl)C2)=O)ccc(S(N)(=O)=O)c(Cl)c1 C1(OC)(CNC(c2cc(-c3ccccc3)no2)=O)CCN(C(C2CC2F)=O)C1 N1(C(C(CC)CC)=O)CCCC2CN(c3c[n+]([O-])ccc3[N+](=O)[O-])CCC12 CC1=NOC2(C1)CC(C(=O)NC(C1CCCN1C(=O)C(=O)Cc1cccs1)C)C2 c1(C(N)=O)cc2cc(NC(C34CCCC3CC(=O)CC4)=O)ccc2[nH]1 C1(CNC(=O)C=CC=C(Cl)Cl)CC2CCC1N(C(=O)CCC1CC1CC1CC1)C2 c1(OCC(=O)NCC2(NC(c3nn[nH]c3Cl)=O)CCOC2)ccccc1C(F)F c1(CC(=O)NCCCNC(c2c(C)c(Br)n(C)n2)=O)cn2c(C)cncc2n1 N1(C(c2c(C)noc2C(F)(F)F)=O)CCCN(C(=O)C(F)C(F)(F)F)C(C)C1 C=CCCCCCCC(=O)NC1CN(C(c2ccc(C(F)(F)F)o2)=O)CC1OC C1(C(=O)NCC2CC(C(=O)NC3(CCCF)CC3)CO2)CC2(C1)CC2(F)F C(=O)(C(C(C)(C)C)n1ccnn1)N(C)CC1CN(C(CC2(NC(C)=O)CC2)=O)C1 C=CC1(C(=O)N2CC(O)CCO2)CCN(C(=O)Cc2ccc(C)nc2)CC1 c1(C(=O)NCc2cc(C(N3C(CC)CC(O)C3)=O)no2)cc(=O)n(C)cn1 CC1CC2(CCN(C(C3CNC(=O)CN3C(=O)CCC(N)=O)=O)C2)CO1 c1(C(=O)NCC(CCOC)NC(c2cscn2)=O)cc(COC)oc1C CC1C(NC(c2cnn(C)c2OCc2ccccc2)=O)CCCN1C(N)=O c1(C(=O)OCCc2ccc(Cl)c(Cl)c2)nc(Br)n2ccsc12 C1(NC(c2ncsc2C(F)(F)F)=O)CCCN(C(=O)C(c2ccccn2)O)C1 c1(C(=O)NC2CC(NC(c3nnc(O)nc3O)=O)C2)cc(F)c(F)cc1Cl N1(C(C(COC)(C)O)=O)CC2CCCCC2(CN=c2nc(C)cc(C)[nH]2)C1 CN1CCCC(CC(N2CC(O)(C(C)(C)CNC(=O)C=C(Cl)Cl)C2)=O)C1 c1(C(N2CCC(C3CCCN3C(c3ccnnc3)=O)C2)=O)ccc(O)c(F)c1 CC1CCCN(C(=O)C(=O)N(C)Cc2nc(-c3ccco3)no2)C1 CC1CCN(C(=O)CCCC(=O)C2CC2)CC1NC(=O)C(C1CCCCC1)O CON1CCC(C(=O)NC(C)CCN(C)C(c2ccc(C#N)cn2)=O)CC1 c1(NC(C)C)cccc(-c2nn[nH]n2)c1F.n1(C(C)C)ncc2c1NC2=O C1(C#N)(C(=O)NCCC(=O)NCCn2c(CC)nnc2)CCCOC1 C1(CN(C)C(C23CSCC2C3)=O)CCCN1C(C1(n2cccc2)CCCC1)=O C1(OCC)CCC(C(=O)NCCCNC(=O)C(c2ccnn2C)C)CC1 CC(CNC(=O)C(F)n1ccnc1)CC(=O)N1CCCC1CC1CC1 C(=O)(C1=C(C)OCCS1)N1CCN(C(CCSCCCC)=O)CC1CCC C#CCC(C(=O)NCC(F)F)NC(=O)CC12CCCC1C2 N1(C(c2c(C(C)C)onc2)=O)CCC(C(=O)N(C)Cc2cnn(C)c2)C(O)C1 N1(C(CCCNC(C)=O)=O)CC2CC(O)C1C2NC(c1ccn(CC(C)C)n1)=O C1(CNC(CC2C(CNC(CCCOC(C)=O)=O)C2)=O)CCOC1(C)C CC1COc2ccc(C(CNC(=O)CC3CS(=O)(=O)C3)N(C)C)cc21 C1(NC(C2N(C(c3ncn(CC)c3)=O)CC=CC2)=O)CC=C(C(C)C)CC1 N12CCC3CC1CN(C3)CC2=O.c1(CC)ccc(NCC#N)cc1 C=CC(C)(O)CC(=O)NCC=CCNC(C1CC(COC)C1)=O CN1CC(F)CC1C(N1CCC1CNC(=O)CCc1cccnc1)=O c1(C(=O)NCCC(C)N(C(CCc2scc(C)n2)=O)C)cnc2sccn12 Cc1nc(NC(C2CSCCN2Cc2ccc(O)c(I)c2)=O)c(C#N)n1C O=C(CC1=CCCCC1)NC1CC(CCNC(C2CCCCC2C2CC2)=O)C1 CCCCC(C(=O)NCC(N1CCCCC1)=O)NC(=O)C(F)C(=O)OCC C(=O)(C1=COc2ccccc2O1)NC1CC(NC(CCNC(=O)NC)=O)C1 c1(C(N(CCC(C(C)C)NC(CC2(C=C)CCC2)=O)C)=O)ccc(C)nc1C Cc1ccc(C#N)cc1C(=O)NC1C2CC3C1C3C2C(=O)NCC1CC(=C2CC2)C1 N1(C(c2ccnc(C)c2C)=O)CCC2(CC1)CC2NC(=O)CCn1cccn1 C=CCC(C)(C)CC(=O)N1CCC(NC(c2cc(CC(C)C)[nH]n2)=O)C12CCC2 CC1(C#CC(=O)NCC2CC3CCC2N3c2ccnc(C3CCC3)n2)CCCO1 C1(Cl)(C(N2CC(C(N)=O)(CNC(C3CCCC3)=O)C2)=O)CC12CCC2 c1(C(=O)NC2C(C(=O)NCC(CC)(C)OC)C2(C)C)cnc(Cl)n1C c1(C(=O)NC2CC3CN(C(Cn4c(C)cnn4)=O)CC32)ccnc2c1CC(=O)N2 c1(CNC(C(CC#C)(C)C)=O)nc2c(s1)CN(C(C1(c3cc[nH]n3)CC1)=O)CC2 CC1CC(NC(C2C=CCN2C(=O)CCC(C)(C)C)=O)CC(C)(C)C1 C1(NC(c2cnn(C(C)C)n2)=O)(CNC(=O)CCNC(N)=O)CCCCC1C CC(=O)CC(C)(C)CC(=O)N(C(CNC(c1ccc(Cl)cc1C)=O)C1CC1)C C1(C(=O)NCCc2ccncc2)CCN(C(c2cccc(F)c2O)=O)CC1O c1(OC)ccc(C=CC(N2CCC(NC(=O)Nc3c(F)cccc3I)C2)=O)cc1 C1(CNC(=O)C(=O)NCc2cccc(Cl)n2)CCCCN1C(C1CC1CF)=O N1(C(CN(CCC)C)=O)CCC2(CC1)CC(C)N(C(C1CC3CCC3C1)=O)C2 N1(C(CC=C(C)C)=O)CCC(NC(C2CCCN2C2CCCC2)=O)CC1C c1(OC)c(Br)cc(C(=O)NCC2CCN(c3nccc(C)n3)CC2)cc1[N+](=O)[O-] CC1CCC(NC(C2(CN(C)C)CC2)=O)CN1C(=O)CC1(C2CC2)CC1 N1(C(=O)OC(C)(C)C)CCC(C(=O)NCC2OCC23CCC3)C12CCC2 C(=O)(C(CCC=C)NC(=O)CC(C)SC)NC(C#C)(C)C CC#CC1CCN(C(=O)C(C)(CNC(=O)CCOC2COC2)CC)C1 Cc1nc2c(o1)CCN(C(=O)COC(C)(C)CNC(C1COCC1C(N)=O)=O)C2 C1(N(c2cccs2)C(N2CCC2)=O)CCN(C(=O)CC2CCC(=O)O2)CC1 C1(CNC(c2c(C)nc(CCC)o2)=O)CN(C(=O)CC2CCCSC2)CCN1C N1(C(C=C(C)C2CC2)=O)C2CCC(C2)C1C(=O)OC(C)(C)C.C12(CC1)C(=O)N2 c1(C(N2C(C(=O)NCCOCC(C)C)C(C)CC2)=O)cc2cccnn2c1 c1(C(=O)NCCCN(C(=O)C(CO)C(C)(C)C)CC)cccc2ccoc12 C(=O)(C1=NOC2(CCN(Cc3cc(Br)cc4[nH]ccc34)C2)C1)N1CCC(OC)C1 N1(Cc2cncc(OC)c2)CCC(O)C(C(=O)Nc2cc(OC)ccc2I)C1 N1(C(C2(OC)CS(=O)(=O)C2)=O)CCCN(C(=O)Cc2ccc(F)c(C)c2)CC1 C1(C(NOc2cc(C)no2)=O)Cc2ccccc2C1C c1(C(=O)NC2(CC)CC2)ccc(CNC(=O)CC2CC2(Cl)Cl)nc1 C1(NC(c2c(OC)nsc2)=O)C2CC3C(C2)C13C(=O)NOCCSCCO c1(OCCNC(=O)NC(c2ncccn2)CC)ccccc1O N1(C(=O)CCOCC2CCCO2)CC(O)CC1C(=O)NC1C2CCC1CC2 C(=O)(C(C)(C)C1=CCN(C(=O)CC=C(C)C)C1)NC(CC)C(C)(F)F c1(NC(C(=O)NCc2ccc3c(c2)CCOC3)=O)n[nH]c2ccc(C(=O)O)cc12 CC1(C)CCC(C(=O)NCc2nc(C3CC3)n[nH]2)(NC(=O)CCOCC2CC2)C1 CN1CCCCC(C(=O)NCC2CC3CCC2N3C(C2CCCCN2C)=O)C1=O N1(CCCCC)CCCC1CNC(c1cc(C(F)(F)F)cs1)=O c1(C(=O)NCC#CCNC(C2(C)CCNC2=O)=O)n[nH]c2c1CCC2 CC(C)(C#Cc1cn(CCO)nn1)N(C(=O)C(C1(O)CCCCC1)(F)F)CCO N1(C(C(C)(C)OC)=O)CCC(C2CN(C(=O)C(CO)C(F)(F)F)C2)CC1 CCCCCCC(=O)NC(CCCOC)C(=O)N(C1CCC1)C1CCC1 C(=O)(C(C)(C)C(=O)OC(C)(C)C)N(CCC)CCNC(=O)Cc1sc(C)nc1C N1(C(C2CC(=C3CCC3)C2)=O)CC(O)(C(F)C(=O)NC2C(O)CC2O)C1 C1(C(=O)NCC(C)NC(CCCC(=O)NC(C)C)=O)C(C)OC(C)C1C N1(C(=O)C2CC2)CC2CC(C1)CN(C(c1coc(O)n1)=O)C2.C12(CC1)C(=O)N2 n1(CC(=O)NC23CCN(C(c4cccnc4)=O)CCC2C3)cnc2ccccc12 N1(C(CCN(CCC)C)=O)CC(NC(=O)CCC2CCCC(=O)N2)C(F)C1 c1(C(=O)Nc2c(C)cccc2)ccn2c1CS(=O)(=O)CC2 N1(C(c2ncc(CC)s2)=O)CCC(NC(=O)C(C(C)C)NC(=O)COC)C1C N1(c2cc(F)nc(-c3ccccc3)n2)CC2C3CCC(CC3)C2C1 c1(OCCC)cc(NCC2(CNC(c3ccc([N+](=O)[O-])o3)=O)CC2)nc(C)n1 N1(C(C(C)SCCCC)=O)CCOCC1CC(=O)NCCC(O)C(F)F c1(CC)cc(N)c(C(=O)NCC(C)(O)CNC(c2cn[nH]c2)=O)cc1F C1(Cl)(C(COC)=O)CC1C(=O)NCC(=O)OC(C)C C1(C(C)(C)NC(=O)Cc2ccsc2)CCN(C(C2CCCN2S(C)(=O)=O)=O)CC1 c1(C(=O)NCCC(CNC(CCCCC#C)=O)O)cc(C)c(OC)c(C)c1 CC(=O)CCCC(C)C(=O)NC(Cn1cccn1)C(=O)NCC1(C)CC2(CC2)C1 C1(NC(c2cnc(C)s2)=O)CN(C(c2ccc(C#N)c(C)n2)=O)CC1N=[N+]=[N-] C(=O)(CCC(F)F)NC1CC(CNC(CC=CCC)=O)C1 Cc1ccc(N2CCC(CN(CC(C)O)C(=O)Cc3cccc(F)c3)C2=O)cc1 CC1(CNC(c2cccc(CN=[N+]=[N-])c2)=O)CCN(C(C2CCCC3CC23)=O)C1 Cc1scnc1C(=O)N(CCC(c1cccs1)NC(C1CCC1)=O)C N1(C(N(c2ccccc2)CC)=O)CCC(C)CC1CSC1CCC1 C=CCCCCCC(=O)N1CCC(NC(=O)CCCN2CCCC2)CC1 C#Cc1cc(C(=O)NC2CN(C(C3CC34CCCC4)=O)CC2CO)cc(F)c1 N1(C(c2c(C#N)nc[nH]2)=O)CCC2CC2(NC(=O)C2=COCCO2)CC1 CC1CN(C(C2Cc3ccccc3O2)=O)c2cccc(Cl)c2O1 C(=O)(C(C)S(C)(=O)=O)NC(CC(C)C)CNC(=O)C=CCOc1ccccc1 c1(CC(=O)NCC2(CNC(C(C(C)C)CN(C)C)=O)CC2)cccc2c1COC2 N1(c2n(CCC=C)c(-c3ccc(OC)cc3I)nn2)CCOC(C)(C2CC2)C1 C1(C(C)NC(c2cc(C3CC3)on2)=O)CCCN(C(=O)C=CC2CC2)C1 C1(NC(C2C(=C)CC2)=O)CCN(C(=O)CC2CCC(=O)N2C)C12CC2 CC1(C)CCC(O)(C(=O)NC2CC(F)(CNC(=O)CCNC(=O)CO)C2)CC1 N1(C(CC(C)(C)OC)=O)C(CNC(=O)C(C)(C)C(C)(F)F)CC2COCC12 CC1CN(C(c2cnnc(O)c2)=O)CCC1NC(c1cnc[nH]1)=O CN1C(=O)CCC1C(=O)NCC1CCN1C(c1n[nH]cc1C1CCC1)=O C1(OC)CC(O)CN(c2nnc(-c3ccc(F)c(F)c3)n2C)C1 C(=O)(CS(=O)(=O)C(C)(C)C)N1CCCC(N(C(=O)CC2C=CCC2)C)CC1 c1(C(=O)NC23CC(CNC(C4C(C(=O)OC)CC4)=O)(OC2)C3)c[nH]cc(F)c1=O N1(C(CS(CC)=O)=O)CCC2CN(C(c3c(F)cccc3Br)=O)CC2C1 C#Cc1ccc(C(=O)N(C2CN(C(c3csc(CC)n3)=O)CCC2C)C)cc1C C1(C)(CC(=O)N(CCCOC)C)CCN1C(=O)CCOCCCOC CN1CCC(C(N2CC(NC(c3ccnc(C(F)F)c3)=O)C(C)(C)C2)=O)S1(=O)=O C(=O)(C(CCc1cnn(C)c1)N1CCCC1COC(C)(C)C)NC(CC)C C1(CCC)(NC(C2CCC(COC)O2)=O)CCN(C(c2cccc(Cl)c2Cl)=O)CC1 c1(C(N2CC(C(=O)Nc3ccc(OC)nc3)C2)=O)cc(C(C)C)cc(F)c1 C1(C(N(C2CCN(C(=O)OC(C)(C)C)C2)C)=O)CCC(C(N)=O)CC1 N1(C(C2CCC(C(N)=O)CC2)=O)CC(C2CCCN(C(=O)C(F)C3CC3)C2)C1 CC1CC(CNC(C2(CC3CC3)CC2)=O)CN(C(C2(F)CCCCCC2)=O)C1 c1(OC)csc(C(N2CC(OC)CC2CNC(C2CC(N(C)C)C2)=O)=O)c1OC c1(C(N2CC(C=C)C(NC(=O)CC3CC3CC)C2)=O)c(C)cc(C)oc1=O CC(CNC(c1ccnn1C1CCC1)=O)(CO)NC(=O)CCCC1CCOCC1 CCCCC(CNC(C1CCC(N(C)C)CC1)=O)NC(c1[nH]c(C)cc1C)=O CCCCC(O)C(=O)NCc1cc(O)nc(CNC(c2cc(O)n(C)n2)=O)n1 c1(C(=O)NCc2nc3ccccc3[nH]2)nnn2c1CN(Cc1occc1Br)CC2 N#CC1(C(N2CC3CC3(CNC(=O)CCC3CCC3)C2)=O)CCCOC1 c1(C(=O)NC23CC(CNC(C4C(C)OCCC4)=O)(C2)C3)cc2ccsc2s1 N1(C(COC)=O)CCC2(CCCN2C(c2cnccn2)=O)C1 c1(CC(=O)N(C(C(=O)OC)C)C2CC2)sc2ccccc2c1C C1(CC(=O)N(CCC(c2cccs2)NC(C(C)C2CC2)=O)C)CCC=CCC1 C(=O)(C1=CC2(CCOCC2)C1)NC1C2CN(c3snc(C(=O)OC)n3)C(C2)CC1 c1(OC)cccc(C(O)C(=O)NCC(C)NC(=O)Cc2cnc(C)[nH]2)c1 N1(C(c2cnc(C(C)=O)s2)=O)CC2CCC(CNC(=O)C(C)(C)C(C)O)(C2)C1 CCCCCC(C)C(=O)N1CC2CN(Cc3cccc(SC)c3)CC12 N1(Cc2c(CC)cccc2)CC2(CN(C(c3ccc(C)nc3)=O)CC2CO)C1 N1(C(C23CC(C(C)(C)C)(C2)C3)=O)CC2CN(C(C3CC3C#N)=O)CC2C1 c1(C(N(C2CCCC2)CCOC)=O)cc2c(s1)CCC(C(C)C)C2 C(C(=O)NCC12CC(NC(=O)CC3CC(=O)NC3=O)(C1)C2)(C(C)C)SC N1(C(CCCC#N)=O)CCC2CCCC12C(=O)Nc1cnn(CCO)c1 CCC(C(=O)NC1(c2ccccc2)CN(C(=O)C(C)n2cccn2)C1)C1CCC1 Cc1ccc2c(c1)C=C(C(=O)NC(C)CN(C(=O)C=CCF)C)CO2 CP(C)(=O)COCC(=O)NCC1CCC(NC(c2ccc(Br)s2)=O)C1 C1(CCNC(c2onc(C)n2)=O)CCN(C(=O)CN(c2cccs2)C)C(C)C1 CS(=O)(=O)C1CN(CCCO)CC1NS(=O)(=O)CC1CCC(F)(F)CC1 c1(CC)c(C(=O)N(CC(O)CNC(=O)C(C)n2ccnc2)C)ccn1C C=CCCCCCCCC(=O)NCCC1CCC(NC(c2[nH]cnc2C#N)=O)C1 C1(OC)CN(N2CC(O)C(O)CC3(CCOCC3)C2)CC1c1cnn(C)c1 Cc1ccc(S(=O)(=O)N(c2ccc(F)cc2C(F)(F)F)C(C)C)cc1C C1(NC(=O)Cc2ccc(Cl)s2)C2CC(O)C1N(C(c1ccnc(C3CC3)n1)=O)C2 c1(C(N2C(CC)CN(Cc3cc(Br)cc(Br)c3)CC2)=O)cccc2c(I)n[nH]c12 C1(C(=O)NC2CCN(C(C3CC(CC)C3)=O)C2C2CC2)CCc2c[nH]nc2C1 N1(C(c2c(C)ocn2)=O)CC2CCC1C(CNC(c1sc(C(C)C)nc1C)=O)C2 C1(C2CC2)(C(=O)NCC(CCCC)NC(C2CC2(C)CCOCC)=O)CC=CC1 N1(C(c2cn(CC)nc2)=O)CC2CC(CNc3cc4nncn4cn3)CC1C2 C(=O)(C(F)(F)CC)N(CC(C)N(C(C1C(CC)C1)=O)C)C CC(C)CC(O)C(C)C(=O)NCC=CCC(=O)NC(C)(C)CCF C1(NC(CCSC)=O)CCC(CNC(c2ccccc2C(N)=O)=O)CC1 c1(C(=O)NC2CCN(C(c3c(C)snc3)=O)C(C)C2)c(F)ccc(N)c1F Cc1c(NC(=O)C(N2CCC(CN(C)C)CC2)c2ccnn2C)cccc1F c1(C(N2CC(NC(CCC=C)=O)C(CO)CC2)=O)ccc(O)c(C)c1C N1(C(CCC=CC)=O)CC(C(=O)NC2CCC(C3CC3)C2)CC1(C)C N1(C(C2CC(=C)C2)=O)CCC2CCN(C(c3ccc(O)c(N)n3)=O)CC2C1 C1(CCOC)CCN(C(=O)CCNC(C2(CSC)CCOC2)=O)CC1 c1(OCC)cccc2c1OCC(C(=O)NC(C)C(C)NC(=O)CN(C)C(N)=O)C2 C12(C(=O)NCC(CNC(C=NOC)=O)(C)F)CC=CCN1CCC2 C1(NCC2CCC(CCC)CC2)CC2(CCC2)C1OC.c12ccccc1OC2 Cc1ncnc(C(N2CCN(C(=O)CC3CCC(C)O3)CC2)=O)c1C N=c1[nH][nH]cc1C(=O)NC1CC(CCNC(c2[nH]nnc2C2CC2)=O)C1 CC(C)CCCCCC(=O)NC(C)CCCNC(=O)Cc1ccccc1CC#N c1(C(=O)NC2(COC)CCN(C(=O)C(C)=C(C)C)CC2)n[nH]c2c1CC(C)CC2 C1(C(=O)NC(CN(C(=O)C(=O)NCC(F)(F)F)C)(C)C)CC2CC1CO2 c1(C(N(CCN(C(C2(C(=O)OCC)CCO2)=O)C)C)=O)ccnc(Br)c1N c1(OC)cc(OC)cc(NC(N2C3CN(Cc4cc(Cl)cc(I)c4)CC23)=O)c1 CCC(C)C(C(=O)NC1CCC(CO)CC1)N(C(=O)C=CCF)C C12(NC(CC(C)CN(C)C)=O)CCC(C(=O)NCCN3CC(OC)C3)(CC1)C2 N1(C(C(CCCC)O)=O)CC2CCCC(C1)N2C(c1scnc1CC)=O C1(OC)CCCN(CCC(=O)N(C2CCCC2O)C)C1 C(=O)(CC1=CCOCC1)N1CCCC(CNC(=O)Cc2ccsc2Cl)C1 C(=O)(C(CC)C(C)O)N1CC(CN(C(Cn2ncc(C(=O)OC)c2)=O)C)OCC1 c1(-n2ncc(C(N3CCC(c4cn(C5CCC5F)nn4)C3)=O)c2)ccccc1F CCCCCCCC(=O)NCc1ocnc1C(=O)Nc1cnc(C)nc1C C1(C(C2CCCO2)N(C(CC=C(C)C)=O)C)CCN(C(=O)CC2(N(C)C)CCC2)CC1 N1(C(c2ccc(CNC(C(C3CCOC3)OC)=O)o2)=O)CC(CO)C1(C)C C1(NC(=O)CC2CC2)CC2(C1)CC(C(=O)NCC(O)C(F)(F)F)C2 C=CC(F)(F)C(=O)N1CC(O)(C(=O)NCCNC(c2occc2COC)=O)C1.CC O=C1CC(CC(N2CCC(O)(C(=O)Nc3sncc3C(N)=O)C2)=O)C(=O)N1 c1(C(N2C(C)CC(NC(c3cnc(C)nc3)=O)C2)=O)cc(C)c(F)cc1Cl Cc1sc(=O)n(CC(=O)N(C)CC2CCCN(C(c3cc(Cl)c(Cl)[nH]3)=O)C2)c1C N1(C(CCc2ccnc(C)n2)=O)CC2CN(C(C3(C)CCCC3O)=O)CC2C1 c1(C(c2n(CC=C)nnn2)NCc2sccc2C(=O)O)ccc2c(c1)CCOC2 Cc1ccc(CN(C)C)cc1Br.N1(C2CNC2)C(C2CC2)C1 CCCCC(C(=O)N(CC(C)(C)CNC(=O)C(CCC)C1CCC1)C)N(C)C C1(CNC(C2(C)CCCS2(=O)=O)=O)CC2(CCN(C(=O)CC34CC(C3)C4)C2)CO1 CC1Cc2cccc(C(=O)NC3CCCCN(C(=O)CCc4ccco4)C3)c2O1 Nc1ncccc1C(=O)NCCn1cc(CNC(c2coc(C3CC3)n2)=O)nn1 C(=O)(CCCC(=O)N1CCOC(CN(C)C(C2CCCC2)=O)C1)NCCC Cc1cc(NC(c2csc(N(c3ccccc3Cl)C)n2)=O)n(C(=O)N)n1.CCO C(C(=O)NC(C)C)(C(C)(C)C)NC(C1(C)CN(C(C(C)OCOC)=O)C1)=O S(=O)(=O)(c1ccc(NCC(=C2CCSCC2)C2CCOC2)c(C#N)c1)NCCC=C c1(C(=O)NCCC(C)NC(C23CCCC2C3Br)=O)cc(C#N)cn1C N1(C(CC(C)(C)O)=O)CCN(C(=O)C(C)(O)c2ccccc2)CC1c1cn[nH]c1 c1(C(N(CC(O)CNC(=O)CC2(CO)CC2)C)=O)cc(Br)c2nccnc2c1 C1(CCCNC(C2CC(C)OC2)=O)CCN(C(=O)Cc2nc(C3CC3)cs2)CC1 c1(-c2nc(CC(=O)NC(C3(C)CC3)C)[nH]n2)cccc(Br)c1 N1(C(C(CC#C)(C)C)=O)CCCC(NC(c2cc(C(N)=O)cn2C)=O)C(F)C1 c1(C(=O)NCC2(O)CN(CCc3cn(CC)nc3)C2)c(C)nn(C)c1C C(C(O)C(F)(F)F)NCC1N(C(c2ccccc2)=O)CC1 CCN(CCO)NC(=O)C(C)OC(c1cc(S(N)(=O)=O)cc([N+](=O)[O-])c1)=O N1(C(CC(COC)C)=O)CC2CCN(C(c3ccc(F)cc3OC)=O)C2C1 C(=O)(C1=NN(C)C(=O)CC1)NC1C(OC)CN(C(=O)C(O)CC(C)C)C1 N1(C(CC(C)c2cccnc2)=O)CCC2(CCN(C(=O)C3=CCCCO3)C2)C1 c1(C(N(C2CCCN(C(C(C)C#N)=O)C2)C)=O)ccc2[nH]c(=O)c(=O)[nH]c2c1 c1(C(=O)NCC2N(C(C(C)C)=O)C3C(C2)C3)nc2c(Br)cccn2n1 N1(C(C2CCC(=O)N2)=O)CCOC(C2(C)N=N2)C1.C1(N)CCCCCC1.CS CCC(C)(C)CCCC(=O)N1CCCC(C)(C(N2CC(=O)NC(=O)C2C)=O)C1 CC(C(C)(C)C(=O)NCCCC(N)=O)NC(=O)CN1CC(=O)NC1=O C1(OC)CC(CNC(c2ccc(-c3ccc(C)o3)s2)=O)N(C(c2ccco2)=O)C1 c1(NC)ccc(C(=O)NC2CC(C)N(C(=O)COCCc3ccccc3)C2)nc1 CC(C)C(C(=O)NCC1(O)CN(C(=O)C(c2ccc(Cl)cc2)C)C1)C(C)C c1(C(=O)NC2CCN(C(C(CC)n3nccc3C)=O)C2)cc(C)c(N)cc1Cl C1(CNC(c2csnn2)=O)CC2(CCN(C(c3cn4ccnc4s3)=O)C2)CO1 c1(CN(C(C2CC(=C)CN2C(C2CCCOC2)=O)=O)CC)cccc2nc[nH]c12 N1(C(C(CSC)O)=O)CCC2CCN(C(c3sc(CO)nc3C)=O)C2C1 c1(C(=O)NCCC(CC)(CC)NC(c2ccco2)=O)ccc(=O)n2c1COCC2 c1(C(=O)NC)ccc(C(=O)NC2(CF)CN(C(=O)Cc3cncs3)C2)cn1 Cc1cc(=NCC2CC2C2CCCC2)[nH]c(=NCC2(CF)CC(F)(F)C2)[nH]1 C1(OC)CCCCC1NC(C1CC(CNC(=O)C(C2CCC(=O)N2)C)C1)=O N1(C(C2CCSCC2)=O)CCC2C(CCN2C(c2cnc3[nH]ccc3n2)=O)C1 C(=O)(C(CC(F)F)N(C(=O)CCC1CCCO1)C)NC1C(OCC)CC1 N1(C(CC2N(C(C(C(C)C)CN(C)C)=O)CC(O)C2)=O)CCCC2(CCCO2)C1 C(=O)(CCCCCNC(C)=O)NCC(C)N(C(C(CCC)C)=O)CC CCS(=O)(=O)CC(=O)N1CC(F)(C(=O)NCCOCCC(C)C)C1 c1(C(N(C(C)C(=O)NC(c2ccns2)C)CCC)=O)cn(C)nc1OCC C(=O)(C(=O)C(C)CC)N1CC(C(=O)OC(c2n(SCC)ncn2)C)C(OC)C1 Cn1ccn2cc(C(=O)NCC34CCC3CN(C(=O)C#CC3CC3)C4)nc2c1=O O=C(C1=CCCS1)NCCc1ccc(CNC(=O)CC2CCC(O)C2)cc1 C(=O)(C(C)CCC(C)(C)C)NC(c1cn(CCC=C(CC)CC)nn1)(C)C C1(CNC(C=CCOCCOC)=O)CC(NC(C2CCCCC2)=O)C1(C)C c1(-c2cc[nH]c2)nc(-c2cn(-c3ccccc3F)nn2)n(CCO)n1 C12(NC(c3cnc(CC)s3)=O)CCCC1N(C(=O)CCCn1cccn1)CC2 C=CC(C)(CC)C(=O)NCC(=O)NCC1(C#N)COC1 c1(OC)ccc(F)cc1C(=O)NC1(CNC(c2c(C)ccnc2O)=O)CCOC1 CN1CC2CCC(NC(=O)CCCNc3ccccc3[N+](=O)[O-])C2C1 C1(CC(=O)N(C(C)C)CCNC(C2CC(=O)NC(=O)C2)=O)CCCC(C)(C)CC1 C1(C)(CC)CC(NC(c2cn[nH]c2)=O)CN1C(=O)CCSc1ccc(F)cc1 C#CC1CCN(C(=O)COC2CCN(C(c3ccc(C)cc3)=O)C2)C1 C1(C(N(CC(C)NC(C2CS(=O)(=O)C2)=O)CC)=O)CCC(C(=O)OC)CC1 CN1CCN(C2(CNC(C3(O)CCSCC3)=O)CCC2)CC1 N1(Cc2cccc(OC(C)C)c2)CC2CN(C(c3ccc(I)c(Br)c3)=O)C2C1 c1(C(N2CC(C3CN(C(CC(C)O)=O)C3)C2)=O)cc2n(n1)CCCC2O C(CNC(=O)C(=O)N(CC(F)F)CC1CC1)(C(F)(F)F)N(C)C C(=O)(C1=CCCOCC1)N1CCC(NC(c2c(C)ncnc2)=O)C1(C)C S(=O)(=O)(c1ccc(Cl)cc1)N1CC(C(=O)NCCCOC=C)SCC1 C1(CN(C(CC)C)C)CC=CCC1 CCC(C(=O)NCC1(NC(c2c(F)cccc2F)=O)CC12CCC2)C(F)(F)F C1(NC(c2c(OC)ccnc2)=O)CCCN(C(=O)CC2CCCCC2(C)C)CC1 c1(OC)n[nH]c(C(=O)NCC(N2CCN(C(=O)C(=O)N(C)C)CC2)C(F)F)c1Cl c1(C(N(C)CC2CCCN2C(C2CCCCC2)=O)=O)ccc(F)c(O)c1 c1(C(c2nnnn2C2CCCC2)NC2(SCC)CCC2)ccc2nonc2c1 C1(NC(c2scnc2C(F)F)=O)CCCN(C(C2CC3(C2)CC3F)=O)C1 C(C(C(=O)N1CCOCC(CNC(C2CCCC(C)C2)=O)C1)C(F)(F)F)OC C1(NC(c2cc(CCCCC)no2)=O)CCCCCN(C(=O)COC2CC2)C1 C1(NC(=O)Cc2ccon2)CN(C(=O)CCC2CC2)CC2(CCOCC2)C1 CCCC(C)CCNC(=O)C(c1ccnn1C)NC(C1CC2(CC2)CO1)=O c1(C(=O)NCC2CC3(CC3)CN2C(c2cnns2)=O)cc(Cl)c2n[nH]cc2c1 CN=C(NC1CC1c1ccncc1F)N1CCN(CCC(=O)OC)CC1 C1(NC(Cc2nc(C)sc2Cl)=O)CCCC12CN(C(C1CCCOCC1)=O)C2 N1(C(c2cccc(F)n2)C(=O)NCCCCCC)CCC(C)C(F)(F)CC1 C1(CCNC(c2c(C)cco2)=O)C(C)CCCN1C(c1cc2n(n1)CCO2)=O N1(C(c2cccc(CC)c2)C(=O)NCc2ccccc2Cl)CCNC(=O)CC1C C(=O)(C1=NNC(=O)CC1)N1C(C)(C)C(CNC(=O)C=CC(F)(F)F)CC1 C(=O)(C1OCCc2c(O)cccc21)NC(C)(CO)C(F)F c1(NC(CCC2(C)N=N2)=O)cncc(C(=O)NCCC2CCCC3CC23)c1 c1(C(C)C)ccc(O)c(C(=O)NCCNC(=O)C2=NOC(C)C2)c1 c1(C(=O)OC)ccc2c(c1)OCO2.n12nc(cc1C)C(=O)N1C3CN(CC13)CC2 c1(N(CC(=C)Br)C)nc(N2CC(C(N)=O)C3(CC3)C2)c2c(n1)CCCCC2 C1(CC(=O)NC2(NC(=O)C(C3CCCOC3)=O)CC(CO)C2)CC2(CC2)CO1 N1(C(c2nn(CC)c(C)c2)=O)CCC2CC(NC(=O)C#CC3CC3)CCC2C1 C(CCCCCNC(=O)CN1CCCS1(=O)=O)N(C(=O)C1=COCC1)C C1(NC(=O)NCC(C)OC(F)F)CC2(CNC2)S(=O)(=O)C1 C=CC(C)C(C)C(=O)N(CCCNC(c1cc(OC)ccc1NC)=O)CCO c1(OC)csc(C(N2CC(O)(CCNC(C3CC(CF)C3)=O)C2)=O)c1OC Cc1ncc2n1CC(C(=O)NC1CCC(CCNC(=O)CCN(C)CCO)C1)CC2 C(=O)(C(O)CC(C)(C)C)NC(C1(O)CN(C(c2cccc(SC)c2)=O)C1)C C(=O)(C(C)(C)CSCC)NC(COC)C(=O)NN1CCCCC1=O c1(C(N(CC(CNC(C(C)C2CC2)=O)O)C)=O)ccc2c(c1)CN(C)C2 c1(C(=O)Nc2nc(C)c(C(=O)NCC3(F)CCC3)s2)cc(Br)ccc1Cl C(=O)(CCS(C)(=O)=O)N(CC(c1ccncc1)C)C1CC1.c12cccnc1C(=O)N2 c1(C(N2CC(O)CC(NC(CP(C)(C)=O)=O)C2)=O)ccnc2cc(Cl)ccc12 C(=O)(C(CCOC)NC(C1CC2(CCC2)C1)=O)NCC(CC)CO N1(C(c2ccc(CC)cc2)=O)CC2(CC2)CC1CC(=O)NCc1cc(C)ns1 c1(CN(C(=O)N(c2ccccc2)CC)CCc2nc[nH]n2)ccc2c(c1)COC2=O N1(C(CCSCC(C)C)=O)CCC(O)(CCNC(=O)C(C)(C)C(C)C)CC1 C(N=c1[nH]c2cccc(F)c2o1)C1CC(C)N(C(C2CC=CCO2)=O)C1 CC1(C(N2CCC(c3cn(CCCCF)nn3)C2)=O)CCCCCC1 C(=O)(C(CNC(C1CCCN1C(C)=O)=O)C(C)(C)C)N1CCN(C(C#C)C)CC1 CC1CCN(C(c2ncccc2N)=O)C1CNC(=O)C(C)(C)c1cnsc1 CCC(C(C)O)NC(=O)C(C)(C1CC1)N(C)C(C1CC(=C2CC2)C1)=O C#CCCCCCC(=O)N1CCC2(NC(=O)CC(C)(O)C3CC3)CCCC12 Cn1ccc2sc(C(=O)NC3CCC(Cn4cc(C5COCC5O)nn4)C3)cc12 c1(N(CC(=C)C)C)nc(=NC(CCO)C2CCC(F)(F)CC2)[nH]c2ccsc12 CCCC(C)(c1nnnn1CCC1CC1)NCc1csc(-c2ccncc2)n1 c1(CNC23CCC(C(=O)OC)(CC2)CC3)ccc2c(c1)Cc1ccccc1-2 C1(O)(C(=O)NCC(C)CNC(=O)COc2ccsn2)CCOCC1 CCCC(CNC(c1cn(CCO)nn1)=O)C(=O)N(C)CCN1CCCC1=O CC1CC(NC(C2(N(C)C)CC2)=O)CN1C(c1cccc(N2CCCC2)c1)=O N1(C(COCCOCC)=O)CCC(C(=O)NC2CCOC2C2CC2)C(O)C1 c1(SCCC)ccc(NC(C2(Oc3ccccn3)CCOC2C)=O)cc1 Cc1ccn2cc(C(=O)NC3CC4CCC3N4C(=O)CC34CCCC3C4)nc2c1 c1(COC)cc(C(=O)N(CCNC(=O)C=C(CC)CC)CCOCCO)cs1 C1(C(N2CCCN(c3ccccc3)CC2)=O)CCc2cnccc2N1 C1(NC(C(COC)(C)C)=O)CCC2(CC1)CC(NC(=O)CSC)C2 C1(c2nc(C(C)OCCOC)nn2-c2cccc(Cl)c2N)CN2CCN1CC2C CCC(C)(C)C(C(=O)N1CCC(NC(=O)C(C)(C)c2ccno2)CC1)OC c1(C(N2CC(C)N(C(C3CC4(CC4)CO3)=O)CCC2)=O)cc2cc(F)ccc2o1 C1(NC(c2cccc(OC(C)C)c2F)=O)C2CCC1CN(C(=O)C(C)O)C2 N1(C(c2cc(C(=O)OC)on2)=O)CCOC(CNC(=O)C(c2cncn2C)O)C1 N1(C(C(C)(C)OCC)=O)CC2C(C(=O)N(C)C(c3ccncc3)C)C2C1 c1(C(N2CC(C3CC3)C2)C(=O)NC2CCC2)cccc2nonc12 C(C)(CCC(C)(C)C)NC(C(CC#C)NC(=O)CC=C(C)C)=O c1(OCC)ccc(F)cc1CC(=O)NCCC1(NC(=O)C=CC(C)C)CCC1 c1(C(N2C3C(NC(C(CC)(CC)CO)=O)CC(C3)C2)=O)cnc2n1CCCCC2 C(C)(CCC#N)(c1n(C(C)C)nnn1)NC(C)Cc1ccco1 C1(C(=O)NCCC(C)NC(c2cc(SC)ncc2)=O)CC2CCC1CC2 C(=O)(CC(C)(C)CC(=O)N1CCCC(O)(CNC(=O)C(C)N2CCC2)C1)OCC Cc1[nH]nc2c1CCC(C(=O)NC1CCCCCN(C(c3ccc[nH]3)=O)C1)C2 C(=O)(C1CSc2ccccc21)N1CC(C(N)=O)(CNC(CCC=CCC=C)=O)C1 c1(OC)ccc(SCCC(=O)NC2CN(Cc3ncc(Cl)n3C)CC2O)cc1 c1(C(c2nnnn2C2CC2)NCC(C2CC2)OC)ccc(C)s1 C1(N(C(CN(CCC)C)=O)C)CCCN(C(=O)C(O)C(C)(C)C)CC1 c1(CC)cc(N(C)CCc2ccnn2C2CC2)n(C)n1 O=C(CC(Cl)Cl)NCCC1(C(=O)NC2CCC(CC3CC3)C2)CC1 C(=O)(CCS(=O)(=O)N(C)C)N(C)CC1CCN(C(c2cc(CC)n(C)n2)=O)C1 C1(CC)CN(C(C2CC(O)C2)=O)CC1NC(C1CC=CCC1)=O C1(CNC(CSCCC)=O)CN(C(=O)CCn2ccc(C)n2)C2(CCC2)C1 c1(CCC)onc(C)c1C(=O)NC1CCCC(NC(=O)CCCN2CCCCC2)C1 CCCCCC(C)(CC)C(=O)N=S1(=O)CCC2(CC1)CN(C(=O)C(C)C)CCO2 CC(C)C(C)CC(=O)N1CCC(OCC(=O)NC2CC3(CCC3)C2O)C1 C(=O)(C(C)N=c1cc[nH]cc1)NCC12C(CN(C(CCC=CC)=O)C1)C2 CC(C)CC(F)C(=O)N1CCCC(NC(=O)CCc2cccnc2F)C1C c1(C(=O)NC2CN(C(C(CCC)(C)C)=O)CC(O)C2)cccn2nnnc12 c12c[nH]nc1C(=O)N(OC)C2.C1(CC2CCOC2=O)CCCCC1 C1(C(=O)NCC2(NC(C3C(C(C)C)(CC)C3)=O)CCC2)C(=O)ON=C1C c1(C(=O)NC(C)Cn2cc(-c3cn[nH]c3)nn2)cc2c(nc1O)CCN(C)C2 N1(C(c2c(CCC)[nH]cc2)=O)CC2CCOCC2(NC(=O)C(=O)NCC)C1 c1(C(=O)NCCCN(C(C2C(C)(CC)C2)=O)CCO)cc(OCC2CC2)ccc1F C1(C(=O)NCC(C)(C)NC(=O)CC2CCCC(CC3CC3)O2)CCCCC1O C1(NC(=O)CC2C=CCCC2)(CO)CCN(C(=O)CSC2CCCC2)CC1 c1(C(=O)NCC(C)N(C(c2cc(OC)cc(F)c2)=O)C)cc2n(c(=O)c1)CCS2 O=C(C1=Cc2ccccc2C1O)NC1CC(CNC(C2(CO)CC2)=O)C1 N1(C(C2CCN(CC#C)CC2)=O)CC2CC1CC2NC(=O)COc1ccccc1 N1(C(CCC(=O)NCC)=O)CCCN(C(c2cc(Br)co2)=O)CC1CO C1(C(CC)C)CCN(C(=O)CNC2(c3nnc(C)o3)CC2)C1 C=C(C)CN=C(NCc1ncoc1C)N1CCN(C)C2(CCC2)C1 C#CCCCCCC(=O)N1CC2CCCC2(CNC(c2cnn(CC)c2C)=O)C1 N1(C(n2cc(Cl)c(C(F)(F)F)n2)CNCC(F)F)CC(C)OC(C)C1 CC1CC=C(C(=O)NC(CC(C)(C)C)C(=O)N(CCCn2ccnc2)C)CC1 C=C=CC(C)C(=O)N1CCCC(NC(=O)C(C)SCC)C1 N1(C(c2cnn3c2OCC3)=O)CC2OCCN(C(c3cc[nH]n3)=O)C2C1 N1(C(C)=O)CCc2cc(CC(=O)NC3CCCCN(CC(=O)N(C)C)C3)ccc21 C1(NC(c2c(C)nc[nH]2)=O)CCN(C(c2cc(Cl)nnc2Cl)=O)C(C)C1 C(=O)(CS(=O)C(F)(F)F)NC1CC(C)(NC(CC(c2ccc(F)c(F)c2)C)=O)C1 c1(C(N2CC(NC(Cc3c(C)cco3)=O)C(C)C2)=O)cc2ccccc2cc1N N1(C(C(=O)NCCOCCCC)=O)CC2CC1(NC(=O)C(C)SC)C2 Cc1cc(OCC(C)NC(N2CCC(C)C(N(C)C)C2)=O)ccc1Cl CS(=O)(=O)CC(F)(F)CC(=O)NC1CCC(NC(=O)CC(F)(F)Cl)C1 CC1(C)CCN(C(c2c[nH]nc2-c2cncs2)=O)CC1NC(C1CCCCC1)=O C1(CNC(C(C)OCCOCC)=O)CCN(C(=O)C=CC)CC1(F)F N1(C(COC(CNC(c2ncc(C)c(C)c2)=O)(C)C)=O)CC(C)N(C)C(C)C1 C(=O)(C(O)CCNC(C1CC(O)C(F)C1)=O)NC1C(OC)C(O)C1 CC1OC2(C)CC1(C(=O)NC1CCCC1CNC(c1ncoc1C1CC1)=O)C2 CCC(C)C(=O)C(=O)NCC(CC(N1CC2CCC=CC12)=O)C1CCC1 C12CCN(CC1O)C(=O)C(COC)NC2=O.N1(CC(=C)C)CCCC1 CCCCC(O)C(=O)NCCN(C1CCCCC1)C(=O)CCc1ncccc1C c1(C(=O)NC(CNC(C2CCCO2)=O)CO)ncnc2ccsc12 N1(C(CCCCOC)=O)C2COCC1CC(NC(=O)CC1CCCCN1C)C2 c1(NC(C(N2CCNC2=O)C)=O)ccccc1CNC(=O)C(C)(F)F C1(C)(C(=O)NCCCC(=O)NC2CCN(CC)CC2)CC2C=CC1C2 CCC(CC(=O)NCc1ncccc1C(=O)NC1CCCC(C)C1C)C1CCC1 C(CC(C)C)(C(=O)N(CCC(=O)NC)C1CC1)NC(C(C)NC(=O)NC)=O C1(C(N2CCCC2CNC(=O)OC(C)(C)C)C)CCCN(CC2=COCCO2)C1=O C(c1cccnc1)=C(C)C(=O)OCC1CCOC1C C(c1ccc(F)c2ccccc12)=CC(=O)NC1CC(S(=O)(=O)c2ccccc2)C1 CC(C(=O)NCC12COC(CNC(=O)CCCN(C)C)(C1)C2)C(C)(F)F CC1=NOC(C(=O)NC(C)CN(C)C(C2(C)CC(=O)C2)=O)C1 c1(C(=O)NCC(CNC(=O)CC2C=CCC2)O)conc1-c1ccccc1 C(=O)(CC(F)(F)C(F)(F)Br)NCC(C)N(C(=O)Cc1cocn1)C N1(c2c(C)cnc(C)n2)CC(CNC(C2(O)CCCCCC2)=O)OC(C)(C)C1 c1(C(=O)NCC2CC(NC(c3cc(OC)ns3)=O)C2)c(CO)noc1C c1(NC(C2CCN(C3CCN(Cc4scc(C)n4)C3)CC2)=O)c(F)cccc1F c1(C(C(=O)N(CCC)Cc2ccccc2)O)ccc(Cl)c(Br)c1 c1(CNC(CCC(=O)NC(c2ccccc2)C)=O)nc2cccnn2c1Br N1(C(C(CC)COC)=O)CCC(NC(=O)CC(C)c2ccccc2)C(F)(F)CC1 C(c1ccncn1)=CC(=O)NCC1CC(NC(C2(c3cccs3)CCCC2)=O)C1 c1(OCCCCNC(c2nc(C3CC3)cs2)=O)ccc(F)cc1 N1(C(C=CCC)=O)CCCC2CN(C(C3Cc4ccc(C)cc4C3)=O)CC12 c1(SC)cc(F)ccc1C(=O)NC1CN(C(c2cnccc2C)=O)CC1O C(=O)(C(C)CC(C)(C)C)N1C(CN(C(CCc2nc(C)c(C)o2)=O)C)CC(F)C1 c1(CC(=O)NC2C(NC(C=CC=CCC)=O)C2)cccc(COC)c1 c1(CC)c[nH]nc1C(N1CC=CC1C(=O)NCCNC(C1CCC1)=O)=O C1(CNC(c2cn(C3CCOC3)cn2)=O)CCCCCN1C(=O)Cc1cnns1 CC(C)(C(=O)O)C(C(F)(F)C(F)(F)F)NC(c1[nH]ccc1C1CC1)=O C1(CNC(CCOCC)=O)CC2CCC1N(C(c1ccc(=O)n(C)n1)=O)C2 N1(Cc2c(C)c[nH]n2)CC2CCN(C(c3cc(I)c(F)cc3F)=O)C2C1 c1(CC)ccc(NC(=O)CC2CCCN(C(=O)COC3(C)COC3)C2)cc1N c1(CN(C2CCN(C(=O)CCSc3cn[nH]c3)C2)CCC)ccccc1OC C1(NC(C(C)C(C)(F)F)=O)CC1C1CCN(C(=O)CC(F)(F)Cl)CC1 c1(C(=O)NCCCC2(CNC(=O)COc3cccnc3)CC2)cc(Cl)nnc1O N1(C(C(CN(CC)CC)F)=O)CCCC2(CCCN2C(=O)C#CC2CC2)C1 N1(C(c2c(C)[nH]c(C#N)c2)=O)CCC2CN(C(c3ccn(C(F)F)n3)=O)CC2C1 C1(CCOC)CN(C(=O)C=C2CCOCC2)CCN1C(=O)CC1(C(F)(F)F)CC1 N1(C(C=Cc2c(C)ccnc2)=O)CC2(CCN(C(=O)C(=O)NC(C)C)C2)C1 c1(COC)ncc(C(=O)NCC(C)Nc2cc(C(F)F)nc3ncnn23)c(O)n1 c1(C(=O)OC)[nH]c(=NC(C)C2CCN(C(c3ncc(OC)cn3)=O)CC2)sc1C c1(C(N2CCCN(C(C(CC)(C)F)=O)CC2)=O)cc(Cl)cc(C)c1N N1(C(CC(OCC)OCC)=O)CCCCC(NC(C2(C)CCCC2C)=O)C1 C1(NC(CNC(c2cccc(OC(C)(C)C)c2)=O)=O)C2CC3COC1C3C2 C1(C(=O)NC2C3CC2N(C(=O)COCC2CCOC2)C3)CC1C1CCOCC1 CC1COC(C)(C)CN1C(=O)C(Cc1ccco1)NC(=O)Cn1[nH]cnc1=N C(C(CC1CCCC1)C(=O)N1CCOC(CC)C1)NC(C(C=C)OC)=O N1(C(c2ncc(NCC3(C(=O)OCC)CC3)cc2C)=O)CCC2(CCC(OC)C2)C1 Cc1ccc2c(c1)CC(NC(c1cccc([Si](C)(C)C)c1)=O)N2C(=O)OC(C)(C)C C1(CCC#C)CCCN(C(C2CC2C(C)NC(=O)CCNC(=O)CO)=O)C1 C1(CC(=O)NC)CN(C(=O)Cn2cccn2)CCN1C(c1cocn1)=O N1(C(CC(C(=O)OC)C)=O)CCC2(CC1)CC2CNC(C1(OC)CCCCC1)=O C(=O)(C(O)CC(F)(F)F)N(CC(=O)Nc1ccc(F)c(CO)c1)C1CC1 N1(C(C2NC(=O)C(F)C2)=O)CC2CCCC(C1)N2C(=O)COc1cccc(Cl)c1 Cc1c(C(N2CCC(C(C)NC(C34CC(C3)C4)=O)C2)=O)cnn1CCO Cc1cc(O)nnc1C(=O)NC1CN(C(c2coc(Cl)c2)=O)CCC1C(F)(F)F c1(C(N2C(C(C)=O)CSC2)=O)ccc(Oc2ccc(C(F)(F)F)nc2)cc1C C1(C(=O)NCCCCC(C)NC(CC2(COC)CC2)=O)CCn2c(C)nnc2C1 N1(C(C(C)Cn2cccn2)=O)CCC(NC(c2cnn[nH]2)=O)CC1C C#CC1(C(=O)NCC2CCC(C(=O)NCCn3cncn3)O2)CCCCC1 N1(C(C(C)C2CCOC2)=O)CC2(CNC(c3ccn(C4CC4)n3)=O)CCC1CC2 C1(CC)CN(C(c2coc(CNC(c3cnc(OC)s3)=O)n2)=O)CC(=O)N1 N1(C(c2scc(C)n2)=O)CC(CNC(C2CC=CCO2)=O)OC2(CCC2)C1 c1(OC)c(C(N2CCC(NC(c3ccoc3)=O)C2C)=O)ccc(Cl)c1C C1(NC(C(C=C)O)=O)CCC(C)(CNC(c2cn(C)nc2Br)=O)C1 CON1CCC(CC(=O)NC2CC2NC(=O)C=Cc2ccccc2C)CC1 N1(C(c2ccc(OC)o2)=O)CCC(C)(C)C(NC(=O)CN2CCC(C)C2)C1 CCCCCC(O)C(=O)N1CCCC1CCNC(c1cnc(C)s1)=O C1(C(=O)NC2CN(C(c3cnc(CC)s3)=O)C(C)C2)COC2(CO)CC1C2 CCC(C)(CNC(C1CCCC1)=O)NC(C1C=CCCC1)=O c1(NCC2C(NC(C(C)C)=O)CC2)ccc(C(=O)NC(C)(C)C)s1 C1(C(=O)NC2(C(=O)NCC)CC2)CC(OC)CN1C(c1c(C)cnn1C)=O CC12CCC(CC(N3CCC(O)(CNC(=O)CC#N)CC3)=O)(CO1)C2 c1(C(N2CCC(C(=O)Nc3n(C)nnc3)C2)=O)ccnc(N2CCCCC2)c1 CC(O)(C(=O)N1CC2CC(NC(=O)CN3C(=O)CCC3=O)C1C2)C(F)(F)F c1(N(CCCN(C)C2CC2)C(c2ccccc2)=O)ccccc1N(C)C C=C=CCC(=O)NCCNC(C1CCC1c1ccccc1)=O.c12nc(no1)SC2 O=C1CCCC(CC(N2CC=CC(NC(=O)CCCc3ccccn3)C2)=O)C1 C1(C(N(C)Cc2ccc(C)cn2)=O)CCC(O)CN1C(C1CCCN1C(C)C)=O C(=O)(CCCCC(F)F)N1CC(CNC(CC2CC(C)(C)OC2)=O)C(C)(C)C1 C#Cc1ccc(C(N2CC(NC(=O)Cc3c(C)n[nH]c3C)C(C=C)C2)=O)cc1C CC(C)CCCCCC(=O)N(CCCCN(C)C(C1C=CCCC1)=O)C C(=O)(C#CC1CCCO1)N(C)CC1(OC)CC1.C(c1cccnc1)=C(C(=O)O)C CC(C(=O)NCc1nc(C(=O)Nc2cnn(CCF)c2)co1)C(C)(C)C C1(C)(NC(C(C)OCCOC)=O)CCN(C(C2CC2[N+](=O)[O-])=O)CC1 C(=O)(C(F)C(F)(F)F)NC1C(C)(CNC(=O)C=Cc2ccsc2)CCC1 CC1CCC(CO)CN1C(=O)COC1CC(NC(=O)C=Cc2ccco2)C1 C1(C(=O)NCc2nc(C)c(C)o2)(C(=O)OC(C)(C)C)CCC2CCCC12 N1(C(CCCOCC=C)=O)CCCC(C(C)NC(c2cccc(OC)n2)=O)C1 CCC(CNC(=O)C(C)C#N)(CC)NC(c1cc(C2(C)CC2)n[nH]1)=O N1(C(C(C)CC2CCC2)=O)CCC(O)(C(C)NC(=O)CCC2CCC(O)CC2)C1 c1(C(N2CC3C(NC(c4ccc(C(C)C)o4)=O)(C3)C2)=O)ccc2ccncc2c1 C1(CNC(=O)COC2CC(NC(=O)CC3CCC(O)C3)C2)CCCCNC1=O c1(OC)ccc(O)c(C)c1.C1(C(N2CC3(C2)C(=O)NC3)=O)(CO)CC(C)(C)C1 C1(NC(c2cc(CC)oc2C)=O)CCN(C(c2sc(OC)nc2C)=O)CC1F C=CCCCC(=O)NCC1CN(C(c2ccc(CC)cn2)=O)C2CC12 C1(C(C)C(N2CC(C3(C)CC3)C2)=O)CC2(C1)CN(C(c1cnccn1)=O)C2 C#CCCCCC(=O)NCc1cc(C(N2CC(=O)NC(CC)C2)=O)no1 C(=O)(C1=NNC(C(F)(F)F)C1)N1C(CCSCC(=O)NCC2CC2)CCC1 c1(C(N(CC(=O)N(CC(F)(F)F)C(C)C2CC2)CC)=O)ccccc1 C1(CNC(c2cc[nH]c2)=O)C2CCCC1N(C(C1CCN(C(C=CC)=O)CC1)=O)C2 C12(NC(C(C)=C3CC3)=O)CCC(CC1n1cc(COc3c(C)ccnc3Br)nn1)C2 N1(C(C(C(C)OC)NC(C2CCN(C)C2)=O)=O)CCC2(CNC(=O)N2)C1 n1(CC)nnc(C(N2CCC(C3CCCN3)C2)=O)c1C Cc1oc(CNC(c2cc(C3CC3)on2)=O)nc1C(=O)NC1CS(=O)(=O)C1 C#CC1CN(C(C2CCN(C(=O)Cn3cnnc3)CC2O)=O)CCN1C c1(C(=O)NC(CCN(C(CCN(CCCCC)C)=O)C)C)ncoc1C(F)(F)F N1(C(C2CCN(C(C(CC=C)OC)=O)C2)=O)CC2C=CCC(C2)C1 Cc1cc(C(=O)NC2CN(C(=O)CCn3c(C)csc3=O)CCC2C)nc(O)n1 c1(OC)cccc(N=c2[nH]ccc(C(=O)NC(C)CCCNC(=O)C(C)O)n2)c1 c1(C(N2CCN(C(C(C)C#N)=O)C(c3nccn3C)C2)=O)nc2ccccc2[nH]1 C(=O)(CC(C)CC(C)(C)C)N1C(C(=O)NC2CCC3(CCCC3)C2)CC(C)C1 c1(C(N(CCC)CCNC(=O)CCn2cccn2)=O)csc(C(C)(C)C)c1 C1(N(C(c2c(C)n(CCO)nc2)=O)C)CN(C(c2cc(Cl)ccn2)=O)CC1(C)C C1(C(=O)NCC2(CF)CC2)CC2CCC(C1)N2C(=O)CC1CCCOC1 c1(C(=O)NC2C(NC(c3cc([N+](=O)[O-])c[nH]3)=O)C2)ncc2ccccc2c1O C1(C(=O)NC2CC(C)(NC(=O)C(C3(O)CCCC3)F)C2)CN(S(N)(=O)=O)C1 Cc1ccc(C)c(-c2nc(-c3cc(CO)ccn3)nn2Cc2ccccc2F)c1 Cn1nc2c(c1C(N1CCN3CC(F)CC3C1)=O)CN(C(=O)C(N)=O)CC2 C1(=O)C(C(C)C)C(C)N1.c1(C(=O)NC(C(=O)N(CC)CC)C)ccnc(C)c1N C1(C(=O)NCc2ccc(O)cc2)CCN(C(c2scnc2Cl)=O)CC1O C1(C(N2CC(CNC(=O)C(F)(F)C3CCCC3)C3CC23)=O)C2(CC2)C12CC2 c1(NCc2onc(-c3ccc(NCC)nc3)n2)oc2c(OC)cccc2c1C N1(C(C(C)OC(C)(C)C)=O)CC(C(C)(C)O)(CNC(C2CCCCS2)=O)C1 c1(NC(CC2OCCN(S(CCCC)(=O)=O)C2)=O)cc([N+](=O)[O-])c(F)cc1C C(c1cc[nH]n1)=CC(=O)NCCN(CCOC)C(C1CC(n2cccn2)C1)=O c1(C(N(CC(C)CNC(=O)CC2COCC2(C)C)C)=O)cccc2c1CCN2 CC(F)(F)C(C)(C)C(=O)NC1CC(C2CC2)(NC(=O)CCC(F)(F)F)C1 c1(C(=O)NCCCC2N(C(C(CC)N(C)C)=O)CCC2)noc2c1CCCC2 c1(N2CC(NC(c3cccc(O)c3)=O)C(F)(F)C2)ncnc2cc(Br)sc12 N1(C(CN2CC(C)(OC)C2)=O)CC(CC(=O)NCc2sccc2C)C2(CC2)C1 N1(C(C=NOC)=O)CCC2(CC1)CC2CNC(=O)C=Cc1cccc(F)c1F N1(C(CC2C(C)=NNC2=O)=O)CCC2(CC2C(=O)NC(c2ccco2)CO)C1 C(C(=O)N=c1cccn[nH]1)N1CCN(S(C(C)C)(=O)=O)C2(C1)CC2 N1(C(C(n2ncc(C)c2)C)=O)CC(F)CC1CN(C(=O)C(O)C1CCC1)C C(=O)(C(O)CC(C)C)NC1CN(C(C2CCC(CC)O2)=O)CC1F c1(-c2cn(CC3CN(C(C4(C=C)CCOCC4)=O)C3)nn2)cc(Cl)cc(Cl)c1Cl c1(C(=O)NCC2N(CC(N)=O)CCOC2)ccc2c(c1)COC2 c1(C(=O)OC)ccc2c(c1)CCC2NC(=O)C(=O)NCCC1CC2CC1C2 C12(C(=O)NCc3nnc(C)o3)CCC(CC1)N(C(=O)CC(=O)N(C)C)C2 c1(C(N(C2CCN(CC(=O)N(CC(F)(F)F)C)C2)CC)=O)ccc(O)nc1Cl N1(C(c2cc(C)c(C(F)F)cn2)=O)CC2(CCCCN(C(C3CCCC3)=O)C2)C1 Cc1cccc(Cl)c1CNC1C=CCN(C(C2CCCCC2)=O)C1 c1(CNC(CC2CCC(C)C2)=O)nc2c(s1)CN(C(c1coc(Cl)c1)=O)CC2 N(C)(C(=NCCCSC)NCC12CCCC(C)(CO1)C2)CCCCOC C1(C(N2C(CNC(Cc3c(C)nn(C)c3)=O)COCC2)=O)CC2C=CC1C21CC1 C1(OC)CC(CNC(C2CCC(F)CC2)=O)N(C(c2n[nH]c(C)c2Cl)=O)C1 c1(SCC)cc(NC2CN(CC)CC(C)O2)c(OC)c(F)c1 N1(C(c2cc3c(s2)CCC3)C(=O)NC(CC)C)Cc2cccc(C(F)F)c2C1 N1(C(C(CC#C)(C)CC)=O)CCC2(CCCN(C(=O)Cc3cccs3)C2)C1 c1(C(=O)NCC2C(CNC(CCOCCCOC)=O)C2(F)F)c(C)n[nH]c1C c1(CCC(=O)OCC(=O)Nc2ccc(CC(N)O)s2)ccc(O)nn1 Cc1cc(C(F)(F)C(=O)N2CCC2CNC(=O)COCC(C)C)cnc1Cl C#Cc1ccc(CNC(=O)C(=O)NC2C3CC4C(C3)C24C(=O)O)cc1 c1(CC(C)NC(C2CC3CC3N2C(=O)CS(C)(=O)=O)=O)ccc(O)c(O)c1 N1(C(C2C(=C)C2)=O)CC2(NC(c3c[nH]ccc3=O)=O)CC1C2 C1(OC)CC(C(=O)O)CN(CCCC(=O)NC2CCCOC2)C1 N=c1ccn(CCCOCc2ccc(Cl)s2)[nH]1 N1(C(C2(c3ccc(Cl)nc3)CC2)=O)CCC2CN(C(C3CCC4CC34)=O)CCC12 C(=O)(C(F)C(C)CC(C)(C)C)NCC(CNC(c1c(OC)cnnc1)=O)CO c1(NCCCC(=O)OC)ccccc1OCC(O)CNCc1ccoc1 CC1(C)CC2(CC(C(=O)NCC34CCC3CCN4C(=O)C=Cc3ccco3)C2)C1 N1(C(C2CN3CCN2CC3)=O)CC2COCC2(C(=O)NCc2n[nH]cc2CO)C1 Nc1c(C(N2CCC(C(F)C(=O)NCC3(CF)CC3)C2)=O)cccc1F C1(C(=O)OC)CS(=O)(=O)CC(=O)N1.c1(N(CC)CC)nc(SCC)nc(=N)[nH]1 c1(C(=O)NC(C2CCN(C(C3CCC(SCC)CC3)=O)C2)C)cc(O)ccc1F Cc1nc(O)c(C(=O)NC2CCCCCN(C(C3C=CCC3)=O)C2)nc1C c1(CC)c(C(=O)NC2CCN(C(=O)C(O)CCSC)CC2)csc1C N1(C(CCC#C)=O)C(C=O)CCC12CC2.c1(N)cccc(SC)c1 Cc1nc(C(=O)NCC(C)(C)NC(=O)CC(C)C(F)F)ccc1C#N C1(CNC(C2(C(=O)NC)CCC2)=O)(NC(c2n[nH]c(=N)s2)=O)CCOCC1 C1(CC#C)CCN(C(C2(CN(CCO)CCN(C)C)CC2)=O)CC1 c1(OCCN(CC)CC)cccc(OCCN(Cc2ccccc2F)CC)c1 Cc1oc(S(=O)(=O)N(CCF)CC2CC2)cc1C(=O)NC1CC(NC(=O)CO)C1 C(C)(CCC(=O)NCC1CCC(C(=O)NC(c2n[nH]c(C)n2)CO)CC1)SC c1(CNC(c2cnc(OC)s2)=O)cc2n(n1)CCN(C(=O)CC1CCC(C)C1)C2 Cn1cc(C(=O)NC2COCC2CNC(C2(F)CC=CC2)=O)nn1 CC(C)C(F)(F)CC(=O)NC(C)CC1CN(C(=O)C(C)Oc2cccnc2)C1 C1(CC)N(N2CCC(S(N)(=O)=O)C2)CC12CCC2 c1(C(=O)NC(C)CN(C(=O)Cc2ccsn2)C)oc(Br)nc1C(F)F c1(C(=O)NC2(CC(=O)NCCC(CCC)O)CC2)cc(C#N)ccc1N c1(NCCC(C)C2CCCO2)nccnc1C#N Cc1ccc(C=CC(=O)NCCC2COCCN2C(c2csnc2C)=O)cc1Cl c1(C(C)C(=O)NC2CCC(NC(=O)Cc3cn[nH]c3)CC2)ccc(F)c(F)c1 C(=O)(C1COc2cc(C)c(C)cc21)NC1CC(CCNC(CC=C)=O)C1 Cc1cc(C(=O)NC2CCCCC2CO)cnc1F.N12CC(C(F)(F)C1)NC2=O c1(CCNC(N(C)CCC=C)=NCC2CCN(C)C2)c[nH]c2cc(F)c(F)cc12 N(C(=NCCC(C)(O)C1CC1)NCCF)CC1C(C)OCC1 C(=O)(CC(C)C(F)(F)F)N1CCC(NC(C(CCSC)O)=O)C(C(N)=O)C1 C1(C(N(C2CN(C(c3ncccc3Cl)=O)CC2(C)C)C)=O)CCCCCS1(=O)=O C=CC(C)(C)CC(=O)NCc1csc(C(=O)NCC(C)=C(C)C)c1 N1(C(c2cc(COC)[nH]n2)=O)CC2(CCCC(CNC(=O)C(C)(C)CSC)O2)C1 N1(C(c2sccc2OC(F)F)=O)CCC2(C1)CN(C(C1(F)CC=CCC1)=O)C2 N1(C(c2cc(OC)c(Br)cc2F)=O)CC2CCCCCCC12 Cn1ncc(C#N)c1C(N1CC2CC1C2C(=O)NC(CCO)C(F)F)=O c1(CN(CC(=O)NC(CSC)CC(=O)O)C)ccc2c(c1)CCC2 C1(C)(CC)C=C(C(=O)NCC2(O)CCN(C(=O)Cc3csc(C(C)C)n3)CC2)C1 C12(C(=O)NC3(C(N4CCC5CC45)=O)C(C)C3)CC(C#N)(C1)C2 N1(C(CCC=C)CN2CCC(=O)CC2)CCc2c(ccnc2N(C)CSC)C1 c1(OC)ncc(NC(c2cc(F)cc(F)c2)C)cc1Br N1(C(C2N(C(C)=O)CCC2)=O)CN(Cc2ccc(C)o2)CC1CO C1(CC)CN(C(c2ccc(Cl)o2)=O)CCN1C(c1ccc(C#N)s1)=O c1(C(N2C3CN(C(c4c(CC)nccn4)=O)CC32)=O)ccc(C)c(Cl)c1 C1(N(C(=O)COCc2ccccn2)C)CN(C(C2CC(=O)C2(C)C)=O)CC1(C)C N1(CCC=C)CCC2(CC1)CC(n1cc(C(O)CC)nn1)CCO2 c12ccc(s1)S(=O)(=O)NCC2.C(=O)(C(C#N)CN(C)C)OC(C)C C(=O)(C(C)(C)C(C)(C)C)N(C)CC1CCCN(C(C2(C)ON=C(C)C2)=O)C1 C#Cc1ccc(CC(=O)NCC2CN(C(=O)COCCCC(C)C)CC23CC3)cc1 c1(C(=O)NCC2C(NC(CC=C(C)C)=O)CC2)cc(Cl)c(Br)cn1 c1(CC)ccc(C(N2CC(OCCNC(=O)C(CC)OC)C2)=O)c(Cl)c1 C(=O)(CCC1=NNC(=O)CC1)NCC1C(C)CCN(C(C2(F)CC2)=O)C1 C(CC(=O)NC(C)(C)CC(C)(C)C)(C(F)(F)F)NC(C1C(=C)C1)=O CC(CC(C)(C)C)C(=O)N1CCN(C(c2coc(C(F)(F)F)c2)=O)CC1 c1(C(C)(C)C)ccc(C2CC2C(=O)NCC2CN(C(C3(C)CCCO3)=O)C2)cc1 c1(N2CCC(C)(F)C2)nc(=NCc2cc(Cl)cc(Cl)n2)[nH]c2c(F)cccc12 CCC(C)CCC(=O)N1CC(C(=O)NCc2cnn(CCF)c2)CCC1C CN1CC=C(C(=O)NC(C(=O)NCCN2CCC2)C2CC2)C1 C1(OC)CN(C(C2CN(C(=O)C(C)(F)c3ccon3)CC2C)=O)CC12CC2 N1(C(c2cn(C3CCCC3)nn2)C(=O)NCCCF)CCCCC12CC2 c1(Cn2c(C(c3cn(CCCO)nn3)OCC)nnn2)nc2ccccc2s1 C(=O)(C1CCCc2nc[nH]c21)N1CC2C(CNC(C=CCOC)=O)C2C1 c1(C(=O)NCC2(NC(=O)C(F)CC3CCCCC3)CC2)cnn2ncccc12 N1(C(=O)Cc2ccsn2)CC2CCCN(C(c3ncn4c3CCC4)=O)C2C1 N1(C(c2c(C)noc2C)=O)CCCC(CCNC(C2CC3C(C2)C3(F)F)=O)CC1 C(=O)(CS(=O)(=O)CCOC)NC(C(C(N1CCCC(CC)C1C)=O)(C)C)C C1(CC(N2C(CN(C)C)C=CC2)=O)CC2(C1)CN(C(C1CCCCC1(C)C)=O)C2 c1(C(C)C)nc(=NC(=O)OC(C)(C)C)n(C)[nH]1.C12COCC1CC(=O)N(CC)C2 N1(C(C2(CCCC)CC2)=O)CCC(C)(C)C(NC(=O)CCCCC(=O)NC)C1 Cc1cc2[nH]c(C(=O)N(CC(C)NC(=O)CC=Cc3cccc(F)c3)C)cc2o1 Cn1ccc(C(=O)NC2CCCC2(C)NC(C2CC2c2ccco2)=O)cc1=O C1(NC(CCS(=O)(=O)NC)=O)CN(C(=O)CC(C)P(C)(C)=O)C2(CCCCC2)C1 N1(C=O)CCOCC2(COCCN2C23CC4CCC(CC(C4)C2)C3)C1 c1(CC(=O)N(CC(CC)NC(=O)CCc2cc(OC)no2)C)csc(C)n1 c1(OC)ccc(Cl)c(C(c2nnnn2C2CC2)NC(C)CC2CCOCC2)c1Cl c1(-c2n(-c3cn(C)nc3)nc(C3CCCO3)n2)cc(-c2cc[nH]n2)nnc1O C1(Cn2cc(C3N(C)CCC3)nn2)CCCC2(CN(C(=O)CC3CCOC3)C2)O1 N1(C(c2c(CC)nco2)=O)CCCC(NC(=O)CC(C)(C)OC)C1C C1(C(=O)NCC(CC=C)NC(=O)C=CC)CC2CC(=O)C1O2 C12(C(=O)NCC(COC)(O)CO)CCCC1N(C(=O)C1=CCCC1)CC2 C1(CC)(NC(C2CC(C)(C)C2)=O)CCN(C(=O)CC2CCS(=O)(=O)C2)CC1 N1(C(CCC(=O)NCC)=O)CCC2CCCC12CNC(c1nccnc1SC)=O C1(CNC(=O)CC2CCCCO2)CC(O)CN1C(=O)C=CC(F)F C(C(CC(=O)N(C1(CCC)CC1)C)OC)NC(C1(CC)CCC1)=O c1(C(N2C(CNC(Cc3c(C)cccc3)=O)CCC2)=O)cc(C#N)ccn1 c1(C(N(C(C)CNC(=O)Cc2csc(Br)c2)C)=O)cc(C(F)F)ncn1 C1(C(=O)Nc2cccc(C(C)=O)c2)CCCCN(C(=O)C(O)C(C)(C)C)C1 C1(C(=O)NCC(CC)(C)NC(c2nc(O)c(C)s2)=O)COCC2(CCC2)O1 C(=O)(CCCCCCNC(=O)CNc1ccccc1Cl)NC1(C)CC(=C)C1 N1(C(c2c(CNC(c3ccc(O)cc3)=O)[nH]cc2)=O)CC2OCC(OC)C2C1 c1(CCCC(=O)NCC(CC=C)NC(=O)C(C)CC=C)ccc(Br)cc1 n1(CC)cc(C(=O)NC2(CCNC(=O)CCC3CCCN3C)CC2)c(C)n1 c1(OC)nc(C(F)(F)F)ccc1C.C1(CSC)CCC(C)O1 C(=O)(CCCC(=O)NC(C)CC(=O)N1CCC(CF)C1)OCC C(CC(C(=O)NCC1CCCCS1)NC(=O)CCc1cnn(C)c1C)OC c1(CNC(C(C(C)O)NC(C2CCCCC2)=O)=O)c(F)cc(Cl)cc1Br C(=O)(C1=C2CCCN=C2NN1)NC1C(NC(C=C(C)C)=O)CCOC1 c1(N2C(CNC(c3c(CC)nc[nH]3)=O)C(C)CC2)nc(C2CC2)nc2c1CCC2 C1(F)(CNC(CCSCC)=O)CCCN(C(c2cc(O)ccc2Cl)=O)C1 c1(C(=O)NC(C)(CNC(=O)Cc2cccc(O)c2)CO)coc2c1COC2 N1(C(CC=CCC)=O)CC(NC(c2coc(-c3cccnc3)n2)=O)C2(CC2)C1 c1(CC)ccc(F)c(C(=O)NCC(CNC(=O)CCC(C)C)S(C)(=O)=O)c1F c1(C(=O)NC2C(Cn3cc(-c4ncn(C)c4)nn3)CCC2)cc(F)c(Cl)cc1Cl C1(CNC(C2CCOCC2)=O)CC2(CCN(C(c3c(F)cccc3F)=O)C2)CO1 c1(C(=O)NC2(C3CN(C(C4(CCC)CC4)=O)C3)CC2)cc(F)cc2nn(C)cc12 O=S(=O)(c1cnc(NC2COCCC2O)c(Cl)c1)NCc1cc(F)ccc1F C1(NC(c2c(CC)nco2)=O)CCOCC1NC(=O)CC1(O)CCOC1 C(=O)(C1CCCn2cc(C)nc21)NCCCNC(CC(CC)CN(C)C)=O C12CCCCN1C(=O)CC2.c1(NC(C(C)C2(O)CCC2)=O)n[nH]cc1C1CC1 c1(C(=O)OCC)nnc(SC)nc1N1CC=CC1C(=O)N(CC)CC1(C)COC1 O=C1CC(C(=O)NCC#CCNC(C23CC2COC32CC2)=O)=NN1 N1(CCC)C(=O)CCC1C(=O)NC(C)CNC(c1oc(C(F)F)cc1C)=O c1(-c2onc(-c3ccc(N(C)C)nc3)n2)ccc2occc2n1 C(CC#CC(C)(C)C)NC(CCC(C)NC(=O)CC1CC(=O)NC1=O)=O C1(C(N2CC(C)(CSC)C2)=O)N(C(=O)C(C)C2CC2)CC12CCCC2 C1(NC(C(=Cc2ccco2)C)=O)C2CC(O)C1N(C(c1cnnc(O)c1)=O)C2 CC1CCC(O)(C(=O)NCC23CC(NC(c4csc(Cl)n4)=O)(C2)C3)CC1 C1(C(N(C2C(N(C(=O)C=CC=C(Cl)Cl)C)CCCC2)C)=O)CC2C=CC1C21CC1 CC(C)(C)CCC(=O)N1CCC(CC(=O)NC2(c3ccon3)CC2)C1 N1(C(C2CC(=C)C2)=O)CCC(N(C)C(c2sccc2C(=O)OCC)=O)CC1 c1(C(=O)NC2CCC(N(C(=O)CCc3ccccn3)C)C2)ccc([N+](=O)[O-])s1 C1(C)(C(=O)NCCCC2N(C(c3cc(OC)n(C)n3)=O)CCC2)CCCC1(F)F n1(C(C)C)cc(C(=O)NC2CN(C(=O)C(C)N(C)C)CC23CC3)c(O)nc1=O C#CCC(C)(C)CNC(=O)CC(C)(C)N(C)C(C1CCC1(OC)OC)=O CC1(C)C2CCC1(C(=O)NC1CCC1CNC(C1(c3ccccn3)CC1)=O)CC2 C1(CNC(c2nc(OCC)oc2)=O)CC(C)N(C(c2cnn(CC)n2)=O)C1 c1(C(N2CCC(CN(C)C(C34C=CC(CC3)C4)=O)C2)=O)cccc2nncn12 N#Cc1nccc(N2CCC(O)C2C(=O)NCCc2ccccc2)n1 c1(C(=O)NCC2(CN(C(C(C=C)O)=O)C)CC2)cc2c(=O)[nH]ccn2n1 CN1Cc2ccccc2CC1C(N1CC2CC2(C(N2CCOCC2CO)=O)C1)=O N1(C(c2c(C(C)C)occ2)=O)CC2CCN(C(c3cc4n(n3)CCOC4)=O)C2C1 [N-]=[N+]=NCC(F)CCNC(C1(CNC(=O)Cn2nccn2)CC1)=O C(=O)(CCCCC(F)(F)F)NCC12OCC(NC(c3nccc(C)n3)=O)C(C1)C2 C1(NC(C)=O)CN(C(c2ccc(Cl)o2)=O)C2(CCC2)C1.n12nnc(n1)C2 CC(C)CC(C(=O)NCC=CCl)ONC(C1CCC2CC1CO2)=O c1(C(C)C)nn(CC(=O)NCC2(CSC(C)C)CC2)c(=O)o1 C1(C(N2CCC(NC(C=CCC)=O)(CF)C2)=O)Cn2c(C)nnc2CN1C c1(CC)cc(F)ccc1C(=O)NC(CO)C(C)NC(=O)Cn1ccc(C(F)F)n1 C1(NC(C2CC(=C)C2)=O)CN(C(C2(C(=O)OC)CC2C(F)(F)F)=O)CC(C)(C)C1 C1(CNC(C2(CCOCC)CCC2)=O)CC(NC(=O)C(O)c2ccsc2)C(O)C1 N1(C(CCOC)=O)Cc2[nH]nc(C(=O)NCCN3CC(C)(O)C3)c2C1 N1(C(CC=CCC)=O)CCC(C)(CNC(C2C=CCS2)=O)C1 N1(C(c2c(CCC)nsc2N)=O)CC(C)C(N=c2ccc(C#N)c[nH]2)C(C)C1 N1(C(Cn2c(C)ccn2)=O)CCCC(CCNC(C2CC3CCC2C3)=O)C1 c1(C(=O)NC2C(CC)CN(C(=O)CN(C)C3CC3)CC2)c([N+](=O)[O-])cnn1C CP(C)(=O)c1cnc(C(=O)NCC2CCC2NC(C2COCCC2(F)F)=O)nc1 N1(C(CC(=O)NCC)=O)CCCC(N(C)C(c2ccc(C(N)=O)[nH]2)=O)C1 Nc1ccc(O)c(C(N2CCC(OCCNC(C3CCOC3)=O)C2)=O)c1 N1(C(=O)OC(C)(C)C)CC2CC(F)C1C2C(=O)NCc1ccco1 C1(C(N(C)CC2N(C(C=CC(CC)=CC)=O)CC(F)C2)=O)CC2CCC(C1)C2O C(C(O)CC(=O)NCC1=NOC(C)C1)NC(c1cn(CC=C)nn1)=O c1(OC)cc(C(=O)NC23CC(C(N4CC(C)SC(C)C4)=O)(C2)C3)c(Br)cn1 N1(C(C2CC2(C)Br)=O)CCC(CNC(C23CC(C2)C3)=O)C1 Cc1cc(CNC(=O)C(CCF)NC(c2cccnn2)=O)c(C)s1 n1(CC)nc(C(=O)NCc2cnn(C)c2C(=O)NOCC(C)(C)O)c(C)n1 N1(c2ncc(C)o2)CCC2(CC1)CCN(C(=O)CCOc1ccc(Cl)cc1)CC2 S(=O)(=O)(c1ccccc1)NCC(=O)NCCNC(C1OCC(C)(C)OC1)=O C(C(C)(C)CC(=O)NCCC1CCCC1(C)C)NC(C(CO)N(C)C)=O c1(C(N2CCC(c3ccon3)C2)C(=O)O)cccc(N=[N+]=[N-])c1.C(CC(=O)N)=C(C)C C(=O)(C(COC)CC(C)C)NCC(CC=C)NC(c1nscc1Br)=O N#Cc1cccc(NC(C2(NC(C3CC3c3cccs3)=O)CCCC2)=O)c1 C(C(F)(C(=O)N(c1ccsc1)C)C(C)C)NC(C(C1CC1)OC)=O C1(COCCC)CCCN(C(=O)CC2CCN(C(C3(CCCF)CC3)=O)C2)C1 C1(NC(C(C)N(CC)CC)=O)CC2CCC(C1C)N2C(=O)C(CC)CC(C)C N1(C(c2n(CC#C)ccc2)=O)CC2CC2(C(=O)NC(C)CCC2CC2)C1 CCCC(O)(CN(C(c1ccn(-c2ccccc2)n1)C(=O)NC1CC1)C)CCC C1(NC(c2ccc(F)nc2F)=O)CN(C(C2COCCO2)=O)CCC1(F)F c1(C(N2C(CNC(C(c3ccc(Cl)cc3)CC)=O)CCC2)=O)cccc(F)c1N C(N=c1[nH]c(Cl)ncc1Cl)C1CCC(C)C(NC(C2CC3CCC(C2)C3)=O)C1 c1(C(N2C(C(C)NC(c3c(C)nsc3C)=O)CCCC2)=O)ccc(N)c(F)c1 N(C(=NCCCCl)N1CCC(O)C(C)C1)CC(C(=O)NC)(C)C CC1CC(NC(=O)Cc2cc(F)ccc2F)CCN1C(=O)Cn1cccn1 c1(C(=O)NCC(C)(CNC(C2(C)CCCC2O)=O)OC)ccc(N(C)C)nc1 n1(CC(=O)NCC(CNC(C(C)(F)c2ccccc2)=O)F)nc(O)ccc1=O Cc1cc(C(=O)NCC(C)(C)CNC(C2(C)CC2(F)F)=O)cc(C)c1O c1(C(N2CC3CN(C(CN(CC)CC)=O)C3CC2)=O)cnc2c(c1)N(C)CCO2 N1(C(C2OCCN(C)C2)=O)CCC(NC(c2cnc(S)n2C)=O)C12CC2 C1(C(C)NC(c2cncn2C)=O)CN(C(c2cc(Cl)cs2)=O)CCO1 N1(CC(=O)NCCN(C(=O)CCSC)CC)C(=O)NC2(CCCC2)C1=O C(CS(=O)(=O)Cn1cc(-c2cc[nH]n2)nn1)NC(C1CCN(c2n(C)ccn2)C1)=O C1(CNC(=O)C2=CCC2)C2CCCC1N(C(c1cnc3ccoc3c1)=O)C2 C1(n2cc(CCCOC)nn2)CN(C(=O)CNC(=O)CC2CCOCC2)CC1C C=C=CCCN=c1nc(N(CCCO)C)c2c([nH]1)CCC2 C1(F)(C(=O)NCc2ccc(C(C)C)o2)CCN(CC2CC(F)(F)C2)C1 N1(c2nnc(CC)s2)CC2CC(NC(C3(CC)CCC3)=O)CC2C1 c1(C(=O)NCCC(C)NC(c2cc(OC)ns2)=O)ccc(C(O)CF)cc1 c1(CCC(=O)NC(C)CCCNC(=O)C(C)S(C)(=O)=O)ccc2c(c1)CCCO2 C1(CC(N2CC(C(C)NC(c3c(C)csc3)=O)C2)=O)CCCS1(=O)=O C(=O)(C(F)(F)C(C)(C)O)NC1CCN(C(Cc2ccc(C)cc2Cl)=O)CC1F CCC(CC(=O)NC1(C)CC(NC(=O)CCN2CCCCC2)C1)OC CC1(C)CCCC(CC(=O)NCC(C)(C2CC2)NC(=O)CCCCNC(N)=O)C1 c1(C(=O)NCCN(C(=O)COC(c2nccs2)=O)CC)cccc[n+]1[O-] CC(C)CS(=O)(=O)CC(=O)N1CCCC1CNC(C1(N2CCOC(C)C2)CC1)=O C(C)(CN=c1[nH]nc(C2CC2)o1)NC(c1c(C)oc(C2CC2)n1)=O c1(NCc2c(CC)nn(C)c2)nc(N2CC3CC2C3CO)nc2sccc12 c1(N(C)C)nc(C(=O)NC2CC(CNC(=O)CCc3ccccc3)C2)[nH]c(=N)n1 CC1CN(C(=O)CCC2CCOC2)CCCN1C(c1ccc2nn[nH]c2c1)=O c1(C(N(CC(=O)NC2CCC3(CC3)C2)CCC)=O)cc(CO)c(C)o1 N1(C(C(CCCC)CC)=O)CCC2OCCN(C(=O)CSc3cn[nH]c3)C2C1 Cc1cscc1C(=O)NC(Cc1ccco1)C(=O)N(C)CC1(O)CCOC1 c1(C(N(CC(=O)NC(C(O)CO)C2CC2)C(C)C)=O)c[nH]c(C#N)c1 c1(C(=O)NCC2(C(C)NC(C3CC3Cl)=O)CC2)ccn(CCF)n1 c1(OC)ncnc(C(N2CC3CC(CNC(c4cc(CO)on4)=O)C3C2)=O)c1F C1(CNC(C2(CC(C)C)CCCC2)=O)COCCN(C(c2cc(C#N)no2)=O)C1 c1(C(=O)NC(C2OCCN(C(c3ccc(C)nn3)=O)C2)C)cnc(C)cc1C c1(C(=O)NC2C(C)N(C(c3sccc3F)=O)CCC2)nn(C)c2c(=O)[nH]cnc12 c1(CN(c2nccc(C(=O)OC)n2)C2CC3CNCC23)c(F)ccc([N+](=O)[O-])c1F C(CC1CC1)(C(=O)NCCC1CC(F)C1)NC(C(C1CCOCC1)C)=O C(=O)(C(C)(CNC(=O)C(C)CCC)CC)NC(C(CC)CC)C C(=O)(CC1OCCc2sccc21)NC1C(C)N(C(=O)C=CC(C)(C)C)CCC1 C=C1CCN(C(C2CCC(C)(C)CC2)=O)C(C(=O)NC(C2CCCCC2)C)C1 c1(CCNC(CC)=O)ocnc1CNC(=O)C(c1cnn(C)c1)NC(C)=O C1(C(N(Cc2n(C)c(O)nc2)C(C23CCN(CC2)C3)=O)=O)CC12CC(F)(F)C2 C1(CNC(=O)CNc2ccccn2)CN(C(=O)Cn2cc(F)ccc2=O)CC12CC2 CC1CC(C)N(C(c2cc(Cl)c([N+](=O)[O-])[nH]2)=O)CCN1C(=O)C1=CCCCCC1 C(=O)(C(C)CN1CCCC1)NCC(C)CNC(=O)CSCc1ncccn1 c1(CCC)cc(C(=O)NCCN(C(=O)CC(C)COC)CC2CCCC2)ccn1 CC1CN(C(c2cc(O)ncn2)=O)CC(C)N1C(=O)C(C)(C)Cc1cnn[nH]1 C(C(CNC(C1CCCC(C)(C)O1)=O)S(C)(=O)=O)NC(C1(CC)CCCCC1)=O C1(NC(CC2(C)CCOCC2)=O)CC2CCC1CN2C(c1ccnc(S)c1)=O c1(C(N)=O)ccc(C(=O)NC2(CNC(=O)C(O)C(F)F)CCCCC2)cn1 C(=O)(CC(C)C(F)F)N1CC(CCCCNC(COCC(=O)NC)=O)C1 N1(C(c2nc(C)oc2C)=O)CC2CC(NC(=O)Cc3ccco3)CC2C1 c1(SCCC)ccc(C(=O)NC2CN(C(c3ccc(CC)cc3)=O)CC2C)cc1 c1(C(C)C(=O)NC2C=CCN(C(=O)CCc3nncn3C)C2)ccc(F)c(Cl)c1 C(CCCC(C)(C)C(=O)NNC(=O)c1c[nH]nc1Br)NC(C(C=C)C)=O N1(C(c2n(CC)ccn2)=O)CCC2CCN(C(c3c(C)nn(C)c3C)=O)CC12 N1(C(CS(CC)=O)=O)CCC(C(=O)N(CC(O)COC)C)C1(C)C c1(C2(C(=O)NCC(CO)NC(C3(C)CC(C)C3)=O)CCC2)ncccc1F c1(C(=O)NCC(CC=C)NC(c2ccsc2-n2cnnn2)=O)cc2n(c1)CCC2 Cc1c(C(N2CC(F)(c3ccncc3)C2)=O)[nH]ccc1=O N1(C(c2ccc(C)o2)=O)CC(C)CN(C(=O)CCc2nc(C)no2)CC1C N1(C(=O)CC2CC2)CCOC2CCN(C(=O)C(c3ccc(Cl)cc3)(F)F)CC12 C1(NC(c2cc(CN(C)C)on2)=O)CCN(C(C2CCCN2N=O)=O)C12CC2 c1(COC)nc(=NC2CS(=O)(=O)CC2NC(c2c(Cl)ccc3c[nH]nc23)=O)s[nH]1 c1(C(=O)NC2CC3CC(C2)N(C(=O)C=CI)C3)ccc2ncc(=O)[nH]c2c1 c1(C(=O)NC(CC(C)NC(C2(O)CCCC2)=O)C)ccc2nc(O)cn2c1 C(=O)(C(C(C)C)c1ccccc1)NCC1CC(NC(C2(C)CC(=C)C2)=O)C1 C1(CC(=O)NCC2(C)CSC2)C(NC(c2cc(CC3CC3)on2)=O)C1(C)C CN1CCCCC1C(N1CCCC(n2cc(CNC(=O)C=C3CCC3)nn2)C1)=O C1(CC(=O)OC)CN2N3CCCC(CC3)C1C2.C1(CO)CC1 c1(C(N2CC3C(CNC(C(Cc4cc(C)on4)N)=O)(C3)C2)=O)ccc(Cl)c(F)c1 C1(NC(C(C)CN2CCOCC2)=O)CCCCN(C(C2(n3cccn3)CC2)=O)C1 N1(CCN2C(CCC(=O)NC(CCCCCC)=O)CCC2)C(=O)NC(C)(C)C1=O C(C(=O)N(CCC(=O)NC(C)C(C)NC(=O)OC)CCO)(C(C)C)OC c1(C(=O)NCc2cncc(C(=O)NCC(C(C)C)CO)c2)cnn(C)c1C#N C1(C(=O)NCCCCOC(C)C)CCN(C(=O)C(O)CC2CC2)C1 N1(C(CCSCCC)=O)CCC2(CC1)CC(NC(=O)C(C1SC(=N)NC1=O)C)C2 C1(CNC(C(=O)OCC)=O)CN(C(c2ncc(OC)cc2F)=O)CC(C)(C)O1 N1(CC)C(C)CN(C(C2CCN(C(C3CC(=O)CCO3)=O)CC2)=O)CC1C N1(C(c2sc(C)c(O)n2)=O)CCC2(CC1)CN(C(=O)Cc1ccoc1)CC2CO Cc1cccc(C(N2CCCC2CN(C(=O)Cc2ccc(F)c(Br)c2)C)=O)c1F C(CC(C(=O)NC(C)C(C1CC1)OC)NC(=O)Cc1ccoc1C)OCC c1(C(=O)NC(C(C)NC(CCc2cc(C)no2)=O)C)cc(C#N)ccc1F C(C(=O)NCC(C)(C(C)C)NC(=O)C1=CCCC1)(C(C)C)OCC N1(CC(=O)NCC2C(C(N(C(C)C(=O)N(C)C)CCC)=O)C2O)CC2CC2C1 c1(C(=O)NCC2CCCN(C(C3(C)CCCCO3)=O)C2)cc2ccccc2s1 C(=O)(C1SCCc2ccccc21)N1C(CNC(C(C)SC(C)C)=O)CC2(CC2)C1 C(=O)(N1CCCCCO1)C1OCCN(C(c2cncc(C#N)c2)=O)CC1 Cc1cncc(C(=O)NCC2(O)CCN(C(=O)C(N)=O)C2)c1C C(=O)(CCCC(C)=O)NC1CCCN(C(C(c2ccccc2)OC)=O)C1 C12(C(=O)NCC(C3CCN(C(c4cnc(C5CC5)s4)=O)CC3)F)CCCC1OCC2 C=C(C)C1OCCCC1C(=O)NCC1C=CCN1C(=O)CC1CN(C(C)=O)C1 C#Cc1ccc(C(=O)NC2(CC=C)CCN(C(c3coc(C(F)F)c3)=O)C2)nc1 N1(C(Cc2ccc(OC)cc2)=O)CCC(C)(C)C(NC(C2CN(C)C2)=O)C1 c1(C(=O)NC(C2CCOC2)CNC(CC2CC(=C)C2)=O)cc(C(=O)OC)n(C)c1 N1(C(C(CN(C)C)C(C)(C)C)=O)CCC2C(=O)OCC12C c1(OC)cccc(NC(C2CCN(Cc3cc(C4CC4)[nH]n3)CC2)=O)c1F C1(C(N2CCCCC(NC(=O)C(O)CC(F)(F)F)C2)=O)CC2(CCOCC2)CO1 N(C1CCCc2nc(C)[nH]c21)CC(=O)OC.C12CC(C(F)(F)F)(C1)N2 CN1CC(O)CC1C(=O)NCCCCCCN(C)C(C1CC2CCC2C1)=O C1(C)(NC(C(CC#C)C)=O)CCN(C(=O)Cc2cc(Cl)n(C)n2)CC1 C1(C(=O)NCC(C)NC(C(C(=O)OC)C)=O)CC(=O)N(OC)C1 CC1=C(C(=O)N2CC3CC2C3NC(c2coc(C)n2)=O)CCCO1 c1(C(N2CC3C(CNC(CCC4C(C)(C)C4)=O)(C3)C2)=O)cc(N)cc(O)c1 c1(C(N2CCC(CNC(C3(C)CCOCC3)=O)C2)=O)ccc2c(c1)CC(=O)N2 C(C)(CN=c1ccnc(N2CCn3c(nn(C)c3=O)C2)[nH]1)NC(=O)OC Cc1ccccc1C=CC(N1CCN(C(c2cncnc2C)=O)C(C)C1)=O C#CCC(CC(=O)NCCCO)NC(=O)CCCCC=C c12cc(cc(F)c1)O2.C1(CC)CCOCCN1C(=O)C(N1CCC(CCO)C1)=O C1(C)(CCNC(C(C2CCOCC2)OC)=O)CCN(C(c2cnc(C)o2)=O)CC1 c1(C(=O)NC(COCC)C(=O)NCC=CC(C)(C)C)cc(F)n(C)n1 c1(C(N(C)CC2CN(C(C3(SC)CCC3)=O)C2)=O)cc2nn[nH]c2cc1F C1(NC(c2ccc(CCC)[nH]2)=O)CCN(C(=O)CCCN2CCCCC2)CC1F c1(C)ccc(-c2csc(N)c2)cc1.N1(NCCCCCC)CCC(C(C)(F)F)CC1 C#CC1(C(=O)N(C(C)C(C)CC)C2CC2)CCN(C(=O)C=C(C)C(C)C)CC1 CC(C)(C(=O)NNC(=O)c1ccc(O)cc1Cl)C1CCCNC1 n1(CC=C)cc(C(N2CC(CO)(NC(c3conc3C)=O)C2)=O)nn1 C1(CCCNC(c2cn(Cc3ccccc3)nn2)=O)C=CS(=O)(=O)C1 C(C1Cc2ccccc21)Nc1ncc(C#C)cn1.c12cccc(c1)CNC2=O c1(NC(C2CN(C(c3ncc(C)s3)=O)CC(F)C2)=O)cccc2c1CCC2 c1(C(N2C3CN(Cc4ccc(CCBr)cc4)CC23)=O)cc(F)c(Br)c(F)c1 C1(CC)CN(C(c2cn(C)cn2)=O)CCN1C(c1[nH]cnc1-c1cccnc1)=O n1(CC(=O)NC2C(CNC(CN(CCCCCC)C)=O)CCC2)ccccc1=O C1(C)(C(=O)NCCN(C2CCCC2)C(c2ccc(SC)o2)=O)CC2CC2C1 Cc1ccc(F)cc1C(=O)NC1CC(NC(C2CCC3CC23)=O)CC1O c1(C(=O)NC2(CF)CCN(C(CCCCC)=O)C2)cnn2c(Cl)cccc12 C1(C)(C(=O)NC(c2nc(C(=O)NC3CN4CCC3CC4)co2)C)CCCN(C)C1 c1(OCC)ccc(O)c(CNC(c2ccc(C#N)cn2)c2ccccc2F)c1 N1(C(C(C)=C(C)C)=O)CCC2(C1)CN(C(C1CC3CCC1O3)=O)C2 C1(OC)CC2CC(C(N3CCN(CCCNC(C4(C)CCCC4)=O)CC3)=O)CC12 c1(C(N2C(C)C(NC(=O)CC3(N(C)C)CC3)CC2)=O)cnn2c1S(=O)(=O)NCC2 O=S(=O)(c1c[nH]nc1-c1ccccc1)N1CCC(NC2(C#N)CCCCC2)C1 N1(C(C2CCN(C(Cc3nc(C)on3)=O)CC2O)=O)Cc2cccc(O)c2C1 N1(C(C(C(C)C)O)=O)CC2CC1CN(C(c1ccn3c1CSCC3)=O)C2 C1(NC(c2n[nH]cc2Cl)=O)CC2(CCCCN2C(=O)C(C2CCOCC2)F)C1 Cc1ccc(F)c(OCC(=O)NC2(C)CCCN(C(=O)C(C#N)=CC3CC3)C2)c1 O=C(CCCC(F)(F)F)NCCC1CCN(C(=O)CCC2CCOC2)C1 c1(C(=O)NCCN(C(C2CC2(C(C)C)CN(C)C)=O)CC)c(F)ccc(N)c1F C(C)(CC(=O)N1CCC1Cc1cn(-c2ccc(Br)c(F)c2F)nn1)(C(F)(F)F)OC c1(C(N2CCN(C(CC(C=C)CC)=O)CC2C)=O)ccc2ccccc2c1F C(=O)(CS(N)(=O)=O)N(C(C)C)CCNC(=O)CCN(C)Cc1ccccc1 c1(OC)cccc(CN(C)CCNC(=O)OCc2ccc(C(=O)O)cn2)c1F C(C1C(C(=O)NCC2(NC(=O)C(C)NS(=O)(=O)CCCC)COC2)C1(C)C)=C(C)C Cc1ccn(CC(=O)NC2COCCN(c3nnc(C)s3)C2)c(=O)c1 c1(C(N(C)CC2C3CN(C(C(CC(C)C)OC)=O)CC32)=O)nc2ccccc2s1 CC1(C)C(CNC(=O)CN(c2ccncc2)C)CCN1C(=O)CC1COCCO1 Cc1ccc(C(N2CCC(C(=O)N(CC(N3CCOCC3)=O)C)C2)=O)c(=O)n1C CC1CCn2cc(C(N3CCC(c4nnc5ccccn45)C3)=O)nc2C1 C(=O)(CCCCC(=O)c1ccccc1)NC1N(C(CSC)=O)CC(O)C1 CC(CS(C)(=O)=O)C(=O)N1CC2CCN(C(=O)C(C3CCCCCCC3)O)C2C1 N1(C(c2c(OC)scc2)=O)CC2CCCC2(NC(C23CC(C(F)F)(CO2)C3)=O)C1 c1(CNS(c2ccc(NC(c3ccc(N)nc3)=O)cc2)(=O)=O)ccc([N+](=O)[O-])cc1Br CC1CN(C(=O)C(c2ccc(F)cc2)=O)CC1NC(=O)CC1CCC(=O)N1 C1(CNC(C(CC)(C)CC)=O)CN(C(=O)CCCc2csc(C)n2)C2CCN1C2 CCC(C(=O)NCC1CC1NC(c1sccc1CN(C)C)=O)c1ccccc1 CC1(C)CCN(C(c2ccc(OC(F)(F)F)cn2)=O)CC1.C12CCCC1C(=O)N2 C1(F)(CNC(C2CC=CCC2)=O)CCC(CNC(C2CC(O)C2)=O)C1 C1(NC(CCCC#CC)=O)COC2CN(C(C3C=CCCC3)=O)CC12 CCC(O)C(F)(F)C(=O)NCC1CN(C(c2ncccc2Cl)=O)CC1(F)F C1(CC=C)(C(=O)NC(c2csnn2)C)CN(C(=O)CCC2CC2(C)C)C1 C1(CC(N2CC(C(N3CCC3C3CCCC3)=O)(SC)C2)=O)COCC(C)O1 N1(C(C(C)CC2CCCC2)=O)CCC(CN(C)C(C2(C)CC2C)=O)CC1 CC(C)CC(C)C(=O)N(CC(C)(C)CNC(=O)CC1CN(C(C)=O)C1)C C1(C)(CNC(C(n2cc(CO)nn2)C)=O)CCN(C(=O)C=C2CCOCC2)CC1 C1(C(=O)NC(C(C)C)C2CCC2)C2CCC(C2)C1C.C12CCN(CC1)C(=O)C2 CN=c1cc(C(=O)NCCCC(C)NC(=O)CCCc2nccs2)cc[nH]1 c1(C(N(C)CC2N(C(CCC(=C)C)=O)CCOC2)=O)cc(C)c2c(c1)CCC2 c1(C(=O)NCC(C(=O)O)N(C)C)c(C#N)ncn1C C1(C(=O)NCc2nc(C)c(C)o2)CN(C(C2CCCO2)=O)C2(CCC2)C1 CC1CCC=C1C(=O)NCC1(CNC(=O)COC2CC(F)(F)C2)CCC1 C(C(C(=O)N(C)CC1COCC1O)N(C)C)NC(CCNC(=O)NC)=O C1(C(=O)NCCCCNC(c2occ(C)c2)=O)CSC(c2ccccc2)=N1 C1(NC(=O)OC(C)(C)C)CCCOC1CC(=O)NC1(CC(N)=O)CCOC1 c1(C(N(CCNC(=O)C(C)OC)CC)=O)cc(COC(C)(C)C)n(C)n1 C1(CNC(CN(C=O)C2CC2)=O)CN(C(c2ncncc2F)=O)CC12CC2 c1(C(C(=O)NCC(F)F)N(CC(=O)OCC)C)cc2ccccc2o1 C(=O)(C(F)(F)C(F)(F)C(F)(F)F)NCC1OCCN(C(c2ccoc2)=O)C1 c1(C(c2nnnn2C2(C)CC2)NC(c2cccc(F)c2)(C)C)ncc(F)cc1F N1CC(O)(CO)C1.c1(C(C(=O)NC(C)(C)C)N2C(COC)CC2)cn(C2CC2)cn1 C1(NC(CN(C)C(C2CCC(C)(C)C2)=O)=O)CCN(S(C)(=O)=O)CC1 C1(c2c(OC)cccc2)CN(C(=O)C2=CCCC2)CCN1C(C1CC(C)C1)=O CCCCC(C(=O)NCCN1CCCC1=O)N1CCC(C)(CC)CC1 Cc1coc(C=CC(=O)NC2CCC(C)(CNC(=O)C(C)(C)CC3CC3)C2)n1 N1(C(c2c(C)nc(O)s2)=O)CCC2(CC2C(=O)Nc2ccc(O)c(CO)c2)C1 CC1CN(C(=O)Cc2cccs2)CCC1CNC(=O)COCCO C1(O)(CNC(CCNS(CC)(=O)=O)=O)CCN(C(=O)CC(C)SC)CC1 C1(NC(=O)CC2CC3CC3C2)CCC2CC1CN2C(C12CCCC1C2(F)F)=O c1(OC)cccc(CCC(C(=O)NCC(F)Cl)N(C(C)CS(C)(=O)=O)C)c1 N1(C(CCCCCC)=O)CCCCC1C1CCCN1c1cc(O)ncn1 N1(C(c2ccc(F)s2)=O)CCOC2CN(C(C3(F)CC3)=O)CC12 C=C(C)CCCC(=O)NOCC(=O)NCC1C=CCOC1 C1(COC)CN(C(c2coc(C(F)F)c2)=O)CCN1C(=O)CCS(N)(=O)=O c1(OC)ccc(-c2ccccc2C(=O)N(C)C)cc1C(F)F C(=O)(CCC(=O)NCC1CC(NC(=O)Cc2cc(Cl)n(C)n2)C(O)C1)NCCC c1(CCC(=O)N(C(C)C(=O)N(C)Cc2nc[nH]n2)CC)cn(C)cn1 N1(C(c2ccc(-n3cnnn3)cn2)C(=O)NC)CCCC(N(C)C)CC1 Cc1ccc(Cl)c(C(=O)NCC2CN(C(=O)C(C)OCC(C)C)CC2O)c1N N1(C(c2nc(C(N3CCNCC3)C)oc2)=O)CCC(N2CCNC(=O)C2)C(C)CC1 CC1OCCC1(F)C(N1CC=CC(NC(=O)C(O)CO)C1)=O C1(NC(CSCC#C)=O)CCCC(CC(=O)NCC2CNC(=O)C2)C1 c1(C(=O)NC2CC(C(C(=O)N(C3CCCCC3)CC)F)C2)nnc(O)nc1O C12(C(=O)NCC3(CNC(=O)Cc4cccnc4)CCCO3)CCC(F)(CO1)C2 c1(OC(C)C)cccc(C(=O)NCCC2CCN(C(=O)C(C)N(C)C)C2)c1Cl N1(C(C(C)C2CC2)=O)CCC(C2(O)CN(C(=O)CC(C(F)F)C(C)(C)C)C2)CC1 CC1(OCC(=O)NCC(C2CCC2)NC(C2CC2CF)=O)CCOCC1 CC(CC(=O)NOC(C)(C)C)NC(C1CCCCC(=O)N1)=O C1(C(=O)NCCCCC(C)NC(CCC(=C)C)=O)CN2CCCC2CO1 C1(CNC(CC(CN(C)C)O)=O)CC(C(=O)NCC(F)(F)C(N)=O)=NO1 C1(CNC(CN(CC)CC)=O)CC(F)(F)CN1C(c1cc(C(F)F)ccc1C)=O CCC(CC)(CCNC(C1CC=CCC1)=O)NC(C1(C)CCCN1C(C)=O)=O C1(NC(=O)CC2(NC(=O)CCn3ccnc3)CCC2)Cc2ccccc2C1 N1(C(COC)=O)CCCC(C2CCN(C(C3(c4cccs4)CC3)=O)C2)C1 Cc1cccc(C#CCNc2cc(I)n(C)n2)c1 CCN=c1[nH]c(C(=O)NC2CN(C(=O)CC=C(Cl)Cl)C(C)(C)C2)cs1 c1(CC)noc(COCC(=O)NCCC(C)NC(C2(Cl)CC2(C)C)=O)n1 c1(CC)nc(C)c(CNC(C2CC(=O)NC(C3CCNCC3)C2)=O)c(C)n1 c1(NC(C(C)NC(=O)NC)=O)ccc(F)cc1F.C12(C)CN(C1)C2=O c1(CC(=O)N(C(C)CCNC(=O)C=CCN2CCOCC2)C)nocc1C1CC1 C1(C(N2CSCC2C(N2CCC23CCC3)=O)=O)(OC)CCCOC1 N1(C(C(C(C)C)SCC)=O)CC(CC(N2CC(N(CC(C)C)C)C2)=O)C2(CC2)C1 c1(OC)cc(C(=O)NC2CC(C)(NC(=O)C(C)NS(C)(=O)=O)C2)cnc1O CC1CCc2c(C(=O)NC3(C)CCC(NC(=O)Cc4ccoc4)CC3)csc2C1 c1(C(=O)NC2CN(C(=O)CNC(=O)C3CC3)CC2F)ccc(Br)c(Cl)c1F c1(C(N(c2nccc(C)n2)C2CCNC2)=O)ccc2c(c1)c(C)c(C)n2C1CC1 N1(C(c2nc(C3CC3)cs2)C(=O)NCC=C)CCC2(CC1)CC(CO)C2 C1(NC(c2c(CC(C)(C)O)cccc2)=O)CC2CC1N(C(C1(O)CC1)=O)C2 C=C(Cl)CC(C(=O)NCc1nnc(O)n1C)NC(=O)C(C)COCC c1(C(=O)NC2CCN(C(C(C)OCC#C)=O)CC2C)nc(O)c(C#N)cc1C c1(CNC(C(CC)OC)=O)cnn2c1CN(C(C1CN(c3nncs3)C1)=O)CC2 C1(CC2CCCC(C)N2Cc2ccsc2)Cc2cccnc2C1 c1(C(C(=O)NCC2CC2)N(C2CC2)CC)ccc(C(C)(C)C)cc1 N1(C(c2nc(CC)oc2)=O)CCCC12CCN(C(=O)C(F)C(C)C(F)(F)F)CC2 N1(S(CC)(=O)=O)CC2(CCC(NC(c3cc(Br)ccc3C)=O)CC2)C1 N1(Cc2cc(C)c(-c3cnn(C(C)C)c3)nn2)CCCCNC(=O)C(F)(F)C1 C1(C)(CNC(c2cc(COC)sc2)=O)CCCN1C(c1c[nH]nc1C)=O c1(CN(C(c2csnc2C)C(=O)NCC)C)cccnc1OC Cc1nn(CC(=O)NC2COCC2NC(C2CCC(C)(C)O2)=O)c(=O)n1C C1(C(=O)NC(CC)C(C)O)CC=CCN1C(C1CCCC1F)=O c1(OC)ccc(F)c(C(N2CCCN(C(c3cnn(C)c3)=O)CCC2)=O)c1N c1(C(=O)NC2C=CCN(C(C3CCN(C)C3=O)=O)C2)c[nH]c2nccc-2c1 C#CCCC(C(=O)NC(C)C=C)NC(C1(O)CCSCC1)=O CCCCC(CC)C(=O)NC1(CO)CCN(C(=O)Cc2nc[nH]n2)C1 c1(OC)cc(C(=O)NC2(CCCNC(c3csc(Cl)n3)=O)CC2)on1 N1(C(C(CC)N(C)CC)=O)CCN(C(c2cccc(C#N)c2)=O)CC1C1CCC1 c1(C(N2CC3C(NC(C(C)N4CCC4)=O)(C3)C2)=O)cc2c(Cl)nccc2o1 N1(C(C=Cc2n(C)cnc2)=O)CC2(CCCCN(C(c3cccnn3)=O)C2)C1 c1(CC(=O)NCc2cc(CC(=O)NCC(COC)O)no2)ccc(Br)cc1 Cc1c(C(=O)NCCCCNC(C2(C)CCC(C)(C)CC2)=O)nn2ccccc12 Cc1ccc(F)c(C(=O)NCC(CO)NC(=O)C(C)(C)CN2CCN(C)CC2)n1 C(=O)(C1=CS(=O)CCC1)NCC(C)N(C(CN1CCC(C)CC1)=O)C c1(CCN2CC(CC)OCC2)ccnc(OC(F)F)c1Br C(=O)(C(C)(C)CNC(c1nc(Br)sc1Br)=O)NCC N1(C(C2(C#C)CC2)=O)C2CCC1CC(C(N1CCCC(OCC)C1)=O)C2 CC1CC2CN(C(=O)CCS(C)(=O)=O)CC2N1C(c1cccc2ccncc12)=O C1(CC(=O)NCC2(C(=O)OC)CC2)CN(C(=O)Cn2nccn2)C(C)(C)C1 Cc1cc[nH]c1C(N1CCC(N(C)C(c2csc(CS(C)(=O)=O)n2)=O)C1)=O C=CC1COCCN1C(C1CC(F)CN1C(c1ncccc1N)=O)=O N1(C(CCSC)=O)CCC(NC(=O)CCCn2nc(C)nc2C)C(OC)C1 C1(C(N2CCC(NC(C3CC3(Cl)Cl)=O)C(O)C2)=O)C2CCCCCCC12 CCCCCCCCNC(=O)C(=O)NCC(F)CNC(=O)CN(C)C(C)=O Cc1c(Cc2nc(CSC3CC3)nn2C(C)C(C)C)noc1-c1ccccc1 c1(C(=O)NC(C=C)C)cc2ccc(-c3cc(C)cnc3OC(C)C)cc2o1 C1(NC(c2cnc(C)s2)=O)CC12CCN(C(c1c(F)cncc1F)=O)C2 C(=O)(C(CSC1CC1Cl)NC)NCCCOCC C(=O)(N=c1ccn(C)[nH]1)C1(O)CCN(C(c2c(C)nc[nH]2)=O)CC1 C1(CC(=O)NC2CC2CNC(c2cnc(C3CC3)o2)=O)CCCOC1 c1(CC)ncncc1C(=O)NC1CC2(C1)CC2C(=O)NCc1cc(C(N)=O)co1 N#Cc1cccc(C2(C(=O)NCC(O)CNC(=O)CCCC3(CO)CC3)CC2)c1 N1(C(CCC(C)NC(c2cc(=O)n(C)cn2)=O)=O)CC2CC1C(F)(F)C2 C1(C(=O)NCc2c(C)c[nH]n2)CC(O)CN1C(=O)C(C)C C(=O)(C(F)(F)C(N)=O)NCC1(NC(=O)Cc2ccc(SC3CC3)cc2)CCOC1 c1(C(N2CCCC(F)(CNC(C(CO)N(C)C)=O)C2)=O)cc2ncccc2s1 c1(C(=O)NC(CN(C(C(CC)SC)=O)C)(C)C)n[nH]c2c1COc1ccccc1-2 C1(C(=O)NCC2CCN2C(c2ccn3c2CCCC3)=O)CCc2ccccc2N1 C(C(=O)N1CCC(N(C(=O)CC2CCC2(C)C)C)CC1)(C(C)C)NC(=O)OC c1(C(=O)NC2(C)CC(NC(C=C(C)I)=O)C2)ccc(CO)nc1 c1(C(=O)NCC(C2CCOC2)NC(c2ccc(O)nc2)=O)ccc(O)nc1Cl C#CCC(C)(C)C(=O)N1CCCC1CNC(=O)Cc1cccc(CC)c1 C(C(C)(C)CC(=O)NCCCN(C)C(C)C)NC(C1C(COC)C1(C)C)=O c1(C(=O)NCC2C3N(C(c4c(OC)scc4)=O)C(CC3)C2)cc(N)c(O)c(F)c1 c1(CN2CC(F)(C(=O)NC3CC(C#N)C3)C2)nc(Br)ccc1F C1(O)(C(=O)NC2CN(C(CC3C(C)(C)CCO3)=O)C2)Cc2ccccc2C1 CC(C)C(C(=O)N1CC(NC(c2ccc(CSC(F)F)o2)=O)C1)c1cnn(C)c1 C1(C(=O)NC2CCCN(C(C3(C#N)CC(C)C3)=O)C2)CCC2(CCC2)CC1 c1(C(CC)NC(C2(CNC(=O)CC(=O)OC)CC2)=O)ccc2nccnc2n1 C(CCCCC(=O)NC1(CNC(C2(C)CCCC2C)=O)CCC1)=CC c1(NC(C(C)C)CNC(c2cc(C(C)(C)C)no2)=O)cc(=O)n2ccccc2n1 c1(SC)ccc(CCC(=O)NC2CC(C)(CNC(c3cccnc3)=O)C2)cc1 C(=O)(CCC(C(C)C)NC(C1C2CCC(F)C12)=O)N1CC(C#C)C(O)C1 C(=O)(C(F)C(C)CNC(=O)C(C)(C)c1ccno1)NCc1nc(C(C)C)on1 C(=O)(C1=CCCSC1)N1CCC(CCNC(C(C(C)C)SC)=O)C1 c1(CNC(=O)NC(C(CCC)(C)C)C)cccc2occc12 c1(C(=O)OCC)cc(Br)ccc1N(C)Cc1sc(C)cc1C c1(NC(=O)OCc2c(C)cccc2)cc(Cl)nc(-c2ccccc2)n1 C1(C(F)(F)F)(CNC)CC2CN(c3nnc(-c4ccc(C)nc4)n3C)CC2C1.C=O C(C(C)C(C)(C)C)N(C(C(CSCC)NC(c1cnsn1)=O)=O)C C1(C(=O)NC(CNC(CC(=O)OCC)=O)(C)C2CCC2)CCC2CC1C2(C)C N(C(=NCCCF)NCC1CCCCC1C)Cc1ccnc(OC)c1F c1(N(CCC)C(C2C=CCCC2)=O)cccc(-c2nc(Br)nn2C)c1 CC(CC(=O)NC1C2CC1N(C(c1ccc3c(c1)CC3)=O)C2)CC(C)(C)C c1(C(C(=O)NCCN(C(c2c(CC)csc2)=O)CCOC)C)cccc(Cl)c1 CC(C)(CC(F)(F)F)C(=O)NC1COCCC1NC(=O)CN1CCCOC1=O C(C)(CN=c1[nH]nco1)(C(C)C)NC(=O)Nc1cn(CCOC)nc1 N1(C(C2(CCC)CC2)=O)CCCC(CNC(=O)C(C(C)(C)C)C2CCCC2)CC1 c1(C(N2CC(C=C)OCC2)C(=O)NC2CCCC2)cccn2ccnc12 N1(C(=O)CSC2(O)CCC2)CCC(=C(F)F)CC1 O=C(CCCn1cc(-c2cccnc2)nn1)NCc1cscn1 C1(C(=O)NCCC2CC(NC(c3ncn(CC)c3)=O)C2)(CC)CC=CCC1 c1(OCC)ccc(NC(=O)CCOCC(F)F)cc1O.C12(COC)CN(C1)C2=O C1(NC(c2cc(OCC)no2)=O)CCCC(N(C(=O)CN(C2CCCC2)C)C)C1 N1(C(C=C(C)C(=O)O)=O)CC2CC(C1)N2C(=O)NCCc1ccc(C)cc1O N1(C(c2cnn(CCC)c2C)=O)CC2CCC(NC(C3(C(C)C)CC3)=O)CC2C1 C1(CC(=O)N(C(C=C)C)C)CN(C(c2ccc(CC#N)cc2)=O)CC1C C1(C(N2C(C(N3C(CO)CC(OC)C3)=O)CCC2)=O)C2CCCCC12 c1(NC(C2C(OC)CN(C(C3CN4CCC3CC4)=O)C2)=O)cc(C)cc(O)c1 c1(C(n2cc(C3COCCN3C(c3ccc(Cl)nc3)=O)nn2)C)ccccc1F c1(N2C(NCCN3CC(C)OC(C)C3)COCC2)ncc2nc(Cl)nc-2[nH]1 N1(C(C(C)C(=O)N2CCOCC2)=O)C2CCC1CN(C(C1(CF)CC1)=O)C2 N1(C(C(Cc2ccoc2)NC(C2CC(=C)C2)=O)=O)CCC2(CCOC2)C1 Cn1nc(C(N2CC(F)CC(F)C2)C(=O)NCCON)c(Br)c1Cl c1(CC(N2CCOCC2C(=O)NCCC2(C(F)(F)F)CC2)=O)ccc(Cl)cc1Cl c1(C(=O)Nc2n(C)ccc2)ccc2c(c1)CN(S(=O)(=O)C1CCOC1)CC2 Cc1nc(C(=O)NCCC(F)(F)Cn2cc(C3OCCO3)nn2)cc(O)n1 N1(C(C2(C)CCCOC2)=O)CCCN(C(c2c[nH]cc2Br)=O)CC1 c1(OC)cc(C(=O)NC2(CNC(c3ccnc(C)n3)=O)CC2)cnc1O c1(CCNC(CCN(C(=O)CC(=O)NC2CC2)CC#C)=O)ccccc1 Cc1cc(CCCNC(C2CCN(C(=O)Nc3ccccc3)CC2)=O)cc(C)c1 c1(C(=O)NC(CNC(C(C(C)(C)C)SC)=O)CCOC)cc(C)ccc1[N+](=O)[O-] c1(SCC(=O)NC(C)CC2CN(C(c3nc[nH]n3)=O)C2)ccccc1O N1(CCCC(C)C)CCOCC1=O.n12nnnc1C2COC.C(C)(C(=O)NC)N C1(NC(Cc2n(C)ccc2)=O)CCCN(Cc2ccc(Cl)cc2O)CC1 CCCCC(CNCc1cnc(-c2cccc(C#N)c2)s1)CC C1(C(C)NC(=O)C=CI)CCCCN1C(c1cccc(F)c1)=O C(=O)(CCCCC#N)N1CCC(C(=O)NOCCO)(CC)C1 c1(C(N(C)CC2CCN(C(c3c(C)nsc3N)=O)C2)=O)cc2cccc(Cl)c2o1 C(C)(CC(=O)NCCCCN(C)C(c1cn(C(C)(C)C)cn1)=O)SC C1(NC(C(C)Oc2cccc(C)c2)=O)CN(C(c2ncn(C)n2)=O)C(C)(C)C1 CC(C)C(F)C(=O)NC1CCC(CNC(c2ccccc2Br)=O)CC1 c1(C(=O)NCC(C)CN(C)C(C23CC(C)(CO2)C3)=O)cc(F)c(F)cc1O c1(C(N2CC(C(=O)NC(C3CCN(C)C3)CC)C2)=O)ccc(C)c(C)n1 C1(NC(=O)OC(C)(C)C)CC2(C1)CC2NCCCc1nnc(C2CC2)s1 C1(NC(C=C(CC)CC)=O)CN(C(=O)Cn2nnc(C)n2)CC12CCOCC2 c1(C(=O)NCC(C)(C)NC(COCc2onc(C)n2)=O)c2c(c[nH]c1=N)CCC2 C(=O)(C(C(C)(C)C)c1cc[nH]n1)NC1CN(C(C2(C)CCCS2)=O)C1 N1(C(C(CC)C#N)=O)CCCC(N(C(=O)C=Cc2cccs2)C)CC1 CN1CCCCC1C(N1CCC(O)(CNC(C2(C(F)(F)F)CC(F)(F)C2)=O)C1)=O C(=O)(CC1COc2ccccc21)C1CCCC(CC)C1.c1(OC)cc(C)c(OC)c(N)c1 c1(C(N2CC3C(NC(C4CC(c5ccccc5)C4)=O)(C3)C2)=O)ccc(F)c(F)c1 CC1COCC(CC(=O)N(CCc2ccccc2)CCO)O1.c12cccc(n1)NC2=O N1(C(C(C)c2cccs2)=O)CSCC1C(=O)NC1CCNC1=O C#CC1(C(=O)NCC2(C(=O)OC)CC2)CCN(C(C2CC3CC2CC3=O)=O)C1 C12(NC(C3COCCO3)=O)CC1CN(C(=O)Nc1ccccn1)C2 C(=O)(C(C(C)(C)C)NS(C)(=O)=O)N1CC(CCNC(c2c(C)cco2)=O)OCC1 N1(C(C2N(C)CCC2)=O)CC2CC1CCC2NC(C1COc2ccccc2O1)=O n1(CCC2(CCO)CN(C(COC(C)(C)C)=O)C2)ccccc1=O.c1(=O)c(=O)[nH]1 N1(C(C(C)CC(C)(C)C)=O)C2CCCC1CN(C(=O)C(N1CCCCCC1)C)C2 N1(C(C(OC)OC)=O)CCN(C(=O)C(c2cncn2C)O)CC1c1ccncc1 CCCC(C(=O)NC1CCN(C(=O)C(C(C)O)N(C)C)CC1)NC(N)=O C(=O)(C1=CCCCC1)N1CCCC(C(C)NC(c2nc(Cl)c(Cl)s2)=O)C1 Cc1ccc(N)c(C(=O)N(C(=O)C(c2cccnc2)C)CCCNCCO)c1F C(=O)(CCC(=O)NC1CCCCC1CC)NCCC.C12CN(CCO1)NC2=O C1(NCc2c(CC)cccc2)CN(C(C2CCS(=O)(=O)C2)=O)CCC1F C(=O)(C(=O)NNc1ncc(Br)cn1)NCc1c(C(=O)OC)ccs1 c1(C(N2CC3C(NC(c4ccnc(C5CC5)c4)=O)C3C2)=O)ccc(F)c(O)c1 C(=O)(C1=CCS(=O)(=O)C1)NCC(CNC(Cc1c(CC)cccc1)=O)O C1(C(=O)NCC2C(NC(c3ccc(CC)cn3)=O)CCC2)CCC(C#N)CC1 C1(CC(=O)NC(C)CNC(c2cn(C)[nH]c2=N)=O)CC2(CCOCC2)CO1 C1(C(=O)OC)N(C(C(=O)Nc2ccc(F)cc2C)C2CC2)CCSC1(C)C CC1CC(CC(=O)NC(C)CC(C)(C)C)CN1C(C1CC1c1ccco1)=O c1(C(N2CCN(C(C3CC3F)=O)C(CC(F)F)C2)=O)cn2ncccc2n1 C(CC(=O)N1CC(CNC(=O)C(C2CC2)SC)C1)NC(=O)OC N1(C(c2c(C)[nH]c(C(C)(C)C)c2)=O)CC2CCC1CN2C(C1CC1(C)Br)=O N#Cc1cc(NCC2CCCC23CCNCC3)c(Cl)cc1Cl c1(C(N(C(C)CCNC(C2(F)CCC2)=O)C)=O)ncn(-c2ccccc2)n1 CCC(C(O)C(C)C)NC(=O)CCCOc1ccc(NCC[Si](C)(C)C)cc1 c1(C(C(F)(F)F)OC(C2CC3CCC2C3)=O)ccccc1Cl C1(N(C(CCCC)=O)C)CN(C(c2cccc(N(C)C)n2)=O)CCC1O C1(=O)C2=CCN(C2)C(=O)C(CCN(C)C)N1.C(=O)(CCCN(C)C)OC c1(N2CCC(C)S(=O)CC2)ccc(S(=O)(=O)N2CCc3ccccc3C2)cc1Br C1(CNC(c2oc(C)c(Br)c2)=O)CCCCCN1C(C1CC1C(N)=O)=O N1(C(Cc2c(C)cco2)=O)CC2CCCC(C1)N2C(c1c(Cl)noc1C)=O N1(C(Cc2cc(C)c(Cl)cc2)=O)CC(CNC(=O)C2=NNC(=O)C2)C2(CCC2)C1 c1(C(=O)NC(CCCNC(c2c(OC)cccn2)=O)C)noc2c1CCCC2 C1(C(=O)NCc2ccc(S(C)(=O)=O)s2)(OC)CCCC(C)(C)C1 N1(C(COCCC=C)=O)CC2(CCN(C(=O)CC3CCCC(=O)N3)CC2)CC1C C1(CNC(c2nnc(C(C)(C)C)s2)=O)CC(NC(=O)CCC(F)(F)F)C12CCC2 C(c1cc(F)c(O)c(F)c1)=CC(=O)NCC1(NC(C(CCC)C)=O)CCOC1 N1(C(c2ccnc(C)c2N)=O)CC2CCC1CN2C(C1CC2(CCC2)CO1)=O N1(CC(=O)NCC(C)N(C(c2c(CC)n[nH]c2)=O)C)CCP(C)(=O)CC1 N1(C(C2(C)CCCNC2=O)=O)CC(NC(=O)CCC[N+](=O)[O-])C2(CCOCC2)C1 N1(C(CC=C(C)C)=O)CCCOC(CCNC(=O)CN2C(=O)CNC2=O)C1 CC(C1CC1)=C(F)C(=O)N(C1CCCC1)CCNC(=O)Cc1ccsc1 N1(C(CN(CCC)C(C2CCN(CC)C2)=O)=O)CC2(CCCN2C)C1 c1(CN(C(C(c2ccnn2C)NC(CSCC=C)=O)=O)C)ccn(C)n1 c1(OCC(=O)NC2CC(NC(=O)CC3CSCCS3)C2)ccc2cnccc2c1 c1(OC)ccc(C(N2CC(C(F)(F)F)CC23CCOCC3)=O)c2c1CCCC2 C(C(C)N(C(=O)CNC(=O)C=CCSC1CC1)C)OC(C)C n1(CC)nc(C)cc1C(N1CCN(CCCNC(=O)CC(F)F)CC1)=O CC12OCC(CNC(=O)CNc3ccc(F)c(Cl)c3)(CO1)CO2 c1(C(=O)NCC(C(C)(C)C)NC(CC2(COC)CC2)=O)ccc(Br)c(N)n1 N1(C(C(C(C)(C)C)OC)=O)C2CCC1CN(C(c1cnccc1Cl)=O)CCC2 C1(NC(=O)C(c2ccccc2)=O)CCC2(CCN(C(C3CC(F)(F)C3)=O)C2)C1 c1(C(N2CC3C(CNC(c4ncccc4CO)=O)C3C2)=O)cccc2[nH]ccc12 C1(F)(CNC(CN(C)CC)=O)CCC(NC(=O)CSc2cccc(C)c2)C1 Cc1cccc(CC(=O)NC(C)(CNC(C2C(C)C2C)=O)C(C)C)c1Cl C(c1ccc(C)cc1)=C(C(=O)N(CC(CC)NC(C=COCC)=O)CC)C C1(C(=O)NC2CN(C(CC3(C)CCCCC3)=O)C2)CN2CCCCC2CO1 N1(C(CC(CC)C)=O)CCC(CC(N)=O)(NC(C2CCCS(=O)(=O)N2)=O)CC1 N1(C(C2N(C(=O)CSc3nc[nH]n3)CCC2O)=O)CC2CC3CC2C1C3 c12ccc(cc1)C=CC(=O)N1CC(C1)OC(=O)N2.c1(OC)nccc(CC#N)n1 Cc1ccc2cc(NC(C3CCCCN(C)C3=O)=O)ccc2n1 c1(C(=O)NCC2CC(C)(C)N(C(=O)C3=NOCC3)C2)cc(F)cc([N+](=O)[O-])c1N C1(C(=O)NC(C(=O)NCCC2CCC(C)(C)C2)CC2CC2)CCCCC(=O)N1 N1(C(c2cc(C)[nH]n2)=O)CCCC(C2(NC(=O)C(C3CCC(=O)N3C)C)CC2)C1 CC(C)(CC(=O)NCC(C(F)(F)F)N1CCN(C(C2CSC2)=O)CC1)C1CC1 C1(C(C)(C)NC(C2C(C)C2)=O)CCN(C(C2(c3ccccc3)CC2(F)F)=O)CC1 c1(C(N2CCN(C)C(C(C)C)C2)C(=O)NCCCC)cccc(C)c1OC c1(-c2n(CC)c(N(C)CC3CN(C)C4(CCCC4)C3)nn2)ccc2c(n1)NCCC2 c1(C(C(=O)N(CCOC)Cc2c(C)noc2C)(C)C)ccccc1C(F)(F)F Cc1ccc(C=CC(N2CC(NC(=O)C3=CCC(C)CC3)C3CCCC23)=O)c(C)c1 C1(CCNC(c2nc(CSC(C)C(N)=O)sc2)=O)COCC1(C)C N1(C(c2c(C)c[nH]n2)=O)CCC(C)(C)CC1C(=O)NC1CCOC2(CCC2)C1 C1(NC(Cc2ccc(C)nc2)=O)CCCC12CCN(C(=O)CSCC(N)=O)CC2 c1(CNC(C2CC3CCC2O3)=O)ccc(C(=O)NC(C(CO)NC(C)=O)C)cc1 C1(C(N(C(C)CNC(c2nc(Cl)sc2Cl)=O)C)=O)CC12CCOCC2 C1(C(N2C(C3(NC(C(C)CF)=O)CC3)CCC2)=O)CCN(c2cccc(Cl)c2)C1=O Cc1ccn2ncc(C(=O)NC(C)CCNC(C3(NC(N)=O)CCCC3)=O)c2c1 C1(CC(=O)NCC2N(C(c3c[nH]c(=N)s3)=O)CCC2)(N(C)C)CCCCC1 C1(NC(c2scc(C)c2)=O)CCCCCC1C(=O)NCc1noc(C(N)=O)n1 c1(C(N2CCN(C(C3CCCC3)=O)C3CC23)=O)cc(F)cc2ccoc12 c1(C(=O)NCC(CC)NC(CNC(=O)OCC=C)=O)ccc(C(C)CC)nc1O n1(CC)c(C(N2CCC(CCNC(c3csc(COC)c3)=O)C2)=O)cnc1O Cc1ncnc(C)c1C(N1CCN(C(C2CCC3(CC3)C2)=O)CC1CF)=O N1(Cc2n(CC)ccc2)C(=O)CN(Cc2cc(Br)cnc2OC)C1=O c1(OC)nccc(I)c1C(N1CCNC(NCCN2CC(C)OC(C)C2)C1)=O C1(C(N2CC(OCCNC(c3ccn(CCC)n3)=O)C2)=O)C2CCCCCC12 c1(C(N2C3C(NC(C(C)OC)=O)C(C3)C2)=O)cc2cccnc2[nH]1 Cc1c(C(N2CC3CC2CN(C(=O)CCCC(F)F)C3)=O)oc2ccc(Cl)cc12 CN1CCc2cc(C(N3CC4CC4(CNC(=O)C(C)(C)C(F)F)C3)=O)ccc21 C1(C(=O)NCC2CCCC(NC(C3(CC)CCCCC3)=O)C2)COC(C)(C)CO1 C#Cc1ccc(C(=O)N(C2CCN(C(=O)C(C)=C3CCCC3)C2)C)c(F)c1 C1(CNC(c2cccc(OC)c2)=O)CC2CCCC2N1C(=O)CC(C)F C=C(C)CCC(=O)NCCCCC1CN(C(=O)CC(O)C2CCCC2)C1 N1(C(C2CCN(C(C)=O)CC2)=O)CCN(C(c2cnnn2C)=O)C(CCOC)C1 C1(CNC(C(C)ONC(C2C(=C)C2)=O)=O)CCCCC1C(=O)NOCCC(F)(F)F C1(C(=O)NCC(c2ccc(Cl)cc2)NC(C=C(CC)CC)=O)CCCC(CF)C1 C(=O)(C(C)(C)C1=CCN(C(=O)C(=O)Nc2ccc(S(C)(=O)=O)c(C)c2)CC1)OC n1(CCC(=O)NC2CCN(C(C(CC)OC)=O)C2)cc(Br)c(O)nc1=O C(CNC(C1(c2ccno2)CC1)=O)(CC(F)(F)F)NC(C(C)n1cncn1)=O C=CCCCCCC(=O)N1CCN(C(=O)CC(O)COC)CC1N(C)C C1(C(=O)OCC2(CC(F)F)CC2)CCCN(C(=O)Nc2ccco2)C1 N1(CCOC)CCOCC1CCC1CCC(OC(=O)NCc2ccccc2)C1 C1(n2cc(C(N3C(C)CC3)=O)nn2)CCCCCC1.O=C(O)CCC1CC1 c1(C(=O)NC2C3CN(C(CCS(C)=O)=O)C2C3)cncc2ccccc12 CCC(C)C(O)C(=O)NC1CC(F)(CNC(=O)C(F)(F)C=Cc2ccccc2)C1 CC1CCCCN(C(C2CCN2C(=O)C=CC2CCCC2)=O)C1 N1(C(C(C=CC)O)=O)CC(NC(C2CC2(F)F)=O)C(COC)C1 CCCC(CC)C(=O)NC12CC1CN(C(=O)Cc1cnsc1)C2 Cc1cc(F)ccc1C(=O)NCCCCNC(C1COCC1c1ccccc1)=O CCCC(CC)CC(=O)N1CC(OC)CC1CNC(c1ncoc1C)=O c1(C(=O)NCC(=O)N(CC(C)(O)C2CC2)C)cccc(F)c1 N1(C(C(C(C)C)F)=O)CCN(C(c2cc(C3CCC3)on2)=O)CC1C1CCCC1 Cc1ccn(C)c1C(=O)N(CCCNC(=O)C(C)CF)C c1(OC)ncccc1S(=O)(=O)Nc1cc(C)ccc1F.C12CCCCN1C2 C12(C(N(C(C(=O)NCC(Cl)Cl)C3CC3)C)=O)CCN(CC1)C2 N1(C(c2nc(-c3ccncc3)cs2)=O)CCc2c(F)ccc(Br)c2C1 C(=O)(C(C)C(=O)NCC1CCCC1)NC1(CC(=O)OC)CCCCC1 N1(C(C(C)NS(C)(=O)=O)=O)CCCC2(NC(=O)C=Cc3cccn3C)CC2C1 C12(C(=O)NCC(C)N(C(=O)Cc3ccccc3)C)CC(C1)C(C(F)(F)F)O2 N1(C(C=C(CC)C)=O)CCCC2(NC(c3cn(C)cn3)=O)CC2C1 C1(CC(=O)NCCC(C)NC(=O)C=C2CCC(C(C)(C)C)CC2)COCCN1C c1(OC)cc(C(N2CCC(NC(c3c(F)ccc(Cl)c3F)=O)C2)=O)cc(C#N)c1 CCC(F)(F)C(C)(C)C(=O)NCCC1CC(NC(c2ocnc2C(F)F)=O)C1 N1(C(=O)C=Cc2cccs2)CC2CC(NCc3ccncc3)CC(C2)C1 C1(C(N2CC(NC(C(C(C)(C)C)(C)O)=O)C2)=O)Cc2ccccc2CO1 CN1CCC(C(=O)NC2CC2CNC(=O)C=CC(=O)NC2CC2)C1 c1(C(N2CCOCC(NC(C3CCP(C)CC3)=O)C2)=O)cc2ncccc2[nH]1 c1(C(C(=O)NCCC(C)NC(=O)C(C)(C)CF)O)ccc(F)c(Cl)c1 c1(C(=O)NC2CC(C(N3CC(O)(C(C(N)=O)F)C3)=O)C2)cncc(O)c1 c1(C(=O)NC2CN(C(CCOCC=C)=O)C2)cncc(SC)c1 C(C1=NOC2OCCCC12)n1cc(SC2CC(C(N(OC)CCO)=O)C2)nn1 c1(SC(C2N(Cc3nc(C(=O)OC)c(C)s3)CCC2)=O)ccnc2ccccc12 Cc1cc(CCC(=O)NCC(c2ccccc2)OC(=N)O)cc(C)n1.C1C(=O)N1 C1(CC=C)(NC(C2(C(F)(F)F)CC2)=O)CCN(C(=O)CS(=O)CC)C1 Cc1nsc(C(=O)N(C(C(N2CCCC2CCN(C)C)=O)C2CC2)C)c1N c1(OC)cc(C(=O)NCC(C2CCCN2C(C2COCCO2)=O)(C)C)[nH]n1 c1(C(=O)NCC(CCOC)NC(C2(CC(C)C)CCCC2)=O)cnc(O)c(Cl)c1 c1(CNCC2CC3CN(C(C(CC)(CC)CO)=O)CC32)cc(=O)n2ccsc2n1 c1(C(=O)NCC(c2cccnc2)NC(CC=C=C)=O)cccc(CSC)c1 c1(C(C)C)ccc(O)c(C(N2CC3C(NC(C4CCCCO4)=O)C3C2)=O)c1 c1(C(C)(C)C(=O)NC2CCC(NC(C3CS(=O)(=O)C3)=O)C2)ccc2ccoc2c1 Fc1cc(CNCC2CC23CCOCC3)cc(Br)c1 c1(C(N2C(CN(C(=O)CC3CC4(CC4)C3)C)CCC2)=O)ccc2cnnn2c1 C(C)(C)(CN=c1nc(C(C)C)cc(C)[nH]1)N1CCCC(CC(=O)OC)C1 c1(C(=O)NC(c2ccc(SC)cc2)C)ccc2c(CN)c[nH]c2c1 Cc1cc(=NC(C)C2CC(NC(c3ncccc3C)=O)C2)[nH]c(C)n1 c1(OC)ccc(CC(=O)NCC2(C)CCC(NC(=O)C(C)OC)C2)cc1Cl C(=O)(CCNC(=O)N(C1COC1)C)NCC(=O)NC(C)C.c1ccsc1 C1(CC#C)(C(=O)N(C)CCN(C)CCO)CCN(C(=O)CN2CCC(C)C2)C1 C(=O)(C#Cc1cccs1)N1C(COC)CNCC1 n1(CC)cnc2c(NCCCC3CC3)nc(N(CCC(C)O)C)nc12 N1(C(C2N(C)CCC2)=O)CCN(C(CNC(c2cn(C)cn2)=O)C(F)(F)F)CC1 C(C(C)(C)C(=O)NC(c1nnc(C)o1)C)NC(C=C(C)C(C)C)=O CCC(C)C(C(=O)NCC1CC1CNC(=O)C(C1CCCCC1)F)OC C(=O)(C(O)CC(C)(C)C)N(CC(C)NC(c1n(C(C)C)nc(C2CC2)c1)=O)C CCCC(CNC(=O)OC(C)(C)C)C(=O)NCc1cc(SC)n[nH]1.C(C)(C)(C)O N1(C(CCc2onc(CCC)n2)=O)CC(O)CC1CNC(=O)Cc1cnoc1 CN1CCN(Cc2cc(O)no2)C(C(=O)N(c2ccccc2)Cc2cnn(C)c2)C1 c1(C(N2CCC(NC(COCCC#C)=O)CC2C)=O)ccc2ncc(=O)[nH]c2c1 C1(SC(CNC(CCSC)=O)(C2CCC2)C2CCC2)COCC1c1nc[nH]n1 c1(NC(=O)OC(C)(C)C)nc(Cl)c2ccnc-2[nH]1.C1(=O)CCO1.CN1CC1 C1(CNC(CCC(=O)NCCC)=O)CC12CCN(C(=O)C(O)CCSC)C2 N1(C(C(CNC(=O)CCc2ccsc2)N(C)C)=O)CCCC(C2CC2)CC1 Cc1cc2[nH]c(C(N3CCn4c(CCN)nnc4C3)=O)cc(=O)n2n1 C1(CC)C(CC(=O)NCCCN(C(C2(C)CCC2)=O)C2CC2)C1(F)F N1(C(C(CC#C)C2CC2)=O)CC(C(=O)N(C)C(c2ccccc2)C)C(F)(F)C1 N1(C(C(CC)NC(N)=O)=O)CC(C2(NC(c3nccc(OC)c3F)=O)CC2)C1 c1(C(N2CCN(C(CCNC(C)=O)=O)CC2CCO)=O)[nH]nc2ncccc12 Cc1c(C(N2CCC(C(C)NC(=O)Cc3cccc(O)c3)C2)=O)c(Cl)nn1C Cc1cc2c(N(C3CCNCC3(C)C)C(c3cncc(N(C)C)c3)=O)ncnc2[nH]1 C1(CN(C(=O)CSC(C)(C)C)C)CCCN(C(C2CC2c2cccc(Cl)c2)=O)C1 C1(NC(C(C)C)=O)COC2(CCCN(C(=O)Nc3cnc(CC(F)(F)F)s3)C2)C1 O=C(N=c1nc(Cl)[nH]s1)C1=NOC2CN(Cc3ccccc3)CC12 Cc1ccc(N)c(C(=O)NCC2(CNC(C3(C)CC3F)=O)CC2)c1F C1(C(N2C(CNC(Cc3nn(C)c(Cl)c3)=O)CCC2)=O)CCc2ccnn2C1 Cc1cn2cc(C(=O)NC(CNC(c3nocc3C)=O)C(C)(C)C)cc(F)c2n1 C12(CNC(=O)CCN3CCCCC3)CC1CN(C(=O)C(c1cccnc1)O)C2 C(CC1CCc2ccccc21)N1CC(C2CN(C(=O)COc3ccccc3)C2)C1 c12ccccc1NC2=O.N1(C(C)=O)CC(OCCNC(=O)CNC=O)C1 c1(OC)ncc(Br)c(=NC(=O)C2CC3CC3N2Cc2occc2C)[nH]1 C1(CNC(Cn2ncc(CC)c2)=O)C(C)CCCN1C(C1CC(F)(CO)C1)=O N1(C(C2C(OCC)CC2)=O)CCC(CNC(C2CC3(CC3)CN2C)=O)(OC)CC1 C1(CNC(CCc2n(C)ccc2)=O)C2CN(C(=O)CCCNC(=O)C3CC3)CC12 C(CCCCC(=O)NCC12CCC(F)(CC1)C2)N(C(=O)C(O)C1CC1)C Cc1cn2c(C(=O)NCC3CCCCN(C(C4C5CCCC45)=O)CC3)cnc2s1 c1(NC(C(C)S)=O)cncc(C2=CCC(C(F)(F)F)CC2)c1 C=C=CCCC(=O)N1CCC(N(C(=O)CSC(F)(F)F)C)C1 N1(C(c2c(CC)nccc2)=O)CC(NC(=O)C(C)(C)C2CCCO2)CCC(O)C1 Cc1nc(O)c(C(=O)NCC2CCCCN(C(C3(CF)CC3(F)F)=O)C2)nc1C N1(C(C(C2CC2)NC(C)=O)=O)CC2CC(NC(=O)C(C)C3CCCC3)C(C2)C1 N1(C(c2c(C)scc2)=O)C(CNC(=O)C=Cc2cnccn2)CC2COCC12 O=C(CC1CCc2ccccc21)Nc1cccc(NC(C2CC3CCCC3C2)=O)c1 c1(C(=O)NCC2CN(C(C)=O)C(C)C2)cnc2c(c1)N(C)CCO2 c1(C(=O)NC2C(C(=O)NCC(CC)(C)COC)OCC2)cc(C)ccc1F C1(CN)(NC(c2ccc(-c3ccccc3)[nH]2)=O)CCC1O Cc1ccccc1C(=O)NCC(C)NC(=O)COCCC(C)C CC1(NC(=O)NC2(F)CCN(Cc3ccccc3)C2)CCCNC1=O C(C(CC(C)C)C(=O)N(CC(C1CCC1)OC)C)NC(C(CC=C)(F)F)=O Cn1[nH]c(C(=O)NC2CN(C(=O)CCc3ccccc3O)C3CC23)nc1=O C1(N(C(c2ncn(C)n2)C(=O)NCCC#N)C)CC2CCC1O2 CCCCC(O)C(=O)NC1CCCC1N(C(=O)C(c1ccc(Cl)cc1)=O)CC C1(C(=O)Nc2ccccc2)CCC(NC(c2ccn(CC(F)F)n2)=O)C1 C(C(C)(C)CC(=O)NC1CC(F)(F)C1)NC(C1CCN(C)C1=O)=O C(=O)(CS(=O)(=O)C1CC1)N1CC(CC(C)NC(=O)COCCF)C1 N1(C(C(COC)C)=O)CCC(CO)(NC(=O)CNC(=O)CNC(C)=O)C1 CC1CCC(C(=O)NC2C3CC2N(C(=O)C(=O)Nc2ncc[nH]2)C3)CC1C C1(C(N(C(C)C(N2CCC23CCC3)=O)CC)=O)CCCC2(CC2)C1 N1(C(c2cn(C3CC3)nc2C)C(=O)NCCCC)CCCC(F)(F)CC1 CCCCC(CC)CC(=O)NCc1ccccc1CN(C(=O)CC1CC1(C)C)C C1(CNC(C(C)OCC)=O)CC2(CC2)CN1c1ccnc(C)n1 c1(C)cc([N+](=O)[O-])ccc1C.C(=O)(CC(Cc1ccc(F)cc1)NC(=O)N)OC C1(NC(c2c(C)con2)=O)CC2(C1)CN(C(C1(C)CCC(=O)NC1)=O)C2 C(=O)(C1=NOCC1)NC(C1(CNC(=O)CCCn2cccc2)CC1)C C1(NC(Cn2c(C(C)C)ncc2)=O)CCCN(C(C2CN(S(C)(=O)=O)C2)=O)C1C c1(C(=O)NC23CC(CNC(C)=O)(OC2)C3)c2ccccc2cc2ccccc12 C(=O)(C(CCc1cn(CCO)nn1)NC(N1CCCC(C(=O)OC)C1)=O)NC c1(C(C(=O)NC(CN(C(=O)C(CO)N(C)C)CC)C)(F)F)cc(Cl)ccc1Cl c1(-n2cc(C(CC(N)=O)NC(c3nc(CC)oc3)=O)nn2)ccc(Br)cc1 c1(SCC)c(C)noc1NC(c1nc(C(=O)OC)cs1)=O C(=O)(CCCCN1CCOCC1)NCCC1CN(C(CN(CCC)C)=O)C1 C1(C(=O)NC2C(CC)CN(C(=O)C=C(C)c3ccsc3)C2)CCOCC12CCC2 c1(CN(C(C2CCCSC2)C(=O)NC(CC)(C)C)C)cccc2[nH]ccc12 c1(CC(=O)NC2CCCN(C(C3CCC(=O)NC3)=O)C2)cc(F)ccc1Cl N1(C(c2c(C)nc(N(C)C)s2)=O)CC(C2(NC(=O)COC(C)(C)C)CC2)C1 c1(NC(C2CC(NC(c3ccc(C(C)N)cc3)=O)C2)=O)cnccc1[N+](=O)[O-] c1(-c2cn(C(C(=O)NC(c3nncs3)C)C)nn2)ccc(Cl)cc1Cl C(=O)(C(C)(C)C(F)(F)CC)N1CC(NC(CCC(CC)CN2CCCCC2=O)=O)C1 C1(NC(c2n(C)nc(C3CC3)c2)=O)CCC(C)(NC(=O)CC2CCCCO2)CC1 C1(c2nnnn2Cc2ccco2)(NC(C)CCC(F)(F)F)COC2(COC2)C1 C=CC1(CC(=O)NC2(C)CCCN(C(c3cc(C#N)no3)=O)C2)CCOCC1 Cn1c(=O)c([N+](=O)[O-])c(NCC(O)CNC(c2ccco2)=O)c2ccccc12 CCCC(C(=O)Nc1ccc(COCc2cn(C3CC(O)C3)nn2)cc1)C(=O)O N1(CCC(=O)NCC(CNC(=O)C(F)n2ccnc2)CO)CCCS1(=O)=O C=C(C)CCCC(=O)N(CC(C)NC(=O)C(N)Cc1ccccc1F)C C(C)(CCCNC(C1CCCN1C1CC1)=O)NC(C1(CCC)CC1)=O c1(C(=O)NCCCCCN(C)C(c2c[nH]cc(Cl)c2=O)=O)ccn2nnnc2c1 C1(CNC(Cn2c(C)ccn2)=O)CC(C(C)C)CCN1C(C1CC(N(C)C)C1)=O c1(N2CCC(C(=O)OCC(c3nc(C)sc3)=O)C2=O)ccc(F)c(Cl)c1 N1(C(c2n(C(C)C)ccn2)=O)CCOCCC1C(=O)NCC12CCC(C1)C(=O)N2 C1(NC(=O)NCC2CCCNC2=O)CCCN(C(c2ccccn2)=O)C1 C1(C(=O)NC2(SC)CCC2)CCCN(C(C)=O)CC1 Cc1cc(N(C)C)cc(C(N2CCC(C)C2c2cccc(F)c2)=O)c1 C1(OC)(CNC(c2ccnnc2O)=O)CCN(C(=O)C2CC2)C1 Cc1cc(C(=O)NC2CCC(C(=O)NCC3CC4C=CC3O4)C2)ncn1 N1(C(C=CCCC)=O)CC(NC(c2cc(-c3cnn(C)c3)[nH]n2)=O)C(C2CC2)C1 C1(C(N2CCC(N(C)C(c3ccnnc3O)=O)C2)=O)CC2(COC(=O)N2)C1 c1(NCC)ccc(C)cc1C(N1CCC(N(C(=O)CCCF)C)C1)=O c1(CCN(c2nnc(-c3ccc[nH]3)n2CC2CCCCO2)C)ccc(F)c(F)c1 c1(C(C(N2CCC(NC3CCCNC3)CC2)=O)=O)ccc(F)cn1 C(C(C(CC)CC)NCCO)NC(C1(NC)CCOC1)=O c1(CC2CC2)cnc(CSC)nc1.CC(CC(=O)Nc1cn(CCCC)nn1)n1ccnc1 C1(C(=O)NCCC(C)N(C(c2c(C)n(C)nc2)=O)C)CC2(CCCO2)C1 Cc1ccc(C)c(CNC(N2CCN(CCC(=O)O)CC2)=O)n1 c1(CC(N2CC3CCC(C2)N3C(C2C(F)(F)C23CC3)=O)=O)ccc2nn[nH]c2c1 N1(Cc2c(OC)c(SC)ccc2)Cc2cc(OC)c(OC)cc2C2(CC2)C1 N1(CC(=O)NC(C2CCOC2)CNC(c2nn[nH]c2Cl)=O)C(=O)CCC1=O C1(C(C)C(N2CCCC2(C)C2CCC2)=O)NC2CC1CC2O N1(C(c2ccc(N)c(N)c2)=O)CC2OCCN(C(C3CCCCC34CC4)=O)C2C1 C=C(C)C(C)(C)C(=O)N1CCCC(C)(NC(c2ccc(C(C)(F)F)cn2)=O)C1 Cc1cc([N+](=O)[O-])cc(C(=O)NCCC2(O)CCCN(C(=O)C(O)CF)C2)c1C C(c1cc(F)c(F)c(F)c1)=CC(=O)NCCCN(C(=O)CCCCN(C)C)CC c1(C(=O)NCCC(C)NC(C(CC)F)=O)cc(C(F)(F)F)ccc1F c1(C(N(CC(C(=O)N2CC(CC(=O)OCC)C2)(C)C)C)=O)ccc(F)cc1F C#Cc1cc(F)c(C(N2CC3CN(C(=O)C=C4CCCC4)CC3C2)=O)cc1F c1(C(=O)NC2C(CC)CN(C(c3nsnc3O)=O)CC2)cnc2c(Cl)cccn12 C1(C(=O)NC(C2CCCC2)CNC(C2(CCCC)CC2)=O)CC1(C)C C1(N(C)C)(C(=O)NCc2ccc(F)c(N)c2)Cc2ccccc2C1 c1(C(=O)NC2C(C(=O)NCc3cn(C)nc3)C2)cnc2ccc(F)cn12 c1(OC)ccn2c(C(=O)NCC3(c4ccc(Br)cc4)CC3)cnc2c1 C=CC(C)(C)C(=O)NC1C(C(=O)NOCCF)CC1(C)C C1(C(=O)N(CC2CSCCO2)CC2CC2)CC(NC(=O)OC(C)(C)C)C12CCC2 C1(C(N2C(C)(CNC(C3CCC(=O)N3)=O)CCC2)=O)CCC(=O)N(C2CC2)C1 CC1(C(=O)NC2CCC(NCc3ccccc3)C2)CC2(CC2)C1 C1(NCC(C(=O)N(C(C(=O)NCCC)C)C)O)(OC)CCOCC1 CC1CN(C(=O)CCN(C(C2(CO)CCCO2)=O)CC2CC2)CCN1CCO c1(-c2c(C)nc(CC)s2)cc(C(=O)NCCF)cc2[nH]ncc12 N1(C(c2c(C)ccnc2)=O)CCC(O)C(NC(=O)C(C)Oc2cccc(Br)c2)C1 C1(C(N(CC)CC)=O)CCC(CC2C(NC(=O)COCC(C)C)CCO2)CC1 Cc1cc(F)c(C(=O)NC(c2ccc(Cl)cc2)c2ccccn2)c(F)c1 C(N=c1[nH]cnc2ccc(Cl)cc12)c1cc(C(N2CCCCCC2)C)cc(F)c1 CCC(C)(C)C(=O)N1CCCC(N(C(=O)COCCF)Cc2cccc(C)c2)C1 CC1OC(C)C(C)C1C(=O)NCC1(F)CCN(C(C2CCC(=O)O2)=O)CC1 c1(OCC)ncccc1C(N1CC(NC(c2ncoc2C)=O)C(C(F)F)C1)=O C(CN=c1[nH]c(N(C2CC3(CC3)C2)C)nc2ccsc12)(CC(C)(C)C)OC C(=O)(CCCN(C)N=O)NC(CCC)CCCNC(c1ccc(C(C)F)cc1)=O C(CN=c1[nH]c(=N)[nH]c(=NCC(S(C)(=O)=O)C2CC2)[nH]1)c1c(SC)cccc1 CC1(C)CC(O)CN(c2nnc(CN3CCCS3(=O)=O)n2Cc2ccsc2)C1 N1(C(C2(OC)CC2)=O)CC2CN(C(=O)C(C3CCCC3)C3CCCC3)CC2(C)C1.OCF N1(C(C(C(C)NC(=O)CC(=O)NC2CC2)C)=O)CC2COC(=O)C2C1 N(C1CCc2cccc(F)c21)C(C(N1CCc2n(C)nc(Br)c2C1)=O)=O N1(C(C(CCOC)NC(C2(C#C)CCCC2)=O)=O)CC(C)(C)CCC1C Cn1nnc2cc(C(=O)NC3CN(C(C4COC(=O)C4)=O)CC34CC4)ccc12 Cc1cnc(C(N2CC(C(F)(F)F)CCC2C)C(=O)NC(C)C)cc1Br C1(CNC(c2ccc(CC)[nH]2)=O)CCCCN1C(c1n[nH]cc1F)=O c1(C(=O)NCC2COC(C3CC3)O2)cc(C2CCOCC2)on1 CN=c1[nH]cc(C(=O)NCCc2n[nH]cc2C(=O)NCC2(C)C=CCCC2)s1 n1(CC(=O)NCCC2N(C(C=CS(C)=O)=O)CCC2)cc([N+](=O)[O-])ccc1=O C1(CNC(C2CN(C(C)C)C2)=O)CCCC(NC(C2CC2c2cccnc2)=O)C1 CC(C)(C)CC(C)(C)CNC(=O)C(CCC1CC1)NC(C1CCCO1)=O c1(C(c2ccccc2)C(C)COC2CC2)nnnn1C1COC1 C(=O)(C1=C(C)S(=O)(=O)CC1)NCC1(OC)CN(C(c2cc(OC)c(F)c(F)c2)=O)C1 c1(C(=O)NCC2(NC(c3cc(CCO)on3)=O)CC2)csc(-c2ccccn2)n1 N1(C(Cc2ccc(OC)cc2)=O)CCC2C(NC(=O)C(C3CCOCC3)F)C2C1 N1(C(C=CCC)=O)CCC(NC(C2CCCS2)=O)C(F)C1 CCC(C)CC(C(=O)NCc1cccc(F)c1F)NC(=O)CCSC C(=O)(C1=CCCN(C(c2ccc(O)nc2C)=O)C1)NCCSCCCC Cc1c(C(N2CCC(N(C)C(C3CCCSC3)=O)C2)=O)oc2c(F)cccc12 C(C1=NOC2CCCC12)n1c(N2CC(COC)N(C)CC2)nnc1-c1cn[nH]c1 Cc1nccc(C(=O)N(CC(C)(C)C(=O)NC2COCC2N(C)C)C)n1 C1(C)(C(N2CC(C)(NC(COCCOCC#C)=O)C2)=O)COCCO1 N1(C(C2C(OC)C2)=O)CC(NC(c2csc(-c3ncccn3)n2)=O)CC12CCC2 C1(C(=O)NCc2nc(C(N3CC(c4ccon4)C3)=O)cs2)CCOCC12CCC2 c1(C(=O)NC2CN(C(C(CC)NC(C)=O)=O)CC2C)cnn2c1CCC2 C=C(C)CN=C(NCc1ccccc1)N1CCC2(CCCCCC2)C1 c1(C(CC2CC2)NC(=O)NC(CCF)C2CC2)ccc(Br)cc1 C1(C)(C(C(N2CCCC2Cn2cc(C3CCC3)nn2)=O)OC)CCOCC1 CC1CCC(CNC(=O)C=Cc2cnn(C)c2)N(C(=O)Cn2ncnn2)C1 CC12CC(C(N3CC4C(CNC(C5CC(F)C(=O)N5)=O)C4C3)=O)(C1)C(C)(C)O2 N1(C(CN(CC)CC)=O)CCCC(NC(C2CCCCCC2)=O)C1 c1(-c2c(C)nns2)nc(-c2ccncc2)nn1CC(C)(C)C N1(C(Cn2c(C)nnn2)=O)CCC(C)(CC(=O)NC(C)CC2(O)CCC2)C1 N1(C(C(=Cc2cn(C)nn2)C#N)=O)CC2CC(NC(C3CSCCS3)=O)C2C1 c1(C(N2CC(C)(C)C(NC(=O)CCNC(=O)CO)C2)=O)cnc2[nH]ccnc1-2 N1(C(C2C(C)OCC2)=O)CCCCC1C1CCCN(C(c2cccc(=O)o2)=O)C1 N1(C(=O)NCC2(CC3CCC3)CCCO2)CCN(C2CCC2)CC1 N(C(=NCCC(=O)Nc1ccccn1)N1CCC(CSC2CCCC2)C1)C(C=C)C C1(F)(CNC(C2CCC(C)(CC)O2)=O)CCN(C(=O)C(C)(C)CCF)CC1 c1(C(=O)NC2C(NC(C3C(C)=CCS3)=O)CC2)sc(C#N)cc1Cl N1(C(C(CCC)NC(C)=O)=O)CC2CCCC(C1)N2C(c1nn[nH]c1Cl)=O C(=O)(C(C)(C)CS(N)(=O)=O)N(CCC(C)NC(=O)CC1Cc2ccccc2O1)C C1(C(=O)NC23CC(N)(C2)C3)CCOC2(CCCC2)C1.C1(NC(C)=O)CCN(C)C1CC C#Cc1ccc(C(=O)NC(c2ccccc2)CNC(=O)C(C2CC2)OC)c(C)c1 N1(C(C(CC)C)=O)CCC(O)(C(=O)NCc2cn(C)nc2C)C1 C1(C(N2CCC(=CCC)C2)=O)CCCCCN1C(=O)CNC(=O)C1CC1 CC(C)C(C#N)C(=O)NC1(C)CCN(C(c2ccc(C(C)(F)F)nc2)=O)C1 N1(C(c2c(C)c(Cl)ccc2)=O)CC23CCCC2(C1)CN(C(C1CCC(=O)C1)=O)C3 N1(COC)CC(C(=O)NCC(C(C)(C)C)NC(=O)C=C(C)c2ccsc2)CC1=O c1(-c2nc(CSC)nn2C2CCCCCC2)c[nH]c(=NCCO)s1 N1(C(C2CCCN(C)C2)=O)CCC(C(=O)NC(C)(C)CCO)CC1(C)C C1(O)(CC(N2CCC(NC(C(C)Cn3ccnc3)=O)C2)=O)CCOCC1 C(=O)(C#CC1CCOC1)NCC1CC(n2cc(-c3cccc(N)n3)nn2)C1 Cc1[nH]c(=NCC2CN(C(c3cc4c(Cl)nccc4o3)=O)C2)ccc1[N+](=O)[O-] c1(C(=O)NC2(CF)CCN(C(C3C(=C)CC3)=O)C2)cc2c(C)cc(C)nc2s1 C12(CNC(C(C)OCCC#C)=O)CCC(CC1)N2C(=O)C(F)C(C)(C)O CSC1=C(C(=O)N2CCCC2(C)CNC(=O)C(C2CCOCC2)C)CCCC1 N1(C(C2(NC(C3C(C)OCCC3)=O)CC2)=O)CC2CSCC2C1 c1(C(N2CCC(NC(=O)CSC(F)F)(CF)C2)=O)c(Cl)ccc2ccncc12 c1(C(C)C(=O)N(C)CCN(C(=O)CCc2cnn(C)n2)C)ccc(F)cc1 c1(C(=O)NCC(C)(CNC(=O)CCC2CCC(C)O2)OC)cc(C)sc1C N#Cc1cc(C(N2CC3CC(C2)C3(F)F)=O)c(O)cc1N C1(C(N(CC(CNC(CCCOC(C)C)=O)C)C)=O)CC(F)(F)CO1 N1(C(C2N(C)CCOC2)=O)CCC2(CCCN(C(c3cc[n+]([O-])cc3)=O)C2)CC1 CC1Cc2cc(CC(=O)NCC3CC(NC(=O)C(F)(F)CO)C3)ccc2O1 N1(C(Cc2scc(C)c2)=O)CC(C(=O)NC2CC(C#N)C2)C2(CC2)C1 Cc1ccc2c(C(=O)NC3CN(C(C4COC(=O)O4)=O)CC(C)(C)C3)c[nH]c2c1 c1(C2(N(C(C(C3CN(C(=O)C4CC4)C3)OC)=O)CC)CCC2)ccc(C)c(Cl)c1 N1(C(=O)COC2CCCC2)CC(CNC(=O)C2=CCCC2)OC2(CCC2)C1 N1(C(c2cc(OCC)no2)=O)CCC(O)(C(C)NC(=O)C(CC)SC)CC1 c1(OC)ccc(Br)cc1C(N1CCC(NC(=O)CCSCC)C2CC12)=O c1(C(=O)NC2CC(NC(c3c(C)nc(CCC)o3)=O)C2)cncc2ncccc12 C(=O)(C(CC=CCl)c1ccccc1)NCC(CNC(=O)Cc1nonc1C)OC C(=O)(CCCC(C)NC(C1CCC2CC12)=O)NCC(C(C)C)(C)C N1(C(c2n(C=C)nnc2)=O)CCCCC2(CCN(C(c3nccnc3C)=O)C2)C1 Cc1cncc(CNC(C2CC(NC(=O)Cc3nccn3C)C2(C)C)=O)c1 C(=O)(C(C)(C)C(N)=O)N1CC(OC)C(C(N2CCC(C)(N(C)C)C2)=O)C1 c1(C(N2CCC(O)(CNC(c3cnc(O)nc3O)=O)C2)=O)c(F)ccc(F)c1Cl c1(C(N(CC(C)NC(c2cc(F)cc(F)c2)=O)CC)=O)cncc2n[nH]cc12 N1(C(c2cccc(C#N)n2)=O)CCN(C(=O)COCCF)C2(CCC2)C1 C1(CC)C(NC(=O)C(O)Cc2ccccc2)CCN1C(=O)CNc1ccccn1 C1(CNC(C2CC(=C)C2)=O)CC(F)(CNC(=O)C(=O)NCC(F)(F)F)C1 c1(C(N2C(CNC(C(=O)N(C)C)=O)CCCCC2)=O)ccc(S(N)(=O)=O)c(Cl)c1 C1(CC(=O)NCC(CC=C)NC(C2(C)CCCCO2)=O)CCC2(CCCC2)CC1 C(=O)(C(C)(C)CCNC(C1C2CCCC12)=O)N(C(c1cc(C)on1)C)C C(C)(N=c1[nH]c(Cl)nc2c1COCC2)C1CCN(C(C(C=C)(C)CC)=O)C1 c1(C(N(c2nccc(C#N)n2)C2CCC(N)C2)=O)c(F)cc(O)cc1Cl C1(NC(=O)Cn2cccn2)CCC2(CC1)CN(Cc1ccc(F)c(Cl)c1)C2 C1(CCN(C(C)(C)C)C)CC2(C1)CN(C(=O)CC1(C34CCC(CC3)C4)CC1)C2 CC1CCN(C(=O)CC2(c3c(SC4CC4)cccc3)CC2)CC1c1nccn1C Cc1c(S(=O)(=O)NC2CC(C)CCC2=O)sc2c(F)cccc12 Cc1ncnc(C)c1CC(=O)NCC#CCNC(c1ccc(N)c(Br)n1)=O c1(OC)cc(C)c(C(N2CCC(N(C)C(c3nccnc3OC)=O)C2)=O)cn1 C1(N(C)C)CN(C(=O)Cc2cccc(Cl)c2)CC1CNC(C1CCC(O)CC1)=O C1(C(N(CCCC)CC(=O)N(CC(F)(F)CC)C)=O)CC2CC1CC2O N1(C(C(C)NS(CCCC)(=O)=O)=O)CCN(C(c2cnsn2)=O)CC(C)(F)C1 N1(C(CC2C(C)(C)C(O)C2)=O)CC(CNC(c2cnco2)=O)OC2(CCC2)C1 N1(C(Cc2cnc(C)s2)=O)CCC(CO)C(NC(c2sc(CO)nc2C)=O)C1 C(C1(O)CCc2ccccc21)NC(CC(C)C)c1nnnn1CC1CCOCC1 c1(C(=O)NCC2N(C(CCc3c(C)nn(C)c3)=O)CC2)cc2cc(F)ccc2[nH]1 C(=O)(CCN=c1[nH]c(=NC)[nH]c(=NCCc2ccn(C)n2)[nH]1)NCC c1(CC(=O)NCCCN(C(CC2(CSC)CC2)=O)C)cc(Cl)cc2c1OCC2 C1(CN(C(C2N(CC)CC2)=O)C)COCCN1C(=O)Cc1nc(C)sc1Cl C1(NC(CC(=O)NCC#C)=O)C(CNC(c2cccc(F)c2)=O)CCC12CCC2 N1(c2nnc(CC)s2)CCN(C(c2cn(CC3CCOC3)nn2)=O)CC(O)C1 c12nc(C)ccc1C(=O)N1CCN(CC1C)C2=O.c1(NC)nnc(C)cc1O N(C(=NCCCF)N1CCC(C2CCC2)C1)Cc1scc(C)n1 c1(CC)ccc(C(CNC(=O)Cc2ccc(F)cn2)NC(C2CC(O)C2)=O)cc1 CC1CCN(C(=O)CC(C)(C)O)CC1NC(=O)CSc1nncs1 c1(C(=O)NC2C(CNC(C3CCC(C)C3)=O)CCC2)cc2c(cn1)CCCC2 C1(C)(C(=O)NC(CC(C)C)CNC(=O)CCc2cnn(C)c2)CCS(=O)(=O)CC1 Cc1cc2ccc(C(=O)NC3CCC(CCNC(c4cc(CO)[nH]n4)=O)C3)cn2c1 N1(C(C2(c3ccc(C)s3)CC2)=O)CCC(NC(c2cc3sccc3[nH]2)=O)CC1C C=CCCC(C(=O)NCCCNC(=O)C(C)C)NC(C1CCCC12CCC2)=O C(c1c(Cl)nc2ccc(Br)cn12)=CC(N1C2CCCC1COC2)=O Cc1cccn2cc(CC(=O)OCC3(C)CC3Br)nc12 O=C(C#CC1CCCCO1)OCN1CCN(c2ccccc2F)CC1 C(=O)(C(CNC(C1CCCCNC1=O)=O)CCC)NCC1CCN(CCC)C1 N12CCN(CC1)C(=O)C2.CC1(C)CN(C2CCN(C(=O)Nc3ccccc3)C2)C1 CC1CCCC1(C(=O)NCCOC(F)F)NC(c1cc[nH]c1C1CC1)=O n1(CC)ncc2c(C(=O)NC3CN(C(c4ccns4)=O)CC3O)cc(C)nc12 Cc1nccnc1-n1cc(CC2CCCN(CC3=CCCC3)C2)nn1 c1(NC(C2CN(C(C(CC)F)=O)C2)C)ccnc(C2CCCC2)n1 CCC(C)C(O)CC(=O)NC(C)(CNC(C1(C(N)=O)CCC1)=O)Cn1cccn1 N1(C(CC(C)(F)F)=O)CC(NC(=O)COc2ccc(F)cc2)C2CCCC2C1 C=C1CC2(C1)CC(C(=O)N(C1CN(C(=O)CCN3CCC3)CCC1C)C)C2 c1(C(=O)NC2CCN(C(c3c(C)nc(C)o3)=O)CC2)c[nH]c2nccc-2c1 C1(O)(CNC(c2cnc(O)o2)=O)CCCN(C(=O)C2=CCCS2)CC1 c1(CC)nc2c(C(N3CCCC3(C)CNC(=O)CS(C)(=O)=O)=O)ccnc2[nH]1 C(C(=O)NCc1nc(C(=O)NCC2(C)CSC(C)=N2)c(C)o1)(C(C)C)SCC CCC(O)C(C)(C)C(=O)NCCCN(CCO)C(c1cc(C(=O)OC)ccn1)=O c1(C(CC(=O)NC2C(CNC(c3c(C)ncs3)=O)CCC2)C)c(C)n[nH]c1C N1(C(CCCCCC#C)=O)CCCC(C2CN(C(c3ccnn3CC#N)=O)C2)C1 N#Cc1cccc(CNC(=O)Nc2nc(C(F)(F)F)cs2)n1 C1(NC(CCN(C(c2cscn2)=O)CC)=O)CCCCCCC1 CC1(C(=O)NCCCCN2CCC2)CC(O)CN1C(C1CC(=O)OC1(C)C)=O CC1(C)OCC(c2nnnn2CCCC2CC2)(NCC2CCC2CO)CO1 c1(C(=O)NC(C2CCN(C(CCCCSC)=O)CC2)C)cccc(SC)c1O C1(NC(CCCC)=O)COC2(C1)CN(C(C1CC3(CCC3OC)C1)=O)C2 C1(CC)CCOC1C(=O)NCC1(CC(=O)NCCOC2CCCC2)CC1 C1(CNC(n2c(C(=O)OCC)cnc2)=O)C2CC1N(C(=O)C=C1CCC(C)C1)C2 c1(OC)ccc(C(C)C)cc1CN1CCN(C(=O)Nc2ccncc2)CC1C C(=O)(CC(C)(O)COC)NCC(CC=C)NC(c1nn(C)cc1Cl)=O N1(C(c2c(C)[nH]cc2)=O)CCC(C)C(NC(=O)C=Cc2ccc(Br)o2)C1 c1(CC)n[nH]c(=NCC(C)CNC(=O)CCOc2c(C)cccc2C)s1 C#Cc1cc(NC(C2(C)CCCN(C(=O)Cn3cc(Cl)cn3)C2)=O)cc(F)c1 CC(C(=O)NC(C)CNC(=O)CC1OCCCO1)S(=O)(=O)C1CCOCC1 c1(CC(N2CC(CC)N(C(C3CC3C(C)C)=O)CC2)=O)ncn2c1COCC2 C(=O)(C1=CS(=O)(=O)CCC1)NCCN(C(=O)C(S(C)(=O)=O)C1CC1)C C(=O)(CC(C)(C)COC)NC1C(NC(C(CC)=CCCC)=O)C1 c1(CC)ccc(C(N2CC(C)C2C(=O)NC(c2noc(C)n2)C)=O)cn1 CC(C)CCC(O)C(=O)N(CCC(=O)NC1(CO)CCC1)C c1(C(N2CCC(NC(CCC)=O)C2)=O)cc2c(C)n[nH]c2nc1O C1(C(=O)NC(CC(=O)OC)C)(CF)CCN(C(C2CCCN2C)=O)C1 Cc1ccc(F)c(CCNC2CCCC(c3ccccc3)C2)c1 C(=O)(C(C)CN(C(=O)CCCN(C)C(C1CCCN1C)=O)C)OC CCCCC(C(=O)NCC1(C)CC2CC2C1)NC(=O)CCC(C)SC c1(C(=O)NC23C(C)OC(CNC(=O)OC(C)(C)C)(C2)C3)cc(Br)c(F)cc1N c1(OC)cc(F)cc(C(=O)NCC2CCN(C(c3cnns3)=O)CC2C)c1N C1(C(=O)NC2CCCN(C(C3(N(C)C)CC3)=O)C2)CC1C1(C)COC1 Cc1ccn(CC(=O)NC2CN(C(c3cccnc3)=O)C2)c(=O)c1 N1(C(CCN(C(=O)C(C(C)C)NC=O)CC)=O)CCOC2COCC12 C1(NC(C(C)c2ccco2)=O)CCCCN(C(=O)CN2CCC(F)CC2)C1 CCCCCCCCC(=O)N1CCSC(C(=O)Nc2ncc(OC)cc2Br)C1 c1(C(=O)NC(CCCCNC(CC=C)=O)C)cc(F)cc(S(N)(=O)=O)c1 CCCC(C(O)C(=O)N(CCCO)C1CC1)NC(c1cc(C)nnc1C)=O Cc1nocc1C(=O)NCC(F)CNC(C1C=CCCC1)=O N1(C(c2ccc(Cl)nc2)=O)CC2CCN(Cc3ccn(CCF)n3)C2C1 c1(C(=O)NCC2CN(C(c3ccc(Br)o3)=O)C2)cc2n(c1)CCSC2 C1(NC(C2C(COC)(COC)C2)=O)COC2(C1)CN(C(c1ocnc1C)=O)C2 N1(C(C2(CCC)CC2)=O)CC2(C)CN(C(=O)CCCC(C)O)CC2(C)C1 c1(C(N2CCCC(C(C)(O)CNC(=O)Cn3ccnn3)C2)=O)ccc(O)c(Cl)n1 c1(C(=O)Nc2c(Cl)ccc(Cl)c2F)nc2n(c1Cl)CCN(Cc1cocn1)C2 n1(CCOC)ccc(=NC(=O)C2CNC(=O)CN2C(c2n[nH]c(O)n2)=O)[nH]1 c1(C(=O)NC2C(CNC(CCC(=O)OC)=O)COC2)cc(Cl)c(F)cc1Cl C1(CNC(=O)C(=O)Nc2ccc(F)c(Cl)c2F)CCC2C(C1)C2(F)F CCC(CC(=O)NCC(C)CNC(c1cn2ncccc2n1)=O)C(F)F C(=O)(C(CC(F)F)C1CC1)N1CC(CN2CC(c3ccc(OC)cn3)C2)OCC1 C1(CC)CN(C(c2cnc(F)cc2C)=O)CCN1C(=O)C(C)c1cccs1 c1(OCC(=O)NC2CC2NC(c2cc(C(F)(F)F)no2)=O)ccc(F)cc1 N1(C(CN(S(CC)(=O)=O)C)=O)CCC(C2CC2)(CNC(=O)C(C)(C)CF)C1 C(CSC)(C(=O)NC1CC(N(C)C(c2ccnn2Cc2ccccc2)=O)C1)OC C(=O)(C(CO)C(F)(F)F)N(CCCCNC(c1ccncc1F)=O)C C1(CNC(c2cccc(N)c2)=O)CCN(C(C2C3CCCCC23)=O)CC1O c1(C(=O)NC2C(O)CCN(C(C3N(C)CC(O)C3)=O)C2)c[nH]c2ncnc(O)c12 C(c1ccccn1)=C(C)C(=O)NC1CC12CC(NC(=O)CC13COC(C)(C1)C3)C2 c1(OCC)ccc2c(c1)CC(C(=O)Nc1ccc(C=CC(F)(F)F)cc1)CO2 N1(C(CC(C)C)C(=O)NCC(F)F)CCCC(N=c2[nH]nc(C(N)=O)s2)CC1 C(=O)(CCCCCCNC(C1CN(CC)CCO1)=O)NCc1cnc(CCC)s1 c1(C(=O)OCC)ccc(CN2CC=CC2C(=O)N(CCO)Cc2ncc(C)o2)o1 C=C1CCN(C(=O)CC(CC)CC)C(C(=O)NCc2ccnn2CC)C1 C(=O)(CC(C)C(F)(F)F)NCC(CC=C)NC(=O)C(c1ccc(Cl)cn1)(F)F C1(C(=O)O)(CC)CCN(S(=O)(=O)Cc2csc(C3CCC(C(=O)OC)C3)n2)CC1 C1(CC(=O)N(CC(=O)NCCOCCOCCCC)C)CCCCCC1 C(CCC(=O)NCC1CCC(NC(c2n[nH]cc2OCCO)=O)C1)NC(=O)OC S(=O)(=O)(c1ccc(C#N)cc1)NCC(=O)NC1CCCN(C(C(C(C)C)(C)O)=O)C1 N1(C(CC)=O)CCCC(C2CCCN(C(C3CC(C#N)C3)=O)C2)C1 C(C(C)(C)C(=O)NC1C2COCC12)N(C)CC1(C(=O)NOCC2CC2)CC1 Cc1cc(C(=O)NCC2CCC2NC(c2ccc(C3CC3)nc2O)=O)cnc1O c1(NC(C(=O)NCCc2cccc(OC)n2)=O)cc(Br)nc(C(C)C)n1 c1(C(=O)NC2(CNC(C(C)NC(N)=O)=O)CC2)cc2n(n1)CCO2 c1(OC)ccccc1C(CC(C)C)NC(C1CCNC1)C C1(NC(=O)C(O)CC2CCCCC2)CC2CN(C(=O)Cc3ccccc3)CC2C1 N1(C(c2[nH]cc(C)c2)=O)CC(NC(C2CN(C(C)C)C2)=O)CC(C)(C)C1 c1(C(N(C)CC2(NC(=O)Cn3cnnc3O)CC2)=O)ccc(-n2ccnc2)cc1 C(=O)(C(C)(C)C(C)(C)CO)NC1CC2CC(NC(CC(CC)C3CCC3)=O)C1C2 n1(-c2c(C)cc(C)c(C=CC)c2C)c(=O)cc(C)c2ccccc12 C1(C)(C(=O)NCC(CCOC)C)CCN(C(=O)CC2(N(C)C)CC2)C1.NC C1(C(=O)NCC2C(CC(NOCc3scc(C)n3)=O)C2)CC2(C1)CC(C)C2 CCC(O)(CN(C)C(C1COCCC1NC(=O)C(C(C)O)N(C)C)=O)CC N1(C(C(C)SC)=O)CCCC2(C1)CN(C(=O)C(C)(C)OCC(F)(F)F)C2 C=CC1(C(N2CC(CC(F)C(=O)NC(C)COC(F)(F)F)C2)=O)CCCCC1 C12(C(=O)NCC3N(C(C(C)(C)C)=O)CC(O)C3)CC(CO)(C1)OC21COC1 C1(NC(CC2CC(=C)C2)=O)CN(C(=O)COC2CC(F)(F)C2)CC(F)(F)C1 N1(C(C(=O)NC2CC2)=O)CC(O)CC1CNC(C1(F)CCCOC1)=O c1(NC(C)=O)ccc(C(=O)NCC=CCNC(C2C(CCO)C2)=O)cn1.CC N1(C(C(C)OCC=C)=O)CCN(CCNC(=O)CC2C=CCC2)CC1 C1(CC)CN(C)C(=O)CN1C(=O)COC1CC(NC(=O)CCc2nccn2C)C1 Cc1nc(N2CCC(NC(c3cnn(CC(C)C)c3)=O)C2(C)C)c(F)c(C)n1 c1(C(=O)NC2CCC(CNC(=O)CCc3cccs3)C2)ccc2c(c1)NCCC2 CC1OC(C)(C)N(C(=O)OC(C)(C)C)C1CNC(C1CS(=O)(=O)C1(C)C)=O c1(C(N(C2CN(C(c3ccc(OCCC)nn3)=O)C2)C)=O)ccc(O)c(OC)c1 C(=O)(CCS(N)(=O)=O)N1C(CC)C(C(=O)N(C(C)C)Cc2ccco2)CC1 c1(C)ccccc1.c1(C(N(CCOC)CCNC(=O)C=CCOC)=O)sccc1Cl N1(C(CNc2c(C)cccc2C)=O)CC2(CCCC2NC(=O)Cn2ccnc2)C1 N1(C(CCC2CCN(C)CC2)=O)CCOCC(F)(CNC(=O)CSC(F)(F)F)C1 C1(C#N)(C(=O)NCCC2CCN(C(COCC(C)(C)C)=O)CC2)CC12CCC2 N1(C(N(CCN(C(CC(C)=CC)=O)C)C)=O)C(C)CCC1C c1(C(=O)NCC(C)(c2cccs2)NC(=O)COCc2nc[nH]n2)cncc(CO)c1 c1(NC(C2(C(=O)OCC)CC2(F)F)=O)cnn(C(C)C(C)C)c1C c1(NC(C2(COC)CCCOC2)=O)ccccc1S(=O)(=O)C(F)(F)F C(C1=C(C)CCC1)NC(c1nn(C)cc1C)c1n(CCCC)nnn1 C1(F)(C(=O)NCC2C(NC(C3(CC)COC3)=O)C2)CCOC1 c1(NC2CC(NC(CCCCC#C)=O)C2)ncnc2c1ncn2C C(C(C)(C)C(=O)N(CCC=O)OC)OC.C(=O)(CC(C)(C)C(F)F)NCC CCCCN(C(=O)CC1CCN1C(C1(CSC)CC1)=O)C C1(CNC(c2ccn(CCOC)n2)=O)(CO)CCN(C(=O)C2=CCCS2)C1 N1(C(C(C=C)(F)F)=O)CCC(C2(NC(=O)CCc3cncc(F)c3)CCC2)CC1 CC1(OC2(C(=O)NCC(C)(C)NC(=O)CC3CC=CCC3)CCC2)CCCC1 Cc1cc(Cl)cc(C(N2CC(C)(NC(=O)CCNC(C3CCCO3)=O)C2)=O)c1O CC(CCC(=O)NCC1(O)CN(C(c2ccccc2C(F)F)=O)C1)S(C)(=O)=O c1(C(=O)NC(CNC(C2CC(C(F)(F)F)(OC)C2)=O)(C)C)ncn(C)c1C c1(OC)cc(F)c(Br)cc1NC(=O)CC1CCN(c2ccncn2)C1 c1(CC(=O)NCC(C(=O)NCC2CCN(C)C(C)C2)N(C)C)ccc2c(c1)CC2 c1(C(=O)NC2CCCCN(C(C3CC34CCCC4)=O)C2)ccc2occc2c1 c1(C(=O)NC(CCOC)CNC(=O)C(C)CSC(C)(C)C)cccc(CCO)c1 N1(C(CCOCC)=O)CC(NC(=O)C(CC)Oc2ccc(F)cc2)C2(CC2)C1 Cc1ccc(O)nc1CNC(C1CNC(=O)CN1C(=O)CN1CCC(C)CC1)=O C1(C(N2CC(O)(C(C)C)C2)=O)CCC2(CC2)N1C(C12CC1CNC2=O)=O c1(NC(C=CCCC=C(C)C)=O)ccc(-c2ccc(C)s2)nc1 c1(CC)ccc(C(=O)NC(C(=O)NCCC2(CO)CCC2)C2CC2)o1 c1(C2C(C(=O)NCC(CCO)c3ccccc3)CC2)cccc(Cl)c1 c1(C(=O)NCC2(C)CC(NC(COCCC)=O)C2)c(Cl)ccc(C)c1N c1(C(=O)NC2CCC(NC(C3CCC(CCCC)C3)=O)C2)ncn2c1COCC2 C1(CNC(C2(C=C)CCC2)=O)CN(C(=O)C(=Cc2c[nH]cn2)F)CC1C Cc1cc(Cl)ccc1OCC(=O)N(C(C)CCNC(c1ccc(N)c(Cl)c1)=O)C c1(-c2cn(C(C)C(N3CCC(C)C3CC3CC3)=O)nn2)ccc(C(N)=O)cc1 N(C(=NCc1cn(C2COCC2OC)nn1)NCC(C)(C)C)C1CCC(CC)C1 c1(C(=O)NC(C(C)NC(CCCC#C)=O)C)cccc(C#C)c1F C#CCC(CC(=O)N(C1CCCC1C#N)C)NC(=O)CCCn1cncn1 N1(C(C2CN(C(N)=O)C2)=O)CCN(C(C2(O)CCOCC2)=O)CC1CC(F)(F)F CCCCC(CN(C(=O)CCN(C(c1ccc(F)s1)=O)C(C)C)C)CC C(=O)(CC(C)P(C)(C)=O)NCCN(CCOC)C(C1CC(C)OC(C)C1)=O C1(CCCC)(OCCCNC(C(C2CC2(C)Br)OCC)=O)CCCCC1 c1(C(=O)NC2(CO)CCN(C(C(CC=C)NC(C)=O)=O)C2)cc(CC)cc(F)c1 c1(C(=O)NCC2C(NC(CCCCC#C)=O)COC2)cnc2cc(C)ccn12 C1(C(=O)NC(S(C)(=O)=O)COc2ccccc2)CCc2nnnn2C1 N1(C(c2cc(CC)[nH]n2)=O)CCCC(C)C1CNC(=O)C=Cc1ccc(C)nc1 C(=O)(CCCCn1ccnn1)N(CC(C)NC(=O)C(C)(C)c1ccccn1)C C1(NC(c2cc(SC)oc2)=O)CC2CCC(C1)N2c1ncnc2[nH]ccc12 CC1CN(C(=O)CSc2cccc[n+]2[O-])CC1CCNC(=O)CCn1cncn1 c1(CC(=O)N(CCNCCn2cc(CCC)nn2)CC)c(F)cccc1Cl c1(C(=O)NC(CCC)CCCNC(c2ccoc2C)=O)ccc([N+](=O)[O-])cc1F CC(C#N)CCC(=O)NCC(C1CCCC1)NC(c1cn(C2CCC2)nn1)=O C1(COC)CN(C(=O)C(C)(C)c2ccn(C)n2)CCN1C(=O)CCn1cncn1 C12(CNC(=O)C=Cc3ccc[nH]3)CCC1CCN2C(=O)CCc1ccc(O)nn1 C1(NC(=O)C=CCN2CCCC2)CN(C(=O)CC2C=CCCC2)CC12CC2 C1(c2n(-c3ccc(C)cn3)nc(-c3cccc(F)c3)n2)CS(=O)(=O)CC12CC2 C(=O)(CC(C(C)CC)NC(=O)CC1(OC)CCOCC1)NC(CC=CC)CO C#CC(CC(C)(C)C)NC(=O)C=CCN(C)C(C1CCC2(CC1)CC2)=O c1(-c2onc(C(=O)NCCOCCO)n2)cccc([N+](=O)[O-])c1 C1(C(=O)OC)C2CC2CN1C(=O)C1CC1.C=CCCOCCN1C(=O)C1.CN c1(CC)oc(C)cc1C(=O)N(C(C)(C)CC(=O)NC(c1nccc(O)n1)C)C N1(C(Cc2c(OC)nccc2)=O)CCC2CN(C(C3CC(SC)C3)=O)CC12 C1(C(N2CCC(OCC)C2)=O)C2CCN(C(C3OCCC3(C)C)=O)CC12 C12(C(N3CCC(C(C)NC(C(C)(C)OC)=O)CC3)=O)CCCN(CCC1)C2 c1(C(C)C)cccc(F)c1C(=O)NCC1CC(NC(c2cnc(C3CC3)s2)=O)C1 CC1CCCC(C(=O)NC2CCC(N(C)C(c3nccnc3N)=O)CC2)CC1 Cc1ccc(C(=O)NC(C)(CNC(C2CC(F)C(=O)N2)=O)C2CCC2)c(F)c1 N1(C(c2cccc(OC)c2)C(=O)NCC=C)CCC2C(C1)C2(F)F C(CCCCCC(=O)N1CC(O)C(O)C1)NC(C(C)(C)c1ccno1)=O c1(OC)ncc(CN2CCC(C)(NC(=O)CN3CCOCC3)C2)cn1 N1(C(C2C(CC)C2)=O)CCCC1C1CCN(C(=O)CCc2cnn[nH]2)C1 c1(C(C)(C)NC(c2n(CCC)nnn2)C2CC=CC2)cnn2cc(Br)cnc12 N1(C(c2c(C)nc(CCC)o2)=O)CC(NC(c2sc(SC)cc2C)=O)CCC1C C#CCC(C(=O)N1CC(OCC(=O)NC2CC2)C1)C1CC1.C(C)(C)O c1(C(=O)NCC2(OC)CN(C(c3cnc(COC)s3)=O)C2)cn2c(n1)CCCC2 N1(C(COCC#C)=O)CCCC(C2CN(C(c3ccc(O)cc3F)=O)C2)C1 c1(CNC2C3CN(C(C4=C(C)OCC4)=O)CC2CC3)n[nH]c2cc(Br)cc(F)c12 CN1N=C(CC(=O)NC2(C(=O)NCc3cccc(O)n3)CCC(C)(C)C2)CC1=O C1(CNC(C23C(C)OC(C)(C2)C3)=O)N(C(c2cc(Cl)sc2Cl)=O)CCCC1(C)C C(=O)(C(O)C1=CCCCC1)NCC(C1CCCCC1)NC(C1CS(=O)(=O)C1)=O CC1CN(C(C2CN(C(N)=O)C2)=O)CC(C)N(C(=O)Cc2cccc(F)c2O)C1 c1(C(=O)NC2CN(C(CC=CCC)=O)CC23CCC3)ccc(=O)n2c1COCC2 CC(C)C(C(=O)N(C1CCN(C(c2cncs2)=O)C1)CCO)c1ccn(C)n1 Cc1ccccc1-c1cccc(CN(CCCCCCl)CC2CC2Cl)c1 C(=O)(C(C)C(C)C(C)(C)C)NCCCN(C(c1cncc(OC)c1)=O)CC C1(C(=O)NCc2cncc(C(=O)NC(C)CCC3CC3)c2)CCCCC1(C)C C1(CNC(CN(C)C)=O)CCC2(CCC2)CN1C(=O)C=C1CN2CCC1CC2 C=CCC(C(=O)N1CCC(CCNC(c2c(N)cc(Cl)nc2Cl)=O)C1)C(C)C C1(CNC(CC2(NC(c3c(C)snc3)=O)CC2)=O)CCC(=O)NC1C C1(NC(CN(CC)CC)=O)CCC(C(=O)NCCC(O)CCO)C1 CC(C)CC(C(=O)N1CCC=CC1C(=O)NCC1(N(C)C)CCCC1)N(C)C N1(C(Cn2c(C)nc(C)n2)=O)CC2CC(NC(=O)C(O)CC3CCCC3)CC2C1 N1(C(CSCC)=O)CC(CCNC(c2cnc(SC)nc2)=O)C(C)C1 C1(C(=O)NC2(C)CC(F)(F)C2)CCOCCN1C(C1CCC(F)(F)C1)=O C(C)(C(=O)NCC1CCCC1N(C)C)(N(C(C(C)=CC(C)(C)C)=O)C)C1CC1 C1(C(N(C)CC2(O)CCCN(C(=O)CNC=O)C2)=O)CCC2(CCCC2)C1 N1(C(C2CCN(CC)C2)=O)Cc2nccn2CC(NC(=O)CCC2CC(C)C2)C1 N1(C(c2nccc(C#C)c2)=O)CC2CCC1CN2C(c1cnn(CCO)c1C)=O Cc1oc(S(=O)(=O)Nc2cc(Cl)cc(Br)c2F)cc1S(C)(=O)=O N12CCN(C(C3CC3)C1)C(=O)c1cncc(c1)C2=O.c1(CC)cc(C)cc(C)c1 c1(C(=O)NC2C(CNC(P(C)(C)=O)=O)CC2)cc(F)c(F)cc1Br c1(C(=O)NCCC(C)NC(c2cccc(CC)n2)=O)cc2sc(C)nc2[nH]1 c1(C(=O)NC2C(C)CN(C(=O)Cc3nncs3)CC2)cnn2ccncc12 c1(CNC(CCC#C)=O)ccc(CNC(c2ccc(CO)cc2F)=O)c(F)c1 N1(C(C(c2cncn2C)N(C)C)=O)CCC(C)(C)C(NC(C2CC(O)C2)=O)C1 c1(C(=O)NC23CC(CNC(CCC(=O)NCCC)=O)(OC2)C3)[nH]cc2c1CCC2 N1(C(C2C(NC(C3(C)CCSCC3)=O)COC2)=O)CCOC2(CC2)C1 C1(NC(CCC=C)=O)CC1C1CCN(C(c2cccc3sncc23)=O)CC1 N1(CCC)CCCN(C(=O)C=CCC(C)(C)NC(C2OCCCC2(C)C)=O)CC1 C#Cc1cc(C(=O)NCC2CCN(C(C3(F)CC3)=O)CC2C)cc(Br)c1 CC(C)(C)C(C(=O)NC1CCN(C(C23CC4CC2C3C4)=O)C1)N1CCCCC1 c1(C(N2CCCC(N(C)C(c3cnn(C)c3Cl)=O)C2)=O)cc2cccnc2o1 C1(C(=O)NC(C2CCCC2)C#C)CCCCC1(C)NC(=O)C(C)NC=O C1(C(N(CC=C)CCO)=O)CN(C(c2c[nH]nc2Cl)=O)CCO1 c1(COC(C)C(=O)OC2C3CCCC23)cc(-c2ccccc2)nn1C c1(OC)cccc([N+](=O)[O-])c1C(N1CC(O)(CNC(c2ccc(F)cn2)=O)C1)=O N1(C(C2C(C)C(=O)C2)=O)CCOCC1CNC(c1ccn(C(F)F)n1)=O CC1(C)CCN(C(=O)CC2CCCC23CC3)CC1CNC(C1(Br)CC1)=O CC(C(N)C(=O)Nc1ccc(-c2noc(=N)[nH]2)cc1)c1ccccc1 C1(CC)CN(C(=O)C(=O)NC(C)C)CCC1NC(=O)C(=Cc1cccnc1)F N1(CC(=O)NC(C)(C)CCNC(C23CC(C2)C3)=O)CCCCC1=O N1(C(CN(C(C(C)C)=O)C)=O)CCCC(NC(C2(F)CC2(F)F)=O)C1 N#Cc1ccc(N2CCCC(C(F)(F)F)CC2)nc1Cl Cc1nsc(C(N2CCCC(CNC(c3cc(Br)nn3C)=O)C2)=O)c1N c1(NC(C2CN(c3cc(CO)ncn3)CCS2)=O)ccc(F)c(C2CC2)c1 Cc1c(C(N2CC3CC(O)C2C3NC(=O)CCF)=O)nc2sccn12 C1(CNC(COC)=O)CC2(CCN(C(c3c[nH]nc3OC)=O)CC2)CO1 N1(C(CC2(CC=C)CCCC2)=O)CCCC(CCNC(C2CNC(=O)O2)=O)CC1 c1(C(=O)NC2C(NC(c3cn(C)nc3)=O)CCC2)ccc2c(c1)COC2 C1(CNC(c2cc(C)on2)=O)CC2(CCN(C(=O)C=C(Cl)Cl)C2)CO1 N1(C(c2c(CC)[nH]c(=N)s2)=O)CCC2(CCC2NC(C2CC(C)N(C)C2)=O)CC1 CN1CCC(C)(CNC(=O)CC2CCCN(C(C3CC(O)C3)=O)C2)C1 CCCC(C(=O)OC)C(=O)NC(CNC(=O)CC1CCCC(C)(C)O1)CC(=O)OC C1(C(N(C)CC2(C)CCCC2)=O)CCN(CC(=O)N(C2CCCCCC2)C)CC1 C(=O)(CCCCCCCBr)NC(C1CCCN(Cc2cc(F)cc(Br)c2F)C1)C C(c1c(C)noc1C)=CC(N1CCN(C(CC=C(C)C)=O)CC1)=O CC(C)C(O)C(C)C(=O)N1CCC(CF)(NC(=O)C(=O)NCCC(F)F)C1 CCCN(OC)C(=O)C1(C)CC(O)CN1C(c1cc(F)n(C)n1)=O N1(C(CCC(=C)Cl)=O)CCCCN(C(=O)CCCCNC(=O)C2CC2)CC1 N1(CCN(C(CN(C2CC2)CC)=O)C)CCN(C(=O)Cc2c[nH]nc2C)CC1 CCCCCC(C(=O)Nc1cccc(Cl)c1C)N1CCN(C(C)CC(=O)OC)CC1 c1(C(=O)NC(CNC(c2cc(C(F)(F)F)on2)=O)CO)ccc(Cl)nc1O C1(N(c2cn(CCC#C)nc2)C)CCCN(C(C2(NC(C)=O)CCOCC2)=O)C1 N1(C(COC2(C)CN(C(C)=O)C2)=O)CCCN(CCC(C)(C)C)CC1 c1(CC)nc(=N)[nH]cc1C(=O)NC1CCN(C(C2(c3cc[nH]n3)CCC2)=O)CC1 N1(C(CCNC(C)=O)=O)CCN(C(C2OCCOC2C)=O)C(CC(F)(F)F)C1 N1(C(c2[nH]cc(CC)c2)=O)CC2CCC(CNC(c3ocnc3COC)=O)(C2)C1 C1(C(N(c2cccc(C)c2)CC)=O)CCC2(CC2)N1C(=O)C(CC)CCOC c1(C(=O)NC(C(=O)NC(C)CC(F)(F)F)C2(O)CCC2)cc2cccnc2[nH]1 c1(NC(C2N(C(Cc3cnc(C)s3)=O)CC2)=O)cc(Br)ccc1[N+](=O)[O-] c1(NC(N2CCC(CC(=O)NCC(=C)C)CC2)=O)ccc(NC)c(F)c1 c1(N2CC(C)C(NC(=O)CCc3cccnc3F)C2)nc2ncc(Cl)cc2o1 c1(C(=O)NCCOC2CN(C(C3CC(CF)C3)=O)C2)cc2n(n1)CCOC2 N1(C(CCC(=C)Br)=O)CCCC(NC(=O)CC2CC(OC)C2(C)C)CC1 c1(C(N2CCC(C)(CC(=O)NC3CCC(C)(O)CC3)C2)=O)ccc2[nH]ccc2c1 C1(NC(CC=C=C)=O)CCC2(CC1)CN(C(=O)Cc1n[nH]c3ccccc13)C2 CCCC(CCC)CC(=O)N1CCCCC1CCCNC(C12CC(OC)C1C2)=O N1(C(C2N(C(C)C)C(=O)CC2)=O)CCCC(N=c2nc(C(F)(F)F)[nH]s2)(CO)C1 CC1CCCN(Cc2ccccc2NC(=O)COCc2ccccc2)C1 C(C(=O)N(CC(O)CNC(C1CC1c1ccsc1)=O)C)(OCC)OC C1(C(N(C(C)C(C)(C)C)C)=O)(CF)CCN(C(=O)Cc2ccc[nH]2)C1 c1(CCNC(C(C)n2cnnn2)=O)ocnc1CNC(=O)Cc1ccco1 c1(NCC2CCN(C(c3c(C)cc(Br)cn3)=O)CC2)ncc(S(=O)(=O)O)cc1Br C1(C(N2C(C)CSCC2)C(=O)NCc2ccccc2)CCCCC1(F)F Cc1sc(Br)nc1CC(=O)NC1CC(N(C(=O)CN(C)C(N)=O)C)C1 C1(CNC(Cc2n(C)nnc2)=O)CN(C(C2(C)CCOC2)=O)CC12CCC2 N1(c2ncnc3ncn(C)c32)CCCc2c1ccc(Br)c2F N1(C(c2ccc(C)s2)=O)CC2(NC(c3cc(C)n(C)c3)=O)CC1C2 O=C(CS(=O)(=O)c1ccc(Cl)cc1)NCCCOCCNC(c1ccncn1)=O C1(C(CC)CC)CCC(NC(=O)C(=O)NCCCCN(C)C)CC1 C(CCC(=O)NCc1ccco1)N(CCCC)CCOC c1(C(=O)NC(C(C)NC(C(C)N(CC)CC)=O)CO)nc(-c2cccs2)oc1C C(=O)(C(C(C)(C)C)n1cc(Br)cn1)Oc1ccc(C)cc1 CCC(C(C)C)C(C(=O)Nc1ccc2c(c1)OCO2)N1CCCC1c1ccsc1 C#Cc1ccc(C(=O)NC2CCCN(C(C34CCC(CO)(CC3)C4)=O)C2)cc1C Cc1cnc(NCC2(CNC(C3COCCC3(F)F)=O)CCCC2)c([N+](=O)[O-])c1 C(C(C(=O)N(C)CC1CCOC1)C(C)(C)C)NC(CC(C)C)=O c1(C(N(C(C)CC(=O)NCC2CN(C)CCO2)C)=O)cc(O)ncn1 N1(C(CN(C2CCC2)C)=O)CCCC(NC(c2cocc2C(N)=O)=O)C1 c1(COC(C2CN(C(C(=O)NCCOCC)C)C2)=O)cc(Br)ccc1[N+](=O)[O-] C#CCCCCC(=O)NCC1CN(C(=O)C=C(C)C)CCC1C N1(C(C2(C)N(C)CCC2)=O)CC(C2CN(C(=O)CN3CC4CC4C3)C2)C1 CC(C)(C#N)CC(=O)N1CC(CNC(=O)CN2CCC(C(N)=O)CC2)C1 C1(C(=O)NCC(C)N(C(=O)CC(Cl)Cl)C)CC2(CCCO2)C1 c1(CO)ccc(C(c2ccc(Br)cc2)NC(=O)CC2(O)CCC2)nc1 c1(CC)ncsc1C(=O)NCC1CCC1NC(C1CCCN1c1cnccn1)=O C1(NC(c2cn(CCN(C)C)nc2)=O)CC(O)CN(C(C2(C(N)=O)CCC2)=O)C1 N1(c2n(CCCCC=C)nnn2)CC(C)N(C(=O)CCCC(C)C)CC1C CC1(C)CCCC1(C)NC(=O)C(N1C2CCC1CCC2)=O c1(NC(=O)CC2CCN(C(=O)CCC3CCCO3)C2)cc(F)ccc1O c1(Cn2cc(C3(O)CN(C(=O)CCCCC4CC4)C3)nn2)cc(Cl)ccc1Cl N1(C(CCc2c(C)noc2C)=O)CCCC(O)(CCNC(C2CC23CC3)=O)C1 c1(OC)cc(CNC(C2N(CCC(=O)Nc3csc(C)n3)CCC2)=O)ccc1OC C1(NC(C(C(C)C)O)=O)CCCC2CN(C(=O)Cc3ccc(O)c(Cl)c3)CC12 c1(CC(=O)N(C2CCN(C(C3(C)CCCO3)=O)C2)CCC)ccc(O)cc1 c1(C(C(N2C(c3ccc(C)cc3)C(C)C2)=O)(F)F)cc(F)ccc1C C(c1cc2ccccc2o1)=CC(=O)NC1CC(NC(c2n(C)ccc2)=O)C1 C1(C)(NC(C)=O)CCN(C(=O)CC2CN(C(=O)COCCCN=[N+]=[N-])C2)C1 N1(C(c2c(OC)csc2)=O)CC(NC(C2CC23CCOCC3)=O)CC(F)(F)C1 c1(N2C(C)CC(CNC(c3c(CC)oc(C)c3)=O)C2)nc(OC)c(F)c(C)n1 N1(C(C2(CC#C)CCCC2)=O)CCC(C)(CC(=O)NCCCC(=O)NO)C1 c1(C(=O)NC2CN(C(Cc3c(C)cc(Cl)cc3)=O)C(C)C2)ccccc1N=[N+]=[N-] C=CCC(C(=O)N1CCC(NC(c2ccc(CSCC)cc2)=O)CC1)C(C)(C)C C(=O)(CC(CCC)NC(c1nocc1C(C)C)=O)N1CCC(C#C)C1 CCCCCC(O)CC(=O)N1CCN(C(C2CN(C(C)C)C2)=O)CC1C(F)F C#Cc1ccc(C(c2nnnn2C2CCC2)NCC2(CO)CC2)nc1 c1(NC(C(=O)NC(c2noc(C)n2)(CC)C)=O)cc(OC)nn1C c1(OCC)ccc(C(=O)NCC(C)(CO)NC(=O)CCC=CC(C)C)cc1 C=CCC(C(=O)OCC)NC(=O)CCN(CC=C)C(C1C2CCCC12)=O N1(C(CN2CCCC(CC)C2)=O)CCC(NC(c2cc(C)c(C)o2)=O)C(C)(C)C1 Cc1cc(C(=O)NC2CC2CNC(=O)C(C(C)C)N2CCCCC2)c(O)nc1C CC1CN(CCc2ccccc2Br)CCN1c1ccncc1 C1(NC(c2nn(C)c(C(N)=O)c2)=O)CCN(C(C2C=CCC2)=O)CC1(C)C C(=O)(CC(C)C(C)(C)NC(c1ccn2cccc2c1)=O)NCC(C=C)O c1(C(N(CCCNC(=O)CN(c2ccncc2)C)C(C)C)=O)ccc(CO)nc1 N1(C(C=CC=CC)=O)CCN(C(=O)C(c2cccc(Cl)c2)O)CCC1C c1(CN2CC(NC(c3c(C#C)cc(F)cc3)=O)C(O)C2)ccc2nn(C)cc2c1 c1(NCC(=O)NC(C)C(C)Nc2ncncc2C#N)ccccc1[N+](=O)[O-] N1(C(c2ccc(OC)c(I)c2)=O)CCCc2cc(OC)ccc21 C#CCC(CC(=O)N1CCC(COC)CC1)NC(=O)C(CC(C)C)N(C)C C1(CNC(=O)CN2CC3CC3C2)CN(C(=O)CN2C(=O)CNC2=O)CC1O N1(C(CCC2CCN(C)CC2)=O)CCC2(CCN(C(C3(C)CCCCC3)=O)C2)C1 Cc1cc(NC(C2CC(C)CN2C(c2ccc3n[nH]cc3c2)=O)=O)c(F)cc1F c1(C(N(C2CCCN(C(=O)C(C)(C)O)CC2)C)=O)cccc(C(F)(F)F)c1O N1(C(COCC(=O)OC)=O)CCC(CN(C(=O)CSCCC(F)(F)F)C)C1 c1(OC)ccc(C(O)C(N2CC(NC(c3ccccc3F)=O)C(C)C2)=O)cc1 c1(N(C2(C#N)CC2)C(c2cccc(OCC)n2)C)cccc([N+](=O)[O-])c1 c1(C(N2CC(NC(C3(CF)CCC3)=O)CC(O)C2)=O)cc2c(o1)CCCC2 N1(C(CCCCOCC)=O)CCC2(CCCN2C(=O)CC2NC(=O)NC2=O)CC1 c1(C(=O)NCCC2CC(NC(C3(OC)CCC3)=O)C2)cnc(C)nc1 C1(O)(CNC(C2CC(NC(c3cc(C4CC4)on3)=O)C2)=O)CCSC1 c1(CNC(c2c(C)onc2O)=O)cnc(O)c(F)c1.c12ccccc1CNC2=O c1(CC)ccc(CCc2noc(-c3cc(C4CCCN4)[nH]n3)n2)cc1 N1(C(C23CC(C)(OCC2)C3)=O)CCCC(C2CN(C(C3CCCC34CC4)=O)C2)C1 OCC(CC1CCOC1)CN=c1nc(N2C3CCCC2COC3)c2c([nH]1)CCC2 Cc1cn2nc(C(=O)NC3CCN(C(=O)Cc4cnc[nH]4)C(C)C3)cc2c(=O)[nH]1 c1(C(C(=O)NCC(CN(C)C)NC(=O)OC(C)(C)C)O)cccnc1 C1(C2(O)CCOCC2)(C(N2CC3CCN(C(=O)C4=C(Cl)CCCC4)C3C2)=O)CC1 C1(C(C)NC(=O)CCCN(C)C)CN(C(c2ccnc(C(C)(C)C)c2)=O)CCO1 c1(C(=O)NC2C3CN(C(C=CCC)=O)C2CC3)cc(SC)ccc1C C1(CC(=O)NCCN(C(c2ncoc2C2CCC2)=O)C2CC2)CCOC1=O n1(CCCC(=O)NCCC(=C)CNC(=O)C(C)C2CC2)ccc2ccccc12 C1(CNC(c2c(CC)nco2)=O)CCCCN(C(C2CC3C=CC2CC3)=O)C1 N1(C(Cc2nnc(C)o2)=O)CCCC(NC(c2ncc(Br)cn2)=O)C1 C(=O)(C(CC#N)c1ccccc1)NC(C)CN(CC(C)(C)O)CCCCC(C)(C)C N1(C(C(C)N(C(=O)C=CC2CCOCC2)C)=O)CCC2CCN(C)CC12 O(NC(=O)C(CC(=O)OC(C)(C)C)NC(=O)OC)Cc1c(N)cc(C)cc1Br CC1(C)CC2(CC(C(N3CC(O)(CNC(=O)CC4(O)CCOCC4)C3)=O)C2)C1 Cc1cc(Cl)n[nH]c1=NC(=O)C1CCCC1NS(=O)(=O)c1ccc(Cl)cn1 CC(F)(F)C(F)C(=O)Oc1ccc(CN(C2(C3CCCO3)CCCCC2)CC2CC2)o1 C1(c2n(CCC)nnn2)(NCc2cn(C3CC3)nn2)CCC(CC)C1 N1(C(c2cccc(C)c2Cl)C(=O)Nc2ccccc2C)CCC(O)C(C)(C)C1 N1(C2CCN(CCc3csnc3Br)CC2)CCC(F)(F)CC1.c1(C(=O)NC)cnsc1 c1(C(=O)NCC(CN(C(c2c(CC)noc2C)=O)C)O)c(C)ccnc1O C#Cc1cccc(C(N2CC3(C2)CN(C(c2ccnc(OC)c2)=O)C3)=O)c1F C1(NC(c2c(C)csc2)=O)CS(=O)(=O)CC1NC(c1c(C(F)(F)F)coc1C)=O N1(C(C(=O)NCCC2CCCC(C)C2)=O)CC(N)CC2(CC2)C1 C1(C(=O)NCc2c(C(N3CC(CC(C#C)C)C3)=O)n[nH]c2)CN(C)CC(C)O1 C1(c2n(C(CC)(C)C)nnn2)(NC(C)(C)COC)CN(C)CC1C c1(C(=O)NC(C2CCCN(C(c3cc(C)c(C)s3)=O)C2)C)ccc2oncc2c1 CC1CC2CN(C(C3C(C)(C)C3(F)F)=O)CC2N1C(=O)C=CC1CCCC1 C=CCCCCC(=O)NC1(C)CN(C(c2cccc(C3CCOC3)c2)=O)C1 Cc1nn(CC(=O)NCC(C)(C)CN(C(=O)C(N2CCOC2=O)C)C)c(=O)o1 c1(C(N2C3(CN(C(=O)CCBr)C3)CCC2)=O)ccc(I)c([N+](=O)[O-])c1 N1(C(C(=O)NC)C)CC2CCN(C(c3cccc(C4COC4)c3)=O)CCC2C1 c1(CN(C2CCCC2)CC(C)C)c(F)ccc(C#N)c1F C1(NC(c2cc(COC)no2)=O)COC2C(NC(=O)C(F)CC3CC3)COC12 N1(C(C(c2ccnn2C)C)=O)C(CC(=O)NCC(F)(F)C(N)=O)C2CCCC12 N1(C(CCOCC)=O)CCCCC(NC(C2CC(F)(CO)C2)=O)C1 CS(=O)CCC(=O)NCc1cn(CC2(C(=O)NCc3ccc(C#N)o3)CC2)nn1 C1(CNC(CS(=O)(=O)N(C)C)=O)CN(CCCc2ccccc2)CCC1(F)F Cc1ccc(CC(=O)NCC2(C(N3CCN(C)C(CO)C3)=O)CCC2)cc1O C1(CNC(C(CCCC)(C)F)=O)CCC2(CCC2)CN1C(=O)CCOCCC CCCC(C)C(=O)NC(Cn1cccn1)C(N1CCC(C)(CC)C1)=O N1(C(c2scc(C(C)=O)c2)=O)CCCC(N(C)C(c2cc(C)c(C)o2)=O)CC1 N1(C(CCC(=O)NCCC)=O)CCOCC(NC(c2cc(Br)ccc2C)=O)C1 Cc1ccnnc1C(=O)NC1CCOCC1C(=O)NCc1c(C)noc1C N1(C(CCCc2onc(C)n2)=O)CC2CCCC(NC(C3CCNC3=O)=O)C2C1 CC1(NC(=O)CC2(C3CC3)CC2)CC(NC(=O)C(O)C2CCCC2)C1 C1(NC(C2(NC(C)=O)CCC2)=O)CCN(C(c2ccc(CC#N)cc2)=O)CC1F C(C)(C(C)(C)C(=O)NCC(C)(C1(C)CC1)OC)NC(CCC(C)OCCOC)=O Cc1ccccc1C(N1CC(CNC(=O)Cc2ccnnc2O)C1)=O C1(OC(C)C)CC(NCCCc2ccccc2)C1(C)C c1(CC(N2C(C)CC(NC(CCOCCC)=O)C2)=O)c(Cl)cccc1Br C1(CCC(=O)NC2C(CNC(c3cc(C)sn3)=O)CC2)CCCN(C)C1 c1(C(=O)NC(CNC(c2c(C)c(N)cnc2)=O)C)cc2cc(F)cc(F)c2[nH]1 C1(CNC(c2c(C)cc(C)[nH]2)=O)CC2CCC1N2C(c1cc(CO)on1)=O c1(N(C2CNCC2F)C(=O)NC(c2ccccc2)C)ccnc(C2CC2)n1 N1(C(C2CC(C)SCC2)=O)CCN(C(=O)CCN2CCCC2)CC1CO Cc1cc(C(N2CC(CO)(NC(C3CCCC3O)=O)C2)=O)c2c(C)n[nH]c2n1 C1(OC)(CO)CN(C(C23CCC(C2)C3)=O)C1.C1(N(CC(=O)N)C)CCCC1 C1(NC(C2ON=C(C)C2)=O)CCCN(C(C23CC4CC2C3C4O)=O)C1C c1(OC)ccc(C)c(NC(c2ccnc(-c3ccc(-c4nn[nH]n4)nc3)c2)=O)n1 c1(C(N(C)CC2N(C(C3C(=C)C3)=O)CCC2)=O)ccncc1N(C)C Cc1cc(NCC(c2ccc(N(C)C)cc2)=O)nc2ccc(I)cc12 C1(C(=O)OC)(C(=O)NCC2(NC(c3n[nH]cc3C3CC3)=O)CC2)CC2(CCC2)C1 C#Cc1ccc(C(N2CC(CNC(c3cnc(O)c(Cl)c3)=O)CC2(C)C)=O)cc1 c1(C(N(CC(CC)NC(=O)CCCS(N)(=O)=O)C)=O)cccc2oc(=N)[nH]c12 CN1CCc2c(C(N3CC4CN(C(=O)CCCCCl)C4C3)=O)cccc21 C1(CC(=O)NCCNC(C(C)SC)=O)CCCCC12CC2 C12(CC)CN(C(C3CC(C)OC3=O)=O)C(CNC(=O)C(C)(C)CO)(C1)C2 O(NC(=O)C1CCc2c[nH]nc21)C(CC(C)C)C(=O)NCCCCCCF C(=O)(C1SCCc2sccc21)NC(C(C)C)(C)CNC(c1cnnn1C)=O C1(OCC)CC2(C1)CC2C(=O)Nc1cccc(C(N2CC(C(=O)N(C)C)C2)=O)c1 C123CC(C1)(OC21CN(C(=O)C(C(C)O)N(C)C)C1)C(=O)N3.Cc1nc(CO)n[nH]1 c1(C(=O)NC23C(CN(C(CS(CC)=O)=O)C2)C3)ccc2ncncc2c1 O=C(C1=COc2ccccc2O1)NC12CCC(CF)(C1)OC2 C(C1(C)COC1)=CC(=O)NC1(CN(C(=O)Cn2ccc(Br)n2)C)CC1 c1(COC)ccccc1CN1CC2(CC2C(=O)NCc2c[nH]c(Br)c2)C1.OCC c1(C(C(=O)NCC(CNc2nc(C)sc2)(C)F)C)cccc(F)c1 CCCC(C#N)C(=O)NCC1CCN(C(=O)Cn2cnc([N+](=O)[O-])c2)C(C)C1 c1(C(=O)NCCC(C)CCNC(C2CCC(C#N)CC2)=O)ccc2cncn2c1 C1(C(=O)NC2CCCN(C(Cc3c(C)con3)=O)C2)CCCc2ccccc2C1 C1(CC=C)(NC(C2CC(=O)N2)=O)CN(C(c2cn(CCO)nn2)=O)C1 Cc1nc(C(N2CCC(O)(C(C)NC(c3cnccn3)=O)C2)=O)c2n1CCCC2 CCC(CC)CCC(=O)N1CC2(C1)CN(C(C1CCCC(=O)O1)=O)C2 C1(C(N2CC(CCC=C)(C(=O)NC3(C)CCCC3)C2)=O)CC2CCC1C2 N1(C(C(CC(C)C)OC)=O)CCCN(C(c2cncc(N)c2)=O)C(CO)C1 N1(C(C(CC#C)O)=O)CCCC(NC(c2ccc(-c3nnc(C)o3)cc2)=O)C1C C(CC(C)C)(C(=O)N1CCC=C(F)C1)N(C(C1C(OCCN(C)C)CC1)=O)C C1(CN(CCCCCO)C(c2ccc(CC)[nH]2)=O)CN(C(C)C)CCO1 c1(C(C(=O)NC(c2c[nH]nc2-c2cnccn2)=O)N2CCCC2)nc(Cl)c(Cl)s1 C(C)(CO)(CC(C)C)NC(c1cc(CNC(c2ccc(OC)s2)=O)ncc1)=O Cc1ccc(C(=O)NC(CNC(c2scc(Br)c2C)=O)CO)cc1 CC(C)CCCCCC(=O)NC1CCOCC1NC(c1cc2cccnc2[nH]1)=O c1(C(=O)OC)cc(C(=O)NCCN(C2CCCCC2)C(=O)CCC2(C)CC2)co1 C1(N(C)C(c2cc(=O)cc[nH]2)=O)CCCCN(C(=O)C(CO)c2ccccc2)C1 O=C1CC(NC(c2coc(CNC(=O)Cc3cnoc3)n2)=O)CC(=O)N1 CCC(CO)CCNC(C1CCN(C(c2ccn(COC)n2)=O)C1CC)=O c1(CNC(c2c(C)cccc2)CF)ncnc2ncn(C)c12 c1(C(CC(=O)NC(CNC(CN(CCOC)C)=O)C(C)C)C)ccc(F)cc1F C#Cc1c[nH]nc1C(N1CCC(NC(C2CCCC2Cc2ccccc2)=O)C1)=O C1(CNC(c2c(Cl)cn(C)n2)=O)CN(C(=O)C2=COCCO2)CCC12CCOC2 c1(C(=O)NC2C(NC(CC3C(C)(C)CCC3)=O)CC2)cc(Cl)c2n[nH]cc2c1 N1(C(c2ccc(CC(C)C)s2)=O)CCC2(NC(c3nc(Cl)sc3Cl)=O)CC2C1 C1(CN(C)C(C2CC2(C)C)=O)CCCN(C(=O)Cc2ccn(C(F)F)n2)C1 C1(C)(NC(c2nc(C)n(C)n2)=O)CCCN(C(c2ccccc2SCCO)=O)C1 N1(C2CCCC2)CC2CCCC2(Nc2ccc3occc3c2)C1 O=C(CC(C(F)(F)F)n1ccnc1)NCC1CN(C(c2cncc(CO)c2)=O)C1 C1(C)(CC)CCCN(C(=O)C(CCC2CC2)NC(c2ccc(CO)cc2)=O)CC1 N1(C(C=C(C)C)=O)CC(NC(=O)C(CC(C)C)NC(=O)OC(C)(C)C)C2(CC2)C1 C(CC1=CCCCCC1)NC(C1C(NC(C2CC2C2CCC2)=O)CCC1)=O CC1=CCC(C(=O)NC(C)(C)CCNC(=O)CNc2ccc(C(N)=O)cn2)CC1 C(c1ccc(F)cc1F)=CC(=O)NCC1CCCCN1C1CC1 S(=O)(=O)(c1cccc(Cl)c1)NC1(C#N)CN(C(c2cc(F)cnc2Cl)=O)C1 c1(C(N2CCCN(C(C(CCC)(C)CC)=O)CC2)=O)cnc2c(c1)CCCC2 c1(C(N2CCCC(C(F)F)C2)C(=O)NCC2(C)CC2)cc2n(n1)CCCCO2 C12(CNC(=O)CCC3CCCC3)CC(C1)C(NC(=O)Cc1cnns1)CO2 C(=O)(CC(C)(C(F)F)N(C)C)N(C1CCN(C(CC(CC)C(F)F)=O)CC1)C C=C(Cl)C(C)(C)C(=O)N1CCCN(C(c2c(OC)ccnc2OC)=O)CC1 CC1CC(N(C2CCCOC2)C)CN1C(=O)CN1CCCC1 S(=O)(=O)(c1cccc(F)c1)NC(CCN(C)CC1CC(NC(=O)CN(C)C)C1)=O c1(OC)c(C(=O)NC2CCC(C(=O)O)C2)ncnc1Cl C#CCC(C(=O)NCc1cccc(O)n1)NC(c1cnn(C)c1C)=O c1(C(=O)NC2CCCCN(c3nnc(C(C)(C)C)o3)C2)cc(Cl)c(F)cc1F Cc1ccc(Cl)c(OCC2(CCO)CCN(C(=O)C(C)(C)O)C2)c1.C1(C)C(=O)O1 C(C1CCCCC1)=CC(=O)NCC1(O)CC(C(=O)NCCC(C)N(CCC)C)C1 C1(CCNC(CC(C)n2ccnc2)=O)CCCN(C(c2cnn(CCO)c2)=O)C1 C1(NC(C(CC)OCC)=O)CCC2(CC1)CCN(C(=O)CSCCC#N)C2 C1(NC(c2c(Br)n[nH]c2C)c2n(C(CC)(C)C)nnn2)CCn2ncnc2C1 C=CC(C)(CC)C(=O)NC1C2CCN(C(c3ccnn3CC)=O)CC12 c1(CC(C(=O)NC2C(NC(C3(C)CC3)=O)CC2)(C)C)nc2ccccc2[nH]1 c1(CCC(N2CC(NCc3c[nH]c(Br)c3)C(O)C2)=O)ccc(O)cc1 n1(CC)nc(C(=O)NCC2CCC(NC(=O)CSC(F)(F)F)CC2)ccc1=O c1(C(c2n(CCOCC)nnn2)NCc2ncccn2)cc2c(s1)CCC2 c1(C(N(CCC(C)NC(C2(CC=C)CC2)=O)C)=O)cn(CC2CC2)nc1C CCC(CC)CCCC(=O)NCc1ncc(C(=O)NCC(C2CCCO2)O)cn1 C#CCCCN=c1[nH]c(=NCC(C)(F)C(C)(C)F)[nH]c2cc(OC)ccc12 C(=O)(C(F)C(=O)Nn1cc(-c2cncc(Cc3ccc(N)nc3)c2)nn1)OCC c1(C(N(CCNC(c2c(C)csc2Cl)=O)C)=O)cc2ccncc2[nH]1 c1(OC)ccc([N+](=O)[O-])cc1S(=O)(=O)N(C)Cc1cc(Cl)cc(Br)c1 C(C(CSC1CC1)C(=O)N(C)CCOCCO)NC(CNC(N)=O)=O CCC(CNC(C1(C)CC1(Cl)Cl)=O)(CC)NC(C1CC=CCC1C)=O C(CC(=O)NCC(O)CNC(CCNC(C)=O)=O)(c1cccs1)NC(COC)=O CC1C(NC(C2CC2C(F)F)=O)CCCN1C(c1cc(C(F)(F)F)cnc1O)=O c1(C(=O)NC(C2CN(C(C3CN4CCN3C(C)C4)=O)C2)C)coc2ccccc12 N1(C(CNC(CCC)=O)=O)CCC(C(F)CNC(=O)C(O)CCSCOC)CC1 C=CCCN=C(NCC1C=CCCCC1=C(C)C)N1CCc2cc(Br)cnc2C1 N1(C(CC2(C=C)CN(C(=O)C(O)C3CCC3)C2)=O)CCS(=N)(=O)CC1 c1(NC(C2CCC(N(C(=O)CCCNC(N)=O)C)CC2)=O)cc(F)c(F)cc1O C(=O)(C1=CS(=O)(=O)CCC1)NC1C(CC)CN(C(=O)C=Cc2cnc(C)s2)CC1 CC1(C)CC(CNC(C2CC(F)C2)=O)N(C(=O)COc2ccccc2)C1 C#CCC(CC(F)(F)F)C(=O)N1CCC(NC(=O)OC(C)(C)C)CC1 C12(C(=O)NC(CC=C)(C)C)CC(CN1C(=O)Cc1csc(C)n1)C2 C1(C(C)NC(CSCCOC)=O)CCN(C(=O)Cc2cnn(C)c2)CC1 C(C(O)CC(=O)N1CC(O)(CNC(c2nccnc2N)=O)C1)N(C)C C1(NC(C(C)OCC)=O)CC2CC(C1)N(C(=O)Cc1noc3ccccc13)C2 Cn1cnc2c1CN(c1nc(N3CC4CSCC4C3)nc3cc[nH]c13)CC2 c1(C(N(C(CNC(C(C=C)(C)O)=O)C)C)=O)cc(C)c2ncccc2c1C c1(C(=O)OC(C)C)ccc(C)c(S(=O)(=O)NC2CC3C(C(=O)OC)C3C2)c1 N1(C(=O)Nc2ccc(OC)c(OC)c2F)CCCC(C2CCN(C(C)=O)CC2)C1 c1(CC)cccc(C(N2CCCC(CN(C(=O)C(C)OC)C)C2)=O)c1 Cc1n[nH]c(C)c1CC(=O)NC1CCC(CCNC(c2cn(C)nc2Cl)=O)C1 c1(C(C)CNC(=O)C(C2CCC2)NC(=O)C(C)C2CC2)ccccn1 C(=O)(C(C)CCC(C)(C)C)NC1(C(=O)NCC(COCC)O)CCSC1 Cc1ccc(-c2cn(CCNC(C34CCN(C3)S(=O)(=O)C4)=O)nn2)c(C)c1 N1(C(C2C(CCC)CCC2)=O)CC2(C1)CN(C(=O)C(C1CCOCC1)C)C2 C1(C(=O)NCC(C)NC(C(C2CC(F)(F)C2)OCC)=O)CCC(=C2CCC2)CC1 c1(C(N2CCN(Cc3cc(Br)cc(Br)c3O)CC2)=O)cc(F)c([N+](=O)[O-])cc1F c1(C(N2CCC(NC(C(C)Cc3ccccn3)=O)C2)=O)ccc(Cl)cc1 N1(C(C(c2c(C)cccc2Br)NC(C2CCCOCC2)=O)=O)CC(C)(C)C12CCC2 O=C(CCCCOCCO)NCC1CC2(C1)CC2F c1(C(=O)NCCNC(C23OCCCC2C3(F)F)=O)cccc2c1OCCC2 C1(CNC(c2ccc3cc[nH]c3c2)=O)C(C2CC2)CCN1C(c1ccoc1Cl)=O N1(C(c2c(CC)onc2C)=O)CCC(CNC(c2cc(C)cc(C)c2)=O)C(O)C1 c1(C(N2CC(C)OC(C(F)(F)F)C2)=O)noc2c1CN(Cc1cccs1)CC2 CCCC(C)(C)C(=O)NC(C)C(C(C)C)NC(c1cn(C)c(C)n1)=O C(CCCCC(=O)N1CC2C(CNC(c3cc(C)cc(C)c3)=O)C2C1)OC C12(NC(COC(CC)(C)C)=O)COC(C1)C(NC(C1(n3cc(Cl)cn3)CC1)=O)C2 C1(C)(NC(C(C)Cn2ccnc2)=O)CCCN(C(c2ccc(O)cc2)=O)C1 N1(C(C(CC)OCC)=O)CC2CCCC2(NC(=O)CSc2ccccn2)C1 C1(NC(=O)CCCn2ccnn2)(CF)CCN(C(c2ccc(C3CCC3)o2)=O)C1 CC#CCCC(=O)N1CCOC(CC(=O)NCCC2CC2C2CC2)C1 N1(C(c2cnn(CC)c2C)C(=O)NCCOC)C2CCC1CN(C)CC2.C1CO1 c1(C(C)(C)C)cccnc1C(=O)NCCC1CCCN(C(c2coc(Cl)c2)=O)C1 c1(C(=O)NCC2(O)CC(NC(c3c(C)coc3C)=O)C2)ncn2c1CCCCC2 c1(C(=O)NCC2C(NC(c3c(C)ccs3)=O)C2)cccc(C2CCOC2)c1 C(=O)(C#CC1(C)CCCO1)N1C(C(=O)NCC(C)CC(F)(F)F)CC2(CCC2)C1 c1(Cc2scc(C(=O)NCC(C(C)C)NC(C3(CF)CC3)=O)c2)ccccc1F N1(C(C(C)N2CCC2)=O)CCN(C(c2nn[nH]c2Cl)=O)CC1CCO c1(CC)n[nH]cc1C(=O)NCC1(CCNC(c2cc(CO)cs2)=O)CC1 N(C=CC(=O)C(F)(F)F)C(C1CC2(C1)CN(C(c1cc3ccoc3s1)=O)C2)=O C(CN=c1ccc(Br)c(S(=O)(=O)NCCS(=O)(=O)CCCC)[nH]1)SC(C)C CCCCC(CCC)CN=C(NC1CCS(=O)(=O)C1)N1CCC2=C(CCCC2)C1 C(C)(CO)(C(=O)NCC(CNC(=O)CCCc1ccccc1)CO)OC C1(N(C(=O)C=C2CCSCC2)C)CN(C(=O)CCc2ccnn2C)CCC1O C1(N(C(c2ccc(C)cc2)=O)C)CN(C(c2onc(C)c2C)=O)CC12CC2 c1(C(=O)NCC(C)NC(=O)CCCn2ccnn2)c(C(C)(C)C)sc2c1CCC2 C1(C(N2C(CNC(=O)CSc3ccncc3)CC(O)C2)=O)CC(F)(F)C12CCC2 N1(C(C2C(c3cn(C(C)C)nc3)C2)=O)CC2(C1)C(NC(N)=O)CCS2(=O)=O CCC(C)C(C(=O)NC(C)C(C)F)N(C(=O)Cc1cc(C)on1)C c1(CC)cc(OC)ccc1C(=O)NCC(C)CN(C)C(c1cnoc1CC)=O N1(C(c2cnc(-c3ccsc3)s2)=O)CC2CN(C(C3(C(F)F)CCC3)=O)CCC12 c1(COC)nc2ccccn2c1C(=O)N(C1CCCN(C(=O)OC(C)(C)C)C1)C C#CCC(C)C(=O)NC(C1CCCC1)CNC(c1ccc(C(F)(F)F)s1)=O c1(C(N2C(C)CN(C(=O)C3=CCS(=O)(=O)C3)CC2)=O)cc(=O)c2ccccc2[nH]1 C(C(COC)C(=O)NC1(c2ccccc2)CCN(C(c2cc[nH]n2)=O)C1)OC c1(CN(C)C(=O)NCCNCc2c(C)noc2C)cccc(F)c1F C1(NC(c2nc(C(C)(C)C)oc2)=O)CC12CCN(C(=O)Cc1cccnc1)CC2 c1(C(N2CCCC2CNC(C(C=C)(C)O)=O)=O)ccc(C(=O)OCC)cc1O C1(CNC(CCc2nc(C)c(C)[nH]2)=O)CCN(C(C2C3CCC23)=O)CC1O CN1Cc2cc(NC(=O)NCC3CCNC3=O)ccc2C1=O C1(C(=O)NCC2C(CNC(c3c[nH]cc3C3CC3)=O)C2)CC1C1CCCC1 N1(C(c2cc(C3CC3)ccc2O)=O)CCN(C(c2sccc2F)=O)C2(CC2)C1 N1(c2c(C)c(NCc3cc(C(N)=O)no3)ncn2)CCCC2(CC1)CCN(C)CC2 N=C1NC(=O)C(CC(N2CC3CC2C3NC(c2ccc(-c3ccco3)o2)=O)=O)S1 C1(C(N2CC(C)(NC(=O)C=Cc3ncc[nH]3)C2)=O)(COC)C=CCC1 c1(CN(C)C(C2C(CNC(=O)C(O)Cn3cncn3)C2(C)C)=O)cccc(O)n1 Cc1nn(CCO)c2ncc(C(N3CC4COCC4(CC(=O)O)C3)=O)cc12 Cc1ccc(C(O)C(=O)N(C)CC2COCCN2C(=O)C#CC2CC2)cc1 C12(NC(c3scc(C(N)=O)c3)=O)CCN(C(c3cnc(Cl)s3)=O)CC1C2 C1(NC(C(C=C)C2CCC2)=O)CCC(C)(C)N(C(=O)C(CC)C(=O)OCCOC)C1 CCCC(C(=O)NC1CCCCC1CC(=O)N(C)Cc1nncn1C)OC CCCC(C)(C)CC(=O)N1CCN(C(C2CCCC(CF)C2)=O)C(CC)C1 C(=O)(CCCCN=[N+]=[N-])NCCC(C(=O)NCC1CCC(=O)O1)C(C)C c1(C(N2CC(Cc3cn(CC(F)(F)F)nn3)C2)=O)ccc(Br)nc1F N1(C(C(C=C)O)=O)CC2(CCN(C(c3cnc(C)nc3C3CC3)=O)CC2)C1 N1(C(c2c(C)oc(Cl)n2)=O)CC(NC(=O)CC2CCC(F)(F)C2)C2CCCCC12 N1(C(c2c(C)cnnc2)=O)CCOC(C)(CNC(=O)CCCc2cccs2)C1 C1(C(=O)NCc2ccn(-c3ccccc3)n2)CCOC2(CCS(=O)(=O)C2)C1 C1(C(=O)Nc2cnn(C3CC3)c2C)(CC)CCN(C(C2CCC3(CC3)C2)=O)C1 C(CC(F)(F)Cl)SC.C1(C2CCCC2)C(=O)N2CC(C(C)C(=O)N1)C2 c1(C(=O)OC)cc(NC(c2n[nH]c(C)n2)=O)cc(CO)c1 C1(CNC(CN2CC(C)C2)=O)CN(C)CCN1C(c1ccc(C2(C)CC2)cc1)=O c1(C(=O)NCC2(O)CC2)cc2n(n1)CCCN(C(C1(F)CCC1)=O)C2 C=C(C)CC(C)C(=O)Nc1nnc(-c2ccccc2Cl)o1 Cc1cc(C(N2CCC(NC(c3ccccc3OCC(N)=O)=O)C2)=O)ncc1Cl N1(C(c2c(C)n(C)nc2)=O)CCC2C1CCCN2C(=O)CN1CCC(C)C1 N1(C(c2c(C)n[nH]c2C)=O)CCCOC(CNC(c2ccc(C3CC3)cc2)=O)C1 C1(C)(CC)C=C(C(=O)N2CCCC2CNC(C2CC3CCC3C2)=O)C1 C1(CC=C)(NC(=O)C(C2CC2)OCC)CCN(C(=O)Cc2nccs2)C1 CC1CN(C(=O)C=CC2CCC2)CC(C(=O)N(CCCC2CCOC2=O)C2CC2)O1 c1(C(=O)NCC2C(C(N3CC(COC)OCCC3)=O)C2)ccn2cncc2c1 Cc1ccc(C(=O)NN2CC3CN(Cc4cnc5ncccn45)C3C2)cc1[N+](=O)[O-] N1(C(C2CCCC(=O)O2)=O)CCCC(O)(c2ccccc2)CC1 N(C1CCCc2c[nH]nc21)C(C(C)CNC(=O)CCc1cn[nH]c1)=O C12(CNC(c3cn(CCCOC)nc3)=O)CCC1CCN2C(=O)C1=CCOC1 C1(CC(=O)N(C2(CC(=O)N(C(C)CNC(C)C)CC)CC2)C)CCC(=O)N1 Cc1cccc(N)c1C(=O)NC1CC(F)CN(C(C2CC2CF)=O)C1 C(CN=c1[nH]c(Cl)nc2c1CS(=O)(=O)C2)c1c(C)ccc(OC)c1 c1(CNC(C2CCSC2)C)ccc2[nH]nc(Cl)c2c1 C(C)(C)(CCC(=O)NC(C(=O)NCC(=O)N(C)O)C1CCC1)N(C)C C(=O)(C(F)(F)CC(C)C)N1C2CCC(NC(C(c3c(C)noc3C)C)=O)(C2)C1 C1(NC(c2c(C)nsc2)=O)(CNC(c2cc(F)ccc2F)=O)CCCCC1C C(=O)(n1c(CC)cc(=O)n(C(=O)C(=O)OCC)c1=Nc1cc(F)ccc1C)OCC C1(C(=O)Nc2c(SCC)cccc2)CN(C(=O)C(F)C(CC)CC)CC(C)(C)C1 C(=O)(C1=CS(=O)(=O)CCC1)NCC(C1CCCC1)NC(C1(CC)CCOCC1)=O CC1CCC(CNC(=O)CC2(n3cnnn3)CCSCC2)CN1C(=O)CCF c1(C(=O)NC(C)CN(C(=O)C(C)OC2CCOCC2)C)csc(S(N)(=O)=O)c1 CCC(CCc1ccccc1)C(=O)N1CC(C(C)NC(C2CC3CC3C2)=O)C1 c1(CC(=O)N(CC(C)(C)NC(CSCC)=O)C)ccc2c(cnn2C)c1 c1(C(=O)NCc2cn(CCNC(c3cnc(CC)[nH]3)=O)nn2)csc(=NC)[nH]1 C1(NC(c2c(C)n(C)nc2)=O)CCN(C(c2ccc(C#N)[nH]2)=O)CC12CC2 C1(NC(c2nccc(CC)c2)=O)CCCN(C(C2CC(C(C)=O)C2(C)C)=O)CC1 c1(C(C)=O)cccc(NC(=O)C(=O)NC2CN(C(=O)OCC(C)(C)C)C2)c1.C(C)(C)(C)N c1(OC)ncccc1C(N1C(C(N2CC(C)C(O)C2)=O)CC2CC12)=O N1(CCN=[N+]=[N-])CCN(CCN2CC3(CC3)C2c2ccc(F)cc2)CC1 c1(C(=O)NC2C(C)(C)N(C(c3cc(Cl)sc3Cl)=O)CC2)occ2c1CCOC2 C1(CCCC(=O)N(C(=O)CS(=O)(=O)N(C)C)CCOC)CCC(C)C1(C)C c1(CC)cc(C)ccc1C(=O)NCC1C2CN(C(c3cc(O)ccc3Cl)=O)CC12 C1(CC)CCN(C(c2cc[nH]n2)=O)C1C(N1CCC(OCCF)C1)=O C(=O)(C(O)(CN(C)C)C(F)(F)F)N(CC(C)NC(C1(CO)CCCCC1)=O)C C1(NC(c2ncc(C)c(Cl)c2)=O)CC2CCC(C1F)N2C(c1cccc[n+]1[O-])=O c1(C(N2CCN(Cc3cccc(CC)c3)CC2C)=O)cc(F)cc(F)c1Br O=C(C#CC1CCCC1)NCc1cccc(NC(c2ccsn2)=O)c1 CCC(O)C(C)(C)C(=O)N1CCN(C2CCCN(C(=O)CCCN=[N+]=[N-])C2)CC1 c1(C(=O)NCCNC(C(C)OC(C)(C)C)=O)nc(Cl)ccc1OCCF C1(NC(CS(CC)=O)=O)CC2CN(C(=O)C(O)C(C)(C)CC)CC2C1 N1(C(c2c(C)oc(C)c2C)=O)CCN(C(c2cncs2)=O)C2(CC2)C1 C1(CN(C(=O)Cc2cccs2)C)C2CN(C(=O)C(C3CC3)C3CC3)CC12 CC1CN(C(=O)NCc2cc(Cl)ccc2F)CCC1(c1ccccc1)CO C1(CNC(C(CC)NC(N)=O)=O)CN(C(c2coc(Br)n2)=O)CCC1(F)F C(=O)(C(C)CC(=O)N(C1(CC(=O)NCC2(F)CCCCC2)CC1)C)OC N1(CCC2C(C)CCO2)CCSCC1CO C(=O)(CCC(O)C(C)(C)C)N1CCN(C2CCN(C)CC2)CC1.N12CCC(C1)C2=O c1(C(N2C(C)C(C(=O)NC3(C(F)(F)F)CC3)CC2)=O)ccc2cc[nH]c2n1 C1(C(N(C)Cc2ccc(CC)o2)=O)CC12CC(NC(=O)Cc1ccsc1C)C2 C12(NC(=O)C=Cc3ccsc3)COC(CNC(c3csnn3)=O)(C1)C2 C1(CNC2CC(C(=O)NC(=O)Nc3ccccc3)C2)CN(CC(F)(F)F)CCO1 CC1CCC(CO)(NC(C2CCCCN(C(c3cocc3C(N)=O)=O)C2)=O)CC1 Cn1cc(C#N)cc1C(=O)NCc1csc(C(=O)NCC2CCCC3(CC3)C2)c1 Cc1ccc(Br)c(NC(C2CC23CN(C(=O)Cn2cc(Br)cn2)C3)=O)n1 c1(CCC(=O)NC(CNC(C(CCC)OC)=O)CO)cc(C)cc(C)c1 c1(CNC(=O)NC2(n3cnnn3)CCOCC2)ccnc(-c2ccccn2)n1 O(NC(=O)C(C)(C)CCNC(=O)CC1NC(=O)NC1=O)CCCC(=O)OC C(=O)(C1=CC2CC(C1)CC2O)NC12CC(CNC(c3c(CC)noc3)=O)(OC1)C2 N1(C(C=CC)=O)CC(C2CCCN(C(c3c(Br)cc(Br)c(O)c3Br)=O)C2)C1 c1(C(=O)NC(C2CN(C(=O)C(C(C)(C)C)N(C)C)C2)C)ccc2ccsc2c1 c1(C(=O)NC2C(NC(C3(C(N)=O)CC3)=O)CCCC2)ccc2cncn2c1 C1(CNC(c2cc(C3CC3)[nH]n2)=O)C2CN(C(c3sccc3F)=O)CC12 Cc1nc2c(F)cccc2cc1C(=O)NCCN(C(c1ccon1)=O)CC1CC1 c1(NC2C(C)(C)S(=O)(=O)C2)ccc(S(C)(=O)=O)c([N+](=O)[O-])c1 c1(C(=O)NCC(CC=C)NC(c2csc(C(C)(C)C)c2)=O)c(C)coc1C CCCN=C(NCc1ccc(F)cc1OC)N1CCC(C(F)(F)F)(CC)C1 c1(CNC(C(CNC(CCCOC)=O)C)=O)cnc(C)nc1 C1(C(N(CC(CC)(C)OC)C)=O)CCC(NC(=O)CC2CCCC3CC23)CC1 c1(C(C(=O)NCCOCCNC(CC2CCN(C)C2)=O)(C)C)ccccc1Cl C1(NC(c2c(C)nc(-c3ncccn3)s2)=O)CN(C(=O)C2CC2)CCC1CO CC(C)CC(Cc1cc(C(C)C)no1)C(=O)NCC12CC(NC(=O)C3CC3)(C1)C2 C1(CNC(C(C)(C)n2ccnn2)=O)CC2(CC2)CN1C(=O)COC1CCCOC1 N1(C(C(C)N2CCC2)=O)CCC(NC(c2occc2CN2CCOCC2)=O)C1C C(=O)(CCCS(N)(=O)=O)N(C)CC1OCCN(C(CC2CCC(C)CC2)=O)C1 N1(C(C(C)(C)c2ccncc2)=O)CCN(C(C2CCCS2(=O)=O)=O)C(C2CC2)C1 c1(C(N2C(C(C)NC(c3c(SC)n(C)nc3)=O)CCCC2)=O)ccc(O)c(Cl)n1 c1(CCN=C(NC(C=C)C)NC2CC23CCCCC3)cccc2cc[nH]c12 CC(C)CC(C(=O)NC1CN2CCC1C2)ONC(c1cccc(Br)c1)=O c1(C(=O)NC2CCN(CC)C2)cc(-c2cccc(C)c2OC)c2n[nH]cc2c1 Cc1cn(C(C)C)cc1C(=O)NC1C2CN(C(C3(C(=O)N(C)C)CC3)=O)CC12 C(=O)(C#CC(C)(C)CNC(=O)CC1(C)CCOCC1)Nc1ccc(OC)c(C)c1 c1(C(N(C2CN(C(C(C)CF)=O)CC23CC3)C)=O)n[nH]c2cccnc12 Cc1nc(N(C2CCCNC2)C(C2CCC(O)CC2)=O)c2cc(Br)ccc2n1 C(=O)(C(=O)CC(C)C)N1CCC(C(=O)NC(c2ncn(C)n2)C)(OC)C1 C=CC(CC)CC(=O)N(C1CN(C(c2c[nH]nc2[N+](=O)[O-])=O)CCC1O)C N1(C(C2CCCN(C(C)=O)C2)=O)CCC2C(C1)CN2C(c1cnc(O)c(F)c1)=O Cc1c(C(N2CCCC(C)C2CNC(=O)C(C)C)=O)sc2ccccc12 Cc1cc(C(=O)NC2CC3CN(C(C4CN5CCN4CC5)=O)CC23)cnc1O c1(OCCC(=O)NCC(C)CNC(C2CCC3(CC3)C2)=O)ccc(Cl)cc1Cl N1(CC)CC(NC(=O)C(C2CCN(C(=O)CCC3OCCO3)C2)C)C(C)C1 C(=O)(CC(C(F)F)NC(=O)C(C)c1ccco1)NCc1c(C)nc(C)o1 C#CCCN=C(NCc1cc(F)ccc1CS(N)(=O)=O)NCC1CC1CC N1(C(CC(=O)NCC2CC2)=O)CCOC2CCN(C(C3(F)CCCC3)=O)CC12 N1(C(C)=O)CCC2CN(C(C3(C)C=CCC3)=O)CCC12 C(=O)(C1=CC2(CCN(C(c3nc[nH]n3)=O)C2)C1)NCCC(CCC)C1CC1 N1(C(c2cc(C)sc2N)=O)CCCC(C)(NC(C2CN(C(C)C)CCO2)=O)C1 CC1=C(C(=O)NC(CNC(C2CCS2(=O)=O)=O)C2CC2)CC1 C#CC1CN(C(=O)COC2CCC2)CCN1C(=O)C=C(Cl)Cl C1(N(C)C)(C(=O)NC(CNC(c2ncc[nH]2)=O)C2CC2)CCOCC1 N1(C(C(C=C)(C)C)=O)CC2CC(C1)CN(C(C1CNC(=O)CC1C)=O)C2 CCCCC(O)C(C)C(=O)N1CC(O)CC1(C)C(N1CCC(CO)(OC)C1)=O C1(NC(CC=CC)=O)CC(O)CN(C(c2ncncc2Cl)=O)C1 c1(CCC(=O)NC(CC)CNC(C2(CCOC)CC2)=O)ccc2ncsc2c1 c1(CNC(=O)CC2CCCN2c2ncnc3[nH]ccc23)c(F)ccc(F)c1O C=CCCC(C(=O)Nc1ccc(OC)nc1)NC(=O)C=CCCCSC n1(CC)nc(C(N2CC(F)CC2CNC(c2cnsc2C)=O)=O)c(Br)n1 c1(OCC)cc(N)c(Cl)cc1C(=O)NCC=CCNC(C1(F)CCOC1)=O CCCCCCCCNC(c1ccc(COC)[nH]1)=O.c12cc(ncn1)CN2 N(C(=NCCC(C)=O)NCc1c[nH]nc1C)C1CC(OC)C12CCC2 C1(C(=O)NC(C(C)C)CCN(C)C(C2(Cl)CC2)=O)CCc2ncncc2C1 c1(C(=O)NCC(CNc2nccc(CC(=O)OC)n2)O)ccc(C)c(C)c1 CC(CCCNC(c1cn(-c2ccccc2)nn1)=O)NC(c1ncc(Cl)s1)=O Cc1ccc(C2C(NC(=O)CN(C)C)C2)c(C)c1 C1(C(=O)OCC)CCN(C(=O)Oc2scnc2-c2ccccc2)C2CCCCC12 c1(CC(N2CCC(C(=O)NC3CC3COC(C)=O)(CC)C2)=O)c(C)cccc1C CC1COCCC1C(=O)NCC=CCNC(c1cnn(C2CCC2)c1)=O.C1(C)CC1 C1(NC(CN(CC#C)C(C2(SC)CC2)=O)=O)CCC(CC(N)=O)CC1 Cc1cc(C#N)cnc1C(=O)N(CC(C)(C)C(=O)NC1CCCCNC1=O)C Cc1nc(=NC(=O)CCN(c2cccc(Cl)c2O)Cc2ccccc2)o[nH]1 C(=O)(C(C)(C)CN(C)C1CC1)NC(=O)NCCCC(C)CC1(OCC)CC1 C(C)(C)(CC(F)(F)F)NC(C(C)N(C(C(C)NC(CC)(C)C)=O)C1CC1)=O C=CC1CN(C(=O)CCOCCNC(c2cccn2CC)=O)CC1O CCC(C)C(C)C(=O)N(C1CCN(C(=O)C=CSC)CC1)CC1CC1 CC(CC(N)=O)C(=O)NC(C)(C)CNC(c1cnccc1C(F)F)=O CC1CCN(C(c2cscc2C#N)=O)CC1CNC(c1cncnc1C1CC1)=O Cn1nc2n(c1=O)CCN(C(=O)C(=O)NCC1CC3(CCC3)CO1)C2 CC1(C)CCC(CC(=O)NC2(C(=O)NCC3(N(C)C)CCCCC3)CC2)C1 C=CCC(F)(F)C(=O)NCC1CC2CN(C(=O)C(C)SC(F)(F)F)CC12 N1(C(c2ccc(C(=O)OC)s2)=O)CCC(CO)(NC(c2n[nH]cc2[N+](=O)[O-])=O)CC1 c1(-c2nc(C)nn2C)cn(CCN)c(=O)nc1O c1(NC)ccc(C)c(CN2CCC(NC(=O)OC(C)(C)C)CC2)c1 N1(C(C(CCOC)C)=O)CC(C(=O)NCc2cnccn2)C2(CC2)C1 C(=O)(C(C(C)(C)C)OC)NCC(=O)NCC(CNC(CC)=O)CO CN1N=C(CC(=O)NCC23CC2CN(C(C2(C(F)F)CCC2)=O)C3)CC1=O c1(C(N2C3CC(CNC(C4(OC(C)=O)CC4)=O)C2CC3)=O)cc2occc2n1C C1(C)(CNC(c2ccc(COC)cc2)=O)CN(C(=O)CC(C2CC2)C2CC2)CCO1 C12(C(=O)O)CCCC1N(C(=O)CCc1ncc(-c3ccccc3)o1)CCC2 Cc1cnc(N2CCCC2CNC(c2c(C(F)(F)F)cccc2F)=O)nc1C C(=O)(C(C1CCCO1)NC(=O)CNCCC#N)NCCN(C)C(N)=O N1(c2nnnn2C2CCCC2)CCN(C(=O)CC2CCC2C(F)(F)F)CC1.CC(C)(C)O C(=O)(C1=CC2CCCCCCC12)CCN1CCN(c2ccccc2)CC1.O=C1NC1 CC(C(=O)NCC1CN(C(=O)CCc2ccco2)CCO1)C(F)F C12(C(=O)NCC(C)N(C(C(C)=CC)=O)C)CCC(O1)c1ccccc12 n1(CCC(=O)NC2(CNC(C3(F)C(C)OCC3)=O)CCOC2)ccc(O)nc1=O C(=O)(CC1OCc2ccccc21)N(C(CCNC(c1cn(C(C)C)nc1)=O)C)C C1(C(C(=O)NC2CCC(CNC(c3c(C)snc3)=O)C2)(C)C)CCCCCCC1 N1(C(CCc2ccc(C)o2)=O)CCCC(NC(c2ccsn2)=O)C1 C12(CNC3ON=C(C)C3)CN(C(C3(N4CCOCC4)CC3)=O)CC1CCO2 C1(NC(c2cc(C)nn2C)=O)CCC2CCN(C(=O)CCCC3CC3)C12 C1(C(N2CC(C)C(NC(=O)Cc3cn[nH]c3)C2)=O)CC(C)(C)OC1(C)C O=S(=O)(c1ccc(NCC(O)CF)c(Cl)c1)NCC(O)C(F)(F)F C=CC(C)CC(=O)N1CC2CC1C2NC(=O)Cc1ccccc1C C1(CCc2cn(C(c3nnc(C)o3)C)nn2)CN(C(=O)C(=O)OC(=N)O)CCO1 N1(C(C2(N)C(CC)CC2)=O)CC(O)C(C#N)C1 c1(C(C(=O)C(O)C(F)(F)F)=O)coc(=O)c2ccccc12.C12(N)CC1CN(C=O)C2 C#CCCC(C(=O)N(C(CC(C)C)C(N)=O)C)NC(=O)CCN(C)C C#Cc1cnc(C(=O)NC(C2CC=CCC2)C(N2CCC(CF)CC2)=O)c(C)c1 C1(NC(c2nc(CC(C)C)sc2)=O)CN(C(C2CN(C)CC(C)O2)=O)CC1(C)C C1(C(=O)NCC(CC)(C)O)(CC)CCCN1C(c1cncn1C)=O c1(N(C)CC2CCN(C(c3ncn(CC)n3)=O)C2)ncnc2c1SCCC2 c1(CC)cnc(C)c(NC(=O)C(c2cn(C)nn2)NC(=O)CCC(C)=O)c1 c1(C(N2CCN(C(CCC3(C)CC3)=O)C(C(C)(C)C)C2)=O)cnc2ccnn2c1 C#CC1CN(C(=O)Cn2[nH]cnc2=N)CCN1C(C1OCC2CCCC12)=O c1(CN2CCC(C(C)NC(Cc3ccc(C)nc3)=O)C2)ccc(F)cc1C CCC(CC(=O)N1CCCC(c2n[nH]c(CNC(=O)CCF)n2)C1)C(C)C S(=O)(=O)(c1cccnc1)N1C(C(N2CCCC(N3CCCC3=O)C2)=O)CCC1 c1(C(=O)OC)cc2n(n1)CCCN(C(c1cccc(Br)c1[N+](=O)[O-])=O)C2 C1(OC)CN(C(c2nsnc2O)=O)CC1NC(c1cccc(-n2cncn2)c1)=O c1(C(=O)NC2(CNC(C(C)N(CC)CC)=O)CCC2)cccc2ccnn12 CC1=NN(C)C(=O)C1CC(=O)NCC1(CO)CCN(C(=O)C=C(Cl)Cl)CC1 C#CCC(CO)NC(=O)CCNC(=O)CCc1cnco1 C1(C(=O)NC2CN(C(Cn3nc(C)c(Cl)c3C)=O)CC2O)CCn2ccnc2C1 N1(C(C(C)NC(=O)COC2CCCC2)=O)CC2CCC(C1)C(=O)O2 c1(NC2CCCN(C(C(C)Oc3cc(Cl)cc(Cl)c3)=O)C2)cc(O)nc(O)n1 c1(C(=O)NCC2CC(F)(CNC(c3c(CC)nn(C)c3)=O)C2)c(OC)ccnc1F C1(C(=O)NC2CC(N(C(CCCOCC=C)=O)C)C2)CCn2nnnc2C1 N1(C(CCC(=O)NCC)=O)CC(CO)C2(C1)CN(C(=O)C(c1cccnc1)O)C2 C1(C)(CNC(CC2CC(C(=O)OCC)C2)=O)CSCCO1 c1(N2CC(CF)OCC2)nc2c(c(=NC3CCC4CCC34)[nH]1)SCC2 CC(CC(=O)NC1(CF)CCN(C(=O)C(F)=C2CCCC2)C1)C(F)F C1(NC(C2CCC(C)O2)=O)C2CC3C(C2)C13C(=O)NC1CC(O)C(F)C1 c1(C(=O)OC(C2CC2CCN(CCO)Cc2ccccc2)=O)ccnc(C2CC2)n1 c1(C(N2CC(CNC(C(CCCOC)C)=O)C2)=O)nccc(Br)c1O c1(C(C(=O)NCC(CN(C(CN2CC(CC)C2)=O)C)C)C)ccn(C)n1 C12(C(=O)NC(CC)(C)CO)CC1CN(C(=O)CC=CC(C)(C)C)C2 Cc1cc(=O)n(C)cc1C(=O)NCCCCCNC(C1CCC(C)(F)CC1)=O N1(C(Cc2c(NC(c3ccc(OCC)nc3)=O)cccc2)=O)CC2COCC2C1 c1(NC(C2CC2F)=O)c(SC2CCN(C(=O)Cn3ccnn3)C2)cccc1F S(=O)(=O)(c1ccc(=NCC2CC23CCC(F)(F)CC3)[nH]c1)NC(CC)C C(=O)(C(C)(C)C1=CCSCC1)N1CC(CC(C)NC(=O)C(F)C(C)(C)O)C1 N1(C(c2c(C)onc2)=O)CCC(C)C(NC(=O)C=Cc2ccc(C3CC3C)s2)C1 CCC(C)CCC(=O)NCC(C)(CO)NC(=O)CCc1cc(Cl)no1 C=CCCC(C)C(C(=O)NCCCC)N(C)Cc1ccsc1 N1(C(CCCC#CC)=O)CCC(F)(F)C(CNC(=O)CC(O)CN(C)C)C1 N1(C(c2nc(C(C)C)oc2)=O)CCCC(NC(=O)CCc2cccn2C)C1 c1(C(N2C(C(=O)NC(C=C)(C)C)C=CC2)=O)cc2ncccc2[nH]1 CC1Oc2ccc(NC(=O)CN3CCc4ccc(C(=O)O)cc43)cc2NC1=O c1(CC(=O)NCC(C)N(C(=O)CC2CSCCS2)C)cccc(C#N)c1 C#CC1(C(=O)NC2CCC(=O)N(CC)C2)CCN(C(=O)CCCn2ccnc2)C1 c1(C(=O)NCC(C)NC(c2cc(C(C)=O)c(O)cc2)=O)cnc2cccc(C)n12 Cc1ccc([N+](=O)[O-])cc1C(N1CC2CC1CC2NC(c1ccco1)=O)=O Cn1cnc2[nH]c(=NCC3COCC3CO)nc(N3CC4CC4(CO)C3)c12 C(C(C)N=c1cc(C)[nH]c(=NCCCC(=O)OC(C)C)[nH]1)c1ccc(OC)cc1 C1(CNC(c2cc(C)n(C(C)C)n2)=O)CCN(C(C2CCCCC2O)=O)C1(C)C C(=O)(C1CCS(=O)(=O)c2ccccc21)NCC1CN(C(CC(CC)C(C)C)=O)C1 C(=O)(C(C)C(C)C)NC(C1N(C(c2c(C)nc[nH]2)=O)CCC1)C c1(C(=O)NCC(CC=C)NC(c2c(C)cnnc2O)=O)cc(N)cc(F)c1 c1(CC(=O)NC2CCC(NC(C3(C(C)C)CCCO3)=O)C2)cc(F)c(N)cc1F C(=O)(C1CCCn2cnnc21)NC1CCC(NC(c2ccc(CO)nc2)=O)C1 Cc1nc(C2CC2)nc(C)c1C(=O)NC1CN(C(C2CN3CCN2CC3)=O)C1 C1(C)(C(=O)NCc2nc(C)c(C)[nH]2)CCCN(C(=O)C(C)O)C1 N1(C(C2(SC)CN(C(c3ccc(CC)o3)=O)C2)=O)CCCC(F)(F)CC1 C#CCCN=C(NCC(=O)OC(C)(C)C)N1CCC(O)C(CO)C1.C1CCN1 CC1CCN(c2nnco2)CC1NC(c1cccc(Cl)c1Cl)=O C1(C(=O)NC2(C(=O)NCCC(C=C)C)CC(CO)C2)COCCN1C C(c1cccc(F)c1F)=CC(=O)NC1CCC(NC(c2c(C)scn2)=O)CC1 c1(NC(C)=O)ccc(C(N2CC3C(CNC(C4(O)CCOC4C)=O)C3C2)=O)cc1 CC1=C(C(=O)NC2CN(C(=O)CC3CC(F)C3)CCC2F)CCO1 C(=O)(C1=CCCOC1)NCC(C1CCCN(C(CCN(CC)CC)=O)C1)(C)O CC1CC(C(N2CCCC2C2CCN(C(c3cn[nH]c3)=O)CC2)=O)CC(C)(C)C1 C(=O)(CCCN=c1[nH]ccc(=NC(CF)CF)[nH]1)N(c1c(OC)cccc1)C N1(C(C(CC)(C)CNC(=O)CC(COC)COC)=O)CCCOC(C)(C)C1 C1(NC(C2(C=C)CC2)=O)CCCOC1C1CCN(C(=O)C=CSC)CC1 CC(C)CCCCC(=O)N1CCCC(O)(CCNC(C2CC3(C2)CC(C)C3)=O)C1 c1(OC)cc(C(=O)NC2CC2NC(=O)C=Cc2cccs2)ccc1C#N C(=O)(C(C)(C)CN(C(=O)CC(=O)N(C)C)C)NCc1n(C(C)C)ccn1 Cc1cc(N2CCC(c3nc(C)no3)C2)nc(C(C)C)n1 Cc1nc(C(=O)NCC2CCCN2C(c2cc(C(F)(F)F)ccn2)=O)n(C)n1 C(=O)(C(C)(CO)NC(c1scnc1Cl)=O)NC(c1cnn(CCF)c1)C N1(C(C(C)CC(N)=O)=O)CCCC2CN(C(=O)CCCN(C)C)CCC12 c1(NC(C)=O)ccc(F)c(C(N2CCCC(CO)(NC(=O)C(C)C3CC3)C2)=O)c1 C(=O)(C(O)CC(F)(F)F)NC1(C(N2CC(CC(=O)OC)C2)=O)CCC(C)(C)C1 C=CCCC(C)(C)C(=O)NC(C1CCCCN1C(c1[nH]c(C)nc1C)=O)C N1(C(C2CCCC(=O)N2)=O)CCOC(C(=O)NC2C=CCCCC2)CC1 CC(CCCNC(=O)COCC(c1ccccc1)C)NC(c1csc(C2CC2)n1)=O C1(C(=O)NC(C=C)(C)C)CN(C(C2CC(OC3CC3)C2)=O)CC1F c1(CCNS(N(CC)CC)(=O)=O)c[nH]c2c(Cl)cc(F)cc12 S(=O)(=O)(c1cnn2ccc(=NCCC(F)F)[nH]c12)NC(C=C)C1CCC1 c1(NC(Cc2c(C)ccnc2)=O)ccc2c(c1)CN(C(=O)C(F)(F)C(F)F)CC2 N1(C(C2N(CC)CC2)=O)CCC(C)(CC(=O)NCC(C2CC2)OC)C1 c1(C(=O)NC(C)C(C)NC(c2cnc(O)o2)=O)c[nH]c2cc(F)ccc12 Cc1ccc(C(N2CCN(C(=O)CSC(C)(C)C)C3CC23)=O)c2c1CCCN2 c1(C(=O)NC2CCN(C(C(CC=CC)C)=O)CC2O)cc([N+](=O)[O-])ccc1O N1(C(CSc2n(C)nnn2)=O)CC2CCN(C(C3CCNC(=O)C3)=O)CC2C1 C12CCN(CCC1C)CC=CC2.C1(C(NOCC=CC)=O)C2CC3C(C2)C13 C#Cc1ccccc1COC(=O)CC=CC1CCC(CNS(=O)(=O)C(F)(F)F)C1 CC(C)(CNC(c1ccc(C(F)F)o1)=O)CCNC(=O)C=CC1CC1 C(=O)(C(F)(CNC(=O)CC1(N(C)C)CCC1)C(C)C)NCCC(C=C)(C)C C(C(F)F)(C(C)(C)C)NC(C(c1ncccc1F)C)=O.C12C(C1(C)C)NC2=O C1(CNC(c2cc3ccccn3c2)=O)CCCC2CN(C(c3cncs3)=O)CC12 C1(F)(CN(C(=O)CC2CCOC2)CC)CCN(C(=O)CN2CCC(O)CC2)CC1 N1(C(C(C)(C)SC)=O)CCN(CC2CN(C(c3nsnc3O)=O)C2)CC1 N1(C(C(F)=C(C)C)=O)CCC2(CC1)CCN(C(C1CN3CCCC3CO1)=O)CC2 N1(C(CCCCCCC)=O)CCOC2(C1)CN(C(=O)C(C)C(=O)OC)C2 C(C(C(=O)NCCN1C(=O)CNC1=O)C(C)(C)C)NC(c1n(C=C)ncc1)=O c1(SC)cc(C)c(C(=O)NC(C)CNC(C2CC=CCC2)=O)s1 c1(OC)c(C)cc(C(=O)NC(CNC(C2CCCC3(CCC3)O2)=O)CO)cc1C O=C(CCC[N+](=O)[O-])NCC1C2CN(C(=O)CSc3cc(F)ccc3F)CC12 CC(Cc1cccc(F)c1)N=c1nc(N2CCC(C)(C)C2)c2c([nH]1)CCC(C)C2 CC(C)CC(C(=O)N1CCCC(CCC(=O)NC2(CO)CCOC2)C1)C(N)=O Cc1ccc(C(N2CCC(NC(C3CCSC3)=O)C2(C)C)=O)cc1C CS(=O)(=NC(=O)CCNC1CC1)c1cnn2c1CN(c1ncnc(Cl)c1Br)CC2 Cc1cc(C(N2CC3CCC2CN3C(C2(C)CNC(=O)C2)=O)=O)c(C)nc1C N1(C(c2c(NC)cccc2)=O)C2CCC(C2)C1C(N1CC(n2cnnc2)C1)=O Cc1cc(C(N2CC(N(C)C(c3[nH]cc4c3CCC4)=O)C(F)C2)=O)ccc1Cl Cc1ccc(C(=O)NCC2CCCN2C(C2CC3C=CC2C3)=O)c(C(C)C)n1 C=CCC(CC(=O)NC(C)CC(C)(C)O)NC(C1(C=C)CCCCC1)=O c1(C(CC(=O)NC(c2nccc(=N)[nH]2)C)N)cccc(F)c1 c1(N(C(C2CCCO2)C)C)nnc(C2COCCN2C)n1CCOCC1CCOC1 CC(C)CC(C)C(=O)NC(C)(CNC(c1c[nH]cc(Br)c1=O)=O)C1CC1 C1(NC(CNC(CC(C)(C)C)=O)=O)CCCC12CCN(C(=O)Cc1cccs1)C2 C=CC(CC)C(=O)N1CCC(C(=O)N(CC(O)C2CC2)C)(CO)C1 c1(C(=O)NC2CC(CCC(=O)NCC3CC3Cl)C2)ccc2ccoc2c1 c1(C(CF)NC(N(c2cccc(OCF)c2)C(C)C)=O)ccc2c(c1)OCO2 N1(C(C2(C#C)CN(C(c3csnc3Cl)=O)C2)=O)CCOC(C)C1CO N1(C(c2cc(C)oc2)=O)CCC2CN(C(=O)Cc3c(O)ncnc3O)CCC2C1 C(=O)(C1=COCCO1)NCC1(COC)CN(C(=O)C(c2ccc(F)cn2)(F)F)C1 c1(C(N2CC3C(CC(=O)NC(CCCC)C)(CC3)C2)=O)c[nH]c2cccnc12 CC(C)C(CCNC(C1(C)CCOCC1)=O)NC(=O)CSCCC#N c1(C(C)C)nocc1C(=O)N(C)CCNC(C1CC2CC2C1)=O c1(NCc2c(COCC)cccc2)cc(S(C)(=O)=O)cc(Cl)c1Cl n1(CC)nc(C(N2CCC(N(C)Cc3cccc(Cl)c3)C2)=O)cc1C(F)(F)F c1(NCCc2ccc(C)cc2)ncccc1S(=O)(=O)NC1CC(C)CC(C)(C)C1 N1(C(CN(CCC)C)=O)CC2CCC1C(CNC(=O)Cc1ccccc1F)C2 C1(NC(c2cnc(C(C)O)s2)=O)CCCC(NC(=O)C(C)(C)NC(N)=O)C1 N1(C(C2(C#C)CCN(C(=O)C(C)C(C)(C)C)C2)=O)CC2CCCCC2C1C C12COC(C1)CNC2=O.c1cc(CC2CC2)on1.C(C(=O)N)(OC)OCC c1(NC(C(=O)NCC(CC)Oc2c(OC)noc2C)=O)ccc(F)cc1 CC1=CC(C)=NS(=O)(=O)N1CC(=O)NCC(O)CNC(c1cc2n(n1)CCC2)=O C1(NC(c2c(C)coc2C)=O)CN(C(=O)C(C)n2cncn2)C2(CCCC2)C1 C1(CO)CN(C(c2cc(OC)n(C)n2)=O)CC1NC(=O)CN1CCCOC1=O N1(C(CC2N(C(C)C)CCC2)=O)CC(NC(c2ccc(Cl)cn2)=O)CCC1C C1(CN(C2CCN(C(C34CC(C(=O)NC)(C3)C4)=O)C2)C)CC(=O)N(C)C1 C=CC(O)C(=O)NC1CCCC1CNC(=O)CC1(O)CCCC1 CN1CC2CC(C1)N(C(c1ccc(CN3CCNC3=O)cc1)=O)C2 CCCC(C)CC(=O)NCCCCN(CCCNC(=O)Cc1cccn1C)C O=C(N=c1ccn(C(F)F)[nH]1)c1ccc(CC(=O)NCCCC2CC2)c(Br)c1 C1(NC(C)=O)CC2(CCCN(C(C3CC3c3ccc(C#N)cc3)=O)C2)C1 Cc1nn(CC(=O)NC2CN(C(C3CCC(C(N)=O)O3)=O)CC2(C)C)c(C)c1Cl C1(CNC(C(C)N(C)C)=O)CN(C(c2n[nH]cc2Cl)=O)C2COCC2O1 N1(C(C2(OC)CCCOC2)=O)Cc2[nH]nc(C(=O)N(C)CCF)c2C1 N1(C(c2cc(OC)ncc2)=O)CCC2CCN(C(=O)COc3ccsc3C)C2C1 C(=O)(CC(O)CNC(=O)C(C)CN(C)C)N(C(CC)CC)C C(CCN=c1cc(C)nc(OC)[nH]1)N(C(C(C)OC)=O)C c1(CNC(C2CSCCN2C(c2cc(Cl)sc2Cl)=O)=O)ncccc1Cl N1(C(C(C)OCCCC)=O)Cc2[nH]nc(C(N3CCC(C)C3COC)=O)c2C1 N1(C(CCC(C)OC)=O)CCN(C(c2cccnc2)=O)CC1CN(C)C C1(OC)CN(C)CC1N=c1[nH]c(=NCCCc2ccnc(O)c2)[nH]c2c1COC2 C12C=CCN(C1)C(=O)N2CC(F)F.CC(O)COC(=O)OC(C)(C)C C1(C(=O)NC(CC=C)(C)C)CCCN(C(C2(CO)CCCO2)=O)C1 C1(OCCCC)(CN(C)Cc2cnc(OC)s2)CC1(C)C C12(COC)CC(CNC(=O)C(C)SC)(CN1C(=O)CCc1ccccc1F)C2 c1(COC(c2ccc(C)cc2Br)=O)ccc([N+](=O)[O-])cc1Br C1(CC(N2CC(CC(=O)NC(c3ccccc3)C)C2)=O)NC(=O)NC1=O CC1CCN(C(c2cc3occc3[nH]2)=O)C(C(=O)NCC2CCC=CO2)C1 C(CC(C)C(=O)N1CCC(C(=O)N(CCC(N)=O)C)C1C)OC c1(C(=O)NCC2N(C(CNC(N)=O)=O)CCCC2)nc[nH]c2ncnc1-2 N1(C(c2c(C)nncc2)=O)CCC(NC(c2ccnc(F)c2F)=O)C12CCCC2 C(=O)(C(CCC(N)=O)N(C)C)NCC1N(C(Cn2c(C)csc2=O)=O)CCN(C)C1 c1(C(=O)NC2(CC)CCOC2)c([N+](=O)[O-])cnn1C N1(C(c2cncc(C=C)c2)=O)CCC(C(=O)NCc2ccccn2)C(C)(C)C1 C1(OCC)(OC)CC(C)(c2nc(C(F)F)nn2C2CC(OCC)C2)C1.C(C)(C)OO C(=O)(C(c1ccccc1)=C(C)C)N1CC(NC(C2C(CCC)C2)=O)(CO)C1 C1(NC(=O)CN(C)C)CCN(C)CC1C.c1(CCC)ocnc1C(=O)OC N1(C(C2CC(=O)OC2)=O)CCC(F)(CNC(=O)C(F)(F)C2CC2)CC1 C1(C(=O)N(C)C)(COC)CC=CCC1.C12CC(C1)CCNC(=O)C1(CCC1)C(=O)N2 N1(C(CCN(C(=O)Cc2cccs2)CC#C)=O)CC=CCC(C)(C)C1 C1(CNC(CCCOC)=O)CN(C(=O)Cc2cn(CC)nn2)CC(C)(C)C1 C(=O)(CC1OCCc2ccsc21)NCCCN(C(CCC(=C)C)=O)C c1(OCC)c(CC(=O)NC2CC(N(C)C(C3CCCC(C)O3)=O)C2)cccc1Cl C(=O)(CCCC(=O)N1CC(NC(=O)CCn2ccnc2C)CC1C)OCC c1(SC)cscc1NC(=O)CC(C)N(C(=O)C(CO)NC(N)=O)C C1(CNC(c2cc(Cl)sc2Cl)=O)C2CCCC1N(C(=O)CC1CC=CC1)C2 c1(C(N(CC(C)CNC(=O)CCC2CCC(=O)C2)C)=O)ccnc(C(C)(F)F)c1 c1(C(N2C3C(NC(c4c(C)sc(O)n4)=O)CC(C3)C2)=O)ccc2c(c1)C(=O)NC2 Cc1sc(Cl)c(C(=O)NC2(CO)CCCN(C(C3CCCCC3O)=O)C2)c1C Cc1cc(O)c(F)cc1NC(C1CN(C(c2[nH]cc(C)c2C)=O)C2(CCC2)C1)=O c1(OC)cc(CC(N2CCC(CNC(=O)COCCCF)C2)=O)ccc1O c1(NCCN(C(=O)C(c2ccccc2)F)C(C)(C)C)nccc(CO)n1 C1(NC(c2c(C)onc2C(F)(F)F)=O)CCC(C)N(C(C2C3CCCCC23)=O)C1 CCC(C)(C)C(C)CC(=O)NCC1C=CCN1C(=O)CSc1ccc(OC)cc1 c1(C(=O)NCCCCN(C(C(c2cnccn2)C)=O)C)ccc(F)c2ccsc12 CC1CC(C(=O)NCCC2CCCC2(C)C)CN(C(=O)CCc2ncccn2)C1 C1(CNC(C(C=CCCC)O)=O)CC12CCN(C(=O)C=C(C1CC1)C1CC1)CC2 Cc1ccc(C=CC(N2CCC(C)(NC(=O)C3=CCCOC3)C2)=O)cc1C N1(C(C(C(C)C)c2cn(C)nn2)=O)CCS(=O)(=O)N2CCOCC12 CC1=C(C(=O)NCC2(C)CCN(C(=O)CCc3ccccc3)C2)C(=O)OC1(C)C CCC(C)(O)C(=O)NCC1(NC(c2cc(C3CCC3)no2)=O)CC(F)(F)C1 c1(NC(C(=O)N(CCNC(c2c(CCC)nns2)=O)C2CC2)C)ccc(C)cc1 c1(C(N2C(CNC(c3ccc(C)nc3O)=O)CC2)=O)nc2ccc(F)cn2n1 C(CS(N)(=O)=O)N(C(C1CC(C(C)NC(=O)OC(C)(C)C)C1)=O)C c1(C(C2CC2)NCCNC(C(CC)OCC)=O)ccc(C(F)(F)F)cc1 CC#CCC(CO)NC(c1cc(CNC(=O)C(C)CC#N)cs1)=O Cc1c(N)ccc(C(N2CC(F)(F)CC2(C)CNC(c2cncn2C)=O)=O)c1Cl c1(C(N(CC(C)NC(C2(O)CC2(C)C)=O)C)=O)cnn2cccnc12 C(N=C(NC(C)C)N1CC(C)CC(C)C1)c1c(CC)ccc(OC)c1 CC1(C)CC(n2ccnc2-c2cccc(C(F)(F)F)n2)C(=O)N1 C1(NC(C2CN(CCC)C(=O)C2)=O)CCN(C(=O)Cc2csc(CC)n2)C(C)C1 c1(CC(=O)N(C(C)CNC(=O)CNC(=O)CC(C)(C)C)CC)ccc(O)nc1 c1(CC)ccc(O)c(CN2CCC(F)(C(=O)Nc3cccc(C)c3OC)C2)c1 Cc1cc(N)ccc1C(N1CCC(CN(C(=O)CN2CCN(C)C(=O)C2)C)C1)=O c1(CC(C)OC)nc(-c2ccc(Sc3ccccn3)nc2)n(CC)n1 c1(NCCC(C)N(C)C)nccc(=NCc2ccnc(NCCn3ccnc3)c2)[nH]1 C1(NC(CC(CC)CC)=O)CC2CCC(C1)N2C(c1cncc(OC)n1)=O c1(OC)cc2[nH]ncc2cc1C(=O)N(CCC(C)(C)c1ccccc1)C CC1CCN(C(=O)Cc2cc(O)no2)C1c1cn(CCO)nn1 c1(OC)cc(C(=O)N(C)C(c2nc(CSC3CC3)no2)C)ccc1C O=C1NCc2ccc(C(N3CCC(NC(=O)CC(F)(F)C(F)F)C3)=O)cc2N1 C1(C)(NC(C(CCC)NC(=O)COCCCN(C)C)=O)CCCC(C)(C)C1 CCS(=O)(=O)C=CC(=O)N1CCC(C(C)NC(=O)CC2=CCCCC2)C1 CCC(CC)CN=c1[nH]c(=NCC2(C)CC3CC3C2)c2cccc(F)c2[nH]1 CCC(CCC(=O)NCC1CC(C)=NO1)NC(=O)CCCOC(C)C C1(CC=C)(NC(=O)C=CCN(C)C)CCCN(c2ncc(OC)cn2)C1 c1(C(C(N2CC3(CC(NC(C(C=C=C)C)=O)C3)C2)=O)C)cccc2ccccc12 C1(CC=C)(NC(c2cc(Br)co2)=O)CCCN(C(=O)CCCCOC)C1 C1(CC)CN(C(C23CCC(C2)C3(C)C)=O)CCC1NC(=O)CCCC1CC1 C(=O)(CC(C)CF)N(CCCNC(=O)C(F)(F)c1csc(C)c1)CC C1(C(=O)NC2C(OC)CN(C(=O)C(C)(C)CN(C)C)C2)CC2CCC1C21CC1 Cc1ccc2c(c1)CCC(C(N1CC(NC(c3ccn4nccc4c3)=O)C1)=O)O2 c1(C(=O)NC2C(NC(Cc3c(C)noc3C)=O)COCC2)ccc(F)c(F)c1O Cc1ncc(C(=O)NCC2CC3CCC2N3C(=O)Cc2ccccc2C)c(C)n1 c1(C(=O)NCCC(C(C)C)NC(=O)CC(O)C2CC2)nccc2occc12 c1(C(=O)NCC(C)(CO)NC(c2cnn(C(CC)C)c2C)=O)ccc(F)c(F)c1 C(=O)(C1=CCCSC1)N1CCN(C2CCCN(C(C3CCC(C)CC3)=O)C2)CC1 C1(CC(=O)NCCS(CC)=O)CCCCN1C(=O)CCC c1(C(=O)NC2CC(NC(C3CCOC3)=O)C23CCC3)ccc2[nH]ccc2c1 C1(C(NOCC=CC)=O)CCCC(NC(=O)C(C)SC2CC2)C1 c1(C(C)C)ccc(C(=O)NCCCCCCNC(C2CCCS2)=O)cc1Cl C(=O)(CC(C)(C)C(F)F)N(C1CCCN(C(C2COC(=O)O2)=O)CC1)CC c1(CC(=O)NCCC(C)N(C)C(c2ccc(C(N)=O)cc2)=O)ccc(F)c(Cl)c1 c1(N2CCC(=NO)CC2)nc(N2CCCC(N3CCCC3)C2)nc2cccnc12 C#CCC(C)(CC)C(=O)N1CCC(CNC(c2cccc(F)c2C)=O)C(F)(F)C1 c1(C(N(C2CCN(C(=O)C(C)(C)CO)C2)CC)=O)oc2c(Cl)cccc2c1C C1(C)(C)CCC(=O)N(C)CCN1.CCCN(C)C(CC)O C1(NC(c2cnc3n2CCS3)=O)CC2CC(C1)N(C(C1CC3CCC1O3)=O)C2 Cc1ccc(C)c(C(=O)NCCC2CCN(C(c3cnc(O)c(F)c3)=O)C2)c1O C(CO)(C(C)(C)C)NC(c1nnnn1C(C)(C)C)CCOC(C)C C1(NC(c2c(C)nc(O)[nH]2)=O)CN(C(C2CC2C)=O)C2(CCCC2)C1 Cc1cc(C(=O)NC2CN(C(=O)CSCC(C)C)CC2C)nnc1O N1(C(C(C(C)NC(=O)CN2CCN(C)CC2)(C)C)=O)CCCCN(C)CC1 C1(C(N2CCCCC2C2CCN(C(C3CCSC3)=O)C2)=O)(COC)CCOCC1 N1(C(c2c(C)nc(Cl)cc2)=O)CC2CCN(C(c3snc(Cl)c3Cl)=O)CC2C1 O=S(=O)(c1ccc(NC2(CO)CCOC2)cc1Br)NCCc1cccnc1 S(=O)(=O)(c1cccs1)NC(C(CCSC)N(C)C1CC1)=O C(CC(C(=O)N1CCCNCC1)C1CCC1)N(C)C C1(F)(CNC(c2cc(C)[nH]n2)=O)CCCN(C(=O)CC2CCCCC23CC3)C1 N1(CC=C)CCN(CC(=O)Nc2cccc(C(O)CC)c2)C(C)C1=O C1(NC(c2cnc(Cl)cn2)=O)COCCN(CC2CCS(=O)(=O)CC2)C1 CC1OC2(CO)CC1(C(=O)NCC1CCN1C(C1CCC(C)C1)=O)C2 N1(C(C(C)O)=O)CCOCC1CCNC(=O)CSc1ccccn1 c1(C(=O)NCCN(C(C2C(=C)C2)=O)CC)nnn(CCC)c1C(F)(F)F c1(C(=O)NC(CC)(CC)CO)n[nH]c2c1CN(C(=O)CN1CCCCC1C)C2 Cc1c(Cl)cnn1CC(=O)NC(C)C(C)NC(=O)Cc1sc(O)nc1O C1(C2CCN(C(c3cnn(CC)c3C)=O)CC2)(NC(CC(C=C)(C)C)=O)CCC1 C1(CO)CN(C)CCN1C1(C(=O)OCC)CC1.c12nc(oc1OC)CNC2=O C(=O)(CS(=O)C(F)(F)F)NCC1CC(F)(CNC(CC(C)n2ccnc2)=O)C1 C(=O)(CCCN=[N+]=[N-])NCCCC(=O)NC(C)CC1(O)CCC1 N1(C(C(C(C)(C)C)CO)=O)CCC2(CC1)CCN(C(c1csc3nnsc13)=O)C2 c1(CC(=O)NCC(C23CCC(CC2)C3)NC(CCCC)=O)cc(C)sc1C C(=O)(C1=C(Cl)CCOC1)NCC(c1ccc(F)cc1F)NC(CSCCC)=O CN1CCN(C)CC(C(N2CCCC2CNC(C2(C)CCOC2)=O)=O)C1 C1(C(C)NC(=O)CCOCc2ccccc2)CN(C(c2cc(O)no2)=O)CCO1 CCC(C(=O)NC1CC1NC(C1CC(O)C1)=O)Oc1ccccc1 c1(C(N(C(C)CNC(=O)CC2(COC)CC2)CC)=O)c[nH]nc1-c1ccoc1 Cc1ccn2c(=O)c(CNC(=O)NC3(CO)CC(C)(C)C3)cnc2c1 CCS(=O)CC(=O)NC1CC1NC(=O)Cc1cc(Cl)n(C)n1 N1(C(Cc2cc(C)sc2)=O)C2CCC1CN(C(c1cc(O)cc(O)n1)=O)C2 N1(C(CCC2(C)CC2)=O)CCC(NC(C2CCOC2)=O)C(O)C1 CCCCC(c1nnnn1Cc1cccs1)N(CCCn1cc(Br)cn1)CC C12CCC3(CN(C3)N(C3CC3)C(=O)N1)O2.c1(CN)cc(C)nc(O)c1 C1(NC(CCCC#C)=O)CC2CCC(C1)N2CC1CCC(C)C1 CC1CCCCN1CCNC(=O)C(C)(C)NC(=O)CC(C)N(C)C c1(OC)cccc(Cl)c1CC(=O)N(C)CCN(C(=O)CC(O)c1ccccc1)C N1(C(CCCCC=C)=O)CC(CNC(c2cnc(C)[nH]2)=O)CC12CCOCC2 N1(CCC(=O)N(CC(C)(C)NC(C(C2CCOC2)OC)=O)C)CCOCC1=O C1(C(=O)NC(CC#CC)C(=O)NC(C)(C)C)CN(C(C)=O)CCC1(C)C c1(C(=O)NC2C(NC(COCC=C)=O)CCC2)cc(F)cc2nc[nH]c12 C(=O)(C1CCc2cccnc21)NC1C=CCC(C(=O)OC(C)(C)C)C1 CC(C)(F)CN=c1[nH]c2c(c(=NC3CC(Cc4ccccc4)C3)[nH]1)CCCCC2 CCC(C)(CCNC(=O)C(=Cc1cccnc1)F)NC(=O)C(O)CSC c1(OC)ccc2c(=NCCc3ncc[nH]3)[nH]c(=NCCn3ncc(Br)n3)[nH]c2c1 CC1(C)CC(CC(N2CCCC(C)(NC(=O)Cc3cocn3)C2)=O)C(=O)O1 C(=O)(C1=NN(C(C)C)C(=O)CC1)NCC1(C)N(C(CCC=C(C)C)=O)CCC1 C#Cc1cnn(C)c1C(=O)NCC1(CNC(c2sccc2CC)=O)CC12CCC2 C(=O)(CCC(=O)NN(C)C)N1CCCC(CC(=O)NC(c2ccc(Cl)cn2)C)CC1 C(=O)(C(C)(C)S(=O)(=O)C1CC1)N(CC(C)CNC(c1ocnc1C(F)F)=O)C C1(CCNC(COCCCCC)=O)COCCN1C(=O)C(N1CCC(C)C1)=O c1(C(C)C)cc(C(=O)NCC(C)NC(c2ccncc2Cl)=O)cc(F)c1 C1(NC(C(C)(C)CF)=O)CC(F)CN(C(c2cccc(CF)c2)=O)C1 CS(=O)(=O)c1ccc(C(O)CNc2ccc(-c3ccco3)cc2)cc1 C(=O)(C(O)C(C)CC)NCC(CCCC)NC(c1ccc(CN=[N+]=[N-])o1)=O C1(N(C(C2CCC(CCCC)CC2)=O)C)CN(C(=O)C(CC)OC)CCC1O C=CCCCC(C)(c1nnnn1C(C)C(=O)OC)NCC(=C)C Cc1cc(N(C2CNCC2C#N)C(c2cnon2)=O)ncn1 c1(C(N2CCCC2Cn2cncn2)C(=O)NCC)cc(Cl)cc(Br)c1F c1(C(N2C(C3CCN(C(c4cn(C)nn4)=O)C3)CCC2)=O)ccc2nc(S)oc2c1 N1(CC(=O)NCC2CC(Nc3c(NC(C)=O)ccnc3)C2)C(C)=CC(C)=NS1(=O)=O C1(NC(Cn2cc(-c3cn(CCOC)nc3)nn2)=O)CCC(C(F)F)CC1 CS(=O)C=CC(=O)NC1CCCN(C(c2ccc(Cn3ccnc3)o2)=O)C1 N1(C(N2C(c3onc(C)n3)CCC2)=O)CC(=O)Nc2ccc(C(F)(F)F)cc21 N1(C(CCC=CC)=O)CCC(NC(c2ccc(N)c(Br)n2)=O)C(C)C1 c1(C(N2CC(NC(c3c(CC)csc3)=O)C(OC)C2)=O)cc(O)ccc1F c1(CNC(CCNC(N)=O)=O)ccoc1C(=O)NCc1cnsc1 C1(NC(C(n2cc(C)nc2)(C)C)=O)COCCC1NC(=O)Cc1ccc(C)s1 C1(C(=O)NC(CC)(CC)CCNC(=O)C=Cc2cnc[nH]2)CC2CCC(C1)N2C CCCS(=O)(=O)C(C)C(=O)N1CCN(CC(C)NC(c2cc(C)nn2C)=O)CC1 N1(C(CC(C)SC)=O)CCC(NC(c2oc(C(F)F)cc2C)=O)C(C)C1 c1(OC)ccc2oc(C)c(C(=O)NC3CN(C(c4sncc4C)=O)C4CC34)c2c1 C1(C(C)C)C(=O)N1.C1(CN(CCCC)CC(=O)OC(C)C)CC1[N+](=O)[O-] c1(NC(C2(O)CCN(C(CC(=C)C)=O)CC2)C)ncnc2sc(C)c(C)c12 c1(CC(C)C)c(C(=O)NC2CC(NC(C3(C)CCC34CCC4)=O)C2)cnn1C Cc1cc(-c2cn(CC3CCC(C(F)(F)F)O3)nn2)ccc1C#N c1(OCC)ccc(NC(=O)CCC2CCN(C(=O)C=CCO)C2)cn1 c1(C(=O)NC(C)CCNC(=O)CCCCO)cncc(N=[N+]=[N-])c1 C1(C(C)C)CN(C(=O)CCCc2ccccc2)CCN1C(C1C=CC(=O)NC1)=O c1(-c2ccc(C(=O)NC)cc2)ccn2nc(C(=O)NC(CO)CO)cc2c1 n1(CCC(=O)NCC(C)(C)NS(=O)(=O)C2CC2)cc(CCOC)nn1 CCCCC(F)C(=O)N1CCSCC1C(=O)NCC1CCOC1 N1(C(C=C(C)C2CC2)=O)CC(N(C)C(c2n[nH]c(C)c2F)=O)C(F)C1 C#CCCCCCCC(=O)N1CC(NC(c2ccn(CCC(C)C)n2)=O)C(O)C1 C1(C(=O)NC)CCN(C(C2CN(C(=O)Cn3cccnc3=O)CCO2)=O)C1C N1(C(CC(C)F)=O)CCN(C(C2(C)CCCCO2)=O)CC2(C)CCCC12 C(C)(C(C)(C)C(=O)NCc1ccnn1C)NC(C(C(C)O)N(C)C)=O C1(NC(CCC(C)=O)=O)CC(NC(=O)C=Cc2nnn(C)n2)C12CCC2 c1(C(n2cc(NCCN3CCC(C(C(=O)N(C)C)(C)N)C3)cn2)C)ccc(F)cc1 C1(CC(CN2C(c3ncc(C(=O)OCC)[nH]3)CCC2)O)CCS(=O)(=O)CC1 N1(C(C=CC(=O)N)=O)CC(C)OC(C)C1.C1(C(c2cc(C)on2)=O)CCC(CO)CC1 c1(CC)nc(C)c(C(=O)NCC=CCNC(C23CC(C2)C(C)O3)=O)o1 c1(N2CC(c3nnc(C)o3)OCC2)nc(=NCCC2CC2)[nH]c2cccc(F)c12 N1(C(c2cncc(C)c2C)=O)CCC(NC(C2(F)CC=CC2)=O)C(CO)CC1 O=C(C#Cc1ccccc1)N1CCN(c2ncncc2I)CC12CC2 c1(CC)cc(C(N2CC(CNC(c3ccn(COC)n3)=O)CC2C)=O)ncn1 Cc1cccc(C(N2CCCC2C2(C(=O)NC3CC4C=CC3CC4)CC2)=O)c1O N1(C(C2CC=C(C)CC2)=O)CCC(F)(F)C(CNC(c2ccc(Br)c(C)n2)=O)C1 C1(C(=O)NCC2CN(C(c3[nH]cc(CC)c3)=O)C2)CCCCC1(C)C CCC(CC(=O)NCC1(CC(=O)NCC(C)(C)CO)CC1)SC c1(C(N(CCN(CCOCC(C(=O)NC)C)C)C)=O)c(F)cccc1Cl O=C1CC(NC(=O)CC2CC(F)CN2C(C2CCCC3(CC3)C2)=O)CC(=O)N1 C1(C(=O)NCC(C(=O)NCC(CC)(C)Cl)C)C2CC3C(C2)C13 c1(C(=O)CSC)cc2ccccn2n1.C1(OCC)CC2C1(C)C(C(=O)OC)NC(=O)N2 C(CC(=O)NCC1(C)CC1(F)F)(C(F)(F)F)NC(=O)CCC1CCCO1 Cc1nc(N)c(CC(=O)N(C(C)CNC(C2CC=CCC2)=O)C)c(O)n1 c1(CC)cnc(CNC(=O)CC=CCNC(=O)CSCCC#N)o1 N1(C(c2nccc(C)n2)=O)CCC(NC(=O)C(CCS(C)=O)N(C)C)C(C)(C)C1 C1(CNC(C2(CC)CC2)=O)CN(C(=O)C(F)C(F)(F)F)C2COCC2O1 N1(C(CCNC(=O)OC(C)(C)C)=O)CCN(C(=O)CC2COC2)C2CCC12 C1(NC2(c3n(CCCC)nnn3)CN(C(C)=O)C2)CCCC(CO)C1 c1(CC(C(=O)NC2C=CC2)NC(CCN(CC)CC)=O)ccccc1Br C1(C2(O)CN(C(=O)C(CC(C)C)N(C)C)C2)(CNC(CNC(C(C)C)=O)=O)CC1 C(C(C)C(=O)N1CC(CSC)C1)NC(CNC(CC)=O)=O C(=O)(C(C)(C)CC(C)C)N1CCC(C(N2C(CCC=C)CCC2)=O)C1 Cc1ccc2scc(CC(=O)NCCN(C(=O)CC3CC=CCC3)C)c2c1 c1(CC(=O)N(CCC(C(C)C)NC(c2cnn(C)c2)=O)C)c(F)cccc1F C1(C(=O)NC2CN(C(c3scc(C(C)=O)c3)=O)C2)CC(Cc2ccccc2)=NO1 C1(C(N2CC3C(CNC(Cc4n(C)ncc4Cl)=O)(C3)C2)=O)CCC(C)(C)OC1 Cc1c(F)ccc(Br)c1C(N1CCC(NC(c2nc(=N)cc[nH]2)=O)C1)=O C(=O)(C(C)(C)CCCc1ccccc1)NCC(CNC(CC1(CC)CCC1)=O)F C(=O)CCCCCC=O.C1(C)(COCC)CCN(C(=O)CC)CC1 C(=O)(CCCCC(C)(C)C)N1CCC(N(CC#C)C(c2ccsn2)=O)CC1 C1(NC(CC2CC(SC)C2)=O)CN(C(c2cc(C)sn2)=O)C2CCCC12 c1(C(=O)NC(C)CCN(C)C(C2OC3CCC2CC3)=O)ncnc2ccsc12 c1(C(N(CCCNC(C2CC2C)=O)CC)=O)cc2n(c1)CCCNC2=O N1(C(C2CCC(=O)O2)=O)CC2CCCC1C2CNC(c1c(Cl)n[nH]c1C1CC1)=O C1(CC(=O)Nc2csc(-c3ccncc3)n2)CCCN1Cc1ccc(Cl)s1 N1(CCCCCCOC)C(=O)CN(CC23CCCC2C3(F)F)C1=O c1(CC(N2CCOCC(NC(CCC(N)=O)=O)C2)=O)c(F)cc(F)cc1F N(C1COc2cc(Br)cnc21)C(C(C)C(C)(C)C)c1n(CCCOC)nnn1 C1(NC(c2c(CC)c(C)ccc2)=O)CCCCN(C(=O)C(O)CN(C)C)CC1 Cc1cccc(C(N2CCOC(CN(C(=O)C(C)OCC3CC3)C)C2)=O)c1C C1(C(=O)NCCCOCCNC(=O)CCc2cncs2)C2CC3C(C2=O)C13 Cn1cc(C(=O)NC2CC(C(N3CCCC3(C)C(C)(C)C)=O)CC2O)ncc1=O N1(C(c2ccc(Cl)c(Cl)c2)=O)CCN(C(C2CCc3nnnn3C2)=O)CC(O)C1 N1(C(c2ccn(CC)c2C)=O)CCN(C(c2ncncc2C)=O)C(CCOC)C1 N1(C(C(=O)OCC)C)CCN(C(C2(c3cccc(C)c3)CC2)=O)CC1 N1(C(c2cc(C)n(C)c2)=O)CC(NC(C2(c3cccc(Cl)c3)CC2)=O)C(C#N)C1 c1(C(CN2CCCC2)N(C(C2CCCC2)C)C)ccc(F)cc1 C(=O)(CCCCCc1cccs1)N(C(C)CCNC(C1CN(C)C(=O)N1)=O)C C(=O)(C(C(C)(C)C)N1CCNC1=O)NC(CNC(C(n1ccc(C)n1)C)=O)(C)C N1(C(CCCC(=O)OC)=O)CCC2C(CCCN2C(=O)CCC=C(C)C)C1 c1(C(=O)OCCOCC#C)ccc(CSc2cccc(F)c2)cc1F c1(C(C(=O)NCCCC)N(C2CCN(C3CC3)C2)C)nccc2ccccc12 CC(C)CC(CNC(=O)CC1(O)CCCC1)C(=O)N(C(C)CCN(C)C)C c1(-c2nc(-c3ccc(C)cc3)nn2C23CC(C2)C3)c(C)cccc1C c1(NC(=O)CNc2c(C)scc2)ccc(Cc2ccccc2)cn1 CC1CCCC=C1C(=O)N(C)CC1CCCN(C(=O)C(F)(F)c2cscn2)C1 C1(C(F)(F)F)(C(=O)NC(C)C(C)NC(c2cccc(SC)c2)=O)CCCCO1.CC c1(C(=O)NCCC(=C)CNC(=O)Cc2ccc(Cl)c(F)c2)cc(O)nc(OC)n1 N1(C(c2snnc2C2CC2)=O)CCOC2(CCN(C(=O)CCC3CCC3)C2)C1 C1(NC(=O)NC(CSC)(C)C)CCCC(F)C1 C1(CNC(=O)CCc2cccnc2)CN(C(c2ccc[nH]2)=O)CCCO1 N1(C(=O)OC(C)(C)C)C(CNCC2CC3CCC(C2)S3(=O)=O)C2CCC(O)C1C2 N1(C(C2C(CCC)C2)=O)CCC(NC(=O)C(=O)N(C)C)C(F)(F)CC1 c1(CC)cn2c(n1)CC(C(N1CCC(CNC(=O)C(F)CC)(OC)CC1)=O)CC2 C1(C(=O)NCC(C)NC(C2C=CCS2)=O)CCC(F)(F)CC1 N1(C(c2nc(Sc3c(OC)nccc3)sc2)=O)CCC(c2cn(C3CC3)nn2)C1 CC1(C)COCC(CC(N2CC(CNC(C3(c4ccccc4F)CC3)=O)C2)=O)O1 c1(C(=O)NC2CC(F)(CNC(CCC#C)=O)C2)cc(NS(C)(=O)=O)nc(=N)[nH]1 c1(NCc2cn(CCC)nn2)cccc(S(=O)(=O)NC(C)(C)CC)c1 C#CCC(C(=O)N(CC(C)(CC)OC)C)NC(=O)C(CC)N(C)C C(=O)(C1=NOC2(CCC2)C1)NC1CC(C)CN(C(c2cccn3nncc23)=O)C1 N1(C(=O)OC(C)(C)C)CC(OC(C2C3CCCCC23)=O)CC2CCCCC12 C(=O)(CC(O)CC(C)(C)C)NC(C)CNC(C1CCCCN1C(=O)OC(C)(C)C)=O CC(CS(C)(=O)=O)C(=O)N1CCCC(C(C)(O)CNC(c2cnco2)=O)C1 CC1CC2(CCN(C(C3(CC(F)F)CC3)=O)CC2)CN1C(c1cncs1)=O C(CN=c1cc[nH]c(C#N)n1)(N(C)C(c1cnn(C)c1)=O)C1CC1 N1(C(c2c(C)cc[nH]2)=O)CCC2(CC1)CC(N1CCC3OCCC3C1)CO2 N(C1CCCn2cnnc21)C(C1(NC(C2N(C)CCCC2)=O)CCCC1)=O c1(C(=O)NCCC2CCN(C(=O)CCC(F)F)C2)ncc(Cl)cc1Cl c1(C(=O)NCCN(CCC)C(c2sc(CC)nc2C)=O)noc2cc(F)ccc12 C12(NC(c3cn[nH]c3)=O)CCCN(c3nnco3)CC1C2.C1(C=O)(CO)CCCCC1 C(=O)(C(C(C)C)N(CC(C)(C)C#N)CC)N(C(C)C(=O)NC)CCC Cc1ccc2nonc2c1C(=O)NCC(C)N(C(=O)CCCS(C)(=O)=O)C CC(C(=O)N1CCC(C(=O)NC2CCC(=O)N(C(C)C)C2=O)O1)=C1CC1 c1(C(=O)NCC2(CCNC(COC3(C)CCC3)=O)CC2)cc(Cl)cnn1 c1(CCNC(=O)NC2CCc3nccn3C2)c[nH]c2nc(Cl)ccc12 CC1CN(C(=O)C(C)(C)CN(C)C)CC(C)C1NC(=O)CSC(F)(F)F C1(C)(CC)NC(=O)N(CC(N2CC(NC(c3cccn4nncc34)=O)C2)=O)C1=O CC(C)(CCC#N)C(=O)N1CCCC2(NC(=O)C#CC3CC3)CC2C1 C(=O)(C1CCCn2nccc21)NCCCN(C(C(C)Sc1ccccc1)=O)C C1(C(=O)NC)CCC(N=C2NC3=NC2CC2CCC(CNc4c3[nH]cc4)O2)CC1 c1(N2CC(S(C)=O)C2)ncnc2c1ncn2CC1(C)CC1(F)F C#Cc1ccc(C(=O)N(CC(C)NC(C2(C)CCCS2(=O)=O)=O)CC)cc1Cl C1(CCC(=O)NCCN(C)C)CCCC(N)C1 c1(CNC(C2(CC=C)CC2)=O)ccoc1C(=O)NC1CCN(C(C)C)C1 c1(C(C)=O)ccc(OCC(=O)NC2CCC2CNC(C2(CO)CCCO2)=O)cc1 C1(F)(CNC(C2C(CC)C2)=O)CCCN(C(c2cnc3n2CCS3)=O)CC1 C1(C(=O)NCC(CC)NC(C2(C)COCCO2)=O)CC2(CCC2O)C1 CC1CC(N(C(=O)CCCN(C)C(c2csc(Cl)c2)=O)C)CC(C)C1 N1(C(CC=C)=O)CC(F)(F)CC1CNC(C12CCC(C(=O)OCC)(C1)C2)=O CC(C)(CNC(c1conc1CNC(C1CCCC(=O)CC1)=O)=O)CCCO Cc1cccc(O)c1C(=O)N(C(C)(C(=O)NC(C1CCOC1)CO)C1CC1)C Cc1c(F)ccc(C(=O)NCCC2CCN(C(=O)Cc3ccon3)C2)c1N N1(C(c2c(C)nncc2)=O)CCC(C2CCN(C(C3(F)CC3C)=O)C2)CC1 c1(C(N(C(C)CCNC(=O)Cc2cccs2)C)=O)cnn(-c2ccccc2)c1F c1(C(N(C2CCN(C(c3nncn3CC)=O)C2)CCC)=O)ncc(Br)cn1 C1(C)(C(=O)NC2C3CC(NC(c4n(C)cnc4)=O)CC32)COC(C)(C)CO1 C(=O)(C(CC)C(=O)N1CCCCC1C(N1CCCC(F)(F)C1)=O)OCC N1(CC)CCC(C(=O)NCc2cn(-c3cccc(Cl)c3)nn2)C(O)C1 c1(CC(=O)NC2(C(=O)NC(c3ccncc3Cl)C)CCC2)cccc(O)c1 N1(C(c2c(CCC)nco2)=O)CCC(NC(=O)Cn2ncc(Cl)c2C)CC1 C(CC(CO)C(C)C)OCC(=O)NC(C(C)C)C(=O)NC1CCC1 N1(C(C)=O)CCOCC1C(N1CC(CNC(=O)CC2CCC2)C1)=O C1(C(=O)NCC(C(C)(C)C)NC(c2cscc2C#N)=O)CC2CCC1CC2 C(=O)(NN1CCCC1C(=O)NCC1(C)CCC(=O)N1)c1cc(CC)no1 c1(C(=O)NCC(CC)(CC)NC(c2cn(C)nc2O)=O)c[nH]c2cc(F)ccc12 C1(N(C(C=C(C)C)=O)C)CC2CCC(C1)N2C(=O)CCc1ccc(O)c(Cl)c1 C12(CCCCC1)C(=O)N1CCC(O)(C1)C(=O)N2.CC#CC(=O)N(CC)CC N1(C(c2cc(COC)n(C)n2)C(=O)NC2CCCCC2)CCC2CCN(C)CC12 C(=O)(C1=CCCCO1)NC(CC1CN(C(c2ccc(C(C)O)cc2)=O)C1)C c1(N(CCCNC(C2(C(C)C)CNC(=O)C2)=O)CC)ccc([N+](=O)[O-])cn1 c1(CC)noc(CC)c1CC(=O)NCCC(C)(C)NC(c1csc(CSC)n1)=O C(=O)(C#CC(C)(C)C)NCCN(C(COc1ccc(C(CC)=O)cc1)=O)C C1(N(C(=O)CCC2(OC)CCOC2)C(=O)C2CC2)CCc2c[nH]nc2C1 c1(C(N2CCN(CC(N3CCC(C#C)CC3)=O)CC2)=O)cccc2c1CCC2 N1(C(=O)CC=CC(C)(C)C)CC2CCC(CNC(c3n(CC)ncc3C)=O)C2C1 C1(CNC(CN(c2ncccn2)C)=O)CN(C(c2cncn2C)=O)C(C)(C)C1 N1(C(Cc2c(C)nsc2)=O)CC(C(=O)N(CC(O)CO)C)C(F)(F)C1 C(=O)(C1CCCn2c(Br)cnc21)N1CCCN(C(C(C(C)C)(C)O)=O)CC1 c1(OC)ccc2c(c1)C(NCc1nc(Br)co1)CC2 c1(C(N2CCC(NC(Cc3n(C)ccn3)=O)(CF)C2)=O)ccn(O)c(=O)c1 C(=O)(C1=CC(O)C(NC(=O)C#CC2(C)COC2)C1)NC(c1nccc(O)n1)C N1(C(C(Cc2ncn(C)c2)O)=O)CCN(C(C2CCCC2)=O)CC1C(F)F CCC(CC(=O)NCC1CN(C(=O)C(C)C#N)C2(CCC2)C1)CC(C)C CCCC(CNC(=O)CCOCC1CC1)C(=O)NCc1cc(C(C)C)on1 CC1(C)C2CCC1(C)C2C(N1CCN(C(=O)CCC2CCOC2)C(CF)C1)=O C1(NC(C=CC)=O)CCN(C(c2cc(CCO)on2)=O)C1C1CC1 C1(O)(CCNC(C(C)CC2CCCOC2)=O)CCN(C(c2ccoc2Cl)=O)CC1 Cn1cc2c(n1)CC(C(=O)NCCCCNC(c1cscc1C(F)F)=O)CC2 C#CC1CN(C(=O)CC2CCS(=O)(=O)CC2)CCN1C(=O)C(COC)N(C)C c1(C(=O)NC(CN(C(C2CC3CCC2O3)=O)CC)C)nc(O)nc(O)c1N c1(C(N2C(CN(C)C(c3ncccn3)=O)CCC2)=O)nccc(Cl)c1F c1(C(C2CCCN2Cc2ccc(Nc3ccccc3)s2)=O)ccnc(Cl)c1F c1(CC(N2C(CNC(C3(CSCC)CC3)=O)CCC2)=O)cnn(C)c1C C1(C(=O)NCc2n(C)ccc2)CCC(NCC2CCC(O)CC2)CC1 c1(Cn2nnnc2C(C2CCCSC2)NCC=C)ccc(N(S(C)(=O)=O)C)cc1 C(=O)(C1Cc2ccc(Cl)cc21)N1CCN(C(Cc2c(C)nn(C)c2Cl)=O)CC1 CC(C)(C(=O)N1CCC(C2CCCN2C(C2CCCC2)=O)C1)C(F)(F)F N1(C(c2n(C)cc(C3CC3)c2)C2CC2)CCc2nc[nH]c2C1c1ccc(Br)cc1 C1(c2nnnn2C2CC2)(NCc2c(Br)c[nH]n2)CC2(CCC2)C1 N1(C(c2c(CC)oc(C)c2)=O)CCN(C(=O)CCC(C)N(C)C)CC1CF N1(C(c2c(C)n(C3CCOC3)nn2)=O)C2CCC1CN(C(c1c[nH]ccc1=N)=O)C2 C1(C)(C(=O)NCC(CC(C)C)OC)CC(O)CN1C(C1CC2(CC2)C1)=O C1(C(=O)NCC(C)CCCO)CCCN1NC(=O)C1CC=CC1 C1(C(=O)NCCC(C)F)COCCN(C(=O)C2=CCCC2C)C1 N1(C(c2c(CC)con2)=O)C(C)CC2CN(C(C3(OC)CCOC3)=O)CC12 c1(CC(=O)NCCCC(C)NC(c2ccc(C(N)=O)o2)=O)nn(C)cc1Br C1(NC(c2onc(CC)n2)=O)CN(C(=O)CCc2cncc(C)c2)CCC1C Cc1cc(C(=O)NC(C)(CO)C(=O)N2CC(CO)(CO)C2)oc1C N1(C(C(c2n(C)ccn2)(F)F)=O)CCOC(CNC(=O)CCN2CCC2)C1 C(=O)(CCC(C)(F)F)N1CCC(CCOC)(NC(=O)C(N2CCCCCC2)C)C1 C(=O)(CC(C)(C)C(F)F)N1CCC(C(CNC(C=C(C)C(F)F)=O)C)CC1 C1(C(=O)NCC2CCC(F)(CNC(C(COC)C)=O)CC2)CC2(CC(C)=NO2)C1 C1(CCNC(C2(CO)CCCO2)=O)CCN(C(C23CC(CC(F)F)(C2)C3)=O)C1 c1(CCCC(=O)NC2CN(C(=O)C3=CCCS3)CCC2F)c[nH]c2ccccc12 N1(C(C(CC)CC)=O)CCCC2(C1)CN(C(C1(c3ccccc3)CC1C)=O)C2 N1(C(CC(CNC(c2n(CC)nnc2)=O)C)=O)CCOc2ccccc21 c1(C(=O)NC2(CO)CCCN(C(=O)C(O)C(F)(F)F)C2)cc(Cl)ccc1[N+](=O)[O-] C=CC1CN(C(c2cc(C)ccc2OCC)=O)CC1NC(=O)C(C)(C)CO C1(NC(C(C)NS(CCC)(=O)=O)=O)(CNC(=O)C(C)O)CCOCC1 N1(C(c2ccc(C)[nH]2)=O)CCC(C)C(NC(C2(CN(C)C)CCCC2)=O)C1 C1(C(=O)NCC2(C)CCCN2C(c2cnccn2)=O)CCn2nncc2C1 N12CCN(C(=O)C3=NNC(=O)C3)C(C1)NC2=O.c1(OC(C)C)ccc(CO)cc1 C(CN=C(NCC1CCCO1)NCC1CC(F)(F)C1)c1c(C)nccn1 C(=O)(C1=CC2(CCN(C(=O)C(F)CCC)C2)C1)NC(CCCC)CC CC(C)CCC(O)C(=O)N1CCCCC(CNC(=O)CCc2ccc(Cl)nc2)C1 C1(O)(CC(=O)NCC(=O)N(C2CCCO2)C)CN(C(=O)COC(C)(C)CC)C1 Cc1cc(C)c(C(=O)NCC2CC3CCC(C2)N3C(=O)CCCF)cc1Br c1(C(=O)NCC2CC(NC(C(C3CC3)SC)=O)C2)c(C)nc2sccn12 C(=O)(C1OC(=O)c2ccccc21)NCC1CC(NC(C2C(C=C)CC2)=O)C1 N1(C(CCC2C(C)(C)C2)=O)CCOC(CNC(c2ccoc2Br)=O)C1 C(=O)(C1CCC(=O)c2cccn21)N1CCCCC(CNC(COCC(C)C)=O)C1 N1(CCOC)CCN(c2ccnc(NCCSCc3cccc(Br)c3)n2)CC1 N1(C(c2oc(C)c(CO)c2)=O)CC(CNC(=O)C(F)C2CCOC2)CCC1C N1(C(C(CC)NC(N)=O)=O)CCOCC(CNC(C2(C)CCOC(C)C2)=O)C1 N1(C(c2c(CC)nc(C)nc2)=O)CCCC(C2CCN(CC3CCC3)CC2)C1 CC1CCN(C(=O)C(c2cnccn2)C)CCN1C(c1ccc(=O)oc1)=O c1(C(=O)NCC(=C)CCNC(C2COCC(C)O2)=O)c(Cl)ccc(F)c1C c1(OC)ccc(CC(N)C(=O)NC(c2cccc(N3CCOCC3=O)c2)C)cc1Cl C1(NC(CCN2CCN(C)CC2)=O)COC2C(NC(c3ccc(Cl)o3)=O)COC12 C1(C(=O)NCC(C2CCN(C(C3CC(=C)C3)=O)CC2)(C)O)COC2(CCC2)CO1 c1(NS(=O)(=O)Cc2ccon2)nc(Br)c(C2OCCO2)s1.O=C1CO1 C12(CNC(c3c(C)csn3)=O)CCCC1CN(C(c1cccn1C)=O)C2 Cc1ccc2sc(CN(C3CCN(C(=O)OC(C)(C)C)C3(C)C)CCO)nc2c1 CCC(F)C(=O)NCC(O)CN(C)C(c1cnn(C(F)(F)F)c1)=O C1(C(N(C)CC2N(C(C(CC)n3cccn3)=O)CCCC2)=O)CCCC(C)(C)C1 c1(CC)sccc1C(=O)NC(C)(CNC(=O)CCNC(=O)COC)CC C1(C(N2CC(O)(CN(C(C3CN(C)C3)=O)C)C2)=O)CC2CCC1C2 O=S(=O)(c1ccc2c(Cl)ccc(Cl)c2c1)NC1C2Cc3c(F)cccc3C12 C=C1CC2(C1)CC(C(N1CCOC(CNC(=O)C(c3ccc(Cl)cc3)C)C1)=O)C2 CC1(C)CCCN(C(c2cc(C(N)=O)[nH]n2)=O)C1C(=O)Nc1cnc(Cl)nc1 C1(C(=O)NCc2oc(C(=O)NCc3c(C)ccs3)c(C)n2)CC(C2CC2)=NO1 C1(CNC(C(C)=C(CC)C)=O)CN(C(=O)C=CCN(C)C)C2(CCOCC2)C1 c1(C(N2CC3(CN(C(C(C(COC)C)C)=O)C3)C2)=O)ccc2ccncc2n1 c1(C(N(C(CN(C(C(CC)=CC)=O)C)C)C)=O)ccnc(N2CCN(C)CC2)n1 c1(OC)cc(C(=O)NCC(CO)CCCCN)cc2c1OC(C)C2 C1(CNC(CCN(C(CCC)C)C)=O)CC12CCN(C(c1ccsc1CC)=O)CC2 Nc1c(C(=O)NC2CC(NC(=O)CCCc3ccncc3)C2)cccc1O c1(N(C(C23C(CN(C(c4c(CCC)onc4C)=O)C2)C3)=O)C)cccn(C)c1=O N1(C(COCCCCCC)=O)CCC2CCN(C(=O)Cc3nc(C)cs3)CC12 CC(CC(C)C(F)F)NC(=O)C(c1cccs1)NC(=O)CCC(=O)c1cccs1 C(c1ccc(Cl)c(Cl)c1)=CC(N1CC(NC(C(C)OCCC#C)=O)CC1(C)C)=O c1(CC(=O)NC2CN(C(CNC(CCC(C)C)=O)=O)CC2O)ccc(F)cc1Cl c1(C(N(CC(CNC(Cc2cc(C)on2)=O)(C)C)C)=O)cccc([N+](=O)[O-])c1Cl N1(C(C(C2CCCC2)OC)=O)CCC(NC(c2cnncc2C)=O)CC1 N1(C(CCC(C)OC)=O)CCCCC(C(=O)NC(CO)CCC2CC2)C1 N1(C(C(CCC)Cl)=O)CCC2(CCCCC2NC(=O)CSCC(N)=O)C1 O=C(CCC(F)(F)F)NC1(CCCCNC(=O)CO)CC1.C1(CC)CCCO1 c1(C(=O)NCC(CC)NC(c2ccc(F)c(O)c2F)=O)cc(C)sc1S(N)(=O)=O c1(COC)cccc(OC(F)(F)F)c1.C12CC1C(=O)NC1(CC1)CCCNC2=O c1(C(N2CC(CNC(C(C)(C)c3ccccn3)=O)C2)=O)ccc(N)cc1Cl c1(SCC2(F)CCN(C(=O)Nc3ccn(CC)n3)C2)cc(F)ccc1F CCC(C#N)C(=O)N1CC(O)(CCNC(=O)C2CC2)C1 c1(OCC)cccc(C(=O)NC(C2(O)CCN(C(=O)Cn3ccc(C)n3)C2)C)c1 c1(C(N2CC(F)(CNC(c3ccc(F)cc3)=O)C2)=O)sc2cccnc2c1Cl C(=O)(CCC(N)C(=O)O)NC1CCN(Cc2c(CC)noc2CC)CC1 C1(C)(CC(=O)NCC(c2ccccc2)NC(c2ccc(C(C)=O)o2)=O)CCOCC1 C#CCCCCCCC(=O)N1CCC(O)(CCNC(=O)C(O)CC2CC2)CC1 c1(N(C(=O)C=COC(C)C)CCC)cc(C(C2CC2)N(C)C)nc(C)n1 c1(C(=O)N)ccc(O)c(C)c1C.C12(NC(C3ON=C(C)C3)=O)COC(CF)(C1)C2 c1(C(=O)NCC2(F)CC(NC(C(C)n3cccc3)=O)C2)ccc2c(c1)nnn2C c1(-c2nc(COC)nn2C2CCCC2(C)C)cc(C(C)C)ccc1C c1(OC)cc(C(N2CC(NC(c3nc(=N)cc[nH]3)=O)CCC2C)=O)cc(C)n1 C1(CCC)CN2CC1(F)SCC1(CC2=O)CC1.c1(C(=O)NC)nc(OC)co1 c1(NC(c2ccc(C3CCCCO3)cc2)=O)cc2cc(Br)ccc2s1 C1(NC(Cn2ccc(C)n2)=O)CCN(C(C2CSCCS2)=O)CC1C(N)=O C(=O)(CC(C)C(F)(F)F)N1C(CCNC(c2c(C)coc2C2CC2)=O)CCC1 C1(C(=O)NC(C#C)CC)CCN(C(=O)Cc2cccc(O)c2)C(C)(C)C1 N1(C(c2cccnc2)C=O)CC(C)(C)C1c1ccccc1.Cc1cnn(CC)c1 Cc1ccc(NC(C2(NC(=O)C(c3ccnn3C)C)CCN(C)C2)=O)cn1 C1(NC(C2CC(=O)NC2)=O)CC2(C1)CC2NC(=O)Cc1cccc(Cl)c1 c1(C(N2CC(C)CC(NC(c3c(CC)nc(C)[nH]3)=O)C2)=O)ccn2c1CCCC2 N1(C(Cn2ccc(C)cc2=O)=O)CCC2(CC1)CCN(C(c1csnn1)=O)C2 n1(CC(N2CCC(C)(NC(C(C(C)C)O)=O)C2)=O)ncc2cccnc12 c1(N(C)C)cc(C(=O)NC2CCCC(NC(c3nsnc3O)=O)C2)cc(Cl)n1 c1(C(C)OCC)nc(CC(=O)NCC(O)CN(C(=O)Cn2cn[nH]c2=N)C)cs1 N1(C(c2n(C)ncc2Cl)=O)CC2CCCC(NC(=O)CC3(O)CCCC3)C2C1 C12(C(=O)NCC(CC)n3cccn3)CCCC1CN(C(C1CCC(F)(F)C1)=O)C2 Cc1ccc(C(=O)C(=O)NC(C)(C)CN(C(=O)C=Cc2nc(C)co2)C)cc1 N1(C(c2c(C)cccc2)=O)CC(NC(=O)C=CC(C)C)C(C2CC2)C1 C1(CC(=O)NCCCCCNC(=O)CN2CCCNC2=O)CC2CCC1CC2 N1(C(c2[nH]c(=NC)sc2)=O)CC2CCC(C1)N2C(=O)C(=CC1CCCC1)C C12CN(CCCO1)CC2.n1(C2(C(C)CC)CC2)cc(Br)cn1 NC1CC2CC(C1)N(C(C1COCCN(C(=O)CCCN3CCCCC3)C1)=O)C2 Cc1cc(C)n(CC(N2CCCN(C(=O)CCCC(C)(F)F)C(C)C2)=O)c(=O)n1 C=CC(C)(O)C(=O)N(C)CC1(NC(c2ncoc2C2CC2)=O)CC1 Cc1ccc(NC(C2CCCN(C(=O)C(n3ccc(C)n3)C)C2C)=O)cc1C CS(=O)CCC(=O)NCCCN(C1CCCC1)C(=O)C=C(C1CC1)C1CC1 CCCCCCCN(C(=O)COCCCC(=O)NC(=O)C(O)CC1CCCC1)C c1(C(=O)NC)ccc(Cl)c(NCc2cn(C)nc2C(F)(F)F)c1 CCC(C)C(CN(C)C)OC.C(=O)(COCC(C)C)NCCOCCSC C1(CNC(N)=O)CN(C(=O)CCNC(C2CC(=C3CC3)C2)=O)C1 c1(CNC(CCN(C)C(c2cc(Cl)cn2C)=O)=O)ccncc1F c1(C(N2CC(O)(CNC(CCc3c(C)n[nH]c3C)=O)C2)=O)ncnc2c1CCC2 C1(NC(c2c(-c3ccccc3)nc(C)s2)=O)CN(C(C2CC2C)=O)CC(C)(C)C1 N1(C(CCC)=O)CCOC2CCN(C(=O)C=C3CCSCC3)CC12 N1(CCn2c(C)ncc2)CCN(C(=O)C(C)S)CC1.C(=O)(C(C)C)O C1(F)(CC)CCN(C(C2CCC(CNC(c3coc(C)n3)=O)C2)=O)C1 N1(C(C2CC(C)(C)C2)=O)CCN(C(C2C3CCOCC23)=O)CC1CO C(=O)(CC(C(C)(C)C)NC(=O)C(C)C(CC)CC)NC(CC#C)(C)C CC(C)CCCC(C)C(=O)NC(C1CC1C(=O)N(C1COC(C)(C)C1)C)C c1(CNC(C(CC)N(C)C)=O)cccc(C2CCC2)c1 N1(CCNC(c2ccccc2)=O)CCCNC(=O)C1.C12C(C1(F)F)C(=O)N2 c1(NC(C(C(C)(C)C)NC(C2=C(C)CC2)=O)=O)ccc2c(c1)OCC2 c1(C(=O)NCC(CC=C)NC(=O)CCn2cc(Cl)cn2)cc(C)nn1C c1(C(C)(F)F)cc(C(=O)NCC(C)(C)CNC(=O)CC(C)n2cccn2)[nH]n1 c1(C(=O)NCC2C3CN(C(c4nc(C)sc4C)=O)CC32)cc2c(C)nn(C)c2s1 N1(C(C(C)OCC)=O)CC2CC(C(=O)NCC3CC3C(F)(F)F)(C2)C1 c1(C(=O)NC(CC(C)C)CNC(C2(C)CCCC2(F)F)=O)cncc2c[nH]nc12 N1(C(c2c(C)nc(CC)o2)=O)CC(N(C)C(C2CC2c2ccsc2)=O)C(C)(C)C1 C1(C2CCOCC2)(NC(C2(CNC(CCC(=O)OCC)=O)CC2)=O)CC1(F)F.CNC n1(CC(=O)NCC(C2CCC2)NC(C(C)N2CCCC2)=O)cc(F)ccc1=O C(C(C)(C)C#CC(=O)NC1CCCN(CC)C1)NC(c1c(CC)non1)=O c1(CCN2C(C(N3CC4CC3CS4=O)=O)CCC2)cccc2c1OCCO2 C1(NC(C2(C)CCC2)=O)COC2(CCCN(C(C3CC(F)(F)C3)=O)C2)C1 C1(NC(Cc2n(C)ncc2)=O)CCCCC1NC(=O)Cc1cnc[nH]1 C=CCC(C(=O)NC1CN(C(C2CC3CC3C2)=O)C1)OC C1(CC(NOCC(=O)OC)=O)CCCCN1C(=O)C(O)CN(C)C N1(C(C2C(CC)OCC2)=O)CCC(CCNC(=O)C(C)Cc2cnn(C)c2)CC1 C1(C(=O)NC2CCC(NC(=O)C(F)C3CCCC3)CC2)CC12CCOCC2 CC(Cn1c(CCO)ncc1)C(=O)NCCCC(C)NC(=O)C(=O)NC1CC1 C1(CNC(C2CC=CC2)=O)CCN(C(c2cc(O)ccc2Br)=O)C12CCC2 C1(CNC(=O)Cc2cccnc2)COCCN(C(c2cn3c(n2)SCC3)=O)C1 c1(C(=O)NCCCC(C)NC(C(C=C)(C)C)=O)cnc(O)c([N+](=O)[O-])c1 O=C1CCC2(C(=O)NCCCNC(c3ccc4occc4n3)=O)CCCCC2N1 C(c1ccc(Cl)cc1)=CC(=O)NCc1ccccc1C(F)(F)F C1(CC(=O)NCCCNC(=O)NC(CN(CC(C)C)C)=O)CCCOCC1.C(C)(C)(C)O C(=O)(C(C(C)(C)C)N(C)C)N1CC2C(CNC(c3c(C)ccs3)=O)(C2)C1 Nc1c(C(=O)NCC(CO)NC(c2cnn3cnnc3c2)=O)ccc(Br)c1F CC(C(C)(C)C(=O)NC1(C2CC2)CC1)NC(c1cncc(C#N)c1)=O C(=O)(CC(C)(C)CNC(c1ccc[n+]([O-])c1)=O)NCC(C)N(C)C1CC1 N12CC3(COC)CC1(C3)C2=O.c1(CN(C(CCC)=O)CC)cncn1CC C1(OC)CN(C(c2cc(Cl)c(Cl)s2)=O)CC1c1cn(CC2CCC(=O)O2)nn1 c1(-c2cn(CC(=O)N(CCOCC)C)nn2)cc(OC)ccc1Br Cn1nc(CNCC2CCCCC(O)C2)c2c1CCN(c1nnnn1C)C2 C(C1CC1)(C1CC1)=CC(N1CC(O)(C(C)(C)CNC(=O)CO)C1)=O C1(CNC(CCN(S(C)(=O)=O)C)=O)C2CCC(C2)N1C(=O)C1=NOCC1 Cn1c(=O)n(CCC(=O)NCCCCNC(=O)C(F)F)c2c1CCCN2 N1(CC(=O)NCC2CC(NCc3ccc(C(=O)OC)o3)C2)CCN(C)C(=O)C1 N1(C(Cc2c(C)n(C)cn2)=O)CC2COCC2(C(=O)NOCCCC2CC2)C1 N1(C(CNC(=O)OCC=C)=O)CC(CNC(=O)CC2CCCCC2)C2(COC2)C1 N1(C(c2cc(CC)nn2C)=O)CCC(F)(C(=O)Nc2cnc(Cl)c(C)c2)CC1 N1(C(C(=O)N(C2CCN(C(c3cc(OC)n[nH]3)=O)CC2)CC)C)CCC(O)CC1 CCCC(CC)C(=O)N1CCC(C(N2CC=CC2C(=O)NC)=O)C(C)C1 CC1(CCC(N2CC3(CC3)C2)=O)CCCN1C(=O)CCn1cncn1 C1(CC(=O)N(CC(=O)NCCN(C(C(C)C)CO)C)C2CC2)CCC(=O)NC1 N1(C(COC(CC)(C)C)=O)CC(CNC(=O)C(N2CCOCC2)C)C(F)(F)C1 c1(CNC2CN(C(C(C)(C)CCl)=O)CC2F)ccc(Br)c(F)c1O c1(C(N(C(C)CNC(C2CC(C)CO2)=O)C)=O)nc(-c2ccco2)oc1C1CC1 C1(C(=O)NCC2CCC(NC(CC(=C)C)=O)CC2)CCn2c(C)nnc2C1 N1(C(c2oc(CC)c(C)c2)=O)CC2(CCN(C(=O)C(C)C(C)C3CCC3)C2)C1 C1(CNC(c2c(C)snc2)=O)CCCC12CCN(C(C1CCCN1C=O)=O)CC2 c1(C(=O)NC(CC)(CNC(C2CC2C(C)C)=O)CC)noc2c1COCC2 N1(C(c2ccnc(Cl)c2F)=O)CCCC2CN(CCOCC3CCCOC3)CC12 CC1(NC(=O)C(CCC2CC2)NC(=O)CCc2nncs2)CC2CCC1C2 C(N=c1nc2scnc2c(NCC2(CO)CCCC(=O)N2)[nH]1)C1CC(C)C1 N1(C(CCSCCC)=O)CC2CCOC2(CNC(c2cn(C)nc2O)=O)C1 C1(C(=O)NCC2C(NC(c3cn(CCC4CC4)nn3)=O)C2)COC2(CCC2)C1 C1(NC(=O)CN2CC3CC3C2)CN(C(c2cc(Cl)sc2Cl)=O)CCC1F C(=O)(C(F)C(C)CNC(C1(CC)CCOCC1)=O)N(CC#CC)C c1(Cn2cc(C3C4CN(C3)C(=O)CO4)nn2)nnc2ccccn12.CC(=O)CC C1(NC(=O)Cc2cccnc2)CC(C(=O)NCc2ncc(C(F)(F)F)[nH]2)CC1O c1(C(N(CCCCNC(=O)CC2COCCO2)C)=O)cnn(C(C)C)c1F c1(OCCOC(=O)Cn2cc(Cl)cn2)cc(Br)sc1Cl c1(NC(C2CC3(CC(OC)C3)C2)=O)ncnc2c1CCC2 c1(C(=O)NCC(CO)NC(=O)C(c2ccccc2)=O)ccccc1CC#N CCCC(C)(O)CC(=O)NC1COCC1C(=O)N(C1CC(O)C1)C C#CCCN=C(NCC1(C2CC2)CC1)NCC1(Cl)CCCC1 C(=O)(CCC1=NNC(=O)CC1)NC1CC(NC(c2c(C)ncnc2)=O)C(O)C1 C1(CC)CN(C)CCCN1C(=O)CCCCCNC(=O)C=CCCC(C)C c1(-c2c(OC)cncc2)ccn2cc(C(=O)Nc3cnc[nH]3)nc2c1 CC(=NO)C1CC(C(=O)NCC2(C)CCN(C(=O)CC34CC(C3)C4)CC2)C1(C)C Cc1cc(=NCC(C)CNC(c2[nH]c(C)c(C)c2C)=O)[nH]c(C(C)(C)C)n1 C1(COC)CCN(N2CCCC2(C)c2c(C)n[nH]c2C)CC1 CC1=CCSC1C(N1CCC(OCC(=O)N(C2CC(F)(F)C2)C)C1)=O c1(CNC(C(=O)OC)(C)Cc2ccccc2)cccc(Br)c1C CC(C)CC(C)CC(C)C(=O)NC1CN(C(C2CC(=O)CS2)=O)C1 c1(CC)ccc(C(=O)N(C2CN(C(C3CCN(CC(F)F)CC3)=O)C2)C)c(F)c1 CCC(CC)(CC)C(=O)N1CCCC(C)(NC(=O)C(n2ccnc2C)C)C1 CCC(C)C(C(=O)NCC=CC(C)(C)C)N(C(=O)CCc1nncn1C)C C1(NC(=O)COC(F)F)COC2(C1)CN(C(=O)CCCCF)C2 C1(C)(NC(CCc2cc(C)[nH]n2)=O)CCN(C(=O)C(C)NS(C)(=O)=O)C1 c1(N(N2CC(C(C)(C)O)(CNC=O)C2)C)cc(C2CC2)ncn1.C1(F)(C=O)CC1 N1(C(c2n(CC)nnc2)=O)CCOC2(CCN(C(=O)CC3CCC(F)(F)C3)C2)C1 C1(O)(C(=O)NCC(CO)NC(c2coc(O)n2)=O)CCSCC1 N1(C(=O)Nc2ncc(-c3ccc(CC)cc3)s2)CCC(C(=O)OC)C12CC2 N1(C(C(C)Oc2cccc(F)c2)=O)CCCCC(NC(c2nncnc2Cl)=O)C1 c1(C(N2CCN(C(C3N(C=O)CCC3)=O)C(CCO)C2)=O)n[nH]c2c1COCC2 N1(CCC=CC)CC2CC2(C(=O)N(C)C(C)C2CC2)C1 C1(NC(C(CCO)N(C)C)=O)CN(C(=O)Cc2cc(F)ccc2F)CC1C1CC1 c12ccccc1C(=O)NC2c1nnnn1C.C1(CCOC)(NC)CCC1 CC(C)C(CCC(=O)N(C(C)CC(F)(F)F)C)NC(=O)CC12CCCC1C2 c1(SC)ccc(CN2CC(C)(CC(C)C)C2)cc1.c12ccc(cc1)c(=O)[nH]2 C1(NC(CCC#C)=O)CCCCC12CCCN(C(c1cc3sccc3s1)=O)C2 c1(CN(CC=C)C)cn(C2CCC(C(=O)NCCc3ncoc3CC)C2)nn1 N1(C(Cc2c(C)n[nH]c2)=O)CCCCCC1CNC(C1CSCC(=O)N1)=O N1(C(NOCC2CNC(=O)O2)=O)CC(F)(F)C1c1ccc(F)cc1 c1(C(=O)NCC(CC(=O)NCCCCc2cnc[nH]2)OC)ncc(F)cc1F c1(CC2C3CN(C(C(=O)NCC4CCOC4)c4ccoc4)CC32)cccc(Cl)c1 C1(NC(CC(=O)O)=O)CCC(CC(N2CCCC2c2nccs2)=O)CC1 c1(OC)ccc(NC(=O)C(=O)N2CC(OCc3ccc(F)cc3F)C2)cc1S(N)(=O)=O c1(C(N2CCN(C(C34CC(C)(C3)C4)=O)C3C2C3)=O)cccc2scnc12 C1(CNC(C(CCC)NC(c2ccn(C(F)F)n2)=O)=O)CCOCC1(C)C c12nc(C)c(o1)C(=O)NC2.c12nocc1C(=O)NC2.C1(CC)(CO)CC1 c1(CC(N)C(=O)NC23CCCCC(F)(C2)C3)ccc([N+](=O)[O-])cc1Cl c1(C(=O)NCc2cn(-c3cncc(N(C)CC)c3)nn2)scc2c1OCCO2 Cc1cc(C(F)(F)F)ccc1C(=O)NCCOCCOCCNC(N)=O c1(CNC(c2cnc(OC)s2)=O)nc(C(=O)NCCNC(C)=O)c(C)o1 c1(CNC(C(N2C(C=C)CCCC2)=O)=O)cc(C)c(Br)cn1 N1(C(CC(CN(C(Cc2ccn(C)c2)=O)CCO)O)=O)C2CCC1CC(=O)NC2 Cc1cc(C(=O)NCCC2(O)CCCN(C(=O)COC(F)F)C2)c2occc2c1 C12(C(N3CCCC(NC(c4ccc[nH]4)=O)(CO)C3)=O)CCC(O1)c1ccccc12 C(CCCC(=O)NC1(C)CC(NC(=O)Cc2cccc(CC)c2)C1)OCCC=C c1(OC)ccc(Br)c(CNCC2CCC(C(=O)NCCc3ccco3)CC2)c1F C(=O)(C(C(C)(C)C)NC(c1cnn[nH]1)=O)NC(C)CC1CCCC1 C(=O)(CC(CC)C(C)C)NC(COC)CC(N1CCOC(C)(C)C1)=O N1(C(CCC#C)=O)CCC(C)(C)C1C(=O)NCCN1CCCCC1 C1(C(N2CCCC2(C(C)C)CO)C(=O)NC)C2CCCCC12 Cc1cc(C(=O)NCc2ocnc2C(=O)NC2CC(O)C2)cc(C#N)c1 N1(C(C(N2CCCCC2)C)=O)CCCC2C(NC(=O)CN(C)CCO)C(C)(C)C12 C(=O)(CS(=O)(=O)C(C)C)NCC1C(NC(CCc2ccc(OC)c(F)c2)=O)C1 N1(C(c2ccc(SC)o2)=O)CCC(O)C1C(=O)NC1(C)CCCC1C C=Cn1nncc1C(=O)N(C1CCN(C(c2ccc(C(C)=O)cn2)=O)CC1)C c1(NC(C2CC2C(=O)Nc2cc(O)ccn2)=O)cc(Br)ncc1[N+](=O)[O-] N1(C(c2cnc(CC)nc2O)=O)CC2CN(C(c3cc(Cl)no3)=O)CC2(C)C1 C(CCCCCNC(C1CN(C)CCO1)=O)N(C)C(c1cc(Br)cs1)=O c1(-c2onc(C3(N(C)C)CCCOC3)n2)coc2c(F)cc(F)cc12 C(C(CC(C)C)C(=O)N1CC(O)(C(F)F)C1)NC(c1c(C)nc(Br)s1)=O C1(O)(CNC(C2(CC#C)CCOC2)=O)CCCN(C(c2nc(Cl)sc2Cl)=O)C1 C(=O)(C1=CCCS1)NCC1C(NC(CNC(CNC(C)=O)=O)=O)CCC1 N1(C(C(CC[S+](C)C)O)=O)CC2(CCCN(C(=O)CC3CC4(CC4)C3)C2)C1 Cc1cc(C(=O)NCC2CCN(C(c3ncoc3C)=O)C2)ncc1F c1(OC)ccc(Cl)c(C(=O)NC2CCCN(C(=O)Cc3ccc(Br)cc3)CC2)c1 Cc1cc(Br)c(NC(C2CC3CC3N2C(c2cnnc(O)c2)=O)=O)cc1C C(=O)(C(C1=NOC2CC12)N(C1CC2(CCC2)C1)C)NCCC Cn1cc2c(n1)CCCC2C(=O)NCCNC(=O)C1CCCc2ncnn21 c1(NCc2c(C)nc(Cl)s2)cccc2cccc(Cl)c12 N1(C(c2ccc(C)cc2C)=O)CC(NC(=O)Cn2cnccc2=O)CC(C)(C)C1 C1(NC(C(CCOC)C)=O)CN(C(=O)CCCc2nc(C(C)C)no2)CCC1C c1(CCCC)cc(C(=O)NCC2CCCN2C(=O)CN(C)C2CC2)c(C)o1 N1(c2c(=O)cc[nH]n2)CC=CCC12CCOCC2 c1(-c2ccc(=N)[nH]c2)c(C(=O)Nc2ccc(F)nc2F)nc2ccccn12 n1(CC)nc(C(=O)NC(C)C(C)NC(=O)C=Cc2cn(C)nn2)c2c1CCOC2 C1(CNC(C2CN(C(C)C)C2)=O)CC2(CCOCC2)CN1C(=O)C(O)P(C)(C)=O c1(C(N2CCCC(Cc3cccc(C)n3)C2)=O)ccc2c(ccn2C(C)C)c1 c1(C(N2CCC(NC(c3c(C)cn(C)c3)=O)C(CO)C2)=O)cccn2nccc12 c1(C(=O)NC2C=CCN(C(c3n[nH]cc3Cl)=O)C2)cc(C2CC2)nc(Cl)c1 C1(C(=O)NC(CCC)C2CCC2)N(C(c2csc(C)c2C)=O)CCCC1(C)C c1(C(C)C)cnc(CNC(=O)C(N2CCOC(C3(C)CC3)C2)=O)nc1 C1(C(N2CCC(C)(CNC(c3cc(Cl)c[nH]3)=O)C2)=O)CCOC2(CCCC2)C1 C1(Cl)(C(N2CC(CC=C)(C(N3CCC3CC)=O)C2)=O)CCCCC1 c1(C(C)Nc2sc([N+](=O)[O-])cc2N)cc(F)ccc1F c1(C(=O)NC2C(NC(C=C(C)C(F)(F)F)=O)CCCCC2)cnc(C)c(C#N)c1 C(=O)(CCCS(C)(=O)=O)NCC1C(NC(CCn2ncc(C)c2)=O)CC1 N1(C(c2cnc(CC(C)(C)C)s2)=O)CC2CCCC(C1)N2C(=O)COCCCF c1(C(=O)NC(C2CN(C(=O)C(c3ccccc3)N(C)C)C2)C)[nH]nnc1C1CC1 C1(NC(C(CC=C)C)=O)CC2CC1N(C(c1c[nH]nc1-c1ccsc1)=O)C2 N1(C(=O)Nc2ccc(C)c(C)c2)CCC2(CC(C(F)F)=NO2)C1 c1(CC)ncsc1C(=O)NCC1CCCC1C(=O)NOCC(C)C CC(CCCNC(=O)C(C)OC1CCCC1)NC(C1CC1c1ccccc1)=O C(CC1CCC1)(C(=O)NCC1(C(=O)NC(C2CC(F)(F)C2)C)CCC1)OC C1(C(=O)NCC(C2CC2)SC)CCCN1C(C1CCC(C)O1)=O Cc1cc(=O)c(C(N2CC=CC2CNC(=O)C=C(Cl)Cl)=O)cn1C1CC1 C1(C(N2CCC(F)(CNC(CC(CC)C)=O)C2)=O)CC2(C1)CS(=O)(=O)C2 C(CC(C(=O)NC)NC(c1ccc(OCC2CN(C(N)=O)C2)cn1)=O)OC Cc1cc(N)c(C(=O)NC2CC(N(C)C(C3CC3(F)Cl)=O)C2)c(F)c1 C1(C(=O)NC(c2cccnc2)CC)CC12CC(NC(N1CCCCC1)=O)C2 c1(N2CC(C(=O)NCc3cccs3)OCC2)ncnn2cc(Br)cc12 CN1CC(O)CCC1C(N1CC(CC(=O)NCc2nccs2)C2(CC2)C1)=O c1(CC(=O)N(CCC(C)NC(=O)CSCC(F)(F)F)C)cc[nH]c(=N)c1 C1(C(=O)N)CCC2(CC1)CC2.c1(C(NC(C)CCC)=O)ccncc1N(C)C C(=O)(CCCCCCS(N)(=O)=O)N1CCC(C2(NC(C=COCC)=O)CC2)C1 C1(C(N2CCCC(CN(C(=O)C(N)=O)C)C2)=O)CCC2(COC2)OC1 C1(CNC(c2cnsc2)=O)CC2CCC(C1)N2C(=O)CC=Cc1ccccc1 c1(CC)c(C(=O)NC2(C)CC(NC(=O)C(C)P(C)(C)=O)C2)[nH]c2ccccc12 C1(NC(C)=O)COC2(CCCN(C(=O)CCn3ncn(C)c3=O)C2)C1 c1(OC)ccc(C(N2CCC(N(C)C)C(C)C2)=O)c(N)c1 N1(C(c2c(CCCC)ocn2)=O)CCCC(CNC(=O)C(=O)NC2CC2)C1 C1(OC)CS(=O)(=O)CN(CCC2C=CCC(C(=O)OC(C)(C)C)C2)C1 C(=O)(C1COc2ccc(Cl)cc21)NC1C(CNC(C2CCC(C)C2)=O)CCC1 c1(OCC)cc(C(=O)NCC2CCC(F)(F)C2)oc(=O)c1.N12CCC1(C)CC2=O C#Cc1ccc(C(N2CC(C)C2CNC(C2CCCCC2OC)=O)=O)cc1 Nc1cccn(CC(=O)NC2CC(NC(c3cc(Cl)ccn3)=O)C23CCC3)c1=O c1(C(=O)NC2CN(C(Cc3cc(C(C)C)no3)=O)CC2F)ccc(S(C)(=O)=O)s1 C1(NC(=O)NCCN2CCCN(C(=O)C3CC3)CC2)CCC2(CCC2)O1 c1(CC)nc(-n2cccc2)sc1C(=O)NC1CC(C)(NC(c2sc(F)cc2C)=O)C1 CC(=C(Br)Br)NC(CCC)(Cl)c1nnnn1Cc1cccs1 C(=O)(C1=CCC(C)CC1)N1CCC(COC)(NC(=O)C=CC2CCOC2)CC1 Cc1nc(C(N2CCC3(CCCN3C(C3CCC(=O)N3)=O)C2)=O)c2n1CCCC2 c1(OC)ccc2[nH]c(C(N3CCC(F)(F)CC3)=O)cc2n1.C123CC(C1)(C2)CN3 C1(CCC(=O)NC2(C(=O)NC3CCCC3CO)CCCC2)CCC(=O)C1 CCCC(C)(C)C(=O)NCCC1CN(C(=O)Cc2csc3nccn23)CC(C)O1 c1(N(CCC)CCNC(=O)CS(N)(=O)=O)ccnc2nc(C)nn12 NC(=O)CCC(=O)NCC(CNC(c1cccc(OCC(F)(F)F)n1)=O)CO N1(C(C2CCC(CNC(C(C)(C)SC)=O)CC2)=O)CCOC2COCC2C1 C#CC1(O)CCN(C(=NCCc2c[nH]nc2C(=O)OC)NCCOC)C1 N1(C(c2c(C)csc2)=O)CC2CCCC(NC(C3CC(C(C)C)C3)=O)C2C1 CC1=C(C(=O)NC(C2CCCCC2)CNC(=O)CCC(F)F)CCC1 c1(C(=O)NC2CC(N(C(C(C)SCC)=O)C)C2)c(F)ccc(Cl)c1N C1(C(=O)NCC2CC(OC)CN2C(=O)C=C(C)C(F)F)CCc2c(cnn2C)C1 CCC(C)(C)C(=O)NCCCN(C(=O)CN1C(C)CCC1C)C c1(CC)c[nH]c(C(=O)NCC2(O)CC(NC(=O)C(C)OCC(F)(F)F)C2)c1 C1(CNC(c2ccc(OC)o2)=O)CC2CCC1N2C(c1cnnc(O)c1)=O C1(O)(CN(C(C=C(COC)C)=O)C)CN(C(c2csc(C(C)C)n2)=O)C1 N1(CCCC)C(=O)NC(c2csc(NC(C)=O)n2)C(C(=O)OCC)=C1C(F)(F)Cl C(=O)(C(C)CC(C)(C)C)NCC(CO)NC(CC(C)O)=O.CC(C)(C)OCC1CC1 C#CCCCC(C)C(=O)NC1CC2CC1CC2C(N1CC(C2CCCO2)C1)=O O=C(CC1=CCOCC1)NC1CCC(C(=O)NC2CN(CC(F)F)C2)C1 N1(C(CC=CCC)=O)CCC(C2CC2)C1CNC(=O)CCc1cnc(C)o1 CCCC(CCC)C(=O)N1CCOC(C(C)NC(c2ccc(N)c(F)c2F)=O)C1 O(NC(=O)C(C)(CSC)NC(=O)CC(C)C1CC1)CCCC.N1CCCC1 N1(C(C2C(c3cn(CC)nc3)OCC2)C(=O)NCC2CC2)CCC2C(O)CC12 C(C(C(=O)NCC1CC(F)(CNC(=O)C=NOC)C1)C(C)(C)C)OCC=C C1(CC(=O)N(c2ncc[nH]c2=O)C)CC(F)CN1C(C1CN(COC(C)(C)C)C1)=O CC(C)C(C(C1CCCCC1)NC(=O)CCCN1CCCC1)NC(=O)CO N1(C(C(CC)OCC)=O)CC(C=C)(CC(=O)NCCC(C)OC)C1 C(=O)(CC(O)C(Cl)(Cl)Cl)NCC(C)Cc1cn[nH]c1 C1(C(=O)NCC=C)CC(C)(C)CCN1C(=O)C(N1CCOCC1)C C(N=c1cc(C)nc(Cl)[nH]1)C1CC(NC(c2c(OC)cccc2)=O)C1 C(CCC(C(=O)N1CCOC(C(=O)OC)C1)NC(c1ccncc1Cl)=O)OC Cc1ccc2sc(C(=O)NC3CC4CC3N(C(C3(C)CS(=O)(=O)C3)=O)C4)cc2c1 Cc1nocc1C(=O)NC1(CN(C)C)CC1.C12OCCC1C(=O)NC2 C1(NC(CC(C)(C)O)=O)CCCC12CCN(C(=O)C=CC1CCCCC1)C2 c1(CC(=O)NCC2C(C(=O)NCC(CCC)C)CC2)ccc(F)nc1 C(=O)(C1=CCCOC1)NCCCCCCNC(C(c1ccn(C)n1)(C)C)=O C(C(=O)N1CC(C(C)NC(=O)CC(O)C2CCC2)C1)(C(C)C)NC(COC)=O C(CCC(C)C(=O)NCC(C)(C)CC(=O)NCCC1=CCCCC1)OC c1(OC)ccc(CC(N2CCOCC2C(=O)NCc2nc(Cl)sc2Cl)=O)cc1F C(=O)(C1=CC2(CCOC2)C1)NC1CN(C(COCCOCC)=O)CC(C)C1 c1(CCN2CC(CC)OCC2)c(NC(=O)CNS(=O)(=O)N(C)C)ncnc1Cl Cc1ccccc1-n1cc(-c2csc(NC(=O)NC3(C#N)CC3)n2)cn1 CCC(CCC(=O)N(CC(O)(CC)CC)C)NC(c1ccc(O)cn1)=O N1(C(C(c2nc(C)sc2)=O)=O)CCC(CO)C(NC(c2cocn2)=O)C1 CC(C)C#CC(=O)NC(C1CN(C(=O)C(CN(C)C)c2ccccc2)CCO1)C c1(CCC)ncoc1C(=O)N(CCCCCNC(=O)C(O)CN1CCCC1)C N(C(=NCC1C(C(=O)OC)C1(C)C)NC(C)Cc1cccc(F)c1)C(C#C)CC C(=O)(CC(CC)CCCC)NCC12C(CN(C(C(CCCCC)F)=O)C1)CCO2 C1(C(=O)NCC2C(C)(C)CN(C(c3coc(CO)c3)=O)C2)C2CCC3C(C2)CC13 Cc1cc(C(=O)NNC(=O)c2cc[nH]n2)c(C)n1CCC(C)C c1(C(=O)NC2CC(NC(c3cncc(O)c3)=O)C2)c(F)c(F)cc(F)c1F N1(C(COCCCC)=O)CCCC1(C)C(=O)NCC1CC(OC(C)=O)CCO1 Cc1cc2c(C(=O)NC3CC3CNC(=O)CCC3(C)CC3)ccc(C)c2[nH]1 c1(N2C(c3nc(C)[nH]n3)COCC2)ncc(I)cc1Br Cc1cccn2ncc(C(=O)NC3CCCC3c3ccccc3)c12 C1(C(=O)NC2CN(C(C(CC)N(C)C)=O)C(C)CC2)CC2CCC(C1)N2C CC1(C(=O)NCCCN(C(c2cscc2C2CC2)=O)C2CC2)CCCC1O CC1(C)CCCN(C(=O)NC(C(C)(C)O)C2CC2)C1CO C1(CNC(=O)CCCCF)CCC2(CCN(c3nc(C4CC4)ns3)CC2)CO1 Nc1cc(C(=O)NCC(CO)NC(=O)C(F)C(F)(F)F)cc(F)c1Br C1(C(N2CC(C)(OCC(=O)N(CCCCC3CCCC3)C)C2)=O)CC(=O)NC(=O)N1 C1(C(=O)OC(C)(C)C)N(c2ncnc3cnccc23)CC12CCC(F)(F)CC2 c1(-n2cc(C3N(C(C(CC[S+](C)C)O)=O)CCOC3)nn2)ccc(S(C)(=O)=O)cc1 c1(C(N2CCCC(NC(C3C(C)CCC3)=O)CC2)=O)ccc(Br)c(O)c1Br C1(NC(c2c(C(=O)OC)scc2)=O)CCN(C(C23CCCCC2C3)=O)CC1 C1(OCC)CC2(C1)CC2C(N1CCCCC1CN(C(=O)CC(C)(F)F)C)=O C1(NC(C(=Cc2ccco2)C)=O)CN(C(C2CC(C)(C)CN2C)=O)CCC1CO N1(C(c2n(C(C)C)ccc2)=O)CCC2CN(C(=O)C=Cc3ccco3)C2C1 C1(N(C(CCSCCC)=O)C)CCC2CN(C(=O)Cn3cnc(C(N)=O)n3)CC12 N1(C(C=CSC)=O)CC(NC(=O)C(C)N2CCC2)Cc2ccccc21 C1(NC(CC2(C)CC2(Cl)Cl)=O)CCN(C(c2cccnn2)=O)CCC1CO c1(OC)cc(C(=O)NC2CC(O)(CNC(=O)CCCc3nncn3C)C2)sn1 C(=O)(NNc1ccc(Cl)c(C)n1)C(Cc1c(C(=O)OC)[nH]c2ccccc21)=O c1(C(C)=O)ccc(OCCCNC(=O)CN2CCN(c3nncs3)CC2)nc1 c1(C(=O)NCCSCC(=O)NC2(c3ccccc3)CC2)c(C(F)F)cccc1F C(=O)(CC1=NNC(=O)C1)NC(CN(C(C(c1c(C)n[nH]c1C)C)=O)C)C n1(CC(N2CC3C(CNC(C#CC(=O)N(C)C)=O)(C3)C2)=O)ncc2ccccc12 N1(C(C(COC)COC)=O)CCC(C)(NC(=O)CC(C)C2CCCO2)CC1 Cc1ccc(F)cc1C(N1CC(O)CC1C(=O)NC(c1nn(C)cc1O)C)=O CCCC(CNC(=O)Cc1cn(C(C)C)nn1)NC(=O)C=C(CC)CC c1(C(C(=O)NCC(=O)On2cnnn2)N2CCCC2)ccc(C(C)C(F)(F)F)cc1 c1(C(=O)NCC(CNC(CC(CC)C)=O)C(F)(F)F)ncc2cc(Cl)ccn12 O=[N+]([O-])c1cc(Cl)c(Cl)cc1S(=O)(=O)NCC(F)F.c12ccc(cc1)N(CCO)C2 N1(C(c2c(NC)cncc2)=O)CCOCCC1C(=O)NCCC1CCCOC1 C1(CNC(COCC#C)=O)CCCCN1C(=O)CC1CCC(C)CO1 C(=O)(C1CCc2ccccc21)NC1C(C(N(C(C)(C)C)CC2(O)CC2)=O)C1 c1(C(=O)OC)cccnc1NC1CCN(C(=O)C(C)Cc2ccccc2Cl)CC1 N1(C(C(CN(CC)CC)F)=O)CCCC(C)(CNC(c2cnncc2C)=O)C1 C1(NC(C(C(CC)O)C)=O)CCCC12CN(c1ncnc(C(C)(C)C)n1)C2 CC1(O)CCC(CC(N2CCN(Cc3cc(F)ccc3F)C(CF)C2)=O)CC1 C1(N(C)C(C2CC(F)(F)C2)=O)CCCN(C(c2cc[nH]n2)=O)C1 N1(C(C2(CF)CCN(C(c3cc(C)cc(C)c3)=O)C2)=O)CC2CCCCC2C1C C1(NC(C(=O)NCCOCCCC)=O)CCN(C(c2ccccn2)=O)C(CC)C1 N#Cc1ccc(CN2CC(C(=O)NCCC3CC3)CC(F)C2)c(Br)c1 c1(CC(=O)NCCCN(C(=O)COCCOC)CC)ccc(OC)cn1 c12cc(ccc1I)C(=O)N(C)C1CCN(C1)C2.c1(COC)c[nH]c(C(=O)O)c1 c1(C(=O)NC2CCC(F)(CNC(CC3(C)OCCO3)=O)C2)c(F)ccc(F)c1F n1(C2(C(=O)NC3CC(NC(CCN(C)CC)=O)C3)CC2)cc(Cl)cn1 C1(NC(c2c(CC)ncs2)=O)CC2CCC1CC2NC(=O)CCc1ncnn1C C1(C(N2CCC2CC(=O)N(C(C)CC(F)F)C)=O)(OC)CCOC1 O=C(C#CC1CCOCC1)NCC12CCC1CCN2C(C1CC(O)C1)=O c1(C(N(CC(C)NC(c2cccc(Br)c2)=O)CC)=O)cccn2nccc12 c1(COC)ccc(C(=O)NC2CCC(NC(C3CCNC(=O)C3)=O)C2)cc1F c1(C(=O)NC)ccc(C(=O)N(CC(O)CN(C)C(c2nnc(C)s2)=O)C)cn1 c1(C(=O)NCc2cccc(CNC(C(CC)(C)C)=O)c2)c(N)sc2c1CCSC2 C1(NC(C(CC)n2ccnc2)=O)CCC(C)N(C(c2ccc(Br)cc2)=O)C1 C1(COC)CCCCN1C(C1C=CCN1C(=O)CCCC1CCCC1)=O N1(C(CC(CC2CC2)NC(Cc2cc(C)on2)=O)=O)C2CCCC1CN(C)C2 C1(n2cnnn2)(CC(=O)NCC2(C(C)NC(C3CCSC3)=O)CC2)CS(=O)(=O)C1 N1(C(=O)CCc2ncccn2)CCC2CCN(C(C3CCCC3F)=O)C2C1 C1(C(N2CC(OCCOC)C2)=O)CC(C)N1C(=O)CC1CC2CC2C1 N1(C(C2(C)CCOC2)=O)CC2(NC(=O)COC3CC=CC3)CCC1CC2 C(=O)(CC1(O)CCOc2ccccc21)NCC(C)NC(CCCC#C)=O C1(C(N(C)CCNC(=O)CCn2ccnn2)=O)CCCCN1S(N)(=O)=O C=CCC(CC=C)C(=O)NC1CCN(CCCNC(=O)C(O)P(C)(C)=O)C1 C1(NC(=O)CC2(CO)CC2)CC2(CCCN(C(c3csc(Cl)c3)=O)C2)C1 C12CC(C)N(C1)C2.C(c1cnc[nH]1)=C(C)COC Nc1ccc(C(N2CCCC(n3cccn3)C2)=O)c(F)c1 C(=O)(C(O)CCCC)NCC1CN(C(CCC)=O)CC1c1ccc(OC)cc1 c1(N(C(c2c(C)ccc(CC)c2)=O)CC)cn2c(C)cc(C)nc2n1 C=CCC(C)C(=O)NCc1ccc(CNC(C2(C(C)(C)O)CCC2)=O)cc1 C1(C(=O)NC2CN(C(=O)C=C3CCC3)CC23CC3)CC(c2ccc(F)cc2)=NO1 C(C(C)(C)CC(=O)NCC1CCC(NC(C2CC(C)(O)C2)=O)CC1)NC(=O)OC C1(C(=O)NCCN(C)C(c2cc(Br)ccc2N)=O)CN2CCCCC2CO1 c1(C(=O)NC(C)CC2CN(C(C3(C)CC4(CCC4)C3)=O)C2)cnc2occc2c1 N1(C(C(C)C2CC2)=O)CC2CC1C2NC(c1cccc(C2CC2)c1)=O c1(CCCN2C(CC(=O)NCC3(CO)CCC3)COCC2)ccc(Cl)cc1O CCCCC(C)C(=O)N1CCCC(CCC(N2CCN(CC(N)=O)CC2)=O)C1 C(=O)(C1SCCc2ccccc21)N1CC2(N(C(c3n(C)ccn3)=O)CC2)C1 C(=O)(C1=CC2CCC(C1)C2)NCCC1(O)CCN(C(CCc2ncn(C)c2)=O)C1 c1(C(N2C3CC(CNC(c4c(CC)cco4)=O)C2CC3)=O)cc2cccnn2c1 C1(NC(C(F)OC)=O)CS(=O)(=O)N(C)C12CCN(C(=O)C(C)C)CC2 C1(C(=O)NCC(CN(C)C(C23CCC2C3)=O)O)CCOCC1 c1(NC(c2nc(C(=O)OC)oc2)=O)ccc([N+](=O)[O-])cc1Cl C=CCCC(C)(C)C(=O)NC(c1nocc1C(=O)NC1CC(C)(C)C1)C C1(C(=O)NCC(CC)(C)Cl)CC(O)CN1C(c1nccnc1C)=O O=C(CCC(F)(F)F)NC(CNC(C1(C(F)(F)F)CCCC1)=O)C1CCC1 N1(C(c2n(C(C)C)ccc2)=O)CCC2(NC(=O)CCOC3CC(F)(F)C3)CC2C1 c1(C(C)C)n[nH]c(=NC2CCN(C(=O)CCc3cc(Cl)cs3)CC23CCC3)o1 N1(C(C(c2ccccc2)NC(C)=O)=O)CCCN(C(c2cc(C)n(C)c2)=O)CC1 C(=O)(CCCC(C)C)N1CC(CCNC(C(CCSC)OC)=O)OCC1 C(CCC(N)=O)(C(=O)N1CCC(CNC(c2cnn(C)c2)=O)C(C)C1)NC(C)=O Cc1cccc(O)c1C(=O)NCc1ccc(CCNC(C2CC2CF)=O)cc1 c1(C(=O)NCC(O)CNC(C2CCS2(=O)=O)=O)ccc(N2CCOCC2)cc1F C1(C(=O)NC2CC(O)(CNC(c3ccco3)=O)C2)CCc2nnc(O)cc2C1 C12(C(=O)NCC(C(=O)OCC)C)CC1CCN2C(=O)Cn1cnnc1 c1(C(N(CC(CNC(C(C)NC(=O)C2CC2)=O)O)C)=O)cc(O)cs1 c1(CN2CCC(C(O)CCc3cn(-c4ccc(F)nc4)nn3)C2)c(Cl)cncc1Cl C(C(=O)NC1(C)CN(CC(N2CCC(CCO)(CO)C2)=O)C1)(C(C)C)SC C1(C(=O)NCc2cccc(CN(C(=O)C(C)(C)O)C)c2)CC2(CCC2)C1 c1(C(=O)Nc2cc(OC)c(C)cc2C)csc2c1CCN(Cc1[nH]ccc1C)C2 c1(C(N2C(C)CC(NC(c3cnc(S)nc3)=O)CC2)=O)nccc2c1NCCC2 C1(C(=O)NCC2CC2C2CCCO2)(CO)CCS(=O)(=O)CC1 c1(CNC(C(CC)NC(=O)C(O)C2CCCC2)=O)cncc(C)c1 c1(C(=O)NC2CN(C(c3cc(C)c(C)[nH]3)=O)C(C)CC2)n[nH]c2c1NCCC2 c1(NC(CCC2N(C(c3c(C)cco3)=O)CCC2)=O)cc(C(N)=O)ccn1 N1(C(CC(CNC(C(C=C)(C)C)=O)C2CCC2)=O)CC2(CNC(=O)OC2)C1 c1(C(N(C)CC2(O)CN(C(c3scc(OC)c3)=O)C2)=O)c(OC)n[nH]c1C C(C(=O)NC(C)(C)C=CC(=O)NOc1ccc(F)cc1)(C(C)C)OC C1(NC(CCSCCC)=O)CN(C(C2CN3CCC2C3)=O)CC(C)(C)C1 CC1CN(CC(O)COCC(C)C)CCN1C(c1coc(C2CCOCC2)n1)=O CS(=O)(=O)c1ccccc1CN1CCCC(C(=O)NCc2c(Cl)cccc2Cl)C1 c1(OC)cc(F)c(F)cc1C(N1CC2CC1CN2C(c1cc(O)cc(=O)o1)=O)=O Cc1cccc2c(C(N3CCC(NC(c4cc(=N)[nH]c(Cl)n4)=O)C3)=O)n[nH]c12 N1(C(C=CC(C)C)=O)CCN(C)CC1CNC(c1[nH]c(=N)ccc1C)=O N1(C(C(CC)(C)O)=O)CCC(C)(Nc2ncc(F)cn2)CC1 Cc1cc(CNC(=O)CC2(C)CCN(C(C3C4CN(C)CC34)=O)C2)ccc1F Cc1cc(C)nc(N2CCCC(NC(=O)Cn3ccnc3C)C2)n1 c1(C(=O)NCCN(C(C(C(=O)OC)(C)F)=O)C)ccc(O)c(C)c1C Cc1csc(C(=O)NC(c2ccc(C(N3CC(F)(F)C3)=O)cc2)C)c1C c1(OC)ccc(CC(=O)NCCN(CC(C)O)C(=O)Cc2ccoc2C)cc1F N1(C(C(CCC)C(=O)OC)=O)CC2(CCCCN2C(=O)CC(C)C(F)F)C1 CC(C)C(C(=O)NCC1C2CC1N(C(=O)CC(C)c1cccs1)C2)n1cnnc1 C1(C(C(=O)C(C)(C)F)=O)CN(C)CCO1.C(=O)(C(C)C(=O)OC)NCCC Nc1cc(Cl)cc(Cl)c1C(=O)NC1CCC1NC(=O)C=C1CCSCC1 C1(C(C(=O)N(CC#C)CCO)C)CCN(C(c2ccn(C(F)F)n2)=O)C1 c1(CC)nc(C)[nH]c1C(=O)NCC(C)N(C(=O)CCC1CC1(Cl)Cl)C n1(CCC)nnnc1C(c1ccoc1C)NC(C)C(=O)OC(C)(C)C C1(NC(=O)CCn2cncn2)CC2C(NC(=O)CC3CCCNC3=O)C2C1 Cc1cnc2c(S(=O)(=O)NC3COC4(CCC4)OC3)cccc2c1 N1(c2ncc(C#N)cc2Cl)CCC2(CC(C(=O)N=c3occ(Br)[nH]3)=NO2)C1 N1(C(CSC2(c3n(C)ccn3)CCC2)=O)CCN(C(C2C3CCCC23)=O)CC1 c1(C(N2CC3C(CN(C(=O)Cc4nc[nH]n4)C)(C3)C2)=O)c(Br)ccc2c1OCO2 c1(CC)oc(C)cc1C(=O)NC(CN(C(C1(C(F)(F)CC)CC1)=O)CC)CC c1(NS(C)(=O)=O)ccc(C(=O)NNC(=O)c2ccc(N(C)C)cc2)cc1[N+](=O)[O-] Cc1nc(C(N2CCC(O)(CCNC(C3(O)COC3)=O)C2)=O)c(C)s1 C1(CC)CCCC1(C)C(N1CCC(CF)(NC(c2ccc(C(C)C)[nH]2)=O)C1)=O CC1CC(C)N(C(=O)CNS(C)(=O)=O)CCN1C(c1ccc2nc(O)[nH]c2n1)=O C#CC1(O)CC(C(N2CCC(C)C2CNC(c2snc(O)c2Cl)=O)=O)C1 C#Cc1cccc(CC(=O)N(C(C)CNC(C2CC3CCCC23)=O)C)c1 N1(C(C2CC(C)(C)O2)=O)CCC(O)(CNC(=O)CCc2ccccc2)CC1 N1(C(c2ccc(F)c(F)c2)=O)CCOC2(CCN(C(C3CCC=CCC3)=O)C2)C1 C(=O)(C(C(=O)OCC)C(C)C)NC(c1ccccc1F)CNC(CCC)=O.OCC Cc1cc(=NCC2COC(=O)O2)[nH]c(Cc2ccc(OCCCN(C)C)cc2)n1 c1(CCC(=O)NC2(CC=C)CN(C(c3ccncn3)=O)C2)c(C)noc1C C1(CC(=O)NCc2ccc(C(=O)NCC(O)C(F)F)s2)CCCC12CC2 C12(C(=O)NCC(N(C(c3c(C(C)=O)cccc3)=O)C)C3CC3)CC3CC1C2C3O c1(C(=O)NCC(CC)NC(C2CC(F)(CO)C2)=O)cncc(F)n1 S(=O)(=O)(c1cccc(F)c1)NCC(=O)NC1CCC(CNC(C2CC23CC3)=O)C1 N1(C(c2c(C)cc[nH]2)=O)CC2OCC(NC(c3cccn4nccc34)=O)C2C1 C1(C)(CC)C=C(C(=O)N2CCCC(CNC(c3cc(CSC)ccc3Cl)=O)C2)C1 CC1=C(C)CC(C)(C(N2CC(CNC(=O)C=C(Cl)Cl)C(C)(C)C2)=O)CC1 N1(C(C(CC(N)=O)NC(CCC(=O)NCC)=O)=O)CC2(CCCN2C)C1 C(C1CS(=O)(=O)c2ccccc21)OC(c1ccc2c(c1)NC(=O)C2)=O CC(C)C(C(=O)N(CCC(C)NC(C1CC(C2CCC2)C1)=O)C)C(C)C c1(C(=O)NC2CCC(NC(CCC(=O)OC)=O)C2)cc(Cl)ccc1-n1cncn1 c1(C(N2C(CN(C(C=C(CC)C)=O)C3CC3)CCC2)=O)ccc(C)c(C)n1 C1(C(=O)NCC23CCC(CC2)C3)COCCN(C(C2(CCCF)CC2)=O)C1 Cc1ccc(CNC(=O)C(C)NC(=O)Cc2cnccn2)c(F)c1 c1(NC(C2CN(C(=O)CC3CC3)CC(F)(F)C2)=O)ccc2nnnn2c1 c1(CC)sc(C)cc1NC(C1CCCCN1C(=O)CCN(C)C)=O N1(C(CCOC)=O)CCCC2(CC(NC(c3nc(C)c(C)[nH]3)=O)C2)C1 Cc1cccc2cc(C(=O)NC3CCN(C(=O)CC4CCOC4)C(C)C3)[nH]c12 N1(C(CCc2n(C)cnn2)=O)C2CCC1CN(C(c1cc(C(N)=O)n(C)n1)=O)C2 C1(NC(CN2CC(C)(C)C2)=O)CCCCC1C(=O)NC1CC1NC(=O)C(F)(F)F C1(C(N2CCC3C(C2)CN3C(C2CC(O)C2)=O)=O)CC12C1CC3CC(C1)CC2C3 C#CC1CC2(CC2)CN1C(c1ccnc(CNC(=O)C(C)(C)CC(F)F)c1)=O CC1CC(C(=O)NCCC2CCCN2C(c2cnc(-c3cnccn3)s2)=O)=NO1 N1(C(C(=O)OCC)=O)C2CC1CN(C(c1sc(C)nc1C(C)(C)C)=O)C2 N1(C(CCCC(=C)C)=O)CCCCCCC1C(=O)NC1CCC(=O)NC1C c1(C(N2C(C(=O)NOCCCCF)CCC2)=O)ccnc2cc[nH]c12 C1(CC(=O)NCCCCC#CC)C2CCC(C2)N1C(c1cc(C)nn1C)=O C1(OC)C(N=c2[nH]c(=NCCS(=O)(=O)CC)[nH]c3c2CCC3)CC12CCC2 C1(NCCSC)CN(C(=O)C=Cc2nccs2)CCC1F C1(COC)CN(C(=O)C(C)C)CCN1C(c1nn(C)cc1C)=O CC1=C(C(=O)N2CCC(NC(C3CC(F)(F)C3)=O)CC(C)(C)C2)C(C)(C)CCC1 C#Cc1cc(F)c(C(=O)NC2CC3(C2)CC3NC(c2ccn(C)n2)=O)c(F)c1 N1(C(C(CSC)O)=O)CCCC2CN(C(=O)CN(C)Cc3ccccc3)CC12 c1(C(=O)NC2C3CN(Cc4cn(Cc5c[nH]cn5)nn4)CC23)ccc(N)cc1Cl c1(C(=O)NC2(SC)CN(C(CCOC)=O)C2)ccc(C)cc1OCCO C1(CC(=O)NC2CCC(C)(CCCC)O2)C2CCCC2CN1C(=O)OCC(C)(C)C C1(CC)CN(C(c2c[nH]c(C#N)c2)=O)CC1C(=O)NCC1CC1(Cl)Cl Cc1ccc(C(=O)NCC2(CNC(=O)C(C)C(C)O)CCCC2)cc1Cl c1(CSC)cc(C(=O)NC(C)C(C)(C)NC(C23CC4CC2C3C4O)=O)ccc1F Cc1cc(Br)cnc1C(=O)NCC(CC(F)(F)F)NC(C1CC1F)=O C1(OC)CCCN(C(=O)CC(C(C)C)NC(=O)CCC(C)SC)CC1 C1(NC(c2coc(O)n2)=O)CC2CN(C(C3CC34CCCC4)=O)CC2C1 C(=O)(N=c1ccn(C(F)F)[nH]1)C1(C)N(C(COCC(=O)NC)=O)CCC1 CN1CCN(CC(=O)NC2(C(=O)NCC3C(C(=O)NCCO)C3)CCOC2)CC1 O=C1N(C(=O)Cc2ccc3ncsc3c2)CCOC12CCOCC2 C(C(CC(F)(F)F)NC(c1ccnn1C1CC1)=O)NC(c1c(C(C)C)[nH]cc1)=O C(=O)(C1=C(C2CCOCC2)N(C2CC2)C(=S)NC1c1ccc(F)c(F)c1F)OC c1(NCC(CCCCC)O)ncc(C)cc1S(=O)(=O)N1CC2CCOC2C1 Cc1cc(C(=O)NC(CCNC(c2csc(Cl)c2)=O)C(C)C)nn1C1CC1 c1(C(N2C(CO)CC(NC(CNS(CC)(=O)=O)=O)C2)=O)cc2ccsc2n1C N12C3CCC(C3)C1NC(=O)c1c(cccn1)C2=O.C1(OCCN)CCCCC1.CO CCC(CC(=O)N1CCCCC1CCNC(=O)C(C)N(C)C)C1CCC1 c1(C(N2CCCC(NC(CCCC(N)=O)=O)(CO)C2)=O)cn2c(n1)CCCC2 C(C(C)CC(=O)NCC1(C(=O)NOCC=C(C)C)CC2(CC2)C1)OC c1(CC)ccccc1OCCOCC(=O)NCCN(C(=O)C(C)CO)C(C)C N1(CC)N=C(C(=O)N2CCCC(C)C2CNC(=O)CCCCC(C)C)CCC1=O c1(C(=O)Nc2c(CNC(C3C(C(=O)OC)C3)=O)cc(Cl)cc2)cccc(Cl)c1C c1(C(N(C2CCN(C(C(C(C)O)C)=O)CC2)C)=O)cc2c(cn1)OCCO2 C12(C(N(C3CCN(C(c4nnnn4C)C)C3)CC)=O)CC(C)(C1)OC2C c1(C(=O)NC2CN(C(C(CC=C)C)=O)C(C)C2)noc2cc(Br)ccc12 Cc1cccc(C2(C(=O)NCC(CO)NC(c3cccnn3)=O)CCC2)c1 c1(CC)nnc2n1CCC2.C12CN(CC1O)C(=O)c1cnn(c1C)-c1cn2nn1 CONC(=O)CN.C(C(C(=O)N(C)C)N(C)C)NC(C1CC(=C2CCC2)C1)=O c1(OC)ccc(NC(=O)NNC(=O)c2cc(Br)nn2C)cc1 N1(C(C(C)C)=O)CCCC1C(N1CCC(CCNC(c2coc(O)n2)=O)C1)=O c1(C(=O)OCC)ccc2c(c1)CC(NC(=O)C(=O)NCCCCCCCO)C2 CC1CN(C(C2CC3C=CC2C3)=O)CCC1CNC(=O)CC1COC(=O)N1 c1(CNC(c2scc(C)c2)c2nnnn2C2CCCC2)cc(F)nc(F)c1 Cn1c(=O)sc2cc(C(N3CCOCC3)CS(=O)(=O)c3ccc(Br)cn3)ccc12 C12CCCC(C1)C2.C1(=CCC)CCN(C(C2CCOC2)OC)C1 CC(CCc1ccccc1F)C(=O)N(CCCNC(=O)COCC1CCCC1)C c1(N2CCOCC(C(N(CCCCCC=C)CC)=O)C2)ccc2nc[nH]c2n1 CC1CCCC1(C)C(N1CCN(c2cccc(-c3nn[nH]n3)c2)CC1)=O c1(C(=O)NC(C(=O)NC2CCN(C(C)=O)C2)Cn2cncn2)cc(C)c(F)cn1 N1(C(C(N2CCOCC2)C)=O)CC(CNC(c2nn(C)cc2N)=O)CC12CCC2 N1(C(C(CSC)O)=O)CC(NC(c2ccc[nH]2)=O)C(CC(C)(C)C)C1 C=CC1CCCCN1C(=O)C(CC=C)NC(=O)C=Cc1ccnn1C N1(C(C(CC)CC(C)C)=O)CCC(NC(=O)CCCCC(C)C)C2(CCC2)C1 C(=O)(C1=NOC(CNC(c2cn(C)cc2C)=O)C1)N1CC(OCC(=O)NC)C1 C1(NC(c2c(O)nc(CC)c(C)c2)=O)CCC2(CC1)CN(C(=O)C(C)(C)F)C2 c1(C(=O)NCC2CN(C(C(C)(CO)OC)=O)CC2C)cc(S(N)(=O)=O)co1 C(=O)(C(O)C(C)C)N1CC(OCCNC(c2n(COC)ncc2)=O)C1 c1(C(N2C(CNC(C(C=C)(C)C)=O)C(C)(C)CC2)=O)ccc2c(c1)CCN(C)C2 c1(C(CO)NC(CCOCCCNC(C(C)C2CCC2)=O)=O)ccccn1 C=CCC(C)(C)CC(=O)NC1CCCC1CNC(=O)COC(C)(C)C N1(CC(=O)NC2CC(CCNC(=O)CC3CCCC3O)C2)CCC(O)CC1 N1(C(CCC=C=C)=O)CC(CNC(=O)CC2CCC(=O)NC2)C2(CCOCC2)C1 N1(C(CNC(C)=O)=O)CCC2CN(C(=O)COc3ccc(F)c(F)c3)CC2C1 N12CC(C3(CCC3)C1)C2=O.c1(C(=O)NCC2OCC(C)(C)C2)cncc(C#N)c1 N1(C(C2CCC(C(=O)OC)CC2)=O)CCC(C)C(NC(=O)Cc2nnc(C)s2)C1 CC1CC(NC(C2(C)CC(C)(C)C2)=O)CCN1CCCN1C(=O)CNC1=O S(=O)(=O)(c1cccc(=NCC(O)c2ccccc2F)[nH]1)NCC(CCC)OC N1(C(CCc2cnc(C)o2)=O)CC(O)CC1C(=O)N(C)CCN1CCCCC1 N1(C(CC2(C#N)CCC2)=O)CCCC2(CCCN2C(=O)CCn2cnnn2)C1 C(=O)(N=c1ccn(C2CCCCO2)[nH]1)c1c(C2CC2C(F)(F)F)cc(OC)nn1 Cc1ccc(O)nc1CNC(=O)CN(CC(C)C)C(C1CC(=O)C1(C)C)=O C(=O)(CC1=NNC(=O)C1)N1CC(OCCNC(C2(C(=O)NC)CCOCC2)=O)C1 S(=O)(=O)(c1ccccc1)NCC(=O)NCC1(C(C)NC(=O)C2=CCC2)CC1 N1(C(C(CCCOC)C)=O)CCCN(C(=O)C(F)(F)CN2CCCC2)CC1C N1(C(C(CC=C)(C)C)=O)CCC(C2(NC(C3(SC)CCC3)=O)CC2)CC1 C(=O)(CCCCCC(C)O)NCC(CN(C(c1cncc(COC)c1)=O)C)C Cc1nc2ccccn2c1C(C(=O)NCCC#N)N(C1CCCC(C)C1)C c1(OC)cccc(C2N3C(C=CC3)CNC2=O)c1.c1(C(=O)NC2CC2)ccco1 c1(C(=O)NC(CNC(C=CC)=O)(C)C2CC2)ccc(CCc2ccccc2)[nH]1 n1(CCCC)nc(C)c(C(N2CC(O)(CNC(=O)CC3CCOC3=O)C2)=O)c1Cl C(=O)(CCCC1CCC1)NC1(C(=O)NCC(C2CCOC2)OC)CCC1 CCCCCCC(C)C(=O)N1CC2(C1)CN(C(=O)Cn1nc(C)nc1C)C2 C1(CCNC(=O)Cc2cnccn2)COCCN1C(=O)Cc1cncs1 C1(CNC(CCCc2onc(C)n2)=O)CCC(CNC(=O)C(C)C(C)O)CC1 n1(CC)nc(C2CCC2)cc1C(=O)NCC1CC(NC(=O)CCSCC(C)C)C1 C1(C(=O)NC2CN(C(C3CCC(C)CC3)=O)CC2O)CCCC2(CC2)C1 c1(CC(=O)N(C)CC2CCN(C(C3CC(F)(F)C3)=O)C2)csc2nccn12 C1(C(F)(F)F)(C(=O)NC2CN(C(c3cc(C(F)(F)F)c[nH]3)=O)C2)CC=CCO1 CON(CCO)C(=O)COC1CN(C(=O)C=C(C2CC2)C2CC2)C1 C1(NC(=O)COC)CCC(NC(=O)CCCF)C1.c1(C(=O)NCC=O)ccco1 c1(C(=O)NCC2CC(NC(CC(=C)C)=O)C2(C)C)ccc(F)c(F)c1F N1(C(c2c(C)scc2)=O)CCN(C(=O)C(C(C)C)n2ncc(N)n2)C2CCC12 c1(OC)ccc(C(C(C)OC(c2ccc(-n3cccn3)cn2)=O)=O)cc1 C#Cc1cn(C)nc1C(=O)NC(C)CCCNC(c1cn(CC)nc1C1CC1)=O C1(CC(=O)N(CCN2CCCC(C)C2)CCO)CCN(CCCCO)CC1O.CO C(=O)(C1(C)CCCc2ccccc21)NCCN(C(=O)C#CC(C)(C)O)CCC C1(NC(C2CC3CCC3C2)=O)CCN(C(=O)C(F)(F)C2(O)CCCC2)CC1 c1(CN(CCCCCC=C)Cc2ccc(F)cc2)cccn(CC)c1=O CC(C)(C#N)CCCC(=O)N1CCC(NC(=O)C=C(Br)Br)C1 Cc1ccn(CC(=O)NCC2(O)CN(C(c3ccnn3CC(F)F)=O)C2)c(=O)c1 CCC(CC)C(C)C(=O)NCCCCNC(c1cnc2sccn12)=O c1(C(=O)NCc2c(CCNC(C(CC)OC)=O)ocn2)nnc(O)cc1O C1(NC(C(c2cncnc2)C)=O)CCCC(C(=O)NC2(CCF)CC2)C1 c1(N(C)CC)nnc(N(C)CCC2CC2)n1CC(=O)OC(C)(C)C N1(C(C=C(C)C2CC2)=O)CCC(C2CCCN(C(C3CC3(F)F)=O)CC2)CC1 c1(C(=O)NCCCNC(C(n2c(C)cc(C)n2)C)=O)ccc(C(C)(C)C)cc1N CC1(C)CCC(N)C2N1CC(=O)NC1C2=CC=CC=CCC1O N1(C(C(C)=C(CC)C)=O)CCC(CNC(c2nc3ccccn3n2)=O)C12CCC2 N1(C(C2(CCN(C)C)CC2)=O)CCC(O)C(C(=O)Nc2cccc(CO)c2)C1 c1(NC(C2N(Cc3n[nH]c(C)c3C)CCC2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 c1(C(N2C(CNC(c3c(OC)n[nH]c3)=O)C=CC2)=O)ccc(C)c(CO)c1 c1(NC(CC2N(C(c3nc(C(C)C)sc3)=O)CCC2)=O)ncc(Cl)nc1Br C1(C(=O)OCC)(NC(=O)CCN(CC(F)(F)F)C)CCCN(C(=O)C(C)(F)F)C1 CCCCCC(O)CC(=O)NC(C)CCCNC(c1cc(F)cc(Cl)c1)=O c1(C(N2CC(NC(C3CCCS3)=O)CC3(C2)CC3)=O)cc(F)c(F)c(O)c1F C1(CNC(=O)C=Cc2ccco2)CC2CCC(C1)N2C(=O)CCC(F)F c1(C(=O)NC(CN(C(C2(CC#C)CCOC2)=O)C)C)cc2nnn(C)c2s1 C1(C)(CCC)CCN(N(C(C)c2ccccc2)CCO)C1 C1(C2CC2)(NC(C(F)=C(C)C)=O)CCN(C(c2ccc(Cl)cc2)=O)C1 c1(C(=O)Nc2ccnc(C(N3CCC(O)CC3)=O)c2)ncn2c1CCCC2 Cc1nocc1NC(=O)C(C1CCN(C(=O)CC2(C)OCCO2)C1)F c1(C(=O)NC2CC3CCC2N3C(=O)CN2CSCCSC2)cc2cccnn2n1 c1(C(=O)NC2CN(C3CN(C(CNC=O)=O)C3)C(=O)C2)csc2cncn12 Cn1nc2c(c1C(=O)Nc1ncc(Br)nc1I)CN(Cc1ccccc1I)CC2 C(=O)(C1=CCCOC1)NC(CN1CCN(C(C2C(OCC)C2)=O)CC1)(C)C C1(CCC)CN(C(c2ccc(Cl)o2)=O)CCN1C(=O)CCC1CCC(=O)N1 N1(c2ncc(OC)cn2)CCC2CN(C(c3c(F)ccc(C)c3Br)=O)CCC12 N1(C(c2cccc(OC)c2N)=O)CCC2(COC(CNC(C3CC3(C)C)=O)C2)C1 C1(NC(C(c2ccccc2)NC(CC)=O)=O)CCOCC1NC(=O)CCSC1CC1 c1(CNC(=O)NC2CC(CN(C)C)OCC2)cn(CCO)c(=O)nc1O c1(C(=O)NC(CNC(C(CC)(C)C)=O)(C)CC)coc2c1CS(=O)(=O)C2 Cc1sc(C(N2CCCC2CCNC(=O)C(C)CC2CCCCC2)=O)nc1O c1(CC(N2CCN(C(C(CC)F)=O)C(C3CC3)C2)=O)cccc2nonc12 N1(C(C)NC2CCCN(c3cc(-n4ccnc4)ncn3)C2)C(=O)NC(C)(C)C1=O C(=O)(C1=COCCC1)NC(C(=O)NC(CCSC)C)C1CCC1 C1(C(=O)NCCCCCn2cc(-c3c(C)cncn3)nn2)CC(=O)NC1(C)C C1(C(=O)NCC2(CC(C)C)CC2)CCC(C)(C)N(C(C2CCCN2C=O)=O)C1 CCC(C)C(C(=O)N(C)CCOCCNC(=O)Cn1nnc(=N)[nH]1)OC c1(C(N2CCCC(CC(=O)NC3CC3)C2)=O)ccc(N2CCCC2)nc1 N1(C(c2cc(C)on2)=O)CCCC12CCCN(C(c1cc(Cl)cn1C)=O)C2 CN1CC(=O)Nc2ccc(C(=O)N(C)CO)cc21.C12(C(N3CC(O)C3)=O)CC(O)C1C2 CCC(C(=O)N(CCCNC(=O)Cc1cnn(C2CC2)c1)C1CC1)OC C1(CCC(=O)NC2(CC=C)CC2)CCCN(C(C2CC2(C)C(F)F)=O)C1 C1(CC#C)(C(=O)N(C)CCc2cnn(C)c2)CCN(C(c2cc(Cl)no2)=O)C1 C(CCCC(=O)N1CCC(NC(c2cc(CS(C)(=O)=O)c(C)s2)=O)CC1)OCC CC1=C(C)CC(C(=O)N(CCC(=O)Nc2cnc(C)c(C)c2)C)CC1 C1(OC(c2cc(C(C)(F)F)c(Br)cn2)=O)CCCC12CCOCC2 n1(CC)c(S(=O)(=O)N2CCC2CCC(=O)O)cnc1C c1(C(=O)NCc2nc(-c3sccc3-c3ccccc3)cs2)cc(O)ccc1Cl c1(SCC=C)ccccc1C(=O)NC1CCC1CNC(c1ccccc1SC)=O CCC(CC(=O)N(C)CC1(O)CCN(C(=O)CC2(C#N)CCCCC2)C1)C(C)C C1(S(C)(=O)=O)(C(N2C3CC(CNC(CC(C)(C)C)=O)C2CC3)=O)CCOCC1 C1(C(N(CCNC(c2cc(NC=O)no2)=O)CCOCCO)=O)C2COCC12.CO N1(C(c2c(C)cnn2C)=O)CCCN(C(C2CC2C)=O)C(c2ccccc2)C1 c1(C(N(C2CCN(C(=O)C(C)CO)CC2)CC)=O)noc2ccc(Cl)cc12 N1(C(C(C(C)C)=O)=O)CC=C(C(C)(C)C(=O)NCCCCCC2CC2)C1 c1(CC(=O)NCCC2(NC(c3cnc(C)c(N)c3)=O)CC2)cc(Cl)c(F)cc1F c1(N(C(CCC)CO)CCOC)cc(Br)ccc1S(=O)(=O)Nc1cc(C)cc(C)n1 CN=c1[nH]cc(C(=O)NC2CC2CNC(c2ccc(OC3CC3)cc2)=O)s1 C12(C(=O)NC(CC)CO)CCC(C(=O)Nc3cc4ccccc4s3)(CC1)CC2 c1(N2CC(C)C(NC(=O)CC3CCCC3(F)F)CC2)ncnc2sc3c(c12)CCC3 C(CC(C)(C)CNC(=O)CCCOc1ccccc1F)NC(C(CC)O)=O CCC(C)C(C(=O)N1CCC1Cn1cc(-c2ccc(OC)c(N)c2)nn1)N(C)C C1(C(N2CC3C(NC(=O)COCc4ccccc4)(C3)C2)=O)CCCCCCC1 C1(CCC2N(C(CC3(C)CC3)=O)CCC2)CCCCN1C(c1cc[n+]([O-])cc1)=O CCCCCC(C)(c1nnnn1C1CCOC1)NCc1cc(Cl)cs1 Cc1nn(CC(N2CCCC2CNC(c2cscc2C(F)F)=O)=O)c(=O)n1C n1(CC(=O)NCC2CC(F)CN2C(c2cnsn2)=O)cccnc1=O N1(C(c2cc(C)ns2)=O)CC(C(=O)NCc2nonc2C)C2(CCC2)C1 c1(C(=O)NCC2CN(C(C3C(C(=O)OCC)CC3)=O)CC2C)nnc(O)nc1O CC1CN(C(=O)CCS(C)(=O)=O)CC(C)C1NC(=O)C=CCN1CCCCC1 C(CC(C(=O)N(C(C)(C)CC(=O)N(C1CN(C)CC1O)C)C)OC)OC c1(C(N2CCN(C(CC(C)(C)O)=O)C(C#N)C2)=O)cccc([N+](=O)[O-])c1Cl CC1=C(C)CC(C(=O)N(C(C)CN(C)C(c2cn(C)[nH]c2=N)=O)C)CC1 C12(C(=O)NCC(C)(CO)NC(c3ccc(O)nc3Cl)=O)CC3CC(CC(C3)O1)C2 C12(NC(CCC(C)(C)F)=O)CCN(C(=O)CCn3cnccc3=O)CCC1C2 C(C)(C)(CCC(=O)NCCC1CC(NC(C2CCO2)=O)C1)OC C1(NC(C23OCC(C(C)C)(C2)C3)=O)CCCN(C(=O)C(C2CCOCC2)O)CC1 C12CCN(CC1)C2.C1=CC(Sc2csc(Cc3ccccc3)n2)COC1 CN1CCC2(CCN(C(=O)NCC3CCCCN3c3ccncc3)C2)C1 c1(OCC(=O)NCCC(C)CCNC(C2OCCO2)=O)nc(O)nc(O)n1 N1(C(C(CC)C)=O)CCCC(NC(c2cnc(C)c(Cl)c2)=O)C1C CC1(C)CC(CNC(c2cnoc2C2CCOCC2)=O)CN(C(=O)C(N)=O)C1 C1(NC(c2cn(C)nc2C(C)(C)C)=O)CN(C(C2(N=[N+]=[N-])CC2)=O)CC1C1CC1 Cc1ccc2c(CC(=O)N(C)CC3(NC(C4CN(C)CC4C)=O)CC3)coc2c1 c1(C(=O)NCC(CNC(Cc2c(C)cc(C)s2)=O)F)cnn2ccc(O)nc12 CCC(C)(C(=O)NCC1(O)CCN(C(=O)Cc2ccc(F)cn2)C1)C(N)=O C1(C(=O)NC(c2ccc(OC)cc2)CC)CC2COCC(C1)C2N c1(C(N2C(C(C)NC(c3c(CCC)n[nH]c3)=O)CCC2)=O)ccc(C)c(F)c1 c1(CN(C(CC=CC=C)=O)CCCNC(=O)Cn2ncnn2)ccccc1 C(=O)(C(F)(F)C(C)(C)O)N(C(CC)C(=O)NCC(O)COC)C c1(C(C(=O)NCC2CC2)N(CCC)CC2CC2)ccnn1CC c1(OC)nc(=NC2CN(C(c3cccnn3)=O)C2)[nH]c2[nH]cnc12 N1(C(CC2N(C(C(C(C)C)O)=O)CC2)=O)CCOC2(CCC2)C1 c1(C(OCOCC)=O)ccc(C2CC2)cc1.C(CCSC(C)C)NCC C(=O)(CC=C(Cl)Cl)N1CC(SC(c2cn(CC(=O)C(C)(C)C)nn2)CC=C)C1 Cn1cc(C=CC(=O)NC2C(C(N3CCC(O)(CO)C3)=O)C2(C)C)nn1 Cc1sc(Cl)c(C(N2CC(CNC(C3(C)CCC3C(=O)O)=O)C(O)C2)=O)c1C N1(C(C(CC(C)C)CNC(=O)CCCCN(C)C)=O)CCc2ccc(F)cc21 C1(C(NOC(c2ccccc2)C)=O)(NC(C2CC(C)(C(N)=O)C2)=O)CCN(C)C1 c1(OC)ccc2c(c1)OCC2NC(=O)C(=O)NCc1cc(P(C)(C)=O)ccn1 C1(CNC(C2(C(=O)NC)CC2)=O)CC(C)CCN1C(C1CC2CCC1CC2)=O C(C)(CO)(C(=O)N1CC(C(O)C(N2CCOC(CN=[N+]=[N-])C2)=O)C1)OC c1(NC(c2[nH]nc(NC(C3(OC)CC3)=O)n2)=O)c(-c2ccccc2)sc(C)c1C C1(C2CCN(C(c3ccn4cnnc4c3)=O)CC2)(NC(C(=O)NC2CC2)=O)CC1 N1(C(c2cccc(C(C)C)c2)=O)CC2CCC(C(N3CCC(C)CC3)=O)(C2)C1 N1(C(c2c(C(C)C)nns2)=O)CCOC(C(C)NC(C2(CF)CC2)=O)C1 C1(CNC(COC)=O)CN(C(=O)CN2CCCC(CO)C2)C2CC12 CC1=CCCN(C(C2CC(C)N2C(c2nccn2C)=O)=O)C1 CC(C)CC(CNC(=O)C(C)C(C)C)C(=O)NC(C(C)(C)CO)C1CC1 c1(C(N2CCCC(C)(NC(=O)CSc3ccncc3)C2)=O)ccc(F)c(N)c1F C(=O)(CC(CC)CCCC)NC(CC=CC)C(=O)N(C)Cc1ccnn1C c1(C(=O)NCC(CNC(c2c(CC)ncnc2)=O)O)cnc2cccnn12 N1(C(C2CCC(NC(=O)CN3CC4CCC3C4)C2)=O)CCCC12CCOC2=O C1(C(N(CCN(C(COCC(=C)C)=O)CC2CC2)C(C)C)=O)CCc2nn[nH]c2C1 C(=O)(C1=CC2C=CC1C2)NC1C(NC(CC(CC)C)=O)C1 N1(C(c2cc(C#N)[nH]c2)=O)C2CC=C(C(=O)NCCN3CCCOC3=O)C1CC2 CCC(C(=O)N(C(C)CC(C)C)C(=O)CCSCC(C)C)OC1CCCC1 N1(C(C(C)(C)CC#N)=O)CC2(CCC(CNC(=O)C(O)Cc3ccccc3)O2)C1 CCC(C)C(C(=O)N1CCC1C(=O)NCc1ccc(C)nc1O)NC(C)=O CCN=C(NCCC1CC1C1CC1)N1CCN2C(CCS2(=O)=O)C1 C1(CC(=O)NC(C2CN(C(c3cccs3)=O)CCO2)C)CC2CCC1CC2 Cc1ccc(C(N2CC(C)(C)CC2CNC(=O)C(C)n2ccnn2)=O)c(F)c1 c1(SCCN(CCC#N)CC)ccc(Cl)s1.C1(C)CCCO1 N1(C(=O)CCCN2CCCCC2)CCCN(C(C2CC(=C3CCC3)C2)=O)CCC1 c1(OC)ccc(C(N2CCCC2CNC(=O)C(C)CC(C)(F)F)=O)c2sccc12 c1(CCC(=O)NC(C(=O)OC)CCCC2CC2C)ccc(O)c(OC)c1 C1(NC(C2C(OCC)CCC2)=O)CC(NC(c2ncsc2C)=O)C(O)C1 C#Cc1ccc(NC(C2(C#C)CN(C(c3cc(C)sc3C)=O)C2)=O)cn1 C(CC(C)C)(C(=O)N(CCC(=O)NC(C)C(C)SC)C)OC N1(C(c2cc(C)on2)=O)CC2CC2(C(=O)NCC2CC(c3cccc(Cl)c3)C2)C1 C1(NC(c2ccc(-c3cscn3)cc2)=O)COCC1C1CC1 N1(C(Cn2c(C)nc(C)n2)=O)CCC(C)(C)C1CNC(C1CC(=O)N(C)C1)=O C1(CNC(C(C(C)C)OC)=O)CN(C(=O)CCC2(C)CC2)CCC12CCOCC2 CCC(C(C)(C)O)NC(=O)CCC1CCN(C(C2CCC(NC)CC2)=O)C1 CC1(C)Cc2cc(C(=O)NC3CCN(C(C4CC(O)C4)=O)CCC3CO)sc2C1 C1(NC(CC(=O)OCC)=O)CCCC(NC(c2sccc2OC)=O)CC1 CC(C)CC(C(=O)NCCn1ccnn1)ONC(=O)Cc1ccccc1Br C(=O)(C1=CCCCC1C)NCC(C1CC1)NC(=O)C1=COCC1 c1(OC)ccc(C#N)c(NC(c2cc(-c3cnn(CCN(C)C)c3)[nH]n2)=O)c1 Cc1ccc(CC(=O)NC(C)CCN(C)C(C2(C)COC2)=O)cc1Cl N1(C(C(CCSC)O)=O)CC2CCC(CNC(c3cnc(C)[nH]3)=O)C2C1 C1(CCC)C(=O)NCCN1C(=O)Cc1cncn1C(C)C O=NN1CCCC1C(=O)NCCC1CC(NC(C23CC(C#N)(C2)C3)=O)C1 Cc1noc(C)c1C(C)CC(=O)NC1CCN(C(=O)CCc2nc[nH]n2)C1 C1(C(=O)NCC2(NC(c3cn(Cc4onc(C)n4)nc3)=O)CC2)CC(=O)N(O)C1 N1(Cc2c(C(=O)OCC)ccs2)CCSC(C(=O)Nc2ccnc(F)c2)C1 N1(C(c2ncn(CC)c2)=O)C2CCC1(CNC(=O)CC1CCCC(F)(F)C1)CC2 N1(C(c2c(C)ocn2)=O)CC(O)CC1C(=O)Nc1ccccc1CC#N c1(N2CC(C(=O)Nc3c(OC)nccc3C)SCC2)ncnn2ccc(Br)c12 C=CCCCCC(=O)NCC(C)CNC(=O)C(c1ccccc1)OC c1(C(=O)NC2CC(N(C(Cc3c(C)cccc3)=O)C)C2)c(Cl)ccc(F)c1N C(=O)(C1=CCCSC1)N1CCC(N(C(=O)CCCNS(C)(=O)=O)C)C1 C(=O)(C1=CCCOCC1)N(CCCNC(C1CCCS1(=O)=O)=O)CCC CCC(CC)CC(=O)N1CC2CC(NC(C3CCN(C(=O)NCC)C3)=O)C2C1 CC1=CCN(CC(=O)NCc2cccc(OCc3noc(C(F)(F)F)n3)c2)CC1 N1(C(CCCSC)=O)CC2CCC1C2NC(=O)CCC1(C)CCC(=O)NC1 Cc1ccc(Br)c(CC(=O)NCCOCCCNC(c2cc(C)on2)=O)c1 c1(OC)cc(F)c(C(=O)NC(C2CCN(C(=O)C(=O)NC3CC3)CC2)C)c(Cl)c1 C(=O)(CC(C)C(C)C)N1C(CCNC(c2nc(C)n(C)c2)=O)CCCC1 C1(CNC(C(C)NC(CC)=O)=O)CN(C(c2ccc(N)cc2Cl)=O)CC1(F)F c1(C(N2CC(OCC)(CNC(=O)C(C)C)C2)=O)cnc2ccc(C)cn2c1=O CC1CC(CCNC(C2CC(CN(C)C)C2)=O)CCN1C(c1occc1Cl)=O N1(C(c2cncc(N)n2)=O)CCCCC(CNC(c2cc(Cl)sc2Cl)=O)C1 C=CCC(CNC(=O)Cc1ccc(Br)cc1)C(=O)NCCSCCOC C1(CNC(C2(CC#C)CCOC2)=O)CN(C(=O)C(c2cnn(C)c2)=O)CCO1 c1(C(N(CCNC(C2(C(=O)O)CC2)=O)CCc2ccccc2)=O)ns[nH]c1=O Cc1cc(I)ccc1C(=O)Nc1cccc(NC(c2c(Cl)ccnc2Cl)=O)c1 c1(OC)ncccc1C(=O)NCC1CC(NC(C2CCSC(C)C2)=O)C1 C1(CC(=O)OC)CC(NCC2COCCN2)CC(C(F)(F)F)O1.C=CC Cc1ccc(CC(=O)NC2CC23CCN(C(C2CCC(C)C2)=O)C3)cc1F N1(C(CC(C)OC)=O)CCCN(C(=O)Cc2ccccc2F)C(C)C1 C1(CC(C(CCCCCCO)=O)O)CCC2(CCCC2)O1.c1(C2(CN)CC2)ccccc1 C(C(=O)NCC1(CC)CC(C)(C)C1)(C(C)C)NC(COCCC=C)=O C1(CNC(c2nc(COCC)sc2)=O)CC2(C1)CN(C(=O)Cc1csnn1)C2 N1(C(Cc2cccc(OC)c2)=O)CCCCCC1CNC(c1cc(C)c(Cl)s1)=O Cc1cnc(N(Cc2cccnc2)CC2CC3(CCN3)C2)nc1 C1(CNC(c2sc3cc(C)sc3c2)=O)CC2(CCN(C(=O)Cc3ccoc3)CC2)C1 Cc1ccc(C(C)NC(c2cn(CCNC(C3CCCC4CC34)=O)nn2)=O)cc1 CC(F)CC(=O)NC1CCCC1CNC(=O)C(F)(F)C1(O)CNC1 C1(F)(CNC(C2C(CN(C)C)C2)=O)CN(C(=O)C(C)(C)c2ccncc2)C1.C1CC1 Cc1cccc2sc(C(=O)NC3CCC4CC3CN4C(=O)CCCC#N)c(Cl)c12 c1(OC)cccc(C(CNC(C2C(C)CCCS2)=O)NC(c2n[nH]c(C)n2)=O)c1 C1(CC)COCCN1C(c1nc(CNC(=O)CNC(C2CC2C)=O)oc1C)=O Cn1ccc(=NC(=O)c2ccnc(CNCc3cccc(O)c3)c2)[nH]1 n1(CC)cc2ccc(C(=O)NC3CCC(NC(=O)Cn4nccc4C)C3)cc2n1 N1(C(c2nncc(OC)c2)=O)CC2CCC1C(CNC(C1C3CC4C(C3)C14)=O)C2 C=CCC(C(=O)N1CC2(CC(CC(=O)NCC3CCOC3=O)C2)C1)C(C)C N(C)(CP(C)(C)=O)C(C1(NC(c2cnc(C)o2)=O)CCSC1)=O C#CCCC(O)CCNC(C1(CC)CCN(C(=O)CCc2cccn2C)C1)=O Cc1[nH]nc2c1CC(C(=O)NC1CCCC1NC(c1cnc(C(F)F)s1)=O)CC2 c1(C(=O)NC(CCCNC(C(CCSC)OC)=O)C)nc(C)c(C)nc1O CC1CN(C(=O)Cc2ncc(Cl)s2)CCCN1C(c1cnc2[nH]cncc1-2)=O N1(C(C(C)(C)OCC)=O)CC2CCC1C(NC(c1c(Cl)ccc3c1OCO3)=O)C2 C1(CNC(=O)CC2(CO)CC2)CCN(C(c2cc([N+](=O)[O-])c[nH]2)=O)CCC1(F)F CN1CC(C(N2CCCC2(C)CNC(=O)C(CO)c2ccccc2)=O)CCC1=O c1(CC)cc(C(=O)NC2CCC(NC(=O)CC3CC3CC)C2)ccc1F c1(C(=O)NCC(CC=C)NC(=O)C(CO)N(C)C)cnc(C(N)=O)cn1 C12(C(N(C3C(NC(c4nc(C)oc4C)=O)CCCC3)C)=O)CCOC(C)(C1)C2 O(N1CCC(N=c2cc(C)[nH]c(-c3cccs3)n2)CC1)CC N1(Cc2n(CC)nnn2)CCC(O)C(C(=O)NC(C)Cc2ccccc2F)C1 c1(OC)cccc(NCC(=O)N(C)CCNC(=O)C=C2CCC(C)C2)c1 C1(C(=O)NCCCCC(=O)N2CCC(CCCC)C2)CC12CCOCC2 Cc1nc(C=CC(=O)N(CC(O)CNC(c2c(N)cccc2F)=O)C)[nH]c1C C(CC(C)(C)CC(=O)NC1C=CC(C(N2CC3CCC3C2)=O)C1)OC C(C(CC1CCCC1)CO)NC(CN(C(=O)C=CC(C)(C)SC)CC)=O Cc1ccc2oc(N3CC(C)(C)CCC3CNC(=O)C(C)N(C)C)nc2c1 CC1=C(C(=O)NC2CC3(C2)CC3NC(c2c(Cl)c(C)nn2C)=O)CCCC1 N12CC3CC(O)C1C3NC(=O)C=CC2=O.N1(CC(=O)NC2CC2)CCCCC1 CCCC(C#N)C(=O)N1CCN(C(CNC(c2cc(C)c(C)o2)=O)C(F)F)CC1 c1(C(C)C)nc(=NC(C)C2CN(C(=O)COCC3CCOC3)CCO2)s[nH]1 c1(C(=O)NC(CN(C(=O)C(C)CC2CC2)CC)C)ccc(OC)cc1Br N1(C(c2c(C)ocn2)=O)CC2CC2(NC(=O)C(C2CCCC2)C2CCCC2)C1 Cc1cc(CC(=O)OC(C)C)ccc1NC(=O)N(c1ccc(C#N)nc1)C1CC1 N1(C(c2nc(COC)oc2)=O)CCCC(CCNC(C2CC3(CC3)C2)=O)CC1 N1(C(c2c(SC)cn(C)n2)=O)CCC(C)C(NC(C2CCC3(CC3)C2)=O)C1 S(=O)(=O)(c1cccnc1N1CCC(C#N)C1)NCC1OCCN(C(C)(C)C)C1 c12ccncc1-c1nccn1C2.c1(-c2scc(C)c2)cnn(C)c1C Cc1nc2cc(Br)cc(NC(c3ccc(CCc4cccs4)cc3)=O)c2o1 N1(C(CC2CC(C)C2)=O)CC2CCC2(CNC(=O)CCCNC(=O)C2CC2)C1 c1(C(=O)NCC2(C(N3C(CC)CN(C)CC3)=O)CC2)cc2ccccn2n1 C(=O)(C(N)CC1CCCCC1)N1CC(NC(CC2(OC)CC2)=O)C1 N1(C(c2ccn(C)n2)=O)C2CCC1CN(C(C1CC(O)C(F)C1)=O)C2 CC1OC2(C(=O)NCCC3CCN(C(C4CC(C)(C)CO4)=O)C3)CC1C2 c1(C(=O)NC(c2ccccc2F)CNC(c2ccc(C)[nH]2)=O)cncc(N)c1 CC(C)(CC(=O)NC1C=CCC(C(=O)NCc2cccnc2)C1)C1CC1 C(=O)(C(F)(F)C(F)(F)C(F)(F)F)NCC1OCC2CCN(C(=O)OC(C)(C)C)CC21 c1(OC)cc(NC(C2C3CC2N(Cc2scnc2C)C3)=O)cc(F)c1 C(=O)(CCCCC(C)C)NCCC(=C)CNC(c1c(Cl)sc(C)c1C)=O C(C(C)(C)NC(=O)C(F)N1CCCC1)=CC(=O)NCCNC(=O)NC N1(C(C2(CCF)CC2)=O)CCCC1C(C)(C)C(=O)NC(C)CCn1cncn1 CC(C)(C)C(C)(C)C(=O)N1CCOC(CCCNC(=O)CO)C1 Cc1cc(C)c(S(=O)(=O)NCc2ccc(F)c(S(N)(=O)=O)c2)cc1[N+](=O)[O-] c1(C(N2C(CCC)CN(C(=O)C(C)C(F)(F)F)CC2)=O)cc2c[nH]cnc-2n1 N1(C(C2(C(C)C)N(C(c3cc(OC)ns3)=O)CCC2)=O)CCSC2(CCC2)C1 C12(C(=O)NC(CCN(C(c3ccc(C)cc3C)=O)C)C)C3C4C1C1C2C3C41C CC(C)CC(C)C(=O)NCC1(O)CC(C(=O)NCC(O)C2CC2)C1 C1(CC(=O)NC(CN(C(C)=O)C)C)CN(C(=O)CN2CCCNC2=O)CCC1C Cc1cnc(C(N2CCC(CC3CN(C(=O)OC(C)(C)C)C3)CC2)=O)c(F)c1 c1(OCc2[nH]nc(C(N3C(CC(=O)NC)CCC3)=O)n2)ccc(C#N)cc1 N1(C(CNC(C(CC)C)=O)=O)CCN(C(c2coc(C3CC3)n2)=O)CC1C C1(CN(C(C2CCCCO2)=O)CC)CN(C(=O)CCc2cccnc2)C(C)(C)C1 c1(C(N(CC(=O)N(CCOC)CC2CC2)C2CC2)=O)cccc(F)n1 C(CNC(=O)CN1CC2C=CC1C2)(CC(F)(F)F)NC(c1c(C(C)C)cco1)=O N1(C(CCC=C=C)=O)CC(CO)C2(C1)CN(C(C1CC1COC)=O)C2 N1(C(C(C)=C2CCC2)=O)CC2CC(NC(=O)C(C)(C)c3cncnc3)C2C1 CCCS(=O)(=O)CC(=O)NCC12CN(C(=O)C(C)(C)n3cccn3)CC1CCO2 N1(C(c2c(C(C)C)c[nH]n2)=O)CCOC(CNC(C2CC3C=CC2O3)=O)C1 C12(CNC(C3(C#C)CC3)=O)CCC1CCN2C(=O)Cc1ccc(C#N)cc1 c1(CC)cc(N2CCC(CCNC(c3oc(C(C)C)nc3C)=O)C2)ncn1 CC1CCSCCN1C(C1(NC(=O)CC2CCCC2O)CCC(C)(C)C1)=O c1(CC)oc(C)cc1C(N1CCCC(n2cc(CO)nn2)C1)=O.N12CC(C1)C2=O C1(CC(=O)N(CCC)C(C)C)(CNC(C2CC(OC(C)=O)C2)=O)CCC1 N1(C(C(C)OC(=O)OCC)=O)CCCC(C(=O)NCCCc2ccccn2)CC1 c1(N2CCOCC(NC(Cn3c(C(C)C)ncc3)=O)C2)c(Br)cccc1[N+](=O)[O-] C#Cc1cccc(C(=O)N(CCC(=O)N(C(CSC)CC)C)C)c1 C1(CC)(CC)CC(C(N2CCC(C(F)C(=O)N3CC(CF)C3)C2)=O)C1 n1(CC(=O)NCCN(C(=O)C(O)C(C)CC)CCCCCC)c(C)c(C)sc1=O C1(=O)CC(=O)NC2CC2CNC(=O)C12CC2.C(CC)NC(=O)OC.CCN n1(C(C)C)cc(C(=O)NCC2CCN(C(c3coc(C(C)C)n3)=O)C2)ccc1=O CC1CCN(C(C2CC2c2ccccn2)=O)CCN1C(c1cnn(C2CC2)c1)=O C1(c2nnnn2C2COC2)(NCc2c(C)cco2)CC(C)(C)C1 N1(C(c2ccc(CC)cc2)=O)CCOCC(CNC(=O)CC(C)n2cccn2)C1 O=C1CCC(CC(N2CCCC(CCNC(=O)CCc3ncco3)C2)=O)CN1 c1(CC)ccc(C)c(NC(=O)C(F)CC2CN(C(=O)C=C(C)COC)C2)c1 N1(C(C2C(c3cn(C)nc3)C2)=O)CCCCC12CC(NC(=O)CC(F)(F)F)C2 CN1CCC(CC(=O)NC23COC(CNC(=O)CCF)(C2)C3)C1=O N1(C(C(CC)(C)O)=O)CCCC2(CCN(C(=O)CC3CCCC34CC4)CC2)C1 c1(CNC(C(=O)NCC2(CO)CN(CCCOCC(F)F)C2)=O)cccc(Cl)c1 c1(NCC(C)CO)nc(N2CCCNC(=O)CC2)nc2ncn(C)c12 C(CN=C(NCc1cn(C)nc1C)NCC(F)F)OCC=C N1(C(C)=O)CCCCC1C(N1CCC(C(=O)NCCC2CC2C)CC1)=O c1(OC)ccc(N)c(C(=O)N(CC(O)CN(N2CCCC(C=O)C2)C)C)c1.N(C)C C1(C(=O)NC2C(NC(CN3CC(C)C3)=O)COC2)CC(C2CCOCC2)=NO1 C(=O)(NNc1cnnc2ccccc12)N(C(C)Cn1ccnc1)C1CC1 N1(C(C=C2CCC(C)C2)=O)CCCN(C(c2ccc(F)cn2)=O)CC1C C(=O)(CS(=O)(=O)CCOC)N(C1C(NC(C(CC)(C)CC)=O)CCCC1)C c1(CNC(C(CC)N(C)S(=O)(N)=O)=O)ccc(CNC(=O)CCC2(C)CC2)cc1 C1(C(N2C(C)CN(C(=O)Cc3ccno3)C(C)C2)=O)CC(c2ccncc2)=NO1 c1(SCC)ccccc1C(=O)N(C)CCNC1CC1 C1(C(N(C2CC(C#N)C2)CC(=O)N(C)Cc2nccs2)=O)CC12CCOCC2 C1(C(=O)NCC(C2CCOC2)NC(C(CNC(C)=O)(C)C)=O)C(F)(F)C12CCC2 N1(C(Cc2ccc(OC)cn2)=O)CCC(C)(C)C(CNC(=O)C(C)CF)C1 O(NC(=O)CN=c1ccnc(NCCNCCN2CCOCC2)[nH]1)CC n1(CC)ncc(Cl)c1C(=O)NC1CC(F)(CNC(=O)C(c2ccc(Cl)s2)=O)C1 c1(CC(=O)NC2CN(Cc3cccs3)CC(F)(F)C2)ccc([N+](=O)[O-])cc1Br CC1CC=CCC1C(=O)NCC(O)CN(C)C(c1ccc(OCC(F)(F)F)o1)=O c1(C(N2CCN(C(CCN(C)CC)=O)CC2C)=O)ccc2c(c1)nnn2CC c1(C(N2CC(CNC(C(C)CC3CC3)=O)OCC2)=O)ccc2[nH]c(=N)oc2c1 c1(OC)cncnc1C(=O)NC(C(N1CCC(C)(NC(C)=O)C1)=O)C1CCC1 c1(C(C(=O)NCC2C(CNC(c3c(C)[nH]nc3Cl)=O)C2)C)cccc(C#N)c1 c1(C(=O)NCC(C)CNC(=O)C(C)(C)c2ccno2)ccc2nccn2c1 C1(C(=O)NCC2CCCN(C(C=CC3N(C)CCC3)=O)C2)CC2CCC1C21CC1 c1(C(N(C2CCCC2)CCNC(C2CCC(=O)N2)=O)=O)ccccc1F c1(-c2cc(OCC)ncc2)cccc2[nH]nc(C(=O)Nc3nccnc3CC)c12 c1(CC(=O)NC2CN(C(c3cc(Br)no3)=O)C2)ncc(F)cc1F N1(C(CSCCCC)=O)CCC(C(=O)NC(C)C)C12CC2 Cn1cnc2ccc(C(N3CCCCC(CNC(=O)C(O)CC(N)=O)C3)=O)nc12 CCCC(C)C(=O)OCC(=O)N(N1CCCC(Sc2ccc(C(N)=O)cc2)C1)C C(=O)(CN=S(C)(C)=O)N(c1ccccc1)CCN(C(=O)CCN1CCCC1)C(C)C C12(NC(=O)CCN3CCCC3)CCC(CC1n1cc(CCCCCO)nn1)C2 C1(CC)CN(C(C2CCCCC2O)=O)CC1C(=O)NCCN(C(C)C)C1CC1 c1(C(=O)NCC2(NC(c3ccncc3Br)=O)CCC2)cc2cccnc2cn1 N1(C(C2C(C(C)C)CN(C(C3CCN(C)C3)=O)C2)=O)CC2CC(C)C2C1 c1(CNC2CC(C(=O)NCc3cccc(OC)n3)C2)c2c(nn1C)CCC2 Cc1cnc(C(=O)NCCNC(c2onc(C)c2C)=O)cc1C CC(C)CCCCCC(=O)NCC1CCN(C(=O)C(C)Cn2cccn2)C12CC2 N1(C(Cc2cccc(C#C)c2)=O)CCC(F)(F)C(CNC(c2sccc2C)=O)C1 N1(C(c2c(CC)nccn2)=O)CCC2C(CCCN2C(=O)C(C)CSC)C1 C1(N(C(CCCSC)=O)C)CC2CCC(C1)N2C(c1n[nH]cc1C1CCC1)=O c1(C(=O)NC2C(CNC(C(C)CF)=O)CC2)ccc(C(C)(C)C)nc1 CC(C)CC(=O)C(=O)N1CC2C(CNC(=O)Cc3ccsn3)C2C1 CCC(C)C(O)C(C)C(=O)NC(COC)CC(=O)NC(c1nc(C)cs1)C C(=O)(C(F)(F)C(F)(F)F)N(CC(C)(C)NC(C(C1CCC(C)(O)CC1)C)=O)C c1(C(=O)NC2CC(C)N(C(=O)CCSC(F)(F)F)C2)cc2cc(Cl)ccc2[nH]1 C(=O)(CCCCCCn1cc(C(C)(C)NS(C)(=O)=O)nn1)NC(CC)C(F)(F)F CC(CC(=O)N1CCCC(C)(CNC(=O)CC2CC3CCC2O3)C1)P(C)(C)=O Cc1cc(F)ccc1CC(=O)NC1CCCN(C(=O)COCC2CCC2)CC1 C#Cc1ccc(C(N2CC(C)C2C(=O)N(C2CCC2)C)=O)nc1 C#Cc1ccc(F)c(C(=O)NCCOCCNC(c2cc3c(nn2)CCC3)=O)c1 c1(CN2C(C)(C(=O)Nc3cc(C)no3)CC2)ccc(Br)nc1Br CC(C)(C)CCC(F)C(=O)NC(CC(=O)NC1CCC(O)C1)C(F)F c1(CC(=O)NC2CC(C)N(C(=O)CP(C)(C)=O)CC2)cn(C)c2ccccc12 c1(C2C(C(N(CCN(C(=O)C(F)OC)CC)CC)=O)CC2)ccc(F)cc1 N1(C(C(N2CCSCC2)C)=O)CCC(CO)(CNC(=O)CN2CCOCC2=O)C1 Cc1cc(C)n(CC(N2CCCC(C(c3ccccc3)C)C2)=O)n1 C12(NC(CNC(=O)CN(C(C)C)C)=O)COC(C1)C(NC(C1CCOC1)=O)C2 Cc1cc(=NCCCC(C)(C)NC(=O)C=Cc2ccco2)[nH]c(C(C)C)n1 CCC(CC)C(=O)NCC(C)NC(=O)CN(C(=O)C(CC)OC)C CC(C)C(CNC(C1CC2COCC2C1)=O)C(=O)N1CC(C)C(O)C1C(=O)O c1(C(N2CC3C(NC(CN(CCC)C)=O)(C3)C2)=O)cc(Cl)cc2c1CCC2 n1(C(CC)C)nc(-c2ccc(N)cc2)nc1COCC(C)(C)C CC(N=c1nc(N2CC(=O)NC(C)(C)C2)c2ncccc2[nH]1)c1ccoc1 C1(C(N2CC(CNC(C(CO)OC)=O)C(C)CC2)=O)CCC2(CCCC2)CC1 C1(NC2(CC(=O)OC)CCCOC2)CC2(CCCCCC2)C1 c1(CC=CC)ccc2c(n1)CN(c1cccnc1)C2.C1(C(=O)OC)CCC(C)CC1 CCC(C(=O)NCC1CC1CC(=O)NCc1c(C)cccc1C)C(C)(C)CC C(=O)(C(C)(C)N=[N+]=[N-])NCc1c(C(=O)NCCc2nc(C)[nH]n2)occ1 C1(C(=O)NC2(CCOCC)CC2)CCC(n2cc(Cn3ccnc3)nn2)C1 C(=O)(CC1=CCCC1)N1C(C2CCCN(C(CSc3n(C)cnn3)=O)C2)CCC1 N1(C(C2C3(CC(OCC)C3)C2)=O)CC(NC(C2CC3CC3C2)=O)CC2(CC2)C1 C1(CNC(C(C)CC(F)(F)F)=O)CCCC2(CN(C(=O)CC3CCSCC3)C2)O1 CCCCC(O)C(C)C(=O)NCC=CC(=O)NC(c1cnc(C)s1)C Cc1ccc(F)c(CNC2CCN(CC(=O)NCC3CC(=O)NC(=O)C3)C2)c1 c1(C(N(C)CC2(O)CN(C(C(C)SC)=O)C2)=O)ccc(NC)cc1 CC(=O)CCCC(=O)NC(C)(CO)C(=O)Nc1cccc(C)c1 CCCC(F)C(=O)N1CCC2CC12C(=O)NCc1cc(C#N)c[nH]1 c1(CCC(=O)N(C(C(=O)NC2(CC(=O)OC)CC2)C2CC2)C)cncnc1 CC(C)C(O)C(F)(F)C(=O)N(C)CC1CCCC1NC(=O)C(C)Cc1cnc[nH]1 C1(CN(C(COC(CC)CC)=O)C)CCCN(C(=O)CCCC2(NC)CCC2)C1 c1(C2(C)C(NC(C3CC(O)(c4cccnc4)C3)C)C2)cccc(Cl)c1 C(=O)(CCP(C)(C)=O)NCC1(O)CCN(C(Cn2cc(CN(C)C)nn2)=O)C1 C(CCCCCCCO)=CC(N1CC(CNC(C=CC)=O)OC(C(F)(F)F)C1)=O C(N=c1ccnc(C)[nH]1)C1(OCc2cc(OC)c(N3CCCCC3)cc2)CC1 c1(SC)nc(C)c(S(=O)(=O)N2CCCCC2C(=O)NC(CO)CO)s1 Cc1ccc(CCCNC(=O)CCC2CCCN2Cc2ccccn2)o1 C(N=c1ccn2nccc2[nH]1)C1CCCN(Cc2c(OC)cccc2F)C1 c1(C(=O)Nc2ccc(CC#N)cc2)ccc([N+](=O)[O-])c(CO)c1 c1(C(N2CC(C)(C)C(C(=O)NCC3CC34CC4)C2)=O)c[nH]c2cnccc12 N1(C(C(CC)Oc2ccccc2)=O)CCCCC(NC(=O)CC2(C)CCCO2)C1 C1(NC(C(CCCC)O)=O)COC2(CCN(C(c3cncs3)=O)CC2)C1 Cc1ccc(C(C)NC(=O)C(CNC(=O)C(O)C2CCCC2)N(C)C)nc1 Cc1nc(C(N2CCN(C(C3(Cl)CC3(F)F)=O)CC(C)(F)C2)=O)c2ccnc-2[nH]1 c1(CC)cccc(NC(=O)Cc2ccnn2CS)c1.c1(C2CNC2)ccccc1 C(=O)(C1Cc2ccccc21)N1CC(O)(C(CNC(c2occ(C)c2C)=O)(C)C)C1 C(=O)(C(C)(C)CC(F)F)NCC1N(C(C=C(C)C(C)(C)C)=O)CCCC1 C1(CNC(C2CCOC2)=O)CCN(C(C2CC(C(F)F)C2)=O)C12CCC2 c1(C(=O)NCC(CNC(CSCCC)=O)F)cnn(CCF)c1 C1(CNC(c2cc(Cl)c[nH]2)=O)CCCCN1C(c1ccccc1-n1nccn1)=O c1(C(N(CCCOCCN(C(CC2N(CC)CCC2)=O)C)C)=O)ccc(C)n1C c1(OC)cc(C)c(CCC(=O)OC(CC(F)(F)F)c2ccc(F)cc2)c(C)c1 N(C1CCCc2cc(N)ccc21)C(C1(C)CCC(C)(C)CC1)=O C1(CN(C(C2CC(N(C)C)C2)=O)CC)CCN(C(=O)CN2CCOC2=O)CC1 c1(OC)cc(OC)c(NC(N2CC(O)CC2c2ccccc2)=O)cn1.C1(C)CC1 Cc1cc(C2(C(=O)N(C3CCSC3)CC3CCCO3)CC2)cc(C)c1Cl N1(NC(C)=O)CCOCC1CC(=O)NC1CCCC(NC(=O)CS)C1.C(CC1CC1)N N1(c2ncc(C)cn2)CCOCC(NC(=O)C(C2CCCCCC2)N(C)C)C1 c1(C(CNC(=O)C=CC(N2CCOCC2)=O)NC(C2C(C)C2)=O)ccccc1F N1(C(c2c(OCC)scc2)=O)CCCC(C)(NC(C2COC(=O)N2C)=O)C1 c1(C(=O)NCCCN(CC2CC2(F)F)CC2CCCC2)ccccc1C#CC1CC1 C1(CNC(c2cc(CCC)[nH]n2)=O)CCCC(NC(C2(Br)CC2)=O)C1 C1(NC(c2cc(OC)n(C)n2)=O)CS(=O)(=O)CC1NC(=O)C=Cc1ncc(C)[nH]1 c1(OC)ccc(C)c(OC)c1CC(=O)NCC1C2CCC(C2)N1C(=O)CCSC CCC(CC(=O)NCC1CC(C(=O)NC(C)Cn2ccnn2)C1)OC C12(CC(=O)NCCNS(CC)(=O)=O)CCC1CN(C(=O)C(C(C)C)N(C)C)C2 S(=O)(=O)(CC(=O)N1CCC(O)(CN(C(=O)COCc2cccc(C)c2)C)C1)NC Cc1nc(N2CC(O)(C(C)NC(c3ccco3)=O)C2)cc(-c2ccco2)n1 Cc1cn2cc(C(N3CCC(=CCNC(c4cc5n(n4)CCC5)=O)CC3)=O)nc2s1 C1(C)(CC)CC(NC(=O)C2=CCCC2)CN1C(=O)CN1CCSCC1 C1(CNC(C2C(=C)C2)=O)CC2CCC(C1)N2C(=O)C=Cc1ccccc1 CCCCCCCCNC(=O)C(=O)NC(c1ccc(OC)c(OC)c1)C C(=O)(C(F)C(C)C(F)(F)F)NCC(CNC(c1cc(C)c(C)s1)=O)O CCCCCC(O)C(C)C(=O)N1CC(O)(CNC(c2cc3ccccc3o2)=O)C1 c1(C(N(C2CCN(C(=O)Nc3cnnn3C)CC2)C)=O)ccc2scnc2c1 C(=O)(C(O)C(F)(F)F)N1CCC(CNC(c2ccc(CC(C)C)s2)=O)C1 C1(C(N(C2CCCN(C(C34CC(CO)(C3)C4)=O)C2)CC)=O)CCCC(CF)C1 c1(SCC(N2C(c3cn(CCOC)nn3)CC2)=O)nc2ccccc2o1 c1(C(=O)NC(CNCC2(CC(=O)OCC)CC2)CO)cc2ccccc2oc1=O C=CC1(C(=O)NC(C2CCCCC2)(C)C)CCN(C(=O)C=C2CCCCC2)CC1 CC1(C)CN(C(=O)C=CC2CCOCC2)CC(CNC(=O)C(C)(C)CF)O1 c1(OC)cc(CC(=O)NC(C)CCCNC(C2(SCC)CCC2)=O)cc(Cl)c1 C(=O)(C(CC(C)C)C(C)C)N(CC1(CCNC(CSc2nc(C)[nH]n2)=O)CC1)CC C1(O)(CNC(C2C(C(N)=O)C2)=O)CCN(C(=O)CNS(=O)(=O)C2CC2)C1 N#Cc1cnccc1COC(=O)C=Cc1cccc(-c2ccc(Cl)cc2)c1 O=C1C2CCCCC2=NN1Cc1ccccc1CC(=O)OCC(F)F C(S(=O)(=O)CCNC(c1cc(C2CCOC2)[nH]n1)=O)c1cn(CCC(C)C)nn1 c1(OC)ccccc1C(F)(F)F.C12CCC(CC1)C(=O)NS(=O)(=O)C2 C1(C(=O)NCC(CO)N(C)C)CCC(CNC(C2(C)CC=CCC2)=O)CC1 C#CC1(C(N2CCC(CC(F)F)C2)=O)CCN(C(=O)CCc2cnoc2)C1 N1(c2nccc(OCC)n2)CCC2(CCN(C(c3ccc(Br)c(F)c3F)=O)C2)C1 C1(C)(NC(c2cccc(OC)c2)=O)CCC(NC(=O)Cc2ccccc2Cl)CC1 c1(-c2c(C3(C(=O)NC)CC3)cccc2)cc(OC(C)C)c(F)c(F)c1 c1(CC)cc(C(N2CC(OCCNC(C3CC(C#N)C3)=O)C2)=O)c(C)o1 c1(C(=O)NCC2N(C(C(c3ccc(C)o3)C)=O)CC=C2)cnn(C)c1S(N)(=O)=O c1(C(=O)NCc2c(F)ccc(CC)c2)cccc(C#CC2CC2)c1 c1(C(=O)NCC(C)CN(C(=O)CCC2(C#N)CCC2)C)sccc1Cl N1(C(CNC(=O)OC)=O)CCC(C2CCCN(C(c3cccn3C(C)C)=O)C2)C1 Cc1ccc(C#N)cc1C(N1CCCCC1CNC(=O)Cc1nccn1C)=O c1(OCC)cc(CCC(=O)NCCCCCNC(=O)Cc2ccc(C)s2)on1 N1(CCC=CCC)CCCC(NC(=O)CC(C)OC(C)=O)CC1 N1(C(C=CC(CC)C)=O)CCC(CNC(=O)CCn2nc(C)cc2C)(OC)CC1 CC1(C)CCOC(C(N2CCCC2C(=O)NCC2(C)CC2)=O)C1 C1(NC(COCCCCC)=O)CC2CC(NC(=O)CC(C)CC(C)C)CC2C1 N1(C(CC2CC(C)(C)OCC2)=O)CCC2(CC1)CN(C(c1ncc(F)cn1)=O)C2 C1(C2(O)CCOCC2)(C(=O)NCC2CN(C(c3cnoc3)=O)CCO2)CC1 c1(C(=O)NC(CCNC(C(C)OCC)=O)C(C)(C)C)ccnc2ccncc12 C(=O)(CCCC(=O)NCC1(NC(c2coc3c2COC3)=O)CC1)OCC S(=O)(=O)(c1cccc(C(=O)N(C2CCSCC2)C)c1)OCC=C.C1(C)CO1 N1(C(CCOCC)=O)CCCC(C)(C)C1CNC(=O)C(c1c(C)noc1C)C c1(C(=O)NCC(CNC(=O)CC2COC(=O)C2)OC)ccc(F)c(F)c1 N1(C(C2N(CC(C)C)CCC2)=O)CCC(O)(CNC(=O)CCc2cnoc2)CC1 c1(C(N2CCC(CNC(c3ccc(F)cc3I)=O)CC2)=O)ccnc(F)c1Cl N1(C(C2(C(C)C)CCCO2)=O)CC2CC1CN2C(=O)CNS(C)(=O)=O C1(C(=O)N(CC(C)C(C)C)C)(CC)CCCN(C(c2ccc(C(C)C)o2)=O)C1 c1(C(N2CCC(CNC(CCCCC#N)=O)CC2)=O)cc2c(o1)CCCC2 c1(C(=O)NC23CC(CNC(C4CC4[N+](=O)[O-])=O)(C2)C3)nccc(Cl)c1F N1(CCC(=O)NC2(COC)CCOC2)CCN(C(=O)CN2CCC(O)CC2)CC1 N1(c2c(C)c(NCc3ncsn3)ncn2)CCC2(CCCN2C)C1 N1(C(Cn2cc(-c3cnn(C)c3I)nn2)=O)CCC(COC(F)(F)F)C(F)(F)C1 CC1(C(=O)NCC2C3CN(C(=O)Cc4cnco4)CC23)CNC(=O)C1 Cc1ccc([N+](=O)[O-])c(C(=O)NC2CN(C(C3CC4(C3)CC4F)=O)CC2O)c1C N1(C(=O)Cc2ccc(Cl)cn2)CC2CCC(C1)N2C(C1CC1F)=O C1(NC(c2c(F)cccc2Br)=O)CCC2(CC1)CN(C(C1(CC)CCC1)=O)C2 C12(C(=O)Nc3scc(C#N)n3)CC(C1)C(NC(c1cc3occc3s1)=O)CO2 C12CCN(CC1)C2=O.C1(C(N2CCCC2)=O)CN(C(c2csc(O)n2)=O)CCO1 N1(C(C(CCC)OC)=O)CCC(C2CCCN(CCc3cscn3)C2)CC1 Cc1cccc2nc(C(=O)NC(C)(C)CCN(C(=O)C3=COCCC3)C)cn12 C1(C)(COC)CCCN(C(C2CCN(C(=O)CC3(C)CCCC3)C2)=O)C1 C(=O)(C(O)CCCNC(C1CC(C)N(C)C1)=O)NCCC(=C)C C1(C(=O)NC2CCCC2CNC(C2CCC2)=O)Cc2cccnc2C1 CC1(C)C(CNC(C2CCC=CO2)=O)CCN1c1ncc(O)cn1 N1(C(CCNC(COC)=O)=O)CC(NC(C2CC23CCCC3)=O)C(C)(C)C1 N1(C(C2N(CC)CCC2)=O)CC2CN(C(c3ccc(F)c(C#N)c3)=O)CC2C1 N=c1[nH]c2ccc(C(N3CCC(CNC(=O)CCCN=[N+]=[N-])C34CC4)=O)cc2[nH]1 N1(C(C#CC(C)(C)C)=O)CC23CCCCC2(C1)CN(C(C1CC(C#N)C1)=O)C3 N1(S(CC)(=O)=O)CCC2CCC(C1)N2C(=O)NCCc1cn(C(C)C)nn1 CC1CCCCc2cc(C(=O)NCCCNC(c3coc(C(C)(C)C)n3)=O)nn21 N1(C(c2cnc(C(C)C)o2)=O)CCC2(CCC(NC(=O)CC3(CO)CC3)CC2)C1 C1(C(=O)NCC2(NC(C(C)C3CC3)=O)CC2)CN(C)CC1c1ccccc1 c1(C(=O)NCCOC2CCN(c3snc(C(=O)OCC)n3)C2)c(CC)noc1C Cc1nc(N(C)C)sc1C(=O)NC1CC(CCNC(=O)C=CCO)C1 c1(C2(O)CN(C(=O)N(CCc3c(C)nc[nH]3)CC)C2)cccc(Br)c1 N1(c2c(OCCCC)cc(Br)cc2)Cc2ccc(C(=O)O)cc2C1 c1(C(N2CC(O)(C(C)NC(CC=CCC)=O)C2)=O)cccc(C)c1Br C1(N(C(c2c(CNC(c3c(C(N)=O)csc3)=O)noc2)=O)C2CC2)CCS(=O)(=O)C1 c1(C(=O)NCCC2(O)CN(C(C3C(C)CC3C)=O)C2)ccc(CC2CC2)cc1 N1(C(C(CC)COC)=O)C2CCC1C(C(N1CCC=CC1C(=O)OCC)=O)C2 c1(N(C(=O)C#CCNC(C2CS(=O)(=O)C2)=O)CC)ccc(O)cc1 C12(C(=O)NCC(CC)NC(c3cnnc(C)c3)=O)CCC(CC1(F)F)C2 CN1N=CC(CC(=O)NCC(C(=O)NCCN2CCNC2=O)N(C)C)C1=O C(=O)(C(C(C)NC(C1CCCC1O)=O)C(C)C)NCc1nccc(C)n1 c1(C(=O)N(C(C)Cn2cc(CN3CC4CC4C3)nn2)CC)c(Cl)nc2ccccn12 C1(C(=O)OC)CC2(CCC(CNc3cccc(CN(C)CC#N)n3)O2)C1 CC1CN(C(=O)CC2CC3(CC3)CO2)CC1NC(c1cnc(O)s1)=O c1(C(=O)NCCOCCCN(C(c2cc(OCC)n[nH]2)=O)C)ccccc1C c1(CC)nnc(O)c(C(N2CCC(CNC(=O)C(O)CCC(C)C)C2)=O)c1CC CCCCCC(C)(C)C(=O)N(CC(C)CNC(C1CCCN(C(C)C)C1)=O)C c1(NC2CC2F)cc(F)ccc1N1CCCCC1.C1(CNC(=O)N)(C)CC1 CC(C)C(F)(F)CC(=O)NC1CC1CNC(c1cc(N)ccn1)=O C(CC(C)(C)C(=O)NC(C1CCCN(C(=O)C2=C(Cl)CC2)C1)C)OC C1(C(C)C)CCCC1C(=O)N(CCCCCC(=O)CSc1nncs1)C(C)C.N C12(C(=O)NCCN(CCOC)C(c3coc(CO)n3)=O)CCCN1CC(OC)C2.C1CC1 N1(C(Cn2ncc(C)c2)=O)CCC(NC(=O)Cc2cnccn2)C(F)C1 Cc1cccc(CC(=O)NC2(CCCCNC(C3CC4CC4C3)=O)CC2)c1 N1(C(CSCC(=O)OC)=O)CC(=C(F)CNC(=O)CCC2CCCO2)C1 c1(C(=O)NC(CC(C)NC(COCCOCC)=O)C)cccn2c(C)cnc12 c1(C(C)(C2CC2)NC(CC)CNCCS)nnnn1C1CCCC1.C(C)(C)OC C1(NC(=O)CCn2cccc2)CCCCC1.C1(=O)C(=O)N(C2CC2)CCCN1C c1(C(N2CCC(CNC(CCN(C(C)=O)C)=O)C2)=O)cc2c(nn1)CCCO2 c1(C(N2CC(NC(C(C=CCCC)O)=O)C(C(F)F)C2)=O)c(F)ccc(F)c1Cl N1(C(CC2C(C)CCN(C(c3cc(C)oc3)=O)C2)=O)CCC12CCOCC2 C(=O)(CCCCNC(=O)C(C1CCCO1)NC(=O)C(c1ccccc1)C)OCC CC1(C)CC(O)CN1C(C1CCN(Cc2c(I)ccnc2F)CC1)=O N1(C(c2nnc(C)o2)C)CC2(CN(C(c3ccc(F)c(O)c3)=O)CCO2)C1 c1(C(N2CC(C)(NC(=O)C3=C(C#N)CCC3)C2)=O)cnn2c(Br)cccc12 CCS(=O)CC(=O)NCC1(F)CC(NC(c2cccn2-c2ccc(F)cc2)=O)C1 Cc1c(CNC(C23CC(CO2)N(CC2CN(C4CCC4)C2)C3)=O)cccc1F C1(C(N(C)CC)=O)CCCCCN1C(c1sccc1F)=O CCCC(CCCNC(=O)Cc1ccsc1)NC(=O)C=CCOCCOCCO C(=O)(C(C)CC(C)(C)C)NCC(CC)NC(c1cc(O)cc(C#N)c1)=O C#Cc1ccc(C(=O)N(C(CC)C(=O)OC)C)cc1Br N1(C(c2c(Cl)cnc(C)n2)=O)CC2OCC(NC(C3(CC(F)F)CC3)=O)C2C1 c1(C(=O)NC2CC(O)(CNC(C3CCC3(F)F)=O)C2)ccc(F)cc1Br c1(CC(=O)NC2CC(CNC(c3ncc(N(C)C)nc3)=O)C2)ccc(F)c(Cl)c1 c1(C(=O)NCCC2(O)CN(C(C3OCCN(C)C3)=O)C2)ncnc(O)c1F O=C(O)CCCn1cc(CC(=O)Nc2cc(-c3ccns3)on2)cn1 Cc1noc(C)c1CC(=O)NCC1C2CN(C(C3CC(=O)N3)=O)CC12 c1(CC)cncc(-c2cn(CC3CC(NC(=O)C=Cc4ccc(C)o4)C3)nn2)c1 C1(c2cn(COCC)nn2)CC(OC(C2(C(=O)OC)CC2C(F)(F)F)=O)CN1.C(C)C C(=O)(C#CC1CCCOC1)NCC(C(C)C(C)C)NC(c1cccc(CC)n1)=O N1(C(c2ccc(OC)c(C)c2)=O)CCOC2CCN(C(=O)CC3CC3(Cl)Cl)CC12 N1(C(COCCCC#C)=O)CC(NC(c2cc(CO)[nH]n2)=O)CC12CCCCC2 CC(C)CC(CNC(c1cnn[nH]1)=O)C(=O)NC(C)CCc1cn[nH]c1 c1(N(C)Cc2cccc(F)c2)nc2ccsc2c(=NCCN(S(C)(=O)=O)C)[nH]1 C1(C(N(CCCOCCNC(=O)CCn2cccc2)C)=O)COCCN1C=O Nc1c(C(=O)NC2COCC2CNC(C2OCCC2C(F)F)=O)cc(Cl)cc1Cl C(c1cscn1)=CC(=O)NCC1(CN(C(C(C)=CC2CC2)=O)C)CC1 N1(C(C2(CCNC(c3n(C(C)C)cnc3)=O)CCCC2)=O)CCC(O)CC1C C1(NC(C(CC)COC)=O)CC2CCC1CC2NC(=O)COC1CC(F)(F)C1 C1(CNC(C(CCC)(C)C)=O)CC12CCN(C(=O)Cc1ccc(F)cc1)CC2 N1(C(C2C(C)C2)=O)CCCC(C)(CNC(=O)C(F)CC2CCCCC2)C1 Cn1cc(C(=O)NC2CN(C(=O)COCP(C)(C)=O)CC2C(F)F)ncc1=O c1(-c2n(-c3c(C)c(Cl)ccc3)nc(C3CCCCC3)n2)cc2nc(C)sc2[nH]1 c1(Nc2cc(C)cc(N)c2)c2c(nn1C)CCC2 c1(CNC(=O)Cc2cncn2C2CC2)ccc(CNC(c2cnco2)=O)c(F)c1 C12(NC(=O)Cc3nc([N+](=O)[O-])n[nH]3)CCOCC1CN(C(=O)C=CCF)C2 CC1CC(NC(=O)CCC(=O)c2cccc(N)c2)CN1C(=O)C1=CCCC1 C=CCC(C(=O)NC(CNC(=O)CCCc1c(F)cccc1F)C1CC1)C(C)C c1(C(=O)OC)ccc(O)c(NC(C2CCCCC(=O)C2)=O)c1 C(=O)(C#CC(C)C)NCC1CC(NC(c2cc(C(=O)OCC)sc2)=O)C1 CC(=O)C(C)(C)CC(=O)N1CC2COCC2(C(N2CCOC(C(N)=O)C2)=O)C1 C1(NC(N2CCC(C(C)CO)CC2)=O)CC2(Cc3c(OC)scc3)COC1C2 Cc1ccc(CC(=O)NCC(O)CNC(C2(C)COCCO2)=O)c(Cl)c1 Cc1cc(CNC(c2occc2CNC(C2(O)CCOC2)=O)=O)nnc1C C1(NC(=O)C(F)F)C2CC3C(C2)C13C(=O)NCC1CC2(CC2)C(=O)O1 c1(C(CC)CC)cc(C(=O)NC2CC2CNC(=O)CCCn2cccn2)on1 C1(NC(CC=C)=O)C2CCCC1CC(NC(c1cc(=O)c(C)c[nH]1)=O)C2 C1(C(C)C(=O)NCCC2COC(=O)N2)CCN(CCN2C(=O)CNC2=O)CC1 CC1CCC(CC(=O)NC(C)CC2CCN(C(=O)CC(C)N(C)C)CC2)CC1 N1(C(C2N(C=O)CCC2)=O)CC2(CCN(C(=O)C(=Cc3c[nH]cn3)F)C2)C1 CON1CCC(C(=O)NC2(CC(=O)NCC3CCSC3)CC2)CC1 Cc1nc(C=CC(N2CC(NC(C3(C#N)CC3(C)C)=O)C(C)C2)=O)[nH]c1C N1(C(C(CC=C)OC)=O)CC2CC(C(=O)NC3CCCC3(C)N(C)C)(C2)C1 N1(C(c2cc(C(=O)OCC)no2)=O)CCC2CN(C(=O)CCC(C)C)CCC12 C=C(Cl)CC(C(=O)NC(Cc1ccco1)CO)NC(c1cnc2n1CCC2)=O C1(CNC(c2nnn(C)c2C(F)(F)F)=O)CCN(C(c2cc(Cl)cs2)=O)C1(C)C N1(C(C=C(CCN(C)C)Cl)=O)CCN(C(=O)C=CC2CCCN2C)CC1CF c1(CC)ccc(C(=O)NCC(CC)NC(c2ccn(C)c2)=O)s1 N1(C(C#C)=O)CCC2(CCCC2C(=O)Nc2ccc(F)cc2C)C1 c1(C(=O)Nc2c(C)nn(C)c2)ccc(Br)cc1I.c12ncc(cn1)C1CCCN21 C(=O)(C1=NOC(CNC(=O)CN2CC3CC3C2)C1)NCc1c(C)cnn1C c1(CC)nc(C)oc1C(=O)N(C)CCOCCC(=O)N(C)Cc1occc1C CC(CC(C)(C)C)C(=O)NC1CN(C(c2csc(O)n2)=O)CC1c1nccn1C C(C1=NOC2CCCCC12)CN1CC(=O)N(Cc2c(OC(F)F)cccc2Cl)C1=O C1(NC(C2(OC)CC2)=O)CCCC(NC(c2cccc[n+]2[O-])=O)CC1 c1(C(c2nnnn2-c2ccccc2)NC2(CF)COC2)nccc(Cl)c1F c1(CC)cccnc1C(=O)NCC(C1CCCCN1C(c1cccnn1)=O)(C)C c1(C(=O)NC2C3(CCC(NC(C(N)=O)=O)CC3)C2)c[nH]c2nc(F)ccc12 C#Cc1ccc(C(=O)N(C)CC2CC(F)CN2C(C2CN(CC)CCO2)=O)cc1 C1(CCC(=O)NC2C(NC(c3scc(C(C)=O)c3)=O)CCC2)C(=O)NN=C1C Cn1ccc2c(-c3noc(C4CCCCS4)n3)ncnc12 C1(CC(=O)NC23C(CN(C(CCCOCCC)=O)C2)C3)CCC(F)(F)CC1 c1(C(=O)NC2CN(C(c3cc[nH]n3)=O)C2)ccc2nnc(O)n2c1 N1(C(CCC)=O)CCC(C(=O)NCC(c2c(C)c[nH]c2C)=O)(COC)CC1 c1(SC)ncc(C(=O)NC23CC(C(=O)NCc4cnc(C)[nH]4)(C2)C3)cn1 CN1C(=O)CCCC1C(N1CCCC1Cn1cc(Cn2ccnc2)nn1)=O CC1CC2(CC(C(N3CC4CC(NC(=O)Cc5cocn5)C3C4)=O)C2)C1 N1(C(c2cccc(OC(F)F)n2)=O)CCc2c(ncn2-c2ccccc2Cl)C1 CCCCCCC(C)NC(=O)C(CCOCC)NC(=O)CC1(C)CCOC1 C#CCCCCCC(=O)NC1(C)CN(C(=O)CSc2cc(C)ccc2C)C1 c1(CC)cc(Cl)ccc1C(=O)NC(C)CNC(=O)COc1ccc(F)cc1 n1(C(C)(C)C)ccc(C(=O)NCC2CC2NC(=O)CCCc2cccnc2)n1 CN1C(=O)CCC1C(=O)NC1CN(C(=O)CCc2cncn2C)CC1O c1(C(=O)NCc2ccc(-c3cn(C)nc3)s2)cncc(N(C)C)c1 Cn1cnc2cccc(C(=O)NC3CC3NC(c3cnc(S)n3C)=O)c12 C1(CC)(NC(C2CC(=O)N(O)C2)=O)CCCN(C(c2ncn(C)c2C)=O)C1 CC(C)CC(CNC(=O)C(C)c1ccco1)C(=O)NC(c1cncc(F)c1)C N1(C(c2cc3ccccn3c2)=O)CCCC12CCN(C(C1(C3CCC3)CC1)=O)C2 CCC(C)CCC(=O)N(C1CC2CC1N(C(=O)Cc1cc(Cl)n(C)n1)C2)C C#Cc1ccc(C(=O)OC(C)(C)C)nc1C.C12CCN(C(S(N)(=O)=O)C1)C(=O)N2.OCC C1(NC(C(CCC)NC(N)=O)=O)CC2CC(NC(=O)CCCSC)C2C1 C1(C(=O)NCC2CC(NC(=O)Cc3nnc(C)o3)C2)(OC)CCCSC1 C12(OC)CCC1CN(C(=O)C(CC(N)=O)NC(=O)CC13CCC(CC1)C3)C2 c1(C(=O)NC(CCCC)CNC(c2ccnn2COC)=O)cccc2c1COC2 c1(C(=O)NC2C(NC(CNC(N)=O)=O)CC2)cnoc1-c1ccccc1 C1(NC(CCSCCC)=O)CN(C(c2c[nH]cc2CC)=O)CCC12CCC2 C1(OCCNC(CCC=CCC=C)=O)CCN(C(=O)CC(C2CC2)C2CC2)CC1 C(=O)(CC(C)CC(F)(F)F)N1CCC(O)(CCNc2cc(OC)ncn2)CC1 c1(OC)ncc(C=CC(=O)Nc2cccc(CNC3CCC(C4CC4)C3)c2)cn1 Cc1nn(-c2ccc(F)cc2)c(CNCc2nocc2C2CCC2)c1Br C(C(C)(C(C)C)NC(c1nn(C)cc1C)=O)NC(c1nc(NC(C)=O)sc1)=O N1(C(C2C(C(N)=O)CC2)=O)CC=CC1C(=O)NCCF c1(C(N2CCC(C)N(C(C3CCCS3)=O)CC2)=O)c2c(nn1C)CCCC2 C1(C)(NC(CCNC(C2CN(C)C(=O)C2)=O)=O)CCCCC1(C)C C1(C(=O)NC2COCC2NC(C2(CF)CCC2)=O)Cc2cc(Br)ccc2O1 N12CCN(CC1)C(=O)c1csc(n1)C2.c1(SCC)ncnc(=N)[nH]1 N1(C(C2(C)CCCN2C(=O)CC(O)c2ccccc2)=O)Cc2cccc(Cl)c2C1 c1(C(=O)NCC(C)NC(c2c(CC)[nH]cc2)=O)cnn(C2CC2)c1C c1(C(C)C)nc(NCCSc2nccn2C)cc(N2CCC(CO)C2)n1 c1(C(=O)NCC2CC(F)(CNC(CSCC)=O)C2)ccc(Cl)c(S(N)(=O)=O)c1 C1(C(=O)NC(c2nc(-c3ccncc3)no2)C(C)C)CC2CCC(C1)C2(F)F N1(C(c2c(COC)cccc2)=O)CCCN(C(C2CC(=O)N(OC)C2)=O)CCC1 c1(C(COC(C(C)Cc2ccco2)=O)=O)ccccc1C(F)(F)F N1(C(N(c2ccc(F)cc2)C2CC(C)C2)=O)CCCNCC1 c1(C(C(=O)N(CCCN(C(=O)CCC2CCCCC2)C)C)O)ccc(F)cc1 Cc1cc(C)n2nc(CCNC(=O)NC3C(Cl)(Cl)C34CC4)nc2n1 c1(C(=O)NC(CNC(C(c2ccc(F)cc2)C)=O)C2CC2)ccnc2ncnn12 c1(C2C(C(=O)NCC(CC)NC(c3n[nH]c(C)c3O)=O)C2)ccncc1Cl c1(C(=O)NC(CNC(C(C)(C)CC(F)F)=O)(C)C2CC2)cncc(S(C)(=O)=O)c1 CCC(C)C(C)C(=O)NC1CCCC1NC(=O)CC1CCN(S(C)(=O)=O)CC1 C1(=O)CCN(OC)C(=O)C(CO)N1.CCC(CC)n1cccn1 C=C(C)C(C)(C)C(=O)NCCC1CCC(NC(=O)C(C)C)C1 N1(C(C2(CC)CCN(C(c3cc(C)c(C)o3)=O)C2)=O)CCCC(C)(C)C1C c1(C(N2CC3(CN(C(Cc4cc(C)sc4)=O)C3)C2)=O)cc(S(N)(=O)=O)sc1C C1(NC(C(C)OCC)=O)CN(C(c2ccc(C(=O)OC)cc2)=O)CC1F C1(NC(C2OC3CCC2C3)=O)CCC(NC(C2C(Cl)(Cl)C23CC3)=O)CC1 c1(OC)ccc(C(CNC(=O)Cc2cnn(C)c2C)NC(C2CC(C)C2)=O)cc1 N1(C(C(c2ccc(C)cc2)=O)=O)CCN(C(c2ccc[nH]2)=O)CC1CC(C)(C)C Cc1nnc2n1CCN(C(=O)C(C1(O)CCC1)NC(=O)Cc1ccccc1)C2 n1(CC)nc(C(=O)NCC2C3CC3CN2C(C2CC2F)=O)ccc1=O C1(NC(c2c(C)sc(O)n2)=O)CCN(C(=O)C(C)CC(C)C)CC(C)(C)C1 C=CC1(CNC(=O)C(CC)NC(c2nc(Cl)cs2)=O)CCC1 Cc1cc(NC(C23CC2CN(C(=O)C#CC2CC2)C3)=O)cnc1C C1(CC)(CC)CN(C(=O)CC(C2CC2)NC(=O)CC2CCC(O)C2)CCO1 c1(CC(=O)NCC2CC(OC)CN2C(=O)COc2ccsc2)ccc(O)cc1Cl C(=O)(C(C)(C)CCNC(c1cc(Cl)n[nH]1)=O)NC1C(C2C(C)C2)C1 CN=c1nc(C(=O)NCC2CCCN2C(=O)CN2CCC(C)(C)C2)cc(C)[nH]1 C=Cc1cnn(C)c1C(=O)NCC=CCNC(=O)Cc1cnn(C)c1 N1(C(c2cc(OCC)no2)=O)CCC(C)(CNC(=O)CCSc2ccccn2)C1 C1(NC(CCc2onc(CSC)n2)=O)CN(C(c2[nH]c(C)nc2C)=O)CC1C c1(OCC)ccnc(CC(N2CCC(C)(NC(C3CCC(OC)C3)=O)C2)=O)n1 C12(C(N3CCCN(C(CC4OCC(C)OC4)=O)CC3)=O)CCC(N=[N+]=[N-])C1C2 Cc1ncc(Cl)cc1NC(c1nc(C(C)C)n(-c2cccc(Br)c2)n1)=O Oc1c(NCC2(c3ccc(Cl)cc3Cl)CCCC2)cccc1O C#CC1CCC(NC(c2ccc(CNC(C3CCC(N(C)C)C3)=O)nc2)=O)C1 c1(CNC(=O)OC(C)(C)C)cc(C(=O)NC2CC(OCC(N)=O)C2)co1 C1(C(=O)NC(c2ccccc2)C(=O)NCC2(CO)CCN(C)C2)CC(=O)OC1(C)C c1(OC)cc2nn[nH]c2cc1C(=O)NC1CCCCC1NC(=O)CCC(C)(C)C Cc1nc2c(C(N3CC(NC(c4cn(C)nn4)=O)CC3CO)=O)cccc2o1 Cc1c[nH]c(C(N2CCCC2(C)CNC(c2cnn(C(F)F)c2)=O)=O)c1C c1(OC)c(C)cc(C(N2CCN(C(c3ccc(C)cc3)=O)CC2)=O)cc1C N1(C(c2c(OC)scc2)=O)CC2(CCC2NC(=O)C(=Cc2cccs2)C)C1 CC1(F)CN(C(c2ncn(C(C)(C)C)n2)=O)CCN(C(C2(C)CC2(F)Cl)=O)C1 c1(NC(C2(C)CCCN(C(=O)COCC3CCCO3)C2)=O)ccc2ncnn2c1 N=c1cc[nH]c(C(=O)NCC2CC(CNC(C34CCC(C3)C4)=O)CO2)n1 C1(O)(C(=O)NC23CN(C(CC4(CSC)CC4)=O)C(C2)C3)Cc2ccccc2C1 N1(CC2CN(S(c3c(C)onc3)(=O)=O)C2)Cc2ccccc2-c2ccccc2C1 n1(CCNC(NCC(C)C)=NCCc2ccsc2)ccc2c(Br)cccc12 c1(-c2nnc(-c3ccc(-c4n(CC(C)O)ccn4)s3)o2)cc(=O)cc[nH]1 Cc1ccnc(C(=O)NCC2(O)CCN(C(=O)CN3CCCNC3=O)C2)c1O C1(NC(c2c(CC)scn2)=O)CN(C(c2cc(Cl)c(Cl)[nH]2)=O)CC(C)(C)C1 CC1C(NC(c2snnc2C2CC2)=O)CCCN1C(c1cc(C2CC2)on1)=O CN1N=CC(CC(=O)NC2CCCN(C(=O)CC3(O)CCOCC3)C2)C1=O c1(C(=O)NC(c2cccc(F)c2)C(N)=O)scc2c1CCCC2 CCCN=c1[nH]c(=NC2CCCCN(Cc3ccccc3)C2)c2[nH]ccc2[nH]1 C1(C(N2CC(C)(NC(c3n[nH]c(CC)c3C)=O)C2)=O)CC2OC1C1CC21 N1(c2cc(C)nc3n2ncc3)CC2CCC1CN(C(=O)C(C)NC=O)C2 c1(C(=O)NC2(C)CC(NC(C3COCC(C)O3)=O)C2)ccc2nccn2n1 Cc1nc(CNC(=O)C(CNC(=O)CC23CCCC2C3)N(C)C)sc1C c1(C(=O)NCC(C2CC2)NC(C(C)(C)OCC)=O)cc2c(F)ccc(F)c2s1 n1(CCNC(Cc2c(-c3ccc(SCC)cn3)cccc2)=O)ccc2ccccc12 CC1CC(C)(C(=O)NC(CCN(C(=O)Cc2nc[nH]n2)C)c2cccs2)C1 N1(C(c2c(C)nns2)=O)CCCC2(CCN2C(C2CCC(O)C2)=O)C1 C(=O)(C(F)C(F)(F)F)NCC=CCC(=O)N(CC)Cc1ccccc1 CCCC(C(=O)N1CC(c2ocnc2CNC(c2occc2F)=O)C1)C(C)C N1(CCC)CCCC1C(=O)NC(C)CCNC(c1cnoc1C1CC1)=O C(C(C)CC(=O)NCCCC(C)NC(=O)CSCCc1ccccc1)OC C1(C(=O)NCC2N(C(C=CCC)=O)CC(F)(F)C2)CCOC2(CCCC2)C1 CC(C)CS(=O)(=O)CCC(=O)NCCCN(C(=O)CCc1cscn1)CCO N1(C(COC(C)=O)=O)CC2C(NC(c3ccc(CN)cc3)=O)C2C1 c1(OC(CC)C(=O)N2CCCC2C(C)NC(=O)CS(N)(=O)=O)ccccc1C Cn1ncc2c(=O)n(C(=O)CCN3CCSC3=O)cnc12 N1(C(CSC(c2ccccc2)C)=O)CC2CCC1CN2CC1CC(C(C)(C)C)C1 c1(CC)cc(C)ccc1F.C12CCCCC1NC(=O)C(CN(C)C)NC2=O c1(CNC(C2CC2Cl)=O)n[nH]c2c1CN(C(=O)Cc1ccsc1)C2 O=S(=O)(c1ccc(NCC2CCCN2c2ccccc2)c(Cl)c1)N1CCC=C(F)C1 CC(CN=c1cc(C2CCC2)nc[nH]1)NC(c1cc(F)c(F)cc1Cl)=O C1(C(=O)NCC2OCCN(C(c3c[nH]c(=NC)o3)=O)C2)CC(C)(C)OC1(C)C C12(NCCc3nc(C(C)C)sc3)CCCCC1C2Br C1(NC(C2(CCOC)CCC2)=O)CCCC2CN(C(c3cnsc3C)=O)CC12 CCCCC(C)C(=O)N1CC(CCNC(=O)CC=CCOC(=O)OC(C)(C)C)C1 N1(C(C(N(C)O)=O)=O)CCC(O)(CNC(=O)NC)CC1 C1(NC(C(C2CC2)N(C2CCOC2)C)=O)CCCN(CC(=O)Nc2ccccc2)C1 c1(CC)cc(C(=O)NCC2(O)CC(NC(=O)CC3CC=CC3)C2)c(C)nn1 c1(C(N2CCC(C(C)NC(n3ncn(C)c3=O)=O)C2)=O)csc2nccn12 CC(C)(C#N)CC(=O)N1CC(NC(C2CCC(=O)N2)=O)C(O)C1 c1(CC)ccc(F)cc1C(=O)NCC12CC(CN1C(C1CCOC1C)=O)C2 N1(C(c2n(CC(=O)OC)cnc2C)=O)CCCC(F)(CNC(c2cnn[nH]2)=O)C1 c1(CN(C(CCCOC)=O)C)cnn2c1CN(C(=O)C(C)S(N)(=O)=O)CC2 c1(CCCCC(=O)NC2CCC2CNC(=O)COC2CC2)nc2ccccc2s1 C1(NC(C2C(CNC(c3coc(C4CC4)n3)=O)CC2)=O)CC2OC(=O)CC12 Cc1cn2c(C=CC(=O)N(C3C4CCC3CNC4)C(C3CCC3)=O)csc2n1 C=C(C)CC(C(=O)N1CCN(C)C(CN)C1)OCC(=O)C(O)CCSC CCC(CC(=O)NCC(c1ccc(F)cc1)NC(C12CC(C)(C1)C2)=O)C(C)(C)C C1(NC(C2(NC(N)=O)CCCCC2)=O)CC(F)CN(C(C2(Cl)CC2)=O)C1 c1(C(=O)NCC2CC(NC(c3cc(CC)sn3)=O)C2)n[nH]c2c1CSCC2 C(=O)(C1=CCC(C)(C)CC1)NCC(C(C)(C)C)NC(c1cnc(O)n(C)c1=O)=O c1(C(N2CCC(OCC(=O)OC)C2)=O)cc(C#N)[nH]c1C C#Cc1cc(C(=O)N(CCCCC(=O)NCCCC(C)(F)F)C)ccc1C C1(=O)C(CN=[N+]=[N-])NC(=O)CC2C(CC2O)N1.C1(CC=C)CC2(C1)CC21CC1 N1(Cc2ccn(C(C)C)n2)CCC(CO)CC12CC2 c1(CN2CCCC(C(=O)Nc3c(OC)nnc(Cl)c3)C2)cc(C)c(Cl)c(C)c1 C(CN=c1[nH]ccc(=NCC2(C(N)=O)CCCCC2)[nH]1)N(CCC)C(C)C N1(C(C2(NC(c3cccc(CO)c3)=O)CC(F)(F)C2)=O)CCCCCC1 c1(C(=O)NCC(CC)(C)NC(=O)C(F)=CCCF)ccc(C)c(F)c1 N1(C(CN(CCC#C)C)=O)CCCC2(CNC(C3CC(C)=NO3)=O)CCCC12 Nc1cccc(C(=O)CCC(=O)NCC(O)CNC(C23CCCC2C3)=O)c1 c1(C(N2C(C(C)C)C(NC(c3cnncc3O)=O)CC2)=O)ccc(Cl)cc1O C=CCC(CNC(=O)C#CCNC(C)=O)NC(C1CS(=O)C1)=O N1(C(c2c(C)noc2)=O)CCCC(CNC(c2coc(-c3cccs3)n2)=O)C1 C(=O)(C1=NN(C)C(=O)CC1)NCC1(O)CCN(C(C=C2CCC(C)C2)=O)C1 C1(C(=O)NCC2OCC(CNC(CCC#C)=O)C2)CC2(C1)CC(C)(C)C2 N1(C(C=CCC)=O)CC(c2ccccc2)CC(N=c2ccnc(C(=O)NC)[nH]2)C1 C1(C(=O)NC2CC(CCC)C2)(OC)CCN(C(=O)C(C)Cc2cnc[nH]2)C1 c1(OC)ccc(C(N2CCC(CNC(=O)CC(F)F)C2)=O)c(Br)c1F N1(C(=O)Cc2nc[nH]n2)CC2CC(C1)CN(C(c1ocnc1C1CC1)=O)C2 c1(C(N(CCN(C(CSCCOC)=O)CCOC)C)=O)nnnn1C C1(C(N2CC(C)(CC=C)C2)=O)CCCCC1(C)NC(C1CCC(=O)C1)=O CN1CCC(C(=O)NCC2CCC2NC(=O)CCCC2CC2)S1(=O)=O c1(N(CCCOC)C)cc(C(N)=O)nc(-n2nc(C)cc2C)n1 C=CC(CC)C(=O)NC(CO)C(C)NC(c1cnn(CC)c1CC)=O N1(C(COCCSC)=O)C(C)CC2CN(C(=O)CCn3cccc3)CC12 c1(N(C)CC2CCOC2)ccn2ncc(S(=O)(=O)NC3CCC3(C)C)c2n1 c1(C(N2CCCC(N(C(=O)CCC3CC3)CC)C2)=O)c(F)ccc(C#N)c1F c1(C(N2CC(C)(NC(c3cc(COC)oc3C)=O)C2)=O)cccn2nnnc12 C1(F)(CNC(C(c2ccc(F)cc2)OC)=O)CCN(C(C2CCC(=O)N2)=O)C1 C(CNC(c1cccc(COC)c1)=O)(C(C)(C)C)NC(c1c(CCC)nns1)=O c1(C(=O)NC2COCC2CNC(C23CCCC2C3)=O)ccn(C2CCC2)n1 c1(NC(CC2N(C(c3ncc(C)[n+]([O-])c3)=O)CC2)=O)ccc(C)n(C)c1=O Cc1cc(F)c(CC(N2CCC3(C2)CN(C(=O)CC2(O)CCCOC2)C3)=O)cc1F O=C(CCCCCCNC(c1ocnc1C(F)F)=O)NC(CO)C1CCC1 C1(OC)CCCCC1C(=O)NC1CC(CNC(c2ccnn2CC#N)=O)C1 CC1(C)C(C(=O)NCCS(C)(=O)=O)CCN1C(=O)CC=C(Cl)Cl C1(CNC(CC(=C)C)=O)CCN(C(=O)COCc2nccn2C)CC1C Cc1nc(F)ccc1C(N1CC(CC(=O)Nc2cc(Cl)ccc2N(C)C)C1)=O Cc1nn(C)c(N)c1C(=O)Nc1c(C)nn(C)c1Br N1(C(Cn2c(C)cc(C)n2)=O)CCCN(C(c2ccc(F)c(Cl)c2)=O)C(C)C1 c1(OC)cc(C(=O)NCC2COCCN2C(c2ccsc2)=O)cc(C2CC2)c1 C1(NC(CC(CC)C)=O)CC2CC(NC(c3cc(CO)[nH]n3)=O)C1C2 CN1CCC23CC(N(c4cccc(C(F)F)c4)C)C(CC2)C13 C1(CCNC(C2CS(=O)(=O)C2)=O)CCN(C(=O)CC23CCC(CC2)C3)CC1 C1(NC(c2[nH]cc(CC)n2)=O)C(C)CN(C(C2(C3(C)OCCO3)CC2)=O)CC1C C1(C2CCCN(C(=O)C(F)(F)C(F)F)C2)(NC(C2C(C)(C)CCCC2)=O)CC1 Cc1nn(C)c2cc(NC(=O)CC3CCC(C)C3)ccc12 C(C1C(C(=O)N(CC(C)N(C(=O)CCSC(F)(F)F)C)C)C1(C)C)=C(C)C N1(C(C2CCOCC2)=O)CCN(C(C23CC(O)C2C3)=O)CC1CO N1(C(C=CCCC)=O)CCOC2CN(C(=O)C(C(C)C)n3cccc3)CC12 C=CCC(C(=O)N1CCC(C(C)(C)C(=O)Nc2ccc(OC)nc2)C1)NC(C)=O c1(C(N2CCC(C(C)C(=O)NCC3CCC(F)C3)C2)=O)ccc(F)c(Cl)c1 c1(NC(C)=O)ccc(C(N2CCCC2C(C)NC(C2CC(C)=NO2)=O)=O)cc1 C12(NC(C(C)OCC)=O)CC(C)(C1)OC21CCN(C(C2CCC(F)(F)C2)=O)CC1 c1(OC)ccc2c(c1)CCCC2C(=O)NC12CC(NC(=O)CO)(C1)C2 c1(C(N2CCN(C(C(C=C=C)C)=O)C(CCO)C2)=O)nnn2ccccc12 c1(C(=O)NCC2CCCCN2C(=O)C=CC(F)F)cccc(F)c1Br c1(CC(N2C(CNC(c3nc(C(C)OC)sc3)=O)CCC2)=O)cncc(C#N)c1 N#Cc1ccc(Cl)c(C(=O)NCC2CC(CNC(C3(O)CCC3)=O)CO2)c1 CC(C)C(C)(CNC(=O)CCCN1C(=O)CNC1=O)NC(C1C=CCCC1)=O C(=O)(C(C)(C)CC(F)F)NC1CCN(C(c2c(CC)cccc2C)=O)C1 N1(C(C(C2CN(C(C3(CC=C)CCOC3)=O)C2)O)=O)CCCC(N=[N+]=[N-])CC1 c1(C(N2CC3CN(Cc4c(Br)cn(C)n4)C3C2)=O)ccc2c(c1)CCO2 C(=O)(C(F)(F)F)NCC(=O)NC1CCN(C(=O)C(O)c2ccco2)C1 Cc1ncnc(C(=O)NCC2(F)CN(C(=O)C(c3ccccc3)F)C2)c1C Cc1cccc2[nH]cc(CC(N3CCC(C)C(NC(=O)C(F)F)C3C)=O)c12 C=CCCCC(=O)NCC12CC(CN1C(=O)C(C)SC(C)C)C2 Cc1cc(COC(C2CCC2c2ccccc2)=O)c(O)nc1C.C1(=O)CCCN1 c1(C(=O)OCC(C)C)ccc(C2OCCO2)c(F)c1 c1(OC)ccc(Cl)cc1CC(=O)NCCOC(C)(C)CNC(=O)CCCN(C)C C(=O)(C(CC)CCC)N1CCC(C)(NC(COCCCCOCC#C)=O)C1 C1(C(N2CCCC(C(C)C)C2)=O)CC2C=CC1N(C(c1cncn1C(C)C)=O)C2 c1(CNC(C(C)SC(C)C)=O)cccc(C(=O)NCc2ccc(F)s2)n1 N1(C(C=CCCC)=O)CC2(CCN2C(=O)CCc2ncccc2C)C1 C(=O)(CCCN=[N+]=[N-])N1CC(OCCNC(C(CC#C)NC(=O)COC)=O)C1 N1(C(C2C(C)(C)C2)=O)CCN(C(=O)Cc2cnc[nH]2)CC1c1ccc(F)cc1 N1(C(Cc2nc(C(C)C)sc2)=O)CCCC(C2CC2NC(c2cnsc2)=O)C1 C1(C(N2CC(CC(C)NC(=O)CC34CCC(CC3)OC4)C2)=O)CC2(CCC2)CO1 c1(SC)cc(C)nc(N2CCCC(C(=O)NC3CC(=O)N(OC)C3)C2)n1 N1(C(C2(C)CCCO2)=O)CCCC(NC(C2(F)CC=CC2)=O)CC1 c1(C(=O)NC(CCNC(C=C(C)C(C)C)=O)(C)C)ccc2cnoc2c1 c1(C(N(C)CC2(NC(Cc3cncc(C)c3)=O)CC2)=O)ccc2[nH]ccc2c1 C(=O)(C(C)(C)C(C)(F)F)N1CCN(C)CC1CNC(C1(CCO)CC1)=O c1(C(=O)OC)cccc(NC(C2CC2C(=O)Nc2ccc(C)cc2F)=O)c1C C1(C(=O)NCCC(O)CN)(CC)CC=CCC1 N1(C(c2[nH]cc(C)c2)=O)CC(NC(=O)C=Cc2cn(C)cn2)CC12CCCC2 C1(C(C)NC(=O)C(C)(C)c2ccsc2)CCN(C(c2ccc[n+]([O-])c2)=O)CC1 c1(OC)ccccc1OC1CN(C(=O)CC2(N)CCSCC2)C1 N1(C(CNC(CCC)=O)=O)CCC(CNC(c2cnn(C)c2CC)=O)C12CCC2 Cc1ccc(C(N2CCOCC2CNC(=O)C(O)C(C)C)=O)c(O)n1 C1(CCC(C)C)CCC(C)CC1.C(CCO)NC C(=O)(C1=CC2CCCCCC12)N(C)CC1COCCN1C(c1occc1Br)=O C(=O)(CC(C)C(F)(F)F)NCCCC1N(C(C(c2ccc(C)o2)C)=O)CCC1 c1(CCC(=O)NCCC(C)NC(C23CSC(C2)C3)=O)cnc(C2CCC2)o1 CS(=O)(=O)c1ccc(C(=O)NCCOCCCNC(C2CCCO2)=O)s1 C1(NC(c2ccc(C(=O)OC)o2)=O)CCC(NC(=O)C(C)c2ccon2)CC1 N1(CC(=O)NCCNC(C2C(OCC)C2)=O)CCC(OC)C1.C1(OC)(CC)CCC1 CN1CC(C)(NC(=O)CC(C2CCN(c3ccccn3)CC2)N)CC1=O c1(OC)cc(C)cnc1C(N1CC(CCNC(C2CN(C(C)=O)C2)=O)C(C)C1)=O C1(C(=O)NCC(CC)CO)CN(C(=O)C(N2CCCCC2)C)CC1C c1(C(N2CCC(CNCc3cncc(C)c3)C2)=O)cccn2ccnc12 N1(C(c2cc(CC)no2)=O)CCC2(CCCCC2NC(=O)CCCN(C)N=O)C1 N12CCN(C(C3CC3)C1)C(=O)C1CC1CC2=O.CCCCC(=O)N1CCOCC1 c1(C(CNC(c2ccc(-n3c(C)cc(C)n3)nc2)=O)F)cccc(F)c1F c1(C(N(CCNC(c2cnccc2Cl)=O)CC)=O)cn2ncnc2nc1C C12COCCN1C(=O)Cn1cc2nn1.c1(COC(C)(C)C)ncns1 C(=O)(C1=CC2CCC(C1)C2)NC1(C(=O)NC(C2CCOCC2)C#C)CCCC1C N1(C(CNC(=O)OCC=C)=O)CCC(F)C(CNC(=O)C(C)n2cnnn2)C1 C1(NC(c2cc(C3CC3)[nH]n2)=O)CCCC2CN(C(C3CCCCS3)=O)CC12 c1(C(N2CCCC(CNC(C3ON=C(C)C3)=O)CC2)=O)cc(C)cc(C)c1C CC1CN(C(C2(CCN=[N+]=[N-])CC2)=O)CC1NC(=O)CC1CCCN(C)C1 C12(C(=O)OC)CC(CO1)N(CC1CCCN1Cc1ccccc1)C2 C=CCC(CC(F)F)C(=O)N(C)CC1(O)CCCN(C(=O)CCC(C)CC)C1 N1(C(C2(C#N)CC3CC3C2)=O)CC(NC(c2cnc(O)s2)=O)CC(F)(F)C1 Nc1ccc(S(=O)(=O)N(CCC(=O)NC2CC2)CC2CC(C(F)(F)F)C2)cc1 N1(C(C(CC)(C)F)=O)CC(NC(=O)CCc2cnc[nH]2)CC(F)C1 C1(C(=O)NC2C(C)CN(C(=O)C(N3CCSCC3)C)C2)CCC(C2CCCO2)O1 c1(C(N2CCOC(CN=[N+]=[N-])C2)C(=O)NCCCC)ccc(COCC)cc1Br Cn1c(C(N2CC3(NC(C45CCC(CO4)C5)=O)CCC2CC3)=O)ccc1[N+](=O)[O-] CC1Cc2cccc(C(=O)NCCOCCNC(=O)CC3=NN(C)C(=O)C3)c2O1 CC1CC=C(C(=O)NC2CC3CC2N(C(=O)CCc2cnn(C)n2)C3)CC1 C1(CNC(CCS(C)=O)=O)CCN(C(=O)CCSCc2ccc(F)cc2)C12CC2 C1(CC(=O)NCCc2ncc(C)cn2)CCN(C(=O)C2CC2)C12CCC2 n1(CC)ncc(Cl)c1C(=O)NC1(C)CN(C(C2CCCOC2C)=O)C1 C1(C(N2CC[Si](C)(C)C2)=O)CN(C(=O)C2=CCCOC2)C2(CCC2)C1 Cc1noc(Cl)c1CCC(=O)NC1CCCC(NC(C2CC3CCC2C3)=O)C1 CCCC(CCNC(c1cc(CNC(=O)CCC(C)(F)F)[nH]n1)=O)CCC N1(C(c2c(C)cccc2C)C(=O)NC(C)(C)C)CCSC2(CCCCC2)C1 CC1CCOC(C(N2CCC(NC(c3ccc(CN=[N+]=[N-])cc3)=O)C2)=O)C1 C1(CNC(c2nccc(SC)n2)=O)CN(C(C2(N(C)C)CC2)=O)CCC1C c1(C(C(=O)NC2CCC2)N(CCCC)CC)nscc1Br CC(C)(C(=O)N(CC(C)(C)C1CCOC1)C(C)(C)C)C(=O)N1CCCC1 Cc1c(Cl)ccc2[nH]c(C(N3CCCN(C(C4CCOC4)=O)C(C)C3)=O)cc12 O=[N+]([O-])c1ccc(F)c(Br)c1S(=O)(=O)N=c1ccc(-c2ccncc2)n[nH]1 N1(C(CC=CC=C)=O)C2CCC1CC(CNC(c1cc(O)nc(Cl)c1)=O)C2 c1(C(=O)NC2(CO)CN(C(Cc3c(C(C)C)con3)=O)C2)cccc(O)n1 c1(NC2C=C(C)CCC2)nc2ncn(C)c2c(=NCc2csc(C)c2C)[nH]1 C(=O)(C1CCC(=O)c2cccn21)NCCN(C(C1CCC(C)(C)CC1)=O)C1CC1 CC(CC(=O)N(CCCCC(=O)N1CC(O)(C(N)=O)C1)C)C(F)F c1(C(=O)NC2COCC2CNC(C2CC2[N+](=O)[O-])=O)cncc2c1CCC2 CCC(F)(F)C(=O)NCCC1CCN(C(c2ccnc(OCCOC)c2)=O)C1 Cc1cc(N(C(C)CNC(=O)C(C)C(C)S(C)(=O)=O)C)n2ncnc2n1 CCCCC(C(=O)NC(C1CN(C(c2c(C)nn3c2NCCC3)=O)C1)C)C(C)C S(=O)(=O)(c1ccc2c(c1)C(=O)N(C)C2=O)N1C(c2c(C)nc(C)s2)CCC1 c1(NC(C2CCCN(c3nccc(OCC)n3)C2C)=O)cnc2ccccn12 C1(C(=O)NCc2nc(C)sc2)COCCN1C(N)=O N1(C(CCC)=O)C2CCC1C(NC(c1sc(Cl)c(Cl)c1C)=O)C2 C=CC(C)(CCOC)C(=O)NC1CCCN(C(c2cc3cscc3s2)=O)C1C CCCCC(C)C(=O)NC(C1(C(=O)NC(C2CCCC2O)C)CC1)C c1(C(N(C2(CO)CN(C(C3CCOC3C)=O)C2)CC(C)C)=O)ccc(Cl)cc1 c1(C(N(c2ccc(C)c(C)c2)CC)=O)ccc2c(c1)OCCN2C(=O)OC(C)(C)C Cc1ccc(C(=O)NC2COCCN(C(c3cn(C)nc3C)=O)C2)c(I)c1 O=C(C1CCCCCc2ccccc21)NC1C2CN(C(c3cnn[nH]3)=O)CC12 Nc1cccnc1C(=O)NCC1(F)CC(NC(c2ccccc2SC(F)F)=O)C1 c1(NC2CCN(C(=O)OCC)CC2OC)ccc2ncc(Br)cc2c1 CC1CCN(C(C2CC2F)=O)CC1NC(=O)CCNC(c1ccc(N)cc1)=O CCC(CNc1ccccc1Sc1ccccn1)CC(C)O N1(C(=O)C#CC2CC2)CC2(CCN(C(=O)CC3(CSc4ccccc4)CC3)CC2)C1 N1(c2ccnc(C(CC)C)n2)CCn2ncc(CNC(=O)CCC(C)OC)c2C1 Cc1cnn(CC(=O)N(C(C(N2CCC(CCO)C2)=O)C2CC2)C)c1 c1(C(N2CCOCC(NC(C(C)O)=O)C2)=O)c2c(nn1C)CCSC2 N1(C(C=CC=CC)=O)CCC2(NC(=O)CCC3CC(OC)C3)CC2C1 C(=O)(C(Cc1cnc[nH]1)NC(=O)CC(C)F)NC(C)Cc1cnn[nH]1 c1(C(=O)NCCn2cc(CN(CCOCC)C)nn2)cnc2c(c1)OCO2 c1(NC2CCCN(C(C3(c4ccc(O)c(O)c4)CC3)C)C2)ccc(C#N)nc1 C1(O)(CC(=O)NCCCOCCNC(C(=Cc2ccco2)C)=O)CCCN(C)C1 C1(C(N(CCCC)CCO)=O)(NC(=O)C(C)C#N)CC1(C)C N1(CNc2ccc(-c3n(C)c(C(=O)O)cn3)cc2)CCC(F)(c2nn[nH]n2)CC1 N1(C(C2(C=C)CCC2)=O)CCN(C(=O)CC2=CCCC2)C(CF)C1 C1(C(=O)NCC(=O)NCC(C)C)C2CCC(C2)C1NC(c1cc(Cl)cn1C)=O C1(C(N(CC)CC2CC2)=O)CCCCCCN1C(=O)CC1(COC)CC1 C1(NC(C=Cc2nc(C)sc2)=O)C2CC1CN(C(c1nc(O)sc1C)=O)C2 c1(C(N2CCC(C)(NC(C(CSC)OC)=O)C2)=O)nc(Cl)ccc1N Cc1[nH]c(C(=O)Nc2cc(C(F)(F)F)cs2)c(C)c1C(N1CCC(F)(F)CC1)=O N1(C(c2c(CC)n(C)nc2)=O)C2CCC1CC(NC(C1CCN(CC)C1)=O)C2 C1(CNC(c2cccc(C(C)C)c2)=O)(NC(c2cscn2)=O)CCCCC1C c1(C(=O)NCC(C)N(C(C(CC)O)=O)CC)cccc(-n2ccnc2O)c1 Cc1[nH]nc2c1CCC(C(N1CC(C)(NC(c3ccccc3Br)=O)C1)=O)C2 c1(C(=O)NC2(C(=O)NCCCN=[N+]=[N-])C(C)(C)C2)ccc(O)cc1F C1(C(=O)NCCCC=C)CC12CCN(C(=O)CSC(C)(C)C)CC2 Cc1nsc(C(=O)NC2CCN(C(=O)Cn3nccn3)C2)c1Br C1(NC(CC=C=C)=O)CC(NC(c2cnc3[nH]cncc2-3)=O)C12CCOCC2 c1(N(C(c2cc(CCNC(CCCC=C)=O)on2)=O)CC)cnc2ccccc2c1 Cc1nc(C(=O)NC(C)C(=O)N(C2CC(C)C2)C)ccc1C#N c1(OC)cccc(S(=O)(=O)N2CCC23CN(c2cc(C#N)ncn2)C3)c1 c1(CCSCC(=O)NC2CN(C(C3(COC)CCCO3)=O)C2)ccncn1 N1(C(c2c(C)scc2)=O)CC(NC(=O)CC2CCSC2)C(O)C1 N1(C(C)=O)CCCCC1C(=O)NC1CCC(CNC(c2cc(CCO)on2)=O)C1 c1(OC)cncc(C(=O)N(CC(=O)NCCC2CC(C)(C)C2)CC(C)C)c1 Cc1ccc2occ(C(=O)NC3CCCN(C(=O)C#CC4CCCO4)CC3)c2c1 C1(NC(Cc2c(C)non2)=O)CC(O)CN(C(=O)Cc2ccc(F)cc2)C1 c1(C(N2CCC(NC(c3nnn(C)c3C(F)F)=O)C2)=O)cccc2c1CCOC2 CCCC(CCCNC(=O)C(C)Cc1ccco1)NC(=O)CS(=O)(=O)NC c1(C(=O)NC23CC(NC(C=COCC)=O)(C2)C3)cnn2cnc(Cl)cc12 N1(C(C2CCCN(Cc3cccn4nccc34)C2)=O)CCCC2(CCOC2)C1 N1(C(c2cc(C(C)=O)on2)=O)CC(F)CC1CNC(=O)CC(C)(C)N(C)C C1(COC)CN(C(C2(C)COC(=O)C2)=O)CCN1C(=O)C1=COCCO1 Cc1cc(N)ccc1C(N1CCC(NC(C2COCCC2C)=O)CC1)=O C(=O)(CCC(=O)NN(C)C)NCC(CC=C)NC(c1cc(CO)ccn1)=O C(CCCCC(=O)N1CCCC(C(C)C(=O)NC2CCN(C)CC2C)C1)OC CC1CCC(CNC(c2ccc(C(F)F)cc2)=O)CN1C(c1n[nH]cc1Cl)=O C1(NC(c2n[nH]c3c2CCCC3)=O)CCCCN(C(c2ccoc2)=O)CC1 C1(C(=O)NCCCS(C)(=O)=O)C2CCC(C2)C1NC(c1ccnc(Br)c1)=O N1(C(=O)Cc2cc3ccccc3o2)CCN(C(C2(F)CC2)=O)C2(CCC2)C1 C#CCCCC(=O)NCc1csc(CNC(C2CC(c3ccccc3)C2)=O)n1 Cc1cc(=NC(=O)CC2(C)CCCN(C(=O)Cc3cnoc3)C2)[nH]n1C(C)C CC1=NN(C)C(=O)C1CC(=O)N(CC(O)CN(C)C(c1ccnnc1)=O)C C#CC1(C(N2CCC(CC3CC3)C2)=O)CCN(C(=O)CN2CC=CC2)C1 CC1C(NC(C2CC3(CC3)CO2)=O)CCN1C(=O)CC1(C)CC1 c1(N2CCC(N(C(=O)C3=COCCC3)CCC)C2)nccc(S(C)(=O)=O)n1 C(=O)(CC(C)(C)CNC(C1CC=CCO1)=O)N(CCC(C)C)C c1(SC)cccc(C(=O)NC(CO)C(C)NC(=O)CC2(C3CC3)CC2)c1Cl C(=O)(C1=CC2(CCN(C(c3ccc(C)c(O)c3)=O)C2)C1)NC(C=C)C1CCC1 C1(CNC(=O)OC(C)(C)C)CCC2(CC(C(=O)Nc3cncc(Br)c3)C2)O1 c1(NCC(=O)NC2CN(C(c3ncn(C(C)C)c3)=O)C(C)C2)cccc(C#N)c1 C1(NC(c2cnn(CC)n2)=O)CC(CC(=O)N(C)CCC2CCC2)C1(C)C C1(NC(c2cnc(C)n2C)=O)CC2CCC1(C(=O)NC1(C)CSC1)C2 c1(C(N(C(C)C(N2CC(O)CC2CC)=O)CCC)=O)cc[n+]([O-])cc1 C1(C(N2CCCCC(c3cn(CC(CC)C)nn3)C2)=O)CCCCC12CCC2 C1(C(=O)NC(C)(C(=O)NC2COCC2F)C2CCC2)CCCC(=O)C1 c1(C(=O)NCC2(F)CCC(NC(CNS(CC)(=O)=O)=O)C2)cncc(C)c1C S(=O)(=O)(C1CCCCC1)NC1CC(c2ccc(Br)cc2)(C)C1 C=CCC(C(=O)N1CCC(CNC(=O)C(O)CC(=O)OCC)C1)C(C)C.C(C)(C)C c1(NC(N2CCN(C(C(=O)NC)c3cnc[nH]3)CC2)=O)c(C)cc(Br)cc1Cl C1(NC(CC(CC)C(C)C)=O)CC2(CCN(C(c3cnc(NC)cn3)=O)CC2)C1 O=C1NC(=O)C(CNC(C2CCCN(C(c3ccsn3)=O)C2)=O)N1 CCCC(C(=O)NCC1CN(C(C2CC(N3CC(O)C3)C2)=O)C1)C(C)C C1(NC(=O)CCNC(c2cnns2)=O)CN(C(C2COC(=O)N2)=O)CC12CC2 Cc1nc(C2CC2)sc1C(=O)NCC1CN(C(C2OCC2(C)C)=O)C1 N1(C(=O)CSc2ccccn2)CC(NCc2ccc(Cl)c(O)c2)C2(CC2)C1 c1(C(=O)NCCC(C)NC(c2cc(N(C)C)ccn2)=O)cc(F)n(C)n1 CCC(O)C(F)(F)C(=O)N(C(C)C(=O)NCCCC(C)(F)F)C C1(NC(C(c2ccc(F)cc2)(C)C)=O)CCCN(C(=O)Cc2ccon2)CC1 c1(C(C)=O)ccc(C(=O)N(C(C)C(=O)NCCc2nc(C)cs2)C)o1 c1(CC)ccc(C(=O)NCC2CN(C(=O)Cn3cccc3)CCO2)cc1F C1(NC(CCCC#C)=O)CC2CCC(C1)N2C(=O)CC1CCOCC1(C)C C1(CN(C(CC2CC(OC)C2)=O)C)CN(C(=O)Cc2cc(C)ns2)CCO1 C1(NC(c2c(C)snn2)=O)CCC2(CCCN(C(c3nc(Cl)ccc3N)=O)C2)C1 c1(CNC(C2CCCCO2)C)cc(Br)cc(Cl)c1O C1(CNC(C(N2C(CC)CCC2)=O)=O)CC2CC2N1Cc1cccc(OC)n1 C1(C(=O)NCc2occ(C(N(CC(C)(C)C)CC)=O)n2)CN(C)CCO1 c1(OC)ccc(NC(=O)C(C)(C2CCC2)NC(=O)CCCNC(C)=O)c(C)c1 N1(C(=O)Nc2cc(C)cc(Br)c2)CC2(CCCC2)OCC1C C(c1cccnc1)=C(C(=O)NCC1C(C(=O)NCC(=O)NCC)CC1)C C=C(C)CCC(C)NC(=O)CC1(N(C(=O)C(C)COCC)C)CC1 N1(C(c2n(C)ncc2)=O)CCN(C(C2CCCCN2C(=O)CCS(C)=O)=O)CC1 N1(CC(=O)N(CC(=O)Nc2cccc(C(C)=O)c2)C)CC2CC=CC1C2 C1(CNC(CCC=C)=O)(OC)CCN(C(=O)CCc2nc(CC(=O)OC)n[nH]2)CC1 CC(CC1CCCO1)C(=O)NCCn1cnc(C(=O)NCC2(O)CCOC2)c1 N1(C(CC)C(=O)Nc2ccccc2-c2cn[nH]c2)CCCCC1CNC(=O)OC c1(-c2c(C(=O)Nc3c(I)ccc(C#N)c3)ncnc2)cc2cc(Cl)ccc2[nH]1 C1(NC(COCC)=O)CCC2(CC1)CC2NC(=O)C=Cc1cscn1 C(=O)(C1CCc2ccccc21)NCC1(C(N2CCC3CCN(C)CC32)=O)CC1 N1(C(C=CC(=O)OCC)=O)CCN(C(C2CCC(C3CC3)O2)=O)CC1CO C12(NC(CC3CC(SC)C3)=O)CC1CN(C(=O)Cc1sc(O)nc1O)C2 c1(CC(=O)N(C2CCN(C(C(C)C)=O)C2)C)ccc(Br)cc1[N+](=O)[O-] c1(CS(C)=O)cccc(C(=O)NCCC2CCCN2C(C2CNC(=O)N2)=O)c1 C1(C(N2CCC(Br)C2)=O)CCc2nc(-c3ccc4n[nH]cc4c3)sc2C1 N1(C(=O)C(F)C2CC2)CC2CCC(C1)N2C(C1CCC(O)CC1)=O c1(C(N(C)CC2CCCN2C(C2CCOC2)=O)=O)ccc2ccnc(O)c2n1 c1(C(N2C(C(C)NC(C3CCSC3)=O)CCC2)=O)cc2ncccc2cc1Cl C1(NC(C(CCCC)C)=O)CN(C(=O)COCC(C)C)CC2CCCC12 c1(N2C(CCC(=O)NCc3cc(Br)ccn3)CCC2)ncnc2cc(Br)ccc12 c1(NCC(=C)Br)ccc(S(=O)(=O)NCC2(S(N)(=O)=O)CCC2)cc1F CC1=C(C(=O)N2C3CCCC2CC(NC(=O)C(O)CN(C)C)C3)CCC(C)(C)C1 c1(C(N2CC(C(C)NC(=O)CCC(=O)N(C)C)C2)=O)cc2cnccc2[nH]1 Cc1cnc(F)c(C(N2CCC(CNC(=O)CC3(C(F)(F)F)CC3)C2)=O)c1 c1(OCC)ccnc(N2CC(C(C)NC(C3(Cl)CC3)=O)C2)n1 C1(N(C)C(C2CC2C2CC2)=O)CN(C(C2CCCCC2)=O)CC1O CC1=C(C(=O)N2CCOCC2CCNC(=O)CSc2nccn2C)CCC1 C(=O)(C1=CSCS1)NC1C(CNC(C(C)Oc2ccc(F)cc2)=O)C1 C1(NC(C2C(OCC)C2)=O)COCCC1NC(=O)Cc1cc[nH]n1 c1(OC)cc(C(=O)NCC(C)NC(=O)CC2CC2)cc(N)c1OC N1(C(c2cnsc2)=O)CC2C3CCC(C2C1)N(C(C1(CNC(=O)NC2CC2)CC1)=O)C3 N1(C(CC2CCC(OC)CC2)=O)CC2CCCC(N(C)C(C3CCCS3)=O)C2C1 N1(C(c2c(C)oc(CO)c2)=O)CCC(C)(C)C(C(N2CC3(CCCCC3)C2)=O)C1 CC1=CC(C)CN(C(=O)NCC2CC(N3CCOCC3)C2)C1 c1(C(=O)NC(C(C)NC(c2nc(C)oc2)=O)C(C)C)cccc2nonc12 c1(C(N2CCN(CC(C)NC(c3n[nH]c(C)c3Cl)=O)CC2)=O)cc(N)nc(Cl)c1 C1(CN(C(C(C)NC(=O)NC)=O)C)CCCCN1C(=O)CC1(O)CCC1 N1(C(c2c(CC)cno2)=O)CCOCC(NC(=O)C=Cc2scnc2C)C1 C(N=c1ccnc(C2CC2)[nH]1)C1N(CC(=O)N(CC)CC)CCOC1 c1(C(N2CCCC(NC(c3n(CC)nc(C)c3)=O)C2)=O)cc2ccccc2o1 C1(CNC(Cn2c(C)csc2=O)=O)CCN(C(=O)Cc2cncs2)CC1C C(=O)(CC(C)CC(C)C)N(CCNC(c1cncc(C(N)=O)c1)=O)CC C1(CCNC(C=C(C)C(C)(C)C)=O)CCCCN1C(=O)C=CC1CCOC1 N1(C(CC=C)=O)CCC2(CCN(C(c3ncc(C(=O)OC)cc3Cl)=O)C2)C1 c1(C(N2CC3CC3(CNCc3n[nH]cc3Cl)C2)=O)cc(Br)c([N+](=O)[O-])s1 N1(C(c2nc(C)oc2)=O)CC(CNC(=O)COCc2ccnn2C)C2(CC2)C1 C(=O)(CCCC(=O)OC)N1CC(NC(CCSCCC)=O)C2C1C2 N1(CC(C)(C)NC(Cc2c(C)ncs2)=O)CCN(C(=O)C(C2CC2)C2CC2)CC1 N1(C(C2=NOC(C)C2C)=O)CC2(C1)C(NC(c1coc(Cl)c1)=O)CCS2(=O)=O n1(CC(N2CCCC(N(C3CCOC3)C(=O)COC)C2)=O)ccc(=O)cc1C C1(C(=O)NC2CC(C(N3CCC(N(C)OC)C3)=O)C2)(CC2CC2)CCCO1 C(C(=O)NCCC1CN(C(=O)Cc2cccc(C)c2)C1)(C(C)C)NC(COC)=O C1(C(N2C3CC(NC(Cc4nc(C)[nH]n4)=O)(C3)C2)=O)CCS(=O)(=O)C(C)C1 O=[N+]([O-])c1cc(CN=c2[nH]nc(-c3ccc4sc(O)nc4c3)o2)ccc1Cl C(C(=O)Nc1ccc(Cl)cc1F)(C1=CCCSC1)N(CCC)CC1CCOCC1 N1(C(CSc2n(C)nnn2)=O)CC(C2CN(C(c3cccc(N)n3)=O)C2)C1 C(=O)(CCS(=O)(=O)N(C)C)NC1CCCC(N(C2CCCN(C)C2)C(C)=O)C1 c1(C(=O)NC(CCNC(C(C)Cn2cccn2)=O)C)cc(Br)cnc1O O=C1Nc2c(C(N3CC4=C(C3)CN(C(C3CC3Cl)=O)C4)=O)cccc2C1=O c1(OCC)ccnc(N2CCN(C(=O)CCN3CCOCC3)CC2)n1 C(=O)(C(O)CC(F)(F)F)NCC1C(C(=O)NCC(CC=C)(F)F)CCCC1 C#Cc1ccc(C(=O)NCC(C)N(C)C(c2ccc(F)c(CO)c2)=O)cc1Cl c1(C(=O)OC(C)=O)ccc(S(=O)(=O)NC(c2ccc(Cl)cc2)C(N)=O)cc1 N1(C(CSCC(N)=O)=O)CCC(NC(c2ccoc2CC(N)=O)=O)C(C(N)=O)C1 c1(C(=O)NCCCN(C2CN(C(=O)N(C)C)C2)C)csc(S(N)(=O)=O)c1 c1(OC(C)C)nc(C(F)(F)F)ccc1CN1CCN(c2cnccn2)CC1 Cc1cnc(NC(c2ccnc(-c3ccccn3)n2)=O)c(Br)n1 C1(N(C(CCOC)=O)C)CCC2CN(C(c3cc4scnc4[nH]3)=O)CC12 C1(C)(CC)C=C(C(=O)N2CC(NC(=O)CC(C)(C)OC)CC2C)C1 Cc1ccc(C(N2CCCC(CCNC(C3(C(N)=O)CCC3)=O)C2)=O)nn1 Cc1noc(C)c1CC(N1CCC(CNC(=O)C(C2CCCCC2)C)C1)=O c1(C(N2C(C)(CNC(CC3C(C)(C)C3)=O)CCC2)=O)cc(S(C)(=O)=O)co1 Cc1cc(C=CC(N2CCC2(C)CC(=O)NC2CC2(C)C)=O)on1 C(=O)(C(C)CC(F)(F)F)N1CCC(CNC(C(CCC)(C)O)=O)CC1 C1(C(=O)OC)Cc2n[nH]cc2N(C(=O)C(c2ccc(Cl)cn2)(F)F)C1 C1(CC(N2CC3C(NC(=O)Cn4cnnc4O)C3C2)=O)CCC2(CCC2)O1 c1(C(C)NC(C2(c3ncco3)CC2)=O)ccc(NC(=O)NC2(C#N)CC2)cc1 CCCC(C)(CC)C(=O)N1CC(CCNC(=O)C(CSC)OC)(OC)C1 C(CC(C)(C)C)(C(=O)N1CCCC(N(C(=O)CCOCC(C)C)C)CC1)OC Cc1cc(C(N2CC3(C(=O)O)CC3(C)C2)=O)nc(C)c1 C(=O)(C1c2ccccc2C2CC1C2)N1C(CC)CN(C(=O)CC(C)SC)CC1 N1(C(C2C(C3CN(C(C4(C)CCOC4)=O)C3)C2)=O)CCc2nc(O)[nH]c2C1 CN(C)S(=O)(=O)N(C)CC(=O)NC1CN(C(=O)CCc2ccoc2)CC1O C=CCCC(C(=O)OC)NC(=O)CCN(CCO)C(c1cnc(O)n1CC)=O C1(NC)CCCC(NCCOc2ncccc2F)C1 N1(C(=O)OCC)CCC(C(=O)NC(Cc2cncn2C)C(=O)O)CC1 C(C)(CC(=O)N1CCC1CC(=O)N(CC(C)CO)C)=C(C)C c1(C(N(CCC(C)(C)NC(c2cc(CC)sn2)=O)C)=O)cc(C)nn1C1CC1 c1(Oc2cccc(OCC)c2)c[nH]c2cccc(-c3cnc(F)c(Br)c3)c12 C(CS(=O)(=O)NC)(C1CCC1)O.C(CC(C)C)(c1ccsc1)CC O=C(C1CCCn2cnnc21)NC1CC(NC(C2CCCCNC2=O)=O)C1 C12(NC(C(CC)O)=O)CC(CNC(c3cnc(S)[nH]3)=O)(C1)OC21CCC1 N1(C(N(CCNC(CN(C(=O)OC)C)=O)C)=O)CCCS1(=O)=O c1(C(=O)NC2C(CNC(C3(C(=O)NC)CC3)=O)C2)ccc2cc(OC)ccc2c1 C1(C2CC2)(C(=O)NCCC)CN(C(=O)CC(c2cnn(C)c2)N(C)C)C1 C1(C)(C(CC)NC=O)CCCN(Cc2cccc(-c3ccc(N)s3)c2)C1 CC1CCN(S(=O)(=O)CC(=O)N(CCCNC(C2CC3(C2)CC3F)=O)C)CC1 c1(OC)cccc2c1N(C(C1NCC13CCOCC3)=O)CC2 c1(N(C)C)ccc(F)c(C(N2CC(NC(=O)C(O)C(C)(C)C)C3CC23)=O)c1 c1(C(N2C(C)C(NC(=O)Cc3cnns3)CCC2)=O)cccc2oc(=N)[nH]c12 c1(CCC(=O)NC2CCCC2NC(C2CC2C(F)(F)F)=O)cnc(C2CC2)o1 c1(NC(C2CC(F)CN2Cc2cccc(-c3ccsc3)c2)=O)cc(Cl)ccn1 N(C)(C1CN(C(=O)CCCCSC)CCc2ccccc21)C(C1(CC#C)CC1)=O c12cccc(c1)S(=O)(=O)N2.c1(C(N(C)C)=O)cnc(O)c2cncn12 c1(CC)cc(C(N2C(CNC(c3cccnc3CC)=O)CC3CC23)=O)cc(O)n1 c1(C(=O)NCC2CCN(C(=O)C(F)C3CC3)C2)cnc2[nH]nnc2c1 c1(NC(C(N2CC(COC)OCC2)=O)=O)cc(C)ccc1C1CC1 C1(C(=O)NC(C2CCCO2)COC)CCN(C(c2cscc2Cl)=O)CC1 C(C1CCC(=O)c2ccccc21)N1CC(=O)CC12CCC2 c1(C(N(CCC)CCNC(c2ccnn2C2CCC2)=O)=O)cccc2c1OCC2 C(C(CO)(CO)NC(c1ocnc1C)=O)N(C(CC1(CSCC)CC1)=O)C c1(C(c2ccccc2)N(CC(C)C)CC(C)O)ccc(Br)c(C(F)(F)F)c1 N1(C(C2CCC(=O)NC2)=O)CC2(C1)CN(C(C1CCCCCC1)=O)CC2C(=O)O N1(C(C2(C)CN(S(c3c(C)n[nH]c3C)(=O)=O)C2)=O)CCCC2(C1)OCC1CC21 C1(NC(CC(CC)OC)=O)(CC)CCN(C(c2cnn(CC)n2)=O)CC1 CC(CC(C)NC(c1ccnn1-c1ccccc1)=O)NC(=O)CCC1CCOC1 C1(C(N2CCC(CCC(=O)NC3CCCC(SC)C3)C2)=O)CC2CC(=O)C1O2 C(N=c1[nH]c(=NCc2cc(Cl)cc3c2OCC3)[nH]c2c1SCC2)C1OCC(C)C1 C1(C(=O)NCC2N(C(CN(C(C)=O)C)=O)CC=C2)CCn2c(C)cnc2C1 N1(C(CC(CCC)C)=O)CC2CC(C1)CN(C(c1c(C)ncnc1C)=O)C2 c1(SC)c(C(=O)N(C2CC(NC(c3snc(Cl)c3Cl)=O)C2)C)cnn1C c1(C2(C(=O)NCC(CNC(C3(OC)CCC3)=O)(C)O)CC2)ccc2c(c1)OCCO2 C1(C)(N(C(C)=O)C2CC2)CCN(C(C)=O)CC1.C12(CCSCC1)C(=O)N2 Cc1cc(N(C(C)CCNC(c2ccc(F)cc2C)=O)C)nc(CO)n1 C(=O)(CCCCCC(C)O)NCCN(C(=O)C(=Cc1cccs1)C)CC c1(CC(=O)N(CCOCCNC(c2cc(C)[nH]c2C)=O)C)nsc2ccccc12 c1(C(=O)NC2(C)CCN(C(C3COC(C)(C)C3)=O)C2)ccc2c(c1)CCC2=O CC1CC(NC(=O)C(O)CC2CCOCC2)CN(C(c2ccnn(C)c2=O)=O)C1 c1(CC(=O)NC2CCC(NC(C3(C)C(C)C3)=O)CC2)cccc2ncccc12 C#Cc1ccc(C(=O)NC2CCN(Cc3cc(C(=O)NC)co3)C(C)C2)cc1 N1(C(CSCC#C)=O)CC2CC(C1)CN(C(=O)CCCCCC(C)C)C2 N1(C(c2cnc(CCCC)s2)=O)CC2(C1)CN(C(c1n[nH]cc1Br)=O)CC2CO n1(CC)cc([N+](=O)[O-])c(C(=O)NC2CCN(C(=O)C=C(C)C(C)(C)C)C(C)C2)n1 CC(C)C(C(=O)N1CCOC(C(C)NC(=O)C=CC=C(Cl)Cl)C1)C(C)C c1(C(=O)NN2CC(C(C)NC(C3(C(=O)NC4CC4)CC3)=O)C2)cc2ncccc2o1 Cc1cc(C(=O)NCCCCNC(C2(C)CNC(=O)C2)=O)cc2ccoc12 C(=O)(CCCC(C(=O)NCC1CCOCC1)N(C)CCOC)OC C1(CCNC(CC=C)=O)CCCN(C(C2CC(=O)N(C3CC3)C2)=O)C1 C#Cc1cccc(CC(=O)NC2COCCC2NC(c2n[nH]cc2C#C)=O)c1 C(=O)(C(C)(C(C)C)N(C)C)NCCNC(COCC)=O.C1(C)(C)CCCN1 C1(CCCC(=O)NCCOCCCNC(=O)CSC2CC2)CCCC(=O)N1 Cc1cnc2c(C(N3CC(NC(=O)CC4CCCC4)CC(O)C3)=O)cnn2c1 c1(OC)ccnc(CN2CCN(CCCNC(c3cncc(O)c3)=O)CC2)c1 C(=O)(C(CCOCCO)NC(C1(OC)CCCCC1)=O)N1CCC(C(=O)NC)C1 C12(CNC(CC(=O)OC)=O)CC(C1)C(Cn1cc(-c3nccc(C)n3)nn1)CO2 N1(C(Cc2c(C#N)cccc2)=O)CC2(CCC(CNC(c3nc[nH]n3)=O)O2)C1 CCC(C)CC(C)C(=O)NC12CCC(CN(C(=O)CNC(=O)CCC(C)C)C1)C2 C=C(C)C1OCCCC1C(=O)N(CC)CC1CN(C(=O)CCCN2CCCC2)C1 N1(C(c2c(C)ccnn2)=O)C2CC1CN(C(=O)C(N1CCOCC1)C)C2 Cc1c[nH]cc(C(=O)NC(CNC(c2cn(C)c(=O)n2C)=O)CO)c1=O N1(C(CCCc2cc(C)no2)=O)CCC2OCCN(C(c3csnc3C)=O)C2C1 Cc1cccc(C)c1OCC(N1CCC(NCCc2ccccc2Cl)C1)=O N1(C(CNC(=O)O)=O)CC(C)(C)CC1CCNC(=O)CNC(CC=C)=O.C1(OCC)CC1 N1(C(C2NC(=O)OC2)=O)CCC(C2CCN(C(c3snc(O)c3Cl)=O)CC2)C1 C1(CN)CC(C(F)(F)F)CCN1C(C12COCC(C1)C2)=O c1(C(=O)NCC(C)NC(=O)CC2(C)OCCO2)coc(Br)n1 N1(C(C2CCC(CC)O2)=O)CC2(CCN(C(c3ccc([N+](=O)[O-])[nH]3)=O)C2)C1 c1(C(=O)NC2(C)CC(NC(C3C(C)(C)C3(C)C)=O)C2)cc(Cl)ccc1C(F)F c1(C(N2CCC(N(C(=O)C(F)OC)CC)C2)=O)ccnc(C)c1C C(CC1=CCN(C(=O)C(c2ccc(Cl)cc2)O)CC1)NC(c1cnnc(O)c1)=O N1(C(CC(C)F)=O)CCOC2(C1)CN(C(C1CCCCN1S(C)(=O)=O)=O)C2 C(CCCC(CO)NC(c1cccc(OCCF)c1)=O)NC(CS(CC)=O)=O CC(C(=O)N1CC(CC(C)NC(=O)CCc2cnn[nH]2)C1)c1ccco1 C(C(C)C(=O)Nn1ccccc1=O)N(C(C(C(CC)CC)C)=O)C C1(C(=O)NCC(C)(C2CCC2)NC(C(C=C=C)C)=O)CCOC2(CCOCC2)C1 N1(C(=O)Cc2cc(O)nc(O)n2)CCN(C(C2CCCC(O)C2)=O)C(C2CC2)C1 Cc1cc2ncc(C(N3CCC4(CCN(C(C5COC(=O)N5)=O)C4)C3)=O)cn2n1 C1(n2cccn2)(C(=O)N(CC2N(C(CCCOCC)=O)CCC2)CC)CCOCC1 C12CC3(C1)CN(C3)C2.C1(C2C(CNC(Cn3c(C)nnn3)=O)C2)CCCOCC1 C(=O)(C1=CCCN(Cc2cnc(Br)s2)C1)NCC=C N1(C(c2cc(CC)on2)=O)CCN(C(C2CCN2CC)=O)CC1CC Cc1nc(C(C)C)nc(O)c1C(N1CCC(C)(NC(=O)C(O)CC(C)C)CC1)=O C1(CNC(C=CCC)=O)CC(NC(c2ccc(C(C)CC)cc2)=O)CCO1 C1(CNC(CN(C)CCc2ccccc2)=O)CN(C(=O)CC#N)C(C)(C)C1 C1(C(N(CC)CC2CCC2)=O)CC(C)(C)CCN1C(C1CCCCC1(C)C)=O C(=O)(C(O)CCNC(=O)CCNC(=O)OC)NC(CC)C CC1=C(C(=O)NC(C2CCCCC2)C(C)NC(=O)Cc2cncs2)CCO1 C1(CNC(=O)CC2CCC(=O)N2)CC2CN(C(c3cc4ccsc4s3)=O)CC12 c1(CC)conc1C(=O)NCC1CCCC1NC(C1(c2ncco2)CCC1)=O N1(C(Cc2nc(C)sc2)=O)C2CCCC1CN(C(C1CCCC(F)(F)CC1)=O)C2 C1(C(N2CCCC(N(C(c3ncn(C)n3)=O)CC)C2)=O)CCCCC(=O)N1 Cn1cc(C(=O)NC2CN(C(=O)C(=Cc3cccnc3)F)CC23CC3)ncc1=O c1(C(C(N2CC(NC(C3(CCO)CC3)=O)(CO)C2)=O)O)cccc(F)c1 S(=O)(=O)(c1c[nH]ccc1=NCCCn1ccnc1)NC(CCC)CO c1(CNC(C2(COC)CC2)=O)cncc(C(=O)NCC(O)(CO)CO)c1 C(=O)(C1=COCCO1)NC1CC(C(=O)NCc2ncc(CO)[nH]2)C1 N1(CCNC(C=C(C)C)=O)CCC(NC(=O)CCOC2CCCOC2)CC1 C1(C)(C(=O)NCc2occ(C(=O)NC(c3noc(C)n3)CC)c2)CC(C)(C)C1 N1(C(C2N(CC)CC2)=O)CCC(O)(CNC(=O)CC2CCCC(OCC)C2)CC1 c1(C(N(CC(CNC(Cc2ccc(CC)cc2)=O)O)C)=O)ccc2nn[nH]c2c1 c1(OC)cccc(OC)c1C(=O)NCC1CCC(NC(=O)C=C(Cl)Cl)CC1 O=C(CC1COc2ccccc21)NC1CN(C(c2nc3c(Br)cccc3s2)=O)C1 c1(C(N2C(CN(C(C(C)Sc3ccccn3)=O)C)CCC2)=O)ccc(F)c(N)c1 C1(NC(CC2(CNC(c3cc(C)n(C)n3)=O)CC2)=O)CCn2cnnc2C1 C1(C(=O)NCC2CC3(CC(NC(CC(C)(F)F)=O)C3)C2)CCC2C(C1)C2(F)F N1(C(CC(CC)CC)=O)CCC2(NC(c3ccc(SC)o3)=O)CCCC12 N1(C(CCSC)=O)CC(C(=O)NCCCC)C(C)(C)C1.C12CCN(C1)C2 C1(C(=O)NC2C=CCCCC2)CC2(CC2)CN1C(c1cc(O)cs1)=O C1(NC(c2ccc(O)cc2)=O)CC(C(=O)NC2CC3CCC2O3)C12CCC2 N1(C(c2c(OC)nc(-c3ccccc3)s2)=O)CC2CCC1C2N C(=O)(CCC(C)(F)F)N1CC(C(C(=O)N(C)Cc2cncnc2)O)C1 C=CCC(C)(C)C(=O)N1CCCC(C(C)C(=O)NC2(C)CCSC2)C1 c1(C(=O)NC2CCCN(C(C=NOC)=O)C2)cnc2c(Br)c(C)ccc2c1 C(N=c1[nH]c(=NCCOCC2CCOC2)[nH]c2cc[nH]c12)C1CCC(=C)CC1 C1(F)(CNC(C=CSC)=O)CCN(C(c2ccc(C)c(Br)c2)=O)CC1 C(CC(=O)NC(=O)C(CCSC)OC(C)(C)C)(C(F)F)CNC(CCOCC)=O c1(OC(C)C)nn(C)c(Cl)c1NC(N1CCOCC(C(=O)O)C1)=O N1(C(c2cc3ccccn3c2)C(=O)NCCCC)CC(C)OC(C)(C)C1C CCC(C)C(O)C(C)C(=O)NCC(C)(C)CCNC(c1cccc(O)c1F)=O Cc1nc(Cl)nc(N2CCC(N3CCN(C(C4CCCN4C)=O)CC3)CC2)c1Cl CC(Cn1ccnc1)C(=O)N(CCCOCCNC(=O)Cc1coc(Cl)n1)C c1(C(=O)NCC(CN(C)C(C2CNC(=O)N2C)=O)(C)C)ccccc1CC(F)(F)F c1(CC(N2CCN(C(C3C(CCC)C3)=O)C(CC)C2)=O)ccc2c(c1)CCN2C c1(N(CCC)CCNC(C2CCOC(C)C2)=O)nc(C)nc(=N)[nH]1 c1(OC)csc(C(N2CCN(C(C3(CO)CCOC3)=O)CC2)=O)c1OC C1(CNC(C(CC)SC)=O)CN(C(C2(CCF)CCOCC2)=O)CC(C)(C)O1 n1(CC)nc(C(=O)NC2(C(=O)N(C3CCCC3)C)CCCCC2)cc1O C1(NC(C(C)(C)SC)=O)CC2(C1)CC(CNC(C1C3CCCCCC13)=O)C2 N1(C(c2cnc(C(C)O)s2)=O)CC(N(C)C(C2(C(=O)NC3CC3)CC2)=O)C2(CC2)C1 c1(C(=O)NCCCC2N(C(C(COC)C)=O)CCC2)cccc2c1nc(O)n2C N1(C(C=Cc2c(C)ccs2)=O)CCN(C(=O)C(n2nccc2C)C)CC1CCO N1(C(Cc2c(C)cccc2)=O)CCN(C(=O)C(CO)c2ccccc2)C(C#N)C1 Cc1cncc(C)c1C(=O)NC1CCCC1NC(=O)CC(F)(F)F C1(C(C(=O)NCCSC(C)C)F)CCN(C(c2coc(C3CC3)n2)=O)C1 C=CC1(C(=O)NC2CN(C(=O)C(C)CC3CCCC3)CC2C)CCOCC1 CCCC(c1ccco1)NC(=O)CCN(C(=O)C(=O)NC(C)C)C(C)C C=C1CC(C)(C(N2CC(CC(C)(C)CNC(c3cn(CCOC)nn3)=O)C2)=O)C1 c1(C(N)=O)csc(C(N2CC(CNC(c3cn(-c4ccccc4)cn3)=O)C2)=O)c1 C1(NC(C(C)(C)CC2CC2)=O)CCOC12CCN(C(C1(C)CC3CC3C1)=O)CC2 C(=O)(CCN=c1ccc(C)c[nH]1)N1CC=C(CNC(C2(CC=C)CC2)=O)CC1 c1(NC(N2CCC(C(=O)Nc3ccccc3Cl)C2)=O)c(O)cccc1O c1(CCOC(COC(CC)C)=O)cnc(C)o1.C1(C)C(=O)N(CC(C)C)C1 C1(C)(CCC)CCCN(Cc2ccc(-c3ccc(C)c(N4CCOCC4)c3)s2)C1 CC1CN(C(c2cscc2C(F)(F)F)=O)CC1NC(=O)C(C)(C)c1cnn(C)c1 CC(CCC(F)(F)F)NC(=O)CCNC(C1CCCCC(=O)C1)=O Cc1ccc2[nH]c(C(=O)NCCC3CCN(C(c4cocn4)=O)CC3)cc2c1C N(C1CCCc2ccoc21)C(C1CCN(C(CC(COC)C)=O)C12CCC2)=O N1(CC)CCC(CNC(=O)C(c2ccoc2)NC(=O)CCNC(N)=O)C1 O=C(CC(F)(F)C(F)(F)F)NC1CN(C(C2CC2F)=O)C2(CCC2)C1 C(CCOCCO)(C(=O)NCC1CC(=C2CC2)C1)NC(CC(OC)OC)=O c1(CC(=O)NC2C(CCC)CN(C(=O)C(F)n3ccnc3)C2)ccc(F)c(C)c1 Cc1n[nH]c(C)c1CC(N1CC(N(C(=O)CCOCCOC(C)(C)C)C)C1)=O C(=O)(C(CN(C)C)C(C)C)N1CC(NC(C2CCN(CC)CC2)=O)(CO)C1 c1(C(=O)NCC(CCCC)NC(=O)CC(C)(C)C#N)c(OC(F)F)cccc1Cl C(=O)(CC(C)C(F)F)N1C(CNC(C=CCN(CC)CC)=O)(COC)CCC1 CCCC(C)(CC)C(=O)NCc1cc(C)c(C(=O)NCCCN(C)C)o1 C(=O)(CC(C)C(=O)OC)NC1(C(=O)NC(C(=O)OCC)C2CC2)CC1C C1(N(C(=O)C(O)C2CCCC2)C)CN(C(c2ccccc2Cl)=O)CC1O C1(C(=O)NCC(=O)NCC)CC12CCN(C(=O)Cn1cnc(C(F)(F)F)n1)C2 c1(OC)ccccc1C(C)C(=O)NCCCCCCNC(C1(C)CC(F)C1)=O n1(CC(=O)NCC=CCNC(COc2ccc(OC)cc2)=O)c(C)cc(C)nc1=O Cc1ccc(Cl)c(C(=O)N(C)CC2(NC(=O)C(c3ccc(Cl)cc3)CO)CC2)c1 N1(C(c2nc(C)nc(O)c2)=O)CCCCC12CC(NC(=O)C(O)CC1CC1)C2 C1(CC)C(NC(=O)CCc2ncccn2)CCCN1C(c1ccc(Cl)cn1)=O CCC(O)(CC)CCNC(=O)C(=O)Nc1nnc(-c2ccn(C)n2)s1 CC(C)(C(=O)NC1CC(CNC(c2ccc[nH]2)=O)C1)Oc1ccccc1 c1(C(N2CCN(C(C(CCC)CCC)=O)CC2C)=O)ccc2c(C#N)c[nH]c2c1 C1(C)(C(=O)NCC(C2CCN(C(=O)CCCCN(C)C)CC2)C)CCC12CCC2 CC1CCC(O)(C(=O)NCC2CCN2C(C2CCC(C)(C)C2)=O)CC1 C(N=c1cc(C)[nH]c(=NCC2COCC(C)O2)[nH]1)c1n(CC)c(O)nn1 c1(C(=O)NCC2(O)CN(C(C3(C#C)CC3)=O)C2)[nH]nc2ncc(Br)cc12 N1(C(CCCSC)=O)CCC(C(F)(F)F)C(NC(c2cc(C(N)=O)no2)=O)C1 C1(C(=O)NC2CC(NC(c3cc(N)c(Cl)nc3)=O)C2)CC(c2ccccn2)=NO1 N1(C(C(CC)C)=O)CCN(C(c2cc(C)sc2C)=O)CC(C)(F)C1 c1(C(C)NC(C(C)OCCOC)=O)nc(C(=O)NCc2cncn2C2CC2)co1 c1(C2(CNC(=O)NCCC3C(C)OCC3)CC2)cccc(C(F)(F)F)c1 C(CC(=O)N=c1[nH]ccnc1Cl)(c1ccc(Cl)cc1)NC(C)=O N1(CCCNC(CC(C)NC(N)=O)=O)Cc2ccccc2C1 C(=O)(C1=CCN(C(=O)C2=NOC(C)C2C)CC1)NC(C1CCOC1)C#C N1(C(CNC(CN(C)C)=O)=O)CCC(CO)(NC(c2n[nH]c(C3CC3)n2)=O)C1 c1(OC)cc(F)c(CC(=O)Nc2ccc(OC)c(F)c2)cc1F c1(CN2CC(C)(CC(=O)Nc3cc(C)no3)C2)cnc(C(C)C)nc1 N1(C(C)=O)CCCCC(CNC(=O)Cn2c(-c3ccccc3)c(C)sc2=O)C1 C1(CC)CCN(C(=O)CCCNC(CN(C(=O)CSC(F)F)C)=O)CC1 c1(C(N(CCCNC(C2CC2(Cl)Cl)=O)C)=O)cnn(-c2ccccc2)c(=O)c1 C1(O)(CNC(CCSCC)=O)CCCN(C(c2cncn(C)c2=O)=O)C1 CC(C)(C(=O)NNC(=O)Cc1cccc(C#N)c1)S(C)(=O)=O C1(NC(C(C)=C2CCC2)=O)CCC2(CC1)CCN(C(=O)C(C)NC(=O)C1CC1)C2 C1(CNC(c2nn(CCOC)nc2C)=O)CC(N=c2[nH]c(Cl)nc3c2SCC3)C1 C(=O)(C(CCc1ccccc1)N(C1CCN(C2CC2)CC1)C)NC.NC O(NC(=O)C1=CC2(CCN(C(=O)CC(Cl)Cl)C2)C1)CC(C(C)C)O C(CNC(c1cc(O)nn1C)=O)(CC(F)(F)F)NC(CC(CC)C1CC1)=O C1(CCC)(NC(C2CC(C)(C)CO2)=O)CCN(C(=O)C(F)C2CCC2)CC1 Cc1cc(C(=O)NC2CCN(C(=O)COCC(C)(C)C)C2C)nc(C)c1 N1(C(C(C)=C2CCCC2)=O)CC2CCC1CN(C(=O)CN1CCCNS1(=O)=O)C2 c1(C(C)NC(=O)NC2(C3CC3)CCC2)cc2cc(Br)ccc2[nH]1 c1(NCCN(C)C)cncc(NC(C2CCCC2c2ccccc2)=O)c1 N1(c2ncc(OC)c(C)n2)CCC2(CCCN2C(c2ncc(Br)cc2C)=O)CC1 C1(C(=O)NC(C2N(C(CNC(=O)NC)=O)CCC2)C)CCn2ncnc2C1 CC(C)C(F)(CNC(=O)CN1CCN(C)CC1)C(=O)N1CCC1CO C1(O)(CNC(c2sc(C)c(O)n2)=O)CC2CCC(C1)N2C(C1CCC(F)(F)C1)=O CCCCCOCCC(=O)NCC(CO)NC(=O)C(=O)NCC1CC1 c1(CC(=O)NCC2CN(C(CC(CC)OC)=O)C2)cc(Cl)c2c(c1)OCCO2 c1(NC)ccc(F)cc1C(=O)NCC=CCNC(C1(C(O)C(F)(F)F)CCC1)=O c1(NC(CCC2N(C(CCCSC)=O)CC2)=O)cccc(OCF)c1 N1(C(C)=O)CCCC1C1CCCN1C(=O)Nc1cccc2cc(Cl)ccc12 C1(C)(C(=O)NCCN(C(=O)COCC2CCCCO2)CC)CCN(C)C1 C12(CNC(C3ON=C(CC)C3)=O)CCCC1N(C(=O)C(C)C(C)C)CCC2 C1(CNC(C(C)(C)c2cc[nH]n2)=O)CC2CC2N1C(C1CCC(F)CC1)=O c1(C(C)C)nc(N(C)Cc2csc(C3CC3)n2)cc(N2CCC(Cl)=C(Cl)C2)n1 C(=O)(C(CC(C)C)C(C)C)NC1(CC)CCCN(C(c2cn(C)nn2)=O)C1 c1(OC)ccnc(C(=O)NCCC2CC(NC(C3(C)CC3(Cl)Cl)=O)C2)c1N C#Cc1ccnc(C(=O)NC2CC3(NC(=O)CCC4CCCCO4)COC2C3)c1 N1(CCNC(C(C)OCC#C)=O)CCN(C(C2(c3ccno3)CCC2)=O)CC1 N1(C(CC2(C)CCC2)=O)CCC2(CCN(C(C3CCn4c(O)nnc4C3)=O)C2)C1 CCCC(C(O)C(=O)NCc1cccc(C)c1)NC(=O)CCCOC(C)C N1(CC)CCN(C(=O)CC2CCC(NC(c3cc(C)ncc3Cl)=O)CC2)C(C)C1 c1(C(N(C2CN(C(Cc3cn(CC)nc3)=O)CC2F)C)=O)cc(C)c(C)nn1 c1(C(N(C2CCOC2)CC)=O)ccn(CCNC(=O)CCC2CCCC2)c1 C(C)(C(=O)N(CCNC(C1(C(=O)N)CCC1)=O)C1CC1)OC.C1(C(=O)OC)(CO)CC1 c1(N2CCCN(C)CC(C)C2)cccc(S(=O)(=O)N2CC3CCOCC3C2)n1 CC12CN(C(c3sccc3F)=O)CC1(C)CN(C(=O)C1CCCn3nccc31)C2 Cc1nc2cc(C(=O)NC3CCC3NC(c3c[nH]nc3C(F)F)=O)c(F)cc2[nH]1 Cn1ccc2c(C(=O)NC3CN(C(=O)CC(C)(C)C)C4CC34)ncnc12 CC1(C)CC(C(=O)NC2CC(=C3CC3)C2)CN(C(C2(F)CCCC2)=O)C1 N1(C(c2cc(C)c(Br)o2)=O)CCCC(CNC(C2(C)CCCO2)=O)CC1 C(C(C(=O)N(C(C)C(C)C)C)NC(=O)C(C)=CC)OCC c1(N2CC3CN(C(c4sc(Br)cc4Br)=O)CC32)ncc2sccc2n1 c1(C(N2C(COC)CN(C(C3CC3C(F)F)=O)CC2)=O)c[nH]c(C)c(Cl)c1=O N1(C(c2cnn(C)c2F)=O)CCC(NC(=O)Cc2ccc(F)cc2F)CC(O)C1 N1(C(C(COC(C)C)NC(C)=O)=O)CC2(CC2)CC1NC(C1CC2(CCC2)C1)=O N1(C(C(C)C(F)F)=O)CCC(C(=O)NCc2c(F)cccc2F)CC1(C)C C(C(CCC)CC(C)C)NC(C(COCCC)NC)=O C(CC(O)C(=O)N1C(C(=O)NCC2CCNC(=O)C2)CCC1C)N(C)C c1(OC)c(CNC2CC2C(=O)Nc2ccc(Br)c(Cl)c2)cccc1F N1(C(C=CC)=O)CC(C(C)(C)O)(CNC(c2ccn(-c3ccccc3)n2)=O)C1 c1(CN2C(C(=O)Nc3cc(OC)ncn3)CC2)ccc(F)c(F)c1Br N1(C(C(C)Cc2cnco2)=O)CC2(CCCN(C(=O)CN(C)C3CC3)C2)C1 CN1CCC(C)(C(N2CCC(CNC(c3nncn3C3CC3)=O)C(O)C2)=O)C1=O C1(NC(C(C#C)(C)C)=O)CN(C(=O)C(c2cccc(C)c2)(C)C)CCC1CO Cc1nc(CNC(c2cccc(Cl)c2Cl)c2nnnn2CCC2CC2)cc(O)n1 c1(C(=O)OC)c[nH]c(=NCC2CCCC2NC(c2nnccc2C)=O)cc1C N1(C(C2CCCC(=O)CC2)=O)CCC(F)(F)C(CNC(c2cnncc2O)=O)C1 C1(NC(=O)Cc2cnns2)COCCN(C(=O)CCc2cc(Cl)cs2)C1 N1(C(=O)CCn2cccn2)CCC2CCC(C1)N2C(=O)C=CCOC1CCOCC1 C(=O)(C(O)CCCNC(=O)CCc1ccsc1)NC1C(CC)CCCC1 N1(C(c2c(CC)cco2)=O)CCCCC1CCC(=O)NCC(Cl)Cl C1(C(=O)NC2(C)CN(C(=O)Cc3cc(F)c(F)cc3F)C2)COC2CCCCC12 Cc1ccc(C(=O)NC2CC(NC(C3CCCC3(F)F)=O)C2)c(C)c1 C=CCC(F)(F)C(=O)NCCC(CC)(CC)NC(C1CC(CF)C1)=O c1(C(=O)NCC2C=CCN2C(=O)CCc2ccc(Cl)nc2)cc2c(s1)CCC2 C12(NC(CCCOCC)=O)CCN(C(c3conc3CC)=O)CC1C2 n1(CCOC)c(O)nc2ccc(C(=O)NC3CCCCC3(C)C)cc12 C=C(C)C(CC(=O)NC1CCC(C)N(C(C2CNC(=O)N2)=O)C1)OCC N1(C(Cc2cnc(C)[nH]2)=O)CC2(CC2)CC1CNC(C1(c2cccnc2)CC1)=O C1(NC(C(C)C(F)F)=O)CC(C2CCN(C(c3c[nH]nc3C3CC3)=O)CC2)C1 N1(C(c2c(CC)nc(C)[nH]2)=O)CCN(C(=O)C(C)Cn2ccc(C)n2)C(C)C1 c1(C(N2C(CCNC(C(C)SC)=O)CCC2)=O)cc(F)ncc1Br CC1CC(C)CN(C(c2ccc(N(C)C(c3cnn(C)c3Cl)=O)cc2)=O)C1 c1(C(=O)OC)ccc(-n2ccc(C(=O)OC)n2)cc1.c12cc[nH]c1CNC2=O C1(NC(C=Cc2ccc(CC)o2)=O)CCN(C(=O)C(F)(F)COC)CC1(C)C N1(C(c2c(C)ccnc2)=O)CC(NC(=O)C(C)N2CCC2)C2(CCOCC2)C1 CCC(CC(F)(F)F)C(=O)NC1CC(NC(c2cc3nc(=O)ccn3[nH]2)=O)C1 CCCCC(=O)C(=O)NCC(CNC(=O)COc1ccc(F)c(Cl)c1)CO N1(C(c2c(C)ccnc2F)=O)CC2(CCC(C(N3CC(O)CC3C(N)=O)=O)O2)C1 N1(C(C(C(CC)C)OC)=O)CCN(C(c2nc(O)c(C)s2)=O)CCC1C CCC(CC(=O)N(c1ccccc1F)CC)NC(=O)C(C)(C)OCC N1(C(C2(F)C(C)C2)=O)CCCC2(CCN(C(=O)CC(C)(C)CC(F)F)C2)C1 C1(NC(C=CCCC)=O)CCC(C)(CNC(c2cc(C)oc2C)=O)CC1 c1(C(=O)NCC2(F)CN(C(C(C)=CC3CC3)=O)C2)ccc2sc(C)nc2c1 C1(C(=O)NC2CCC3CC23)(COC)CCN(C(c2c[nH]nc2C2CC2)=O)C1 n1(CC(=O)NCC2N(C(CCOCCN(C)C)=O)CCOC2)cc(F)ccc1=O S(=O)(=O)(c1cccnc1)NC1(C#N)CCC(NCc2c(Cl)cc(Cl)nc2Cl)C1 Cc1cn2cc(C(N3CCN(C(=O)CCCC4CCC4)C(C4CC4)C3)=O)sc2n1 C12(C(N3CC(N(C)C(C4CC(CF)C4)=O)C3)=O)CC3CC(F)(C1)CC(F)(C3)C2 C(CCCCC(=O)N1CC(OC(=N)O)C1)NC(c1ccc(C)n1C)=O Cn1nc(C(=O)N(CCNC(C2CC23CC3(F)F)=O)C2CC2)c(Cl)c1Cl C(CO)(C(F)(F)F)NC(CC1CCC(NC(C(C)NC(=O)C2CC2)=O)C1)=O C=CCCCC(C)(C)NC(=O)CCOC1CN(C(C2CCC(=O)O2)=O)C1 N1(c2ccnc(C(C)C)n2)CCC2(CC(NC(=O)CC(C)c3ccncc3)C2)C1 N1(C(C=CC(CC)=CC)=O)CCOCC1CNC(=O)CCc1cc(C)no1 C(=O)(CC1OCc2cc(F)ccc21)Nc1nn2c(=O)cc(C)[nH]c2c1 N1(C(c2cccc(C)c2)=O)CC2(C1)CN(C(=O)CC1CC1C)CCO2 C1(C(=O)NCC2(OC)CCN(C(C3CCC3)=O)CC2)SC2=C1C(=O)CCC2 c1(NC(CC)=O)cncc(C(=O)NCC(CCOC)NC(C2C3COCC23)=O)c1 N1(C(c2c(C)n(C)nc2)=O)CC(CO)C2(CCN(C(=O)CC3=CCCC3)CC2)C1 c1(C(N2CCC(C)(OCC)CC2)C(=O)NC)ccc(C#N)cn1 CCC(C(=O)N1CC(F)(C(=O)NCc2ccc(OC)nc2)C1)C(F)(F)F C(C1c2ccccc2CCN1C(=O)CO)NC(c1ncc(CC)s1)=O C12CN(CC1OCC)C(=O)C1CCN1Sc1cn2nn1.C12(COC)CCCC1C2 c12ccc(c(F)c1)Nc1cnc(s1)C(C)N(CC)C2=O.c1(NC(=O)OC)ccco1 c1(C(C(=O)OC(c2onc(CCC)n2)C)C)cccc(Br)c1 N1(C(c2[nH]c(=N)sc2)=O)CC2(C1)CN(C(=O)CCOCC1CCCO1)C2 C1(N2Cc3noc(n3)C2)C(=O)OCC1(C)C.c1(COC)ccccc1 Cn1nnc2cc(C(=O)NC3CCN(C(C4C5CCC45)=O)CC3)cnc12 CCC(CC)C(C)C(=O)NCC1CCC(C(N2CCS(=O)CC2C)=O)O1 N1(C(C(CC)SC)=O)CC(NC(c2cc(Cl)c(Br)[nH]2)=O)C(C)C1 c1(C(N(C2CCN(C(C3CCCC3O)=O)C2)CC)=O)sc2cncn2c1C c1(CNC(CCCOCCC)=O)nc2c(s1)CCN(C(c1cncnc1)=O)C2 C1(C(N2CC(C(N(CC#C)CC3CCCO3)=O)(SC)C2)=O)CC1C1(C)COC1 c1(N(C2CC2)CC2N(C(=O)OC(C)(C)C)CCC2)cc2sccc2s1 c1(N2CCC(OC)C(C)(C)C2)nc2c(c(=NCC(C)(C)N3CC=CC3)[nH]1)COC2 c1(C(C(=O)NC(C(=O)OC)C)N(C)Cc2cccs2)n[nH]c(C2CC2)n1 N1(C(C=CCOCCOC)=O)CCCCC1CC(=O)NCCCCC1CCCC1 N12CCS(=O)(=O)C(C1)Cc1cn(nn1)CCC2=O.N1(CCC)C(=O)CCC1=O CC(CNC(=O)C=CCN(C(=O)C(C)n1cncn1)C)CO c1(C(=O)NC(C)(CNC(=O)C(F)C2CC2)CO)cc(F)ccc1F C1(C(N(C(C)C2CC2)C2CC2)=O)CCN(C(C2C=CC=CC=C2)=O)C(C)(C)C1 CCCCCC(F)C(=O)NC1CC(CNC(=O)CCn2ccccc2=O)CC1O N1(C(C(CSC)C)=O)CCCC(CCNC(=O)C(F)CC2CCOC2)CC1 c1(NC(C2CSCCN2C(c2cccc(O)c2)=O)=O)ccc2nn[nH]c2c1 C=CCC(C)(C(=O)NCC1CC(C)N(C(c2nn(C)c(Cl)c2Cl)=O)C1)N(C)C C12(NC(C(CCOC)OC)=O)CC(CNC(c3c(F)cccc3F)=O)(C1)OC2C c1(CNC(CCc2onc(C)n2)=O)ccc(CN(C(=O)C(O)C2CCC2)C)cc1 c1(CC)ccc(C(C)C(=O)NC2C=CC(CNC(c3ccccc3)=O)C2)cc1 c1(OCC)ccnc2sc(C(=O)NC3CN(C(=O)C(CSC)OC)CCO3)cc12 c1(SC)nc2ncnc(N3CCCC(CNC(c4nccnc4Cl)=O)C3)c2s1 Cc1cc(N)cnc1C(=O)NCC1CCN(C(C2CCOC2C)=O)CC1O c1(CNC(C2N(C(C=C=C(C)C)=O)CCSC2)=O)ccc(C)cc1F CC1CCC2(CC1)CCN(Cc1ccc(-n3ccnc3)nc1)C2 N1(C(CCCCSC)=O)CCCC(NC(=O)Cc2ccc(F)cn2)C(F)C1 CCC1=NOC(C(=O)NC2CCC2NC(=O)CN2CC(=O)NC2=O)C1 CC1CC(NC(=O)CCc2nccn2C)CCN1C(=O)Cc1csc(C(C)C)n1 CC1(C)CC(CC(=O)NC2(CO)CCN(C(c3c[nH]ccc3=N)=O)CC2)CCO1 Cc1ncc([N+](=O)[O-])n1CC(=O)NCC(C1CCOC1)NC(=O)CCCN=[N+]=[N-] c1(C(=O)NCC2CN(C(C3CC(C)N(C)CC3)=O)C2)c[nH]c(=O)c2ccncc12 c1(NC(C2N(C(CCOC)=O)CCC2)=O)c(Cl)cccc1Br CC1CN(C(=O)C(C)(C)c2cscn2)CC1CCNC(=O)CC1CCCN(C)C1 CC(C)CC(C)CC(=O)NC(C(=O)NCC(F)CO)c1cccs1 C1(NC(CCNC(N)=O)=O)CCCN(C(c2cc(Cl)ccc2N)=O)CC1 C#CCC(C)C(=O)N1CCCC1(CO)CNC(=O)Cc1cc(C2CC2)on1 c1(CC(=O)NC(CNC(CN(C)C)=O)(C)Cn2cccn2)cn2ccsc2n1 N1(C(CCNS(CC)(=O)=O)=O)CC(C)(CNC(=O)Cc2ccno2)CC1(C)C c1(C(=O)NC(CCC(N2CCC(CC)(CO)CC2)=O)(C)C)cncc2[nH]ccc12 C12CCC3(CN(C3)C1=O)O2.c1(C(N)=O)cnc(NC(c2ccncc2Cl)=O)cn1 N1(C(CC(C(=O)OC)C)=O)CCC2(C(N3CCCC(C)(F)CC3)=O)CCCC12 C1(NC(CN(C2CCSC2)C)=O)CN(C(=O)C2=COCCC2)CCC1CO c1(C(N2C(CCCNC(C3N(CC)CC3)=O)CCCC2)=O)cccc(N)c1O c1(C(=O)NC2CC3CN(C(CCOCCN(C)C)=O)CC32)ccnc2[nH]cnc12 N1(C(CCSC)=O)CCOC2(CCC(NC(c3cc(O)c(Br)c(O)c3)=O)CC2)C1 CN1CCCC(CC(N2CCC(NC(C3CC(C(F)(F)F)C3)=O)CC2)=O)C1 C(C(C)(O)CC(=O)N1CCN(CC(=O)NC2CCC(N(C)C)CC2)CC1)OC C(=O)(C(CCF)NC(=O)C(C)NC=O)NC(CC=C)(C)C N1(c2nccc(NC3CC(COC)C3)n2)CCOC2(CCCCC2)C1 C(=O)(C1=NOC2CN(C(=O)CC(C)(F)C(F)(F)F)CC12)OCC c1(C(N2CC3C(NC(CS(CCC)(=O)=O)=O)(C3)C2)=O)cncc(S(C)(=O)=O)c1 c1(OC)cc(C)c(Cl)cc1C(=O)NC1CC(NC(c2ccn(C)c2)=O)C12CCC2 N1(C(CNC(C(CC)C)=O)=O)CC2CCCC(CNC(=O)Cc3cn[nH]c3)(C2)C1 N1(C(C)=O)CC(N(C(=O)COc2ccsc2Cl)C)C(O)C1 N1(C(Cc2n(C)ncc2)=O)CC2(CCN(C(=O)C=Cc3ccncc3)C2)C1 C#CC1(C23C(c4cccc(C(=O)OC)c4)CC(CC2)C3)CCOCC1 N1(NC(=O)OC)CCC(O)(N(C(=O)CCCOC)CC)CC1.C(=O)C1CC1 c1(C(N2C(C)CC(CNC(C(C(CC)C)OC)=O)C2)=O)cc(F)cc2nn[nH]c12 CC1OCCC1CNC(C1(NC(=O)CC2CSC2)CSC1)=O c1(C(=O)NCC(CC(C)C)NC(c2n(CC)nnc2C)=O)cnc(C)nc1C CC(CC(=O)NCC1CCOC1C(=O)N(C1CCCC(C)(C)C1)C1CC1)CC(C)(C)C c1(OC)cc(C)c(Cl)cc1C(=O)NCC1CCN1C(=O)C(C)(C)NC(C)=O N1(C(c2c(OC)cc(=O)n(C)c2)=O)CC2CC3CC2C1C3NC(=O)C=C(C)Cl Cc1cc(C(=O)NCC2CCC(NC(c3ocnc3C)=O)CC2)cc([N+](=O)[O-])c1 c1(C(N(C2C3CN(C(CC(C=C)C)=O)CC32)C)=O)cccc(=S)n1O C1(C(N2CCC(N(C(c3ccn(CC)n3)=O)CCO)C2)=O)CC2(C1)CC(F)C2 C1(C(N(CCCCCC)CCNC(=O)CSC)=O)CCc2n[nH]cc2C1C Cc1cc(C(N2CC3(C2)CN(C(C2(C)CC2Br)=O)C3)=O)cc(N)c1O N1(CC)CCCCC1C(=O)N(C(C)C(=O)N(CC(C1CCCC1)O)C)C N1(C(CSC)=O)CCN(c2ccc(C(N3CCCC(O)C3)=O)cn2)CC1 N1(C(C2(OCC)CCC2)=O)CC(NC(=O)C=CC(C)C)C2(CCC2)C1 C1(C(=O)NC(CC=C)CC=C)COCCN(C(=O)C(C)(C)C2(O)CCC2)C1 NS(=O)(=O)c1cc(C(=O)NC2CN(C(C3CCCO3)=O)CCC2CO)cs1 c1(C=O)cccc(C#N)c1.CC1(OCC=O)CN(N2CCC(CCO)C2)C1 N1(C(C(C(C)(C)C)O)=O)CCC(F)(F)C(NC(c2cc(F)cc(F)c2Cl)=O)C1 c1(C(=O)NCC2CC2NC(C23CCCC2C3)=O)cc(F)cc([N+](=O)[O-])c1Br Cc1ccccc1C(O)CC(=O)N(CCS(=O)(=O)CC)C C1(C)(SC2(C(N(C)CCOCCO)=O)CC2)CCCC1 Cc1snc2sc(C(N3CCCCC3C(N3CC4COCC4C3)=O)=O)cc12 C1(NC(CCCCCOCC)=O)CCN(C(=O)C(C)S(C)(=O)=O)C12CCC2 C(CC(C)(C)C(=O)N1CCC(O)(CCNC(=O)C(C)NC=O)CC1)OC N1(C(c2c(CC)n(CC)nc2)=O)C2CCC1CC(CNC(=O)C(C)SC)C2 c1(CNC(C(C)NC(COC)=O)=O)nc2c(s1)CN(C(C1CCC(=O)O1)=O)CC2 CCC(=O)CCC(=O)NCC1CCCCC1C(=O)NCCOCC(C)(C)C c1(C(=O)NC(CCCC)CN(C(=O)CC2CC=CCN2C)CC)c(C)cccc1Cl c1(C(=O)NC2C(C(=O)NC3CCN(C(C)=O)C3)C2)ccc(OC(C)C)c(F)c1 C(=O)(C(F)C(C)(F)F)N1CCN(CC(=O)NCCC=C(C)C)CC1 C(CC(N)=O)(C(=O)NCCCc1nc[nH]n1)NC(C1C(CC)CCO1)=O C1(NC(C2CCN(C)CC2)=O)CCCCCC1NC(=O)Cn1cnc(C(N)=O)n1 C1(NC(C(F)OC)=O)CCN(C(=O)CNC(=O)CC2CCCC2)C12CCC2 N1(C(c2cnn(C(C)C)c2F)=O)CCC(CNC(c2ccncn2)=O)C12CC2 c1(NC(C(COCC)NC(C(CC)NC(N)=O)=O)=O)cc(C)ccc1C C1(NC(C(C)C#N)=O)CCN(C(c2ccnn2CC(F)F)=O)C(C)C1 C(=O)(N=c1ccn(CCF)[nH]1)C(N1C2CC(NC(COC(CC)C)=O)C1CC2)=O C=CCC(C)(C)C(=O)N(CC(=O)NCC(C)(C)C(F)(F)F)C CC1CN(C(=O)CSCc2ccccc2Cl)CC1(C)CNC(c1ccco1)=O C1(N=c2[nH]nc(C3CC3)o2)(CNC(C(CC)CC)=O)CCCCC1 C#CC1(C(=O)NC(C2CCOC2)C#C)CCN(C(c2ccc(C)cc2)=O)CC1 C1(NC(CCC#C)=O)C2CC3CN(C(C4CCC5(CCCC5)CC4)=O)C1C3C2 c1(C(=O)NCC(CN(C(C(C)SCC)=O)C)O)ncc(Br)cc1C N1(C(COCC=C)=O)CCC(C2CCN(C(c3cnc(C)nc3C)=O)C2)C1 c1(C(=O)OC)ncc(C(=O)NC2CC2NC(C2CC2C2CCCO2)=O)s1 N1(C(=O)OC(C)(C)C)CCC1C#CC(=O)NCc1cnc2n1CCC2 C1(CC(N2CCC(F)(CNC(=O)CCOCC(F)F)C2)=O)CN2CCN1CC2 C1(NC(CC(=O)NCC#C)=O)CCC(CN(C(=O)CC2CCC(=O)NC2)C)CC1 c1(C(C)NC(C2CC(CNC(=O)CCN3CCCC3)C2)=O)ccc(F)cc1F N1(CC2CN(C(C(C)OCC(C)C)=O)C2)CCN(C(=O)Cc2cn[nH]c2)CC1 c1(C(N2CCOCC(NC(c3nn(CC)nc3C)=O)C2)=O)cccc2c1OCC2 c1(CC)n[nH]c(=NCc2ccc(CN(C(=O)CCCC3CCC3)CC)c(F)c2)o1 C1(NC(C2CCN(C)CC2)=O)CN(C(=O)C=CS(C)=O)C2(CCCCCC2)C1 Cc1cc(C(=O)NC(CC2CCCC2)C(=O)N2CC=CC2CF)c[nH]c1=N c1(NC(C2CSCCN2C(=O)CCc2ccc(O)cc2)=O)ccc2ncoc2c1 Cc1cc(C(N2CC(c3ocnc3CNC(=O)C(C)(C)F)C2)=O)n(C)n1 C1(CC(=O)N(C)CCOC2CCN(C(c3cccnn3)=O)C2)CC2(CC2)C1 C1(NC(CN(C2(CO)CC3CCC2C3)C)=O)CC(F)(F)C1(C)C c1(C(=O)NC2CN(C(C(CSC)C)=O)CC2O)ccc(S(=O)(=O)N2CCCC2)o1 C(=O)(C(C#N)=CCl)N1CC(C(C)NC(=O)CCCNC(N)=O)C1 C(=O)(C(O)C(C)(O)CC)O.C(CNC(C)=O)(C(C)(C)C)NC(C(C)(C)OC(C)=O)=O c1(C(N2CCCN(C(=O)COCC3CCC3)CC2)=O)cccc2c1NCCC2 C1(CNC(C(CC)C)=O)CC12CCN(C(c1sc(Cl)cc1Cl)=O)CC2 C(=O)(N=c1nc2n([nH]1)CC(C(F)(F)F)CC2)NC.C(CCC(C)NC=O)N(CC)CC C1(C(=O)NCCN(C(C2(C)CCCC2)=O)CC)CC12CCOc1ccc(Cl)cc12 N1(C(c2c(CC)nc(C)[nH]2)=O)CC(C)CN(C(=O)COC2CCCC2)C(C)C1 N1(C(C(COCC)C)=O)CCN(C(c2cnc(CC)s2)=O)CC1CF C1(CCNC(C(CCSC)O)=O)CCCN(C(c2cc[nH]n2)=O)CC1 c12cccc(c1)NC(=O)C2(F)F.CS(=O)(=O)CC1(C(=O)OC(C)(C)C)CC1 Cc1cc(CNC(C2CSCCN2C(c2cc3ncsc3[nH]2)=O)=O)ccc1Br C(CCCCC(=O)N1CCCC(NC(c2ccccc2C(F)(F)F)=O)C1C)OC C(=O)(C1=NOC2(CCC2)C1)N1CC(NC(=O)CCc2cc(Cl)no2)C(O)C1 CCCCC(CC)CCC(=O)N(C1CCC(NC(=O)C(C)(CC)OC)CC1)C C1(NC(=O)CCF)CCN(C(C2(N3CCCCC3)CCCCC2)=O)CC1F N1(C(COCCOCC#C)=O)CCCC(NC(C2CCN(C)C2=O)=O)C1C CC(C)C1=NOC(C(N2CCC3(CC3C(=O)NC(C)(C)CCF)C2)=O)C1 c1(-c2cn(CC(=O)NCCOCC(=O)O)nn2)cc(F)c(F)cc1F C1(NC(=O)Cn2cncn2)CN(C(C23CCCC(CO2)C3)=O)CC12CC2 c1(C(N2C(CNC(c3cnn(CC)n3)=O)CC2)=O)cc(OC)ccn1 C#CCC(C(=O)N(CCC(C)NC(C1CC(N(C)C)C1)=O)C)C1CC1 C1(C(N(CCCN(C(C(c2ccc(C)o2)C)=O)C)C)=O)NC(=O)OC1C S(=O)(=O)(CC(=O)NCC(C(C)(C)C)NC(=O)CC1CCCCN1C)NC C(C(=O)N1CCC(C(=O)NC2(C(F)F)CCC2)O1)C(NC(CC1(C#C)COC1)=O)(C#N)Br.C1CC1.N N1(C(CC2C(OC)COCC2)=O)CCC2(CNC(c3cnns3)=O)CCCCC12 C12(C(N3CCC(C)(CO)C3)=O)COCC1CN(C(C13CSCC1C3)=O)C2 n1(C(=O)NCCC2CCN(C(C34CC3C4)=O)C2)c(=O)oc2ccccc12 Cc1ccc(C(=O)NC2CCN(C(=O)Cc3cnoc3)C(C)C2)c(O)n1 c1(C(C)C)nnc2n1CCN(C(=O)C=Cc1nc3ccccc3[nH]1)C2C CC(C(C)C(=O)NCCCCN=[N+]=[N-])NC(=O)C=Cc1ccn(C)c1 c1(OC)ccccc1COCCNC(=O)N(C)CC1CCCSC1 C(c1ccc(CC)cc1)=CC(=O)NCCC1CC(NC(CC(=O)NCC#C)=O)C1 c1(C(=O)NCC2CC2NC(c2ccnn2CCF)=O)cc(F)c(F)cc1F CC(CO)C(C)NC(=O)CCN(C(=O)CN(C)C)C c1(CNC(=O)CCc2ccoc2)ncccc1C(=O)NCC(=O)N(C)C C1(NC(c2ccc(C)cc2)=O)CCN(C(c2nc(O)[nH]c(=O)n2)=O)CC1C N1(NC(=NCC)NC)CCCC2CN(CCOC)CCC12.c1(C)sc(C)nc1C c1(NC(c2nc(-c3c(OC4CC4)ccc(C)c3)sc2)=O)cccc(F)c1[N+](=O)[O-] C1(C(=O)NCC(C(=O)NC(CC)COCC2CC2)C)CCCC(=O)C1 Cc1ccn(CC(=O)NC2CC(NC(=O)CSCCC(F)(F)F)C2)n1 N1(C(C(CCC)OC)=O)CCC(C)(C)C1CNC(=O)CN(C)C(=O)OC NS(=O)(=O)c1ccc(CNCc2ccc(-n3cccc3)c(Cl)c2)cc1 c1(C(N(C(C)C)CCNC(=O)CC2CCCCC2)=O)cc2c(ccn2C)[nH]1 C1(c2nc(C(c3cccc([N+](=O)[O-])c3)OC)on2)CCC2CCCCC2C1 c1(C(N2CCCC(NC(C=C(CC)CC)=O)CC2)=O)ccc2snnc2c1 CCC(C)(CCC(C)C)C(=O)NC1CC(NCc2cnn(C)c2Cl)C1 CCCCC(C(=O)NCCCN1CCCC1C)NC(c1ccc(=N)[nH]n1)=O C(=O)(CCCC(F)(F)F)N1CC2(C(NC(C(CC)Sc3nc(=N)[nH][nH]3)=O)CC2)C1 c1(CCNC(=O)Nc2c(C)n(C(C)C(C)(C)O)nc2)cccc2c1OCCO2 CC1(C2CC2C(=O)N(CC(N2CC3CC3C3CC23)=O)C2CC2)COC1 Cc1cc(Cl)cc(C)c1C(N1CCOC(CNC(=O)Cn2c(C)csc2=O)C1)=O c1(CC)nncn1NC(=O)CN(C(=O)CC(C)(C)O)C C1(C(C)C)CCC(C(=O)NCC=CCC(=O)OC)N1C(=O)CC1(C#N)CCC1 c1(CCC)c(C(=O)NC2CC2NC(=O)C(C)c2ccco2)cnn1CCO C1(NC(C(CCCC)C(C)C)=O)CS(=O)(=O)CC1N=c1[nH]nc(-c2ccccc2)o1 N1(C(C(CC)N2CCCC2=O)=O)CC2CCC2(CNC(=O)C(=O)C(C)(C)C)C1 c1(C(=O)NC2C(C(=O)NCCS(C)(=O)=O)CC2)cncc(C#N)c1 C1(C)(CCCC)CCC(C(=O)NC(C)(C)CC(=O)N(CC)Cc2nc(CC)no2)C1 N1(CC(N2CC(N(C(=O)CC3CCC(O)C3)C)C2)=O)CC2CCC1C2 N1(Cc2onc(C(C)C)n2)CCN(C(C)(C)CNC(=O)CC2CN(C)C2)CC1 Cc1ccc(NC(=O)CC2CCN(C(=O)OC(C)(C)C)CC2C)c2[nH]ncc12 c1(NC(C)C(F)(F)F)nc2c(c(=NCC(C)(C)OC3CCOCC3)[nH]1)COCC2 C1(NC(c2cc(C(C)C)n(C)n2)=O)CCCCN(Cc2cnn(C)c2)C1 S(=O)(=O)(c1ccc2[nH]c(=NCC3(C)CC3(C)C)sc2c1)N1CC(CCC)OCC1 c1(C(=O)NCCN(C(C2CC(OC)C2)=O)C2CC2)c[nH]nc1C(F)(F)F c1(NC2C=CC(NC(CNS(CCCC)(=O)=O)=O)C2)cc(Br)ccc1C#N C(=O)(C1CCCc2nncn21)N1CCCC(NC(c2cc(C)c(C)[nH]2)=O)C1 C1(N(C(CC(CCC)C)=O)C)CCC2CN(C(=O)CN(C)C(N)=O)CC12 N1(C(CC(c2ccc(F)cc2)C)=O)CCC(CF)(NC(c2cc(Cl)n(C)n2)=O)C1 N1(C(COCC=C)=O)CC2(C1)CN(C(c1sc3ccsc3c1C)=O)CCO2 C(C(=O)N(OC)C1CCCC1)n1cc(-c2c(CC)n[nH]c2)nn1 N1(C(c2cnc(CC)[nH]2)=O)CC2CCCC(CNC(=O)CC3(CO)CC3)C2C1 c1(NC(C2(C(=O)NCC)CC2)=O)ccc(O)c(OCC(=O)NC2CC2)c1 C(=O)(C(O)CCCNC(C12CCC(CC1)C2)=O)NCC(CC1CC1)OC C(=O)(CCC(C)(C)NC(c1cnc(C)c(C)c1)=O)NCc1nc(C)c(C)[nH]1 N1(C(C2CC(C)C2(C)C)=O)CC2CCC1CN2C(C1C=CCCC1)=O C#CCC(CC(=O)N1CCC(O)(C(C)C)C1)NC(c1sccc1C#N)=O C(=O)(C(C)C(C)(C)C)N1CC(OC)C(NC(=O)CCn2cnccc2=O)C1 N1(C(c2c(F)ccc(N)c2)=O)CCCC2CN(C(C3CC4CCC3O4)=O)CCC12 c1(NC(C(C)NC(c2cccc(CO)c2)=O)=O)cc(C(F)(F)F)ccc1F C1(C)(C(N(CC)Cc2cccnc2)=O)CCCN(c2cc(OC)nc(C)n2)C1 c1(C(=O)NCC2CCN2C(c2cnn3ncccc23)=O)cc2c(nn1)OCCS2 c1(CC(=O)NCCN(CCOC)C(C2CS(=O)(=O)C2)=O)cnc(Cl)cc1C Cc1cc(C#N)ccc1CC#N.C12CC(C)N1S(=O)(=O)C2.C1CNC1 C1(C)(C(N(C(CCC)C(=O)OC)C)=O)CCCN(Cc2ccccc2C)C1 CCC(CC)CC(=O)NC(c1ccccc1F)CNC(=O)C(COC)CC CC(C)(C#CC(=O)Nn1nnc2c1CCCC2)C(C)(C)NC(c1ccc[nH]1)=O c1(C(=O)NCC2(NC(=O)Cc3n[nH]cc3Br)CCCC2)cccc(C(F)F)c1 C1(CNC(C=C(C)C(F)F)=O)CC12CCN(C(=O)CN(C1CC1(F)F)C)CC2 c1(C(N(C(C)CNC(C2CCC(C)CC2)=O)CC)=O)nc(C(C)C)ncc1Cl N1(C(C(C)c2ccco2)=O)CCCCC12CC(NC(=O)CN(C)CCO)C2 C1(CC)CC(C(=O)N(C)CC2CCCN(C(=O)CCP(C)(C)=O)C2)CC(=O)N1 C(CC(=O)N1CCCCCCC1C)(C(F)(F)F)NC(c1cc(C)cc(O)c1)=O Cc1ccc(C=CC(=O)NCC2(C)CC(NC(c3ccc(C)nc3N)=O)C2)nc1 N1(C(CN(CC)CC)=O)CCCC(CN(C)C(C2CCN(C(=O)NC)C2)=O)C1 C1(O)(CC=C)CN(C(C2CC(=O)C2C(F)(F)F)=O)C1 c12nccnc1N1CCCC(C1)C2.c1(C2N(C(C)=O)CC2)ccc(N2CCCC2)o1 C1(CC(N2CCC(NC(C3(C4CCCOC4)CC3)=O)C2)=O)COC2CC1C2 Brc1csc(N2CCCC2c2n[nH]c(C3CC3)n2)c1 CCCC(C(=O)NCCN(CCC)C(C1CC2(C1)CC2F)=O)C(C)C C(=O)(CCC(C)NC(C1(SC)CC1)=O)NC(CC=C)C C1(NC(C=Cc2n(C)cnc2)=O)CCCC12CN(C(C1NC(=O)OC1C)=O)C2 c1(OC)cc(C(=O)NC2CCN(CC3CCCCC3)C(C)C2)cc(Cl)c1 C#Cc1ccc(C(N2CC=CC(NC(=O)Cc3ccc(F)c(Cl)c3)C2)=O)c(F)c1 c1(N(C)C(C2CC2CCNC(=O)COCC2CCOC2)=O)cc(CO)on1 C1(C(=O)NC(C2CN(C(C3(C4CCOCC4)CC3)=O)C2)C)CN2CCCN1CC2 C1(C(=O)NC(C)(C)CCNC(c2ccccc2CC#N)=O)CCc2ccnn2C1 C1(C(C)C)CN(C(c2ccc(O)nn2)=O)CCN1C(=O)Cc1nc[nH]n1 O=S(=O)(c1ccccc1C(F)(F)F)N1Cc2ccc(SCCO)cc2C1 CS(=O)(=O)CCc1cn(CC2CCN2C(=O)Cc2nccn2C(F)F)nn1 c1(SC)ccccc1C(=O)NC1CCC(CNC(=O)Cn2cc(C(N)=O)cn2)C1 Cc1nscc1C(=O)NC(Cc1cn[nH]c1)C(=O)NCC1(CCO)CCC1 Cc1cc(O)c(F)cc1NC(C1(NC(=O)C(C2CCOCC2)O)CCOCC1)=O c1(C(=O)NC(C(C)NC(C(C)Cc2cnc[nH]2)=O)(C)C)cc(Cl)c(F)cc1O c1(NCC2(CO)CC(C)C2)cc(Br)ccc1S(=O)(=O)N1CCC2CC12 C(C(C)C(C)C(=O)NC1(CNC(=O)CSC)CC(F)(F)C1)OC C12(C(=O)NCC#CCNC(c3cnc(COC)s3)=O)CSCC1C2(F)F c1(C(C(=O)NCCCCN(CCCNC(C2SCCS2)=O)C)F)ccccc1 c1(C(N2CCC(c3cn(Cc4cnn[nH]4)nn3)CC2)=O)ncccc1Br C1(C(=O)NC(C2CCN(C(C3(C#N)CCOCC3)=O)CC2)C)CCC(=O)N(C)C1 N1(C(C2(SCC)CC2)=O)CC2CCC1C(CNC(=O)CCc1cc(OC)no1)C2 c1(NC(C2N(C(C(C)C)=O)CCCC2)C)nccc(S(C)(=O)=O)n1 N1(C(C(=O)N(CC(C)OC(C)(C)C)C)=O)CC2CCCC12 Cc1nc(Cl)sc1C(N1CCCC(C(=O)NCCOCC(F)(F)F)C1)=O c1(CC(=O)NCCCN(C(C2CCCCC2(C)C)=O)CC)cc(O)nc(O)n1 N1(C(c2cc(C)c(O)nc2)=O)CCCC2(NC(c3cnnn3C)=O)CC2C1 N1(C(C(C(C)C)OC)=O)CC(C(=O)NC2CSC2)C(C)(C)C1 Cc1ccc(F)c(CNC(c2cncc(CNC3(C)CC3)c2)=O)c1 N1(C(C2CCC(N(C)C)CC2)=O)CCC(C2CC2)C1CNC(=O)CSC(=N)N c1(S)ncc(NC(N2CCC(Oc3ccncc3)CC2)=O)cn1.CCCOC N1(C(C2(COC)CC2)=O)C2CCC1CC(CCNC(c1c(C)nc(C)n1O)=O)C2 C(=O)(C(C)CC(C)(C)C)N1C(C(=O)NCC(CC(=O)NC)C)(COC)C=CC1 C12(C(=O)NC3CC(C=C)C3)COCC1CN(C(c1ccc(CF)cc1)=O)C2 C1(C(N2CCOC(C3CC3)C2)=O)C(CC)CCCN1C(=O)Cc1cncc(C)c1 CC1CCC(C(=O)NC(C2CCCN2C(=O)CN2CCCC2CO)(C)C)C1 N1(C(c2ccc(C)c(O)c2)=O)CCCC12CCN(C(C1CCCCC1(C)C)=O)C2 C(C1CN(C(=O)CCc2ncnn2C)CC1C(N1CC(CC(C)C)C1)=O)=CC C1(CNC(CC2(OC)CC2)=O)C2CN(C(c3ccn(C(C)C)c3C)=O)CC12 CC(C)C(C)C(=O)N1CC(C)C1C(=O)NCCc1cocn1 N1(C(CCCCCC(C)C)=O)CCC2(CC1)CC(C)N(C(c1csc(Cl)n1)=O)C2 CCCC(CC)CCC(=O)NC1(CCNC(=O)CC(C)N2CCCC2=O)CC1 C1(CC(=O)NCC2(Nc3nc(C)nc(O)c3)CC2)COc2ccccc2O1 Cc1cc(CN2CC(O)CC2C(N2CC3CCC2C3)=O)c(C)cc1Br C12(CNC(c3nsnc3O)=O)CC(CCO1)N(C(C1CC3C=CC1CC3)=O)C2 C1(O)(C(C)NC(CCC(=C)C)=O)CCN(C(=O)CSCCN(C)C)CC1 C12(C(N3CC(C)(NC(c4n(C(CC)C)ncc4)=O)C3)=O)CCC(CC1=O)C2 C1(CCNC(=O)OC(C)(C)C)CC(C(=O)NC(c2nnc(O)o2)C)=NO1 C1(NC(CN(C)C(c2ccoc2)=O)=O)CCCCN(C(C2CCCC2(C)C)=O)C1 c1(C(=O)NC2C=CCC(C(=O)NC(CCCC=C)C)C2)c(C#N)ncn1C C1(=O)C(C(C)(C)C)N1.c1(C(N(C(CC)CO)C)=O)cn(CCO)nn1 c1(CN2CC(OC)C(NC(C3C=CC(=O)N=N3)=O)C2)c(F)cc(Br)cc1F C1(CN2C3CN(c4nnc(CC(C)C)s4)C(C3)C2)CC12CCC(F)(F)CC2 C1(O)(CNC(CSCC(N)=O)=O)CCCN(C(c2cncnc2C2CC2)=O)C1 C1(C(=O)NCC2(NC(c3[nH]cc(C)c3)=O)CCCC2)OC2CCC1CC2 c1(C(N(C)CC2N(C(C(CC)SC)=O)CCOC2)=O)cnc(O)cc1C c1(N2C(C(=O)NC(COC)C)CC3(CC3)C2)ncc2c(n1)CCC2 c1(N2CCC(C(=O)OC)(C(C)C)C2)ncnc2cc(-c3ccccc3)sc12 c1(C(=O)NC2CCCN(C(c3cc(C)oc3)=O)C2C)ccccc1N=[N+]=[N-] Cn1nc(C(=O)NCC2CC3(CC3)CN2C(=O)CC2(C)CC2(Cl)Cl)c2c1CCC2 C(=O)(C(C)(C)CNC(=O)CC1CCC(NC(C2CCCN2C)=O)C1)NC C1(C(=O)NCC(C2CCC2)OC)CCCC(NC(c2nnsc2N)=O)C1 c1(COC)ccc(C(=O)NCC2(F)CN(C(c3ncoc3C3CC3)=O)C2)s1 C1(NC(C2(CC)CCNC2=O)=O)CCC2CC1CN2C(=O)Cn1cncn1 C12CCCC(C1)C(=O)N2.c1(CN(C(CN(C(COC)=O)C)=O)C)ccsc1 c1(C(N2C(CCC)CN(C(=O)C(C)CSC)CC2)=O)cnn2cccc(C)c12 C12(NC(C3CC3(Cl)Cl)=O)CCCN(C(=O)Cc3c(Cl)cccc3Cl)CC1C2 c1(SC)cc(C(N2CCCC2CCC(=O)NCC(C)(C)C2CCCO2)=O)co1 N1(C(c2c(C)nc(CCC)s2)=O)CCC(C)C(NC(=O)CC2(O)CCOC2)C1C C(=O)(C1=CS(=O)CCC1)NCCCCNC(CC(C(C)C)C)=O C1(N(C(=O)CC(C2CC2)C2CC2)C)CN(C(=O)C(C2CC(F)(F)C2)O)CC1F N=c1[nH]c(CC(=O)NCC2C=CC(NC(=O)C(=O)Nc3ncc[nH]3)C2)cs1 C(C(C)(C)C(=O)N1CC(C(=O)NC2C3CCCC23)C(C)C1)OC(C)C CC(CCCCNC(=O)CC1CC1(Cl)Cl)NC(C1CC(O)(C(F)(F)F)C1)=O c1(C(=O)NC2C(NC(CCc3nnc(CC)o3)=O)CCCC2)n[nH]cc1[N+](=O)[O-] c1(CC)ccc(C)cc1C(N1CC(CC(C)NC(C2CNC(=O)O2)=O)C1)=O CCCC(C)(CCC)C(=O)NC1CC(CNC(c2ccnc(N(C)C)c2)=O)C1 CC1(C)CCC(C(=O)NC2CC(CNC(c3cnn(CC(F)(F)F)c3)=O)C2)C1 CCCC(C(=O)N(CCCNC(c1nccc(C(=O)OC)n1)=O)C1CC1)NC(N)=O c1(-c2ccc(CN3CCC(C(N(C)C4CC4)=O)CC3)cc2)nc2ccccc2s1 C1(NC(C(C)CN(C)C)=O)CCN(CCNC(C2C3CCC2CC3)=O)CC1 c1(CNC(C2CCC(CNC(C(C)(C)C)=O)C2)=O)ccnc(Cl)c1 C1(NC(C2C(C(=O)OC)C2)=O)CC(NC(c2nn(C)cc2Br)=O)C(O)C1 Cc1cccn2nc(C(=O)NC3CCN(C(c4cncnc4)=O)C(C)C3)cc12 N1(C(c2cccc(C=CC(F)(F)F)c2)=O)CCC2CCC(F)(F)CC2C1 N1(C(c2c(C(=O)NCC#C)cccc2)=O)CCc2[nH]c3ccc(F)cc3c2C1 c1(C(=O)NCC2(OC)CN(c3cc(C(F)(F)F)nc(C)n3)C2)cnc(N)c(O)c1 c1(-n2c(C(O)C3CC3)nc(CC)n2)ccc(S(=O)(=O)C(F)(F)F)cc1 N1(C(c2c(C)c[nH]n2)=O)CCC(c2cn(CC3CCC3)nn2)C1(C)C C1(OC)CN2CCCC2(C(=O)NCC(CC(C)C)NC(c2cnoc2)=O)C1 N1(C(c2c(C)nn(CC(F)F)c2C)=O)CCC(C)N(C(=O)C(C)SC(C)C)CC1 N1(C(CCSCCCC)=O)C(CNC(=O)CCc2ncco2)CC2CC12 CC(CCC(C)(C)C)C(=O)N(c1nc2ccccc2s1)Cc1ncnn1C CC(C)C(O)CC(=O)N1CC(F)(F)CC1C(=O)NCc1nn(C)c(=O)n1C c1(CNC2C(C)CN(C(C)(C)C)CC2C)nc2ccc(F)cc2o1 CCCC(C(O)C(=O)NC(C)(CC)CCO)NC(=O)C(O)CCN(C)C C1(CNC(C(CC#C)C2CC2)=O)C(C)CCCN1C(=O)C(C)CF C1(C)(NC(C(CC)C)=O)CCN(C(C2(c3cc[nH]n3)CCC2)=O)C1 c1(C(N2C(CNC(CSCC)=O)C(C)(C)CCC2)=O)cnc2n1CCCC2C C1(CNC(c2sccc2CNC(C2C3(CC3)C23CC3)=O)=O)CCCC2(CC2)C1 c1(NS(C)(=O)=O)cc(CNC(=O)CS(=O)Cc2ccccc2)cc(C(F)(F)F)c1 C1(NC(Cc2cnc(C)s2)=O)CCN(C(=O)CC(C)c2ccncc2)C1C C(=O)(C1=CCN(C)C1)NCCc1c(CNC(C(CC)NC(=O)OC)=O)nco1 C1(CC(N2C(C=C)CC2)=O)CCN(C(C2CC(O)C(F)C2)=O)C1(C)C C(=O)(CCC(C)(C)[N+](=O)[O-])NC1CN(C(c2cncc(C=C)c2)=O)C(C)(C)C1 C=C(CNC=O)CCN1C(=O)C1.c1(C(C23CCC2C3)=O)ccccc1.C1(C)(ON)CC1 c1(NC(C)=O)cc(NC(c2ccc(Nc3ccccc3)o2)=O)ccc1C C1(CC(=O)N(C(=O)C(C2CCOCC2)C)CCN(C(C)=O)CC)C(C)(C)C1(C)C CC1CC(C)S(=N)(=O)CCN1C(c1cccc2ccccc12)=O c1(C(=O)NC(CC=C)CNC(c2c(C)csc2Cl)=O)ccc(C(C)C)nc1C c1(CC)c[nH]cc1C(=O)NCC1OCCC1C(=O)NCC(c1ccsc1)O C1(CNC(C(C2CCOC2)OCC)=O)N(C(=O)CC(C)SC)CCCC1(C)C CC(C(=O)N1CC2CC(NC(c3ccc(O)nn3)=O)C1C2)C(C)(F)F CCCCC(F)C(=O)N1CCCC(CC(=O)NC(CC)C(C)(F)F)C1 C1(O)(CNC(C(CC)SC)=O)CCCN(C(c2cc(OC)ccn2)=O)CC1 c1(OCC(=O)NCC(CNC(C(C)CC2CC2)=O)(C)C)ccccc1F n1(CC)ccc(=NC(=O)CC=CCNC(c2ccc(F)c(F)c2)=O)[nH]1 Cc1cccc(CCNC2CCOC(c3ccncc3)C2)c1 C1(CNC(C(CSC)OC)=O)CC(C)CCN1C(=O)Cc1cncc(C)c1 C=CCCC(F)(F)C(=O)N1CC2(CCCC2NC(c2cn(C(F)F)c(C)n2)=O)C1 N1(C(C2CC(C)OCC2)=O)CC2CC(C1)C2NC(c1ncccc1C(F)F)=O S(=O)(=O)(c1ccccc1Cl)NCCCNc1c(C(=O)NC(CCCC)C)scc1 c1(C(=O)NCC23C(CN(C(CC4(C=C)CCC4)=O)C2)C3)nnn2c1COCC2 C(=O)(C1CCCc2c[nH]nc21)N(C1CCN(C(=O)CSCCOC)CC1)CCC CC1=C(C(=O)N2CC(NC(c3cc(Cl)cn3C)=O)C2)S(=O)(=O)CCO1 C=CC1(CC(=O)NCCCC(=O)OC)CN(C(=O)C(C)C2CCCO2)C1 CC1CCC(NC(C2CCC(C(N)=O)C2)=O)CN1C(C12CC(CO1)C2)=O c1(C(=O)NCC(C2(O)CN(C(C(C)SC)=O)C2)(C)C)nc(SC)n2ccccc12 c1(OC)ccccc1CNC(C1(C(C)C)CCCN1C(c1cnn(C)c1C)=O)=O O=C1CC(C(=O)NOCC2CCCC3CC23)N(C(=O)CC2(O)CCCOC2)C1 N1(C(C(C)OCC=C)=O)C2CC1CN(Cc1ccc(CC)cc1)C2 C1(CN(C)C(=O)Nc2ccccn2)CCN(C(c2cccs2)=O)CC1 c1(C(N2CC(C)(CNC(CSCC)=O)OCC2)=O)cc2nccnc2cc1F C#CCCCCCC(=O)NC1CCC(C)(CNC(=O)CCc2cc(OC)no2)C1 C1(CNC(C(CC#C)C)=O)CC2CCC1N2C(c1cc(C)cc(F)c1)=O N1(c2ncc(C)cc2C)CCC2(NC(c3ccc(F)cc3Cl)=O)CCCC12 C=C=CCCC(=O)NC(CNC(=O)CCC(C)c1ccccc1)CO c1(CC(N2CC(COC)(CNC(=O)COc3ccsn3)C2)=O)noc(C)c1C#N CC(C)(C)[Si](C)(C)OC.c1(C=O)cc(C2CC2)on1 C(=O)(C1=C(C#N)CCC1)NCCn1cc(C(N2C3CN(C)C(C3)C2)=O)nc1 C1(NC(c2c(C)snn2)=O)CN(C(c2cc3c(o2)CCCC3)=O)CC2CCCC12 Cc1cc(F)ccc1C(N1CC(C)(C)CC1CC(=O)NC(c1ccnn1C)C)=O C(C)(c1cccs1)=CC(=O)NCCN(C(=O)C(CN(C)C)N(C)C)CC.C(C)(C)(C)S Cc1cc(O)ncc1C(N1C2CCC(C2)C1C(=O)NCCC1(C)CCCO1)=O N1(C(CCCC#CC)=O)CCC2(C1)CN(C(C13CC(C1)C(C)O3)=O)CC(C)O2 Cc1n[nH]c(C)c1CC(N1CCCC(C(C)C(=O)N(C)CCO)C1)=O Cc1cc(=NC(COC(F)(F)F)CCO)nc(N2CCOC(CC(C)(C)C)C2)[nH]1 Cc1cnnc(O)c1C(=O)NCC1CC(F)(F)CN1C(c1cccc(CO)c1)=O CCC(CC(=O)N1CCC=C(C(=O)NCc2ncoc2C(C)C)C1)C(F)F N1(C(CC(c2c(OC)cccc2)N)=O)CCN(Cc2ccc(Br)nc2)C(CO)C1 c1(CC)n[nH]c(=NCC(CC)N(C)C(C2CCC(C)(C)CC2)=O)s1 c1(NC(=O)CC2CCCN(C(=O)CCc3ccsc3Cl)C2)ccc(F)cc1CO Cc1nc(O)nc(C)c1CC(N1CCCN(C(C2OC3CCC2CC3)=O)CC1)=O c1(C(N(C(CNC(CC(CC)CC)=O)C)C)=O)ccc2cnnc(O)c2c1 Brc1ccc(-n2nnnc2C(c2cncs2)NCCCOCC2CC2)cc1 c1(N)cncc(C(=O)OC)c1.C(C1CCCC1)=CC(=O)CCN(C1CCCC1O)CC CC(C)C1=CCC(C(N2CC(C(N3CC4(CC(O)C4)C3)=O)C3(CCC3)C2)=O)CC1 Cc1cc(-c2cnc(Cl)c(C(N3CCC(CCO)CC3)=O)c2)ccc1C#N N1(C(c2c(CC)nc(C)[nH]2)=O)CCCC(C)(NC(c2c[nH]c(Br)c2)=O)C1 C=CC(CO)OC.C(C(F)(F)F)N1C(=O)C=C(C)CO1 C=CCCCCCC(=O)NC1CN(C(=O)Cc2cncnc2O)CC1C c1(C(=O)NCC23CC(CNC(C(CC)O)=O)(OC2)C3)cccc(F)c1F N1(C(CC#N)=O)CC(F)(F)CC1CNC(=O)Nc1cccn1Cc1ccccn1 C1(CNC(C(c2cccs2)NC(c2cn(CCOC)nc2)=O)=O)CN(C)CCO1 c1(CN2C(C(=O)Nc3cc(C)c(F)cc3)C(O)CC2)cc2c(Br)cccc2[nH]1 CC(C)(CC(=O)NCC1CCCC(NC(c2cc(=O)cc[nH]2)=O)C1)CC(F)F c1(OC)cc(C(=O)N(C)CCNC(c2nc(=O)n(C)[nH]2)=O)cc(OC)c1O C1(C(=O)NCC2(CC)CCC(=O)N2)CCCCN(C(=O)C(C)C2CCOC2)C1 CC1CCN(C(=O)CCS(C)(=O)=O)CCN1C(=O)CS(=O)(=O)N1CCOCC1 C1(N(C(CN(CC)CC)=O)C)CCCN(C(=O)Cc2ccnn2C2CCCC2)C1 C1(C(=O)NCC2C(NC(c3nc(C)[nH]n3)=O)C2)CC=CCC1C CC(C)C(N=c1[nH]c(Cl)ncc1Cl)C(C)NC(=O)OC(C)(C)C c1(CC)cc(CC(=O)NC(COC)C(=O)NCc2n[nH]c(C3CC3)n2)no1 c1(NC(C2(NC(C)=O)CC2)=O)ccc(N2CCN(C)CC2)cc1 C1(C)(C(=O)NCC2N(C(C(CC)(F)F)=O)CCC2)CCCNC1=O C1(C(=O)NCCC2N(C(c3c(CC)nns3)=O)CCC2)CCC(O)CC1 Cc1cc(C(=O)N(C)CCOCCNC(=O)C2=CCCC2C)ncc1Br c1(C(=O)NC2(CNC(=O)C(O)C3CC3)CCC2)ccc(SCCC2CC2)cc1 C12(NC(C(C)C3CCOC3)=O)CCC(CNC(c3cccnc3S)=O)(CC1)OC2 N1(C(=O)NC2CC(C)=C(C)CC2)CCOC2(CCN(C(=O)OC(C)(C)C)C2)C1 c1(CCC(=O)NCc2c(N)c([N+](=O)[O-])cc(F)c2)nc(O)c2cc(Br)ccc2n1 N1(c2cc(C)nc(NC(c3n[nH]c(=N)s3)C)n2)CCCC(C2CCCC2)C1 c1(C(=O)NC(C)CNC(=O)C(O)C2CCC2)cccc(-c2ccco2)c1 c1(NC)cnccc1C(N1CCCC1C1(NC(c2ccsc2C)=O)CC1)=O c1(CCC(=O)NCCCNC(C2CC2c2cccc(Br)c2)=O)ccc(O)nc1 Cc1ncnc(C)c1C(=O)NCC1(NC(=O)CC2(O)CCOC2)CCCC1 CC(C)(C(F)F)CC(=O)NCCCCCCNC(=O)C(Cl)=CCl C1(NC(C(C)=CC)=O)CC2(C1)CC(CNC(c1cccn1C)=O)C2 C1(C(=O)NCC2C(NC(Cc3c(C)cccc3C)=O)C2)CCn2nccc2C1 C(=O)(C(C)CC(C)C)NCC(C)(CNC(=O)C(C)Cc1c(C)n[nH]c1C)OC c1(NC(C(C)O)C(=O)OC(C)(C)C)ccnc2c1CCO2 C1(NC(Cc2ccc(CCC=C)cc2)=O)CC2CC1N(C(=O)C(CC)OCC)C2 C1(C(=O)NC(C(=O)OCC)Cc2cc[nH]n2)(OCC)CCCC1.C(=O)(COC)N N1(C(C(=O)NCC(F)F)=O)CC2COCCC2(NC(c2csc([N+](=O)[O-])c2)=O)C1 C1(CC)C(NC(C)=O)CCN1C(=O)Nc1ccccc1C(C)(C)C NS(=O)(=O)c1n[nH]cc1C(N1CC2CCC1C(CNC(=O)CCC1OCCO1)C2)=O N1(C(C2CC(C)(O)C2)=O)CCC(N2CCN(C(C3CCC4CC4C3)=O)CC2)CC1 C1(C(=O)OC)CNC(=O)CN1C(c1cccc(F)c1)=O.c12cccc(c1)N2 Cc1cc(N2CCCC(C#N)C2)nc(N2CCOC(CCF)C2)n1 c1(OC)ccnc(C(=O)NCC2N(CC3CCN(Cc4ccccc4)CC3)CC2)n1 N1(C(C2CC(CNC(COCCCC#C)=O)C2)=O)CCC(OC)C1 N1(Cc2c(-c3c(C)nc(OC(F)F)cc3)csc2)CCc2c(F)cccc2C1 N1(C(c2c(CC)nns2)=O)CCN(C(c2ccc(OC(C)C)nc2)=O)C(C)C1 Cc1[nH]nc(C(=O)NC2CCCC2CNC(c2sccc2Br)=O)c1C c12cc(Cl)ncc1NC(=O)C1CC(F)CN(C1)C2=O.C(COCCO)OC N1(C(C(C)(C)CC2CC2)=O)CCC(C2CN(C(C3OCCOC3(C)C)=O)C2)CC1 Cc1nc(C2CC2)nc(S)c1C(=O)NC1CCC(NC(=O)C(C)(C)C(C)C)CC1 c1(C(=O)NCCCC(C)NC(c2cc(OC)c(C)cc2)=O)cc(Cl)cc(Cl)c1O C1(NC(c2c(C)coc2)=O)CCCCC1CC(N1CCC(CC2CC2)C1)=O C=CCCC(C(=O)NCCc1cccnc1)NC(=O)CCC(C)(C)C c1(C(=O)NC(CN(C(C2CC(CCC)C2)=O)C)C)ccn(-c2ccccc2)n1 C1(NC(C(CCNC(C2C(C)CC2)=O)(C)C)=O)CCC(C2CC2)CC1 c1(OC)cc(F)c(C(N2CC3CC(C2)C3NC(C2C3CC4C(C3)C24)=O)=O)cc1F CC1OC(C)C(C(N2CCC(O)(C(C)NC(=O)C3=CCCS3)C2)=O)C1C c1(CC(C)C(=O)NC2(C)CCN(C(=O)C(C)(C)C3CCC3)C2)ccc(C#N)cc1 C(=O)(CCC(=O)c1ccc(Br)cc1)NC1CC(NC(C(COC)C)=O)C1 C(CC(C(=O)NC12CC1CN(C(=O)CCNC(=O)CO)C2)NC(N)=O)SC C(C1CCCC1)=CC(=O)NC1CC(CCNC(CN(c2ccccc2)CC)=O)C1 C1(NC(c2cccc(CN(C)C)c2)=O)CCN(C(=O)COC2CCCC2)C12CC2 C1(=O)CC(C(F)F)CC(CC)O1.C(C)(C)(CC)NC(=O)OC(C)(C)C Cc1ncncc1C(=O)NC(CNC(=O)Cc1ncoc1C)Cn1cccn1 N1(c2nnc(C(=O)OC)s2)CC2CC(NC(c3cc(C(C)(C)C)on3)=O)C2C1 C1(F)(CNC(=O)CNC(=O)C2CC2)CC(CNC(C2CCC2c2nc[nH]n2)=O)C1 Cc1ccnc2c(C(N3CC(C)CCC3CNC(=O)C(C)(C)C(C)C)=O)cnn12 Cc1cc(F)c(C#N)cc1NC(C1CCCCN1C(=O)C1=COCCC1)=O Cc1cc(C(=O)OCCC(C)(C)NC(=O)OC(C)(C)C)c(C)n1NC(N)=O.C(C#N)S CC(CN=C(NCC1CCOCC12CCC2)NCC(F)F)N(C1CCCCC1)C c1(C(N2CC(SC)C(NC(=O)C(C)(C)SC)C2)=O)ccc2ncn(C)c(=O)c2c1 c1(CNC(N(C)Cc2cc(Br)cnc2Br)=O)cc([N+](=O)[O-])nn1C c1(NC(C2C(CC)CN(C(=O)CC(C)SC)C2)=O)cc(CO)cc(F)c1 c1(C2(C(=O)NC3CCCC3C(F)(F)F)CCC2)cc(OC(F)F)ccc1O C1(C)(C(=O)NC2C(CNC(C(C#C)(C)C)=O)CC2)CCC(C)=C(C)C1 C(C(CCC)C(=O)NCC(C)(C)F)NC(COC1(C#C)COC1)=O C1(C(=O)NCCN(C)C)CCCC1CSCc1cn(C(C)C(=O)O)nn1 c1(C(N2CC(NC(CC3(COC)CC3)=O)C3C2C3)=O)cc(Cl)cc2c1OCC2 C1(c2cn(C3(CC4CCN(C(CCCOCC)=O)C4)CC3)nn2)CCCCC1F C(=O)(C1CCCc2nn(C)cc21)N(CC(C)CNC(c1cnn(C)c1F)=O)C N1(C(c2ccc(C(Cl)Cl)cc2)C(=O)NCCSC)CCC(C)C(CO)C1 CCCCC(=O)C(=O)N(CC(C)(C)CNC(=O)CCc1scnc1C)CC CC1(CNC2CC2C(F)(F)F)CCN(C(N2CCOC(c3nc(C)cs3)C2)=O)C1 CCCC(C(=O)N1CCC(C)(CNC(c2ccc(C(F)F)nc2)=O)C1)NC(N)=O C=C(C)C(CC(=O)N1CCOC(CN(C)C)C1)OCC.C12(CC1)C(C)NC2=O C(CN=c1c(-c2sc(SC)nc2C)c[nH]cc1C)c1c(OC)cccn1 N1(C(c2[nH]cc(C)c2)=O)CCN(C(C2CC(C#N)C2)=O)C2CCCC2(C)C1 c1(NCc2cc(C)nc3n2ncc3Br)[nH]c(=NC2CCC(Cl)(Cl)C2)nc2c1ncn2C c1(C(N(CC(C)NC(C2CCCN2C2CC2)=O)C)=O)c(C(F)F)cccc1C(F)F N1(C(C=CC)=O)CCN(C(c2ccccc2Br)=O)CC1c1cn[nH]c1 N1(CCNC(=O)NC(CC)CN2CCCC2)CCC2(CC(n3ccnc3)C2)C1 c1(SCC(=O)NC2CC(NC(=O)C=CC3CCOC3)C2)ccc(C(F)(F)F)cn1 C(=O)(N=c1cc(Br)n(C)[nH]1)Nc1scc(C(C)C)n1 c1(C(=O)NCCC2CC(NC(c3cc(OC)n[nH]3)=O)C2)nn(C)cc1Cl CC1=NN(C)C(=O)C1CC(N1CC=CC1CNC(=O)OC(C)(C)C)=O C=CC(C(=O)N1CSCC1CC(N1CCC1(C)CC)=O)OC C(CCCCCNC(C1CCCC(=O)O1)=O)N(C(CC1N(C(C)C)CCC1)=O)C c1(OC)cc(C(N2CCC(CNC(c3ccccc3F)=O)C(C)C2)=O)ccc1F CC1CN(C(c2cccc(C(=O)O)c2)=O)CCN1C(c1ccc(O)c(=O)cc1)=O C1(NC(C(CN(C)C)NC(CNC(CCC)=O)=O)=O)CCC(CO)CC1 N1(C2c3cc(on3)NC2=O)CC=C(CC(=O)NC)CC1.C(=O)(C)OC.C(CC#N)SC N1(C(c2c(CC)ocn2)=O)CCC(CNC(c2cnn(CCF)c2)=O)C12CC2 c1(C(C)(C)C)ncc(C(N2CCSCC2CO)=O)cc1O C1(CNC(C2C(OC)CCC2)=O)CN(C(c2ccncc2F)=O)CCN1C Cc1ccc(Cl)cc1C(=O)NC(C1CN(C(c2c[nH]c(C(N)=O)c2)=O)CCO1)C Cc1cccc2oc(N3CC4(CC4)CC3CNC(C3C4CCCC34)=O)nc12 Cc1cnc(C)c(C(=O)NC(C)CC2CN(C(=O)C=Cc3cn(C)cn3)C2)c1 C1(NC(C(C(CC)(C)C)O)=O)CC2CCC(C1C)N2C(=O)C=Cc1ccccn1 C1(NC(c2c(OC)cc(N)cc2)=O)CCN(C(C2CCSCC2)=O)CCC1CO C#CC1(NC(=O)C(CC)N(C(=O)C(C)CC(C)(C)C)C)CC2CCCC12 C12(CNC(C3C(C(N)=O)C3)=O)CCC(CN(C(=O)CN3CC4CCC3C4)C1)C2 C12(C(N3CCCN(C(C)=O)CC3)=O)COCC1CN(CCOc1ccccc1)C2 C1(C(N2CC(OCC(N3C(CNC(CC)=O)CCC3)=O)C2)=O)CCC(C)(O)CC1 CC1(C)CC(=O)CCN(Cc2cccnc2)C1.n12cc(nn1)C2 c1(OCC(C(=O)N(CCNC(=O)Cc2cocn2)CC)OC)ccc(Cl)cc1C C1(CCNC(c2c(COC)noc2)=O)NC(=O)NC1=O.C12(CCOC1)C(=O)N2 N1(C(c2ccn(C)c2)=O)CCN(C(=O)CCS(N)(=O)=O)C(c2ccccc2)C1 C1(NC(CN(c2cc(NC3CCCSCC3)ncn2)C)=O)CCS(=O)(=O)C1 c1(C(N(C2CCCC2)CCNC(c2coc(C(F)F)c2)=O)=O)ccc(Br)nc1N C=CCCCCN(C)C(C1(C)C=CCN1C(=O)COC(C)(C)CC)=O c1(C(=O)NCC(C(C)C)NC(C(CC)NC(N)=O)=O)cc2c[nH]cnc-2n1 c1(CCCNc2cn(C3CN(C(C(=O)OC)=O)C3)nc2)cccc(C)c1 c1(OC)nc(C)c(C(c2nnnn2CC2CCCO2)NCCCF)c(C)c1Cl Nc1sc2c(c1C(N1CC3(CCC(CNC(=O)C4=CCCC4)O3)C1)=O)CCC2 N1(C(CCC=C)=O)CCC2(CC1)CC2C(N1CCOCC(C(=O)O)C1)=O C#CCC(CC(F)F)C(=O)NC1CC(CO)(NC(C2CCN(C(C)(C)C)C2)=O)C1 Cc1cc(F)c(NC(C2CC(=O)CN2C(c2csc(=N)[nH]2)=O)=O)cc1C Cc1ccc2c(c1)CC(C(=O)NCC1CCC1NC(c1cc(Cl)cnc1O)=O)S2 C1(NC(CCc2cc(C)no2)=O)CN(C(=O)C(O)CC(C)C)C2CCCC12 C(=O)(CC(C)(C)N(C(=O)CCC1CCC1)C)NCC(CC)CO N1(C(COCC)=O)CC(NC(c2nc(C)n(-c3ccccc3)n2)=O)C(CC)C1 C(=O)(C(CC)C(C)(C)CC)NCc1c(C(=O)NC(CCCC=C)C)con1 C1(C(=O)NCC2(C)CC(C)(C)C2)CCN(C(c2ncc(F)cc2F)=O)C1(C)C CC1Cc2cc(C(=O)NCC3CN(C(c4ccc(O)nc4)=O)CC3C)ccc2O1 C(N=c1cc(C)c(S(=O)(=O)NCC(C)(C)CCC)c[nH]1)C1C(C=C)C1 N(C1CS(=O)(=O)c2ccccc21)C(CC1C(C(=O)OCC)C1)=O n1(CC)nc(C(=O)NC2CN(C(C3CCC(C(N)=O)CC3)=O)CC2C)c(C)n1 N1(C(c2cc(CCC)on2)=O)CC2CCC1CN2C(=O)C1=NOC(C)(C)C1 C(C)(CCCC(=O)N1CCC(C(C)(C)O)C1)NC(C(CC=C)C)=O C(C(=O)N1CCCC(CNC(c2nc(Br)c[nH]2)=O)C1)(C(C)C)NC(C)=O c1(C(C#N)NC(C2(F)CN(C(=O)C3CC3)C2)=O)ccccc1Br C1(CC)CN(C(=O)CCCNC(=O)OC)CCN1C(=O)CC(C)c1ccccc1 Cc1ccc2c(c1)CN(C(C1(NC(=O)CC(=O)NCC3CC3)CC1(C)C)=O)C2 O=C(N=c1ccn(Cc2cccs2)[nH]1)c1ccc(=O)n(C2CC2)c1 C(CCCCCCCO)=CC(=O)NC(Cc1csc(Cl)c1)C(=O)O C1(NC(c2occ(C)c2)=O)CN(C(c2ccc(O)cc2Br)=O)CC2(CC2)C1 C(N=c1ccnc(N2CC(C(N)=O)CC(C)C2)[nH]1)C1(OCC)CC1 N1(C(CC(C=C)C)=O)CCOCC(C)(CNC(c2c(Cl)c(C)nn2C)=O)C1 c1(CCNC(C(c2ccco2)NC(CC(C)n2cccn2)=O)=O)ccncc1F N1(S(CCC)(=O)=O)CCCN(C(c2ccc(F)cc2OCC)=O)C(C)C1 c1(CN2CC(c3cc(N(C)C)nn3C3CCCC3)C2)ccc(N)c(N)n1 c1(OC)cc(C(=O)NC2CC3CN(C(=O)C(C)O)CC23)c2c(c1)CCO2 O=C(C1CCOc2ccccc21)NCC1(CNC(C23CCCN(CC2)C3)=O)CC1 C1(C(=O)NCc2cccc(C)c2)CCC2(CC1)NC(=O)N(C)C2=O C(=O)(C1CCc2ccccc21)N(C1CCN(C(=O)CCOC)CC1)CC c1(SCC(=O)NCC(C[N+](C(C2CCCC2(C)C)=O)([O-])NC)OC)ccccc1Cl Nc1c(C(=O)NCCCN(CCO)C(c2cncnc2)=O)cccc1F c1(OC)ccc(Cl)c(C(N2CCCC2C(N2CC3C(C2)C3(C)C)=O)=O)c1F c1(OCC(=O)NCCCC(C)NC(CSCCC)=O)ccc(Cl)c(C)c1 CC1NC(=O)C2=C1N(c1ccc(Br)cc1)C(=O)NC2c1cc2c(Cl)cccn2n1 C1(N(C(=O)C(Cl)=CCl)C)CCCN(C(c2cccnc2S)=O)C1 Cc1ccc(F)cc1CC(=O)NC1C2CN(C(C34CSCC3C4)=O)CC12 N1(C(c2c(C)csc2)=O)CCC(C)C(CC(=O)NC(Cc2ccco2)CO)C1 CC1CCN(C(c2cccc(Cl)c2)=O)CC1N(C(=O)CC1CC2CCC1O2)C N#Cc1cc(S(=O)(=O)N2CC3(CN(C(c4cnncc4C(=O)O)=O)C3)C2)ccc1Br C1(C(=O)NCc2c(C)occ2)CC(=O)CN1C(C1CC(=O)C1(C)C)=O CC1(C(F)(F)F)c2cc(Br)ccc2CCN1C(=O)C1=NOC2CCCC12 c1(C(N2C(C)CC(CNC(=O)CCCCC3CC3)C2)=O)ccc(N=S(C)(C)=O)s1 c1(C(C)(C)C)nc(CNC(=O)C(N2CCC(OCCF)C2)=O)cs1 C1(C(=O)NCC(C)(C)OC(C)C)CC12CCN(C(=O)CC1CCCCC1)C2 C(=O)(CCCCCCNC(N)=O)NC(C)(C)C.C1(=O)CC(=O)OC(C)CN1 CC(C(=O)NCCCC1CN(C(c2cc(C(F)(F)F)c[nH]2)=O)CCO1)S(C)(=O)=O C(c1ccc(F)cc1)=C(C)C(=O)NCC(C)NC(c1ccc(N)cc1F)=O C12(CNC(CCc3cn(C)nc3)=O)CCC1CN(C(c1ccnc(O)c1F)=O)C2 N1(C(C2N(C)C(=O)CC2)=O)CCC12CN(Cc1ncccc1O)C2 N1(CCC2C(C)CCCC2)CC2(C)CC1CO2 N1(C(C#CC(C)C)=O)C2CCC1CC(N(C(=O)CCC1CC1(Cl)Cl)C)C2 N1(C(CNC2CC(OC(C3CCN(C)C3C3CC3)=O)C2)=O)CC(O)C(C2CC2)C1 Cc1cn2c(n1)C(C(=O)NC1CCCC(NC(=O)CCc3cnoc3)C1)CCC2 C(C(=O)N(CC(C)OC)C)(C(C)(C)O)NC(C1(CC=C)CCCC1)=O c1(CC(=O)NCCNC(C(C)OCCOCC)=O)cc(F)ccc1Br CCC(C)C(O)C(=O)N1CCC(n2cc(C(C3CCOC3)C)nn2)C1 c1(CC(=O)NCCC(C)(C)NC(CC(C(C)C)C)=O)nc2c([nH]1)CCCC2 c1(OC)ccnc(C(=O)NC2(C)CC(NC(=O)CCc3csc(C)n3)C2)c1OC c1(CN(c2cncs2)S(=O)(=O)Cl)ccco1 N1(C(=O)CC2(CCNC3CCOC3)CC2)CCC2(C(=O)Oc3ccc(F)cc3)CC2C1 CC1(NC(=O)CCc2cc[nH]n2)CCN(C(C2CC2C(F)(F)F)=O)C1 C=CCCC(C(=O)N1CCCC(C)C1)NC(c1cc(C)cc(F)c1)=O C=CC1(C(=O)NC2CC2CNC(c2cc(N)ccc2Br)=O)CCCCC1 C1(C(=O)NCC2(CCNC(C(CSC)(C)C)=O)CC2)Cc2cc(C)c(C)cc2O1 C1(C(N(c2ccc(Cl)cc2)C)=O)CCC(C)(C)N(C(=O)C2=CCCOC2)C1 N1(C(C(CCOC)(C)C)=O)CCc2c(c(CNC(C3CCC3OC)=O)nn2C)C1 c1(C(=O)NC2CCCCCC2NC(C2CCCS2)=O)ccc2nonc2c1 Nc1ccc2[nH]c(C(=O)NCc3cccc4c3NCC4)cc2c1 N1(CCc2cn(CCSCC3N(C(C4CC=CC4)=O)CCC3)nn2)CCCCCC1 c1(CNC(C(c2ccoc2)NC(CC(C)=C(C)C)=O)=O)ccc(F)c(C)c1 C1(NC(C2C(CC)CCO2)=O)CN(C(c2coc(Cl)n2)=O)CCC1C C(N=c1cc(C)nc(C)[nH]1)c1ncc(-c2c(F)ncc(C)c2)nc1 C1(O)(C(=O)NCC2CCC(NC(c3ccc(C)nn3)=O)C2)CCCC(C)CC1 C1(NC(c2c(Br)cn(C)n2)=O)CN(C(=O)COCCF)C2(CCCC2)C1 C1(CC(=O)NCC2(CNC(C(COC(C)=O)C)=O)CCC2)CC2CCC1O2 N1(C(C(CCSC)O)=O)CC2CN(C(c3ccc(-n4cc(C)cn4)cc3)=O)CC12 c1(CNC(C(CC2CCC2)N(C(C(=O)OC)=O)C)=O)sc(C)cc1C N1(C(C(C)n2cnnn2)=O)CCC2(CC1)CN(C(=O)CSC(F)F)C1COCC21 C1(F)(C(=O)NC(C)CCCCNC(C2CCC2(C)C)=O)CCCCCC1 N1(C(Cc2cc(NC(C3CCN(C)C3C)=O)no2)=O)CCC(C(C)OC)CC1 c1(CN2C(C(=O)N(CCO)Cc3ccco3)CCC2)cc(F)cc(Br)c1 c1(C(=O)NC2C(C)CN(C(=O)C3=CCC3)CC2C)ccc2nc(C3CC3)oc2c1 c1(C(N2CC3C(NC(CCCC(=C)C)=O)C3C2)=O)cc2c(=O)[nH]ccn2n1 Cc1csc(CC(=O)NC(C)CC(C)NC(=O)C(C)Cc2ccco2)c1 N1(C(c2cccc(CC)c2)=O)CCC2CN(C(C3(CC#N)CCCCC3)=O)C2C1 N1(C(=O)OC)C2CCC1CC(N(C)C)C2.C(CCC1CNC1=O)N Cc1c(C(=O)N(C(C)CNC(C2(Cl)CCCC2)=O)C)cccc1F c1(C(=O)NCC(=C)CCNC(=O)COC(F)(F)F)ccc(=O)n(C)n1 c1(C(=O)NCC(C)CNC(c2[nH]c(=N)sc2C(F)(F)F)=O)ccc(C2CC2)nc1 C1(CC(=O)NNC(=O)C2OCCO2)C(F)(F)C12CCOCC2 C1(C2CCN(C(c3cc4c[nH]cnc-4n3)=O)C2)(NC(c2cnco2)=O)CC1 c1(C(N2CCN(C(C3C4CC5C(C4=O)C35)=O)CC2CF)=O)nccn2ccnc12 N1(C(C2(CC)CN(C(=O)C(C)c3cccs3)C2)=O)CCC(C)(C2CC2)C1 c1(-c2ccc(C)cc2C)cc(=NC(C)c2[nH]c(C)nc2C)cc[nH]1 N1(C(c2c(C)oc(C#N)c2)=O)CC(C(=O)NCc2nnsc2CO)CCC1(C)C C12(C(N(CCN(C(c3cc(CCC)nn3C)=O)C)C)=O)CCOC1CCOC2 C(=O)(CC(C)NC(=O)CCC1CCC(NC(=O)C(C)N(C)C)C1)OC C(=O)(C#CC1(C)CC1)N(CC(=O)NC(CC(C)C)C)C1CCC1 O=S(=O)(NC1CC(c2ccccc2)C1)N1CCCC2(CCCNC2=O)C1 c1(C(=O)NCCC(C)NC(C=C(C)C(C)(C)C)=O)cnc(S(C)(=O)=O)s1 c1(C(C(=O)NC)NC2CC3CC3C2)cc(C2CC2)[nH]n1 N1(C(C(CC)CC)=O)CC2CCC2(CNC(=O)C=CS(C)=O)C1 CCCCC(O)CCC(=O)N1CCCOC(CNC(C2(C)CCN(C)C2=O)=O)C1 C1(CC)CCC(C(=O)NC2(C)CN(C(C3(CF)CCOCC3)=O)C2)CC1 C(=O)(C(C)(C)CCCO)NC1CN(C(c2c(=O)ccn(C)c2)=O)CC1(C)C N1(C(C2C(C)(C)OCC2)=O)CCC2(CCC2)C(NC(=O)C(=O)NCC(F)(F)F)C1 CC1CCC(NC(c2cc(=O)n(C)cc2Br)=O)CN1C(=O)C(C)CC(N)=O Cc1oc(C2CC2)nc1C(=O)NC1(CF)CN(C(C2CC3(CC3)CO2)=O)C1 CCCC(C)C(C)(c1nnnn1C)NCc1ccc(-c2cnco2)cc1 C1(NC(c2nc(C(C)=O)sc2)=O)CCCN(C(C2(C)CCCC2)=O)CC1F C1(CCC(N2CCCC2CO)=O)CCN(C(c2cncnc2C2CC2)=O)CC1 N1(C(CC)=O)CCC(NC(c2ccc(CN3CCCC3)s2)=O)C(F)C1 N1(C(C(C2CCCC2)OC)=O)CCCC(C)(NC(C2CN3CCCC2C3)=O)C1 N1(C(C(=O)NC(C)C)=O)CC(O)(C(C)(C)CNC(=O)CC2(C)OCCO2)C1 c1(C(=O)NCC(C)(O)C2CCCC2)ccc(C(N2CCC2C)=O)cc1.CN CCC(C(=O)N(CCC(=O)NCC(C)(C)N(C)C)CC)NC(N)=O Cc1ccccc1CC(=O)NC1CN(C(C2(CF)CC2)=O)CC1C(F)F c1(OCCCC)ccc(C(N2CCNC(NCC(C)CC)C2)=O)cc1OC C1(C(N2CCC(F)(CNc3nccc(OCCC)n3)C2)=O)CN2CCN1CC2C c1(C(=O)OC)c(NC(C2CC2C(=O)Nc2ccc(C(=O)OC)o2)=O)cncc1F c1(NC(C2C(NC(C(C(C)C)=O)=O)CCC2)=O)cccc(C#N)c1[N+](=O)[O-] c1(NCC2OCC(C)C2)[nH]c(=NCC2(C(F)(F)F)CC2)nc2c1ncn2C c1(NC(c2sccc2NC(C2CCCO2)=O)=O)c(F)cc(Br)cc1[N+](=O)[O-] c1(C(N(CCOCCCN(C(C2C(C)(CC)C2)=O)C)C)=O)cccc([N+](=O)[O-])c1 c1(CC(=O)NC2CCN(C(C3(C)CC=CCC3)=O)C2)c(F)cccc1F N1(C(C2C(=C)CC2)=O)CC2(C1)CN(C(=O)Cn1nc(C)c([N+](=O)[O-])c1C)CCO2 C1(CNC(Cc2c(C)nsc2)=O)(NC(=O)C(O)CC2CCCCC2)CCOCC1 c1(C(=O)NC2CC(CNC(C3(OC)CCSC3)=O)C2)cnc2c(c1)COCC2 c1(C(C)=O)cnc(Cl)[nH]c1=NC1CCN(C(c2nnn(C)n2)=O)CC1C C1(NC(CCCCC#C)=O)CC2(CCC(CNC(c3cnnc(C)c3)=O)CC2)C1 N1(C(C2CC(C(C)C)C2)=O)CCCC(N(C(=O)C(C)C2CCCC2)C)C1 c1(C(=O)NC(C)CCNC(=O)C2=CCCSC2)c(Br)cncc1[N+](=O)[O-] N1(C(C(C)NC(N)=O)=O)CCCC2(C1)CC2(F)F Cc1ccc(C(=O)NC2CCN(C(c3cc(C(N)=O)cn3C)=O)CC2)cn1 c1(C(=O)OC)cnc(NC=O)s1.c1(C(C)N(C)C)nnc(CN)s1 c1(C(=O)NC(CN(C(CCSCCCC)=O)C)(C)C)cc(CC(C)C)on1 N1(C(C2CCC(C(N)=O)CC2)=O)CCCC(C2CN(C(=O)C3=NNC(=O)C3)C2)C1 CN1CCC2C(CCN2C(C2(C)CN(C(C3CCC4(CC4)C3)=O)C2)=O)C1 C12(CC(=O)NCC(Cc3ccccc3)NC(C3(CC)COC3)=O)COCC(C1)C2 CCCCC(CNC(c1cnccc1N(C)C)=O)NC(=O)CC(=O)NCC1CC1 C1(C)(CC)CC(NC(c2ccc(C(C)(C)C)s2)=O)CN1C(=O)CC=C(C)C Cc1sc(Br)cc1C(=O)N(C1CCOC1)Cc1ccc(O)cc1 C(=O)(CCCC(=O)N1CCCC(N(C(=O)CC2CCCCC2O)C)CC1)OC C1(CC(=O)NC2CC(CN(C(=O)C3=COCCC3)C)CC2O)CCCC(C)(C)O1 C(CC1=CCN(C(=O)C(C)(F)C(C)(C)F)CC1)NC(C(C1CCOCC1)C)=O C1(CC=C)CCCCN1C(=O)CNC(=O)CC#N C1(NC(C2CCC(NC(=O)C3=CCCC3)C2)=O)CCC(C2CC2)C1 N1(C(Cc2cc(C)sc2)=O)CCC2(CC1)CC(NC(=O)CCC1CC1)CO2 c1(NC(c2cc(OC)ns2)C)cc(C)c(S(=O)(=O)N2CCCC(O)CC2)cn1 c1(CNC(CC(CN(C)C)(C)C)=O)ccc2c(c1)C(=O)N(C)C2 c1(C(=O)NCC(C)NC(c2cc(C(F)(F)F)c[nH]2)=O)cccc2cccc(O)c12 C1(C(=O)NCC2CC(C(C)(C)C)C2)(CO)CCN(C(=O)C(c2cccn2C)=O)C1 C1(OC)CC2(C1)CC(C(=O)NCC(C)(C)CCNC(=O)CC(C)C(F)F)C2 C1(NC(CSCCCC)=O)CCC2CC1CN2C(=O)CCCOc1ccccc1 CC1CN(C(=O)Cn2nnc(=N)[nH]2)CC1CNC(c1cn(C2CCCC2)nn1)=O C1(C(N2CCC(SC)CC2)=O)CN(C(=O)C=CC(F)F)C2(CCC2)C1 Cc1cc(CC(=O)NC2CCN(C(c3ccc4c(c3)CC4)=O)C2(C)C)cc(F)c1 c1(C(=O)NCC2CCC(C)N(C(=O)COC(C)(C)C)C2)cccc2[nH]ncc12 N1(C(c2ccc(C3C(C)(C)CC3)nc2)=O)CCOCC1(C)c1ccccc1 C1(C(=O)NCCC(C)F)C2CCCC2CN1C(=O)CC1CC=CCN1C O(N(CC)C(=O)C1CC=CC(NC(=O)CN2CCC(C)C2)C1)CC C1(CCCNC(C(COC)OC)=O)CCCCN1C(=O)C=C(C)c1ccco1 C1(C(=O)NC(CC(=O)OC)C)CCCN(CC(=O)Nc2ccccc2)CC1 N(C)(C(=NCCF)NCC1C2CCC(F)(F)C12)CCNC(=O)OC Cc1cccc2c1C(C)CC2CC(=O)N1CC2(C1)CN(C(c1ccsc1Cl)=O)C2 CCCC(C)(O)C(=O)NCC1CC(C(N2CCC(n3cnnn3)C2)=O)C1 O=C1CC2(CCC2)C(C(N2CCN(C(C3(CO)CCOC3)=O)CC2)=O)CN1 c1(C(=O)NC2CC(NC(=O)CCSC3CC3)C2)cc2ncccn2n1 C(N1CCC(P(C)(C)=O)C1)N1C(C)c2ccccc21 Cc1ccnc(C)c1C(=O)NC(C)C(C)n1cccn1.c12nc(c(C)o1)NC2=O C1(F)(CNC(C(n2ncc(C)c2)C)=O)CCN(C(=O)C(F)C(C)C)CC1 c1(C(=O)NC2CCC(N3CCN(C(C)=O)CC3)CC2)cc(O)c2ccsc2n1 c1(C(=O)NC2CS(=O)(=O)CC2NC(C2(O)CCCC2)=O)cnc2n1CCOC2 Cc1c(C(=O)N(CCC(=O)O)Cc2cccs2)sc2[nH]cnc(=S)c12 C1(C(=O)OCC)CN(C(=O)C(C)(F)n2c(C(C)C)nnc2S)CCO1 N1(C(CCNC(=O)OCC)=O)CC2C(CC(=O)N(C3(C)CC3)C3CC3)C2C1 c1(CNC(=O)NCCC2CCOC2)ccc(CO)c(Cl)c1 N1(C(C2C(C(=O)OC)C2)=O)CC(NC(c2cccc[n+]2[O-])=O)CC2(CCC2)C1 C(=O)(CCC(C)CNC)NCC1CCN(C(C(C)OCC=C)=O)CC1 C12CCCCN1C(=O)C1(CC1)NC2=O.C=CC(O)C(=O)NCc1ccccc1 c1(CC)cc(C(N2CCC(NC(c3ncccc3F)=O)C(O)C2)=O)cc(Cl)c1 N1(C(c2ccc(C)cc2C)=O)CC2CCCC1CN(C(=O)COC(C)C)C2 C1(CNC(C(c2ccc(F)cc2F)C)=O)CC2CN(C(C3CCCS3)=O)CC12 C1(C(=O)NCC2CN(C(C(CC=C)NC(C)=O)=O)C2)CCC2(CCOCC2)O1 c1(C(=O)NCC2CCC(NC(c3ccc(CC#N)cc3)=O)C2)cc2n(n1)CCC2 N1(C(Cc2c(C)n[nH]c2)=O)CC2CC1C2NC(C1CCC1C)=O c1(C2(C#N)CC2)cccc(C(F)(F)F)c1.c1(N2C(=O)NCC2)ccccc1Cl C1(NS(Cc2c(Cl)ccc(OC)c2)(=O)=O)CNCC1C1CCOC1 N1(C(c2n[nH]cc2Cl)=O)CCC(CF)(NC(=O)C(c2ccccc2F)(F)F)C1 c1(C(=O)NC2(CC=C)CN(C(c3nsnc3O)=O)C2)coc2c1COC2 CC(C)(C)CC(O)C(=O)NCCCCCCC(=O)NCCCC1(O)CC1 C1(CC(=O)NCCN(CCC)CCOC)CC2CCC1(NC(C1CCC1)=O)C2 C1(NC(C2CN(c3cn(CCCC#C)nc3)C2)=O)CCCC2(C1)CC2(F)F c1(C(=O)NC(C(=O)NC(C)CCCCCO)CC2CCC2)c[nH]c2cccnc12 c1(C(=O)NC2(C)CCC(NC(C3N(C)CCCC3)=O)CC2)ccn2c1CCC2 c1(C(N2CCC(C(=O)Nc3c(C#N)cc(Br)cc3)C2)=O)ccc(O)c([N+](=O)[O-])c1 N#Cc1csc(C(=O)NCC2CCCCN2C(c2cnc(N(C)C)s2)=O)c1 n1(CCC#C)c(N2CCC(CCCOC)CC2)nnc1-c1ccc(C)o1 O=C(C(F)(F)CCn1cc(-c2ccsc2)nn1)NCC1CCS(=O)C1 C1(NC(c2c(C)cco2)=O)CN(C(=O)COc2ccccc2Cl)CC1CO C1(CNC(CC2(CNC(=O)Cn3nccn3)CC2)=O)(SC)CC2CCCC12 CCC(CCCC(=O)NC(C)(CO)C1CC1)NC(c1coc(C(C)C)n1)=O c1(C(=O)NC2C(CC)N(C(=O)COC3CC=CC3)CC2)cnc2[nH]c(C)nc2c1 c1(C(=O)NC(c2ccc(Cl)cc2)C)cc2c(nc1Cl)CCS(=O)(=O)C2 c1(C(=O)NCC2CN(C(c3ccnc(C)n3)=O)C(C)C2)ccc(C(F)F)c(Cl)c1 n1(CCSCC)nnnc1C(c1ncoc1C(F)F)NC1(C)CCC1 c1(C(=O)OC)cc2cc(c1O)Cn1c-2ncc1.n1(C(C)C)nccn1 C(=O)(C(C)CCCC(C)C)N1C2(C(NOCCN(C)C)=O)CCCC2CC1 CC(C)CC(CNC(c1ccc(CCO)cc1)=O)NC(c1cc(Cl)n(C)n1)=O C1(NC(c2cccc(COC)n2)=O)CC(O)CN(C(C2C3CC4C(C3=O)C24)=O)C1 N1(C(C=C(C)c2ccccc2)=O)CC2CC(C1)CN(S(=O)(=O)C1CC1)C2 C(=O)(C1SCCc2sccc21)NC(CNC(c1cc(C)n(C)c1)=O)(C)C N1(C(CCC2CCCCN(C(c3cccc[n+]3[O-])=O)C2)=O)CC2CCC(C1)C2O C1(C(C)(C)NC(CNC(CC)=O)=O)CCN(C(=O)C(F)=C2CCCC2)C1 C(CC(O)C(=O)NCC1CCN(C(C2CCCC2c2nc(S)n[nH]2)=O)CC1)SC N1(C(c2ccc(C3CCC(=C)CC3)cc2)=O)CC2CCOCC2C1 Cc1nc(C=CC(=O)NCCC2=CCN(C(=O)OC(C)(C)C)CC2)[nH]c1C C12(C(N3CC(CNC(c4c(CC)oc(C)c4)=O)OCC3)=O)CCCN(CCC1)C2 N1(C(CCC2OCC(C)(C)C2)=O)CC(C)(C)C(NC(=O)COC(F)(F)F)C(C)(C)C1 n1(CC(=O)NCC2CC(Cn3cc(C(CC)(C)O)nn3)C2)ncn(C)c1=O C(C(C)(C)CC(=O)N(C1CCCN(C(=O)C(C)CC(N)=O)C1)C)OC N1(C(c2cccc(OCC(C)C)c2)=O)CCC2(CC(NC(C3CC3Cl)=O)C2)C1 C1(NC(=O)NCc2n(CC)ccn2)CCC(CCC(=O)NC(C)C)CC1 Cn1nccc1C=CC(=O)NC(C1CCOC1)CNC(=O)C(C)(C)n1cc(Cl)cn1 CCC(C)(C)CCCC(=O)N1CC(C(=O)NC(CO)CC(C)(C)C)C(C)C1 C1(C2CCC2)(C(=O)NC(C2CN(C(C3(CC(C)C)CCCC3)=O)C2)C)CC1 N1(C(CCC#C)=O)CCC2(NC(=O)Cn3ccc(Br)cc3=O)CCCC12 CC(C)CC(O)C(C)C(=O)N1CCN(C)CC1C(=O)NC1CCCC(C2CC2)C1 C1(C(=O)NCC2CN(CCN3CCCC3=O)C2)CC2CCC(C1)S2 C1(C(=O)NC2C(NC(=O)CC3(n4cccn4)CC3)C2)CCS(=O)CC1 c1(CC)ncc(C(=O)NC2CCCN(C(c3ccnc(Cl)c3N)=O)C2)c(C)n1 C1(CC)CN(C(=O)COC(F)(F)F)CCN1C(C1CCN(C)C(=O)C1)=O N=c1[nH]c(CC(=O)NCC2(CNC(C3CC3CF)=O)CC2(F)F)cs1 C1(NC(C(C)C)=O)CCN(C(C2(CF)CC2)=O)CCC1(F)F c1(C(C)OCC)nc(NC(=O)NCc2nc(CN(C)C)ns2)cs1 c1(C(=O)NC2CC(C(=O)NC3CN(C)CC3(F)F)C2)nccc2cc[nH]c12 C1(NC(=O)CCC=Cc2ccccc2)(CF)CCN(C(C2CCCCS2)=O)C1 c1(C(N2CC(C(=O)Nc3c(OC)cccn3)SCC2)=O)ccnc2ccccc12 C1(O)(Cn2cc(CC=C)nn2)CCCN(C(c2nc3sccn3c2Br)=O)C1 Cc1c(C(N2CC(CO)(NC(=O)Cc3cccs3)C2)=O)ccc(F)c1F C1(OC)(OC)CCN(C(CCC=C(C)C)C(=O)OC)CC1 C1(CNC(C(CC=CCC)C)=O)CN(C(c2cnc(CC)nc2O)=O)CC1(C)C CCCCC(CNC(=O)CCS(=O)(=O)N(C)C)NC(=O)CCCc1ccccc1 c1(C(=O)OC)cnc(N=S(C)(C)=O)c(Nc2ccc(F)cc2)c1 c1(C(c2n(CCC3(C)CC3)nnn2)N)noc2c1CCC2.C1(COCO)CCOC1 Cc1ccc(C(=O)COC(=O)CC2COC(C(F)(F)F)C2)cc1 N1(Cc2cc(C)on2)CCCC1C1CCCCN1C(c1cc(C2CC2)no1)=O N1(C(C(C)CF)=O)CCCC(C)C1CNC(c1cnn(C2CC2)c1)=O C1(NC(CCC)=O)C2CC1N(C(c1c(C)nc(C)n1O)=O)C2C Cc1cc(C(N2CC(C)(NC(C3CCC4CC3CO4)=O)C2)=O)cc(C)c1C N1(CC)CCCC2(CCCN(C(=O)CCCCc3ccc(C(F)(F)F)cc3)C2)C1 CC(C(=O)N1CC(C)(NC(c2cnn(C3CCOC3)n2)=O)C1)C(F)F N1(C(CCCCCOCC)=O)CCC2CN(C(C3CCS(=O)(=O)N3)=O)CC12 N1(C(c2c(C)n(C)cc2)=O)CCC(N(C(=O)CSCCC(F)(F)F)C)C(C)C1 C1(OCCC)CCCN(C(=O)C(O)C2(N)CC2)C1 Cc1nc(C(N2CCCC(NC(=O)C(c3ccc(Cl)cc3)C)C2)=O)nn1C c1(-c2n(-c3cccc(SC)c3)nc(C)n2)cnn2c(C)c(C)ccc12 c1(C(=O)OCC)ccccc1C(N1CC(C)(NC(=O)CC(C)SC)C1)=O C12(C(=O)NCCOCCNC(C3CCN(C)C3)=O)CCC(C(F)F)(CC1)C2 N1(CCOC)CCN(C(=O)C(C)=CCNC(=O)CCCn2cccc2)CC1 C1(CC(=O)NCC(CC)NC(=O)CNC(=O)CCc2ncccn2)CNC(=O)C1 N1(C(c2cn(C)cn2)C(=O)NC(C(=O)OCC)C)CCC2(CCC(O)C2)CC1 C1(CNC(COCCC#C)=O)CN(C(c2ccccc2CC#N)=O)CCO1 c1(C(N2CC(C)C(NC(c3cc4ncccc4s3)=O)C2)=O)coc(S(N)(=O)=O)c1 Cc1cccc(F)c1C(=O)N(CCC(C(C)C)NC(=O)CC1SC(=N)NC1=O)C C1(CNC(C2(C(C)(F)F)CCC2)=O)CC2(CC2)CN1c1nc(CC2CC2)ns1 CC1(C)CCC(O)(CNC(C2(CNC(=O)CCC3(C)N=N3)CCCCC2)=O)C1 C(=O)(CC(F)(F)C(F)(F)F)NCC12C(CN(C(c3c(N)c(O)ccc3Cl)=O)C1)C2 CC(C)(C)C(C#N)C(=O)NCCc1cc(C(=O)Nc2cccc3c2CCC3)no1 Cc1cnc(N2CCC(C(N)=O)CC2)c(S(=O)(=O)NC2CCCCNC2=O)c1 Cc1ccc(Cl)c(O)c1C(N1CCCC(NC(C2CNC(=O)N2)=O)CC1)=O c1(NCC2NCC(CC(=O)OC)OC2)ccc2nccn2c1C c1(C(N2C(CNC(CC(=C)C)=O)CCC(C)C2)=O)onc2c1CCCC2 N1(C(C2ON=C(C)C2)=O)CCC(CNC(=O)CC=CC(C)(C)C)C(C)C1 N#Cc1cc(C(N2CC3(C2)CN(C(C2C4C5CCC(C5)C24)=O)C3)=O)ccc1F C1(CC(=O)NC(C2CCN(C(C3CC(O)C3)=O)C2)(C)C)CC2CCC(C1)N2C c12c(cccc1Cl)NC2c1n(C)nnn1.c1(CC2CCC2)cncc(C(F)F)c1 C(=O)(CN=c1cc[nH]cc1)N(C)C.C12CCN(C13CCC3)C(=O)N1CCCC(C)C21 C1(C#N)(C(=O)NC(CN(C(c2cncc(OCC)c2)=O)C)C)CCCCCC1 C=CC1(CC(=O)NCC2(CC(C)C)CCC2)CN(C(=O)COC2CC=CC2)C1 C1(NC(c2cc(OC)n[nH]2)=O)CN(C(=O)CCCC(C)(F)F)CCC12CCC2 CC(C)C(C(=O)Nc1ccc2ncnn2c1)C(C)NC(=O)C(O)CN1CCCC1 N1(C(CCN(CCC)C)=O)C2CCC(C(=O)NCc3n[nH]c(C)n3)C1CC2 c1(N2CC(NC(C(Cc3ccccc3)OC)=O)C(C)CC2)ncn(C)c(=O)c1Br c1(-c2ncc(C)o2)cccc(C(N2CC(COc3ccccc3Cl)CC2=O)=O)c1 c1(OC)ccccc1OCCC(=O)NCC1(O)CCN(C(=O)C(C)NC(N)=O)C1 C1(C(N2CC(CCNC(c3c(C)nsc3N)=O)C(C)C2)=O)CCc2c[nH]nc2C1 N1(C(C2(OC(C)=O)CC2)=O)CCC(O)(CNC(=O)CC2CCC(=O)NC2)CC1 c1(NCc2ccc3ccn(C)c3c2)ccnc2c1ccn2C N1(C(C=CCN(C(c2cc(CC)no2)=O)C)=O)CCN(C)C2CC12 C(=O)(C1=CCCN(C)C1)N1CCC(C(=O)Nc2cccc(C#C)c2)CC1C(C)C C1(CC(=O)NCC2(COC)CCCO2)CC(C)N(C(c2c[nH]cc2C)=O)C1 CC1(C)CC1(NC(c1cccnn1)=O)CN.c1(C(C(=O)O)N)ccccc1 C1(N(C(CSCC=C)=O)C)CC2CCC(C1)N2C(c1cnc(N(C)C)o1)=O Cn1c(C(N2CCCC(CCCCNC(=O)C(F)C3CCC3)C2)=O)ccc1C#N N1(C(c2c(C(C)C)n[nH]c2)=O)CC(O)CC1(C)C(=O)NCCCc1cccnc1 Cc1ccnc2c(S(=O)(=O)Nc3ccc(N4CCC(C)C4)cc3)cccc12 C1(C(=O)NCCC(=O)NCCC(CCC)C2CC2)CN(C)CC(C)O1 C=Cc1cc(C(=O)NCC2CCN2C(c2cc(CC)ccc2N)=O)cc(F)c1 c1(C(C2(c3ccc(Cl)cc3)CCC2)NCC(C)SC)ccccc1F C1(NC(C2CCN(CC)C2)=O)CC2CCC1CC2NC(=O)C(C)NC(N)=O c1(C(N2CC(CCNC(C(C)(CO)OC)=O)OCC2)=O)cc2ccsc2c(O)n1 Cc1coc(C(N2CC(OCCNC(=O)CN(C3CCCCC3)C)C2)=O)c1C CCC(C)C(C(=O)NCC(C)(C)CNC(=O)C(CC)C(C)C)N(C)C C1(CCC(C)(C)NC(=O)CSC2CC2)CCN(C(=O)C(F)C2CCC2)CC1 N1(C(C2N(C)CSC2)=O)CC(F)(F)CC1(C)CNC(=O)CC1CCOCC1 CCC(C)C(C(=O)NCCN(C)C(c1ncc(C)cc1OC)=O)NC(=O)OC N1(C(C(CC(C)C)NC(CCCOC)=O)=O)CCC(C2CC2)CC1 CC1C(C(=O)NNC(=O)CC2CCC(COC(C)(C)C)O2)CCN1C(=O)OCC S(=O)(=O)(c1cccc(Cl)c1Cl)N1CC(NC(c2scc(C)n2)=O)C(F)(F)CC1 c1(OCC)ccc(N)c(C(N2CCCC2C2(NC(c3ccns3)=O)CC2)=O)c1 c1(C(N2CC(NC(c3c(OC)cccc3Br)=O)C(C)C2)=O)nc2ncccn2n1 C1(NC(c2c(CC)[nH]cc2)=O)CCC12CN(C(c1cc(C(N)=O)co1)=O)C2 C(=O)(C1=CS(=O)(=O)CCC1)N1C(CCNC(c2cnc(SC)n2C)=O)CCC1 S(=O)(=O)(c1ccc(NC(C)(C)CO)c(F)c1)N(C(CSC)C)C C1(CNC(=O)CC2(NC(c3cn(CCO)nn3)=O)CCC2)CC1C1CCCC1 [N-]=[N+]=NC1CCC(C(=O)NCC2CCCOC2c2ccccc2)CC1 CC1CCC(C(=O)NCC2CCN(C(=O)C3=CCCC3)C2(C)C)C(=O)N1 C1(O)(C(C)NC(Cc2ccc(CCC)cc2)=O)CCN(c2nnnn2C)CC1 c1(C(N2CCC(F)C2)=O)cc2ccc(-c3ccc4c(c3)CCOC4)cn2n1 C1(NC(c2nc(C)[nH]n2)=O)CC(=O)N(C2CN(C(=O)Cc3ccc(Cl)cc3)C2)C1 N1(C(CCC=CC(C)C)=O)CCC(NC(=O)COc2ccsc2)CC1C C(=O)(C1=CCC2CCC1N2C(c1ccc(N)cn1)=O)NCc1c(C)nn[nH]1 C=CC(C)N=c1[nH]c(=N)[nH]c(=NCCC(=O)NCC(=O)NCC)[nH]1 c1(C(=O)NCC(C2CCC2)NC(C(C)O)=O)ccc(S(C)(=O)=O)cc1Br Cc1cnn(CC(=O)NC(CNC(C2(N3CCOCC3)CCC2)=O)CO)c1 C(=O)(C1NCCc2nc(C)ncc21)NC(c1ccc(COC)cc1)C C1(NC(C(C2CN(C(C3CCC3)=O)C2)OC)=O)CCOC(C)(C)C1 C(C(CC1CC1)C(=O)NCCc1cn(C)nn1)NC(C1(C(C)=O)CC1)=O c1(C(C(=O)NCC2(OC)CCN(C(CCC#C)=O)C2)C)cc(C)cc(F)c1 c1(-c2cn(C3CN(C(CNC=O)=O)C3)nn2)ccc(CO)c(F)c1 O=C(C(F)Cc1ccccc1)NC1(CNC(C2CC2(Cl)Cl)=O)CC1 C1(NC(C2(CNC(C(C)n3cnnn3)=O)CC(C)(C)C2)=O)CC2(CCC(O)C2)C1 C=CCC(CNC(c1scnc1C)=O)NC(=O)CC1CCCCO1 C(c1ccccc1)=C(OC)C(=O)N(CC(C)NC(=O)CCc1nc(C)no1)CC c1(C(=O)NCC2C(C)CCN2C(=O)CCC[N+](=O)[O-])ccc2cc[nH]c2c1 C(=O)(C(C(C)(C)O)NC(C1CCCS1)=O)NCCC(CCC)O C1(CCNC(CC=C=C)=O)CCCN(C(=O)CCc2ccc(CC)cc2)C1 c1(COC)nccc(N2CCC(CN(C)C(c3ccc(C)cc3)=O)CC2)n1 N1(C(CCCC#N)=O)CCCCCC1Cn1cc(C(C2CC2)OC)nn1 C1(C(=O)NCC2(C(=O)NCC3=CCN(C)CC3)CC(=C)C2)CCCCC(=O)C1 CC1(C#CC(=O)NCC(O)CNc2ccc([N+](=O)[O-])c(O)n2)CCCO1 C1(CNC(=O)CSC)CCCCCN1C(=O)Cn1cc(Cc2ccccc2F)nn1 c1(NC2CCOC2)ccc2n[nH]cc2n1.c1cc2cc(c1)CO2 c1(OC)cc(C)c(OCC(=O)OC(C(F)F)C2CCCO2)cc1C Cc1ccc(CNC(C2CCN(C(C3COCC3(C)C)=O)C2C)=O)cc1 Cc1cc(F)c(NC2CC3CC2CN3)cc1N N#Cc1ccsc1C(N1CC=CC(NC(=O)CN2CCC(C(F)(F)F)CC2)C1)=O C1(C(=O)O)(Nc2nnc(C3CC3)s2)CCC2CCCC12.CCCN1C(=O)N1 C1(NC(C2C(C=C(C)C)C2(C)C)=O)CCCN(C(=O)CC2(OC)CCCC2)CC1 c1(C(N2CCN(C(CC3(C=C)CC3)=O)CC2C)=O)cc2oc(Br)cc2s1 CN1CCOC2CN(C(C3(C)C=CCN3C(C3CC3c3ccccc3)=O)=O)CC12 C(CCCC(c1ccc(Cl)cc1)NCC(C1(CO)CCCC1)=O)OC Cc1cc(S(=O)(=O)N2CCC2C(=O)Nc2cc(C(C)C)nc(Cl)c2)c(F)cc1Cl c1(C(N(C2CCN(C(=O)C(C)(C)CF)C2)CCC)=O)ccc(C(C)=O)cc1F C1(C(=O)NCCNC(=O)CNC(=O)NCc2ccco2)C2COCC12 C1(CC(=O)N(C)CC2CCCN2C(=O)CCn2cncn2)COC2(CCC2)CO1 C=CCC(CC)C(=O)N1CC2C(NC(c3cc(CSC)ccc3OC)=O)C2C1 C=CC(C)(CC)C(=O)N1CCCC(CCNC(=O)CCCOC2CCOCC2)C1 c1(OCC(N2CCN(C(C3(C)CC3)=O)CC2CCO)=O)ccc2c(c1)CCCC2 c1(C(=O)NC(C2CCOC2)CC)ccc2c(c1)NC(=O)CCS2 c1(C(=O)OC)ccc(C(=O)N(CC(C)NC(C2CCCC(O)C2O)=O)C)c(F)c1 C1(NC(COCCCC)=O)CCCOC12CCN(C(=O)C(C)(C#N)CC)CC2 c1(CCC(=O)N(C(C)CCNC(=O)CCC[N+](=O)[O-])C)c[nH]c2ccccc12 c1(C(=O)NCC(C)N(C(Cc2scc(CC)n2)=O)C)ccc(S(C)=O)cc1 CC1CCCC1N(C)C(c1cn(CCNC(=O)CCNc2ncccn2)cn1)=O c1(C(N2CCN(C(c3n(C)c(C(F)(F)F)cc3)=O)CC2)=O)cc(Br)cnc1O CCC(CC)C(c1nnnn1CCSC)NC(c1cc(Cl)ccn1)C c1(N2CC(C(N3C(C(=O)OC)CSCC3)=O)OCC2)nc(C)ncc1C#N c1(C(=O)NCc2ccccc2-n2cc(Cc3nn[nH]n3)nn2)cccc(Cl)c1 c1(-c2cn(C3CC(NC(C4(Br)CC4)=O)C3)nn2)ccc(C2CC2)cc1 N1(C(c2c(C)nc(C3CC3)[nH]2)=O)CCC(C2(O)CN(C(c3ccco3)=O)C2)CC1 N1(C(c2cnc(NCC)c(Cl)c2)=O)CC2(COC(CNC(=O)C(C)C(C)C)C2)C1 c1(OC)ccc(C(=O)N(C)CCN(C)C(C2CCCC(F)C2)=O)cc1OC(F)F c1(C(=O)NCC(C)N(C)C(C2(n3ccnn3)CC2)=O)cc2c(F)c(F)ccc2[nH]1 C(CC(CC)C(=O)N1CCC(F)(CNC(=O)CC)C1)=CC.c12cccc(c1)N2 c1(C(N(C(CC)CNC(c2c[nH]nc2C(F)F)=O)C)=O)cccc(C#N)c1C CC1CN(C(=O)CCc2ccc(C3CC3)cc2)CC1CC(=O)NC(=O)CCF N1(CC(N2C(C3(NC(=O)C=CCF)CC3)CCC2)=O)C(=O)CNC1=O c1(COCC)cc(C)on1.C1(=O)C(CC2CC2)N1.C1(CC(=O)NC)CC(F)C1 c1(OC)nc(Br)cnc1NC(C1C(O)CCN1C(c1ccc(O)cn1)=O)=O c1(NC(C)=O)cccc(C(N2CCCC(C3CC(N)CCO3)C2)=O)n1 c1(C(=O)NCC(CC)NC(c2ccn(C3CCC3)n2)=O)cnc(C(C)(C)C)o1 N1(C(CNC(C)=O)=O)CC2(CNc3nc(NC(C4CCCO4)=O)sc3)CC1C2 N1(CCC(=O)NCC(=C2CN(C(Cc3ccn(CC)n3)=O)C2)F)CCN(C)CC1 C1(CCNC(c2c(C)coc2)=O)CC(F)(F)CN1C(c1n[nH]cc1Cl)=O c1(OC)cncnc1C(=O)N(C(C)CCNC(=O)CCc1nnc(C(C)C)o1)C C1(CC(=O)N(C(CCCC)C)C)CN(C(C2(CC)CC2)=O)CCO1 c1(C(=O)NC(C2CCN(C(=O)C(F)=C3CCCC3)C2)C)cccc2c1CC(=O)N2 C1(CC=C)(NC(=O)C(=O)NC2CC2)CCN(C(c2c[nH]nc2C(C)C)=O)C1 C(=O)(CCS(C)(=O)=O)NC(C(=O)NCC(=C)Br)Cc1cc[nH]n1 c1(C(=O)NC(CNC(C(CC)CC2CCCC2)=O)C(C)C)cc(N)cc(F)c1 c1(C(N(C2CCN(C(C3OCC(C)C3)=O)CC2)C)=O)ccc(Br)nc1O c1(C2(NC3C(NC(=O)C=Cc4cc[nH]n4)C3)CC2)ccc2ccccc2c1 c1(CN(C2(O)CCOC2)C(C(N)=O)C2CC2)cc2c(cc1OC(F)F)OCO2 CC1(C)OCC2CC12C(=O)NCC1CCN1C(c1nocc1Cl)=O c1(C(=O)NCC=CCNC(CC2(C(=C)F)CCC2)=O)cc(C(C)C)ncc1Br CCCC(C(=O)NCCF)OC.C1(=O)CN1CC(N)=O c1(C(=O)NC2CC(CC(C)C)OCC2)cc(S(C)(=O)=O)ccc1F CC1CCCCN1CCC(=O)N(C1CCCCC1NC(c1ccnnc1O)=O)C CC1(C(=O)NC2CCCC2NC(C2(C3CCCO3)CC2)=O)CC1(F)F c1(N2CCC(C3N(C(C(CCC)C)=O)CCC3)C2)cc(C(C)C)nc2ncnn12 c1(C(N2CCN(C(C#CC3(CC)CC3)=O)C(C)CC2)=O)ccc2oc(=O)oc2c1 N1(C(c2c(C)nccc2)=O)CCCN(C(=O)C(F)CC2CCCCC2)CC1C C(=O)(C(=O)N=c1ccn(C(=O)N(c2cccc(Cl)c2Cl)c2ncc[nH]2)c(O)n1)NC CC1C(NC(c2cc3c(F)cccc3s2)=O)CC2CCC1N2C(c1cnns1)=O c1(CN2C3C(C(=O)Nc4ccc(CO)o4)C(C3)C2)cccc2cnccc12 Cc1ocnc1C(=O)NC(C(=O)NCCC(F)(F)Cl)c1ccco1 C=CCC(CC)C(=O)NC(C)(C)CCCNC(c1c(-c2ccsc2)noc1C)=O C1(NC(CN(C(=O)OC(C)(C)C)CCc2n(C)ncc2)=O)COCCC1C1CC1 CCC(C(=O)NCC1CC(NC(C2CCCN2C)=O)C1)C(C)(C)CC N1(C(C2N(C(C(C=C)CC)=O)CCC=C2)=O)CCCC2(CCOC2)C1 Cc1[nH]nc(C(N2CCC3C(NC(C45C(=O)C6CC4C5C6)=O)C3C2)=O)c1[N+](=O)[O-] C123CC(CO1)(C2)NC3=O.C(=O)(C(CN(C)C)N1CCCCC1)NCCOC CC(=O)CCCCC(=O)N1CC2C(CNC(c3ccnc(CO)c3)=O)C2C1 C(=O)(CCC(=O)NC1CCCCC1NC(=O)C(C)(CC)OC)NCC(=O)OCC C1(C)(C(=O)NCC(CC(C)C)NC(CC2ON=C(C)C2)=O)CCCS1(=O)=O c1(C(N2CCCC(C(=O)NC)C2C)C(=O)NC(CC)(C)C)ccc(C)c(C)n1 CCC(COC)C(=O)N1CC(C(=O)Nc2cscc2C)(CC)C1 C(=O)(CCC(C)(C)F)NC(C1(O)CCN(C(C(C2CCC(C)O2)F)=O)C1)C N1(c2cccc(-c3cscn3)c2)C(=O)NC(C2CCC2)C1=O.C=CC c1(C(N(C(C)CNC(C2CC=CCC2)=O)C)=O)ccc(CO)cc1F Cc1oc(C(C)C)nc1C(=O)NCC1(F)CC(NC(=O)OC(C)(C)C)C1 c1(CNC(CC(C)C)=O)cnn(C)c1C(N1CCOCC1CC1CC1)=O c1(C(=O)NC2C(N)C2)ccc(O)c(F)c1F.Cc1cnc(C=CC=O)[nH]1 C1(C)(c2cn(CCCCC=C)nn2)CCCN1C(=O)C(C1CCCCCC1)C N1(C(c2cc(C(CC)CC)no2)=O)CC2(CCN(C(C3(F)CCOC3)=O)C2)C1 c1(C(=O)NCCn2cc(C(=O)NCC(=O)OCC)nn2)cc2cc(C)ccc2s1 N1(C(c2c(CC)n[nH]c2)=O)CCCCC1CNC(=O)Cc1nonc1C C1(C(=O)OC)Cc2c[nH]nc2CN1C(=O)N(C)Cc1ccc(SC)s1 C1(C(=O)NCCC2(CNC(C(C)OC3CC3)=O)CCCC2)CCCC12CC2 c1(C(=O)NC(CNC(c2nncs2)=O)CO)cc(Br)n[nH]1 c1(C(=O)NC(C)(CNC(C23CSCC2C3)=O)CO)cccc(C(F)F)c1F O=C(C(O)CC(F)(F)F)NCC12CCC(CC1)N2C(=O)CC1CCCO1 C1(C(=O)NCC2CCC(NC(c3cc(=NC)[nH]cc3)=O)C2)CC2C=CCC(C1)C2 COn1cnc(C)c1C(=O)NC1CCCCC1CC(N1CC(O)(CN(C)C)C1)=O Cc1cc(F)ccc1NC(=O)C(N1CCOCC1c1nc[nH]n1)C1CCOC1 c1(CC(=O)OC)cc(=NC(C)C2CCC2)[nH]c(OC)n1 CC(Cc1ccncc1)C(=O)NCCC1(NC(c2[nH]ncc2Cl)=O)CC1 Cn1nc(CNC(C2CCS2(=O)=O)=O)cc1C(=O)NCCn1ccc(=O)cc1 c1(NC(c2cc(CNC(Cc3scc(C)c3)=O)oc2)=O)ccccc1O C1(CNC(C2C(C)CC=CC2)=O)CN(C(=O)CCCC#N)C2CCN1C2 c1(OC)ccc(Cl)c(C(=O)NC2CC(CNC(c3ccncn3)=O)C2(C)C)c1 N1(C(c2c(C)c[nH]n2)=O)CC(NC(=O)CC(O)C2CCCC2)Cc2ccccc21 C1(NC(C2(C3(C)CC3)CC2)=O)CCCC2CN(C(=O)Cc3ncccc3F)CC12 N1(C(c2c[nH]c(=NC)o2)=O)CCC(CNC(=O)C(C)CS(C)(=O)=O)C(F)(F)C1 CC(C(=O)NC1CN(C(C2CC(F)(CO)C2)=O)CC2(CC2)C1)C(C)S(C)(=O)=O Cc1cccc(C)c1C(N1CCC(C(F)C(=O)NC2CC(O)C2)C1)=O N1(C(Cc2ncc(CC)[nH]2)=O)CCCN(C(c2cccc(O)n2)=O)CC1 c1(C(N2CC(NC(C=CCOCCOC)=O)C(O)C2)=O)ccc(C(F)(F)F)c(N)c1 c1(NC(C2CC2F)=O)cccc(F)c1-c1ccc(OC2CNC2)nc1 C1(C(=O)NC(C(C)C)CN(C)C)CC(NC(=O)CC2CC2)C(O)C1 c1(C(=O)NCC(C)CNC(=O)COC(F)(F)F)ccc(OCCF)cn1 N1(C(COCCCC#C)=O)CCCC(NC(=O)C(=O)NCC(F)F)CC1 c1(CS(=O)(=O)NCc2cccc(C(=O)OC)n2)c(C)cccc1C CCC(CC)(CC)C(=O)NCC1CC(C)CCN1C(=O)CS(C)(=O)=O c1(NC)cccc(C)c1C(N1CCC(CF)(NC(c2coc(N(C)C)n2)=O)C1)=O N1(C(C=NOC)=O)CC(C)CCC1CNC(c1cc(C(C)C)on1)=O c1(NC(C2CN(C(=O)CCCc3ccc(Cl)cc3)C2)=O)ncc([N+](=O)[O-])cc1O Cc1cnn2cc(C(=O)N(CCCN(CCC(C)(C)C)C)C)cnc12 C1(C(=O)NC(c2cccc(OC)c2)C)CC2(CC2)CN1Cc1ncc[nH]1 C(C)(C)(CCCF)NC(C(CN(C)C)NC(C1CC(=O)CS1)=O)=O c1(C(C(=O)NCC(CN(C(c2c(CC)scc2)=O)C)O)OC)ccccc1OC c1(C(=O)NC(CC)CNC(=O)C2=NOCC2)cc(C2CCCCC2)n(C)c1C c1(C(=O)Nc2cc(C(=O)Nc3cc(COC)no3)sc2)ccc(C)cc1C C1(Cn2cc(-c3n(C)cnc3)nn2)CCN(C(C2CCNC(=O)C2)=O)CC1 CC1CC2CN(C(=O)COc3ccsc3)CC2N1C(c1cnc(C2CCC2)s1)=O N1(C(c2c(OC)ccs2)=O)CC2CCC(CNC(=O)CC3CCCC3O)C2C1 Cc1nc(-c2ccco2)sc1C(C)N(C(=O)CCc1nc[nH]n1)C C1(NC(c2c(C)coc2)=O)CC2(C1)CC(NC(c1ccn(C)n1)=O)C2 O=C(CS(=O)(=O)C1CC1)NCC1CCC(CNC(=O)COCC2CCOC2)C1 c1(C(N2CCC(N(C(CCOC)=O)C3CC3)C2)=O)ccc2c(c1)C(=O)OCC2 C=CCCCCCC(=O)N1CCC(F)(CNC(C2(C(C)(C)C)CCCC2)=O)CC1 C=CCC(CC)C(=O)NCC1CN(C(c2cc(C(C)C)cnc2O)=O)CC1C C1(C(=O)NCC(CNC(c2cccc(N)c2)=O)F)Cc2cc(F)cc(F)c2O1 Cc1nn(-c2ccc(F)cc2)c(C)c1CNCC#CCN1CCCC1 C#CC1CCCCN1C(c1cccnc1CNC(=O)C(C)CSC)=O c1(Cc2n(CCCOC)c(N(c3ccccc3)C)nn2)cc(C)cc(C)c1 CC(=O)C(C)CC(C)C(=O)NC1CCOC(C(=O)NCCCN2CCOC2=O)C1 C=CC1CC1C(=O)OCC1(CC(=O)OCC)CC1 c1(C(N2C(CNC(CC=C(C)C)=O)COCC2)=O)cnc2n1C(C)CCC2 N1(C(CCC=C)=O)CCN(C(=O)CSc2ccsc2[N+](=O)[O-])C2CCCCC12 CN1CCC(N2CC(C(N3CC4CC3C4CNC(C3CCO3)=O)=O)CC2=O)CC1 C1(C(=O)NC(C)CC(=O)O)C2CN(C(=O)CN3CC4CC4C3)CC12 c1(C(C)C)ccoc1C(=O)N(CC(C)CNC(C1CC(=C2CCC2)C1)=O)C c1(C(N(CCCNC(C2CC(C)SC2)=O)CCO)=O)ccc(-n2ccnc2)cc1 c1(CC)cccc(F)c1C(N1CCN(C(c2nn(C)cc2Br)=O)CC1C1CC1)=O C(=O)(CCCN=c1nccc[nH]1)NCC(CNC(C(C(C)C)(C)O)=O)C n1(C(C)C)ncnc1CNC(=O)C(CN(C)C)NC(=O)CCCn1ccnc1 c1(-c2n(C)ncc2)ccc2nnc(C(=O)Nc3scc(O)c3C#N)n2c1 C(=O)(C1=CCC(C)(C)CC1)NC1C(CNC(c2c(C)cc(Cl)cc2)=O)CC1 N1(C(c2nc(C)c(C)[nH]c2=O)=O)CCCCC(C2CN(C(C3CCOC3)=O)C2)C1 C1(OC)CCCCC1C(=O)NC(C)CCNC(=O)C(F)(F)C1(O)CCC1 C(C(=O)N(C)CCNC(=O)C)=CCOCCOC.C1(COCC)CC1C c1(C(=O)NC(CNC(C2C(C=C(C)C)C2(C)C)=O)(C)C)ccc(S(C)(=O)=O)s1 C1(C2C(=O)N2)CCN(CC=C)CC1.N1(CC(=O)NCC)CCCC(NC(C)=O)C1 O=S(=O)(c1ccc(NCCCSC(F)(F)F)cc1Br)NCC(C1CCCC1)O Cc1ccc2c(c1)CCN2C(C1CCC(F)CN1)c1ccccc1 N1(C(C2C(CC)CCCC2)=O)CC(CNC(=O)C(C)(C)C(C)C)C2(CCC2)C1 Cc1ccc(C(=O)NC(C)C(C(C)C)NC(=O)CC(C)(C)C2CC2)nc1C c1(C(=O)NCC2(NC(CC(CC)OC)=O)CCCC2)cccn2cncc12 C1(C(=O)NC2(CCC)CC2)C=CCN1C(=O)C=CCN1CCOCC1 C(=O)(C1=C(C)CC1)N1CC(CC(C)NC(C(c2cnn(C)c2)OC)=O)C1 C1(CC(=O)NCC2N(C(c3cc(C)c(Cl)s3)=O)CC(O)C2)CCCC(C)(C)C1 c1(N2C(C(=O)OC)CCC2)ccc(CN2CCOC(c3nnn(C)n3)C2)cc1 c1(C(=O)NC(CNC(C2OCCN(C)C2)=O)C2CC2)cc(F)cc(F)c1 c1(C(C(=O)NC2COC2)N(CCCC)CCCC)ncccc1C N1(C(C2(CC=C)CCN(C(c3cnn(C(F)F)c3)=O)C2)=O)CCC(=O)N(C)CC1 C(=O)(C(C)SC(F)(F)F)N(CCOCCN(C(=O)C=CC(N)=O)C)C C12(C(=O)NCCC3(O)CN(C(CNC(CC)=O)=O)C3)CCOCC1C2 C1(CC)CC(C(=O)NCCCc2ccsc2)CCN1C(=O)CC1CC(C)(C)CO1 C#Cc1cc(C(=O)NCC2CN(C(=O)CC=C=C)CC23CC3)cc(N)c1 C(=O)(C(O)C(C)CC)NCCN(CC(C)O)C(c1ccc(CCCCC)o1)=O N1(C(C2(CC)CC2(F)F)=O)CCC(CNC(C2CSC2)=O)C(C)C1 c1(C(N(CCCNC(C(C(CC)O)C)=O)C2CC2)=O)ncccc1N=[N+]=[N-] C(=O)(C1=C(Cl)CCOC1)N1CC(C(C)C)N(C(c2cc(Cl)ncc2O)=O)CC1 C1(CN=c2[nH]nco2)(CNC(c2ccnc(C3CC3)n2)=O)CC12CCC2 C(CC(C)N=c1nc(NC2CC2)[nH]c2c(C)nn(C)c12)N(CCC)CCO Cc1cc(C)c(C(N2CC(O)(C3CCCN3Cc3cn(C4CC4)nn3)C2)=O)cc1O N1(C(C2N(C)CCN(C)C2)=O)CCC2CC2(C(N2CCCCCC2)=O)CC1 N1(c2ncn(C)c(=O)c2)CCC2(CC1)CN(C(c1cc(C(C)(C)C)n[nH]1)=O)C2 N1(C(CCc2cc(C)no2)=O)CCN(C(C2CN(C)CCO2)=O)C(C)C1 N1(C(COC(C)C)=O)CCC2CCC12CNC(c1c(I)cnn1C)=O c1(CCC(=O)NC(C)CNC(=O)C(C)Cc2ccco2)ccc(Cl)cc1Cl N1(C(C(C)NCc2cc(I)ccc2C(=O)O)=O)Cc2ccccc2C1 CC(c1ccccc1C)=CC(=O)NC(C1CCCC1)CNC(=O)C#CC(C)(C)C c1(C(=O)NCC2(C)CCCN2C(=O)COCC2(F)CC2)ccn2cncc2c1 CCCCC(CNC(C1(SC)CC1)=O)NC(C1CCS(=O)(=O)C1)=O C=CCC(CC)C(=O)NC1(CC)CCN(C(=O)C(C)(C)c2cscc2C)CC1 N1(C(c2c(CC)[nH]nc2Cl)=O)CC2CCC(NC(=O)CNC(N)=O)(C2)C1 C1(C(=O)NCC2ON=C(CC)C2)CN(C(C2CCC(C)(C)C2)=O)C2(CCC2)C1 c1(OC(C)C(=O)NCC2C(Cn3cc(CO)nn3)C2(F)F)cccc(F)c1 N1(CC)CCc2cc(-c3ccnc(NC(=O)NC(C)CF)c3)ccc21 C(CC(C(=O)OC)OC(c1cnsc1C(=O)OC(C)(C)C)=O)OC C1(C(=O)NCC(CC(C)C)NC(=O)CCF)CCC(C)(C)CO1 c1(C(=O)NC(C(C)C)C(C)NC(c2c[nH]cc2C2CC2)=O)cc2sccc2n1C CC1CC(C(=O)NCC2CCC(NC(=O)COc3cccc(F)c3)CC2)C1(C)C Cc1noc(C)c1C(C)C(=O)NCCCN(C(=O)Cn1nnnc1C)CCO c1(Nc2scc(CC)n2)cnc2c(c1)c(C)nn2CC1C(C)(C)C(OC)C1(C)C c1(C(=O)NC(C)CCCNC(=O)OC(C)(C)C)ccnc(I)c1F Cc1nc(C)c(-c2nnc(N3CCCC(OCC(C)C)C3)n2CO)s1 N1(C(C2C(=O)OCC2)=O)CCCC12CCN(C(c1csnc1Cl)=O)C2 c1(C(=O)NCC2N(C(c3c(C)ncs3)=O)CC=C2)c(C)nn2cc[nH]c(=O)c12 c1(OC)c(C(N2CCC(O)C(C(=O)Nc3c(Br)cnn3C)C2)=O)cccc1F N1(C(c2ccc(N)cc2O)=O)CCC(C2CC2)(NC(=O)CSCc2cccs2)C1 N1(C(CCC(C)N(C)C)=O)Cc2[nH]nc(C(=O)NC(C)(C)CCCF)c2C1 C#CCCCC(C)C(=O)NCCC1(NC(=O)CCN2CCCCCC2)CC1 c1(CCC(=O)OC)cc(C(=O)N(C2CC(=O)NC2=O)C(C)(C)C)c(C)o1 C1(CN(C)C(c2snc(O)c2Cl)=O)CCCN(C(=O)C2=CCCO2)C1 N1(C(c2cccc(SCC)c2)=O)CC2CCCC2(NC(=O)CCF)C1 Nc1cnc(Nc2cccc(C(=O)Nc3ccccc3F)c2)cn1 C1(NC(c2cccnc2O)=O)CCCCN(C(C2CC(CC(F)F)C2)=O)CC1 c1(OC)ccc(SCCC(=O)NCC2CCCN(C(=O)CN(C)C)C2)cc1 C1(C(=O)NC(C(=O)NC(CC(=O)NC)C2CC2)COC)C2CCCCC12 N1(C(C(C)(CO)OC)=O)CCOC(C)(CNC(=O)CSC)C1 C1(CC(=O)NCC2(N(C(=O)C(C)(C)c3ccccn3)C)CC2)SC(=N)NC1=O C1(C(=O)NCCS(CC)=O)CCCCCN1C(c1n[nH]c2c1COC2)=O C1(C(N2C(CNC(c3ccnc(C)c3N)=O)CC2)=O)Cc2ccc(F)cc2O1 Cc1c(Cl)nc[nH]c1=NCC(O)CNC(c1cc2cccnc2s1)=O CC1(C)OC(=O)CC1C(=O)N(CCC(=O)NCC1CCC1(F)F)C1CC1 N1(C(c2cc(C)no2)=O)CCC(CCNC(c2ccc(O)c(N)n2)=O)CC1C Cc1nn(C)c2c(NCC3CCCC3(C)C)nc(N(CCO)CCOCCO)nc12 C1(C(=O)NCCCCC(C)NC(C(C)C2CCCO2)=O)CN(C)CC(C)O1 c1(C(=O)NC(C)CC2CN(C(=O)C=Cc3cnc[nH]3)C2)cnc2c(c1)CCCC2 N1(C(c2c(C)n[nH]c2)=O)CCOC(CN(C(=O)C(F)CC2CCCCC2)C)C1 C12(C(N(CC(=O)NC(C)(C)C)C)=O)CC(CO)(CN1C(C1CC3(CC3)C1)=O)C2 c1(C(N2CCC(NC(C3(OC)CC3)=O)CC2C2CC2)=O)ccc2c(n1)CCC2=O c1(NC(c2cc(C)no2)CC)cc(N2CCC(O)C(F)C2)nc(C(F)(F)F)n1 CN(C1CCc2c(F)cccc21)C(=O)NCC1CCC1CF C1(NC(c2cc(C(C)C)on2)=O)CCN(C(=O)COC(C)(C)C)CC1F c1(OCC(=O)NC(C)CCCNC(=O)CNC(c2ccco2)=O)ccc(Cl)cc1 N1(C(c2cn(CCNC(CSCC#C)=O)nc2)=O)Cc2ccc(O)cc2C1 c1(CCC)ncc(C(N2CCC(CNC(C3(c4nc[nH]n4)CC3)=O)C2)=O)s1 c1(N(CC(C)(C)C)CC)cc(N(CC(C)C#N)C)nc(C(F)(F)F)n1 c1(C(N2C(C)CC(CNC(c3cc(C4CCC4)[nH]n3)=O)C2)=O)cnc(O)cc1O C1(NC(Cc2cc(C)on2)=O)CC2CN(C(C3CCn4ncnc4C3)=O)CC2C1 c1(CNC2CCN(C(c3c(C)ccc(Br)c3)=O)C2)ccc(C)c(C#N)c1 c1(C(N(C2CN(C(C3CCC(C)(C)C3)=O)C2)C)=O)nc2ccccc2[nH]1 C1(CNC(C2CN(C(C)C)C2)=O)CCCCN(C(=O)CC(C)O)C1 N1(C(C(CC)F)=O)CCC2(CCC2)C(CNC(c2cccc3cccnc23)=O)C1 c1(C(N(CC2N(C(CC(=C=C)C)=O)CCCC2)CC)=O)nnn2c1C(=O)NCC2 c1(C(=O)NC(C(C)(C)C)CNC(C2CCCC23CCC3)=O)cccc(C#N)c1F c1(OC)ccc(C=CC(=O)NC2(CF)CCN(C(C3(C#N)CC3)=O)C2)cc1F c1(OC)cccc2c(N3CCCC3C(=O)O)ncnc12.n12cc(nn1)CSCC2 N1(C(C(C)(F)F)=O)CC2CC1CN2C(=O)CCc1ccc(F)cc1Br CC1(C)CC2(CO1)CN(C(C1(F)CCCN(C(=O)COc3cccnc3)C1)=O)C2 CC1CCC(C)(C(=O)NCC(C2CC2)NC(=O)Cn2nnc(=O)[nH]2)CC1 C(=O)(CC1=CCN(C(C2CC(F)(F)C2)=O)CC1)NC(C#C)C(C)C CC(CCS(C)=O)N(C(=O)C(=O)C1CC1)C CCC(C(=O)NCC(C(C)C)NC(c1nc(C)no1)=O)Sc1ccccc1 c1(C(N(CCC(C)NC(=O)Cn2nnc(=O)[nH]2)C)=O)coc(-c2ccccn2)n1 C1(C(=O)NC(CNC(C2CN(C3CCOCC3)C2)=O)C2CCC2)COC(=O)C1 C1(NC(c2cc(CO)[nH]n2)=O)CN(C(=O)Cn2ncc(Br)n2)C2CC12 c1(CC)ccccc1-n1nnnc1C(C)NCC1(c2ccnn2C)CC1.C1(S)CC1 S(=O)(=O)(c1cccc(Cl)c1)NN(CCNC(=O)NC1CC1C(F)F)C1CC1 C1(CNC(CCC#N)=O)CCCCC1NC(=O)Cc1nncn1-c1ccccc1 C=C1CCN(C(=O)CS(=O)CC)C(C(N2CCNC(=O)CC2)=O)C1 c1(C(=O)NCCCCNC(C2C(C)(C(=O)OCC)C2)=O)cnc(C2CCC2)s1 O=C(C1=NOC2(CCOC2)C1)NC1CN(C(c2ccc(F)c(C(F)(F)F)c2)=O)C1 c1(OCC(=O)NCC2CCN(C(C(CC)CC)=O)C2C)cc(C)ccc1F Cc1nccc(C(=O)NCC(C)(C)CN(C)C(C2(CN(C)C)CC2)=O)c1C C(CN=c1[nH]c2cccc(F)c2s1)CCNC(c1c(OC)nccn1)=O C(=O)(CCCC(C)C)NCC1(CO)CCN(C(c2c(C)nc(C3CC3)o2)=O)C1 c1(C(N2CCC(c3ccccc3)(N(C(CC=C)=O)C3CC3)C2)=O)c(O)cccc1Cl C1(CC(=O)OC)(CC)COCCN1C(=O)CC(N)CN(C)C Cc1nc2cc(C(=O)NCCC3CCCNCC3)c(F)cc2[nH]1 c1(C(N(C2(C3CN(C(=O)CN(C)S(N)(=O)=O)C3)CC2)C)=O)cc(F)c(O)c(F)c1 CCCCC(C)C(=O)NC1(C(=O)NCCOc2cccnc2)CCSC1 N1(C(C(=O)NCC)=O)CCCC(NC(c2oc(CC(C)C)nc2C)=O)C(F)C1 Cc1c(C(=O)NCC2(NC(=O)C=CCN3CCCC3)CC2)cncc1N c1(C(N2CCC(C(=O)NCc3cncs3)C2)=O)cc(Cl)nc2n[nH]cc12 CC1CCC(CC(=O)NCCCCCCN(C(=O)CCCN2CCCC2)C)OC1 CC1CCN(C(=NCCC2(C)CC2(F)F)NCCF)C1 C1(NC(C(C=C=C)C)=O)CCCN(C(=O)OC(C)(C)C)CC1 N1(C(C(C=C)(F)F)=O)CCN(C(c2ccc(C)n2CC)=O)C(c2ccncc2)C1 c1(C(=O)OC)ccc(C(N2CCN(c3cc(NC(C)=O)ncn3)CC2)=O)cc1F c1(OC)cccnc1C(=O)NC1CN(C(c2cc(C3(C)COC3)no2)=O)C1 C1(CNC(c2ccc(F)cc2CO)=O)CC2CCCC2N1C(=O)CCC1CC1 O(NC(=O)C(CN(C1CCC1)C(=O)CC1(C)CCOC1)CC1CC1)CC(C)C c1(CC)cccc(C)c1C(=O)NCC1(F)CCCN(C(C2ON=C(C)C2C)=O)C1 c1(C(=O)NCCN(C(=O)CC2CCCOC2)C2CC2)cnc2ccccc2n1 c1(C(=O)NC2CN(C(C3C(OCC)C3)=O)CC2C)cc2ccoc2cc1F O=S(=O)(c1cccc(=NC2CCCc3sccc32)[nH]1)N1CCOCC1C1CC1 c1(N2C3CN(c4nc(C)nc(-c5ccco5)c4)CC32)ncc2c(ccn2C)n1 N(C(=NCCCF)NCC1CCN(C(C)C)C1)Cc1c(OC(C)C)nccc1 C1(CNC(C(CC=C)CC)=O)CCC12CCN(C(=O)C(C)(C)CC)CC2 C(=O)(CC(F)(F)C(F)(F)F)N1CCC(Cn2cc(CCOC(C)=O)nn2)C1 N1(C(C2CC(NC(c3cccc(I)c3)=O)C2)=O)CCC12CCCCC2 c1(OC)csc(C(=O)NCC2CN(C(C3CN(C(C)=O)C3)=O)CC2C)c1OC c1(OC)cccc(CC(CC(=O)O)NCc2oc(CO)nc2C)c1 c1(C(=O)NCC2C(CC)CCN2C(c2sc(O)nc2C)=O)cccc(C#N)c1 N1(CC)CC(CNCC2(NC(c3ccc(CO)s3)=O)CC2)CC1=O c1(NC(c2n(CC)ncc2[N+](=O)[O-])=O)nc(Br)c2n1CCCC2 C(CNC(=O)C(COC)N(C)C)(CC(C)C)NC(C1(CC#C)CCOC1)=O C(=O)(CCCCc1cnn[nH]1)N(C1CN(C(=O)C=C(Cl)Cl)C1)C c1(C(=O)NCC(C)NC(=O)Cc2cnc[nH]2)cccc2nc(O)n(C)c12 c1(CC)[nH]nc(C(=O)NC2CC(CNC(=O)COCC3CCC3)C2)c1Cl C(C(F)(F)C(=O)N1CCC(F)(CNC(=O)C=CCN2CCCC2)C1)N(C)C C(C(C)(C(C)C)NC(=O)COc1ccc(Br)cc1)NC(C(CC)C)=O.COC C(c1cnn(C)c1)=CC(=O)NC1C(CNC(c2c(CC)noc2)=O)CCC1 C(=O)(C(CNC(c1ccc(O)nc1)=O)C(C)(C)C)NC(c1ccccc1O)C c1(C(=O)NCC2N(C(CC(CC)CN(C)C)=O)CCCC2)cc2c(nn1)CCC2 c1(CC)nocc1C(=O)NCCC1(CNC(=O)C=CC(c2cnn(C)c2)=O)CC1 C1(NC(c2[nH]cc(CC(C)C)c2)=O)CC2CCC1C(NC(C13CC(C)C1C3)=O)C2 C(=O)(CC(=O)N(C(C)CNC(=O)C(C)CNC(=O)C(C)C)C)NCC#C N1(C(C2CC(O)(CNC(c3n[nH]c(O)n3)=O)C2)=O)C2CCC1CC(O)C2 N1(C(=O)Nc2c(-n3ccnc3)ccc(C)c2)CCc2nc(C)sc2C1 c1(C(CNC(C(COCC)n2cc(CO)nn2)=O)=O)cccc(C(=O)O)c1F C=C(C)CCCC(=O)N1CCN(C2CCN(C(=O)C(C)C3CCCO3)C2)CC1 N1(C(C(C=CCCC)O)=O)CCC2(CCCN(C(c3cn(CC)nn3)=O)C2)C1 C(=O)(C(CNC(=O)C(CN(C)C)CC)CCC)NCc1cn(CC#C)nc1 O=C(CCCCCc1ccc(F)cc1)NC1CC(CNC(c2ccccn2)=O)C1 C1(C(N(C2(CC(=O)NC3(CC(N)=O)CC3)CC2)C)=O)CCC1(F)F C1(NC(C(=O)N(C)C)=O)CC2CN(C(C3CC3c3cnc[nH]3)=O)CCN2C1=O CCCCCC(C)(C)C(=O)NC(CC(=O)N1CC2(C)CC1CCO2)CC(C)C C1(NC(C(NOC)=O)=O)CC2CCC1C(NC(C1CC3COCC3C1)=O)C2 C=CCCC(CC(C)C)C(=O)N1CCC(NC(=O)CC2OCCC2(C)C)C1C N1(C(CC(=C)C)=O)CCC(NC(c2ncoc2CCCC)=O)CC1C Cc1ccc(C(N2CCCC(C)(NC(=O)C(C)C#N)C2)=O)cc1Br C1(CNC(C2C(C)=C2)=O)CN(C(c2occ3c2CCC3)=O)CCC1(C)C c1(C(=O)NCCCNC(C(C(CC)CC)OC)=O)c(O)nnc2c1CCC2 C1(NC(C(C)N2CCC2)=O)(CNC(C2(c3ccccc3)CC2(C)C)=O)CCCC1 c1(SC)nn(C)cc1C(=O)NCCC1CCN(C(C2OCC2(C)C)=O)CC1 N1(C(C#C)=O)CCc2ccc(NC(c3ccc(SC(C)C)c(C)c3)=O)cc21 C1(OCCc2cc(C)no2)CCC(F)(F)C1 C1(C(=O)NC(C)CC(C)NC(=O)Cn2cc(N)cn2)(CC)CCNC1=O C(=O)(C(C)(C)C(=O)N1CC(NC(=O)C=CCN2CCC2)C(C(F)F)C1)OCC N1(C(c2ccc(C(C)C)cc2)=O)CCN(C(c2cc(N(C)C)n(C)n2)=O)C(C)C1 c1(NC(C2CCCN2Cc2cc(Cl)sc2Cl)=O)c(Cl)ccc2cccnc12 C1(C(=O)NC2CCC(CNC(c3cc(C)oc3C)=O)C2)CC2CC2CC1C Cc1ccc(C)c(SCC(=O)NCCCCN(C)C(c2ccc(CSC)o2)=O)c1 c1(C(C)=O)cn(C)nc1C(=O)NC(C)CC(C)NC(C1CCC(C)O1)=O O(NC(=O)C(C)C(C)NC(c1coc(CC)n1)=O)CC C(C)(C)(C(C)CC(=O)NC1CN(C)CC1(F)F)NC(CCSCC)=O c1(C(=O)NC(CN(C(=O)CCNC(C)=O)CC)C)csc2c(OC)cccc12 Cn1cnc(C(=O)NCC2CCC(N(C3CC(O)C34CCC4)C(=O)C3CC3)C2)cc1=O C=CCC(C(=O)NCCC1(NC(CC(F)C2CCC2)=O)CCCC1)OC N1(C(Cn2ncc(C)c2)=O)CC2CCOC2(CNC(=O)C(C)OCC2CC2)C1 c1(SCCCCN2CC(NC(c3ccccc3)=O)C2)cc2cccnc2[nH]1 Cc1noc2nc(C(=O)NC3CCC(C)(CNC(C4(CCO)CC4)=O)C3)ccc12 C(=O)(C1CCc2ccccc21)NCC(C)N(C(=O)Cn1nnc(=N)[nH]1)C n1(CC)ccc(C(=O)NC23CC2CN(C(C2C4CCCC24)=O)C3)cc1=O C(CCCCN=c1cc(C)nc(SCC)[nH]1)NCC(=O)NC(C)C c1(CC(N2CCCC(NC(CC(COC)COC)=O)C2)=O)c(C)nc(C)nc1O C1(CN(C(CC2(COC)CCCC2)=O)C)CCN(C(=O)C(C)NC=O)CC1 CC(C)C(C)(C)C(=O)NC1C2CN(C(C34CCC(CC5CC5)(CC3)C4)=O)CC12 c1(C(N(CC(O)CN(C)C(C2(C(C)(C)C)CCCC2)=O)C)=O)cc(C#N)ccn1 C(=O)(CS(=O)(=O)NC(C)CC)NCC(C)(C1CCC1)NC(C(C=CCCC)O)=O c1(C(=O)NC=O)c[nH]nc1CCSCc1ccc[nH]1.C1(C=O)CC(Cn2ccnc2)C1 C1CCCS1(=O)=O.c1(C(CCC)NC(C2CN(C(N)=O)C2)=O)cn(CC)nn1 C(C(O)C(=O)N1CCC(N2CCC2)C1)NC(CS)=O.C=CCNCCC C1(C(N(CC(=O)NCC(C)O)C2CC2)=O)CCCC(F)C1 c1(C(=O)NC2CCCN(C(c3n(CC)ccc3)=O)C2C)cccc2c[nH]nc12 N1(C(C2(C(=O)OCC)CC2)=O)CCCC12CCCN(C(=O)Cc1cn[nH]c1)C2 CN1N=CC(CC(=O)N(C2CCCC2)Cc2ccccc2)C1=O C1(NC(=O)Cn2cnc(Br)n2)CC(CO)N(C(C2CC3CCC3C2)=O)C1 C#CCCCCC(=O)N1CC(=O)NCC1C(N1CCC(O)(C#C)C1)=O C1(C)(C(N(CCSC)CC)=O)CCN(C(C2(CCOC)CC2)=O)CC1 C1(NC(c2cncs2)=O)CN(C(C2CCCCS2(=O)=O)=O)C2CCCCC12 c1(C(=O)OC(CC=C)C(=O)NC2(C=C)CCCCC2)c(Cl)oc2ccccc12 N1(C(C2(C#C)CN(C(=O)C(C)=C3CCCC3)C2)=O)CC(C)C(C)C1C C12(CC)CN(C(c3cncc(C)c3)=O)C(CNC(=O)CCCOC(C)(C)C)(C1)C2 Cc1ccc(C=CC(=O)NC(C)(C)C(C)NC(c2cc(O)nc(O)n2)=O)cn1 c1(N(C)CC2CCCCO2)nnc(-c2ccccc2C)n1CC1(CO)CCCC1 C(=O)(CC(F)(F)F)NC(C1(CNC(CC2C(C)CC2)=O)CCC1)=O.C12CN(C1)C2 N1(C(C(C)(C)c2cccs2)=O)CC2CC(O)C1C2NC(C1CCCS1)=O C(=O)(CNC(=O)COC)N(CCC)CCOC.C1CO1 N1(C(C(=O)NCC)=O)CCN(C(c2ccncn2)=O)C(c2cccc(F)c2)C1 Cc1ccc(C(=O)NCCC2CN(C(=O)COC3CCOC3)CC(C)O2)c(Cl)c1 c1(C(=O)NCCOCCN(C(c2c(C)ccnc2C)=O)C)sccc1S(N)(=O)=O N1(C(C(C)SC)=O)CCOC(CN(C(=O)Cc2cnsc2)C)C1 CCCC(C)CC(=O)N1CC(O)(C(F)C(=O)NC2CC(=O)N(O)C2)C1 Cc1ccc2scc(C(=O)NC3CCN(C(=O)CCCC(C)(C)C)CC3F)c2c1 C1(F)(CNC(C2(CC)CC2(F)F)=O)CCCN(C(c2ncccc2O)=O)C1 c1(C(=O)NC(CN(C(C(CC)C)=O)C)(C)C)ccc(C2CC2)cc1 C(=O)(C1CCSc2ccccc21)N(C(c1cn(CCS(C)(=O)=O)nn1)C)C c1(CC(=O)NC(C)CCNC(C2(C3CCCCO3)CCC2)=O)ccc(Cl)cc1F Cc1cc(C(N2CCCC2C(N2CCCC(C)CC2)=O)=O)ccc1O C(C)(C)(CC(=O)N1CC(O)(CN(C(=O)Cc2ccccc2C(F)(F)F)C)C1)OC c1(OCC)cccc(C(=O)NC2CC(C#N)C2)c1F CCCC(C)(O)C(=O)N(C1CCC(CNC(c2ccc(Cl)s2)=O)CC1)C C1(CS(C)(=O)=O)CN(C(C23CC(F)(C2)C3)=O)CCN1C(=O)CC1CCCOCC1 c1(C(=O)NCC(CCOC)NC(c2ccc(C)o2)=O)ccc2c(c1)OCCC2 c1(OCC(C)(C)NC(C2CCC(CN)C2)=O)ccc(F)cc1 c1(C(=O)NC2(CNC(=O)COc3ccccc3F)COC2)cc(Br)ccc1O N1(CCn2cc(C3(C)CCCO3)nn2)CCC(C(=O)CC2COCCO2)CC1 C(N=c1[nH]c2cc(F)c(F)cc2s1)C1CCCCN(C(c2nc(CC)oc2)=O)C1 c1(C(=O)NC(C2(O)CN(C(C3(CO)CC3(F)F)=O)C2)C)cncn1C c1(CC)n[nH]c(=NCC2CN(C(c3ccc(OC(F)(F)F)cc3)=O)C2)s1 Cc1cc(Cl)c(C(N2CCC(CNC(=O)CCCCNC(N)=O)C2)=O)cc1F C1(NCC(N)CC(F)(F)F)CCc2c(cnn2Cc2ccccc2)C1 N1(C(c2n[nH]c(C)c2C)=O)CCCC(C)(C)C1C(=O)NCC(c1cccs1)C CCC(CC(C)C)C(=O)NC1CN(C(=O)C2=CCCC2)CCC1O c1(CC)ccc(C)c(C(N2CCC(C)(CCNC(C3CC(OC)C3)=O)C2)=O)c1 N1(CCC)CCCCC1Cn1cc(CNc2ccccc2C)nn1 n12cc(cn1)C(=O)NCC2.n1(CCOC)cc(-c2csc(C)c2)nn1 c1(C(=O)N(C)Cc2cc(N(S(C)(=O)=O)C)nn2C)ccc2ccoc2c1 N1(C(c2ccsc2)=O)CC(C2CN(C(C3CCSC3)=O)C2)C1 c1(C2CN(C(Cn3cc(CNC(C4CCC(F)(F)C4)=O)nn3)=O)C2)cnc2n1CCOC2 c1(C(=O)NCC2CC(Nc3nc(C)nc(=N)[nH]3)C2)cnc2[nH]c(O)nc2c1 N1(C(C2C(=C)C2)=O)CC(NC(c2ccnc(OC)n2)=O)C2(CCOCC2)C1 C1(NC(CN(C(C)C)C)=O)C2CC3C(C2)C13C(=O)NC(C)C(C)(C)N(C)C CC1CCCC(C(=O)NCc2nocc2C(N(C)CP(C)(C)=O)=O)CC1 N1(C(C=CCCC)=O)C(CNC(=O)C(C)(C)OCCC(F)(F)F)CC2CC12 c1(C(=O)NCCC2CCCN(C(CC(COC)C)=O)C2)cn2cccnc2n1 n1(C2(CNCC(CC)F)CC2)cnc2ccccc12.C12CCN(CC1)C2=O c1(C(=O)NC2CCC(NC(C3N(C)CCCC3)=O)CC2)ccc(O)c(CO)c1 N1(C(c2c(C)nccc2)=O)CC2(CCN(C(=O)CSc3cccs3)CC2)C1 O=C(O)C(CN1CCCC1c1cccc(C(F)(F)F)c1)Cc1ccc(Br)cc1 N1(C(CC(C)SC)=O)CCN(C(c2cccc3cnsc23)=O)C2(CC2)C1 N1(C(c2c(CCC)nns2)=O)CC(NC(C2(CCF)CC2)=O)CC(F)C1 c1(NC(C)CNC(c2cncc(Cl)n2)=O)ncnc2ccc([N+](=O)[O-])cc12 N1(C(c2cnccc2Cl)=O)CCC(N=c2[nH]c3cc(F)cc(F)c3o2)C1 N1(C(CCc2ccc(N(C)C)nc2)=O)CC2CCC1CN2C(=O)C=CCN(C)C c1(NC(C(N2CC3C(CC(=O)NCC)C3C2)C)=O)csc2c(OC)cccc12 C1(CC(=O)NCC2(F)CC(CNC(c3cc(C(F)F)no3)=O)C2)CCC2CC12 c1(C(=O)NC2C(C#N)C2)c(-c2cccc(Cn3cccn3)c2)cncc1F c1(-c2onc(C)n2)ccc(C(=O)NC(C)C(C)NC(C2(O)CC2)=O)cc1 C1(CNC(C=CC)=O)CN(C(c2nnn3c2COCC3)=O)CCC12CCOC2 C(=O)(CS(=O)CCC(F)(F)F)NC(CNC(C=NOC)=O)(C)CC(C)C CC(O)(CC(=O)N1CCCC(F)(CNC(c2ncc(Cl)cc2F)=O)C1)C(F)(F)F C1(CNC(c2ccnc(C(F)F)c2)=O)CC2(CC2)CN1C(=O)COc1ccon1 C(CCCCNC(=O)CCc1cn[nH]c1)N(C(CC1C(C)C1)=O)C c1(COC)c(C(=O)NCC2CC(NC(C34CC(C)C3C4)=O)C2)cnn1C c1(CN(C2C(C)CCNCC2)C(=O)C(C)(F)F)ccc2c(c1)OCCO2 C(C)(CC(=O)NC1CCC(NC(=O)C(F)n2ccnc2)CC1)(C(F)(F)F)N(C)C N1(C(COCCOCC#C)=O)CCC(C(=O)NCC2C=CCCC2)C(C)(C)C1 C12(NC(c3c(C)nc(CC(C)C)s3)=O)CCN(C(C3(C#N)CC3)=O)CC1C2 C1(N(C(c2cn(CC(CC)O)nn2)=O)C)CCN(C(C2(CO)CCOC2)=O)CC1 N1(C(c2nccc(N)c2Cl)=O)CC2CC1CCN2C(=O)CN1CCCNC1=O Cc1c(C(N2CC3CCN(C(=O)CN4CC(=O)NC4=O)C3C2)=O)sc2nccn12 Cc1oc(CO)cc1C(=O)NCC(C)(F)CNC(C1(C)CCCC1C)=O N1(C(Cc2ncc(CC)[nH]2)=O)CCC2C(CCN2C(=O)C(C)NS(C)(=O)=O)C1 C(CCCCCC(=O)N1CC(CNC(=O)C(=Cc2cccnc2)F)C(C)C1)SC c1(C(C)C)ccc(C(=O)N(CC(C)CN(C(C2CCOC2)=O)C2CC2)C)o1 C1(NC(C(C)C(C)O)=O)CCN(C(=O)Cc2cccs2)CCC1CO C1(C(=O)NCCOCCN(C)C(c2cc(=N)[nH]c(=N)[nH]2)=O)Cc2cscc2C1 c1(CC(=O)NCC(C)NC(C2(F)CCOCC2)=O)ccc(C(N)=O)nc1 N1(C(C(C)c2cccs2)=O)CC2CC(NC(c3cnc4ccccn34)=O)CC2C1 C1(C(=O)NCC(C(=O)NC)(C)C)CC(Nc2c(C(=O)NC)nccn2)C12CCC2 c1(CNC(CC)=O)nc(C(C)Nc2ncc(C3(O)CCC3)s2)cc(NC)c1C.C(C)C CC(CN=c1ccc(S(C)(=O)=O)c[nH]1)N(C(=O)CCc1ccon1)C Cc1cc(C(N2CCCN(C3CC3)CC2)C(=O)NC(C)C)c2c(c1)CCC2 C=C(C)C(O)CC(=O)NCC1(CNC(=O)C(C(C)(C)C)SC)CCCC1 c1(C(N2CCC(C(C)(Cl)NC(C3CC3C3CCC3)=O)C2)=O)ccc(F)cc1F N1(C(C2N(C(C)C)CCC2)=O)CCCC(C(=O)N(C)C(c2ccc(F)cc2)C)C1 N1(C(C(=O)NC(C)C)=O)CC2CC2(NC(=O)CCC2CC(C)(C)CO2)C1 C#Cc1ccc(C(=O)N(CC(C)NC(c2cccc(C3CC3)c2F)=O)C)nc1 C1(NC(C(c2ccccc2)C)=O)CCN(C(=O)CCC2CCCCC2)C1C1CC1 c1(C(C)=O)cnc(Cl)[nH]c1=NC1CCCC(NC(c2ccc3cnccc3c2)=O)C1 C1(C(=O)NC(C(C)NC(C23CCC(CO)(CC2)C3)=O)CO)CNC(=O)CC1(C)C Cc1cccc(C(N2CCCC2(C)CCC(=O)N(C2CCOC2)C)=O)c1 C1(NC(c2c(OC)ccs2)=O)CN(C(C2(C)COC(=O)C2)=O)CCC1F C12CCC(CC1)NC2=O.C(=O)(CN(CCO)CCO)N(C(C)C)CCF C(=O)(CCCCC(=O)N(C)C)NCC1(NC(CCc2nnc(C(C)C)o2)=O)CCC1 N1(C(C(c2ccccc2Cl)C)=O)CC(NC(=O)CCCC2CCC2)C(O)C1 C1(CC(=O)NCCCCNC(C(c2cccnc2)OC)=O)CCCC(F)(F)C1 CCCCC(C(=O)N1CCC(CCC(=O)NCCCn2ccnc2C)C1)N(C)C c1(NC(=O)NCCC2CC(CO)C2)ccnc2[nH]ncc12 N1(CCc2cn(CC(N3C(C(C)C)CCC3)=O)nn2)CCC(CO)CC1 CCC(C(C)(F)F)NC(=O)COC1CN(C(=O)CC(F)(F)F)C1 c1(C(=O)NCC(C(C)C)(C)NC(c2ccnnc2)=O)cccc2c1OC(F)(F)O2 C#CCC(C)(CC)C(=O)NCCC1CC(NC(C2(C#N)CCSCC2)=O)C1 c1(CNC(C(CNC)(C)C)=O)ccc(OC)c(-c2n[nH]cn2)c1 Cc1sc2ccccc2c1C(N1CC(O)(C(C)NC(C2CC3CC3C2)=O)C1)=O N1(C(C(COC)C)=O)CC2CCCC(CNC(=O)CN3CCC(O)CC3)(C2)C1 c1(CNC(c2ccc(OC)cc2)=O)ccc(-c2nn[nH]n2)c(O)n1 C(c1cn(C)cn1)=CC(=O)NC1C(NC(c2ccc(C(C)=O)o2)=O)CC1 C(=O)(C(C)(O)C(F)(F)F)NCCCCC1CN(c2nnc(CC(C)C)s2)C1 Cc1nc(N2CCCC3(NC(C4CCNC4=O)=O)CC3C2)c2cnn(C)c2n1 Cc1nccc(C(N2CC(C3CC3)(C(N3CCCC3CC(C)O)=O)C2)=O)c1N c1(CC)oc(C(N2CCCC(CNC(C3CCCC(CF)C3)=O)C2)=O)cc1C c1(C(=O)OC)nccc(N(CCCNC(c2ccc(C3COC3)cc2)=O)C(C)C)n1 C1(NC2CCCN(CCC(C)(C)C)C2=O)CC2CCC1N(c1ccccn1)C2 N1(CC(=O)NCCCOCCC(=O)NCC2N(CC)CC2)CCNC(=O)C1 c1(C(N2CCC(CN(C(=O)CNC(C3CCC3)=O)C)C2)=O)sccc1C#N C#CCCCCC(=O)NCCCN1CCC(NC(c2cccc(CCO)c2)=O)C1 c1(C(C(=O)OCCC=C(C)C)C)cccc(Br)c1 N(C(=NCCn1cccc1)NC(C)C1CC1)Cc1c(Br)cn(CC)n1 C1(NC(C2C(C)(CC)C2)=O)CCC(C(=O)NCC2(N(C)C)CCCC2)CC1 Cc1ncc(C(N2CCC(O)(CN(C)C(C3CCC(=O)N3C)=O)C2)=O)cc1N N1(C(CC2CCC(C)C2)=O)CCOCC(CN2C3(C(=O)NC4CC4)CC(C2)C3)C1 C1(C(=O)NC2(CN(C(=O)C(CO)N(C)C)C)CC2)(OC)CCCCC1 C1(C(=O)NCCCC(C)NC(=O)CCC(F)(F)F)CCCC(C)(C)C1 c1(C(N(CCN(C(=O)CCNC(=O)CO)C(C)C)C)=O)c[nH]c(Br)c1 C1(NC(C(C)NC(C)=O)=O)COC2(C1)CN(C(C1CC1c1ccccc1)=O)C2 Cc1ccc([N+](=O)[O-])c(C(N2CCC(NC(c3ccc(Cl)s3)=O)C2)=O)c1 N1(C(CC2C(C(C)(C)C)C2(C)C)=O)CCCC(CNC(C2C3CN(C)CC23)=O)C1 N1(C(CCc2scc(C)n2)=O)CCC(NC(=O)C(F)=CC2CC2)CC1C C1(O)(C(N2CC(OC)C(NC(=O)CC(C)F)C2)=O)CC2(CCOCC2)C1 N1(C(C(C(C)NC(C(=Cc2ccco2)C)=O)C)=O)CC2CCN(C)C2C1 C1(C(=O)NCCC(C)(C)NC(=O)Cn2cc(C3CC3)cn2)CCC(C#N)C1 Cc1ccc(NC2CCC(NC(=O)OC(C)(C)C)C2)c2cccnc12 C1(NC(=O)Nc2cccc(C(N)=O)c2)CCn2nnnc2C1 C1(NC(C2N(C=O)CCC2)=O)CN(C(c2cncc(F)c2)=O)CC2(CCC2)C1 N1(C(C2(NC(c3cc(C)on3)=O)CCCC2C)=O)CC2CC(C)C2C1 C1(O)(C(C)NC(C2CC(C)N2C(c2sccc2Cl)=O)=O)CCCCC1 C(=O)(CCCN=[N+]=[N-])N1CCC(O)(CNC(C2CC(C)(F)C2)=O)C1 C1(c2n(C)cnc2)CN(C(=O)C2=CCC2)CC1NC(c1cc(Br)c[nH]1)=O Cc1ccc(Cl)c(O)c1C(=O)NCC=CCNC(C1(C)C=CCCC1)=O Cc1cccc(S(=O)(=O)NCCC(C)C(F)(F)F)c1Cl C(=O)(C(F)CC)NCC(CNC(N1CC(CCC)C1)=O)OC c1(C(=O)NCCC2(NC(CCC#C)=O)CCCC2)c(OC)cccc1Cl CC(C)(O)CC(=O)NCC1(CNC(=O)Cc2ccnnc2O)CC1 c1(C(N(CCNC(CC(C)C(C)(C)C)=O)C2CC2)=O)cc2c(cn1)COCC2 N1(c2cc(NC(CCCN(CCO)CC)C)ncn2)CCC2(CCCCC2)C1 Cc1conc1C(=O)NC(C1CCN(C(=O)C(C)ONC(=O)OC(C)(C)C)C1)C N1(C(C2(C#C)CC2)=O)CCCC(C2(NC(=O)C(C)NC(=O)NC)CC2)C1 C(=O)(CC(C(F)F)c1ccsc1)NCCC(C)NC(=O)C=CC=C(Cl)Cl c1(CNC(C(C)(C)COC)c2n(C(CC)C)nnn2)ccc2ccccc2c1C C(C(C)C)(C(O)C(=O)NCCN(C(C1(c2ccccc2)CC(C)C1)=O)CC)OC c1(CCNC(C2CN(CCN3CCCC3)CCC2O)=O)ccc2c(c1)OCO2 c1(SCC(=O)NCC2C(NC(CCCOC)=O)CCC2)nc2ccccc2[nH]1 C(=O)(C(C)(O)C(C)(C)C)NCC(C)NC(c1nccn2cnnc12)=O C1(NC(CCc2nc(C)sc2)=O)CC2(C1)CC(NC(c1onc(C)c1C)=O)C2 CN1CC(NC(=O)N(C)C)CC12CCC2.C12CCCN(C1)C(=O)Cn1cc2nn1 c1(-c2n(CCCC#N)c(N3CCS(=O)CC3)nn2)ccn2ccnc2c1 N1(C(CCc2cc(OC)c(C)o2)=O)CCN(C(=O)Cc2cnsc2)C(C)CC1C CC(C)C(CC(=O)N(CC(C)C(=O)NC1CC1)C)NC(=O)C#CC(C)(C)C CC(C)C(CNC(=O)CC1(NC(=O)C(c2cncnc2)C)CCCC1)NC(N)=O C1(F)(CNC(C=CCOC)=O)CC(NC(=O)C=Cc2cocn2)C1 N1(C(C2CCCC(C(=O)OC)C2)=O)C(C)CC2CN(C(c3coc(Cl)n3)=O)CC12 C(CC(C)C(=O)N1CCC(CC(=O)NC(CCOC)C(C)C)C1)=CC c1(-n2cc(CC(C(F)(F)F)N3CCOCC3)nn2)ccc2cccc(Cl)c2n1 C1(N(C(c2cc(OCC)no2)=O)C)CCCC(NC(=O)C(C)(C)c2cnco2)C1 c1(NC(C2(NC(CC=C)=O)CC(CO)C2)=O)cnc(Cl)c(C)c1 c1(C(N2CCCC(NC(c3cc[nH]n3)=O)(CO)C2)=O)cc(Br)ccc1[N+](=O)[O-] N1(C(CCC(C)(C)F)=O)CCC2(CC1)CCN(C(=O)CN1CC3C=CC1C3)CC2 c1(CCNC(N(CC(CCC=C)O)C)=O)ccc(Br)c(OC)c1 Nc1c(Cl)ccc(F)c1C(N1CCCC1CNC(=O)CCc1cccc(F)c1)=O C(=O)(C1CCc2ccccc21)N1CCCCC(C(=O)NC2CN(C)NC2=O)C1 C1(NC(=O)CNC(N2CCCC2)=O)CC2(CCCN2C(C2CCCNC2=O)=O)C1 C=CCC(C)(CC)C(=O)N(C(CC)CC(N1CC2(C1)CC2(F)F)=O)C c1(CC)nc(N2CCCC(NC(c3c(C(F)(F)F)cnn3C)=O)CC2)[nH]c(=N)n1 c1(CNC(C(C)C2CC2)=O)nnc2n1CCN(C(c1ccc3c(c1)CCC3)=O)C2 Cc1ccc(C(=O)NC(C)C(C)NC(c2cnn(C)c2C(F)F)=O)c(N)c1Cl N1(C(C2(C)CCN(C(c3c(C)cc(CC)o3)=O)C2)=O)CCC2(CCC(O)C2)C1 N1(C(c2ccc(CC)cc2O)=O)CCc2nc(NC(=O)CCOCC)sc2C1 c1(NCC2CCC(CC)O2)ccc(=N)[nH]n1 Cc1ccoc1C(=O)NC1CCCC1NC(c1cc(Cc2ccccc2)[nH]n1)=O O=C(C#CC1CCOC1)NCCC1CCCN(C(C2CN(S(N)(=O)=O)C2)=O)C1 N1(C(c2ccc(C(C)C)s2)=O)CCN(C(C2CSCCS2)=O)C(C(C)(C)C)C1 C1(CC(=O)OC(C)(C)C)CC(O)C12CCC2.c1(C(=O)O)cc(C(=O)NC)cs1 N1(C(=O)Cc2ccc(Cl)cc2)CCCC2C1CCN2C(=O)Cc1ccncc1 N1(C(C(C)O)=O)CC(C2CCCN(C(c3[nH]c(=N)ccc3Br)=O)C2)C1 c1(N(C)CC2CCCN(C(=O)CCc3cnn[nH]3)C2)nnccc1C#N CC(C)C(O)CC(=O)N1CC(F)(F)CC1CNC(c1cnn(C(C)(C)C)c1)=O c1(C(N)=O)c(C(=O)Nc2cnc(OCC3CCC3)cn2)cccc1C c1(C(=O)NCC2C(C)CN(C(=O)C(C)OCC3CC3)C2)c[nH]c2cccc(Cl)c12 c1(C(c2nnnn2CCCC2CC2)NC(C(=O)NCC(C)C)C)ccnc(F)c1 c1(C(N2C(C)CC(NC(c3csc(O)n3)=O)C2)=O)cccc2nonc12 C1(C(N(C(CC)CC)C2CC2)=O)C=CC(NC(c2cnsc2C)=O)C1 c1(C(N2C(CNC(C3CCO3)=O)CCC2)=O)ccc(Cl)c(C(F)(F)F)c1 C1(C2CCNCC2)(C(CNC(C(C(C(C)C)=O)(C)C)=O)=O)CCOCC1 CN1CCC2(CC1)CC(O)CN2CC1CCCC(F)C1 c1(C(=O)NCC2N(C(C(C)n3cccc3)=O)CCOC2)noc2ccc(Cl)cc12 c1(C(N(C(C2CCC2)C)C)C)cccc2ccccc12 C(CCCCC(=O)NC1CN(C(C)C)CC1C)N(C(c1c(C)con1)=O)C N1(C(C=C(CCC)CCC)=O)CC(C)(C)CC1CC(N1Cc2c[nH]nc2C1)=O c1(C(N2CC(CC(C)(F)F)C2)=O)cc(=O)c2ccc(F)cc2o1 C1(C(=O)NCC=CCNC(c2c(C)nn(C(C)C)c2)=O)CN2CCN1C(C)C2 c1(C(=O)NC(CN(C(C2CC(OC)C2)=O)CC)C)cccc(Cl)c1 C(c1ccnn1C)=CC(=O)N(CCOC)CC1CCCN(CCC)C1 CCC(C)(CC)NC(=O)C(C)CNC(=O)CCN(C)CCO c1(OC)cc(CC(=O)NCC2CCC2NC(c2cc(=O)c(OC)co2)=O)ccc1Cl C=CC(C)(O)CC(=O)N1CC(OCC(=O)NC2CCC3CCC23)C1 c1(CCC(N2C3(CN(C(c4ccc(=O)oc4)=O)C3)CC2)=O)nc2ncccn2n1 C1(C)(C(=O)NCCC(C(C)C)NC(C(CCCOC)C)=O)CCCCNC1=O N1(C(CC(CCC)CC)=O)CCC2(CCCN2C(=O)C(C(C)C)SC)C1 CC(C)(CC(=O)N1CC(NC(c2sc(F)cc2Cl)=O)C(O)C1)CC(F)F c1(C(N(CC(C)(C)NC(=O)CC2CCCOC2)C)=O)c(F)cc(Cl)cc1Cl c1(CC)cnccc1C(N1CC2C(C(N3CC(C)=C(C)C3)=O)C2C1)=O CC(CNC(C12CSCC1C2)=O)CC(=O)Nc1ccc(F)nc1 N1(C(c2cccc(SC)c2)=O)CCCC(CNC(C2C(C(=O)OCC)C2)=O)C1 c1(CC(=O)NCC(CNC(c2csc(-c3ccc(C)o3)n2)=O)OC)n[nH]c(C)n1 c1(CNCC(C)N(C)C(C23CCC(CC2)CC3)=O)ccc(N(C)C)c([N+](=O)[O-])c1 c1(NC(C=CC(CC)C)=O)nn(C)cc1N N1(C(CC(C=C)(C)O)=O)CC(C2CCCN(C(c3cn(C)cn3)=O)C2)C1 C(CC1=CCOCC1)NC(CNC(CCCOC)=O)=O C1(C(=O)NC2(CO)CN(C(C(CC(N)=O)O)=O)C2)Cc2c[nH]cc2S1(=O)=O.C(N)(=O)N N1(C(C2(C#C)CC2)=O)CCCC(C2CCN(C(=O)C(O)P(C)(C)=O)CC2)CC1 C1(NC(CN(CCC)C)=O)CC2(CCN(C(=O)C(C)CC(F)(F)F)CC2)C1 C1(CCCNC(Cc2cn(CC)nn2)=O)CN(C(=O)C(C(C)O)N(C)C)CCO1 Cc1ncc(C(N2CCCC2CCNC(c2ccc(C(N)=O)[nH]2)=O)=O)c(O)n1 C1(NC(c2n[nH]c(C)c2Cl)=O)CN(C(C23CC(F)(C2)C3)=O)CC1S(C)(=O)=O c1(-c2cn(CC3(C(C)NC(=O)C(O)Cc4cnn[nH]4)CC3)nn2)cnccc1Cl N1(C(C(Cn2ccc(C)n2)C)=O)CC2OCCN(C(c3coc(C)n3)=O)C2C1 C(=O)(C(CC)CC(F)F)N1CCCCC(NC(C(CC=C)OC)=O)C1 c1(C(C(=O)NC2CCC(CNC(CN(CCOC)C)=O)C2)(C)O)cccc(C)c1 N1(C(COC(CC)C)=O)CCC(C2(NC(=O)C3=CCCOC3)CC2)CC1 C(C(=O)N1CCCC1(C)C(N1CCC(CN=[N+]=[N-])C1)=O)(C(C)(C)C)OC Cc1cc(N2CC(C(N)=O)C3(CC3)C2)nc(=NCCN(C)CCO)[nH]1 c1(C(=O)NC2C3CN(C(CC(C(C)C)O)=O)CC2C3)cncc2c(O)nccc12 C(=O)(C(F)CC(C)(C)NC(C1CCO1)=O)N(CC(CO)OC)C C1(N(C(C(C)OC2CCCCC2)=O)C)CC2CC1N(C(C1CCCCCC1)=O)C2 C(=O)(C#CC1CCCO1)NC1(C)CCN(C(c2nc(OC)c(C)s2)=O)C1 N1(NCC)CCCC(C(=O)NCc2n(CC(=C)C)ccc2)C1.C(C)=O C=Cc1cncc(C(=O)NCC2(OC)CN(C(c3cc(C#N)ccn3)=O)C2)c1 Cc1ccc(NC(C2(C(C)(C)C)CCN(C(=O)CCC3CC3)C2)=O)c(Br)c1 C1(CN(C(CCN(CCC)C)=O)C)COCCN1C(=O)C=Cc1cscn1 C(=O)(C1=NOC(C)(C)C1)NC1C2(CCN(C(C=CCNC(=O)OC(C)(C)C)=O)C2)C1 C1(NC(=O)C(O)C2CC2)(CF)CCN(C(=O)CC2CCC=CCC2)C1 C1(C)(NC(CN2CCC(C)CC2)=O)CCN(C(C2CC2C(F)(F)F)=O)CC1 C(=O)(C(C)(F)C(C)(C)F)N(C(C)(C)C)C(=O)NCC.c1(C(C)C)n[nH]c(C(C)N)n1 C1(C(=O)NC2C(NC(CCC(C)(C)F)=O)COC2)CSC(c2ccccc2)=N1 Cc1cn2cc(NC(C3CCCN3C(c3csc(C)n3)=O)=O)ccc2n1 C#Cc1cnn(C)c1C(=O)NCC1(C(N2CCC3(CSC3)C2)=O)CC(=C)C1 CC1CCCC(C)N1CC1(O)CC1.N1CC2CC1CN2C(=O)Nc1cc(CO)on1 c1(C(=O)NC(CNC(C(CC)C)=O)C)cc(Cl)ccc1OCCN(C)C N=c1[nH]nc(CC(=O)NC2CC(F)(CNC(C3CCCCC3)=O)C2)s1 C1(NC(Cc2n(C)cnc2)=O)CCCCN(C(=O)CCc2nc[nH]n2)C1 Cc1cc(=NCC2CC=CCC2)[nH]c(N2CCC(N3CCC(O)C3)CC2)n1 Cc1ncnc(C)c1C(=O)NCCOCC(=O)NOCCC(F)(F)F c1(C(=O)NCCCC(=C)Cl)nc(CNC(C2CSC2)=O)oc1C C(C)(C)(C(O)CO)N(C(C(CC)NC(=O)CN(C(=O)C(C)C)C)=O)C C(=O)(C(O)Cc1cnc[nH]1)N(CC(CN(C(=O)C(=O)N(C)C)C)O)C c1(C(C)=O)cc(C(=O)NCC(C)(C)OCCNC(c2nnn(C)n2)=O)c(C)o1 CC1CN(C(c2ccc(CO)cc2)=O)C(C)CN1C(=O)C(O)CC1CCCC1 CCCC(C)CC(=O)NCCC1CN(C(c2cccc(C)c2O)=O)CCO1 Cc1cc(Cl)cc(Br)c1NC(C1CCSC(C(F)(F)F)C1)=O O=C(CC1OB(O)c2ccccc21)Nc1ccc(Cl)c(I)c1 C(=O)(C(F)(F)C(O)C(C)C)NCC1(C)CCCN(C(C2(OC)CCCOC2)=O)C1 c1(C(N2CC(CCNC(C(C)C(C)(F)F)=O)C2)=O)cccc2nc(O)oc12 c1(C(=O)NCCC2(NC(c3cnc(CC(C)C)[nH]3)=O)CC2)cccc2oncc12 C1(C(=O)NCC(C2CC2)NC(c2cc(C(=O)OC)on2)=O)CN(C)C(=O)N1 Cn1cc2ccc(C(=O)NC3CN(C(C4CCS4(=O)=O)=O)CC3C3CC3)cc2n1 Cc1ccc(C)c(C(=O)NC(C2CCCCN2C(C2CC3(C2)CC(O)C3)=O)C)c1 C1(C(=O)NC2CC(C(C)Nc3ncncc3Br)C2)CCCCN1N=O N1(C(C(C)(C)c2cccnc2)=O)CC2(C1)CN(C(C1CC13CCCCC3)=O)C2 c1(NC(NCc2nnc(C(C)(C)C)s2)=NCCOCCO)nc2ccccc2o1 CC1(C)CN(c2cncc(C#N)n2)CC1NC(=O)C#CC1CC1 N1(C(C(F)=CC)=O)CC2CCC(C1)N(C(c1ncc(C)cc1Br)=O)C2 C(=O)(C1CCCc2nc[nH]c21)NCCC(CNC(Cc1c(C)cccn1)=O)O N1(C(CS(=O)(=O)NC)=O)CC(C)N(C(=O)CCC2CCCO2)CC1C c1(C(=O)NC2(C3CN(C(CCOCCC)=O)C3)CC2)cncc2nnn(C)c12 C(C1C(C)C1(Cl)Cl)=CC(=O)N(C(CC)C1CC1)CC CC1COC2(C1)CN(C(=O)CC1(CO)CC1)C2.C12(CCOC1)C(=O)NC2 c1(C(=O)NC(C(C)C)CCNC(=O)C(N2CCC(C)(O)C2)C)cc2c(s1)CCC2 C1(C(=O)Nc2ccc(CC(C)C)cc2)CCCN(c2ccc(Br)cc2)C1=O CCC(CC(=O)NC(C)(CSC)C(=O)NCC(C)(COC)CO)C1CCC1 Cc1nc2cncc(C(N3CCC(CNC(=O)C4=CCSC4)C34CC4)=O)c2[nH]1 N1(C(CC(C)(F)F)=O)Cc2ccccc2C(NC(c2ccc(F)s2)=O)C1 C(CN=c1[nH]nc(CO)s1)O.c12cccc(c1F)NC(=O)N1CCCCC21.CC C1(=O)C(C)(O)CCN1.C(=O)(C(C)CN(C)C)NCCCOC(C)C c1(CNC(NC(C)CC2CCCO2)=NCC2CC2)nc2cc(Br)ccc2o1 c1(C(=O)NCC(C(C)C)NC(C(=Cc2cnc[nH]2)C)=O)cc(C(F)F)nn1C c1(C(=O)NC2CC(C)(NC(CCC(C)C)=O)C2)cc2sccc2[nH]1 CCCCC(CN=c1[nH]nc(C2CC2)s1)NC(c1sc(CC)nc1C)=O CC(CNC(C1CN(C2CCOC2)C1)=O)(C1CC1)NC(=O)CC1CC=CC1 C(=O)(C(CCC(N)=O)N(C)C)N1CCCCC(NC(CCCOC)=O)C1 C(=O)(CC(F)(F)C(F)F)OC(COC)(C)CNC(c1cccc(OC)c1N)=O C#CCC(C)(CC)C(=O)NCCC(O)CNC(c1nc(C)n(-c2nc[nH]n2)n1)=O Cc1cccc(C(=O)NC2C=CC(CNC(=O)Cc3csc(C)n3)C2)c1 N1(C(c2cc(C(C)(C)C)n[nH]2)=O)CCN(C(c2ccnc(O)c2)=O)C2(CCC2)C1 c1(C(=O)OC)ccncc1C(=O)NCCC1(NC(C2(CC(C)C)CC2)=O)CCC1 c1(C(=O)NC(CNC(=O)CCc2ccncn2)CO)c(O)cc(F)cc1F C1(NC(c2cn(C)nn2)=O)CCN(C(=O)CCC(F)F)C1c1ccccc1 c1(OC)ccc(C)cc1C(N1CCCC(NC(c2ncc(F)cc2F)=O)CC1)=O C=CC1COCC1NC(=O)COC(C1CC2(CC2)C1)=O c1(-n2cc(NC(C(=O)NCCOCC=C)=O)nn2)ccc(N(C)CCO)cc1 N1(C(C(C)(C)O)=O)CCC2(CC(NC(c3ccnc(C(F)F)c3)=O)CO2)C1 c1(C(=O)OCCCc2c(F)cccc2Cl)cc2n(n1)CCCCC2=O N1(C(C(N2CCOCC2)C)=O)CCC2(CCN(C(=O)C(F)(F)CO)CC2)C1 CS(=O)(=O)c1coc(CNC(C2CCN(CC(F)(F)F)CC2)=O)c1 Cn1ncnc1CCC(=O)NCC1CCN(C(=O)COC2CCOC2)C1 Cc1cc2c(Br)ccc(C(=O)NC3(CF)CCN(C(=O)C(C)O)C3)c2o1 N1(C(c2c(CNC(CCC(=O)NCC)=O)nnn2C)=O)CCOCC12CC2 N1(C(C2C(CCC)CCC2)=O)CCC2(CC1)CC(NC(=O)CC(C)C(F)F)CO2 CC1(CNC(=O)CCC2CCOC2)CCN(C(C2(C(F)(F)F)CCOCC2)=O)C1 C1(N(C)C(C2CCC(c3ccccc3)CC2)=O)CCCN(C(=O)CC2CC2)C1 N1(C(COc2cccc(C)c2)=O)CC2(CC(NC(=O)CCC[N+](=O)[O-])CO2)C1 C1(NC(c2c(CC)con2)=O)CN(C(C2(C#N)CCCOC2)=O)CCC1C CC1CCC(NC(=O)CCCn2cncn2)CN1C(=O)C=CC1CCC1 c1(OC)ccc2c(C(=O)NCCC3CCN(C(C4(C)CC4)=O)C3)cnn2c1 C(C(O)CC(=O)NCCC1(NC(C2(c3cccnc3)CC2)=O)CC1)N(C)C C(C1=CCCOC1)N(C(CCN(C(CNC(C1C(C)C1)=O)=O)C1CC1)=O)C C12(CC3(CC3)C1)C(=O)NC2.N1(C(CN2C(=O)CSC2)=O)CCOC2CC12 CC1C=CCCC1.C1(Cn2cc(-c3cncs3)nn2)C(CC(C2CC2)=O)C1(F)F Cc1c(CC(N2CCC(NC(=O)COCCOc3ccccc3)C2)=O)ncn1C C1(C(=O)NCC2(CNC(Cc3cn(C)nn3)=O)CC2)CCC2(CC1)CC2 N1(C(c2cc(C)n(C(C)(C)C)n2)=O)CC2CC(NC(c3cc(O)no3)=O)C2C1 Fc1ccc2c(c1)C1C(C2)C12COCCNC2.c12nc3cccnc3cc1N2 c12ccccc1[nH]c(=O)n2CC.n1(CCO)ccc(-c2ccncc2)n1 c1(C(=O)NC(CC=C)CNC(C)=O)ccc(OC)c(S(C)(=O)=O)c1 CC1CCN(C(c2cc[n+]([O-])cc2)=O)CC1CC(=O)NOCC1CCCC1 c1(C(=O)NC2CN(C(c3ccc(N(C)C)cc3)=O)C2)cc2cc(Cl)ccc2[nH]1 c1(C(N(CC(C)CNC(=O)CC2CCCC23CC3)C)=O)c(O)nnc2c1CCC2 c1(C(=O)OC)ccc(NC(=O)C2=C(C)OCCS2)c(Cl)c1Cl c1(CC(N2CCCC(CNC(C3CC3F)=O)C2)=O)coc2cc(Cl)ccc12 C(=O)(CCC(C)(F)F)NC(CNC(CC1N(C(C)=O)CCCC1)=O)(C)CO c1(NC(=O)CCCSC2CCN(C(C34CC(C3)C4)=O)C2)ccc(F)cc1.C1C(=O)N1 C1(C(N2CCC(CCC)C2)=O)CC2CN(C(=O)C(C)(C)OC)CC2C1 N1(C(C(C=C)(C)CCOC)=O)CCC2(CCC2NC(c2cc(Cl)on2)=O)CC1 C(=O)(CCCC(F)(F)CO)N1CCCC(C)(NC(c2cc(C)n(C(C)C)n2)=O)C1 c1(CC(=O)NCCC(C)C)ccc(C)cc1.C1(=O)C(C)OC(=O)CN1CCC.CC CC1=C(C(=O)NC2CC3CN(C(=O)C=Cc4nc(C)co4)CC3C2)CCCO1 c1(C2CCOC2)ncc(C(=O)NC(C)CN(C)C(C2CC(O)C2)=O)s1 N1(C(C2CCN(CC)C2)=O)CC2CCCC2(NC(=O)C2=CCN(C)C2)C1 c1(C(=O)NCC2(C)CCN(C(C=C3CCC(C)C3)=O)C2)cc2c(s1)CN(C)CC2 CCC(C)(C)C(=O)N1CCCC1CNC(=O)C(=O)N(C)C N1(C(C=CC(=O)OCCCC)=O)CC(NC(=O)C(C)CC#N)CC(O)C1 C(C)(C(C)CCSC)NC(c1n(CCCCCC)nnn1)c1ccc(Cl)s1 C1(CC(=O)NC(c2cn(C)cn2)C)CCN(C(=O)CC2CNC(=O)O2)CC1 N1(C(CCCNC(=O)C2=COCCC2)=O)CCCN(C=O)CC1 c1(CC(N2CCC(N(C(C(CC)O)=O)C)C2)=O)coc2ccc3ccccc3c12 S1(=O)(=O)c2ccc(nc2)NC2CCCC(C2)N1.CC(=O)NCCN(C)C CCC(C)(CO)C(=O)NC1CCC(CC(N2CCOCC2CCO)=O)CC1 N1(C(C(C(C)NC(=O)Cn2ccnn2)C)=O)CC2(CCCCC2)C1 CC1CC(c2nnnn2C2COC2)(NCCC2(C(F)F)CCC2)C1 CC1CN(C(c2ccc(Br)o2)=O)CCC1NC(=O)C=CC(N)=O C(=O)(CC(C)C(=O)OC)N1C(C(N2C(C(=O)OC)CCC2C)=O)CCC1 C1(C(=O)NC(CCC#C)C)CN(C)CCN1C(c1cccnc1O)=O N1(C(C2(C)CCOCC2)=O)CC2CN(C(C3CC4OC(=O)OC4C3)=O)CC2(C)C1 C(=O)(NNC(=O)CN1CCCC1CO)C12CC(CNC(=O)OC(C)(C)C)(C1)C2 C(CC1=CCCCC1)NC(C1(NC(C2(c3ccno3)CC2)=O)CCSC1)=O N1(C(C#CC(C)C)=O)CCCC12CCN(C(c1ccn3ncccc13)=O)C2 c1(CCNC(C2(CC)CCCC2)=O)ccc2c(c1)CN(C(=O)C1=CCOC1)C2 Cn1c(Cl)cnc1-c1ccc(C(Cc2noc(Cc3cccs3)n2)C(C)(C)C)o1 C1(C(=O)NCc2scc(C(N(CCC(C)O)C)=O)c2)CC(C)(C)CN1C Cc1cc([N+](=O)[O-])cc(C(=O)NCC(CO)NC(c2ccn(C(C)C)c2C)=O)n1 C1(OC)CN(C(=O)Cc2cscn2)C(C)(CNC(=O)CNS(N)(=O)=O)C1 N1(C(=O)CONC(c2ccc(O)nc2)=O)CC2C3CCC(C3)C2C1 C1(C(C(=O)NC)N(CC(C)S(C)(=O)=O)C)CCN(CC(F)F)CC1 CCCC(C)(C)CC(=O)N1CCC2(CC1)CC2NC(=O)C(CC)C(C)C Clc1ccc(-c2csc(CSc3cccc(Cl)c3)n2)cc1 N1(C(C(CCC)O)=O)CC2CC(C1)CN(C(C1CCCN1C1CCCC1)=O)C2 c1(NC(CC2(F)CN(C(=O)OC(C)(C)C)C2)=O)ccc(N=[N+]=[N-])c(F)c1 CC1=C(C(=O)NC2(CF)CN(C(c3cc(C)nc(O)c3)=O)C2)CCO1 C1(C(=O)NCCCC(C)NC(C=C(CCC)C)=O)CCC(C(=O)N(C)C)CC1 C1(CNC(C2(OC)CCN(C(C3CC(C)C3)=O)C2)=O)CN2CCC1CC2 C(C(C(C)C(C)C)NC(=O)CN1CCCC1=O)NC(CCc1c(C)cccn1)=O N1(C(C(CC)N(C)C)=O)CC2CC(C(=O)NCC3(SC)CCCC3)C(C2)C1 N1(C(C(C(CC)C)O)=O)CC2(C1)CN(C(c1cc3c(=O)[nH]ccn3c1)=O)CCO2 N1(C(C2CN(C(C)(C)C)C(=O)C2)=O)CC2CCCN(C(=O)C=C3CCC3)C2C1 c1(C(=O)NCCC(CNC(C2(CC=C)CC2)=O)(C)C)ccc(F)c(F)c1N C(=O)(CCC(F)(F)CN=[N+]=[N-])N(CCNC(c1cnsn1)=O)CC c1(C(=O)NC(C)(CNC(=O)C=CCF)C2CC2)cnccc1Cl C(=O)(C(C)(CC)CC)NCC(CC(=O)NC(C#C)(C)C)O CC1C(C(=O)N2CC(C)(OCC(N3CCC3c3ccco3)=O)C2)=NOC1C C1(CNC(CP(C)(C)=O)=O)CCC2(CO1)CC(NC(C1CC(O)C1)=O)C2 c1(C(N(CCCOC)CCNC(=O)CSC2CCCO2)=O)ccccc1C C(C(O)C(=O)Nc1ccccc1)NC(C1C(C(C)(C)C)CCC1)=O C1(C)(C(=O)NC2(CNC(C3C(C)CCCC3)=O)CC2)CCC2(CC1)OCCO2 N1(C(c2cc(C)c(O)c(N)c2)=O)CC2CN(C(c3ccn(C)c3)=O)CC2(C)C1 c1(C(=O)NC(c2ccc(Br)nc2)CC(C)C)ccc(N2CCCC2)c(F)c1 N1(C(c2cc(Cl)c(F)cc2F)C(=O)NC(C(=O)OC)C)CCCN2CCCC2C1 N1(CCC=CC)CCC(=O)N(Cc2cccc(Cl)c2O)C1=O C(=O)(CC(CC)CC(C)C)NC(C(=O)Nc1c(CC)nn(C)c1)CC(F)(F)F C(c1ccc(S(=O)(=O)N2CCOCC2)cc1)=CC(=O)NCc1cccc2n[nH]cc12 n1(CC)cc(C(=O)NCC2COCC2NC(=O)Cc2cc(C)nn2C)c(C2CC2)n1 C12(C(=O)NCc3cc(C)[nH]n3)CCCC1CCN2C(c1cc2ncccc2[nH]1)=O C(=O)(C(C)CC(C)CC)NCc1c(CNC(C(F)=C(C)C)=O)cccc1 CCC(CC)(CO)C(=O)NC1CCN(C(c2cccc(C3CCC3)c2)=O)CC1F N1(C(c2cc(OC)n[nH]2)=O)CCC(CCNC(C2CSCN2C(C)=O)=O)CC1 c1(CC(C(=O)NC(C#C)C2CC2)NC(=O)C(O)C(C)C)ccccc1Br c1(CCC(=O)N(CC(CC)NC(c2sc(=N)[nH]c2C)=O)C)cccc(F)c1 N1(C(=O)C=CI)CCOC2(CCN(c3cc(Cl)ncn3)C2)C1 N1(C(c2c(CC)nco2)=O)CC2CC(C1)N2C(C1COCC(C)O1)=O Cc1cc(=O)ccn1CC(=O)NC1CC2CC(NC(=O)CC(C)F)C1C2 c1(C(=O)NC(c2cccc(OC)c2)C(=O)OC(C)C)c(Br)nc2n1CCOC2 N1(C(CNC(CNC(C)=O)=O)=O)CCCC(CN(C(=O)Cc2ccn(C)n2)C)C1 c1(C(=O)NCCOC2CN(C(=O)COC)C2)sc(F)cc1C.CCC(C)n1cccn1 C(=O)(CCN=[N+]=[N-])NC(C(=O)NCCCC#C)CC1CCOC1 Cc1ccc2nc(C(=O)NC3CCCC34CCN(C(=O)CC3CC3)C4)cn2c1 CC(CCC(C)(C)C)C(=O)N(C)CC1(NC(=O)C2=CSCS2)CC1 Cc1cnn2c(C(=O)N(c3ccc(O)cc3F)Cc3ccccc3)cc(Cl)nc12 c1(C(=O)NC2CN(C(c3c(C)cc(C)nc3)=O)C3C2C3)ccc2c(c1)COC2=O CCC1=C(C(=O)N2CCC(C(=O)NOCC3CC3)C2(C)C)CCCO1 N1(C(CC2CC(=O)C2)=O)CC2CC(NC(c3n[nH]cc3Cl)=O)C1C2 n1(-c2nc(C(C)OCCOC)nn2C(C)C(C)(C)C)cnc2ccccc12 C1(NC(c2cnc(NC(C)=O)o2)=O)CN(C(C2CSC2)=O)CC1F N1(C(CC(CCC)C)=O)CC2(CCC(CNC(=O)COCC3CCOC3)O2)C1 c1(C(N2CC(N(C)C(C3CCC(=C4CCC4)CC3)=O)C2)=O)ccc(N)c(CO)c1 N1(C(C2CCCN(C)C2)=O)CC2(CCCC2NC(=O)CS(=O)(=O)N(C)C)C1 N1(C(C2(CC)CCN(C(=O)Cc3csnn3)C2)=O)CC(C)CCCC1C C(=O)(C(CC(F)(F)F)NC(=O)CC(CN(C)C)NC(=O)C(C)CCOC)OC N1(C(c2c(C)[nH]cc2)=O)CCC(C)(C)C1C(N1CCCC(C)(O)C1)=O CC(CCNC(C1(NC(=O)CC(F)F)CC1)=O)CC(C)(C)C C1(C(=O)NCC2CCN(C(CCc3cn(C)nc3)=O)C2)CCOC(=O)CC1 C1(NC(C2CCCC(F)(F)C2)=O)CCN(C(=O)CCC2CC(F)(F)C2)C12CCC2 c1(C(N2CC(O)(CNC(=O)COCc3nc[nH]n3)C2)=O)cc(C(F)F)ccc1F C(=O)(C1CCCn2ncnc21)NC1CN(C(c2c(C)nc(CC)s2)=O)CC1(C)C CCC1=NOC(CC(=O)NC2(CCOC)CCN(C(C3CC(C#N)C3)=O)C2)C1 C1(NC(C2C(C)(C)CO2)=O)CN(C(=O)COC2CCCCCC2)CC12CCC2 C1(CC#C)(C(=O)N(CCCNC(=O)CC2CC2(Cl)Cl)C2CC2)CCOC1 c1(-n2c(C3(OC(c4nnc(SCC(Cl)=CCl)s4)C)CC3)nnn2)ccccc1C c1(C(=O)NC(CC2CCC2)C(=O)NCCCO)ccc(CO)cc1 C12(CNC(C3N(C(C)=O)C(=O)CC3)=O)CCC(C1)N(C(C1CC1(C)C)=O)C2 C1(Cc2cnc[nH]2)C(=O)NC2CC(C2)N1C.C(=O)(CCC1CC1)N1CCC1 CC1CC(NC(c2ncoc2C2CC2)=O)CN1C(=O)C=Cc1ccnn1C c1(C(=O)NC2C(CNC(c3c(CC)non3)=O)CC2)ccc2ccnc(O)c2n1 c1(C(N2CCC2CCCCCn2cc(C3CC=CCC3)nn2)=O)ccc(O)cc1 N1(C(C(C)NC(COC)=O)=O)CC(CNC(c2snc(Cl)c2Cl)=O)C(O)C1 N1(C(C(C(C)C)OCC)=O)CCC(CNC(=O)CCNC(=O)CO)C(F)(F)CC1 CC(C)C(C)(CNC(C1OCCC1C)=O)NC(=O)C(Cl)=CCl c1(C(N2C(CNC(CC(=O)NCC)=O)CC3(CC3)C2)=O)cc(C)c2c(c1)CCC2 c1(CNC(N2CC3C(C(=O)OC)C3C2)=O)ccc(C)nc1C c1(C(N2CC(NC(CCCCOC)=O)C(F)C2)=O)cc(C)nc(O)n1 c1(C(=O)OC)ccc(C(N2CCCC(C(C)NC(C3CCC(=O)N3)=O)C2)=O)nc1 C1(OC)CC2CC(c3nnnn3C3CCCC3)(NCC3CC4(CC4)CO3)C2C1 N1(C(c2c(C)c[nH]n2)=O)CCc2nc(CNC(C3CC3C3CC3)=O)sc2C1 C(=O)(C1=CCCN(C(=O)CC2(CSC)CC2)C1)N(C(C=C)C1CC1)C c1(NC(c2ccc(CNC(C(c3ccccc3)OC)=O)s2)=O)cc(C)ccc1C c1(C(N2CC(CN(C)C(c3cccc(OCCF)c3)=O)C2)=O)cnnc(O)c1 N1(C(C=CC2N(C(Cn3c(C)ccc3C)=O)CCC2)=O)CCCC2CCCCC12 N1(C(C2C(CC)OCC2)=O)CCC2(CC1)CC(NC(c1ccoc1)=O)CCO2 c1(CN2CC(C)(CNCc3ccc(Br)nc3F)C2)c[nH]c2cccc(C#N)c12 C(=O)(C(COC)CC(C)C)N1CC(C(=O)NCC(F)C2CCC2)(COC)C1 CC1CN(C(c2ccco2)=O)CCC1CNC(=O)CCc1ccc(C(F)F)cc1 c12ccccc1-c1ccc(cc1)CN1CCN(CC1)C2.C1(C(C)=O)CC1=C C1(C(N2CCOC(C(F)(F)F)C2)C(=O)NCC(=C)C)CC2CCC1CC2 CC1CCC(=CC(=O)NCCCC(C)NC(c2ccn(C3CCC3)n2)=O)CC1 C1(C(N(CCC(=O)N(C(CSCC)C)C)CCO)=O)CC(C)=NO1 c1(C(N2CC(CC)N(Cc3ccc(O)cc3)CC2)=O)cc(Cl)ccc1[N+](=O)[O-] N1(C(C(C)(C)F)=O)CCC(F)(F)C(CNC(C2(CC3CCCC3)CCCC2)=O)C1 C1(C)(CC)C=C(C(=O)NC2(C(=O)NCC(O)CC3CCC3)CCCCC2)C1 C1(C(=O)NCC(CNC(C2(NC(C)=O)CCCC2)=O)CO)CC=C(C)CC1 c1(NC(c2ccc(COC)[nH]2)=O)c(C)cnn1C.C12CC1C(=O)NCCNC2=O N(C1C(=O)Nc2c(Cl)cccc21)c1nccc(N2CC(=O)NC(CO)C2)n1 N1(C(C(N2CCC(C)C2)=O)=O)CCN(C(=O)C=Cc2ccc(C(N)=O)o2)CC1CF c1(CNC(=O)NCCCc2scc(C)n2)ccsc1S(C)(=O)=O c1(OC)ccc(Cl)c2c(=O)[nH]c(C(N3CCC(C)C(CO)C3)=O)cc12 c1(CN2CCCC(CNC(C(C(=O)OC)C)=O)C2)ccc(C)c(C)c1 C1(C(N2CCC(NC(=O)CCc3nnc(O)nc3O)C2)=O)CCC2(CCC2)CO1 N1(C(c2cc(O)no2)=O)CCC(O)(CNC(C2(C(F)(F)F)CCC2)=O)C1 N1(C(CN(C(C(C)C)=O)C)=O)CCCC1C(=O)NCCCc1nccs1 N1(C(C2CN(CC)C(=O)CC2)=O)CCC2(NC(=O)CC3CC3C)CCCC12 C1(N(C(Cn2ncc(C)c2)=O)C)CC2CC1N(C(C1CCC(=O)C1)=O)C2 CC(C)C(O)C(=O)NCC1(CCCNC(=O)Cc2csc(=N)[nH]2)CCCC1 c1(OC)cc(OC)c(CN(c2cccn(C)c2=O)C)c(C#N)c1 C1(NC(CC2ON=C(C)C2)=O)CCC(F)(CNC(=O)Cn2ccc(C)c2)C1 c1(C(=O)Nc2c(CC)ccc(F)c2)cc([N+](=O)[O-])ccc1OC C=CC(C)(C)CC(=O)NCC(C(F)(F)F)N1CCN(C(=O)CC2CSC2)CC1 N1(C(c2n(CCC)ncc2)=O)CC(NC(c2coc(OCC)n2)=O)CC1C C(=O)(CS(=O)(=O)C(C)(C)C)N1CCC(OC2CN(C(C(C(C)C)C)=O)C2)CC1 C12(NC(CC(=O)OCC)=O)CC(C)(C1)OC21CCN(C(=O)C(C)(O)COC)CC1 c1(N2CCc3c(ccc(C(=O)OC)c3F)C2)nccc(=NC(C)CS(C)=O)[nH]1 C1(C(=O)Nc2nccc(C(N3CC(OCC)(CF)C3)=O)n2)(CO)CCCC1C C(C1=CCN(C(C2CCC=CO2)=O)CC1)NC(CC1(OC)CCC1)=O c1(CC(CN(C(=O)CN2CCC(CO)C2)C)NC(C)=O)ccc(C)cc1 c1(C(N(CCCN(C(=O)C(O)CC(C)(C)C)C)C)=O)cc2c(cn1)OCCC2 c1(NCC2CN(C(CC(C)Sc3ccoc3)=O)C2)ncnc2cnccc12 NC(=O)CC(O)C(=O)N1CCCC(CO)(NC(c2cccc(C(F)F)n2)=O)C1 C1(CC(=O)OC)(NC(=O)Cc2cccc(F)c2)CS(=O)(=O)C1 N1(C(C(CCC)CC)=O)CCC(C2CC(NC(=O)Cc3sc(C)cc3C)C2)CC1 C12(C(=O)NC3CC(NC(C(CCC)c4ccccc4)=O)C3)CCN(CC1)CC2 CC(CS(C)=O)C(=O)N1CC(OCC(=O)NC2CC(=O)N(C3CN(C)C3)C2)C1 c1(CC)ccc(C(C(C)(C)CC(=O)c2ccccc2)COC)cc1 CCCC(C(=O)N1CCN(CC(C)NC(=O)CCCS(N)(=O)=O)CC1)C(C)C C1(CNC(CNC(CCC)=O)=O)CCCN(C(=O)C(C)(CC2CCC2)OC)CC1 N1(C(CN(CCOC)C)=O)CC(CNC(=O)CN2CCOCC2)CC1C C1(CC)C(C(=O)N(C2CCC2(C)C)C)CCN1C(=O)CNC(=O)OC c1(C(N2CCC(NC(c3ccc(CC)cn3)=O)C(F)C2)=O)ccn2c1CCCC2 n1(CC)ccc(C(=O)NC2(CC(=O)NCc3cnn(C)c3)CCC2)n1 CCC(CC(=O)N(CC(C)N(C)C(C1(F)CCCCC1)=O)C)SC C(=O)(C1=CCOCC1)NCc1cc(C(N(CC(C(C)C)OC)C)=O)on1 C(C)(C)(C(=O)N(CCCNC(c1cn(CC2CCCO2)nn1)=O)C1CC1)OC Cc1ccc(Br)cc1NC(=O)CCCCCc1n[nH]c(NC(=O)CN(C)C)n1 N1(C(C(=O)NC)CCC2OCCO2)CCC(C)=C(Br)C1 N1(C(C(CC2CN(C(C3OCCN(C)C3)=O)C2)F)=O)CCCC2CNC(=O)C12 c1(C(=O)NCCN(C)C(c2coc(Br)c2)=O)cc(OC(F)F)cc(F)c1 C(=O)(C1=CCCSC1)NC(c1ccccc1F)CNC(C1(C)CC1)=O c1(C(=O)OC)ccc(C(=O)NC2C(C(=O)Nc3ccccc3Cl)C2)c(Cl)c1 c1(CNC(c2c(CNC(c3c(C)csc3)=O)cnn2C)=O)cc(F)c(Br)cc1F C(=O)(N=c1cc2n([nH]1)CCCC2)C1CC(O)C1NC(C1=NOC(C)(C)C1)=O C1(C(=O)NC2CC(CNC(C(C(CC)C)=O)=O)C2)CCC2CC1C2(C)C C1(O)(CNC(CSCC=C)=O)COCCN(C(c2csc(-c3ncc[nH]3)n2)=O)C1 N1(C(C2(CC#C)CCCO2)=O)C2CCC1CN(C(c1cccc(CCO)c1)=O)C2 C1(CC(=O)NCC2CC(NC(c3cc(CCC)[nH]n3)=O)C2)CCCCC1C c1(NC(C(C)OC(c2cccc(C(=O)O)c2F)=O)=O)ccc2c(c1)OCCO2 C1(C(N(CC(=O)NCC(C)(C)C)C(=O)CN(C2CCC2)C)=O)CCCCC1 CN1C(=O)CCC1C(=O)N(C1CCCCC1)CCNC(=O)CC1CCC1 c1(C(N2CC(NC(C(C)(F)F)=O)C(F)C2)=O)cc(F)c(F)c(F)c1 N1(S(CCOCC)(=O)=O)CC(NCc2cccc(Br)c2Br)CC(C)C1 c1(CC(=O)N(C2CN(C(=O)CCc3cnn(C)n3)C2)C)ccnc(C2CC2)n1 n1(CCC)nc(C(=O)N(C2CCNCC2)CC)ccc1=O C1(NC(CC2(COC)CC2)=O)CN(C(=O)C(C)(C)CC2CC2)CC1C(F)(F)F C1(C)(CNC(c2cnn(C(C)C)n2)=O)CCN(C(=O)C(F)C2CCOC2)CC1 Cc1cnc(NCC2CCCC2NC(=O)CSc2ccccc2)nc1 Cc1cc(NC(c2nncs2)=O)ccc1NC(=O)C(C)n1cncn1 c1(C(C)OC(C)(C)C)ccccc1.C12CC1NCOC(=O)NC2 C1(NC(C(CC=CCC)C)=O)CC12CCN(C(c1c[nH]c(=N)s1)=O)CC2 N1(C(CCC(C)OC)=O)CCCC(C)(CNC(c2cn(C3CCCC3)nn2)=O)C1 CCC(C)(C)CC(=O)NCCCC(C)NC(=O)C(C)C1CCCO1 CCCCCCCN(C(=O)CC1CN(CCNC(C)=O)CCO1)C(C)C c1(N2CC(NC(c3c(C)oc(CO)c3)=O)C(C)(C)C2)ncc2c(n1)CCOC2 C1(C(=O)NC(C2(C(N(C3CCN(CC)CC3)C)=O)CC2)C)CC2C=CC1CC2 c1(CC)oc(C(=O)NC2CCN(C(=O)C(c3cn(C(C)C)nn3)=O)C2)cc1C N1(C(c2nn(C)c(Cl)c2)=O)CC(NC(c2ccc(I)cc2O)=O)CC(F)(F)C1 C1(NC(C2N(S(CC)(=O)=O)CCC2)=O)CC2CC1N(C(=O)CN(C)C(C)C)C2 c1(CC)ccc(NC(C23CC(CO2)N(C(=O)CC2CC2(C)C)C3)=O)c(C)c1 c1(CC)cc(C)cc(NC2CCCN(C3CCOCC3)C2=O)n1 CC1CN(C(=O)C(C2CCCCC2)O)CCC1Nc1ncncc1Br C12(NC(C(CNC(c3cc(C(N)=O)no3)=O)O)=O)CCN(CC1)CC2 C=C(F)C1(CC(=O)NCC(C)(C)NC(c2ccc(CN(C)C)[nH]2)=O)CCC1 c1(C(N2CCC(N(C)C(c3cnc(O)c(Cl)c3)=O)C2)=O)ccc(C#N)cc1F CCCC(CC)C(=O)N1CCOCC1CNC(c1cnn[nH]1)=O C1(CNC(c2c(OC)ccs2)=O)CCCC1CN(C)C(=O)C(CO)N(C)C N1(C(C(CC)=CC)=O)CCC(C)N(C(=O)C(c2ccncc2C)C)CC1 c1(C(=O)NCC(C(C)C)NC(c2ccn(CCC)n2)=O)cccc(C(F)F)c1 Cc1n[nH]c(C)c1S(=O)(=O)N1CCC2(CC1)CN(C(C1CC1F)=O)C2 c1(CC(=O)NC2CCC(CNC(CCC3CC(OC)C3)=O)C2)ccc(C)nc1Cl Cc1ccc(C(N2CCN(CC(=O)NC3CCCC(C)C3)CC2)=O)c(O)n1 CCC(C)C(C)CNC(C1(NC(=O)Cc2cnn(C)c2C)CCCC1)=O c1(CNC(c2cccc(SCC(F)(F)F)c2)C)ccc(F)cc1Br C1(CNC(COCCC#C)=O)CN(C(c2cc(C(F)F)[nH]n2)=O)C2(CCC2)C1 C(=O)(CC(C)C(C)(C)C)N(C(CC(=O)NCCCC#C)(C)C)C c1(CC)cc(C(=O)NC2CC2NCCOC(F)(F)F)cc(C)n1 Cc1coc(C(=O)NCc2cccc(CNC(=O)Cc3ccco3)c2)c1C C(C1c2ccsc2CCN1C(=O)CC1CC1)NC(=O)CCOCC1CCOCC1 Cc1c[nH]c2ncc(C(=O)NCCC3CCCCN3C(C3CC(C)(F)C3)=O)cc12 C(c1ccc2ccccc2c1)=CC(=O)NC12C(CN(C(C3N(CC)CC3)=O)C1)C2 c1(CC(N2CCC(F)(CNC(COC)=O)C2)=O)ccc(Br)cc1C(=O)O N1(C(COC)=O)CCCCC1CCNC(c1cc(CO)on1)=O.C(=O)(CSC)N(C)C C(=O)(C1=NNC(=O)C1)NC1CC(CNC(c2cc(SCC)ncc2)=O)C1(C)C N(C1CCCc2c[nH]nc21)C(C1N(C(CC(C)(C)OC)=O)CCCCC1)=O c1(C(=O)NCC(C2CC2)NC(C(C)SC)=O)ccccc1C(C)(F)F Cc1cc(=O)n(C)cc1C(N1CC(C(N)=O)(CNC(C2(C)CCCC2C)=O)C1)=O Cc1ccc2[nH]c(C(N3CCC(C)C3CNC(=O)CC3C=CCC3)=O)cc2c1C c1(C(=O)NC2(CNC(C3CC3(F)Cl)=O)CCCCC2)csc2c1CCCC2 Nc1ccc(-c2cn(C3(C(=O)Nc4cc(Cl)c(F)cn4)CC3)nn2)cc1[N+](=O)[O-] N1(C(c2c(OC)nsc2)=O)CCCC2(CC(NC(=O)C3=CSCCO3)CO2)C1 C1(NC(c2ccc(C)o2)=O)CC2CC(C1)N(C(c1ccc(CC#N)cc1)=O)C2 C1(C#N)(C(N2CCCN(C(C(=O)NC(C)C)=O)C(CO)C2)=O)CC2CCC1CC2 c1(C(=O)NCCC2CC(NC(CCOCCN(C)C)=O)C2)[nH]nc2ncccc12 c1(-c2c(C#N)ccnc2)nc2c(s1)CC(C(=O)NCCn1cc(CO)nn1)CC2 CC(C)(F)CC(=O)NC1CCN(C(=O)C2CC2)C1n1cccn1 Cc1cccnc1S(=O)(=O)N1C(=O)CCC1C(N1CC(O)C(O)C(O)C1)=O Cc1nc(C)n(CCC(=O)NC2CCN(C(=O)CSCCC(C)C)C2C2CC2)n1 c1(C(C(=O)NC(CC)CN(C)C(c2csnc2C)=O)OC)ccc(F)cc1 c1(C(N(C)CCC2CCN(C(C3CC3F)=O)CC2)=O)ccnc2ccccc12 CCC(C)(CNC(=O)C(n1cc(Cl)cn1)C)NC(c1ccn(C)c1)=O c1(C(=O)NCC2C(CNC(c3cc(C(C)=O)oc3)=O)C2)cc(C)nc(O)c1[N+](=O)[O-] N#Cc1ccc(C(N2CC3(CC(CC(=O)Nc4cc(Cl)ccn4)C3)C2)=O)cc1F C1(C(N(CCN(C(=O)C(F)(F)CO)C(C)C)C)=O)CC2CCCN2C(=O)N1 N1(C(C2CCCC2)=O)CCCC(O)(Cn2cc(C(C3CC3)C3CC3)nn2)CC1 Cc1ncnc(C)c1CC(N1CCC(NC(C2CCOC(C(C)C)C2)=O)CC1)=O N1(C(C(c2cn(CC)nc2)(F)F)=O)CCOC(CNC(=O)C(C)(C)CC2CC2)C1 C1(CNC(=O)CNC=O)CCC(F)(F)C1.C12(COC)CN(C1)C2=O N1(C(c2cc(C)sn2)=O)CCC2(CCC2NC(C2CNC(=O)CC2(C)C)=O)CC1 N1(C(CC(=O)NCC)=O)CCN(C(=O)C(CC)SC)CC1CO N1(C(C2(CCC=C)CC2)=O)CCN(C(=O)C=Cc2cncnc2O)C(C2CC2)C1 CC1CC(NC(=O)CCCCCF)CN(C(c2cccc(C(F)F)c2F)=O)C1 N#Cc1cccc(C2CC2C(N2CCC(CNC(C3CC4CCC(C3)O4)=O)C2)=O)c1 C1(c2cccs2)(CC(O)COCCC(F)(F)F)CCCCC1 Cn1cc(C(=O)O)c(C2CCCN(C(C3CC3c3ccccc3Br)=O)C2)n1 C1(NC(COCC=C)=O)CCCC(C(=O)N(c2cncc(C)c2)C(C)C)C1 c1(CC(=O)N(CCNC(=O)CC2CC=CC2)CC)ccc(O)cc1Cl c1(OC)ccnc(CNCC2CN(Cc3ccccc3)CCS2)c1F C(CCN=c1cc[nH]cc1[N+](=O)[O-])N(C)C(C1(C)CCC(=O)N1)=O Cc1nc(Cl)ccc1CC(=O)NC1CC2CC(NC(=O)C(C)(C)CO)C2C1 N1(C(C2(COCC)CC2)=O)CC2CC1CC2NC(=O)CC(C)c1ccccc1 C1(C(=O)NC(C#C)C(C)(C)C)CCC2(CC2)N1C(=O)CS(=O)CC Cc1cc(C(N2CCC(CCNC(c3csc(Cl)n3)=O)CC2C)=O)c(N)c(F)c1 c1(N2CCN(CCOC)CC2)nc(=NCC(C)n2cccn2)[nH]c2c1CCCC2 Cc1cnc2n1C(C(=O)N1CC(NC(=O)CNS(=O)(=O)c3ccccc3)C1)CCC2 C1(C(=O)NCC=CC(=O)N(CC(O)CF)C)CCOC1(C)C c1(CC(N2CC(OCC(=O)NC3(COC)CCC3)C2)=O)cc(C)on1 c1(N2C(CCNC(c3ccc(CC4CCCC4)cc3)=O)CCC2)nccnc1F c1(CC(N2C(C)CCCC2)=O)cc(F)c([N+](=O)[O-])cc1F c1(OC(C(N2C(CNC(c3cc(C)ncn3)=O)CCC2)=O)C)cccc(C)c1C N1(C(c2ccccc2F)=O)CCN(N2CCCC2)CC1CC(F)F.O=CCN N1(C(CSC)=O)CC(C)(CNC(=O)CC2CC3C=CC2C3)CC1(C)C C12(C(N(CCN(C)C)CC)=O)CCN(C(c3cccc(CC#N)c3)=O)CCC1C2 N1(C(C2C(CC)CCO2)=O)CC(C)(C)CC1C(=O)NOCCOCc1cnn(C)c1 C(=O)(CCCCC(=O)NC(C)(C)C(C)NC(c1csc(O)n1)=O)NC CCC(O)C(C)(C)C(=O)NCC(CC(=O)NC1(CO)CC(OC)C1)C1CCC1 Cc1cc(N2CCC(CC(C)(C)C)C2)nc(N(CCCCN(C)C)C)n1 c1(CCNC(c2cc(OC)n(C)n2)=O)cc2cccnc2[nH]1 C1(CC(=O)NC2CN(C(C3CCC(CC)CC3)=O)CC2F)CCC(C)(C)CO1 N1(C(C(C)(C)CF)=O)CCC2(CCCCC2NC(c2cc(O)nc(Cl)c2)=O)C1 C=Cc1ccccc1-c1cc(C(=O)NC(CO)C(=O)OC)n[nH]1 CCC(CC)C(=O)NC1(C2CN(C(C3CC3c3cccc(C)c3)=O)CCO2)CC1 N1(Cc2c(OC)cccc2)CCCC2(C=CCO2)C1.C1(=O)CCN1 CC(C(=O)N(C)CC1CN(C(c2ccc(C3CCCOC3)cc2)=O)C1)C(F)F C(=O)(C(C)(C)CC(=O)NCC1CC(C)N(C(C2CC3(CC(=O)N3)C2)=O)C1)OCC c1(NC2(c3n(C4(C)CC4)nnn3)CCCSCC2)ccc(F)c(S(N)(=O)=O)c1 Cc1csc(=O)n1CC(=O)N(C1CCCS(=O)C1)C(c1ccccc1)C c1(OC)cc(C(=O)NCC(CC(F)F)c2ccccc2)cc(NC)c1OC N1(C(c2ccc(C)cc2)=O)CC2(CCC(Nc3cc(C(C)C)nc(C)n3)CC2)C1 O=C(CCCCNC(C1CC1C1CCCO1)=O)NCc1cn(C2CC2)nn1 C1(CNC(CCc2onc(CCC)n2)=O)CN(C(c2ccc(F)o2)=O)CCO1 C(=O)(CCS(=O)(=O)CC(C)C)NCC(CCNC(C1CC=C(C)CC1)=O)O CCC(CC(=O)N1CCC(CO)(CNC(=O)COc2cn[nH]c2)C1)CC(F)(F)F CC1(NC(c2ccc(O)c(Cl)n2)=O)CCC(NC(=O)C(C2CCOCC2)O)CC1 C1(C=O)C(C)CCN1N(CC)CC.c1(C=O)cnc(NC(=O)C=CCOCCO)o1 CCC(CN(C)C)CC(=O)N1CCCC(NC(=O)C(=Cc2ccco2)C)C1C C1(C)(C(=O)NC(C=C)C2CCC2)CCCN(C(c2cc(C(N)=O)co2)=O)C1 c1(C(=O)NC2C3CN(C(C(COC)Cl)=O)C(C3)C2)cc(Cl)cc2cccnc12 CCN=C(NCC1CCC(F)(F)C1)NC1CCCC(F)C1 S(=O)(=O)(c1c(Cl)cc(Br)cc1Cl)N1C(C)(C)CCC(c2c(C(C)C)nnn2C)C1 N1(C(C=CSC)=O)CCCN(C(=O)CNC(=O)Nc2ccc(F)c(F)c2)CC1C C1(NC(CCC#CC)=O)COCCN(C(=O)CCCSC(C)(C)C)C1 C1(C(N(CCN(CC(C)C)CC)CC)=O)CC2OC1C1CC21.C1(=O)CN1.C(=O)(C1CC1)N N1(C(CCC=C(C)C)=O)CCC(O)(C(C)CNC(=O)CCc2ccc(C)nc2)C1 C1(C)(CNC(C=CSC)=O)CC(F)(F)CN1C(C1CC2(CCCC2)CO1)=O c1(C(=O)NCC(C)CNC(C2CCC(O)CC2)=O)ccc(N(C)C)cc1F N1(C(c2n(C)c(F)nc2)=O)CCC(NC(c2cc(O)nc(O)c2)=O)C(F)C1 N1(Cc2ccc(-c3ccc(C(=O)NC(C)(C)C)cc3)cn2)CCn2cncc2C1 Cc1ccc(Cl)c(OCC(=O)NCCN(C(C2C3CC4C(C3)C24)=O)C(C)C)c1 c1(N2CCC=C(C)C2)ccn2ncc(S(=O)(=O)NCCc3cc(O)ccn3)c2n1 C=CCC(C(=O)NC(CO)C(=O)NCc1ncc(CC)s1)C(C)C N1(C(C2(CC)CCOCC2)=O)CCN(C(=O)CCCC(F)F)C(CCOC)C1 CS(=O)(=O)C(C(=O)NCC1CCCCC1NC(c1cn(CCO)nn1)=O)C1CC1 Cn1ccc(CCC(=O)NCCOC2CCN(C(=O)CC3OCCO3)C2)n1 N1(C(CCOCC#C)=O)CCCN(C(c2ccc(F)cc2NS(C)(=O)=O)=O)CC1 C(=O)(CN=c1[nH]c2c(c(=NC3CC3C3CCC3)[nH]1)COCC2)Nc1ncc(C)nc1 N#Cc1ccccc1C1CCN(C(=O)CCCn2ccnn2)C1 N1(C(C(C)(C)F)=O)CCC(CNC(=O)C=Cc2ccco2)CC1 Cc1cc(CNC(=O)COC2CCN(C(C3(Cl)CC3(F)F)=O)C2)cc(C)n1 C1(N(C(c2c(C(F)(F)F)cnn2C)C(=O)NC2CCC2)C)CNC(=O)C12CC2 Cc1nnccc1C(=O)NC1CC(C(C)NC(C2CC(OC(C)(C)C)C2)=O)C1 c1(C(N2CC(=C(CNC(COCCC=C)=O)F)C2)=O)cc(F)ccc1Br c1(C(N2CC(CCc3cn(CC(CC)CC)nn3)C2)=O)cc(C)ccc1F CC(C)C(C)CC(=O)NCC1CCC(CNC(=O)CC2CC(C(C)(C)C)C2)C1 N1(C(CC2CC(CC)C2)=O)CCCOC(CCNC(=O)CCn2cncn2)C1 c1(C(=O)NC2C(NC(=O)CCc3ccoc3)CC2)ccc(Br)o1 C1(CC(=O)OCC)CCCCN1C(c1cnn(C(F)F)c1)C(=O)NCC1COC1 C1(CNC(C2(SC)CC2)=O)C(C)CCCN1C(c1nc(O)c(C)s1)=O Cc1nc(-c2ccccc2)ncc1C(N1CCCN(C(C2C(C)C2C)=O)CC1)=O c1(CC(=O)NCCCC(C)NC(c2cnc(CC)[nH]2)=O)coc2cc(C)ccc12 c1(C(=O)NC(CCNC(CC2CC(OCC)C2)=O)C)ccc(C)nc1N C(C)(C(=O)NC12CC(C1)N(c1nnc(C)s1)C2)(C(C)C)NC(C)=O C(=O)(C(C)CC(F)(F)F)NCC1N(C(c2cc(C)n(C(F)F)n2)=O)CCC1 N1(C(CC(=O)NC)=O)CCCCC(NC(c2ccc(=O)n(CCOC)c2)=O)CC1 C1(C(C)C)N(C(C2(NC(=O)CC3CCCC4CC34)CC(F)(F)C2)=O)CC1(C)C C(=O)(C1=C(C#N)CCC1)NC1CCC(NC(Cn2c(=O)sc(C)c2C)=O)C1 CC(=O)CCCCCCC(=O)N1CCC2(CCOC2)C(C)C1 C1(NC(C(C2CCOC2)OC)=O)CCCCC1CNC(=O)CCC=C(C)C N1(C(C=CC=CCC)=O)CC(F)CC1C(=O)Nc1cnn(C(F)(F)F)c1 C1(C(N)=O)CN(C(=O)CN2CCC(OC)C2)CC1C(C)C.C12CC(C1)CNC2=O N1(C(C2CN(C(C(CC)NC(N)=O)=O)CC2C)=O)CC2CC1CN2C C1(NC(c2cnc[nH]2)=O)CC2(C1)CN(C(C1CC=CCC1)=O)C2 C1(C(=O)NC2CC(CNC(C34CCCC3CC4)=O)C2)CCCN2CCCC12 N1(C(C(C(C)C)n2cnnc2)=O)CCCCC(N=c2[nH]nco2)C1 C1(C(=O)N(C2CC(NC(C3CC(OC(F)(F)F)C3)=O)C2)C)(NC(C)=O)CCOC1 c1(C(N2C(CCCC)CCC2)=O)cc2ccncc2c(O)n1 C1(C(N(CCCCNC(=O)C(F)=C2CCCC2)C)=O)(CF)CC1(F)F c12ccc(s1)c(=O)n2CCC.C1(C(=O)NCCCSC)CC(C(=O)OC)C1 C1(C(=O)NCCCCN(C)C)CCOCC1NC(c1nccnc1N)=O C1(C(=O)NCc2cc(OC)nn2C)CN(C)CCN1C(c1cnc(Cl)s1)=O N1(C(C(C)CF)=O)CC=C(CCNC(c2cc(-c3ccccc3Cl)no2)=O)CC1 CC(CF)CC(=O)N(C)Cc1ccc(CNC(C2CC(C)(C)CO2)=O)cc1 C1(C(=O)NCc2cccc(-n3cc(C(COCC)C)nn3)c2)CCC2(CCC2)C1 C(CNC(c1ccc(O)cn1)=O)(C(C)(C)C)NC(C1CN(C(C)=O)C1)=O n1(CCC(=O)NCC2CCC(CC)CC2)cnc2ccccc12 c1(NC(C)=O)cc(C(N2CC3(CC3)CC2C(=O)Nc2cnc(C)s2)=O)cc(C)c1 CC1CCC(CNC(C23CCC(C2)C3)=O)CN1C(=O)CNC(=O)C1CC1 C(=O)(C#CC1CCC2(CC1)OCCO2)N(CCN(C(C(C(CC)C)OC)=O)C)C C1(C(=O)NCC(C)(C(C)C)NC(c2c(C)cc(SC)o2)=O)CC2(C1)CS(=O)(=O)C2 N(C1CCc2cc(CNC(C3CC(O)C3)=O)ccc21)C(c1ccc(CC)cn1)=O Nc1ccc(F)c(F)c1C(N1CCC2(CC(NC(C3CCCN3C=O)=O)C2)C1)=O C(CCCCC(=O)NCCN(C(c1ccc(CO)o1)=O)C1CC1)OC CCC(CC(C)C)C(C(=O)NCc1ccc(OC)cc1)N1CC2COCCC12 C1(CCC)COCCN1C(=O)CCN(C(=O)COC(F)(F)F)C1CC1 CCCCCC(O)C(=O)N1CCC(NC(c2nn(C)c(C3CC3)c2C)=O)C1C C1(NC(C(CC=C)C)=O)CC2CN(C(C3CCC(C)O3)=O)CC2C1 n1(CC)nc(C(C)C)cc1C(N1CC(NC(C2(C)CC=CCC2)=O)C(O)C1)=O c1(OC)cc([N+](=O)[O-])ccc1C(N1CCN(C(=O)COCCN(C)C)CC1)=O Cc1nc(C(=O)NCC2(C)CCC(NC(c3cccc(C(N)=O)n3)=O)C2)n(C)n1 c1(C(N2CCC(CC)C2C(=O)NCc2nnn(C)n2)=O)cc(O)cc(F)c1 N1(C(=O)Cc2cccs2)CCN(C(=O)C(F)(F)C2CC2)CC1c1cccc(F)c1 c1(C(=O)NCCOCC(N2CCC(CC)C2)=O)ccc(C)cc1C c1(C(=O)NC(C2CCCCN2C(c2nnn(C)n2)=O)C)cc2ccccn2c1 Cn1cnc2c(C(=O)Nc3ccc(NC(c4ccccc4)=O)nc3)cccc12 c1(C(=O)NCC(CN(C)C(C2CCCN2CCCO)=O)(C)C)ccc(CO)cc1 C12CC(C)CN(C1)C(=O)C2.CCC(C)C(=O)N1CCC(NC(=O)OC)C1 c1(C(N2C(CCNC(C3C(=C)CC3)=O)CCCC2)=O)cc(C)c(N)cc1F C(=O)(C1CCCc2ncnn21)NCC1(OC)CN(C(=O)CC2CC(C)OC2C)C1 CC(C(=O)NCC(C1CC1)NC(C12CC(C)(CCO1)C2)=O)C(F)(F)F C12CC(O)CN1C(=O)CCC1CCC(C1)NC2=O.C1(CN(C)C)CC(C)(O)C1 c1(OC)cnc(Cl)cc1C(=O)N(CCCNC(C1CC12CC2)=O)C(C)C C1(NC(=O)OCC)CC(O)CN1N1CC2C=CC2C1 c1(CCC(=O)NC(CCOC)CNC(c2ocnc2C2CC2)=O)ccccc1Cl N1(C(CCC)C)CC(C(N2CC(NC(C3CC(=O)N(C)C3)=O)C2)=O)CC1=O C1(NC(Cc2n(C)ncc2Cl)=O)CC(O)CN(C(c2cnc(O)cc2O)=O)C1 c1(C(=O)NC(COC)CC(=O)NC2C=CC(CO)C2)cc2cccnc2[nH]1 c1(C(N(CCC)CCNC(=O)C(C(C)C)n2cncn2)=O)cc(N)cc(O)c1F c1(C(=O)NC(C2CCCN2C(C2CC2C2CC2)=O)C)cccc(C2CC2)c1 c1(NC)c(C(=O)NC2CC3CN(C(=O)CC4CC4C)CC3C2)cccc1[N+](=O)[O-] C1(C(=O)NC(CNC(C(CSC)O)=O)(C)C)CN2CCN1CC2C C1(CNC(c2ccn(CCCC)n2)=O)CN(C)CCN1C(=O)Cn1ncnn1 N1(C(=O)NC2Cn3c(C)cnc3CC2)CCN(C)C2(CCC2)C(C)C1 N1(C(C)=O)CCN(C(=O)Nc2cc(Cl)cnc2C)c2c(Cl)cccc21 c1(C(=O)NCc2ccc(C(=O)NC3(CC#C)CCC3)o2)cc(O)cc(=O)o1 c1(Cn2ncc(C(=O)NCC(C)NC(C3C(=C)C3)=O)c2)ccccc1F C1(C(CNC(C(C)n2cnnn2)=O)=O)(NC(C2(Cl)CCC2)=O)CCCC1 N1(C(C(N2CCCC(CC(=O)OC(C)C)C2)=O)=O)CCC2(C1)CN(C)C(=O)CO2 c1(C(N(C2CCCOC2)C)=O)cccnc1CNC(c1ccccc1F)=O N1(C(CCCOC)=O)CCCCC(NC(=O)C=CC2CCCO2)C1 c1(CC)ccc(C)c(C(=O)NC2CCCCN(C(c3cscc3OC)=O)C2)c1 N1(C(c2nnc(CC)s2)=O)CC(NC(c2ncccc2OC)=O)CC2(CC2)C1 c1(C(=O)NCC(CNC(C2CC(C(C)(C)C)C2)=O)O)cccc2[nH]ccc12 c1(C(=O)NC2CCCCCN(C(C(C)O)=O)C2)cn(C)c2ncccc12 C=CCC(C)(C)CC(=O)N1CCC(CC(N2CCC2(C)CC)=O)CC1 N1(C(C(n2cc(-c3c(OC)ccs3)nn2)C)=O)CCOC(c2ccccc2Cl)C1 c1(CC)ccc(C(=O)NCC(C2CCN(C(C3(O)CCOC3)=O)CC2)F)cn1 c1(CC)cc(C(=O)NC2CN(C(=O)CC3CCOC3=O)CC2F)cc(Cl)c1 CN1CCC(C(=O)NCc2nccn2C)(NC(=O)CC2CCCOCC2)C1 c1(N(C)Cc2c(C)cnn2C)nccc(=NCC2C(F)(F)C23CCCC3)[nH]1 C#Cc1cccc(C(=O)NCC2CCN(C(=O)CCc3nnc(C)o3)C2)c1Cl C1(CC(=O)N(CCCOCCN(C(=O)CCF)C)C)(CO)CCC1 C(C(C)(C)CNC(=O)COCC1CCCOC1)NC(C1C(OCC)C1C)=O N1(C(C2(COC)N(C(CCC(=O)NC)=O)CC=C2)=O)CC2CCCC(C1)N2C C1(C2CC2)(C(=O)NCC2(F)CC(NC(CNC(C)=O)=O)C2)CCOCC1 CC(C)C(C(C)NC(=O)CC(C)(C)C)NC(c1ccnc(C(F)F)c1)=O C1(NC(c2cc(OC)no2)=O)C2CC1N(C(=O)CN(CC(C)C)C1CC1)C2C c1(C(=O)NCC2CN(C(C3CC34CC4(F)F)=O)C2)cccc2c3c([nH]c12)CCC3 N1(C(C(C=C)(C)O)=O)CCN(C(c2cc(C3CC3)n(CC)n2)=O)C(CC)C1 c1(CNC(C2CCCCCC2)CC)cnc2ccccn12 c1(C(N2CCC(O)(C(C)NC(c3nc(CCC)sc3)=O)C2)=O)cnc(O)c(F)c1 C1(NC(CC2(NC(C)=O)CC2)=O)CCN(C(c2cc3sccc3[nH]2)=O)CC1O c1(OC)cccc(C=CC(N2CC(N(C)C(c3ccn(C)c3)=O)C(C)(C)C2)=O)c1 C1(NCCNC(CCCCCc2n(CC3C(C)C3)nnn2)=O)CCC(=O)NC1(C)C C(=O)(C1CCCn2cc(C(C)(C)C)nc21)NCCCN(S(C)(=O)=O)C C(=O)(CCCC(F)(F)CO)NC(CC(C)C)(C)CNC(c1c[nH]nc1F)=O C(=O)(CC(C)P(C)(C)=O)NCCNC(c1[nH]cc(OC)c(=O)c1)=O C1(NC(c2ccc(COC)cc2)=O)(CNC(=O)COCC(F)F)CC2CCC1C2 C1(=CC(=O)NCC(CCNC(C2CC=C(C)CC2)=O)O)CCOc2ccccc21 N1(C(COCCCC)=O)CCCC(NC(=O)CCC2CCCC(=O)N2)CCC1 CC(C)C1=NOC(C(N2CC(F)(F)CC2CCNC(=O)C=Cc2ccsc2)=O)C1 O=C(CC(C(F)F)N1CCOCC1)NC1CC(F)(CNC(c2nc(Cl)cs2)=O)C1 c1(C(=O)NCCCCNC(=O)Cn2cc([N+](=O)[O-])cn2)cccc2onnc12 C1(NC(c2ccc[nH]2)=O)CN(C(c2cnn(C3CCCC3)c2)=O)CCC1O CC1(C)CC(O)CN1C(=O)CC1CC(NC(=O)CNc2ncccn2)C1 c1(OC)cc(C)c(CC(N2CC3(CCCN3C(c3ccoc3C)=O)C2)=O)c(C)c1 c1(C(=O)NCC(CC=C)NC(C2C=C(C)CS2)=O)ccc(C(C)C)cc1F c1(CC)cc(C(=O)OCc2cn3cc(Br)ccc3n2)cc2c[nH]nc12 N(C1CCc2c(C)cccc21)C(=O)Nc1n(C)nc(C)c1Cl C1(N(C)C)CCCC(CCCCNC(=O)NCc2cc(=N)[nH]o2)C1 CC(O)C(C(N)=O)NC(c1ccc(CNC(c2ccc(C(F)F)o2)=O)cn1)=O N1(C(=O)NCCCl)CCC2CN(Cc3ccnc(F)c3)CC12 CC1CC(c2cn(CC(F)(F)F)nn2)CCN1C(c1cc(Cl)sc1Br)=O CC1CN(C(=O)C=CCNc2ccccc2)CCC1NC(=O)COC1CC=CC1 C12CCN(CC1)CC2.c1(CNC(CCSC)=O)ncnn1C(C)(C)C c1(C(=O)NCC2N(C)CCN(C(C3CC(=O)N3)=O)C2)nc2cncnc2nc1O C1(OC)CN(C(=O)CCC2CCCOC2)CC1NC(c1cc(C)cs1)=O N1(CC)C(=O)CCC1C(=O)NCCC(C)CCNC(=O)C(F)(F)C1CC1 C(=O)(CC1COc2ccccc21)NCCNC(C(C(C)O)(C)C)=O Cc1ccc(C)c(OCCC(N2CC3(NC(C4CC(CCO)C4)=O)CC2C3)=O)c1 C1(C)(C(N2CC(OCCNC(CC(CC)C3CC3)=O)C2)=O)CC2C=CC1C2 N1(C(C2(N(C)C)CCC2)=O)C2CCC1CC(NC(C1(C)CCC(=O)NC1)=O)C2 C12(CCC(=O)NC(c3ccn(C)c3)(C)C)CCC(CC1)C2 c1(NC(=O)NCCC(=O)NCc2ccccc2Br)cccc2c1NCC2 c1(C(N2CCC(NC(CCC=C(C)C)=O)C2C)=O)nc(Br)n2ccccc12 C1(NC(C(CC)C(C)C)=O)CN(C(=O)C(C)(C)C2CCCC2)CC(F)(F)C1 C1(NC(c2cc(C(=O)OC)[nH]n2)=O)CCN(C)C(NC(=O)NCc2ccco2)C1 N1(C(C(C)OCCC=C)=O)CC2CC1C2CNC(c1ccc(C(C)(C)C)nc1)=O N1(C(C2(C#C)CC2)=O)CCC(N(C(=O)Cc2ccn(CC)n2)C)C1 Cn1cc(C(N2CC=CC2CNC(=O)CCN2CCOCC2)=O)cn1 C1(c2n(CCSC)nnn2)(NC2CCC3(CC3)C2)CCCC(C2CC2)C1 CON1CCC(C(=O)NCCC(=O)NCCC(F)(F)CO)CC1 N1(C(C2N(C(C)C)CCC2)=O)CCCCC(N(C)C(c2cn3c(n2)SCC3)=O)C1 CN1C(=O)C(C(=O)NC(C(=O)NCc2ccc(Cl)cc2)C2CCCC2)CC1=O C(c1cc(F)c(O)c(F)c1)=CC(=O)NCC(F)CNC(c1cnnc(O)c1)=O c12ccc(nc1)C(=O)NC1CC(C1)CCNC(=O)CNC2=O.C1(CC2CC2)CC1 N1(C(CCc2ccc(C)o2)=O)CCC(NC(C2CCN2S(C)(=O)=O)=O)C(O)C1 N1(C(C(CC)(C)C)C(=O)NCc2ccccc2Br)Cc2ccc(O)cc2C1 N1(C(c2scc(C)c2C)=O)CC2(CCN(C(=O)Cc3ccsn3)CC2)C1C(C)C C12(C(=O)NC3CCN(C(=O)COc4ccsn4)C3)CC=CC(C1)OC2 c1(C(N2CC(C(=O)NC3CCCN(C)C3)NCC2)=O)ccc2nncn2c1 c1(C(N2CCC(CC(C)C)C2)=O)cn2c(n1)CCN(C1CCC(C)(C)C1)CC2 NS(=O)(=O)c1ccc(CC(=O)NCCCCC(CO)NC(=O)CC2CCCO2)s1 N1(c2ccnc(C)n2)CC2CCC(NC(c3coc(C(C)C)n3)=O)CC2C1 c1(CC(=O)NCCOCCNC(=O)Cc2ccns2)ccc([N+](=O)[O-])cc1Cl C(=O)(CC(C(F)F)OC(C1(C(c2ccccc2)OC)CC1)=O)OCC C(=O)(C(C)(O)Cc1ccccc1)NCCCCNC(CC1(OCC)CC1)=O c1(OC)ccc(C(C(=O)O)NCc2cc(-c3ccc(Cl)cc3)on2)cn1 C1(COC)(CNC(=O)CC(c2c(C)noc2C)C)CCCN1C(=O)C(C)C1CC1 C1(NC(CCc2ccc(C#C)cn2)=O)CC2CCCC(C1)N2C(=O)C(C)CC Cc1ccncc1C(=O)NC1CC1C(=O)Nc1cnsc1 C#Cc1ccc(CNC2(O)CN(C(=O)CN3CCC(OC)C3)C2)s1 CC1CN(C(=O)CC2CCCN2C(=O)Cc2cc(Br)ccc2O)CCC1O C1(CNC(C2CCN(CC)C2)=O)CN(C(=O)C=CCN2CCCC2)CC12CC2 Cc1occ(C(F)(F)F)c1C(N1CC(CNC(=O)C=Cc2cscn2)C(O)C1)=O c1(C(N(CC(C)NC(C=CCC)=O)C)=O)ncnc(C)c1C N1(C(c2c(C)n[nH]c2)C(=O)NCC2CCOCC2)CCOC(CC(C)(C)C)C1 c1(C(=O)NC(CNC(C2(COCC)CC2)=O)(C)C)nn(C)c(=O)cc1C C1(C(C(=O)NC)N(C2CCN(C(=O)OC(C)(C)C)C2)C)CCC(C(=O)OC)CC1 C1(C)(C(N2CCC(C(C)NC(=O)C=CCOC3CCOCC3)C2)=O)CC=CCO1 Cc1c(NCc2conc2C(F)(F)F)ncc2ccccc12 N1(C(C2(C(F)(F)F)CC=CCO2)=O)CCCCC1CC(O)C(F)(F)F c1(C(=O)NC2CCCN(C(C3(CO)CC(C)(C)C3)=O)C2)cc2ccsc2s1 c1(CC)ccc(Br)cc1C(=O)NCC12CCC1CN(C(=O)CC13CC(C1)C3)C2 c1(C(=O)NC2(C)CCN(C(c3c(C)n[nH]c3C)=O)C2)ncc2[nH]ncc2n1 c1(C(=O)NC2(CO)CCN(C(c3c(CC)oc(C)c3)=O)C2)ccc(Cl)c(OC)c1 C1(NC(c2cccc(OC)n2)=O)CCC12CCN(C(C1CCCN1C=O)=O)CC2 Cc1sccc1C(=O)NCC(F)CNC(=O)C(F)(F)C1CCOCC1 C1(CC)CN(C(=O)CC2CCN(C)C2=O)CCN1C(=O)Cc1ccc(OC)nc1 C1(CNC(c2ccc(C)nc2O)=O)CC12CCN(C(C1(CO)CCCO1)=O)CC2 c1(OC)cc(C(=O)NCC23CCC(C2)N(C(=O)COC(F)F)C3)ccc1C O=C1NC(C(=O)NC2CC2CNC(=O)Cn2cc(C3(CO)CC3)nn2)C2CCC12 C12(CNC(c3c(CCC)n[nH]c3)=O)CC(CO1)N(C(c1ccc(C3CC3)s1)=O)C2 C(C(C)(C)C(=O)NC1CC2(C1)CC2CNC(C1CN(S(=O)(=O)C(F)F)C1)=O)OC c1(CCC(=O)NCC2CC(O)CN2C(=O)CN2CC=CC2)cnc2n1CCOC2 C1(NC(c2nc(C(C)OC)sc2)=O)CN(C(c2cc(C3CC3)[nH]n2)=O)C(C)(C)C1 N1(C(CCCC=C)=O)CCC2(CCCCN(C(c3c(C)nn(C)c3OC)=O)C2)C1 N1(C(CN(C2(CS(N)(=O)=O)COC2)C)=O)CCCCC1CN(C)C c1(OC)cc(O)ncc1-c1nc(-c2ccoc2)nn1CCSC.C1(C)CCCCC1 C1(C#N)(C(N2CCC(C)(NC(C3CCCSC3)=O)C2)=O)CC2CCC1CC2 C(CCC(C(=O)NCCc1ccccc1)N1CCC(C)C1CO)OCC C=CC1OCCC1C(N1CCCC1CCC(=O)NCCC1(C)CCCC1)=O C1(NC(=O)Nc2c(OCC)ccs2)CCCCCC1C(c1ccccc1)O CC1CN(Cc2ncc(Cl)nc2Cl)CCN1C(C1CCC(=O)N1C)=O c1(C(=O)NCCC(Cn2cc(C(CC)OC)nn2)F)ccc(F)c(OC)c1 C1(CC(C)NC(c2ccn(C3CCCC3)n2)=O)CCN(C(=O)CNC=O)CC1 c1(CC(N2C(C(C)(C)CNC(C34CC(C3)C4)=O)CCC2)=O)cnc2n1CCOC2 C=CCCC(C)(C)CNC(C(CC)CC=C)C1CCCCC1 N1(CC(=O)NCC(O)CNC(c2cnc(O)nc2O)=O)Cc2ccccc2C1 N1(C(C2N(C(C(OC)OC)=O)C3C(O)CC2C3)=O)CCc2ccncc2C1 c1(C(=O)NCC(C2CCCC2)NC(C(n2cnc(C#N)n2)C)=O)cnn(C)c1Cl CC(C)CC(C)(CNC(=O)CCOCC1CCC1)NC(=O)CSc1nncs1 Cc1nc(C(CO)NC(=O)CC2CC3CC3C2)no1 C(=O)(CC1=NN(C)C(=O)C1)NCCC1(O)CCCN(C(C(C)SC(C)C)=O)C1 CC1CN(C(c2ccnc3ccnn23)=O)CCCN1C(C1CC=CCC1)=O N1(Cc2cnc(C)[nH]2)CC(NC(c2cc(Cl)c(Cl)c(Cl)c2)=O)CC(F)(F)C1 C1(NC(c2n(CC=C)nnn2)(C)CCBr)CS(=O)(=O)C12CCOCC2 C(=O)(C(CC(C)C)C(C)C)NCC#CCNC(c1c(C)nc(N)cn1)=O N1(CC(=O)NC(C2CCCN2C(c2cc(Cl)ns2)=O)C)CCC(C)(O)C1 C(C)(CC(=O)N1CC(F)(CNC(C2(C)CC2(F)F)=O)C1)(C(F)F)N(C)C Brc1ccc(CN2CCOCC2)c(N2CCOC(c3cccs3)C2)c1 N1(C(COCCCC)=O)CCCC(OC)C1C C1(NC(CCN(C)CC)=O)CCC2(CC1)CC(NC(=O)Cn1ccc(C)n1)C2 c1(C(=O)Nc2cccc(C(C)O)c2)ccc2nc(F)ccc2c1O c1(C(=O)NC2CCN(C(=O)CSCC3CCCCO3)C2)ccc2nncn2c1 c1(C)cc(C)c(Br)cc1F.C1(OC)CCC(C(N2CC3CC3(CN)C2)=O)CC1 N1(N2CCCCCCCC2)CC2CCN(C=O)CCC2C1.c1(CC=O)cnccn1 CCC(CC(=O)NC(C)C(C)(C)CO)N(C(=O)C=CC1(C)COC1)C Cc1ccc2[nH]c(CN3CCC=C(C(=O)Nc4ccc(NC)cn4)C3)cc2c1 CCCC(O)CC(=O)NC1CN(C(=O)Cc2ccc(C3CC3)cc2)CC1CO c1(C(=O)NC2CN(C(COC)=O)CC(C)(C)C2)cc2c(Br)c(F)ccc2[nH]1 C(=O)(CC(C(F)(F)F)P(C)(C)=O)NCC(CCNC(C(C)(C)CC#N)=O)O Cn1ncc2c(C(N3CC(F)(F)CC3C(N3CCC(C)(O)C3)=O)=O)cc(Br)cc12 c1(OC)cc(OC)cc(C(=O)NC2COCC2NC(C2CC2(F)F)=O)c1 C(N=c1[nH]c(=NC(C)c2ccc(Cl)cc2)[nH]c2c1COC2)C1CC(=C)C1 C(C1CC1)(C1CC1)=CC(=O)NCC1(CNC(=O)CCNC(C2CCCO2)=O)CC1 c1(C(=O)NC(CN(C(c2cn[nH]c2)=O)CC)C)ccc(N)cc1[N+](=O)[O-] C1(NC(c2c(C)scn2)=O)CN(C(=O)CC=CC(C)(C)C)CCC1CO N1(C(C2CC3C=CC2C3)C(=O)NCCCC)CCCN(C=O)CC1 N1(C(c2nc(C)oc2)=O)CCCC2(CCCN2C(c2cc(Br)ccc2F)=O)CC1 C1(NC(=O)CN2CCS(=O)CC2)CN(C(=O)Cc2cc(F)cc(F)c2)CCC1F N1(C(c2c(CCNC(=O)CCC3CCC3)n[nH]c2)=O)CCOC(C(F)F)C1 Cc1c(C(=O)NC(C)C(C)NC(c2cncc(F)c2)=O)cccc1C#N C(=O)(CC(C)C(F)F)N1CC(OC)C(C(=O)Nn2cc(-c3cccc(C)c3O)nn2)C1 C(CCC(=O)N(CCN(C)C(c1occc1C(C)C)=O)C(C)C)OCCC C(CCCC(=O)N(C)CC1CCCN(C(=O)CCSc2ccccn2)C1)OC N1(C(C2=NOC(C)C2)=O)CCN(C(=O)CC2(C)CC2(F)Cl)CC(O)C1 c1(C(=O)NC2CN(C(C(C)(C)Cc3cnn[nH]3)=O)C2)nccc2[nH]ccc12 C(C(CNC(=O)C(Cc1ccco1)NC(=O)CSc1ccccn1)C(C)C)OC c1(OC)ccc(C(=O)C(=O)NCC2CCC(C)CN2C(c2cccs2)=O)cc1Cl c1(C(=O)NC2CC3(CN(C(CC(COC)COC)=O)C3)C2)ccn2nncc2c1 c1(NC(C2C(NC(C(N3CCOC3=O)C)=O)COC2)=O)cncnc1C C1(CNC(c2ccc(CC)s2)=O)CCN(C(=O)CCC(C)C)CC1O N1(C(c2nc(CC)oc2)=O)CCC(O)(C(C)CNC(=O)CCCC2CCCC2)C1 c1(OC)c(O)cc(C(N2CCCC2C(=O)Nc2cc(Br)c(C)c(Br)c2)=O)cc1O C12(C(N3CCC(O)(CN(C(C(CCN(C)C)O)=O)C)C3)=O)CCC(O)(CC1)CC2 C(=O)(C(C)C(O)C(C)C)N1CCC(=C)CC1C(=O)NC1CCSC1 C(=O)(C1CCCc2sccc21)NCC(C)N(C(c1c(C)n2c(nc1)ncn2)=O)C N1(C(CC2(C=C)CC2)=O)CCC(O)(CNC(c2cnc(C(C)(C)C)[nH]2)=O)C1 C(=O)(C#CC(C)(C)C)NCC(C)(C)NC(=O)CCCn1c(C)ncc1 C1(C(=O)NCCn2ncc(C)c2)CN(C(=O)CC23CCCC2C3)C(C)(C)C1 c1(OC)cc(OC)c(Cl)c(C(N2CC3(NC(=O)C(C)N4CC(C)C4)CC2C3)=O)c1 CC1(C#N)CCN(C(C2CC3C=CC2N(C(c2c[nH]nc2C2CC2)=O)C3)=O)CC1 CC1C2CCC(C2)C1C(N1CC2CC2C1C(=O)NC1(C)CC2(CC2)C1)=O c1(C(N2C(C(C)NC(=O)Cc3cc[nH]n3)CCC2)=O)cc(S(=O)(=O)N(C)C)cn1C C=CC(C)C(=O)NCC(C)CNC(=O)C(c1cncn1C)O C(=O)(C(CO)C(F)(F)F)N(C1CC(C(=O)NC(C2CCCO2)CC)C1)C CCCCC(C)CCC(=O)NC(C)CN(C)C(c1ncc(OC)nc1OC)=O Nc1c(C(=O)OCC(=O)NCC(C2CCOC2)O)ccc(Cl)c1Cl C(CC(C)C)(C(=O)NC(Cn1cncn1)C(=O)N1CCC(CC2CC2)C1)OC CC1CCN(c2nccnc2F)CC1NC(c1cnn(C)n1)=O CN1C(=O)CC(NC(c2nc(NC(=O)Nc3ccccc3)cn2C)=O)C1=O C1(C)(C(=O)NC(C(=O)OCCC)C)CC(O)CN1C(=O)CCc1cc(C)on1 c1(CC(=O)N(c2ccncc2)C2CC2)csc2nccn12.O=C1COCCN1 N#CC1CCCC(C(=O)NCC23CC(NC(C4CCC(=O)N4C4CC4)=O)(CO2)C3)C1 C1(C(N(C)CC2N(C(C3(C)CC(=C)C3)=O)CCC2)=O)CSCC(=O)N1 C1(NC(c2c(OC)nsc2)=O)(CO)CCCN(C(c2n[nH]cc2C)=O)C1 N1(C(C2(C)CCCO2)=O)CCC(NC(C2CC(c3ccccc3)C2)=O)CC(O)C1 C(=O)(CCCCCCN=[N+]=[N-])N(CCCCCCNC(=O)CC1CCC1(C)C)C N1(C(C(CC)CCOC)=O)C2CCCC1CN(C(c1cn3ccccc3n1)=O)C2 c1(N2C(COC)CCC2)nn2cc(C)nc2s1.c12ccc(cc1)C(C)(C)C(=O)NC2 N1(C(c2c(C)oc(C(C)C)c2)=O)CC(N(C)C(C2CCOC2)=O)C(C)(C)C1 C1(CNC(c2ccncc2O)=O)CCCN(C(C2(C3CC3)CC=CC2)=O)CC1 N1(C(c2c(C)cc[nH]2)=O)CC2(CCN(C(C3CC3c3ccccn3)=O)CC2)C1 N1(C(c2ccsn2)=O)CC2CCC1C(CNC(C13CCC(CO1)C3)=O)C2 N1(C(C(C2CN(C(c3cncc(F)c3)=O)C2)OC)=O)CCN(C)C(CO)C1 C1(NC(CC2(OC)CCCC2)=O)CC1C1CCCN(c2nnc(C(N)=O)s2)C1 Cc1cc(Cl)ccc1OCC(=O)Nc1ccc(SCCCCNC(=O)CO)nc1 C1(NC(c2cnnc(Cl)c2)=O)CCCCC1NC(c1occc1C1CC1)=O C1(NC(C=CC(C)C)=O)CN(C(c2cnc(Br)s2)=O)CC1F C1(C(=O)NC(CC)CNC(c2nnsc2C)=O)CCCCC1O N1(C(C=C(C)c2cnn(C)c2)=O)CCC2(CCC2)C(CNC(=O)C(F)=C(C)C)C1 c1(C(C)C)ccccc1NC(C1(C)CN(Cc2cc(Br)c[nH]2)C1)=O C1(CCO)CCCN(c2nnc(CO)n2CCO)C1.c1(OCCO)ccccc1Br C1(C(=O)NC(C)(C)CCNC(C2CC2(C)C)=O)CCS(=O)(=O)C12CCC2 N12CC=CC1(C)C(=O)NCc1cnoc1C2=O.C(CN(C)C(=O)C1CC1)OCC c1(C(N2CCC3CC23C(=O)NOCCCCC2CC2)=O)c[nH]c2cccnc12 c1(C(=O)NC2C(CNC(C3N(CC)CC3)=O)CCC2)ccc(N)c(F)n1 N1(C(C(C2CC2)OC)=O)CCCC(C2(NC(C3Cc4ccccc4O3)=O)CC2)C1 C1(C(=O)NCC2CN(C(c3cccc(F)c3)=O)C2)CC2(CCOCC2)CO1 c1(C(=O)NCC2N(C(C3C(OC)C3)=O)CCCC2)cc(Br)cc(O)c1 Cc1ncnc(O)c1CCC(N1CC(NC(=O)CCCF)CC(O)C1)=O C1(F)(C(=O)NCCN(C)C(c2cc(OC(F)F)n(C)n2)=O)C2CCCCC12 O(C1CCc2cc(Br)cnc21)C(C(C)Cc1cccc(F)c1)=O C(=O)(C(C(C)O)N(C)C)NC(C(CO)NC(c1cc(C(C)(F)F)n[nH]1)=O)C N1(C(=O)CC2(c3ccccc3)COC2)CC(C(N2CCCC2)=O)C2(CC2)C1 c1(C(C(=O)N(C2C3CN(C(=O)Nc4ccccc4F)CC23)C)O)cccc(Cl)c1 C1(C(=O)NCC(c2ccncc2)O)(CC)CCCN(C(=O)C=Cc2cc[nH]n2)C1 c1(C(=O)NCC2CC(NC(C(CC=C)N(C)C)=O)C2)ccc(N)cc1Br C1(CC)CCC(C(N2CCCC2(C(=O)NCC(F)(F)CO)C(C)C)=O)CC1 N1(C(CN2C(=O)CSC2)=O)CCN(C(c2cccc3cc[nH]c23)=O)C2CCC12 c1(CC)[nH]nc(C(=O)NCC2C=CCN2C(C2CC(O)(CCC(C)(C)C)C2)=O)c1Cl N1(C(C2C(CC)C2)=O)CCC(CNC(=O)C2=CC(C)(C)C2)C(CC)C1 c1(CS(=O)(=O)NCC2(NC(c3c(OC)c[nH]n3)=O)CC2)ccc(Br)cc1 C1(C(=O)NC2(c3cn(C)nc3)CC2)CC(O)CN1C(=O)C(C)(F)c1ccon1 O=C(O)CCN=C(NCC1CCCCNC1=O)N1CCCCC1 Cn1nncc1Nc1cnc(C(F)(F)F)s1 C1(CC)C(NC(c2ccccc2Br)=O)CCN1C(=O)C(C)NC(C)=O Cc1ccc(C(=O)NNC(=O)CN2CC(N(C)C)C(C)C2)c(C)c1 N1(C(N2CC3CCC2CN3)=O)CCCC1C1CCCN1C(c1cccs1)=O N(C(=NCCC1CC1(Cl)Cl)NCC1CCCCCCC1)C(C)C c1(C(=O)NC2CC(C)C2)cnc2nc(NS(=O)(=O)C3CCCCC3)ccc2c1 C1(CCNC(C2(SCC)CC2)=O)CCN(C(=O)Cn2ccc(C)c2)CC1 c1(CNC(C(C)OCC(C)C)=O)nocc1C(=O)N(C)CC1(O)CN(C)C1 c1(OC)cccc(CN2CCC(C(=O)NCCc3ccccc3C)CC2)c1F C=C1COCCN(C(c2cnc(C(F)F)s2)C(=O)NC2(C)CC2)C1 N1(C(C(c2ccnn2C)C)=O)CC2(C(N3CC4(C)CC3CCO4)=O)CCC1CC2 c1(CCC(=O)NCCC(C)NC(=O)C(C)(C)CO)ccc(Cl)cc1Br C#Cc1ccc(C)c(NC(C2C(C)CCN2C(=O)C(C)=C2CC2)=O)c1 c1(C(N2CCC(C(C)NC(c3c(C)c[nH]c3)=O)CC2)=O)ccc2c(C)nnn2c1 C(=O)(C#CC1CCCCO1)NCCN(C(=O)CCC1CC1(Cl)Cl)CCOC CC1(C)C2CCC1(C(=O)CO)CC(NC(c1c(Br)cc(Cl)cc1F)=O)C2 CC1C(=O)N(CC(=O)NCC2CCC(C)C2)C(=O)C1C C(=O)(C(C)S(=O)(=O)C(C)C)N(CCNC(=O)Cc1ccc(Cl)cc1)CC N1(C(COC)=O)CCC(O)(C2CCN(C(C3CC4C(C3)C4(F)F)=O)CC2)C1 N1(C(C(CC)OC)=O)CCC(C2(NC(=O)CN(C(=O)COCCSC)C)CC2)C1 C1(Cn2c(C3(SCC)CCCC(CC(=O)NC)C3)nnn2)CC2CCC1(CO)C2 CC1CC(NC(=O)C(C)N(C)C)CCN1C(=O)C1CC1 N1(C(C=CC(N)=O)=O)CCC(NC(c2cnn(-c3ccncc3)c2)=O)C(O)C1 N1(CCC)C(=O)CCC1C(=O)N(CCCNC(=O)CCCC#N)CC N1(C(CCC=C)=O)CCOCC(CNC(c2nn(C)nc2Br)=O)C1 C(CCO)(C(F)F)N(C(C(N(C(CCC)=O)C)C1CC1)=O)C C1(C(=O)OC)Cc2c[nH]nc2CN1c1cc(Br)nc(C)n1 Cc1cc(C(=O)NC2C=CC(C(=O)NCCC3CC=CC3)C2)[nH]c1C c1(OC)ccc2c(N3CCNCC3C(=O)Nc3cc(O)ncn3)ncnc2c1 Cc1c(C=CC(N2CC(NC(=O)CNC(=O)C3CC3)CC2(C)C)=O)cnn1C N1(C(c2ccc(OC)nc2)=O)CCC(C2CCN(C(=O)C(C)P(C)(C)=O)CC2)C1 c1(OC)ccc(C(=O)NCC(C)(C)NC(=O)CS(=O)(=O)C(C)(C)C)cc1[N+](=O)[O-] N1(C(CCOC(C)C)=O)CCN(C(c2ccccc2C(C)(C)C)=O)CC(O)C1 N(C(=NCC(C)C)N1CCC2(CC(C(F)F)=NO2)C1)Cc1ccc(CC)nc1 c1(CC)ccc(NC(C2CC(NC(=O)CCc3ccsc3)C(O)C2)=O)cc1 c1(CC(=O)NC(C2(O)CN(C(C3CC4(C3)CC(O)C4)=O)C2)C)cccc(Cl)c1Cl c1(CC=CC2C(CC(N3CCC(CC)C3)=O)C2)cccc(OC)c1 N=c1nnn(CC(=O)NCC(CO)NC(c2nn[nH]c2Cl)=O)[nH]1 c1(OC)nn(C)cc1C(N1CCCC1(C(=O)NC1(C(C)C)CC1)C(C)C)=O O=C(C#CC1CCCC1)NCC1COCCN(C(=O)C(c2cccc(Cl)c2)O)C1 CCCC(C)CC(=O)N1CC2(CNC(C3CN(C)C3)=O)CCC1C2 C(=O)(CCC(O)C(C)(C)C)NCC1(NC(C2CCC(CCCCC)O2)=O)CC1 c1(CC)cccc(NC(C2(NC(=O)CC3CCCC3C)CC2)=O)c1 c1(C(N2CC(CC)N(C(=O)C3=CCSC3)CC2)=O)cnc2n1CCOC2 CCC(C)C(C)(O)CNC(=O)C(C(C)O)NC(=O)CCC(F)(F)F CN1C(=O)CCc2ccc(C(=O)N(CCn3cc(C4CCC4)nn3)C3CC3)cc21 c1(OCCC(C)C)cccnc1C(=O)NC(C)CNC(=O)C=Cc1cscn1 O=C1NCC(C(=O)NCC#CCNC(=O)CCCn2cccn2)N1 C#Cc1ccc(CC(N2CCC(NC(=O)C=C3CCN(C)CC3)C(O)C2)=O)cc1 c1(CN2C3(CN(c4nc(SC)nc(C)c4)C3)CC2)c(Br)cccc1[N+](=O)[O-] C(C(=O)N1CC(O)CCO1)NC(N(C)C(C)=O)=NCCN(S(C)(=O)=O)C(C)C C#Cc1cccc(C(N2CC(CCNC(C3CCC4(CCC4)CC3)=O)C2)=O)c1Cl c1(OC)c(C(N2CC(OC)C(NC(=O)Cn3ncn(C)c3=O)C2)=O)cccc1N C(=O)(CC(CC1CC1)N(C(=O)CC(C)(C)C)CCO)N(CC(C)C)CCO O=C(C1=C(Cl)CCC1)NC1CC(NC(c2cccc(-n3cncn3)c2)=O)CC1O c1(CC(=O)NCC2CCCCC2NC(=O)CCc2cccs2)ccc(F)cc1 N12CC(CC(C)C1)C2=O.c1(NC(C)=O)ccc(C(=O)NCCN(C)C)cc1 C(C1=NOC2CN(C(c3scc(C)c3C)=O)CC12)NC(COCCOC)=O c1(C(=O)NCC2(CCNC(c3ccon3)=O)CC2)cccc([N+](=O)[O-])c1O c1(OC)noc(C)c1C(=O)NC(C)CCCCNC(c1cc(SC)c(C)o1)=O C(CC(C(=O)N1CCC(COC(C)=O)C1)NC(c1cc(Cl)no1)=O)=CC c1(OC)cc(C(=O)NC(C2CN(C(=O)CC(=O)NC3CC3)C2)C)cc(Cl)n1 C1(OCC)COCCC1CC(=O)NCC(C)(C)NC(=O)Cc1cncc(CC)c1 C(C(C)CC(=O)N(C1CCC(F)(F)C1)C)NCC1(CCNC(C)=O)CC1 C1(C(=O)NC2CN(C(c3cc(CCC)n(C)n3)=O)CC2C)CN2CCN1CC2 C1(NC(C(C)SCCCC)=O)CC(C)CN(C(c2cncc3c2CC3)=O)C1 CC1=NS(=O)(=O)NC=C1C(=O)N1CCCC(NC(=O)CCc2ccc(Cl)s2)CC1 C(=O)(NNC(=O)C(=O)c1cccc(Br)c1)C1CC(C)NC1=O C1(NC(=O)CC2CCCC2)CN(C(C2CC2c2ccccc2)=O)C2CCCC12 c1(CCC)sc(C(=O)NC(C)(CNC(=O)C(C)c2ccsc2)CO)cc1CC C12(CC)CC(NC(c3cc(CNC(=O)C(C)n4cccn4)on3)=O)(CO1)C2 C1(CC)CCN(C(C2CC(=O)N(C)C2)=O)C(C(=O)N(C)Cc2ccc(C)cn2)C1 C(=O)(CCCC(=O)NCC(=O)NC(C)=O)N(C1C(CN(CC)CC)CCCC1)C O=C(C#Cc1cccc(F)c1)N1CCc2nccn2CC1 C1(C(C)NC(C2(CCC)CC2)=O)CN(C(c2cncnc2C2CC2)=O)CCO1 C1(OC)CC(=O)NOCC(C2CC2)O1.C(C)(C)(C)OC c1(C(=O)OC)ccc(F)c(CN2CCC(F)(CO)C2)c1.C1(C=O)(CO)CCNCC1 O=C(N=c1nc(O)[nH]c(O)n1)C1CCN1c1ncnc2ccc(Br)cc12 CN(NC(=O)Nc1ccc(Cl)c(OC(F)(F)F)c1)C(=O)OC(C)(C)C C12(NC(c3c(Cl)ccc(OC)c3F)=O)CCCC1N(c1nnco1)CCC2 c1(C(=O)NCC(CNC(c2ccc(OCC)nc2)=O)C)nccn2ccnc12 N1(C(c2c(CC)nc[nH]2)=O)CCC2CN(C(c3ncc(C)cc3OC)=O)CCC12 N1(C(c2c(C)onc2Br)=O)CCN(C(C2CC2F)=O)C(CO)C1 C(=O)(C(C)(C)CN1CCN(C)CC1)NCCOCCNC(CC(CC)OC)=O C#Cc1ccc(Cl)c(C(=O)NCc2cn(CCNC(c3cncn3C)=O)nn2)c1 C1(NC(c2n(CC)ncc2)=O)CC=CCC1C(=O)NCC(C)CC(C)C CC1(CNC(=O)C=C2CCCC2)CCC(NC(=O)CSCc2ccccn2)C1 Cc1nn(C)cc1C1CCC(C(C)C)N1C(=O)Cn1nnnc1C N1(C(CCN(CCC)C)=O)CCSCC1CCNC(c1cc(C)n(C)n1)=O C1(CCC(=O)NCCN(C(=O)C2=CCOC2)Cc2ccccc2)CCCC(O)C1 N1(C(CCc2onc(C)n2)=O)CCCN(C(=O)CN2CCC(C)C2)C(C)C1 c1(C(=O)NCC(CNC(C(C2CCCOC2)OC)=O)(C)F)cc(Cl)n[nH]c1=N Cc1cc(C(=O)N(C)Cc2ccc(CNC(C3(C#N)CCOC3)=O)cc2)ccn1 CC(C)(C)C(O)C(=O)NC(C)(CNC(=O)CCc1cc(Cl)cc(Cl)c1)CO C1(CNC(CCOC)COC)(CO)COCC2CCCCN12 c1(OC)cccc2c(N3CCC4(CNC(=O)OC(C)(C)C)CC4C3)ncnc12 C1(CN(C(c2cocc2C)C(=O)NCc2ccccc2)CCC)CCCCC1C C#CCC(CC(F)F)NC(=O)C1=NOC(CNC(c2ccc(C(N)=O)[nH]2)=O)C1 C12(NC(CC(CC=C)NC(=O)Cc3cc(C)cs3)=O)CC3CC(CC1C3)C2 c1(NC(C2CCCCC2CO)=O)ccc(CNC(c2ncn(C)c2)=O)cc1F C(=O)(C(F)(F)C(F)(F)C(F)F)N1CCC2C(NC(CS(CC)(=O)=O)=O)C2C1 C1(C(COCC2(C#C)CCC2)=O)CC2C=CC1C2 C(CN=c1[nH]c(C2CC2)nc(=N)[nH]1)N(C(C1C(OCC)C1)=O)C C(=O)(C1=CCC(C)(C)CC1)N1CC(C)(NC(c2c(Br)cn(C)n2)=O)C1 C1(C(C)C)C(NC(C2(CF)CC2)=O)CCN1C(c1csc(-c2ccco2)n1)=O C(C1CCOCC1)=CC(=O)NCC(C(C)C)NC(=O)Cc1ccn(C)n1 c1(C2C(C(N(CCN(C(CC(F)(F)F)=O)CC)CC)=O)C2)cccc(Cl)c1Cl C1(c2nnc(C(C)C)o2)CCCCN1C(C1CC(C)(c2ccccc2)C1)=O C(=O)(C1=CCC2(COC2)OC1)NC1C(NC(c2cc(OC)c(C)cc2)=O)C1 c1(C(N2CC3(C(C(=O)NC(c4cnccn4)C)C3)C2)=O)ncc(Cl)cc1Cl C1(N)CC(O)CN1C(=O)CCCCN(C)CC1CN(C(=O)C2CC2)C1 c1(COC(C(CC(F)C(N)=O)OC)=O)nc2ccccc2n1C c1(C(=O)NCC2CCN2C(=O)CCOC2CC2)c(C(F)(F)F)nc2n1CCCC2 N1(C(c2ccc(OCCCl)cc2)C(=O)NC(CC)(C)C)CC(O)CC(O)C1 c1(OC)cccc(O)c1C(N1CCCC(C)(C(N2CCC(CO)C2)=O)C1)=O c1(NC(c2cncc(CNC(C(CC=CCC)C)=O)c2)=O)cn(CC)nc1C#N C(=O)(CCCCCF)OCC(c1ccc(C#N)cc1)C C1(C(N2CC(c3c(C)nn[nH]3)C2)=O)CC1C1CN(C(C2CC2(Cl)Cl)=O)C1 CC(CS(C)(=O)=O)C(=O)NC1CCC1NC(c1cc(O)nc(N(C)C)n1)=O C1(OC)CC(CNC(c2ccsc2)=O)N(C(C2CC(C)OC2C)=O)C1 c1(C(=O)NC2(CO)CCN(C(=O)CCc3cncs3)C2)cc2ccccc2[nH]1 c1(C(=O)NC(CC)CN(C)C(C2(N(C)C)CC2)=O)cccc(C(C)(F)F)n1 C1(C2CCN(C(C3(CF)COC3)=O)C2)(NC(C(CC(C)C)OC)=O)CC1 n1(CC(=C)C)nnnc1C(c1ccc(C)o1)NCc1cccs1 C1(C(=O)OC)CCCN(CC#CCCOC(C)C)C1 C1(NC(CC(CC)O)=O)CCN(C(C2(N3CCCC3=O)CC2)=O)CC1C C1(N(C(=O)CCc2nc(O)n[nH]2)C)CN(C(=O)Cn2ncn(C)c2=O)CC1(C)C C(N=c1[nH]c2ccccc2o1)C1C(NC(CSC)=O)CCCC1 C(=O)(C1=NN2CCCN=C2N1)NCCC(Cc1ccccc1)NC(C(C)SC)=O C1(NC(Cc2cn(CC)nc2)=O)CC(F)CN(C(=O)CN2CCOCC2=O)C1 C1(C(=O)NCC2(NC(c3[nH]c(=NC)sc3)=O)CCOCC2)COC2(CCC2)CO1 N1(C(=O)CN2CC=CC2)CCCCC2(CCN(C(c3ccc(Br)o3)=O)C2)C1 c1(NC(c2ccc(NC(C)=O)cc2)=O)cc(C2=CCC(O)CC2)ccn1 c1(CN2CCC(n3c(C)ccc3C)CC2)nnn2c1CCC2 c1(NC(C2N(C(c3nc(C(C)C)oc3)=O)CC=C2)=O)ncc(Cl)cc1O C1(OC)CC(CNC(=O)COCc2ncc(C)o2)N(C(=O)CC(C)F)C1 N1(C(C2CCCC2C(C)C)=O)Cc2ccccc2C1.CC(C)C1C(=O)N1C(=O)C N1(C(CC2(NC(C)=O)CCC2)=O)CCCC(CN(C(=O)C(C)(C)OC)C)C1 C(=O)(CC(F)(F)F)NCCCC(C)NC(C1CCC(c2ccccc2)O1)=O O=C(C1=CCSC1)NCCC1CC(NC(c2ccnc(-c3ncc[nH]3)c2)=O)C1 c1(C(N2CC3(CN(C(C4C5C(=O)C6C(C5)C64)=O)C3)C2)=O)cccc2[nH]ncc12 N1(C(c2n(C(C)C)ncc2)=O)CCC(CNC(=O)CC2CCCCC2)CC1C N1(CCC(N2CC(CC(C)NC(=O)CCF)C2)=O)Cc2ccccc2C1=O c1(C(=O)NC(CNC(c2onc(CC)c2C)=O)C)ccc2c(c1)C(=O)OC2 c1(C(=O)NCCCC(CO)NC(c2c(CC)nns2)=O)ccc(S(C)(=O)=O)s1 C(c1ccc(Cl)cc1F)=CC(N1CC(CC(=O)NCC(O)C(F)(F)F)OCC1)=O CC(C)C(C(=O)NCCC(C)NC(c1cnccn1)=O)c1cnn(C)c1 N1(C(C(C)C2CCCO2)=O)CCN(C(C2CC(O)C2)=O)C(C)C1 C#Cc1ccc(C(=O)NC2CC2NC(=O)C(C)CN2CCOCC2)cc1Cl C1(CNC(c2c(CC)nco2)=O)CCN(C(=O)CSc2cccc(Cl)c2)CC1C c1(NC(C2CCN(Cc3ccc(OC)cc3Br)C2)=O)ccc2c(c1)c(Br)nn2C C(=O)(C(O)CC(C)(C)C)NC(C1CCCC1)CNC(C(C)(C)OC(C)C)=O c12ccc([N+](=O)[O-])c(c1)NCC2C.C1(CNC(=O)NCCOC)(CO)CC1(F)F N1(C(c2cnc(Cl)cc2F)=O)CC2CCN(C(=O)COc3ccncc3)C2C1 c1(CC)c(C(=O)N(CCCCN(C)C(C2CCCN(C)C2)=O)C)ccn1C CC1CCCC1(C)C(=O)NCCCCNC(C1CC(C(=O)OC(C)(C)C)C1)=O C(N=c1[nH]cc(Cl)c(C)c1C#N)C1CN(C(C(C(CC)C)C)=O)CC1C(F)(F)F CN(Cc1ccc(Cl)s1)N1CC2(CC(C(=O)NS(C)(=O)=O)CO2)C1 N1(C(c2c(CC)ocn2)=O)CCOC2(CCN(C(C3CCCC34CC4)=O)CC2)C1 c1(C(=O)NC(CNC(C)=O)C(C)(C)C)c(NC(=O)N(C)C)cccc1F C(CN=c1ncc(C(C)(C)O)c[nH]1)OCC(=O)N(C)CC1CC(C)N(C)C1 C1(C(=O)NC(C(=O)NCCN2CC(OC)C2)C2C(C)C2)CCC(=O)O1 C(=O)(CS(=O)(=O)CC(F)(F)F)NCC(CNC(c1c(CC)ccc(OC)c1)=O)O CC#CCC(C(=O)N(CC)CC1CCOC1)NC(=O)C(C)C(C)(C)C C12(NC(CCCn3ncc(C)c3)=O)CCCCC1N(C(=O)CC1(C=C)CCC1)CC2 N1(C(c2c(SC)ccs2)=O)CCCC(NC(=O)Cc2c(C)noc2C)C(F)C1 c1(C(N2CC(O)(C(C)NC(c3cn(C)nn3)=O)C2)=O)ccc(F)cc1 c1(C(N(CC(CNC(c2c(C)cns2)=O)C)C)=O)cccc(NC(=O)C2CC2)c1 C(C)(C(=O)NC1(C(=O)NC2CCNC(=O)C2)CC1)(C(C)C)OC N1(C(c2c(CCC)n(CC)nn2)=O)CCN(C(=O)CC2CC2)C(CCO)C1 n1(CC)nnc(C(=O)NCC2(O)CC(CNC(c3cocn3)=O)C2)c1C C12(C(=O)NC(CCOC)C(=O)NC(C)Cc3nn[nH]n3)CCCC1OCC2 Cc1[nH]c(-c2ccccc2)c(C)c1C(=O)NNC(=O)c1cnsc1.C1CCO1 N1(C(c2cccc(OCc3ccc(F)cc3)n2)=O)CCCC2(CCNC2)CC1 C1(OC)CC(CO)N(C(=O)C(C)(C2CC2)N(C(=O)Cn2cnnc2O)C)C1 N(C(=NCCCCl)NCC1CCCO1)Cc1c(C(F)(F)F)csc1 C=CCC(C)C(=O)N1CCCC1C1CCN(C(=O)C(=Cc2cccs2)C(=O)NC)CC1 n1(CC)nc(C(=O)NC(Cc2ccccc2CC)CC(=O)NC2(C)CC2)cc1C N1(C(C(C)NC(N)=O)=O)CC(NC(C2COC(C)C2)=O)CC2(CCC2)C1 Cc1ncccc1C=CC(N1CCCC1C(=O)NCCc1cccc(O)c1)=O c1(C(=O)NC(C)CC2CN(C(=O)CCn3cncn3)C2)nn(C)c2c1C(O)CCC2 N1(C(C(=O)NC2(c3ccn(C)n3)CCC2)=O)CC2CC(C(F)F)CC2C1 c1(C(N(CCCNC(c2nc(C#C)sc2)=O)CC)=O)cc(C)ccc1S(N)(=O)=O c1(C(N2C(C(=O)Nc3c(C)noc3C)CCCC2)=O)cc(Cl)cnc1Br C(C(COC)CC(=O)NCC1CN(C(C2(C(C)(F)F)CC2)=O)CCCO1)OC c1(C(=O)NC2CCN(C(C(C)NC(=O)NC)=O)CC2C)ccc2ocnc2c1 c1(OC)ccccc1C1CCN(C(=O)C(N)Cc2nonc2C)CC1 c1(C(=O)NCC2C(CNC(C(C)(C)OCC)=O)C2(F)F)ccc(F)c(C)c1 C(=O)(C(CN(C)C)CC(C)C)N1CCN(CCNC(c2cnn(CC)n2)=O)CC1 C(CCC(=O)N(C1(CC(C)C)CC1)C)OC(C)C.c1c(=O)n1 CCC(CNC1CCC(C)(CN)C1)(CC)SC CC(CC(C)(C)C)C(=O)N(C(=O)CC(C)(C)Cc1ccccc1)C(C1CC1)C1CC1 C(=O)(CC(CC)CC)NC1(C)CC(C(=O)NCCC=CC=C)C1 C1(CNC(COCC(C)C)=O)(CNC(=O)Cc2ccco2)CC1(F)F C(C1CCCc2ccccc21)N(C(C(=O)NCCc1ccc(C)c(F)c1)=O)C C(=O)(C(CNC(=O)CC(F)(F)F)CC(C)C)N(CCCO)CC CC1CCN2CCN12.C1(CC=O)C=NN(C)C1=O.c1(NC=O)c[nH]nc1C(F)(F)F N1(C(C2(c3cccs3)C(C)C2)=O)CCCC(CN(c2cn[nH]c2)C)CC1.C1C(=O)N1 Cc1nc(S)sc1CC(N1CCC(C(C)NC(=O)C(c2ccc(Cl)s2)=O)CC1)=O c1(OC)cc(C)[nH]c(=NCC2CCCC2NC(c2cc(C)oc2C)=O)n1 c1(CC(=O)NC2C(C)CCN(C(C3COC(C)C3)=O)C2)cc2ccccc2o1 C(=O)(C1CCCc2ncnn21)N1C(CNC(=O)CSc2nncs2)C(O)C(O)C1 C(CN=c1[nH]c(=NCc2ccsc2)[nH]c2c1CS(=O)(=O)C2)c1nc(O)n(C)c(=O)c1 C1(CNc2c(C(=O)OC)scn2)CCCN(C(C2(Cl)CC2(C)C)=O)C1 C1(NC(C2OCCC(NC(c3c(C)[nH]c(C#N)c3)=O)C2)=O)CCN(C)CC1(C)C C1(C#N)(C(=O)NCC2CC(NC(C(COC)O)=O)C2)CCCCC1 C1(C(N2CC(CCCC)N(C(c3cnc(S)n3C)=O)CC2)=O)CCC2CC1C2(C)C C1(NC(=O)Nc2n(C)nc(C3CCCO3)c2)CC(C2CCCC2)C1 Cc1cccc(C(=O)N(C)CCC2CCCCN2C(=O)CN(C)C(C)C)c1Cl Cc1sc(C(N2CCC(C(F)(F)F)CC2)C(=O)NC2COC2)c(C)c1Br c1(C(=O)NC23CC(NC(c4ncc(OC)nc4)=O)(C2)C3)cnc2cc(C)ccn12 C1(C(N2CCC(O)CC2)=O)(COC)C=CCN1C(=O)C(C)OCC(C)C N1(C(C(C(C)C)NC(=O)CCc2ccccc2)=O)CCCC(C)(CN(C)C)C1 C1(CC)CC(=O)CC(=O)N1.N12CC(C(C)C1)n1cc(nn1)CC1CCC(C1)C2=O c1(C(=O)N(CCC2(CNC(=O)C3=CCOC3)CC2)C2CC2)cc(C(F)F)ccc1Cl C(CC(C(=O)NCCC1CCCN1C(C1CC1F)=O)OC)OC C1(NC(C(C)NC(N)=O)=O)CC2CC(C1)N(C(c1cc(O)ccc1O)=O)C2 c1(C(=O)NC2CCC(F)(CNC(c3cnns3)=O)C2)cc(F)c(F)c(O)c1F C1(NC(Cc2c(C)n(C)nc2)=O)CC2(CCC(CNC(c3ccoc3)=O)OC2)C1 Cc1cccc(=O)n1CCCC(=O)N(O)Cc1cn(Cc2ncoc2CO)nn1 C1(CNC(c2cnc(C)n2C)=O)CN(C)CCN1C(=O)CCc1cccs1 N1(C(C(CC2CCC2)NC(C2CC(SC)C2)=O)=O)C2COCC1C2 CN1CCc2ccc(C(=O)NC(C)(C)Cn3ccc4ccccc34)cc21 CCCC(C(=O)NC(C)CN(C(=O)C(c1ccccc1F)OC)C)NC(C)=O C=CC(C)(CC)C(=O)NCCCN(C(c1cc(Cl)ns1)=O)C1CC1 C=Cc1cncc(C(=O)NCC2CCN(C(c3oc(C)cc3C)=O)CC2C)c1 c1(OC)cc(N(CC(C)CNC(=O)CCc2csc(C)n2)C)nc(OC)n1 c1(C(=O)NC(CCCCNC(CC(C=C)C)=O)C)c[nH]c2c(Br)cccc12 c1(CCOC)n[nH]c2c1CCCC2.n12nnnc1C(C)(OC)COC(=O)C2 c1(C(=O)NCCOC2CCN(C(CCC(C)OCC)=O)C2)cc(F)cc(F)c1N c1(C2(C(=O)NCC(CNC(c3cc(Cl)cs3)=O)OC)CCC2)cccc(Cl)c1F n1(CC)ncc2c(N(CC(C)SC)C)nc(N(CC(C(C)C)OC)C)nc12 c1(OC)ccc(F)cc1C(=O)NC1CCC(CNC(=O)CC2CCC(=O)N2)CC1 CCC(C)(CO)CN=c1[nH]c(=NCCc2ccnn2C)[nH]c2cc[nH]c12 c1(C(=O)NC(C(=O)N2CC(C(CC)CC)C2)CC2CCC2)cnc(C)nc1 c1(C(N2CCC3(C(C(N(CC(C)(C)O)CCO)=O)C3)C2)=O)cc2ncccc2[nH]1 C(=O)(C1=NOC(C)(C)C1)N1CCCC(Cn2cc(-c3ccc(C)cn3)nn2)C1 C1(C)(C(N2CC(COC)(NC(=O)CCn3cc(C)cn3)C2)=O)C=CCCC1 CCC(CC)(CO)C(=O)N1CC(CCNC(c2ccnc3c2CCO3)=O)C1 N1(C(c2cc(OC(C)C)[nH]n2)=O)CCC(CC(=O)NC2CC3CCC2C3)CC1 C1(NC(CNC=O)=O)CCCC(C(=O)NCCCOC2CCC2)CC1 c1(C(=O)NC2CN(C(C(C)C#N)=O)C(C)C2)cn2cnnc2cn1 C1(C(N(CC(=O)NCCC2CC(OC)C2)C(C)C)=O)CCCC(=O)N1C C12(NC(CCc3ccc(C)s3)=O)CC1CN(C(c1cc(CO)oc1C)=O)C2 Cc1noc(C(=O)NC23CC(NC(C4CCC(C(F)(F)F)C4)=O)(C2)C3)c1C c1(N2CCC(C)C(NC(c3cccc(OC)n3)=O)C2C)ccc([N+](=O)[O-])c(C)n1 C1(NC(C(C)C2CCCC2)=O)CC12CCN(C(=O)C(O)C(C)(C)C)C2 c1(SCC(N2C(CNC(c3cc(CC)on3)=O)CCC2)=O)nc2ccccc2o1 C1(C(=O)NCCCNC(CCNC(COC)=O)=O)COCCC1c1ccccc1 C(C(C)(C)CN(C)C(c1nocc1C(C)(C)C)=O)NC(C(C1CCC1)OC)=O C1(NC(C(C)(C)c2cscc2Cl)=O)CC2CN(C(=O)C3CC3)CC12 C1(NC(c2c(OC)csc2)=O)CC(CNC(c2csc(S)n2)=O)C1(C)C c1(NC(C2C3(C(=O)NCC(C(CC)CC)O)C4CC2CC34)=O)cccn2ccnc12 CCCCC(C)(F)C(=O)NCC1CN(C(=O)COC(C)C)CCO1 N1(c2n(C)c3c(n2)c(Cl)ccc3)CCc2c(Cl)c(Br)cc(F)c2C1 N1(C(C(OC)OC)=O)CCCC1CCNC(c1nonc1C1CC1)=O C(=O)(C1=NOC2CNCC12)N1CC(C(=O)OC)C(CC(C)(C)C)C1 C1(NC(C=NOC)=O)CCCC(CN(C)C(c2cnc(-c3ccsc3)s2)=O)C1 CCCCC(C(=O)NC(CNC(=O)CC(=O)N(C)C)CC)C(C)C C1(C)(NC(CC2N(C(CC3ON=C(C)C3)=O)CC(O)C2)=O)C(C)(C)C1(C)C c1(C(N2CCC(N3CCCC3)C2)C(=O)N)cccc(C(N)=O)c1.C1(SC)CC1 C1(NC(c2ccc(C)o2)=O)CCCC2CN(C(C34CC(C3)S(=O)(=O)C4)=O)CC12 Cn1cc(C=CC(=O)NC2CCCC(N(C(=O)C=CC(F)F)C3CC3)C2)cn1 N12CC(C3CCCC13)C2=O.Cc1noc(C2CCCN2C(=O)CC2(CO)CC2)n1 C1(NC(=O)Cc2ccc(C(F)F)cc2)CC2CC1CN2C(=O)CCC=CBr Cc1ncc2n1CC(CNC(=O)C(C1CCS(=O)(=O)CC1)(C)C)CC2 CCCC(CC)CCC(=O)N1CCC2(CC1)CC2CNC(=O)CCN(C)C(C)=O c1(C(N(C(CNC(c2cc(C)c(F)nc2)=O)C)C)=O)ccc2c(c1)C=CS2(=O)=O C=Cn1nccc1C(N1CCCC1CC(=O)NCC#CCSC)=O c1(NC(C2CC2NC(C2=CCSC2)c2n(CC)nnn2)=O)sccc1S(C)(=O)=O N1(C(=O)CCC2CCCO2)CCC(C(N2CCC2Cc2ccccn2)=O)(CO)C1 c1(C(=O)Nc2cnn(C(C)C)c2C2CC2)cc2cc(Br)sc2s1 C(=O)(CC(C)CCC)NC1C(CNC(C(CCC)NC(N)=O)=O)CCC1 N1(C(CCCC(C)O)=O)CCC2CCN(C(c3c[nH]nc3C3CC3)=O)CC12 O=C(C1=COCC1)NC1CCCC(NC(=O)Cn2ccc(C3CC3)n2)C1 C(=O)(C1=CCCSC1)NCC(CO)NC(C(C)(C)C1CCCCC1)=O CC1CN(C(=O)CN2CCOCC2)CC1CCNC(=O)Cc1nc(=N)[nH][nH]1 N1(C2CC(NC(C3CC3)=O)C2)CCCC(OC)C1.C1(CC(=O)OCC(C)C)(CSC)CC1 c1(C(N2C(C(=O)NC(C3CSC3)C)CC(F)CC2)=O)cc2ccccn2c1 c1(NC(CCCCOC(CCC)=O)=O)ccccc1S(=O)(=O)N1CCCC1 c1(CC(N2C(CNC(c3c(CC)cno3)=O)CC(OC)C2)=O)ccc(C)nc1Cl C=CC1(CC(=O)N(CCCNC(C2C3CCCCC23)=O)C2CC2)CCCCC1 Nc1cc(F)c(C(N2CC(C3(NC(c4csc(O)n4)=O)CC3)C2)=O)cc1Cl C1(NC(C(C)(C)NC(Cc2c(C)n(C)cn2)=O)=O)CCCCCC1(C)C c1(C(=O)OC)ccccc1C(N1CC(CC)C1)=O.c1(C2C(=O)N2)ccccc1.OC C1(C(=O)NC(C)CNC(=O)Cc2nnc(C)o2)(NC(C)=O)CCC(C)(C)C1 C1(n2cnnn2)(CC(=O)NC2C(NC(CC(=O)N(C)C)=O)C2)CCOCC1 C1(CNC(c2cccc(C(F)F)n2)=O)COCCN1C(c1nncs1)=O C=CC(CCC)CC(=O)NCC1CN(C(c2cnc(S)n2C2CC2)=O)CC1(C)C N1(C(c2cc(C)sn2)=O)CCC(NC(=O)CC2(C)CCCCCC2)CC1C c1(C(=O)NC(C2(O)CN(C(CCSCCC)=O)C2)C)cn(C)nc1Cl Cc1ccc(C(=O)NC(C2CCN(C(=O)CCOC3CCC3)CC2)C)cc1F CC1CC=CCC1C(N1CCOC(CNC(=O)C(C)n2ccnn2)C1)=O CN1CCCc2cc(C(=O)NCC3CCN3C(=O)C(O)CN3CCOCC3)ccc21 N1(C(CCCOCCC)=O)CCOC(CN(C(=O)C(F)(F)F)C)C1.C1(=O)CN1 C1C(C)C(=O)NC2CCN(C2)OC(=O)COCC(=O)N1C.N1(C(C)(C)C)CCCC1 C(=O)(C(C(O)C(F)(F)F)C(C)(C)C)Nc1cncc(CCN(CC)CC)c1 C1(C(=O)NCC2(F)CN(C(CSc3n(C)ccn3)=O)C2)CCCC2CCCN12 C1(N(C(CNS(CCCC)(=O)=O)=O)C)CCC2CN(C(=O)C(=O)C(C)CC)CC12 c1(C(C)C)cccc(C(N2CCCC(CN(C)C(C3CC3F)=O)C2)=O)c1 c1(C(N2C(CC)CN(C(=O)CNC(=O)N)CC2)=O)cc2ccccn2c1.N(C)C CCCC(C(=O)NC(C)(C)CCCNC(=O)COc1cccc(Cl)c1Cl)C(C)C c1(CC)c(C(=O)NC2CCCC(NC(=O)CCn3nc(C)nc3C)C2)nnn1C c1(C(=O)NC(C)CNC(c2cc(-c3ccc(F)cc3)cs2)=O)c[nH]c(=N)nc1O CCC(CCCC(=O)NC1CC2(CCCC2)C1)NC(C1(C)CC(F)C1)=O C1(C(N2CC(C3(NC(CCC(=C)Br)=O)CC3)C2)=O)CCc2nncn2C1 O=C(C1=COCC1)NCCCN(C1CCCCC1)C(C1CCC(F)C1)=O c1(NC)ccc(C(N2CC=CC2(C)C(=O)NCCCc2ccncc2)=O)nc1 c1(C(=O)NC(CC)CNC(C2CCC(N(C)C)CC2)=O)ccc2oc(C)nc2c1 N1(C(C(C)C2CCCO2)=O)CCC(C2(O)CN(C(=O)C3=CCCCC3)C2)CC1 c1(C(=O)NCC(CC(C)C)NC(=O)CS(C)(=O)=O)ccc2c(O)n[nH]c2c1 N1(C(C(C2(C)CN(C(CNC(=O)OCC)=O)C2)O)=O)CCCCC(F)(F)C1 C1(NC(C=C(C)C2CC2)=O)CC=C(C(=O)N2CCCC(C(C)C)CC2)C1 C1(NC(C2CN(C(Cc3cccc(C#N)c3)=O)C2)=O)CC2CC1C(O)C2O N1(C(C2(SC)CC2)=O)CC2CC1CC2NC(=O)CCc1cccc(C2CC2)c1 Cc1ccn2cc(C(N3CC4C(N(C)C(C5CCC(=O)C5)=O)C4C3)=O)nc2c1 N1(Cc2cc(OC)c(F)c(F)c2)CC2(C)C(=O)NC(=O)C2(C)C1 CC(C)CC(CC(=O)NCC1OCCC1(C)C)NC(c1c[nH]c2cnccc12)=O C(=O)(C1CCc2cccc(F)c21)NCC(C)(O)CNC(c1cncc(N)n1)=O c1(C(=O)NCC2=CCN(C(C(C(C)C)C)=O)CC2)c(F)ccc2ccncc12 C(N=c1[nH]cc2ncnc-2[nH]1)C1(CNC(c2nc(O)[nH]c(=O)n2)=O)CC1 c1(N2CCC(C)(c3ncc[nH]3)CC2)nc(N2CC3CC3C2)nc2ccccc12 c1(C(=O)NC(C)CN(C(=O)Cn2ccc(O)nc2=O)C)c(F)cccc1[N+](=O)[O-] C1(NC(c2c(C)nn(CCCC)c2Cl)=O)CCC2CC1CN2C(=O)C1=NOC(C)C1 C(=O)(C1CCCc2cncn21)N(CCCN(C(C1N(C(C)=O)CCOC1)=O)C)C c1(C(=O)NCC2(CNC(CNS(CC)(=O)=O)=O)CC2(F)F)nccn2cc(C)nc12 N1(C(C2CCCN(CC)C2)=O)CCC(C(=O)NCCCSC)(OC)CC1 N1(CCC2CCCN(C(=O)OC(C)(C)C)C2)CCc2sc(S(N)(=O)=O)cc2C1 O=C(C1=CCCN(C(c2ccc(F)cc2F)=O)C1)Nc1cc(Cl)cc(Cl)c1Br c1(C(=O)NC2CCCCC2NC(C2CCC(F)(F)CC2)=O)cc2scnc2[nH]1 C1(C(=O)NCC(O)C(F)F)(CC)CCCN1C(c1csc(CO)n1)=O Cn1cnc2[nH]c(=NCC3(C)CCOC3)nc(N3CCC(CCO)C3)c12 CC1(F)CCC(C(N2CCCC(C)(NC(c3ccnc(Cl)n3)=O)C2)=O)CC1 c1(C(c2nnnn2CCCF)NCC2(CO)COC2)ccnc(Cl)c1 C#CCC(C)(CC)C(=O)NC1CC2CC(C1)N(C(c1sc(C)nc1OC)=O)C2 Cc1cccc(C=CC(=O)N(CCN(C(=O)C=Cc2cnccn2)C)C(C)C)c1 C1(C(=O)NCCCCCC)N(C(c2cccnn2)=O)CCCC1(C)C N1(C(C(C)=CC)=O)CCOC2(CCCCC2NC(c2c(OC)ccc(F)c2C)=O)C1 c1(CC(=O)NC2(CC=C)CN(C(c3cc(C4CC4)no3)=O)C2)cn2ccsc2n1 N1(C(CCN(C)CC)=O)CC2CC2(C(=O)NC(c2ccco2)C)C1 c1(C(N2C(CNC(C(C)NS(C)(=O)=O)=O)CC2)=O)cc(C2CC2)ncn1 C1(NC(CNC(=O)OC)=O)CC=CCC1C(=O)NCC12CCC(CO1)C2 C(=O)(CC(CC)C(C)C)N1CCC(C(=O)Nc2cnc(CCC)nc2)C1C N12CCC(C1)C(F)C(=O)C1(CC1)CC2=O.C(=O)(COCCF)N(C)C CC(C)C(C#N)C(=O)NC(C1CCCN1C(=O)C(=O)C=Cc1ccccc1)C C(=O)(C1=CC2CCCCCCC12)NCCC1(NC(COCCCC)=O)CC1 c1(COC)ncc(CNC(=O)C=CCNC(=O)C=CC(F)F)[nH]1 Cc1c(NCCCSc2ccc(Cl)cc2)nc[nH]c1=NCc1cocn1 C(=O)(CCCCCc1cccs1)NC1CN(C(c2cc(CC)c(Cl)s2)=O)C1 c1(CC)cc(F)ccc1C(=O)NCC1CC(NC(c2ccc(C)s2)=O)C1 Cc1csc(=NCC(=O)N2CCCC(C)(NC(C3CC3C(=O)OC)=O)C2)[nH]1 C1(CC(=O)N(C(CNC(C2(C#N)CC2)=O)C2CC2)C)CC2(CCC2)C1 c1(CC2CC(NC(N(CC(CN(C)C)O)C)=O)C2)nnc(O)n1C C1(N(C(C2(C#N)CC2)=O)CC2CC2)CCN(C(=O)CCc2nc(C(N)=O)no2)CC1 N1(C(c2n(CC#N)ncc2)=O)CCC(CNC(C2(C3CC3)CC2)=O)CC1 CCC(F)C(=O)NCCC(C)(C)NC(c1ccc(CC(C)C)s1)=O CN1CCC(C(N2CCC(CCNC(c3csc([N+](=O)[O-])c3)=O)C2)=O)CC1=O c1(CC(=O)NC2C3CN(C(C(C)OCC(C)C)=O)C2C3)c[nH]c2cc(Cl)ccc12 N1(C(c2ccc(OC)nn2)=O)CC(N(C(=O)CC2CC=CC2)C)C2(CC2)C1 C1(C(=O)NCCCc2onc(C)n2)CC=CCN1C(=O)CC1CCCCN1C C(CCCCC(=O)NCC(CC(F)(F)F)NC(c1ccncc1F)=O)OC C(=O)(C1OCCc2ccc(C)cc21)N(CCOC)CCNC(=O)CC(C)C1CC1 Cc1[nH]c(=N)nc(O)c1CC(=O)NC(C(C)NC(=O)CCCN=[N+]=[N-])C(C)C N1(C(c2c(C)n[nH]c2)=O)CC(F)CC1C(=O)NCC1CC1[N+](=O)[O-] CC1CN(C)CCC1NC(=O)CC1CCC(NC(=O)CC2CC=CCC2)C1 C(CN=c1ccc2c([nH]1)CCCC2)C1CCN(C(C(C)(C)O)=O)CC1 N1(C(C2(CCC=C)CN(C(=O)C(C)OC3CCCC3)C2)=O)CC2(CC2)CC1C c1(C(=O)NC(CC)COC)ccc(NC(=O)C=CC2CCCC2)c(S(N)(=O)=O)c1 N1(CCN(c2cc([N+](=O)[O-])ccn2)C=O)CCc2cccnc2C1 C12(NC(C3CCN(C)C3=O)=O)CCCCC1CN(C(=O)CCP(C)(C)=O)C2 C1(N(C(N(C(C)C)CCc2ncon2)=O)C)CC2CC2C1 c1(NC(c2n(C(CC)(C)C)nnn2)c2c[nH]nc2C)ccc(O)cc1C C1(NC(C(C)OCC#C)=O)CC2CC1CN(C(=O)C(C)SCC)C2 c1(C(=O)OC)n[nH]c(=NC2C(C)CN(C(=O)C(C)(C)S(C)(=O)=O)CC2C)s1 N1(C(C(CCC)C#N)=O)CCC2CCN(C(c3ccc([N+](=O)[O-])s3)=O)C2C1 CC(=O)CCCCC(=O)N1CC(OCC(=O)NCc2c(C)cccc2F)C1 c1(CNC(CC2C(C)CC2)=O)ccc(CN(C(=O)CCC2(C)N=N2)C)cc1 Cc1cccc2c1CC(C(=O)NCC(O)CNC(c1ccc(CO)o1)=O)O2 N1(C(C(CCNC(Cn2nc(C)oc2=O)=O)O)=O)CCC2(CC1)CSC2 C#Cc1cccc(CNC(=O)C(C)(CO)NC(c2ccn(C)c2C)=O)c1 N1(C(C(=Cc2ccc(F)cc2)C)=O)CC(CCNC(c2cnsc2)=O)OC(C)C1 C1(NC(CCCC)=O)CN(C(c2cc(C)n(CCO)n2)=O)CCC1CC1CC1 C#CCC(CC(=O)NC(CN(C)C)CC)NC(=O)CS(C)(=O)=O C(=O)(C(C(C)(C)C)NC(C)=O)N1CC(CN(C(Cc2ccc(OC)nc2)=O)C)C1 CCC(C)C(C(=O)N(C)Cc1ncco1)NC(C1COCOC1)=O CC1(C)COCC1(c1nn[nH]n1)NC(=O)COc1cccc(C(F)(F)F)c1 C1(NC(C(CCN(C)C)NC(=O)CC2CCC(=O)CC2)=O)CN(C)C(C)(C)C1 C(CCCCC(=O)NC1CCN(C(=O)Cc2csc(C)n2)CC1C)OCC N1(C(c2c(C(=O)OCC)n(C)nc2)=O)CCC2(C1)CN(C(=O)C(C)CS(C)=O)C2 C1(COC)CCCN1C(=O)CC(C)NC(c1cccs1)=O N1(C(CN(CCC)C)=O)CCC(C)(NC(C2CCCC(F)C2)=O)C1 c1(CC)cc(C)nc(NCC2CCCCC2NC(C2CCOCC2)=O)n1 c1(C(=O)NCC(c2ccccc2)N(C(c2ccco2)=O)CC)cc2ccccn2n1 c1(NCC(C2CCC2)N(C(=O)C=CS(C)=O)C)ccc(C(F)(F)F)cc1[N+](=O)[O-] Cc1cn2cc(C(=O)NCC3COCCN3C(=O)Cc3cc(Cl)n(C)n3)nc2s1 C1(CC=C)(NC(=O)C=CC2CCCC2)CCN(C(=O)CC2CCN(C(C)C)C2)C1 CCS(=O)(=O)CC(=O)N1C(C(=O)NC(CCO)C(C)C)CC2CC12 c1(NC(C2(CNC(C(CC)N(CC)CC)=O)CC=CC2)=O)cc(C)ccc1O C(=O)(CCC(F)(F)C(F)F)NC1C(NC(c2c(C)scc2)=O)COC1 c12ccccc1NC(=O)C2.C1(CC(=O)NC2CC2C(=O)OCC)CCCC(=O)N1 CCCS(=O)(=O)CC(=O)N1CC(NC(=O)COc2ccc(Cl)c(Cl)c2)CC1(C)C c1(SCC)cnccc1C(=O)N(CC(C)NC(=O)CCC1CCCCN1C)C CC(C)CCC(O)C(=O)NC(C1CC1C(=O)Nc1cccc(F)c1)C N1(C(C(c2ccc(C)o2)C)=O)CCC2C(C1)CN2C(c1cn(C(C)C)nc1C)=O C(=O)(C(CO)C(C)(C)C)N1CCN(C(C2C(CC)C2)=O)C(C)C1 N1(C(C(c2n(C)ncc2)NC(c2cnsn2)=O)=O)CCCC2(CC2)C1 c1(C(=O)NCC2CC(CNC(CCC(=C)C)=O)OC2)cnc2cccnn12 c1(CCC(=O)NCC(CNC(C(CC)(C)F)=O)C)ccc2c(c1)OCO2 c1(NCCCN(C)CCO)nc(N2CCC3C(CC2)C3(F)F)nc2sccc12 C1(C(=O)NC2CC(C(F)F)(NC(C3CCCO3)=O)C2)CCC2CC1CO2 C1(C(=O)NC2C(C)N(C(=O)C3=NOC(C)C3)CC2)CC12CCCCC2 C(=O)(C(C)C(C)(C)C)N1C2C(C1)C2.Cc1cn(C)cc1NC(=O)CC(C)F C12CCC(CC1)CN2CCO.C1(C(=O)NC(C)=O)CCCN1C(C1CCSC1)=O c1(O)ccc2c(c1)COC2.C=CC(CC)C(=O)N1CC1CN(CCOCCSC)C O=C(C1=C(Cl)CCOC1)NC1CCC(C(=O)O)CC1 C(=O)(CCCCC(F)(F)F)NC1CN(C(c2cnc(N(C)C)nc2)=O)C2C1C2 N1(C(C2(CC#C)CCN(C(=O)Cc3cncc(C)c3)C2)=O)CCC(C)C(O)C1 C1(C(N(C)CC2CSCCO2)=O)CCCCN(C(=O)C(C)(F)F)C1 C1(NC(COCCCCC)=O)CC2CC(C1)N(C(C1CCCC3(CC3)C1)=O)C2 CN=C(NCCCc1nc(CNC(=O)OC(C)(C)C)no1)NCC1CC12CC2 c1(OC)ccc(C(C)C)c(C(N2CCC(CNC(c3cc[nH]c3)=O)C(C)C2)=O)c1 S(=O)(=O)(CCC(=O)N1CCCC(NC(=O)CC2CSCCS2)C1C)NC N#CC1CN(C(=O)C(F)F)CCN1C(c1ccn2nccc2c1)=O C1(CNCc2cccc(COC)c2)CCC(C)c2ccccc2C1 S(=O)(=O)(c1cccc(C(=O)NC2CCCC(F)C2)c1)NCCC(N)=O N1(C(C(C(C)C)C(C)C)=O)CCC2(CCC(NC(=O)CCc3cscn3)C2)C1 N1(C(CCC#CC)=O)CCCN(C(=O)C(C#N)Cc2ccc(C#N)cc2)CC1C CC(C)CC(C)CC(=O)N1CCCC(C)C1CNC(=O)CC(C)C1CCCCC1 C1(N(C)C(c2ocnc2C2CC2)=O)CC2CC1N(C(c1ccc(Br)cn1)=O)C2 N1(C(C2C(OC(C)(C)C)C2)=O)CCN(C(c2ccncc2F)=O)C(CO)C1 Cc1cn2ccc(C(N3CC4CC(NC(=O)C(C)(O)C5CC5)CC3C4)=O)cc2n1 C1(COC)(NC(=O)Cc2cc[nH]n2)CCN(C(c2nccnc2C(N)=O)=O)C1 Cc1cc(C)n(CCCC(=O)N(C2CCN(c3nc(C(C)(C)C)ns3)C2)C)n1 N1(CCCCOCC(N)=O)CCN(C(=O)Cc2cccc(Cl)c2)CC1 c1(C(=O)NCc2[nH]c(=N)sc2)cc2cc(Br)ccc2c(=O)o1 CCCC(C)CCCC(=O)NC1CCC(NC(c2c(C)nsc2N)=O)C1 c1(N(C)CC2CCCOC2)nc2ccsc2c(=NC2CCCSCC2)[nH]1 Cc1ccc(C(=O)NCC2CCCCN(C(C3(CCF)CCC3)=O)C2)c(O)n1 c1(OC)ccc(OCC(F)F)c(NC(=O)C(=O)NCCCN(C)C(C)=O)c1 C12(CNC(c3nc(CCC)sc3)=O)CC(C1)C(NC(C1(C)CC=CCC1)=O)CO2 c1(C(=O)NC2CC(C(N3CC(C)OCC3C)=O)C2)cnc2ccoc2c1 CC1OC2(C(=O)NCC3CCCCN3C(=O)CC3CCCC3(F)F)CCC1CC2 C1(n2cc(CCCCCF)nn2)CCOC2(CCC2)C1 C(=O)(C(C)CC(C)(C)C)N1CCC(C)C1CNC(c1ccnc(C(F)(F)F)c1)=O N1(C(=O)NC(C)CC(F)F)CCCC(C(N2CCCCC2)=O)C1 Cc1cccn2nc(C(=O)NCC3CC3Cl)cc12 C1(CC=C)(C(N2CCC(C(C)NC(c3ncsc3NCC)=O)C2)=O)CCCC1 CCC(C(=O)NCC(C1CC1)NC(c1ccco1)=O)NC(c1ccccc1)=O CC1CN(C(c2cnc(Cc3ccc(F)cc3)s2)C(=O)NC2CC2)CC(C)(C)C1 C1(C(=O)NC2(CO)CC(F)(F)C2)(CO)CCN(C(=O)COC2CCCOC2)CC1 C(C(C)C)(C(O)C(=O)NCCC(C)NC(C1(C)CCN(C)C1=O)=O)OC C1(CC=C)(C(=O)N(CCC2CC2)CC)CCN(C(=O)Cc2ncccc2C)C1 C1(C(=O)NC2CN(C(COCC)=O)CC(C)C2)COc2ccccc2O1 CC(C)CC(C(=O)N(C)CCc1cnccn1)ONC(c1n[nH]cc1[N+](=O)[O-])=O c1(C(=O)NC2(C3N(C(CCN(c4ccncc4)C)=O)CCC3)CC2)ccc(F)cn1 c1(C(=O)NCCN(C(=O)C=CC=C(Cl)Cl)C(C)C)cc(C(N)=O)cn1C N1(C(CC=C)=O)CCSCC1CCNC(=O)Cc1ccoc1 CN1CC2CN(C(c3c(Br)cc(Br)cc3[N+](=O)[O-])=O)CCN2C1=O c1(OC)nc2c(s1)CCCC2.c1(CC)nc2ncc1C(=O)C1CCCN2C1 C1(C(N2CCCCC(NC(=O)COC3CCOC3)C2)=O)CCCC12CCOCC2 C1(C(=O)NCC(CNC(c2c(CC)n[nH]c2)=O)F)CCCCN1S(N)(=O)=O C1(C(N2CC(OC(C)(C)C)C(CNC(=O)C(N)=O)C2)=O)CC(C(C)C)=NO1 CC1(CNC(c2csc(-c3ccsc3)n2)=O)CCCN1C(C1CC1(C)Br)=O CC(C)(O)CC(=O)N1CCC(C)(NC(c2cc(-c3ccccc3)ccn2)=O)C1 N1(C(c2cnc(C)nc2)=O)CCN2C(=O)C(NC(c3nn[nH]c3Cl)=O)CC2C1 c1(-c2n(C(C(C)C)C)nc(-c3ccc(Cl)cc3)n2)ccc(F)c(F)c1 C1(C(=O)NC(CC=C)CNC(c2cccc(F)c2Cl)=O)CCc2nc[nH]c2C1 C1(C)(OC)CC2CC1CC2NC(C)CC1CCC(F)(F)CC1 C1(NC(C(CC)(F)F)=O)CN(C(C2(C3CCCCO3)CCC2)=O)CC2(CC2)C1 N1(CC(=O)NC2(CCO)CN(C(=O)CC(O)C3CC3)C2)CCC(O)CC1 N1(C(C(C)(C)c2ccccc2)=O)CC2CN(C(c3cccc(O)c3Cl)=O)CC12 Cc1ccnc(C)c1CNC(=O)C1=NOC(CNC(c2ncccc2F)=O)C1 N1(C(C2(C(F)F)CC(=C)C2)=O)CC2=C(C1)CN(C(=O)C(C)(C#N)CC)C2 C1(C)(C(N2CC(OC)C2)=O)CC(O)CN1C(=O)C(F)(F)F c1(OC)ccc2c(CCNC(N3CCCC3Cc3ccncc3)=O)coc2c1 C1(C(N2CCCC(C)(NC(CC(=C)Br)=O)C2)=O)CC2CCC1CC2(F)F C(=O)(C(C)(C)C(F)F)NCC1(C)CN(C2CCN(C(C(C)O)=O)CC2)C1 C(C(C)(C)CNC(=O)Cc1csc(S)n1)N(C(=O)C(C)(C)c1cncs1)C C1(NC(C(CC)n2cncn2)=O)CC1C1CCCN(C(c2c(C)noc2N)=O)C1 N1(C(C(CC)O)=O)CCC(C)(NC(=O)C(C)(C)Oc2ccccc2)CC1 C1(C(=O)NC2(C#C)CC2)(CC)CN(C(=O)C(CC)n2ccnc2)C1 Cc1c(NC(=O)C(=O)NC2CN(C(N)=O)C3CC23)cccc1F O=C(C1Cc2c(Cl)cccc21)NC1(CNC(C2Cc3nccn3C2)=O)CCC1 C12(NC(CC(CC)N(C)C(c3cc4n(n3)CCC4)=O)=O)CCC(CF)(C1)OC2 C=C(Cl)C(C)(C)C(=O)N1CC(NC(=O)CC2(CO)CCN(C)CC2)C(O)C1 CC(CSc1cc(F)ccc1F)N=c1ccnc(NC2CC3(CCC3)C2)[nH]1 C1(C(=O)NC(C)CNC(c2ccccc2Cl)=O)CCCCC(=O)C1 C1(CC(=O)NCC(CNC(C(C)Cc2cnc[nH]2)=O)F)CCC2CC1C2(C)C N1(C(CC=C)=O)CC2(COC(CNC(c3c(CC)cccc3F)=O)C2)C1 C(=O)(C(C)(O)C(F)(F)F)NC1C(C(=O)NC(C(=O)OC)C)CCC1 C1(C(=O)NC(CSC)C)CN(C(=O)C(N2CCOCC2)C)CCC1O C1(C(N2CC(CNC(=O)CC3CSCCS3)C2)=O)OCC2CCCCC12 N1(C2C(C)C2)CCC(NC(C2(NC(=O)OC(C)(C)C)CC2C)=O)C(O)C1 CCCCC(C)C(=O)NCC=C1CCN(C(c2cnc(O)n2CC)=O)CC1 C1(C(=O)NC2CCC(CNC(CC(=C)C)=O)CC2)CC2CCCCCCC12 N1(C(c2c(C)snc2)=O)CCCC1(C)C(=O)Nc1cccnc1 CC1(C)Nc2ccccc2C1NC(C1CCC(C2CCNCC2)O1)=O C(=O)(N=C1C=C(C(N)=O)N1c1ccc(F)cc1)C1CC(C(=O)OC(C)(C)C)C1 C1(C#N)(C(=O)NCC2N(C(CCCSC)=O)CCC2)CC12CCC2 C1(CN(C2CCN(CC(C)C)C2)C(=O)CN(C)C)CCC(C)CC1 c1(CC(=O)NCc2cc(C3CC3)n[nH]2)cc(C(N2CCCC2C2CCOC2)=O)cs1 C(=O)(C#CC1(C)CC1)N1CCCC(CCNC(CC2N(C)CCOC2)=O)C1 Cc1cc(F)ncc1C(=O)NC1(C)CN(C(=O)COc2cc(F)cc(F)c2)C1 c1(C(=O)NC(C(C)NC(=O)CNc2ccccn2)C)c(Cl)cncc1Cl N1(C(C(CC#C)(C)CC)=O)CCCCC2(CCN(C(C34CCC(CC3)C4)=O)C2)C1 C(C1=CCN(C(=O)CCc2cscn2)CC1)N(C(=O)COC(F)(F)F)CCCO C1(C)(NC(C(C=C)CC)=O)CCCCC1C(N1CCC(n2cncn2)C1)=O c1(C(=O)NCc2cc(C(=O)NCCC(C)C)on2)ccn2ccccc12 c1(C(N2CC(O)(C(C)NC(c3csc(CO)n3)=O)C2)=O)cc2ccccc2nn1 N1(C(c2ccc(C)cc2)=O)CCC(O)C(C(N2CCC(O)C(CO)C2)=O)C1 n1(C(C)C)ncc2c(NC(C3CCCO3)C)[nH]c(=NCC3CC3)nc12 C1(NC)CCCN(C(=O)C(=O)NC2CCC(n3ccnn3)C2)C1 c1(NC(CNC(C)=O)=O)ccncc1C1=CCC(C(C)(C)C)CC1 C(=O)(CCC(C(=O)N1CC(NC(C)=O)C1)NC(c1cc(Cl)c(F)cc1Cl)=O)OC Cc1cccc(CCC(N2CCC(NC(=O)CCC=CBr)C2C)=O)c1 n1(CCN2CCN(C(c3csc(Cl)c3Cl)=O)CC2)cnc2ccccc12 C1(C(=O)NC(CNC(C=CCOC)=O)C)CCC(C)O1 c1(C(=O)NCC2N(C(C3(CC=C)CCC3)=O)CCCC2)nc(C)n(C)c1C c1(OC)ccc(C(N2CCN(C(C3CC3F)=O)CC2)=O)c(F)c1 C#CCC(C)(C(=O)NC(C)CCc1cn[nH]c1)NC(=O)COCC(=O)NC N1(C(CCc2n(C)cnn2)=O)CCCC12CCN(C(C1CCN1S(C)(=O)=O)=O)C2 C1(C)(NC(c2ccc(C(=O)NCCCCC(=O)OC)cn2)=O)CCCCCC1 c1(SCC2(C(=O)Nc3cn(C(C)C)nc3Br)CC2)ccc(Cl)nc1Cl c1(OC)ccc2c(c1)CC(C(=O)NC(C)(C)CNC(=O)Cn1cccn1)O2 Cc1oc(-c2cnn(C)c2)nc1C(=O)NC(C)C(C)F c1(CNC(C)C)c(OC)ccc(C)c1C.C1(CC)CS(=O)(=O)CC1N N1(C(C2CCCN2C2CC2)=O)CCC(F)(C(=O)N)C1.c1(C)cnc(S)nc1 C1(NC(C2(C)CCCS2)=O)C=CCN(C(c2cnn(C(C)(C)C)c2N)=O)C1 c1(C(=O)NCC2N(C(C(CC)(C)OC)=O)CC2)cc(C)c2c(c1)CCC2 N1(C(C2C(C)=CCS2)=O)CC2CCC2(NC(C2CC2(F)Cl)=O)C1 N1(C(c2cn(C)nc2-c2ccco2)=O)C2CCC1CN(C(c1cncnc1)=O)C2 c1(C(=O)NC(C)C(C)NC(c2cc(O)ncn2)=O)cccc2c1nnn2C C1(CC)(NC(C2CN(c3nncs3)C2)=O)CCN(C(=O)C(C)OC)CC1 N1(C(C(N2CCC(C)(C)CC2)=O)=O)CC(C(=O)OC(C)(C)C)CC12CCC2 O=C(C1CCCc2nc[nH]c21)N1CCC(N(C(C2CCOC2)=O)CCO)C1 C1(NC(CC2(OCC)CC2)=O)CC(O)CN(C(c2cn(CC(N)=O)nn2)=O)C1 C12(C(N3CCCC(O)(CCNC(=O)CC4CC5CC5C4)C3)=O)CCC(CC1)OC2 c1(C(=O)NC2(C)CCCN(C(CC(C)F)=O)C2)cc2cc(Br)cn2cn1 C1(C(F)F)(CNC(CN2CCC(OC)C2)=O)CCN(C(c2c(C)nsc2N)=O)C1 N1(C(C(F)=CC)=O)CCOC(CCCNC(C2CC(=O)N(C)C2)=O)C1 N1(C(c2c(CC)nns2)=O)CCC2(CC1)CC2NC(C1(OC)CCCCCC1)=O C1(CNC(C(C)SCCCC)=O)CN(C(c2cc(Br)co2)=O)C2(CCC2)C1 C1(CNC(CC2C(C)C2)=O)CN(C(c2cc(CC3CC3)nn2C)=O)CCC1(F)F CC1(C)COC(C(=O)NCC2CCN2C(=O)COC2CCCCCC2)CO1 n1(CCOC)nnnc1C(c1cncn1C(C)(C)C)NC(C1CCCCC1)C C1(NC(CCc2c(C)nn(C)c2)=O)CN(C(=O)COCC2CC2)CC1C1CC1 C(=O)(C(O)CCC(C)C)NCC(C)(CNC(C1CCCCS1(=O)=O)=O)OC c1(CNC(C(C)C(C)O)=O)cccc2c1CN(C(C1(C#N)CC=CC1)=O)C2 c1(C(N2CCN(C(=O)CC3(O)CCCC3)CC2C2CC2)=O)ccnc2[nH]ncc12 C1(CNC(c2ncoc2C2CCC2)=O)CN(C(C2CCCO2)=O)CC12CC2 N1(C(C2(CNC(c3cc(C)c(C)nn3)=O)CC(C)(C)C2)=O)CCCC(C)(O)CC1 c1(C2(CNc3nccc(NC(C4CCCO4)CC)n3)CCC2)ccc(F)cc1F c1(OCC(=O)NCCC(C)NC(=O)Cc2ccsc2)ccc(F)cc1O c1(C(N(CCN(C(COCCCC#C)=O)C)C)=O)c(F)cc(OC)cc1Cl C1(C(C)=O)CC(C(=O)NCC(C)CNC(=O)CC2(CSC)CC2)C1(C)C Cc1cn(C)cc1C(=O)NC(C(=O)NCCCn1nccn1)C1CCOC1 C(CC(C)C(=O)NC(c1ccccc1OC)CNC(=O)COC)OC c1(CNC(C2N(CCCCC)CCC2)=O)cccc(COC)c1Cl N1(C(C=CC=CC)=O)CCCC(C)(NC(c2ccc(Cl)nc2Cl)=O)C1 C1(CC(=O)NC(C(C)C)CCNC(c2ccc(C#N)[nH]2)=O)SC2=NCCN2C1=O C1(CC(=O)NC2CC(CNC(CCc3cn(C)nc3)=O)C2)CCCC(=O)N1 c1(C(N2CCC(CNC(=O)CCC(F)(F)F)C2)=O)ccc2ccc(Br)cc2n1 c1(C(=O)NC2(CNC(C3CC(C(=O)OC)C3)=O)CCC2)sccc1Cl C1(C2CC2)(NC(CN(C(c2ccc(C)n2C)=O)C)=O)CCCC1 c1(NC(=O)NCC23OC(=O)C(CC2)C3)cccc2nccn12.C12CCCN1C2 c1(SC(C)C(=O)NC2C3CC2N(C(=O)CCc2cn(C)cn2)C3)ccc(F)cc1 C1(C(=O)NCCCN(C(=O)C=CC(C)(C)C)C)CCc2ncncc2C1 c1(N(CC(C)CNC(c2cc3ccsc3[nH]2)=O)C)ccc([N+](=O)[O-])cc1C#N C1(C)(CNC(C(C)NC(CC)=O)=O)CN(C(=O)CCNC(C)=O)CCO1 C1(CC(=O)NCC(C)N(C(C2ON=C(C(C)C)C2)=O)C)CCCNC(=O)C1 c1(C(=O)NCC(CO)NC(c2coc(C3CC3)n2)=O)ccn2ccsc12 N1(C(c2n(C)ccc2)=O)CCN(C(=O)COc2ccnc(C(N)=O)c2)CC(O)C1 C1(CN(C(=O)Cc2ccon2)C2CC2)CCCN(C(=O)CCc2nccs2)C1 N#Cc1csc(C(=O)NC2CCOCC2C(=O)NCCc2cccnc2O)c1 N1(C(CNS(CCOC(C)C)(=O)=O)=O)CC(C)CN(C(=O)C2CC2)CC1C Cc1ccc(OC(F)F)cc1C(N1CCC(CO)(NC(C2CC2CF)=O)CC1)=O C(N=c1[nH]c2ccc(S(=O)(=O)N3CCCCC3)cc2s1)C1C(C)(Cl)CCC1 C(=O)(C(O)CCCCC)NCC1(F)CC(CNC(C2C(=C)C2)=O)C1 S(=O)(=O)(c1ccccc1Cl)NC(C1CCC(C)S1)=O c1(CCC(=O)NCC2(C(=O)NC3(CCO)CC3)CC2(F)F)ccccc1 S(=O)(=O)(c1[nH]c(=NCc2ccnn2CC)ccc1Br)NCC(CC)C(C)(F)F C1(C(N)=O)CN(C(C2CN(C(=O)Nc3ccccc3)CCO2)=O)CC12CC2 C(=O)(C(C)(C)C1CCN(C(=O)C(C)NC(=O)C(C)(C)C)C1)N(CCOCC=C)C c1(C(=O)NC2CC(CNC(c3c(C)nc(CC4CC4)o3)=O)C2)nc(Cl)ccc1Cl C1(S(C)(=O)=O)(C(=O)NCC2(COC)CN(C(C3(CC(C)C)COC3)=O)C2)CC1 c1(SC)ccc(C(c2nnnn2C2COC2)NC(C)C(C)C)o1 C1(NC(C2CC(OC)C2)=O)CCC(C)(NC(=O)CCC2NC(=O)NC2=O)CC1 N1(C(CCOCCNC(C2CCCC(C)C2)=O)=O)CCC2(C1)CC2(F)F C(=O)(C1Cc2ccccc21)NCC(C(=O)NCC(CC(=O)OCC)(C)C)C C1(C(N(C)CC2CCCSC2)=O)CCCCC1NC(=O)Cc1cccc(Cl)c1 CC1C(C(=O)NC2(CCO)CCOC2)CCN1C(=O)C(C)c1cccs1 N1(C(COCCCCCC)=O)CCC(CN(C)C(C2CCOC2C)=O)CC1 N1(C(C2CC2(F)Cl)=O)CC2(CO)CC1(C(=O)NCCc1ncccc1F)C2 C(CCCCC(=O)N1CCC=CC1C(=O)NCC1CC(=C2CC2)C1)OCC C1(C(N2CC(C)(CC(=O)Nc3nc(Cl)sc3Cl)C2)=O)CCC(c2ccccc2)CC1 C(=O)(CC(C)(C)CC(=O)NCCC(O)CNC(=O)CCC1CC1)OC CC(C)(O)C#CC(=O)N1CCCC1CC(=O)NCCCN1CC=CC1 N1(C(C(C)n2ccnn2)=O)CC2(CO)CC1(CNC(c1ccoc1)=O)C2 C(C(C)(C)C(=O)NC(C1CCCN(C(=O)CN(C)C(C)C)C1)C(C)C)SC C1(CC(=O)NC2(COC)CC2)CN(C(=O)Cc2ccon2)CC12CC2 C(=O)(C=CCCCC)NCC(CCCC)NC(=O)Cc1cn(C)nn1 C(=O)(C(F)(CNC(C1CNC(=O)O1)=O)C(C)C)N1CCC(CCCC)CC1 CC(C)C(CNC(=O)CN(C1CC(C#N)C1)C(C1CCC1)=O)C(C)C C1(C(=O)NCC(CN(C(=O)C2=CC(C)(C)C2)CC)(C)C)OCC2CCCCC12 c1(SC(C)(C)C)cccnc1C(N1CCC(NC(=O)C2=CCCS2)C1C)=O N1(C(CC2C(OC)CC2)=O)CCN(CCCNC(C2CCCN2C2CC2)=O)CC1 N1(C(CCOCCC)=O)CCC(COC)(NC(C2Cc3nccn3C2)=O)CC1 c1(OC)cc(Cl)ccc1-n1nc(CC2(C)CC2)nc1COC1CCOCC1 c1(CNC(C=CC(C)NC(=O)CC2CC2)=O)cccs1 N1(C(C(C(C)C)O)=O)CC2CC(C3C(=C4CCOCC4)N3C)C1C2.c1ccccc1 c1(C(=O)NCC(C)N(C(CCC=C=C)=O)C)nn2cccnc2c1Cl c1(C(=O)NCC(=C2CCN(C(c3cc[nH]n3)=O)CC2)F)cc2c(Cl)cccc2[nH]1 C(C)(CO)(C(=O)NCc1cc[nH]c1C(=O)NCC1CC12CCC2)OC N1(C(C2C(C)CCO2)=O)CC2CN(Cc3occc3Br)CC2C1 C1(NC(C(COC)C)=O)CCCCCN(C(=O)C(C)(C)C(C)C)C1 N1(C(C(F)=CC)=O)CCC(C(C)(O)CNC(=O)CCC23CCC(CC2)C3)CC1 C1(CC(=O)OCc2c(C(=O)OC(C)(C)C)csc2)CC2CCC1C2 N1(C(c2cccc(-c3ccco3)c2)C(=O)NCC)CC2CCC(O)C2C1 O=C(NNC(=O)Nc1ccccc1F)c1c(Cl)nsc1Br c1(C(=O)NCC(CNC(C2(c3cccc(C)c3)CCC2)=O)C)cnc(Cl)c(N)c1 C1(CC(=O)NC(c2cnc[nH]2)C)COCCN1C(c1cncc(C(F)(F)F)c1)=O N1(C(C2CCN(C(CC3(CSC)CC3)=O)C2C)=O)CCOC(C#N)C1 N1(C(C2(CC)CCC2)=O)CCC(CO)(NC(c2sc(C)nc2C(F)(F)F)=O)CC1 C1(OC)CC2CC(NC(=O)C=CC3CCN(C(=O)CC(C)(O)COC)CC3)CC12 c1(C(=O)NC(C(=O)N(c2ccnc(C)n2)CC)C2(O)CCC2)cncc(OC)n1 C(C(C)CC(=O)Nn1cncn1)NC(CNC(COC)=O)=O c1(OC)ccc(CCC(N2C(CNC(=O)CSCC(N)=O)CC3CC23)=O)cn1 c1(COC)nc(C)c(C(N2CCCC2CCNC(C2(O)CC2(C)C)=O)=O)s1 O=C1NC(=O)C2(CCCC23CN(C(c2cccc(-n4cnnc4)c2)=O)C3)N1 c1(NC(c2ccc(Cl)o2)=O)ccc(NS(=O)(=O)Cc2ccccc2)cc1F C(=O)(C(C)(C)C(=O)NC)N1CCC(c2c(CNC(C(C3CC3)OC)=O)c[nH]n2)C1 c1(NC(=O)NC2CC3(CCC3)C2ONC2CC2)cc(Br)cc2c1OCO2 c1(C(N2CCC(CN(C(CC(C)(C)OC)=O)C)C2)=O)ccc2c(n1)CCC2=O N1(C(c2c(CC)c[nH]c2)=O)CCC2CCCC12C(=O)NC1(C)CC(O)C1 C1(NC(C(CC)(O)c2ccccc2)=O)CCN(C(=O)Cc2ccsc2C)C(C)C1 c1(C(=O)NCCC2N(C(C3C(C#N)C3)=O)CCOC2)cc(O)nc(C2CC2)n1 c1(-n2c(C)c(C(=O)Cn3cc(I)nn3)cn2)ccc(Cl)cc1F CC1CN2CCN1C(C(=O)NCC(C1CC1)NC(c1ccc(C(F)F)cn1)=O)C2 C1(F)(C(N2CC(C(C)NC(C(CC)C)=O)C2)=O)CC=CCC1 O=C(C(F)(F)C1CC1)N1CCC(C(c2cn(-c3cccnc3)nn2)C2CCCO2)C1 C(=O)(C1(O)CCCc2ccccc21)NCCc1c(C)c(Br)ccc1 C1(CNC(c2cnnn2C)COC)CC2C=CC1CC2 c1(OC)cc(Cl)c(Cl)cc1NC(=O)C(=O)NC(C1CCCOC1)C c1(N2CCC(CC)C2)nc(N2CCn3nc(C(C)(C)C)cc3C2)nc2c1CSC2 C(c1ccc(Cl)nc1)=CC(=O)NCCCC(C)NC(C1C=CC=CC=C1)=O C(=O)(C(O)CCC(C)C)N1CCC(CNC(c2nc(C#C)sc2)=O)C1 c1(C(=O)NCC(CCC)C(=O)NCC(F)Br)ccc2n[nH]cc2c1 Cc1cccc(C2(O)CCN(Cc3cn(-c4ccc[n+]([O-])c4)nn3)CC2)c1C C(=O)(C(F)C(C)(C)O)NCC1(CC(=O)N(CCC(N)=O)CC)CC1 C1(N(C(c2ncc(OC)nc2)=O)C)CCCN(C(=O)C(CSC)OC)CC1 c1(N2C3(CC(COC)C3)CC2)ncnc2ccc(F)cc12 c1(CN2C(COC)CN(C(C3CCCC(C)C3)=O)CC2)cc(Br)cc(C)c1O c1(C(N(C(C)C(=O)NCCOC2CCOC2)C)=O)cscc1Cl Cc1ccc2c(N3CCN(C(=O)C(C)(O)CC(F)F)CC3)ncnc2c1 C1(NC(c2cc(C)c(C)[nH]2)=O)CC=C(C(=O)NCC(C)C2CCC2)C1 CS(=O)C=CC(=O)NCC(C1CCN(C(C2CCC(N(C)C)CC2)=O)CC1)(C)C N1(C(C=CC(=O)N(C)C)=O)CCC2CCC(NC(c3cc(Cl)nnc3O)=O)C1C2 N1(C(C(C)NS(CC)(=O)=O)=O)CCOC(C(C)NC(c2cnn(C)c2N)=O)C1 O=C(CCC(=O)NC(c1ccccc1)C(C1CCOC1)=O)Nc1cccc(Br)c1 N1(C(c2c(CC)cco2)=O)CC2CCCCN2CC1CNC(=O)CNC(=O)C1CC1 C(=O)(C(CNC(=O)CSC(F)F)C(C)(C)C)N1CCCC(C#C)C1 N1(C(c2c(C)csc2Cl)=O)CC2OCCN(C(c3c[nH]c(=O)cn3)=O)C2C1 c1(C(CNC(C2(O)CC2)=O)NC(C2CCSC2)=O)ccc(Cl)cc1 N1(C(CCCOC)=O)CCC(C#N)(C(=O)O)C1.c12cccc(c1)NC(=O)OC2 CC(CC(=O)N1CCCC1CN(C(=O)C=CC(C)(C)C)C)CC(F)(F)F c1(OC)ccc2c(Br)cccc2n1.c12nnc(o1)COC(=O)N(CCCC)C2=O C1(C(N2CC(N(C(C(C)CN3CCOCC3)=O)C)C2)=O)CCCCN(C)C1=O N1(C(Cc2c(C)scc2)=O)CCOC(CC(=O)NC2CS(=O)(=O)C2)C1 N1(C(CC=CCC)=O)CCCN(C(=O)CSc2nncn2C(C)C)CC1C N1(C(COCC(C)C)=O)CCCCC(NC(c2cc(C(N)=O)cn2C)=O)C1 Cc1ccc(C(=O)NCC(C2CCCC2)NC(=O)C2=CCOC2)c(F)c1F C1(C(=O)NCCC(CC)CN(C)C)CN(C(C2CC2C(=O)OC)=O)CC12CC2 c1(-c2cnc(OCC)nc2)cc(C(=O)NCC(N)=O)cc2c[nH]nc12 C(C(=O)NCCC1CN(C(c2ccccc2)=O)C1)(C(C)C)N(CC)CC c1(C(=O)NCC(C)(C(C)C)NC(c2ccc(OC)cc2)=O)cnn2c1N(C)CC2 N1(C(COCCCC#C)=O)CC(CC(=O)NCCn2cncn2)CC1C C1C(C)(C)CNC(=O)C(CC(C(=O)NC2CC2)C)N1C(C)C.C(C)(C)(C)OC C12(CNC(=O)CC3CCOC3=O)CC(CN1C(=O)CCC1CCCO1)C2 O=C1NC(c2c[nH]c3c(Br)cccc23)C2=C1CN(c1ccc(F)cc1Cl)C2=O C=C1COc2c(C(N3CC(F)(F)CC3C(N)=O)=O)cnn2C1 C1(N(C(=O)CC2CC3(CC3)C2)CCO)CCN(C(=O)Cc2nc[nH]n2)CC1 c1(C(=O)NCC2CC(NC(C3(OC(C)C)CCOC3)=O)C2)cnc[nH]c1=N n1(CC(=C)C)nnnc1C(C1(c2cccs2)CC1)NC1CCCO1 CC1CC=C(C(=O)N2CC3CN(C(c4cc(C#N)ccc4F)=O)CC3C2)CC1 Cc1nc(F)ccc1C(N1CCOCC(NC(=O)Cc2ccc(Br)cc2F)C1)=O N1(C(c2cc(CCC)on2)=O)CCCC1(C)CNC(c1nocc1Br)=O C(=O)(C1c2c[nH]nc2CN1C(=O)Cc1ccoc1C)NCc1c(C)cccc1 c1(C(=O)OCC)ccnc(Cc2csnn2)c1.C12CN(C1)C(=O)NC(=O)CO2 c1(NC(=O)OCCOC)ccc2cc1NC2=O.c1(N(C)C)ccccc1C(C)C O=C1CC(=O)NC(C(=O)NC2(CC(N3CCOCC3CCO)=O)CCCCC2)C1 c1(C(N2CC(CC)C(NC(=O)CC3CC(C)=NO3)C2)=O)ccc(S(=O)(=O)NC)o1 C1(O)(CNC(CS(N)(=O)=O)=O)CCN(C(=O)CCC(=O)c2ccc(F)cc2)CC1 C1(C(C)NC(COC(CC)CC)=O)CCN(C(=O)C(=O)NCC(F)F)C1 N1(C(CC=CCC)=O)CCC(N(C)C(C2CCSC2)=O)CC1 c1(C(N2CC(C(C)NC(C3(C)N(C)CC(OC)C3)=O)C2)=O)c(O)ccc(Cl)c1F C(=O)(CC1=CCCC1)NC1C(C(=O)NC(C(C(=O)OC)C)C)CCOC1 C1(C(=O)NC(c2ccccc2)C(=O)N2CCCC2)CCN(Cc2n[nH]cc2F)C1 C#Cc1ccc(C(=O)NC2(C)CC(F)(F)C2)cc1.C(=O)(CC=CC=C)NC(=O)C1CC1 C1(C(N(CC(CN(C)C(c2ncoc2C(C)(C)C)=O)O)C)=O)OCCC1(C)C C(C1=CCN(C(=O)C2=CCCS2)CC1)NC(C(C)(C)c1ccccn1)=O C=CCC(C)(C)C(=O)N1CCC(C)C(NC(=O)CCc2cscc2Br)C1 C1(N(C(=O)CC#N)C)CCCC(CF)C1.c12csc(c1)CNC2=O N1(C(c2c(C)con2)=O)CCN(C(=O)CC2CCOCC2)CC1CF C1(C(=O)Nc2cn(C)nc2)C2CCC(C2)C1NC(=O)Cc1csnn1 C1(NC(CC2(C=C)CC2)=O)CC(CNC(=O)C=CCF)C1(C)C C1(C(=O)NCC2CC(F)CN2C(c2cccnn2)=O)CC2(C1)CC(F)(F)C2 N1(C(C(c2ccc(OC)cc2)O)=O)CC2(C1)C(NC(=O)CCCF)CCS2(=O)=O C1(C(=O)NC2CC(CNC(=O)C(C)SC3CCCCO3)C2)(OCC)CCCC1 C(C(F)(F)CCC(=O)NC1CCCCCCC1O)n1cc(C(C)OCC)nn1 CC1(C)C(C(C2CC2)NC(=O)CCc2cccs2)CCN1C(=O)CC(F)(F)F C(C1=CCCSC1)(c1n(CC(=C)C)nnn1)NC(c1ccccc1)CF c1(OC(C)C(=O)NN(C(=O)C=CCF)C)cccc(F)c1.C1(C)(CF)CC1 c1(C(=O)NCC(N(C(CSCC)=O)C)C2CC2)ccc(-c2ccccn2)s1 CC1CN(c2cc(Cl)nc(C(C)(C)C)n2)CCC1NC(c1cc2c([nH]1)CCC2)=O CN=C(NC(C)(C)CN(C)CC=Cc1ccccc1)N1CN(C)C(=O)C1C CC1(C(=O)NOCC2CCCCCCC2)CCCC1(F)F.C1(C=O)CC12CCCC2 c1(OC)ccn2cc(C(=O)NC3CCCC3NC(c3oncc3C)=O)nc2c1 C1(C(N2CC(C)(CC)C2)=O)CC(C)(C)CN1C(C1CC(=O)C1)=O C1(C(N2CC(NC(c3c(OC)ccs3)=O)C(C(F)F)C2)=O)CC2(CCC2OC)C1 c1(N(CC#CCNC(c2nc(C)sc2C)=O)C(C)C)ccccc1[N+](=O)[O-] N1(C(c2ccn(C(C)(C)C)n2)=O)CC2(CCCC2NC(=O)Cc2cnsc2)C1 c1(CC(=O)NC(C(C)NC(c2cnc(C)[nH]2)=O)C)ccc(F)cc1Br C1(OC)(CNC(c2c(Cl)sc(C)c2C)=O)CCN(C(C2(C)CC2F)=O)CC1 N1(C(C(CC)(C#N)CC)=O)CC2OCCN(C(C3CCCSC3C)=O)C2C1 O(NC(=O)C(CNC(c1cnccc1C)=O)C(C)C)Cc1ccc(C)nc1 CC(C)C(C)CC(=O)NCC12CC(NC(C3SC4C=CC3CC4)=O)(C1)C(C)O2 c1(C(=O)NC2CCN(C(CSCC(N)=O)=O)C2)cc2cc[nH]c(=O)c2s1 S(=O)(=O)(c1ccccc1F)NCC(N1CC(NC(C(F)OC)=O)CC12CCC2)=O C1(C(=O)NCC2CCN(C(Cc3ccc(C)o3)=O)C2(C)C)CCOCC12CCC2 c1(-c2nc(NC(C3CCOC3)COC)on2)nccnc1OC C1(C(=O)NCC(C)CNC(=O)CCN2CCCC2=O)CC12CCCCC2 N1(C(C2CCC(NCc3cn(C(C)C)nc3)C2)=O)CCC2SC(=O)C=C2C1 c1(SCC(=O)N(CCCOCCN(C(C(=O)NCC)=O)C)C)n[nH]c(C)n1 N1(C(CCc2nnc(C)n2C)=O)CC2(CNC(C3(C)CC=CC3)=O)CCC1CC2 C=CCN=C(NCc1ccc(NS(=O)(=O)C(F)F)cc1)NC.C1(C)(C)CNC(=O)C1 C(=O)(C1=CC2CC=CCC12)N1CC(O)(CNC(c2[nH]c(CC)c(Cl)n2)=O)C1 N1(C(CCC#C)=O)CCC2(C=C(C(=O)NCC(F)(F)F)C2)C1 C1(NC(CCN(CCC)C)=O)CC2CCC1(NC(c1coc3c1CSC3)=O)C2 C(=O)(C1CCCc2sccc21)N1CC(O)(CN(C)C(C2COCC(C)(C)O2)=O)C1 c1(C(=O)NC2CCCN(C(C3CC=CCO3)=O)C2)cccc2cnnn12 C1OC2CCC1CC2.c1(OC)ccc(NC(=O)NCc2cccc(OC)c2)nn1 N1(CC=C)CCN(C(=O)CCN2CCN(C(=O)C(C)C)CC2)CC1 N1(C(C2CC(N(C)C)C2)=O)CC(F)CC1CNC(=O)C=CC1(C)COC1 C(CCCC(C)(C)C)NC(C(C(C)O)NC(=O)COCCF)=O C1(NC(COCCOC)=O)CCc2c(n[nH]c2C)C1 n1(CC(C)O)cc(CCNC(=O)C(c2cccn2C)=O)nn1 C(CCCCCC)(c1n(CCCC)nnn1)NC(C1CC(C)C1)=O CC1CN(C(=O)Cc2cnco2)CCC1NC(=O)CCCC(=O)N(C)C CC1C(NC(c2cn(C)nn2)=O)CCCN1C(=O)CCc1ccccn1 C1(CC(=O)N(C2CC(C#N)C2)CC(=O)N(C(CCO)C(F)F)C)C(C)(C)C1(C)C c1(CNC(=O)CC2CCC2)csc(CNC(C2CCC(=O)N2)=O)n1 CC(CC(=O)NC(C(=O)NCc1ncco1)C1CC1)n1cccn1 CC(C)(Cc1ccc(Br)cc1)C(=O)Oc1ccccc1-n1ccnc1 CC(N=c1[nH]c2c(c(=NC3CCCS(=O)(=O)C3)[nH]1)CCCCCC2)c1cnc[nH]1 c1(C(=O)NC2CC(NC(c3ncc(OC)cc3F)=O)C2)cc2cc(F)ccc2[nH]1 C(CCCCC(=O)NCC1CC12CCCCC2)N(C(C(c1cnn(C)c1)C)=O)C C1(CCCNC(c2c(C)nco2)=O)CN(C(c2cnccc2N(C)C)=O)CCO1 N1(C(c2cnc(Cc3cccc(Cl)c3)s2)C(=O)NC(C)C)Cc2ccccc2C1 c1(CN2CC(NC(c3cccc(NC(C#C)=O)c3)=O)C2)cnc(Cl)c(C)c1 N1(C(C(CC#C)C)=O)CCC(CCOC)(NC(=O)CC(C)c2cnn(C)c2)CC1 c1(OC)cccc(C(C(=O)NCC(F)CNC(c2nc(C)sc2C)=O)OC)c1 c1(C(N(CCCNC(=O)CCc2cccnc2F)C)=O)ccccc1O C1(CN(C(=O)CCc2cncnc2O)CC)CCCN(C(=O)Cc2ccsn2)C1 O=C(C1Cc2ccc(Cl)cc21)NC1CN(C(c2ccc(Cl)o2)=O)CC(F)(F)C1 c1(C(N2CC(CNC(C(CC)OCC)=O)(COC)C2)=O)ccnc(OC(F)F)c1 N1(C(C2(CC)CCN(C(=O)CC3CCC(OC)CC3)C2)=O)CCC12CCN(C)C2 CC(CC(C)NC(=O)CCC1CC1)NC(c1n[nH]c(-c2ccccn2)n1)=O N1(C(CC(CCC)O)=O)CCC(C(=O)N2CC(C(N)=O)C(C)C2)=C(F)C1 C1(C(CC)OCC)CCN(c2nnnn2C2CCC2)CC1 N1(C(CC)=O)C2CCC1C(F)C(NC(c1cc(C)nc(C(F)F)n1)=O)C2 C(=O)(CC(C)C(=O)N(CC(=O)NC1COC2(CCC2)C1)CCOC)OC CN1C(=O)CN(CC(N2CCC(NC(c3ncnc4sccc34)=O)C2)=O)C1=O C(=O)(CCCn1cncn1)N(C(C)C(=O)NC1CCC1N(C)C)CC C1(C(=O)NC(C2CCN(C(c3csc(-c4ccoc4)n3)=O)C2)C)CC(F)(F)C1 C1(C(=O)NCCCN(C(C2(OC)CCCC2)=O)CCO)CC12CCC(F)(F)CC2 C(=O)(C#CC1CCOCC1)N1CCN(C(c2c(S(=O)(=O)NC)scc2)=O)C(C)C1 c1(C(N2C3CN(C(C4(CC)CC4(F)F)=O)C(C3)C2)=O)c(C)ccc2ccccc12 C1(C(C)C)CCCN(C(=O)CN(C(c2ccnnc2)=O)CC2CC2)CC1 CC1(C)CC(C(=O)N2CCC(CO)C(NC(c3nc4cnccc4s3)=O)C2)=NO1 C(=O)(C1=NOC(c2nc(COc3c(F)cccc3Cl)no2)C1)OCC c1(C(C)C)cc(C(=O)NCCC(O)CNC(=O)CN(C2CCSC2)C)ccc1O c1(C(=O)NCCCCC(CO)NC(C2(C)CC2)=O)cc(Cl)c(F)c([N+](=O)[O-])c1N C(CCC(=O)NC(c1ccccc1)CNC(C12CC(C)C1C2)=O)SC N1(C(c2ccc(OC)cc2OC)=O)CCC2CCC(NC(c3cc(C)c[nH]3)=O)C12 CCCS(=O)(=O)C(C)C(=O)N1CC2CC2(CNC(c2cnc(O)n2C)=O)C1 C1(C(=O)N(c2ncc(C#C)cc2C)CC)CCN(C(C2CC2=C)=O)CCC1(F)F Cc1ccc(-c2ccc(C(=O)NCC(c3cnn(C)c3C)N3CCCC3)o2)cc1 N1(C(C=CCC)=O)CC(CC(=O)NC2CC2(C)C(C)C)CC1(C)C C(=O)(C1=C(Cl)CCC1)NC1C(NC(c2ccccc2S)=O)CCC1 N1(C(COCCCN(C)C)=O)CC2(CC2)CC1CC(=O)NCC(F)(F)CO c1(CC)cc(N)c(C(=O)NCC(CNC(=O)CCCCCN(C)C)OC)c(F)c1 N1(C(C(=O)NN2CCC(NC(=O)Nc3ccccc3)CC2)=O)CC(O)(C2CC2)C1 c1(CCCC(N2CCC3C(C(C)=O)C3C2)=O)ccc2c(c1)CC(=O)N2 c1(C(N)=O)ccnc(C(=O)NC23CC2CN(C(C2CSCCS2)=O)C3)c1 c1(C(=O)NCC(C2CCC2)NC(C(COC)(C)OC)=O)cnc2c(C)cccn12 c1(C(=O)NC(C2CCCN(c3nccc(OC)n3)C2)C)ccc(N)c(Cl)c1 C=CCC(C(=O)NC(CNC(=O)CCNS(C)(=O)=O)C(C)(C)C)NC(C)=O C1(CCC)CN(C(c2ccncc2Br)=O)CCN1C(C12CC(O)C1C2)=O c1(C(N2CCCCC(NC(C3(CO)CCC3)=O)C2)=O)cc([N+](=O)[O-])c[nH]1 Cc1cc(C)n(CC(N2CC(CNC(C3CC3(C)Br)=O)C2)=O)n1 Cc1cc(C)c(C(=O)N(C2CC(NC(c3cc(C4CC4C)on3)=O)C2)C)cn1 CCCC(C(O)C(=O)N1CC2C(C)C2C1)NC(=O)CC1CC(CC)=NO1 C1(C(=O)NC(c2cccnc2)CC)CC12CCN(C(=O)CC1CC=CC1)CC2 C#CC1CC2CCC1N(C(=O)C(c1cnn(C)c1)NC(=O)C1=C(C)OCC1)C2 CCC(F)(C(=O)SCCOC)C(=O)NC(C)CNC(C)=O.C12CCN(C1)C(=O)CO2 C(=O)(C(C)C(C)C(C)(C)C)N1CC2(CCN(C(CCc3cnc(C)s3)=O)C2)C1 CCC(CCC(=O)NCC(O)CC(F)(F)F)NC(c1cccnc1NC)=O N1(C(c2c(CCC)nco2)=O)CCN(C(=O)COC)CC1 C(=O)(C(F)CC(C)(C)C)NC(CC#C)C(=O)NCC(CCC)OCC C(N=c1ccc(Br)c(S(=O)(=O)N2CCCOC(C)(C)C2)[nH]1)c1c(NC)cccn1 C(CCC(C(=O)NOC1CCC1)NC(C1CCCN1C)=O)OC CC1CCC(NC(=O)Cc2cccnc2)CN1CCCOC(F)(F)F N1(C(C2(C(=O)NC)CCC2)=O)CC2(CCOCC2)CC1CNC(=O)CC1OCCO1 c1(OC)ccc2cnc(N3CC4(CCC(NCc5cncs5)C4)C3)nc2c1 c1(C(N2CCC(C)(NC(CN(C3CCCC3)C)=O)C2)=O)cncc(O)c1Cl C1(C2CCN(C(=O)CCC3CC3)CC2)(NC(c2cc(C(=O)OCC)n[nH]2)=O)CCC1 Cc1cccc2oc(N3CCCC(NC(c4nc(O)sc4C)=O)C3C)nc12 c1(C(N2C(COC)CCC2)=O)ccc2nccn2c1.c12cccc(c1)NC(=O)N2 c1(C(=O)NC2(CNC(CC3(C)CC3)=O)CC2)cc(C(F)F)ccc1Cl C1(C(=O)NCC(c2ccsc2)C)CCN(C(=O)CC2CCOC2)O1 c1(CC)ccc(C=CC(=O)NC2CC2CNC(=O)Cn2ncc(Cl)c2C)cc1 CC(C)CC(CNC(c1ccc[nH]1)=O)NC(c1ccnn1CCN(C)C)=O C1(CNC(C=CC)=O)CC(C)(C)CCC1NC(c1cncc(NS(C)(=O)=O)c1)=O c1(C(C)C)ccc(C(=O)NCC2CCC(NC(C3(C)CSC3)=O)CC2)cc1 N1(C(C2CC(OCCNC(=O)OC(C)(C)C)C2)=O)CCC(O)C1.C(C(F)(F)F)C1CC1 Cc1sncc1NC(=O)COC(=O)C(C)OC1CC=CC1 CCCCC(F)C(=O)N(CCCNC(=O)C(C)(C)C(F)F)C1CC1 C1(C(C)(C)C)CN(C(C2CC23CC3)=O)CCN1C(=O)Cc1ccnn1C(C)(C)C C1(C2CC2)(CNC(CCC=CC)=O)CCN(C(C2OCCOC23CCC3)=O)C1 C#Cc1cccc(C(=O)NCCNC(C2(F)CS(=O)(=O)CC23COC3)=O)c1C N1(C(C(CC2CCC2)OC)=O)CCN(CC(C)NC(C2(C)CC(C)(C)C2)=O)CC1 N#CC1CCC(C(=O)NCCCCCCNC(=O)C(F)C2CCC2)CC1 c1(CC)cc(C)cc(CC)c1NC(=O)COCC(=O)N(C1CCOC(C(C)C)C1)CCCC c1(OC)ccc(CN2CCC2CNC(c2cccc(Cl)c2OC)=O)cc1F CC1(C)C(O)CC1(CO)NC(=O)NC1(Cc2ccc(Br)cc2Cl)CC1 c1(NCC)cncc(C(=O)N(CCCNC(=O)C=C2CCC(C)C2)CCO)c1 N1(C(c2ccc(C(=O)NC)nc2)=O)CCOC(C)(CNC)C1.C(C)(C)(C)O N1(C(CCC=CC)=O)CCCCC1C(=O)NCC(O)CF C(CNC(c1ccc(Cl)s1)=O)(C(C)C(C)C)NC(c1c(C)cc(C)[nH]1)=O C1(NC(C2(C#C)CCCC2)=O)CC2(C1)CN(C(=O)C=CC(=O)NC1CC1)C2 C1(C(=O)NCC(C)CN(C(=O)C(c2cccc(F)c2)O)C)CN(C)CCO1 C(=O)(CCC(C(=O)NC(C)(CNC(c1cnn(C2CC2)c1)=O)CO)OC)OC N1(C(C(CC=CC)C)=O)CCC(C)C(N(C(=O)CN(C)C(C)=O)C)C1 C(=O)(C(C)CC1CCC1)NCCCOCCC(=O)N(CC)Cc1cccs1 C(=O)(CC(CC(C)C)NC(c1cc2ccccn2c1)=O)N1C(CC=C)CCCC1 N1(C(C(C2CCN(C(c3cncc(CO)c3)=O)CC2)C)=O)CC(F)C(F)C1 C(CC(=O)Nn1cc(-c2nn[nH]n2)c(O)nc1=O)c1nnc(C)s1 N1(C(c2cnc(C)s2)=O)CCCCC1CC(=O)NCC1CC2(CC2)CO1 c1(OC)ccc(Br)c(C(N2CC3CN(C(=O)Cn4cccn4)CC3C2)=O)c1F c1(CC)ccc(C)cc1C(=O)NC1CC1CNC(=O)Cn1cncn1 Cn1c(=O)ccn(CC(=O)NCC2CN(C(=O)CC3(O)CC3)CC2(C)C)c1=O CC1(C)CC(C(=O)NCCOCCNC(c2cn3cnnc3cn2)=O)CNC1=O c1(C(N2CC=CC(NC(C(c3c(OC)cccc3)=O)=O)C2)=O)cc(Cl)ccc1N Cc1ccc(C(N2CC(NC(=O)CC3CCCSC3)CC23CCC3)=O)cc1C#N CC(CC(F)(F)F)OC(CNCC(F)(F)Br)=O C1(NC(C2C(C#C)C2)=O)CC2CN(C(=O)C=Cc3cnc[nH]3)CC2C1 CC(CC1CC1)C(C(=O)NCCC1CC1)N1CCN(S(=O)(=O)C2CC2)CC1 C(C(C)(O)CC(=O)NC1CC(O)C1CC(=O)NCC(n1ccnn1)C)OC C1(NC(=O)CN2CCSCC2)COC2CN(C(=O)CC3CCC(F)(F)C3)CC12 c1(C(=O)NCCCCN(C(C2(C)N(C)CC(OC)C2)=O)C)ccc2cncn2c1 c1(N2CCC(CC=C)(NC(C3C4CC5C(C4)C35)=O)CC2)cc(O)nc(=O)n1C C(=O)(C1CSc2ccccc21)NCC(=O)N(CCCN(C(=O)C(C)(C)C)C)C Cc1cc(OCC(=O)NC2CCC(CNC(=O)C(O)C3CC3)C2)ccc1Cl c1(SC(C)C)cc(O)c(F)c(F)c1.CC(C)C(O)C(=O)N1CCCC(CO)C1 CC(=O)CCCCC(=O)NC1CCCC(C(N2CCOCC3(CC3)C2)=O)C1 Cn1nnnc1C(c1nc[nH]n1)NC(CCC(C1CC1)N)=O.C1(C)CC1 c1(CCCN2CC(CCNC(=O)N(C)C)OCC2)ccc(Cl)c(F)c1 CC1CCCN(CC(C2CC3CC3C2)=O)C1.c1(OC(F)F)ccccc1CC(=O)O C1(N(C(c2nc(OC)oc2)=O)C)CN(C(=O)Cc2ccccc2Cl)CC1O N1(C(C(CSC)(C)C)=O)CC2OCC(NC(C3CC4(CCCO4)C3)=O)C2C1 N1(C(c2c(C)c[nH]c2)=O)CC(NC(=O)CCn2cnc([N+](=O)[O-])c2)CC12CCC2 CCCC(CNC(c1ncccc1CC)=O)C(=O)NC1CC(C(C)O)C1 N1(C(CS(=O)(=O)NC)=O)CCC(NC(c2cnn(CCF)c2)=O)C(F)(F)CC1 C12(C(N(CCCCNC(CC3CCC(C)O3)=O)C)=O)CC3CC1C2C3(F)F C1(C(=O)NC(C2N(C(CCCOCCC)=O)CCC2)C)CS(=O)(=O)CC12CC2 c1(OC)cccc2c(N3CC4CC3CN4Cc3ncc[nH]3)ncnc12 c1(C(C)NC(c2c[nH]nc2C(C)(C)C)=O)ccc2c(c1)CN(C(C1(Cl)CC1)=O)C2 C=CC(CC)CC(=O)NCC(CO)NC(=O)C(C)=CC1CC1 N1(C(C(CCOC)NC(c2cccnc2OC)=O)=O)CCCOCC1C c1(N2CCC(NC(C(C)OCCOC)=O)C2C)cc(=O)n(C)cn1 CC1Cc2cccc(C(=O)NCC3CCCCN3C(c3ncccc3F)=O)c2O1 C1(C(=O)NC2C(CC(=O)Nc3ccc(O)nc3)CCCC2)CCC2(CCC2)C1 n1(C(C)C)ccc(=NC(c2cccc(OC(F)F)c2)c2nnnn2C2(C)CC2)[nH]1 Cc1nc(CC(N2CCC(O)(C(C)CNC(=O)COC3CCCC3)C2)=O)c(C)s1 C=CC1OCCC1C(=O)NC1(CF)CCN(C(=O)CC2(CS(C)(=O)=O)CC2)C1 C1(C(C)C)C(=O)NCCN1C(=O)NC1CCC(c2ccc(Cl)cc2)C1 C1(C(=O)NCC2(C(=O)NC3CCCC(C)CC3)CC(=C)C2)C2CCCCCC12 C(=O)(C(C)(C)CS(N)(=O)=O)N1C(CNC(c2cc(C)cc(Cl)c2)=O)CC1 c1(C(N(C2C3CN(C(C4ON=C(C)C4C)=O)CC32)C)=O)sc2ncccc2c1Cl CC(=O)CCCC(=O)N1CC(CNC(c2cccnn2)=O)C2(CC2)C1 C(=O)(C1SCCc2sccc21)NCc1ccc(CNC(CC(C)C)=O)cc1 c1(C(=O)NCC(CNC(c2ccnc(C3CC3)n2)=O)O)cccc2oc(O)nc12 C=C(C)CCC(=O)NC(CNC(c1ccncc1OCC(F)(F)F)=O)C(C)C c1(C(=O)NCC2(O)CN(C(c3cc(F)cc(Br)c3Cl)=O)C2)ccc2cncn2c1 N1(C(=O)CCCC2CCC2)CCCC(F)(CNC(C2(C3CCCCO3)CC2)=O)C1 C1(CCNC(c2ccc(CC)o2)=O)COCCN1C(=O)C(c1ccccc1)SC C(C(C)C#N)N(C(CN(C(=O)C=CC1CCC1)CCOC)=O)C c1(C(N(CC(CN(C(=O)CC2C(C)(C)C2(C)C)C)O)C)=O)ccc2c[nH]nc2n1 c1(C(N2C(CNC(=O)CSC(C)C)CC(OC)C2)=O)ccc2c(c1)OCCO2 C(=O)(C#CC1CCOCC1)N1CCC(NC(c2nnn(COCC)c2N)=O)C1C c1(C(=O)NC2C3(CC(NC(C4(C)CNC(=O)C4)=O)C3)C2)nc2cccnc2s1 N1(C(C2CC(C)C2)=O)CCC2(CC1)CCN(C(=O)CCC(N)=O)C2 C=C(C)CN=C(NCC1CCCCS1)N1CCC(SC)CC1 C1(C(=O)NC2CCN(C(CCOC)=O)CC2)CCc2n[nH]cc2C1C C(CCSC)(C(=O)NOC(C)(C)C)NC(COCCOC)=O.c1(C)ccccc1 c1(C(=O)NC2C=CC(CNC(c3ccn(C(C)C)n3)=O)C2)coc2c1COC2 C1(CNC(C(C)=C2CCCC2)=O)CN(C(c2cccc(N)n2)=O)CCN1C N1(C(C(C(C)C)c2ccccc2)=O)CC2(CO)CC1(CNC(=O)C(N)=O)C2 c1(C(=O)NCC(C)NC(c2c(O)ncc(SCC)c2)=O)cnn2c(N)ccnc12 N1(C(=O)C2CC2)CCC2CN(C(C3(c4ccsc4)CC3)=O)CC12.C1CCCO1 N1(C(C(CSC)OC)=O)CCC(O)(C(C)NC(c2cc(F)ccc2O)=O)CC1 c1(C(N2CCCC(N(C(C(CC=CC)C)=O)C)C2)=O)cc(CC)ccc1F C=C(Cl)CC(C(=O)NCC1(S(C)=O)CC1)NC(=O)CC1CCCNC1=O C(=O)(CC(C)C(F)(F)F)N1C(CNC(c2c(OC)cccn2)=O)CC(F)(F)C1 N1(C(C(C)OCOC)=O)CCCC1CN(C(C1(C(F)F)CCCO1)=O)C1CC1 CC(CNC(=O)COC(C)(C)CNC(C1(CC2CCC2)CC1)=O)CC(F)(F)F c1(C(=O)NCCCCN(C(=O)CSC2CCOC2)C)cc(OCC(F)F)ccn1 c1(C(=O)NCc2ccc(C3CCCC3)cc2)cccc2c(C(=O)O)nccc12 c1(OC)c(C(=O)NCC2CC(NC(=O)Cc3nnc(C)s3)C2)cnn1C N1(C(c2cc(OC)ncn2)=O)CCCC2CN(C(=O)CC3CC3)CCCC12 N1(C(C2(C#C)CC(=O)C2)=O)CC2(C=C(C(=O)NC3CCCC3(C)CO)CO2)C1 c1(NC2CCN(C(c3ccc(F)cc3)C)C2)nc(=N)[nH]c(=NCC23CC(CO2)C3)[nH]1 C(=O)(CCCC(C)(C)O)OC(C)(C)C.C1(C(C)C)C(=O)C2CCCN(C2)N1C c1(C(=O)NCC(C)N(C(=O)CCc2cn(C)cn2)C)cc(O)nc(Cl)c1 CN1CCOC(CN(C(=O)C(c2ccc(C(C)(C)C)cc2)N)C)C1 C1(NC(C2CC(OC(C)C)C2)=O)CN(C(=O)CC2CCCOCC2)CC1C1CC1 C1(NC(c2cnc(C)n2C)=O)CCN(C(=O)C(=Cc2cccnc2)F)CC1C C=CC(C)CC(=O)N1CC2CC1C2NC(c1cc(CNS(C)(=O)=O)oc1C)=O C(=O)(C1CCCc2nc[nH]c21)NC1CCN(C(c2c(N)nc(Cl)cc2)=O)C12CC2 N1(C(C(CC)NC(c2ccco2)=O)=O)CC2CC(C1)C2NC(c1cnsn1)=O N1(C(C2CCCSC2)C(=O)NC(C)C)CCCCC2(CCC2)C1 N1(C(C(C(C)C)F)=O)CCCC(O)(CNC(C2CCC(C(=O)OC)CC2)=O)CC1 c1(OCC(N2CCC(C)(NC(C(CC=CC)C)=O)C2)=O)c(C)cc(Cl)cc1C Cn1nc(NC(=O)NCC2CCC(C(C)(C)C)CC2)c2c1CCCC2 C#Cc1cnc(C(N2CCC(O)(C(C)NC(C3(C)CCCS3)=O)CC2)=O)c(C)c1 C1(F)(C(N2CCC(OCC=C)C2)=O)CCN(C(c2n[nH]c(O)n2)=O)CC1 c1(OC)cccc(F)c1C(C)NC(=O)C(=O)N(CC(c1ccc(C)cc1)O)C c1(C(=O)NC(CNC(c2[nH]cc(C)c2)=O)C2CC2)ccccc1N1CCCC1=O Cc1coc(C(=O)NC(c2ccccc2)C(=O)NCC(O)CF)c1 C1(C(=O)NC(CNC(COc2c(C)cc(Cl)cc2)=O)C)CC2CCCCN2C1 C1(NC(c2ccc(Cl)o2)=O)CN(C(c2cc(Cl)ccn2)=O)CC12CC2 c1(CC)cc(F)ccc1-n1nc(CCCO)nc1C1CC12CCOCC2 S(=O)(=O)(c1ccc(C#N)c(NCC=CBr)c1)N1Cc2c(nn(C)c2N)C1 n1(CC)nc(C(=O)NC2CCC2CNC(C2COC(=O)N2C)=O)c(Br)n1 c1(C(=O)NC(C(C)NC(c2cc(C(F)F)n(C)n2)=O)C)sc2cccnc2c1Cl C1(CNC(=O)C(O)c2ccco2)CCCC1NC(=O)CCc1cocn1 C1(CCNC(=O)COCCc2ccc(Cl)cc2)CSCCN1C(=O)C(O)CF C#Cc1ccc(C(=O)NCCC(C)N(C)C(c2ccn(CC(C)C)n2)=O)cn1 N1(C(C(C)(C)C)=O)CCCC(C2CCN(C(=O)C3=COCCC3)C2)C1 CC1(c2nn[nH]n2)CCCN(CCS(C)=O)C1 CCC(C)(C(=O)N1CCC(N(C(=O)Cc2cc(-c3ccccc3)on2)C)C1)OC N1(CC=C)CC2CCC(C1)N2c1ccncn1.c12ccccc1C(=O)OC2 N1(C(C2C(CC)C2)=O)CCC(C)N(C(c2ccc(-n3ccnc3)c(F)c2)=O)CC1 C1(NC(C(C)(C)c2ccno2)=O)CN(C(C2CC2c2cccc(O)c2)=O)CC1O C#CC1(C(=O)NC2CC23CCCCCC3)CCN(C(C2CC(O)C(F)C2)=O)CC1 c1(-n2cc(CNc3cc(C)c(I)cn3)nn2)cccc2c1OC(C)(C)CC2=O C(CN=[N+]=[N-])(C(=O)Nc1ccc(O)nc1)NC(C=C1CCC(C)CC1)=O C(c1cncc(C)c1)=CC(=O)N(C1CCN(C(C2CC2(C)C)=O)C1)CCC C=CCC(CC=C)C(=O)NC(C)CCC(=O)N1CC(CC23CC(C2)C3)C1 c1(C(=O)NCC2C(C)CN(C(c3cccc(=O)o3)=O)C2)[nH]nc2c1CCC2(C)C N1(C(C(C)OC(=O)CCc2ncccn2)=O)CC2C(Cn3cnnn3)C2C1 C(=O)(C(=O)CCC(C)C)NCc1c(C(N(CCCCCC=C)C)=O)n[nH]c1 c1(NC(=O)CN2CCN(Cc3ccc(C(=O)OC)o3)CC2)ccc(O)c(OC)c1 c1(CNC(N(C2CCOC2)CCOC)=O)nc2cc(Cl)ccc2o1 c1(OC)ccc(C(C(=O)Oc2ncc(C3(O)COC3)s2)OC)cc1 C1(NC(c2c(OC)nc(Cl)cc2)=O)CN(C(C23C=CC(CC2)C3)=O)CC(F)(F)C1 C(=O)(C(O)C(F)(F)F)N(C(CNC(c1coc(Br)n1)=O)C1CC1)C Cc1ccc(Br)c(NC(C2CN(Cc3ccc(N(C)C)cc3)CCS2)=O)n1 CC1CC(CNC(c2cc(C3CCC3)on2)=O)CN1C(=O)CN1CCSCC1 CS(=O)(=O)CC(=O)N1CCC(C2N(C(c3cncc(Br)c3)=O)CC2(C)C)CC1 C(CCC1CCC1)(C(=O)NCC(CO)OC)NC(C(C1CCC1)OCC)=O C1(C(N(CC(F)F)C)=O)CC(C)N1C(=O)CCC1CCCC1 N1(C(C(C(C)C)C)=O)CCC2(CCC(NC(c3ccsc3Cl)=O)C2)C1 CCC(O)C(C)C(=O)NCC1(NC(C2CN(CC(C)C)C2)=O)CC(F)(F)C1 C1(C)(CC(=O)NCC(C)N(C)C)CC(NC(=O)CN2CCCC2CO)C1 C(=O)(C1(C)OCCc2ccccc21)N1CCCC(NC(CS(CC)(=O)=O)=O)CC1 C(C(=O)NOC1CCC1)(c1ccco1)N(C(c1cc(CCC)[nH]n1)=O)CC c1(C(=O)NC(C)CCCNC(C2(C)C(C)(C)C2(C)C)=O)ncc(Cl)c(N)c1Cl c1(C(C)CC(=O)NC2(CNC(c3cnn(C)c3)=O)CCCC2)ccc(F)c(F)c1 n1(CC(=O)N(CCC)CCNC(c2csnc2C)=O)nc(C)n(C)c1=O C1(C(N2C(CNC(c3c(CC)[nH]cc3)=O)CC(F)C2)=O)Cc2ccccc2C1 C(=O)(CCCC(=O)OC)N1CCC(COCC(=O)NC2CC(OCC)C2)C1 Cn1nc2c(c1CNS(=O)(=O)c1cscc1Br)CCCC2 C1(NC(CCCC(=O)N(C)C)=O)CC2CC1CN(C(=O)C=CC1CCCCC1)C2 C(=O)(CC(C(=O)NC1CC(N(C)C(c2cnc(C)c(C)c2)=O)C1)NC(C)=O)OC C1(NC(C2N(C(c3c(CC)c[nH]c3)=O)CC(O)C2)=O)CCCN(O)C1=O n1(CC)cc(Cl)c(C(=O)NCC(C2CCCCC2)NC(C2CCC(C)(C)C2)=O)n1 Cc1ccc(CC(=O)N(C2(C(N3CCC(F)(C(N)=O)C3)=O)CCC2)C2CC2)cc1 C12(CNC(C3(C(C)(C)C)CCCC3)=O)CC1CN(C(=O)CC1CCCC13CC3)C2 c1(C(N2CC(NC(C3CC(OCC)C3)=O)C(O)C2)=O)cn2c(n1)CC(C)CC2 S(=O)(=O)(c1ccccc1F)NC1(CC2CCCN(C(c3ncon3)=O)C2)CC1 C1(CCCCCNC(C(C)OC2COC2)=O)CCN(C(c2nonc2N)=O)CC1 C=CC(C)(C)C(=O)NCCC(C1CCCN1C(C1COCCN1C(C)=O)=O)(C)C Cc1c(C(=O)NCC2(NC(=O)C(C)O)CCOC2)cnn1-c1ccccc1F Cc1cc(C(=O)NCC2(NC(=O)CC3CCC(C)O3)CCOCC2)n(CCO)n1 N1(CC(=O)N(CCNC(c2c(C)con2)=O)CCOCCO)CC(=O)NC1=O C1(Nc2cc(OC)ncn2)CC(NC(c2cc(SC)c(C)o2)=O)C12CCC2 COn1cnc(C)c1C(N1CCC(NC(c2cc(C)n(CCO)n2)=O)C1)=O O=C(C1=CC(O)C(O)C(O)C1)N1C(C(=O)Nc2cc(F)c(Br)c(F)c2)CSCC1 c1(OC)ccc(Cl)c(CNC(=O)Nc2ccc(Nc3ccccc3C)cc2)c1F C1(CC)CC(C(=O)N(C)CCNC(C23CCCC(C2)OC3)=O)CC(=O)N1 O=C1CCC2CCN(C(=O)CCCc3cccc(-c4nn[nH]n4)c3)C1C2 CCC(CC)CC(F)C(=O)NC1CC2(C1)CC2C(=O)NCCC1CC(C)C1 C1(CNC23CC(NC(c4c(=N)[nH]c(C5CC5)nc4)=O)(C2)C3)CCCCC12CCC2 c1(C(N(CC(C)NC(=O)C(=O)N(C)C)CC)=O)ccc2c(c1)N(C)CC2 c1(C(=O)OCC2(C)CCC(C(=O)OCC)C2)onc2c1CCCC2 c1(OCC)nc(C)ccc1C(N1CC(NC(=O)CCNS(C)(=O)=O)CC(C)C1)=O c1(NC)c(C(=O)NCC2CCN(C(c3cc(O)nc(O)c3)=O)C2)cccc1N Cc1cc(C(=O)NCc2ccc(CN(C(=O)C=CS(C)=O)C)cc2)c(C)nc1C c1(NC(=O)OCC(=O)NCC(=O)OCc2onc(CC)n2)cccc(C)c1 c1(-n2c(CO)nc(C3CCOCC3)n2)ccc(OCc2c(CC)noc2)c(C)c1 c1(C(=O)NCCOCCCN(C(=O)CCn2cnc(=N)[nH]2)C)ns[nH]c1=O Cc1nn(CC(N2CCCC(CO)(NC(=O)CN(C)C)C2)=O)c(C)c1CO c1(C2(C(=O)NCC(CO)NC(C3(C)CCC(=O)N3)=O)CC2)cccc(F)c1F C(=O)(CC(C)(C)N)NCCCCNC(C=CC=CC)=O.C(C)(=O)N CC(C)CC(CCO)NC(C1CN(C(c2cc(N)cc(F)c2)=O)CC1(C)C)=O Cc1c(NC(C2CCN(C(=O)C(C)n3ccnc3)C2)=O)cccc1F N(C(=NCCN1CCOCC1)NC1CCS(=O)(=O)C1)Cc1cn(CCF)nc1 c1(Cn2c(N3C(C(C)C)CN(C)CC3)nnn2)ccc2c(c1)CCCNC2 Cc1[nH]nc(C(=O)NC2CN(C(=O)CC3CCC=CCC3)CCC2F)c1[N+](=O)[O-] CCCCC(CC)CC(=O)NCC(C)(CC)NC(c1[nH]nnc1CC)=O C(CCC(C)C(=O)N1CCN(CCN(C)C(c2cnn(C3CC3)c2)=O)CC1)OC C12(CNC(CCCC(C)=O)=O)CN(C(c3cc(O)cc(O)n3)=O)CC(F)(C1)C2 C#Cc1cccc(C(N2CCCC(C)(CNC(c3ncn(CC)n3)=O)C2)=O)c1Cl C1(NC(CC2COCC(C)O2)=O)CCc2onc(C(=O)NC3CCCCC3)c2C1 Cc1nc(N2CC3C(NC(C4(C)CNC(=O)C4)=O)C3C2)c2cnn(C)c2n1 Cc1cncc(CC(=O)NCc2ccc(C(=O)N(C3CCCC3C)C)nc2)c1 C1(NC(C(C2CCCC2)OC)=O)CN(C(=O)C(C)O)C2CCCC12 C1(C(=O)NCC(C(C)(C)O)F)C2CC(O)C(C2)N1C(c1cc(Cl)ns1)=O c1(C(=O)NCC2CN(C(Cc3c(C)nn(C)c3)=O)C2)cccc2c1CCC(=O)N2 Cc1cc(CC(N2CCCC(N(C(=O)CN3CCC(C)(O)C3)C)C2)=O)cc(F)c1 N1(C(c2cc(CCC)[nH]n2)=O)CC(CNC(C2CCSC2)=O)C(C)C1 CCC(CC(=O)NC1CC2CCC1C(NC(=O)CCC(N)=O)C2)C(C)C N1(C(C2(C)CC(=C)C2)=O)CC2(CC(NC(=O)C=Cc3cnccn3)CO2)C1 N1(C(C(C(C)C)SCC)=O)CCC2(CC2NC(c2ccnc(C)c2)=O)C1 CC1(C(=O)NCC2CCCN(C(=O)CCOC3CCOC3)C2)CCOCC1 Cc1cc(C(N2CC3C(NC(=O)C(C)(C)C(N)=O)C3C2)=O)n2nccc2n1 N1(C(c2ccc(C)s2)=O)CCC2(CCCN(C(=O)CCCCN(C)C)C2)CC1 C(=O)(C(F)(F)C(F)(F)C(F)(F)F)N1CC2CN(C(C3CC(C(=O)O)C3)=O)C2CC1 c1(C(N(C)CCOCCNC(c2cc3ccsc3n2C)=O)=O)cnc2[nH]cncc1-2 C1(NC(c2cscn2)=O)C=CCN(C(=O)CCC(F)F)C1 C(N=c1[nH]cnc2c1COC2)c1c(CNC(C2(O)CC2)=O)cccc1 C1(NC(CCCOCC)=O)CC2CCC1(C(N1CCC(NC(=O)OC)C1)=O)C2 N1(C(c2c(CC)nc[nH]2)=O)CCCC12CCN(C(c1nnn3c1CCC3)=O)C2 CCCCC(=O)NCC1(C(=O)NC2COCC2CC)CC=CC1 c1(C(N(CCN(C(C(C)OCCC=C)=O)C)C)=O)cc(N)c(OC(F)F)cc1F N(C(=NC(F)C1CCCCC1)NC(C)(C)CC)CC(C=C)(C)C C(C)(CN=c1nc2[nH][nH]cc-2c(O)n1)CNC(CCNC(COC)=O)=O Cn1nc(C(F)(F)F)c2cc(C(=O)O)sc12.C12(CCCC1Sc1ccccc1)NC2 N1(Cc2nc(C)oc2)CCCCC1CNC(c1c(Cl)cnn1C)=O c1(C(=O)NC2C(NC(C(C)OC)=O)C2)cccc(C2(F)COC2)c1 c1(NC(N2C(NC(CC(C)c3cnn(C)c3)=O)C=CC2)=O)nc2ccccc2s1 C(N=c1nc2c(c[nH]1)CCCC2)C1CC(NC(CN(C)C)=O)C1(C)C c1(SC)ncc(C(=O)NC(C)CC(C)NC(=O)Cc2c(C)cccc2Cl)c(O)n1 C1(NC(c2c(C)n(CC(C)(C)O)nc2)=O)CCN(C(c2n[nH]cc2Br)=O)C1(C)C N1(C(C=Cc2c(C)n(C)nc2)=O)CCCN(C(c2ns[nH]c2=O)=O)CC1C N1(C(C2C(C)(C)C2)=O)CCCC(N(CCO)C(C2C3CCC2CC3)=O)C1 CN(C)C(=NCC1(c2ccc(Br)cn2)CCC1)NCC1CCC(C(F)(F)F)O1 c1(C(=O)NCC(COC)C2CC2)ccc(C2CCCCC2)cc1C c1(C(N2C(C)(CNC(C3CCCS3)=O)CCC2)=O)cc(O)c2ccoc2c1 C1(C)(CNC(CC2(C(=O)OC)CC2)=O)CC(NC(=O)CCCF)C1 C(=O)(CC(CN(C)C)C(F)(F)F)NCc1scc(CNC(c2[nH]cc(C)c2)=O)n1 n1(CC)nc(C)c(CC(=O)NCC2CC(C)(C)CN2C(=O)C(C)C2CC2)c1C C1(C(=O)NCCN(C(C(CC)F)=O)C)CCc2cnn(CC)c2C1 CCC(CC(=O)N(CCNC(=O)C(=CC1CCCCC1)F)C1CC1)C(C)(C)C c1(C(=O)NCC=CCNC(c2cc(=O)cc(Cl)[nH]2)=O)ccn2ccnc2n1 N1(C(C2(C)CC(=C)C2)=O)CCC(CC)(NC(=O)Cc2c(C)cnn2C)CC1 C1(NC(C2N(C(C(C)C)=O)CCC2)=O)CCN(c2ccc(C(F)(F)F)cc2)CC1 c1(C(=O)NC(CCNC(C2C(C)(CC)C2)=O)(C)C)ccc(C=CC(=O)OC)cc1 CCC(CC)(CN=c1[nH]c2c(c(=NCC3CCC(C)(C)O3)[nH]1)COC2)SC C1(CNC(CCOC(C)=O)=O)(COC)CCN(C(C2CCOC2C)=O)CC1 C(CCC(C)C(=O)N1CC(CCCCNC(=O)CCn2cncn2)C1)OC Cc1nc2ccc(C(=O)NCC3CCCCN3C(c3cnco3)=O)cc2nc1C CCCCCCCCC(=O)N1CC2CCC2(CNC(c2ccccc2OC)=O)C1 C1(OC)CN(C(c2cc(C(F)(F)F)c(Cl)cn2)=O)CC1NC(C1CC(CF)C1)=O Cc1nnsc1C(C)NC(=O)CCCNC(=O)CC1CCOC1C C1(C(N2C(c3cccc(F)c3)COCC2)(CCl)C2CC2)CC2CCC(C1)C2O N1(C(c2cc(C)c(F)c(C)c2)=O)CC2CCN(C(c3cccnc3S)=O)CC2C1 C(=O)(CC(C)(C(F)F)N(C)C)NC1C2CN(C(C3CC(CC)NC(=O)C3)=O)C1C2 C1(CNC(CCS(C)(=O)=O)=O)CN(C(=O)CN2CCCCC2)C2(CCOCC2)C1 Cc1cc(C(F)(F)F)ccc1C(N(C)C(=NCc1cccs1)NCC(C)(C)CO)=O N1(C(C2CC(CC)C2)=O)CCOCC1CC(=O)Nc1sccc1C(=O)OC(C)C C1(NC(c2c(C)cncc2C)=O)CC2CC1CN(C(=O)C(C)C1CCOC1)C2 CC1(C)COCCC1NC(C1CC2(CC2)CN1C(=O)CN1CSCC1=O)=O Cc1cccc(C(C)C(=O)NCC(C)NC(c2cnc(S)n2C)=O)c1 c1(OC)ccc(C(N2CCOC(C(C)NC(C3CC(OC)C3)=O)C2)=O)cc1C C(c1ccc(F)cc1F)=CCN1C(C(=O)NCCc2ncco2)CCCC1 O=C(C1CS(=O)(=O)c2ccccc21)NC1C=CCN(C(c2cn(C3CC3)nn2)=O)C1 N1(C(=O)NCC(c2cccc(Cl)c2)OC)CCC(S(=O)(=O)C(F)F)C1 Cc1c(Cl)c(C(=O)N(CCC(C)NC(c2cc(Cl)c[nH]2)=O)C)nn1C Oc1c(CNCC2CC2C(F)(F)F)cccc1Br c1(OC)cccc2c1OCC(CNC(=O)N(C1CCN(c3cc[nH]n3)C1=O)C)C2 CCC(CC)CCC(=O)NCC1CCCN1C(=O)C(c1cccc(F)c1)F c1(C(N2CC(C)CC(NC(CNC(=O)NC)=O)C2)=O)cc(C)c(O)c(N)c1 c1(C(N(c2nc(SC)nc(C)c2)C2CC3(CNC3)C2)=O)ccc(F)c([N+](=O)[O-])c1 CN1CCOCC1CC(=O)NC1CC(CNC(=O)C(c2ccccc2)N(C)C)C1 CCC(CCC(=O)NCC1(O)CCCC1(C)C)NC(C1CCC(CC)CC1)=O C1(NC(c2cc(C)ncc2)=O)CN(C(c2sc(Cl)c(Cl)c2C)=O)CCC1C Cc1nc(C2CCC2)oc1C(=O)NC(C1CN(C(c2c(Br)nnn2C)=O)C1)C Cc1ccc(C(N2CC(N(C(=O)C(c3cn(C)nc3C)O)C)C(O)C2)=O)c(C)n1 c1(OC)ccc(C(N2CCC(NC(=O)CSS(C)(=O)=O)C2C(C)(C)C)=O)c(F)n1 N1(CC(NOCCC(C)O)=O)CCN(C(C2CCC(=O)CC2)=O)CC1 CC1CN(C(c2cnc(N(C)C)nc2)=O)CCN1C(C1COC2COCC12)=O N1(C(C2(CC(C)C)CC2)=O)CCC(CN(C(=O)CC2CSCCO2)C)CC1 c1(CNC(=O)NCC(=C)C)cn(C)nc1Br C1(NC(C(CCC)N(C)C)=O)CCC2(CC1)CN(C(=O)C=C(C)C)CCO2 c1(CCNC(C(C2CCOC2)NC(CC2N(C(C)=O)CC2)=O)=O)ccccc1C c1(C(C2CC(=C3CCC3)C2)NCc2n(SC)nnn2)ccc2cc(Br)ccc2c1 O=C1CN(C(=O)C(F)CC2CN(C(c3cc(CCO)on3)=O)C2)CC2(CC2)N1 S(=O)(=O)(c1ccccc1[N+](=O)[O-])N(C(c1nc(CC)oc1)=O)Cc1ccccc1F C1(CC)CN(C(=O)CCC2CCCN2C)CCN1C(=O)Cc1sccc1Cl C1(NC(C23CC(C)(C2)OC3(C)C)=O)CN(C(=O)C=CC2CC2)C2(CCCCC2)C1 C1(C=C)CCCN(C(=O)C=CCN(C(=O)CC(C2CC2)C2CC2)C2CC2)C1 C1(NC(C(C)CC#N)=O)CC(C(=O)NCC(C)(C)N2CCCC2)=CC1O C1(O)(CNC(C2CC(C(C)(C)C)OCC2)=O)CCN(C(c2cc(O)no2)=O)CC1 c1(C(=O)NCCCC2(NC(=O)C3=COCCC3)CC2)cnn2cc[nH]c(=O)c12 N1(C=O)CC2(CCN2C(=O)CC2CCOC2)C1.c1(C2CCCCC2)cccc(F)c1 N#Cc1cccc2[nH]c(C(=O)NC3CC3CNC(c3ccsc3Cl)=O)cc12 CC(C)CC(CNC(c1cc(C(C)(C)C)n[nH]1)=O)NC(=O)CSc1nc[nH]n1 c1(SC)ncc(C(N2CC(F)CC2CNC(C2(CO)CC2)=O)=O)n1C C(CCCC(=O)NC(C)C(C)NC(c1cnn(CC(F)F)n1)=O)OCCC=C c1(C(=O)NC2CN(C(c3cnc(N)c(Cl)c3)=O)CC23CC3)ccc2c(c1)COC2 N1(C(c2cn(CCC=C)nn2)=O)CC2CN(C(c3ccsc3Cl)=O)CC2(C)C1 c1(OC)ccnc(C(=O)NCCCC(C)NC(c2cc(C3CC3)ncn2)=O)c1F C#Cc1ccnc(C(=O)NCC2(C)CCCN2C(c2ccc(C)c(NCC)c2)=O)c1 c1(C(=O)Nc2cnn(C3CCCNC3)c2)cc(I)cc(Br)c1Cl CC1Cc2ccccc2N(C(c2cc(F)c(N)c(F)c2F)=O)C1C C1(CNC(=O)Cc2ccc(F)cc2)CCN(C(=O)Cc2cc[nH]n2)CC1 c1(SC(=O)Nc2noc(Cc3cccc(Cl)c3F)n2)sc2ccccc2c1Cl N(C1CCCc2occc21)C(C(CCSC)NC(C1CCN(C)CC1)=O)=O N1(C(CC2(N(C)C)CC2)=O)CC(NC(=O)CC2(C(=O)OCC)COC2)CC(O)C1 N1(C(c2cc(C)oc2)=O)CCCC(N(C)C(c2cc(C3(C)CC3)n[nH]2)=O)C1 c1(CCNC(Cc2nc(NC(c3c(C)ncs3)=O)sc2)=O)ccc(Br)cc1Cl C(CC(C)C(=O)NCC1CCC(C(=O)N(CC)Cc2ccc(F)cc2)C1)=CC N1(C(C(CC=CC)NC(C2CCC(C)(C)OC2)=O)=O)CC2COCC2(C)C1 O=C(C#CC1CCCOC1)NC(CNC(c1cnc(C2CC2)[nH]c1=N)=O)CO C1(CC)CN(C(C2COCCC2(F)F)=O)CCN1C(c1cncc(C(C)C)c1)=O C12(NC(C3C(CC)OCC3)=O)CCC(NC(c3ccc(N)c(F)c3)=O)(CC1)C2 Cc1nc(C)c(-c2nc(CCN(C)C)nn2C(C)C(F)(F)F)nc1C N1(C(CC2CN(C(C3(F)C(C)(C)C3(C)C)=O)CC23CC3)=O)CC2(CCNC2=O)C1 Cc1oc(C)c(C(OCOC)=O)c1C.C1(N)C2CN(C(c3cn(C(C)C)cc3C)=O)CC12 c1(C(CC)CC)nc(Cc2ccc(OC)cc2)n(-c2ccccc2SC)n1 c1(OC)ccc(C(c2nnnn2C2CCCCC2)NCc2occc2Cl)c(F)c1 Cc1cc(C(=O)N=c2cco[nH]2)cc2ccoc12 C1(NC(c2ccsc2)=O)CC2CN(C(C3CCS(=O)(=O)N3)=O)CC2C1 c1(SC)ncc(C(=O)N(C2(NC(=O)Cc3ncn(C)c3C)CCC2)C2CC2)cn1 CC(C(=O)NCC1(CN(C)C)CCC1)N(C(=O)CCn1cccc1)C N1(CCCCC2(C)OCCO2)CC(C2=NOCC2)C1 c1(C(=O)NCCCC2N(C(C(CC=C)C)=O)CCC2)ccc(F)c(F)c1F C1(O)(C(C)NC(c2[nH]c(O)nc2C)=O)CCN(C(=O)COCCF)C1 N1(C(C=CCOC)=O)CCC2CC12C(=O)NCC#CC#CCO c1(C(CC(=O)NC2C(CNC(C3C(OC(C)=O)C3)=O)C2)C)cccc(F)c1 N1(C(C(COC)NC(C)=O)=O)CCCC1(C(=O)NC(C)CC(N)=O)C(C)C C1(CNC(c2c(OC)csc2)=O)CCC(N(C)C(c2scnc2C(C)C)=O)CC1 c1(OC)cc(Cl)c(C(N2CCC(c3cn(CCO)nn3)(N(C)C)C2)=O)cc1Cl c1(Cc2n(CCCCCC)nnn2)ccc2cccc(C)c2n1.C1CCC(C)(C)N1 c1(C(=O)NCCCCNC(c2nc(CC)sc2)=O)cc2n(n1)CCCC2=O C1(NC(C2CCOC2)=O)CCC2CNCC2C1 CCCC(CNC(=O)CCC(=O)N1CCOCC1)C(=O)O.c12cn(nn1)CC2 C1(NC(c2n[nH]c(O)n2)=O)CCC2CN(C(=O)CC3CC3)CCC2C1 C#CC1(NC(=O)C=CCNC(c2ccc(O)nc2C)=O)CCCOC1 C1(O)(C(C)NC(=O)CCc2ccc[nH]2)CCN(C(c2c(N)cccc2Cl)=O)CC1 N1(C(C(c2ccccc2)OC)=O)CC2(C1)CN(c1cc(O)ncn1)C2 c1(C(=O)NC(C2(O)CN(C(C(CC(CC)C)C)=O)C2)C)ccc(F)c2ccsc12 OC1CC2CC1CC2CN1CC2CC1C2.c12cccc(c1)CO2 C1(CC)(NC(=O)CCNS(=O)(=O)CC)CCN(C(=O)CNC(=O)C(F)(F)F)CC1 c1(C(N2CC(O)(CN(C(C3CC(C)(CC)C3)=O)CC)C2)=O)cncc(C(C)C)c1 c1(NC(Cn2cc(COc3c(C)cnc(Cl)c3)nn2)=O)ccc2c(c1)NC(=O)C2 c1(CN(C)Cc2cncc(C(N)=O)c2)cc(C#N)cs1 C1(NC(=O)CCCn2ccnn2)CCCC(c2ccccc2)C1 N(C(=NCCC1CCOC1)NCc1cccc(Br)c1)C(C)C1CC1 C(C(C)(O)C(=O)N(C)CCOCCN(C)C(C1(F)CCOC1)=O)OC c1(OC)ccccc1C(=O)C(=O)NCCC1(CNC(=O)CCc2cncs2)CC1 N12C(C)CN(CC1C)C(=O)C2(C)C.C(C(=O)CCCC(=O)OC)OC(COC)C N1(C(Cc2c(C)occ2)=O)CCC(F)C(NC(c2csc(-c3ccoc3)n2)=O)C1 c1(C(=O)NC(C)CNC(=O)CC2CCNC2=O)cn(C)nc1-c1ccco1 C(C1CN(C(c2sccc2F)=O)Cc2ccccc21)NC(c1[nH]n(C)c(=O)n1)=O c1(C(N2C(CNC(C(ON=C(C)C)C)=O)CC(O)C2)=O)cc2cccn2c(O)n1 c1(NC(C2C3CC2N(C(C2CC4C=CC2C4)=O)C3)=O)ccc(F)c(F)c1F N1(C(c2cccc(-c3c(OCC)c(C)ccc3)n2)=O)CC(O)C(O)C(O)C1CO C1(NC(c2c(C)ncn2O)=O)CC12CCN(C(=O)COCc1cccc(Cl)c1)C2 C(=O)(C(O)CC(C)(C)C)N1C(C(C)C)CCC1C(=O)NCCC1COCC1O C1(C(=O)NC(C(C)C)CNC(C2CCCCS2)=O)CCCC(C)CC1 c1(OC)nc(N(c2cnn(-c3ncccn3)c2)CC2CCNC2)ncc1F NS(=O)(=O)c1ccsc1C(=O)NCC(CO)NC(c1ccccc1CO)=O C1(NC(Cc2ccc(OC)nc2)=O)CC2CC1CN(C(=O)C=CC=C(Cl)Cl)C2 c1(CN2CC(C(C)NC(=O)C=Cc3cccc(O)c3)C2)cc2n(n1)CCCC2O CCC(C(N)=O)NC(C1CCN1C(c1cnn[nH]1)=O)=O C1(C(=O)NC2CC(OC)CN(C(C=CCC)=O)C2)CCn2c(C)nnc2C1 CC(C)C#CC(=O)N1CC2C(CN(C)C(c3csc(Cl)n3)=O)C2C1 c1(C(C)C)ccc(C(=O)N(C)CCOCCNC(=O)CCc2ccoc2)nc1 c1(-c2scc(NC(c3cncnc3)=O)n2)ccc(O)cc1F C12(C(N3C4C(NC(c5cc(F)ccc5O)=O)CC(C4)C3)=O)C3CC(CC13)C2(F)F c1(C(=O)NC(C)CC2CN(C(c3cc(C#N)on3)=O)C2)ccc2ncccc2n1 c1(C(=O)NCC(CC)NC(=O)CCC2CC2(C)C)cc(Cl)c(F)cc1F C(=O)(C1=CCC2CCC1N2C(=O)CCOCC(C)C)NCC(CC=C)(C)CO C1(CC)(CC)CC(NC(=O)CCn2cnnn2)CN1C(=O)C(O)C1CCC1 C12CCN(C1C)C2=O.C1(CC)C(CNC(c2cc(C(C)C)on2)=O)C1(C)C c1(C(N2CCCN(C(C(CSC)C)=O)C(C)C2)=O)cc2nc(C)cc(C)n2n1 c1(C(=O)NCC(CCOC)NC(=O)C(F)Cc2ccccc2)cccc(F)c1 Cc1ccc(O)cc1CN1CCC(C(=O)Nc2ccc(C(N)=O)cc2)C(O)C1 CCCC(C)CCCC(=O)NCC12CCC1CN(C(c1cnc(CC)[nH]1)=O)C2 C(C)(C(=O)N1CCC(NC(c2cc(C(F)(F)F)n[nH]2)=O)C1)(C(C)C)OC c1(C(=O)NCC(CNC(=O)C=CCO)F)ocnc1-c1ccccc1 CCCCCCC(C)C(=O)NCCC(C)N(C(=O)C=Cc1cncc(OC)c1)C C123CC1CCN2C3=O.C(=O)(C(C1CC1)NC(C1(CCl)CC1)=O)OCC.C(C)(C)O C1(CC#C)(C(N2CC(CO)C2(C)C)=O)CCN(C(c2cc(C)oc2CC)=O)C1 N#Cc1ccc(C2CC2C(=O)NC2COCC2NC(C2CC3(CC3)C2)=O)cc1 CON(C(=O)c1ccnc(P(C)(C)=O)c1)C1CCN(c2ccccc2C)C1=O N1(C(c2cc(C)nnc2C)=O)CC2(C=C(C(=O)N3CCCCC3C(C)O)CO2)C1 N1(C(CCC#CC)=O)CC(CO)C2(C1)CN(C(=O)C(C)(O)C(C)C)C2 n1(CC=C)ccnc1C(=O)NCC1C=CCN1C(c1cnc(C2CCCO2)s1)=O N1(C(c2n(C)c(=O)ccc2)=O)CCC=C(C(=O)Nc2cc(C(C)(C)C)no2)C1 C(=O)(C(F)CCC(C)(C)C)N1C(C(=O)NC(CC(C)C)C)CC2(CC2)C1 n1(C(C(N2CCCCC(CO)C2)=O)C2CC2)nc2ccccn2c1=O Cc1ccc(C#N)cc1NC(C1CCCC(NC(=O)C(O)c2ccsc2)CC1)=O N1(C(C2C(CC)C2)=O)CC2(CNC(=O)C(C)C3CCCO3)CC(F)(C1)C2 CC1(C)CCCC(c2cccc(COC(C34CC3CN(S(C)(=O)=O)C4)=O)c2)C1 C1(CC)CCCN(C(=O)CC(C)C(F)F)C1C(N1CCCC(C(C)C)CC1)=O N1(C(c2nncc(C)c2)=O)CC(C)CN(C(=O)Cc2csc(NC=O)n2)CC1C c1(OC)ccc(CC(=O)NCC(O)CNC(c2sccc2C2CC2)=O)cc1 C1(C(N(C)CC2N(C(C3CCC(=C)CC3)=O)CCC2)=O)C2CCC(F)(F)C12 C(N=c1[nH]c2c(c(=NC3CCC3C3CC3)[nH]1)CCC2)c1cc(O)nc(O)n1 c1(OC)ncc(F)c(=NC(=O)C2CC23CN(Cc2cc(C)cc(Cl)c2)C3)[nH]1 CCC(C)(CCNC(C1CCOC(C)C1)=O)NC(c1cn(CCO)nn1)=O N1(C(C(=O)NC(C(=O)OC)C)c2cccs2)CCNC(=O)C1(C)C.C1C(=O)O1 CCCCC(F)C(=O)N(C(C(=O)N(CCCCC)C)C(C)OC)C c1(C(=O)OC)oc(CO)nc1C.C1(C(N2CCCC2CC2CC2)=O)(N)CC1(C)C C1(NC(=O)CC2(NC(C3CCCCO3)=O)CC2)CCCC(F)C1 C(CC(C)N(CC(C)O)C(=O)NCCOCc1cscn1)SC C(N=c1cc(N(C)C)nc[nH]1)C1N(C(C2(C=C)CCOCC2)=O)CCC1 C1(O)(CCNC(Cc2nc(CC)sc2)=O)CCN(C(=O)COC(C)(C)C)CC1 N1(C(C(C)NC(c2ccoc2)=O)=O)CC(NC(C2(C)CC2)=O)C(C)C1 N1(C(C(C)SC(C)C)=O)CC2(C=C(C(=O)Nc3cncc(F)c3)CO2)C1 C1(C(=O)NC2C(CNC(c3cscn3)=O)C2)COCC1C(=O)Nc1ccccc1 CC1(C)CN(C(C2(C#N)CCCO2)=O)CC1C(=O)NCC(C1CC1)C1CC1CC.CO N1(C(C2C(c3cn(C)nc3)OCC2)=O)CCC(C)(NC(C23CC(CO2)C3)=O)CC1 C=CC1(CC(=O)NCC2CC2(F)F)CN(C(C2(C)CC2(F)F)=O)C1 C(=O)(C(F)C(F)(F)F)N(CC)Cc1ccnc(N2CCC(C)C2C)c1 Cc1cc(N2CCC(F)(CO)C2)nc(=NCC2CCC(CO)O2)[nH]1 c1(C(N2CC(F)(CNC(=O)C(O)c3ccco3)C2)=O)ccc(-c2ccco2)nc1 CCC(C)(CCC(C)C)C(=O)NCCNC(=O)C(C1CCCCC1)N(C)C C1(CNC(C(C)CC2CCCC2)=O)C(C)CCCN1C(=O)CCCOC(C)(C)C c1(N2CCC(CC=C)(NC(c3cc(C)n(CC)n3)=O)C2)ncc2ccsc2n1 C(=O)(C(CC(C)C)ONC(c1oc(C)nc1C)=O)N(C(C1CCOC1)C#C)OC c1(OC)ccc(C(=O)NC2CCCC2NC(=O)C(c2ccc(Cl)cc2)C)cc1N C1(NCc2ccc(NC(C(C)C)=O)cc2)C2CC(O)C1N(C(=O)C(C)=CCO)C2 c1(C(C)=O)cc(C(N2CCC(O)(CNC(C3CCOCC3)=O)C2)=O)ccc1C c1(COCC)ccc(CN2CC(NS(=O)(=O)Cc3cccc(Br)c3)C(O)C2)cc1 C1(C(N2CC(N(C(c3ncc(C)cc3C)=O)C)C2)=O)C2CCC3(COC(=O)C13)O2 C(=O)(CC(C(F)F)n1cccn1)NC(CNC(c1n(C(C)C)ccn1)=O)C C1(c2c(NC(=O)NCC(=O)Cc3cnc[nH]3)cccc2)COCCC1(F)F N1(C(C)(C)C)CC2(CCC(CS(=O)(=O)NCCc3nc4ccccc4[nH]3)C2)C1 c1(OC)cc(NC(C2CC2NC(C2CCC(=O)NC2)=O)=O)cc(Br)n1 CC1CN(C(=O)CC2CC(F)(F)C2)CCC1CNC(=O)CSc1nc[nH]n1 C(=O)(C(F)CCC(C)C)N1CC2C(CC(=O)N(CC(CC)C)C)C2C1 C1(CNC(=O)CCC2CCC2)CCN(C(c2cc3cccnn3c2)=O)CC1(F)F c1(C(C)=O)cc(C(=O)NC2(CCNC(=O)Cc3csc(C)c3)CC2)oc1C c1(N2CCCN=C3N=C(NS3)NC2=O)ccc2c(c1)CCC(C)N2.C(C)(C)(C)OC CCC(C(=O)N1CC2C(C(N3CC4(C3)CN(C(C)=O)C4)=O)C2C1)C(F)(F)F N1(C2(C)C(NC(C(C)NC(=O)CN)=O)C2)CCCCC1 C1(OC)CC(NC(C2(N(C)C)CC2)=O)CN(C(=O)C=Cc2ccc(C)s2)C1 C1(CC(=O)NC(C)(C)COC(F)(F)F)CCCN(C(=O)CCCNS(C)(=O)=O)CC1 CCCC(CCC)C(=O)N1C(C(N2CCOCC2COC)=O)CC2CCCC12 C12(C(N(CC(C)NC(c3cc(Cl)cc(F)c3F)=O)C)=O)CC(C)(C1)OC2(C)C N1(C(C2CCN(OC)CC2)=O)CC2CCCC2(NC(=O)COc2ccn(C)n2)C1 c1(C(=O)NC(C)(C)CCNC(=O)COc2ccon2)c(F)ccc(Cl)c1F C1(C(N(CCNC(c2ccn(C(C)(C)C)c2)=O)CC)=O)CC12CC(O)C2 CC1CN(C(c2ccc(Cl)nc2O)=O)CCC1NC(c1c[nH]nc1C(F)F)=O c1(C(=O)NCC(C)N(C(=O)CCC2CCCO2)CC)ccc(OCCF)cc1 C1(OC)C(NC(=O)CN(C(=O)C=CC2CCCC2)CC2CC2)CC12CCC2 S(=O)(=O)(c1ccc(=NCC2CCCO2)[nH]c1)NS(CC1(C)CCCO1)(=O)=O C1(C(=O)NCC2C(C)C2)(NC(=O)CSCCCN2CCC2)CC(O)C1 C(=O)(C(O)CC(C)(C)C)N1CCC(NC(C2(C)CCN(C(C)C)CC2)=O)C1C N1(C(C(=O)Nc2n(C)cc(I)n2)=O)C2CC3CC1CC(C2)O3 C1(C)(CC(=O)NCC)CCN(C(=O)Cn2cc(-c3cc(OC)nn3C)nn2)C1 Cc1c(C(N2CC=CC2CNC(C2CCCOC2)=O)=O)cnn1C1CCOCC1 C1(C)(CNC(COC2(C)CCC2)=O)CCC(NC(c2cc(C3CC3)c[nH]2)=O)C1 C1(C(=O)NC2C(c3onc(C)n3)CC2)CC1C1CN(C(=O)CCc2ccccn2)C1 C1(CNC(c2c(C#C)c[nH]n2)=O)C2CCCC1N(C(=O)Cc1c(Cl)cnn1C)C2 c1(C(=O)NCCCOCCC(=O)NCC=CCC)cccc(OC)c1F c1(NC(=O)Nc2cccc(C3COC3)c2)ncnc2sccc12 Cn1ncc([N+](=O)[O-])c1C(=O)NC1CCC(CNC(=O)C(Cl)=CCl)CC1 CCCC(C)C(=O)NCCC(O)CNC(=O)C=CSC C1(C)(C(N(CC=C)Cc2cn(CC3CCCOC3)nn2)=O)CCS(=O)(=O)C1 c1(CNC(COC(C)=O)=O)ccc(C(C)NC(c2cn[nH]c2)=O)cc1 CCCCC(C)CCC(=O)N1CCCC(C)(CNC(c2ncn(C(C)C)n2)=O)C1 C1(NC(C(C)C)=O)COC2(C1)CN(C(C1(C)CCC(F)(F)C1)=O)C2 O=C(CC(C(F)(F)F)n1cccn1)NCC1(O)CCCN(C(=O)CCC2CC2)C1 N1(C(C(C)N(C)CC)=O)CC(OC)C(NC(c2ccc(-c3scnc3C)cc2)=O)C1 C1(C(=O)NCc2occ(C(=O)NC3(c4nccs4)CC3)n2)CC2(C1)CC21CC1 N1(C(C(C)OC)=O)CCOC2(CCC(NC(=O)Cn3ncc(Br)n3)CC2)C1 c1(CC)cscc1C(=O)NCC=CCC(=O)N1CCC1CO C1(CNC(=O)CC2CCCO2)CC2COCC2N1C(c1cc(Cl)cc(Cl)n1)=O N1(C(c2[nH]cc(C(C)=O)c2)=O)CC(NC(=O)Cn2c(C)c(C)sc2=O)CCC1C C(=O)(CCC(F)(F)F)N(CC(=O)NCCOCC=C)C N1(C(C2CCCC(C)C2)=O)CCC(CNC(=O)CNC=O)C1(C)C C1(NC(C=Cc2ccc(C)o2)=O)CC2CC1CN(C(c1cc(C(C)C)no1)=O)C2 c1(C(N2C(CNC(C(COC)OC)=O)CC2)=O)cccnc1C c1(C(=O)OCC)c[nH]cc1C(=O)N(C)CCNC(C1(c2ccc(C)o2)CC1)=O C(C(=O)NC1(CCC(=O)N2CC(OCCF)C2)CCC1)(N(C)C)C1CC1 N1(C(CCCOCCC)=O)CCCC(C(=O)NCCC(C)C(C)(C)C)C1C C(=O)(C1CCCc2c[nH]nc21)NC1C=CCN(C(c2c(C)cc(=O)oc2C)=O)C1 C1(NC(=O)CCCSCc2ccsc2)CCC(F)(CNC(C2(F)CCCC2)=O)C1 Cc1ccccc1C=CC(=O)NCC12CC(CO1)N(C(=O)C(C)OCC1CC1)C2 C1(N(C)C(C2CCC3(CC2)CC3)=O)CCC(=O)N(C2CC2)C1 CN1CCCC(C)(C)C1N(CCC1CC1)CCO c1(C(=O)NCC(C)N(C(c2n[nH]c(C)c2C)=O)C)cccc([N+](=O)[O-])c1Br c1(N2CCC(CCNC(C3(C)CCOCC3)=O)C2)ncnn2c(Br)ccc12 C1(C(N(C)CC2CCN(C(c3occc3F)=O)C2)=O)CC(C2CC2)=NO1 c1(C(=O)NCCCN(C(=O)CC(C)(C)COC)CC)ccc2nnn(O)c2c1 c1(CNC(c2ccc(OCOC)cc2)=O)cc2cc(C)ccc2[nH]1 N1(C(C(Cc2ccco2)NC(COCCCN(C)C)=O)=O)CCC(NC(N)=O)C1 n1(CC#C)cccc1C(=O)NCCN(C(=O)C(F)C1CCC1)C(C)C CCC(CNC(C1CC2C=CCC(C1)C2)=O)N=c1[nH]c2ccc(O)cc2s1 C1(C(C)C)CN(C(=O)CNC(=O)C2CC2)CCN1C(=O)NC1CC2CC2C1 Cc1cc(Cl)ccc1OCC(=O)NC1CCCC1CNC(c1cnoc1C)=O c1(N2C(C(=O)OC)CCCC2)nnc(-c2[nH]nnc2C(N)=O)n1CC(C)C C(=O)(C(C)CC(C)C(C)=O)NCC(C)NC(CC(C(F)(F)F)n1ccc(C)c1)=O CC1=C(C)CC(C)(NCC2(C#N)CCN(CCO)CC2)CC1 S(=O)(=O)(c1cc(C(F)(F)F)ccc1C)N1C(c2n[nH]c(C)n2)CC(OC)C1 C(C(C)C(=O)N1CC(CCNC(=O)CCc2ncco2)C1)OCC c1(C(=O)O)cc(Cl)nc(SC)n1.C1(C(=O)NCCF)(OCC)CC1 Cc1cc(C(=O)N(C)Cc2cncn2C)ccc1Br N1(C(c2cnc(CC)nc2)=O)CCN(C(=O)C(CO)N(C)C)CC1CCO C1(CNC(c2cccc(OC)n2)=O)CC2(C1)CN(C(C1(C)CC(C)C1)=O)C2 c1(NC(C(CN(C)C)NC(C(CCC)C#N)=O)=O)cncc2ccccc12 C=C(C)CC(C)C(=O)NC(C)CNC(=O)COCC c1(C(N2C(C(CNC(C(C(C)C)CO)=O)(C)C)CCC2)=O)cc2oc(Cl)cc2[nH]1 N1(CC)CCOC(NC(=O)NC(CCSC)C(C)C)C1c1ccccc1 O=C(C1=CCCCCC1)NCCCN(C1CCCC1)C(c1cnc(Cl)s1)=O CC1CN(C(c2ccc(C3(F)COC3)cc2)=O)CC1NC(c1cnsn1)=O.C1CC1 CC(C)CC(O)C(C)C(=O)NCC(C)C(=O)NCC(C)C(C)C CC(C)CC(C)(O)CNC(CCc1ccccc1)C(F)(F)F n1(CC)nc(C(N2CCCC2C(N2CC3C(OC)C3C2)=O)=O)c(=O)c2ccccc12 C(=O)(CS(=O)(=O)CC)N1CCC(N(C(C(C)OCC)=O)C)CC1 N1(C(c2c(COC)n(C)nc2)=O)CCCN(C(=O)CCCc2ccsc2)CC1 c12ccc(c(Cl)c1)S(=O)(=O)N2CC.C1(CCCC)CCC(NCCF)C1 N1(C(C(C)(C)C2CCCO2)=O)CC2OCCN(C(=O)Cc3ccoc3)C2C1 c1(OC(CC)C(=O)N2CC(O)(CNC(=O)CCOCCOC)C2)ccccc1C Cc1ncc(CNC(C)C)c(C)n1.C123C(C(OC)C1C2)n1cc3nn1 CC(C)C(CCc1ccccc1)C(=O)NC(C)CNC(c1ccc(N)c(O)c1)=O N1(C(C2CC(N(C)CC)C2)=O)CCN(C(=O)C(C)(C)F)CC1CC(F)F CC(CNC(=O)CSS(C)(=O)=O)(Cc1ccccc1)NC(=O)CC1CCCOC1 CC1(C)OC2(CNC(=O)CCN3CCC3)CC1(NC(c1cc(F)c(F)cc1Cl)=O)C2 N1(C(C(C)O)=O)CCCC(C)(C)C1CNC(c1n[nH]c(C2CC2)c1Br)=O C=CC1(C(=O)NC2CCOCC2F)CCN(C(=O)C=CCOCCOC)CC1 c1(CC(=O)NC(CN(C(C(C2CCC2)OCC)=O)CC)C)cc(CC)n(C)n1 CC1CN(CC(=O)Nc2csc(-c3occc3Br)n2)CC(C)(F)C1 c1(CC(N2CCCC(C)(CNC(C(CC)SC)=O)C2)=O)csc2cc(C)sc12 C1(F)(NC(c2ccc(OC)cc2C)=O)CS(=O)(=O)CC12CCC2 C12(CNC(C(CC)CC)=O)CCCC1N(C(=O)COCCCF)CCC2 c1(CN(C)C)ccc(C(=O)NC2CCC(C)(CNC(=O)CC(C)(C)C)C2)cc1 c1(OC)c[nH]c(C(=O)NCC2(NC(C3CNC(=O)N3)=O)CCCC2)cc1=O C1(NC(CN2C(C)CCCC2)=O)CCCCCN(C(=O)C(C)C(F)(F)F)C1 C1(CC)CC(C(N2CC(=C(F)CNC(=O)CC3COC(C)(C)C3)C2)=O)CCC1=O O(C=C(C#N)C(=O)N1CCCC1CN(C)C(c1cc(C(C)(C)C)c[nH]1)=O)CC CCCCCCN(C)C(C1CCOC1CNC(=O)CNC(C1CC1C)=O)=O N1(C(C(CCC2CC2)NC(c2c(C)nccc2)=O)=O)CCC(O)C1C N1(C(c2n(CC)ncn2)=O)CC2CCC(C1)N2C(c1cc(C)c(F)cc1Cl)=O C1(NC(c2cc3ccccc3s2)=O)CN(C(C2(F)CCOC2)=O)CC2(CCC2)C1 C1(CN(C(C2C(=C)CC2)=O)C)CCCN1C(c1cc(Cl)c[nH]1)=O c1(-c2nnc(C)o2)cccc(CNC(C2CC(=O)N(c3ccccc3F)C2)=O)c1 C12(NC(CC(=C)Br)=O)CCN(C(c3cnc(C4CC4)nc3)=O)CC1C2 C1(NC(C2(COC)CC2(F)F)=O)CCCN(C(=O)C=Cc2ncc(C)[nH]2)C1 CN1CCC(C(=O)NC(CNC(c2csc(-c3ccccc3)c2)=O)C2CC2)CC1 C12(C(=O)NCc3cc(C)no3)C(NC(C3CC3(C)Br)=O)C3CC1C2C3 Cc1ccc(O)c(CC(N2CCCC2(C)CNC(=O)COc2cc(C)on2)=O)c1 n1(CC(=O)NC2CC(NC(C(C)CF)=O)C2)nc(-c2ccccc2)oc1=O N#Cc1cccc(Br)c1C(=O)NC1CCC(NC(c2cc(F)c(F)cc2Br)=O)C1 C(=O)(CCCCCSC)NCCOCC(=O)OC.c1(O)ccc(C(C)C)cc1 CC(C(C)C)=CC(N1CC(OCC(=O)NCC2CC(O)C2)C1)=O Cc1c(-c2ccccc2F)o[nH]c1=NC(=O)NCC1CCN(C)C1 c1(C(=O)NC2(CNC(COCCC)=O)CC2)c(F)ccc(OCC)c1N.CC CCC(CC(F)F)C(=O)NCCC(C(C)C)NC(C1CNC(=O)CC1(C)C)=O n1(CC=C)cccc1C(=O)NC1CCCC1CNC(c1scnc1C1CC1)=O C(C)(C)(C(C)NC(c1ccnn1CC1CCC1)=O)NC(CN(CCC)C)=O c1(NC(CSCCc2ncc(C)s2)=O)nc(C)c(Sc2cccs2)s1 CC1(c2cn(-c3ccccc3CO)nn2)CCOCC1.c1(C(=O)N)cccc(CO)c1 c1(C(C(=O)NCCC#C)NC(=O)C(C)NC(N)=O)cnn(C)c1 C1(NC(=O)CCC2CC2(F)F)C2CC3C(C2)C13C(=O)NCc1cn(CCO)nn1 Cn1cc(-n2cncc2CN2CC(NC(=O)Nc3ccccc3)C2)cn1 c1(NC(C2CCCC2NCc2c[nH]c(Br)c2)=O)ncc(F)cc1O C1(NC(=O)C=Cc2cscn2)COC2(CCN(C(c3ccccc3CO)=O)C2)C1 C=C(C)CCC(c1nnnn1CC)NCC1CCN(CC(=O)OC(C)(C)C)CC1 C(=O)(C(C)CC(N)=O)NCC1(COC)CN(C(=O)C(C)(F)c2ccccc2)C1 c1(C(=O)NC(CNC(C(C)=C(CC)C)=O)(C)C)cncc2c[nH]nc12 C#CCCC(O)C(=O)N1CCN(C(C2SCCS2)=O)C(C)C1 CC1(C(N2CC3CCC3(NC(c3csc4nnsc34)=O)C2)=O)CCC12CCC2 c1(CNC(=O)CCc2cnc[nH]2)cnn(CCNC(=O)CCC2CCCOC2)c1 N1(C(c2c(SC(c3csc(-c4ccccc4)n3)C)nn[nH]2)=O)CCCCC(C)C1 C1(CNC(c2cnc(C)s2)=O)CC12CCN(C(=O)CCn1cc(Cl)cn1)CC2 c1(-n2cc(CNC3CCN(C(CCC)=O)C3)nn2)ccc(S(=O)(=O)N(C)C)cc1 c1(OCC(=O)NC2CCCCC2NC(=O)CCC2CCC2)cc(F)cc(Cl)c1 C12(CC)CN(C(C3CC3F)=O)C(CNC(c3nn(C)c(C)c3Br)=O)(C1)C2 c1(CS(=O)(=O)NCC2COC3(CCCCC3)O2)ccc2sccc2c1 c1(C(=O)NCC2CC(F)CN2C(C2CCCOCC2)=O)cc2cc(Cl)cnc2o1 C(=O)(CCCC(=O)N(C1CCCCN(C(c2cc(C)oc2C)=O)C1)C)OCC Cc1nc(C(=O)NC2(C)CCN(C(=O)CCN3CCCCCC3)C2)ccc1C#N N1(C(c2cncc(OC)c2C)=O)CCC2CN(C(c3ccncc3O)=O)CC2C1 C(=O)(CC(C)(O)COC)N1CC(CCC)C(NC(C2CC(F)CN2C)=O)C1 N1(C(C(C#C)(C)C)=O)CCN(C)C(CNC(=O)Cc2ccccc2C)C1 CC1(C(=O)NCC(O)(C2CC2)C2CC2)CCc2cc(Br)ccc21 CCCC(C)(CC)NC(c1conc1C1CC1)c1nnnn1CC(F)F C1(C(=O)NCCN2CCC(CO)C2)CCN(CCc2nccs2)C1 c1(CN2CCC(CC(N3CCC(F)(F)C3)=O)C2)ccc(F)c(F)c1Cl N1(C(CNC(=O)OC)=O)CCC2(CCCC2CNC(=O)CNC=O)CC1 C(C(C(=O)NCC(N1CCCCC1)C)C(C)(C)C)NC(C(c1ccc(C)o1)C)=O N1(C(C(=O)NC(=O)NC)C)CC2CN(C(=O)CC3C(C)(C)C3(C)C)CC2C1 CC(C)C(C)(CNC(=O)C(O)Cc1cn(C)cn1)NC(=O)CCCn1ccnn1 C1(CNC(COCCCOC)=O)CCC(NC(=O)COC(F)F)C1 N1(C(c2nnn(C)c2C)C(=O)OCC)Cc2nccn2CC(c2ccccc2)C1 c1(C(=O)NCCC(C)(C)NC(c2cc(CC)nc(O)c2)=O)cnc2ccnn2c1 N1(C(CN(C2CCC2)C(C2N(C)C(=O)OC2)=O)=O)CCC2(C1)CC2(F)F N1(C(c2ccc(CCC)cc2)C(=O)NC2CCCC2)CCOC2(CCCSC2)C1 CC1CN(C(=O)CCNC(=O)C(C)CC#N)CC(C)(C)O1 N1(C(Cc2c(C)noc2Cl)=O)CCN(c2ncnc3c2COC3)CC(O)C1 c1(C(=O)NNC(=O)C(=O)N2CCCC(C(=O)OC(C)(C)C)C2)ccc(Cl)c(Cl)c1O C(=O)(C(C)CC(C)C(C)=O)N1CCC(C(N(CCCC)CC)=O)(CO)C1 Cc1cc(C)c(C(=O)NC(CNC(=O)CCn2ccc(C)n2)CC(C)C)cn1 c1(C(N2CC(CCCCNC(COCC(=O)NC)=O)C2)=O)cc(N)cc(F)c1 C1(NC(C(C)N(C(C)=O)C)=O)C2CC3CN(C(c4cnc(C(C)(C)C)o4)=O)C1C3C2 C(c1ccc(-c2ccccc2)s1)=CC(=O)NCCCNC(C12CCCCC1C2)=O CC(C)C(C)CC(=O)NCC1CN(C(c2ccc(C3COC3)cc2)=O)CC1O C1(CC)Cc2c(Br)cccc2CN1CCC(=O)NCCOC C1(C(N2CCC(NC(c3ccc(Cl)cc3F)=O)(CO)C2)=O)Cc2cccnc2C1 C#CCC(CC(F)F)C(=O)N(CC(O)CN(C(=O)Cn1nnnc1C1CC1)C)C N1(C(C(C)OCCCC)=O)CC(C)(C)OCC1CNC(=O)CC(F)(F)C(F)F N1(C(CC=C(C)C)=O)CCC2(CC1)CC(NC(=O)C1=NOCC1)CO2 c1(C(=O)NCC2N(C(C3(CC#C)CCCC3)=O)CC2)cnc2n1CC(C)CC2 Cc1cccc(-c2nc(C(N3CC(C#N)C3)=O)cs2)c1C N1(C(C(C(C)O)N(C)C)=O)CCOC2(C1)CN(C(C13CCCCC1CCCC3)=O)C2 N1(C(c2nc(C)nc(O)c2)=O)CC2C3CCC(C2C1)N(C(c1occc1C)=O)C3 C(=O)(C(C)CN(C)C)N.C(C)(C(=O)NCC(C)(C)OCCNC(C)=O)SC c1(C(=O)NC(C2CCCCC2)C(=O)NCCC2(O)CCC2)cnc2ccccn12 c1(NC(C2C(C)(CNC(Cc3cn(C)nn3)=O)C2)=O)ccc2c(c1)OCC2 C1(NC(C(C2CCCC2)OCC)=O)CCCC2CN(C(C3COC(C)C3)=O)CC12 CC(C(=O)NC1CCN(C(=O)COC(F)(F)F)CC1F)C(F)(F)F C1(NC(c2n(CCC)nc(C)c2)=O)CN(C(=O)CCS(C)=O)CC2CCCC12 CCC(CC)(CO)C(=O)NC1CC(F)(CNC(=O)Cc2cc(F)ccc2F)C1 c1(-c2c(C(=O)NCc3cc(C)on3)ncs2)ccccc1C C1(C(=O)NCC(c2cnc[nH]2)C)CSCN1C(=O)Cn1cccc1 CCC(C(=O)NC1CC(C)N1C(=O)C(C)(F)c1ccon1)NS(C)(=O)=O c1(CCC)nc(C(=O)NCCCCCC2CC2)co1.C1C(=O)N1C(C)C C1(CC(=O)N(c2ccn(C)n2)CC(=O)NCCC)CCN(C(=O)CC)C1 N1(C(CCc2ccc(C)nc2)=O)C2CCCC1CN(C(=O)C(C)C1CCCC1)C2 CCC(C)(C)CCCC(=O)NCC1CCC(F)(NC(C2CCCO2)=O)C1 C1(O)(CCNC(CNC(C)=O)=O)CCN(C(C2CCCCC2O)=O)C1 C1(NC(CCc2cc(OC)no2)=O)CCCN(C(c2ccncc2)=O)C1C C1(NC(CC2C(C)C2)=O)CCC2CN(CC3CCCOC3)CC2C1 N1(C(C=NOC)=O)CCCC2(CNC(c3cc(F)c(F)cc3F)=O)CCCC12 Cc1[nH]nc2c(C(=O)NC3CCCC3CNC(=O)CCCC(C)(C)C)cccc12 c1(C(=O)NCC(C2CC2)NC(C2C(C)(C)COC2)=O)ccc(O)c(F)c1 C1(CN(C)C(C2CC=CC(NC(=O)C(C3CCOCC3)F)C2)=O)CCC(=O)NC1 Cc1ccc(CSCC(=O)NCC(C)NC(=O)CC23COC(C)(C2)C3)cc1 N1(C(COCc2c(C)ncs2)=O)CC2CC(NC(C34CC3COC4(C)C)=O)C1C2 Cc1cnc(C(N2C3CC2CN(C(c2cnn(CCF)c2)=O)C3)=O)cc1Cl Cc1cc(C(=O)NCCC2CC(C(=O)NC3CC(C)N(C4CC4)C3)C2)cc(Cl)n1 c1(C(=O)NC2CCN(C(=O)Cc3ccc(F)cc3Cl)CC2O)cn2c(n1)COCC2 C(=O)(CCCCC(C)C)N1C2CN(C(CCCCCOCC)=O)CC1C2 c1(NC(N2CCOCC2C2CC(F)(F)C2)=O)cccc(I)n1 CCC(C)(C(N)=O)NC(C1CCCC(NC(=O)CCc2ncccn2)C1)=O C1(OC)CC(NC(c2ccc(C)cc2)=O)CN(C(=O)C(C(C)C2CC2)N(C)C)C1 N1(C(C2(COC)CCCO2)=O)CC2(C1)CN(C(C1(COC)CCOC1)=O)C2 c1(OC)ccc(C=NNc2cccc(C(C)C(=O)OC(C)(C)C)c2)cc1 C1(C)(C(=O)OC)CC(OC)CN1C(c1cc(Cl)c(Cl)[nH]1)=O CCCC(C)CC(=O)N1CC(CC(C)NC(=O)CN2CCCNS2(=O)=O)C1 c1(C(C)(C)CNC(=O)Nc2ccccc2)ccc([N+](=O)[O-])cc1 C(=O)(C(C)(C)C(=O)NC1CCCCC1NC(C1CCCCS1)=O)OCC C1(CCC(=O)Nc2cn(CC(N3CCOCC3)=O)nn2)CCc2ccccc2C1 c1(C(N2C(C)CC(CNC(=O)Cn3cncn3)C2)=O)cc(N)cc(F)c1 CCCCCC(F)C(=O)N1CCC(NC(c2c[nH]nc2CC)=O)C1 c1(C(=O)NCCNC(CN(C)CC)=O)cc2c(nn1)CCCO2 N1(C(C(C)(F)F)=O)CCC(CNC(c2c(F)ccc(F)c2Cl)=O)C12CCC2 c1(CC(=O)NC2CC(F)(CNC(C(CC#C)C)=O)C2)cccc(C)c1C Cn1nc(O)cc1C(N1CCC(Cn2cc(Cc3nn[nH]n3)nn2)CC1)=O c1(C(N2CCC(NC(CCOCC(C)C)=O)C(F)C2)=O)ccc2nc[nH]c2c1 C1(NC(=O)OCc2ccc(F)cc2)CC(F)(F)CC1O C12(CNC(=O)NCCS(=O)(=O)NC)CCCCC1NC(=O)C2 c1(C(N2CC3CC2C3NC(C2(F)CCC2)=O)=O)cnn2c1CCCC2 c1(CC(N2CC(NC(C(C)C3CC3)=O)C2)=O)nn(C)cc1Br n1(CC(=O)NC(CNC(=O)C(=O)NC2CC2)CO)ccc(C2CC2)n1 C1(C(N(CCNC(C2CC2C(F)(F)F)=O)CC)=O)(CC)CCOC1 N1(C(c2c(NC)cnnc2)=O)CCC(C(=O)N(C2CN(C)C2)C)CC1C c1(NC(C2C(C(=O)OC)C2)=O)ccc(OC)c(Cl)c1.C12COC(C1)CN2 Cn1nc(C(N2CCC(CNC(c3ccc(Cl)s3)=O)CC2)=O)c2ccccc12 CN(C)S(=O)(=O)N(C)CC(=O)NC12CC(NC(c3cc(Cl)ccc3O)=O)(C1)C2 c1(C(=O)OC)cnccc1CNC(=O)Nc1ccnn1CC1CCCCC1O c1(C(N(C)CC2N(C(C(C3CC3)OCC)=O)CCCC2)=O)sccc1S(N)(=O)=O C1(CNC(=O)CCC2CCOC2)CC2CC2N1C(C1CC(=O)N(CC2CC2)C1)=O C=C(Cl)C(C)(C)C(=O)NCC1CC2(CC2)CN1C(C1CC(C#N)C1)=O c1(OC)ncccc1CC(=O)NC(C1CCCN1C(c1ccncc1Cl)=O)C N1(C(C(OC)OC)=O)CC2CCCC(NC(C3CCS(=O)(=O)C3)=O)C2C1 C=CC(CCC)CC(=O)NCCOCCCN(C(=O)CC1CC=CC1)C c1(NC(C2(F)CCN(C(C(CCCC)O)=O)C2)=O)cc([N+](=O)[O-])ccc1Br C#CCCN=C(NCC(CC)(CC)N(C)C)NCC12CCC(CC1)CC2 C12(C(N3CC(CC)SCC3)=O)CC(C)(CN1C(=O)CCCC(C)C)C2 N1(C(c2c(C(C)C)cccc2)=O)CCCN(C(c2c[nH]cc2C2CC2)=O)CC1C Cc1conc1C(=O)N(CC(C)O)CCNC(=O)Cn1ccc(CC(C)C)n1 N1(C(CC(C)C)=O)CCC(C2CC(NC(c3n[nH]c4ccc(O)cc34)=O)C2)C1 C(=O)(C(C)(O)CC(F)F)NCC(=O)N1CCC1C.N1(C(=O)NC)CCCC1.CC=O N1(CCC)CC(C(N2CC(NC(c3nocc3C3CC3)=O)C(F)C2)=O)CC1=O N1(C(Cc2c(C)ccs2)=O)CCC(NC(=O)C=CC(=O)N(C)C)C(O)C1 N1(C(C(CC(=C)C)OC)=O)CCN(C(c2c(CC)noc2C)=O)CC(O)C1 C1(CNC(c2c(C(C)C)ocn2)=O)CCCCN(C(=O)C(O)C(F)(F)F)C1 c1(CNC(=O)COc2ccccc2[N+](=O)[O-])cc(C2=CCS(=O)(=O)CC2)cs1 c1(C(=O)NC(CN(C(c2cc3nc(C)sc3[nH]2)=O)C)C)cc(C)cc2c[nH]nc12 N1(C(C(C)OCC#C)=O)CCCC(C(=O)NCC=C)C1 c1(N(C)Cc2cc(C)no2)ncc(N)c2ccccc12 CC1(C)CCN(C(=O)C=CCN2CCCC2)CC1NC(=O)CC1(C)CCC(=O)N1 c1(C(=O)NC(C(=O)OC)Cc2cccnc2F)c(C)cccc1C C1(C(N(CCC(=O)OCC)C)=O)C2CCN(C(=O)C(c3cncn3C)O)CC12 N1(C(C=CC)=O)CCC(CNC(c2ncccc2OC)=O)C(C)C1 c1(NC(N2CC3(C2)CN(C(c2ccc(O)cc2)=O)C3)=O)cc(Br)cc(Cl)c1O C(C(=O)N(CC(=O)NCC1(c2ccoc2)CC1)C)(C(C)C)SC c1(C(N(CCCNC(c2nc(C)n(C)n2)=O)CC)=O)c(C)oc(C)c1Br C1(F)(CNC(C2CCCN(C(C)C)C2)=O)CCCN(C(=O)CC2CC2(C)C)CC1 C(=O)(CCCCCSC)OC.C12(C)CCCN1C(=O)OC2.C(C)(C)(C)O C1(C(=O)NCC2(OC)CCN(C(c3cn[nH]c3)=O)CC2)C2Cc3ccccc3C12 c1(NC)nc(C)c(S(=O)(=O)N2CCOCC(C(=O)NCC3CCCC3(F)F)C2)s1 C1(NC(c2cc(C)ns2)=O)CN(C(c2cc(Cl)cnc2O)=O)CC2(CCC2)C1 C1(O)(CN(C(Cc2c(CC)con2)=O)C)CCN(C(c2ccc(CO)nc2)=O)C1 C(=O)(C1CCCc2n[nH]cc21)NCC(C)NC(=O)C(O)c1ccsc1 C(C(C)(C)C(=O)N1CCCC(OC2CCC2)C1)[SH](n1cc(CCN(C)C)nn1)C C(N=c1[nH]c(N2CCC(CO)(OC)C2)nc2cc[nH]c12)C1C(CC)C1 c1(NC(C2CCN(C(CN(CC)CC)=O)CC2(C)C)=O)ccc2c(c1)OCCC2 c1(OCC)sccc1C(N1CC(OCC(=O)NC(c2ccc(O)s2)=O)C1)=O c1(NCc2c(C(F)(F)F)cccc2)nccc(=NCC2CCCC23CC3)[nH]1 c1(OC)ccc(CN(C=O)Cc2ncn3ccccc23)cc1C#N c1(OC)ccc(I)cc1C(N1CC(NC(c2ccncc2C)=O)C(F)C1)=O c1(-n2cc(CN(C(C)C)Cc3ccccc3)nn2)cnccc1Cl c1(C(=O)NCC=CCNC(C(CC)CC)=O)c[nH]c2nc(Br)ccc12 C(CC(O)CC(=O)N1CCC(OCCNC(=O)CCc2ccccc2F)C1)SC C=C(Cl)CC(C(=O)NCCC(CC)CO)NC(C1CC2(C1)CC21CC1)=O C1(C(N2CC(COC)(CNC(C3C(C)CC3C)=O)C2)=O)CCS(=O)(=O)CC1 CC(CCCc1ccccc1)C(=O)NCCN(CCCN(C)C)C(C1CC1C)=O CCC(C(=O)NC(C)CC1CN(C(C2(CC(C)C)CC2)=O)C1)OC1CCCCC1 c1(C(N(CCCNC(C2(Cl)CC2(C)C)=O)C(C)C)=O)ccc(C(N)=O)cn1 c12ccc(Cl)c(c1)C(=O)N1CC3CC1CN3C2=O.c1(CC)cccc(OC)c1 c1(CC)nc(C(N2CCCC2C(=O)NCC(C)(O)CO)=O)cs1 C1(OC)(CNC(=O)C(N2CCCC2)C2CC2)CN(C(C2(C)CC=CC2)=O)C1 C1(NC(C2CN(C(N)=O)C2)=O)CCOCC1NC(c1cc[nH]c1)=O c1(C(=O)NCC(O)CNC(C2C(F)(F)C23CC3)=O)cc(F)cc2nc[nH]c12 C1(C(=O)NC(Cc2ccc(Br)cc2)C(F)(F)F)C2Cc3c(Cl)cccc3C12 c1(CN(C(C2OCCN(C(C3(CC)CCCO3)=O)C2)=O)C)cccc(F)c1F c1(C(=O)NC(C(C2CCCCC2)NC(c2c(CC)onc2)=O)C)cccc(F)c1 C1(C(=O)NCC(CNC(c2ccc(CC)o2)=O)(C)O)CNC(=O)C(C)(C)C1 N1(C(CCC=C)=O)CCC2CN(C(=O)CCc3nccn3C)CC12 c1(C(N2CCN(C(CC(CCC)C)=O)CC2COC)=O)c(F)ccc(Cl)c1F C(=O)(C(CNC(C1(F)CC1)=O)CC1CCCC1)N(CCCC(O)CO)C c1(OC)cc(C(=O)NC2CCCC(NC(C3(N4CCCC4)CC3)=O)C2)cc(N)c1O C1(CNC(NCOCC(C)(C)CN)=O)(N)CCCSC1.CCO c1(CCC(=O)NC(C2(O)CCC2)C(=O)NC(COC(C)C)C)ccccn1 CN1CCc2cc(C(=O)N(C3CN(C(c4n[nH]c5c4CCCC5)=O)C3)C)sc2C1 N1(C(c2cccc(NC(C)=O)n2)=O)CC(F)(F)CC1C(N1CC(=O)NC(C)C1)=O N#Cc1ccccc1C(N1CCC1CC(N1CCC(O)(CC2CC2)C1)=O)=O C(=O)(C1=NOC(CNC(C2CC3(CCC3)C2)=O)C1)NCc1cnc(C)s1 C1(C(C(=O)NCCOCC)N(c2ccc(Br)cn2)C)CCCC(C)(C)C1 N1(C(C23CCCC2C3)=O)CC2(CCN(NC(c3[nH]cc(CC)c3)=O)CC2)C1 C1(C(=O)NCC(C)CNC(=O)C(c2ccccc2F)(F)F)Cc2nnsc2S1 C(=O)(C(C)(C)OC(C)=O)NC1C(CNC(C2N(C(CCC)=O)CC2)=O)CC1 CC(C)(C)C(O)CSc1nnc(C2CCC2)n1Cc1csc(-c2cccs2)n1 C1(C(=O)NCCCSC)CN(CCNC(c2coc(C(N)=O)c2)=O)CC(C)(C)C1 C1(CNC(C(C(C)C)O)=O)CCC2CN(C(=O)CC3(O)CCCC3)CCC2C1 C(=O)(C(C(C)CC)CCCSC)NCC.N12CC(C)(C1)NC(=O)C2=O.CCCCO C(N=c1cc(C)nc(-c2ccccn2)[nH]1)C1CCN(C(C(CC)C)=O)C1 C1(CC(=O)N(CCOCCCNC(CNC(=O)NCC)=O)C)C=NN(C)C1=O C1(C(N2C(CN(C(=O)Cc3ccc(N)cc3)CC)CCC2)=O)CCCC(C)(C)C1 Cc1c(CC(=O)NCC2COCCN2C(=O)C2=CCCC2)cnn1C Cc1ccc(CNC(C2CCN(C(c3nn(C)cc3Br)=O)CC2O)=O)c(F)c1 N1(C(C(CC)O)=O)C(C(=O)Nc2cnc(Br)cn2)CCC1C C12(CNC(CC(=O)N(C)C)=O)CC(NC(c3cc(F)c[nH]3)=O)(C1)C(C)(C)O2 C(=O)(CC(C)CC(C)C)N.Cc1ccc(F)c(C(=O)Nc2ccc(OCC)c(C)c2)c1 N1(C(c2c(-c3ccc(OC)cc3C(F)(F)F)ncs2)=O)CCc2n[nH]cc2C1 CC(C)(C)C(C#N)C(=O)NC1(CNC(=O)C=Cc2cccc(Cl)c2)CCCCC1 N1(C(c2nc(OCC)sn2)=O)CCCCC1C(C)NC(c1cc(Cl)c(Cl)[nH]1)=O C1(C2(O)CCN(C(C34CCCCC3CCC4)=O)CC2)(NC(C2CC2(Cl)Cl)=O)CC1 c1(OC)cccc(Cl)c1C(=O)NC1CCCC1C(=O)Nc1ccc(C)nc1 C1(N(C(=O)CCSc2ccccn2)C)CCCCN(C(C2CCC2C#N)=O)C1 c1(C(N2CC(NC(COCC)=O)C(OC)C2)=O)c(OC)ccnc1OC c1(C(N2CCN(C(C(CCC)NC(N)=O)=O)C(CC)C2)=O)c(F)cc(N)cc1F c1(Cc2cn(CC(C(C)C)(C)O)nn2)cc(F)cc(Cl)c1 C1(NC(CC(C)(C)O)=O)CN(C(=O)CCC=CBr)C2(CCCOC2)C1 C1(C(N(CC)Cc2cccnc2)=O)CCCCCN1C(C1COC(=O)N1C)=O c1(NC(CCN(C2CC(O)(c3ccncc3)C2)C)=O)cccc(Cl)c1 C1(O)(C(N(CC(=O)OC)C)=O)CCN(C(c2nccc(C)n2)=O)CC1 C(=O)(C(S(C)(=O)=O)C1CC1)NCC(C)(C1CC1)NC(C(C)C1CCC1)=O CCC(CCC(=O)N1CCCC(F)C1)NC(C1CC2(CC2)CO1)=O C1(NC(c2n(C)ncc2Cl)=O)CCC(C)(CNC(C23CC2CCC3(F)F)=O)CC1 N1(C(C(CC(=C)C)NC(c2cnn(CC)c2C)=O)=O)CCN(C)C(=O)C1C N1(C(CC)=O)CC(Nc2nc(OC)cc(OC)n2)C2(CCOCC2)C1 C1(NC(C2CCS(=O)CC2)=O)CCCN(C(C2CC(OC(F)(F)F)C2)=O)CC1 N1(C(C(C)OCCCC)=O)CCC(CO)(NC(c2cc(C(F)F)cs2)=O)C1 CC(C)C(C)(O)C(=O)N(C)CC1CCCN(C(=O)C2=CCCOC2)C1 c1(C(=O)NCC23CC(CNC(CCCC(C)O)=O)(OC2)C3)cnc2ccccn12 CCC(CNC(=O)CC1CCCN1C(=O)C(Cc1ccco1)NC(C)=O)CC c1(OC)cc(-c2ccc(CNC(c3cccc(=O)n3C)=O)nc2)ccc1O c1(-c2c(C(=O)NC3CC(NC(c4cncs4)=O)C3)c[nH]c2)ccccc1F C1(C(=O)NC(C2CCCC2)CNC(CC(C(C)C)C)=O)CC2CS(=O)(=O)CC2C1 C1(CNC(C(CC)(C)OC)=O)CC12CCN(C(C1CCN1C1CCCC1)=O)CC2 c1(SC)cnc(-c2cn(C(=O)NC3CN(C)C(C(F)(F)F)O3)nn2)nc1 c1(C(=O)NCC2C(CNC(C3CCC(C)(F)CC3)=O)C2)noc2ccc(Cl)cc12 C1CCCCC(=O)N1.CC1CCN(c2ncc(-c3ccccc3)cn2)CC1 c1(CC(N2CCC(NC(C=CC=CC)=O)C(CC)C2)=O)nc2c([nH]1)CCCC2 Cc1nsc2ncc(C(=O)N(C3CN(C(=O)C(c4ccnn4C)O)C3)C)cc12 CC1(C)C2CC1CN(C(C1(CCNC(C3CC(C)(O)C3)=O)CC1)=O)C2 c1(SSCC2CC(NC(=O)CCC(=O)N(C)C)C2)c(C(N(C(C)C)C)=O)cccc1F.N c1(C(=O)NCC(C(C)C)NC(=O)Cc2cccc(Cl)c2F)cc(O)cc(O)n1 CCCC(C(O)C(=O)NC1CSC1)NC(=O)CN1CC(C)(OC)C1 c1(C(N2CC(C)OC(CCNC(c3cn[nH]c3)=O)C2)=O)c(Br)ccc(F)c1F Cc1onc(C(=O)NCCCCCNC(c2cnoc2C(C)C)=O)c1Br C(=O)(C1=CC2CCCCC12)N(C1CC(NC(c2ccc([N+](=O)[O-])c(O)c2)=O)C1)C c1(C(N2CCC(CNC(C3C(C(C)O)C3)=O)C(C)C2)=O)ccc(Cl)c2occc12 c1(SCCC(=O)N(CCNC(=O)Cc2ccns2)C2CC2)cccc(O)c1 CON(C(=O)CC1COCCO1)C1CN(C(=O)OC(C)(C)C)C1 O=C(N=c1cc(CCO)[nH][nH]1)c1cc(F)ccc1NC(=O)CSc1ncccn1 Cn1c(C(=O)NC2CCC(CNC(c3ccsc3)=O)C2)cc2cc([N+](=O)[O-])ccc12 C1(C(CNC(c2cc(C)sc2)=O)F)CCN(C(=O)CC(C)O)CC1 N1(C(C=CCC(C)(C)NC(CC2CCC(C)O2)=O)=O)CCNC(=O)CC1 Cc1ccc(C(=O)C(=O)N2CCC2CNC(C2CCC2C)=O)cc1 C1(CNC(C(CC=C)OC)=O)CN(C(=O)Cc2nccn2C)CC1(C)C c1(C(=O)NC2CN(C(C3C(c4cn(C)nc4)CCO3)=O)C2)cnccc1Cl C1(C)(CC)C=C(C(=O)NCC(C)(C2CC2)NC(=O)CN(C)CCO)C1 CCCC(CC)CCC(=O)N1CSCC1C(=O)N(C1CC1)CC Cc1cc(F)c(C(F)(F)F)cc1S(=O)(=O)N1CC(C2OCCO2)CC1(C)C c1(C(=O)NC2C(F)CCN(C(COC(C)C)=O)C2)occ2c1CCOC2 C1(NC(c2sccc2NC(c2ncoc2C)=O)=O)(CC)CCOC1.N(CC)C c1(C(=O)O)ccc(C(=O)NC2CC(n3cc(C4CCOC4)nn3)C2)cc1C1CC1 c1(C(N(CCNC(CCCCSC)=O)C)=O)nc2c(Br)cccn2n1 c1(C(N2CCCC(NC(CC3C(C)(C)C3)=O)C2)=O)cc2c(nn1)CCC2 C(=O)(C1=CCSC1)N1CC(OCC)(CNC(C2CCC(OC)C2)=O)C1 C12(C(=O)NC3(C)CCC3)COCC1CN(Cc1cc(C(C)C)no1)C2 c1(COCC)cncc(NC(C2CC(CF)C2)=O)c1.c12nc(cs1)CNC2=O c1(OC)ccccc1NC(C1(O)CCN(C(=O)COCC(C)C)C1)=O c1(C(=O)NCC2CCN(c3snc(SC)n3)C2)ccnc(C2CCC2)n1 c1(C(=O)NCC(CC(C)C)NC(=O)CCn2cccn2)ncc(C(N)=O)cc1Cl N1(C(CN(CCOC)C(c2ncccc2F)=O)=O)CCN(C)C(C)(C)C1 c1(CC(N2CCCC(CN(CCOC)C)C2)C)cc(C#N)ccn1 c1(C(=O)NC2C(CNC(=O)CSc3ccccc3Cl)C2)c[nH]cc(Cl)c1=O C1(C(=O)NCCCN(C(C(CCOC)C)=O)CCO)CCC(C)(C)CO1 C(CC(C)P(C)(C)=O)NC(C(n1cc(-c2ccc[n+]([O-])c2)nn1)C)=O N1(C(C2(CC=C)CCN(C(c3cc(CC)no3)=O)C2)=O)CCC2(CC(OC)C2)C1 n1(CCC)nccc1C(=O)N(CC(C)NC(C1(CO)CCCO1)=O)C CC1(C(=O)N(CC(=O)Nc2cn(C3CC(O)C3)nn2)CC2CC2)CC2CCC1O2 CN1C(=O)CCCC1C(N1CCOCCC1C(=O)NCC1CCCC12CCC2)=O C=CCC(C)C(=O)N1CC(CC)(NC(=O)CCCn2ccccc2=O)C1 c1(C(N2C3CC(CN(C(C(C)SC(F)(F)F)=O)C3)C2)=O)cn(C)c(=O)n(C)c1=O C(=O)(C1CCCc2ncnn21)N1CCN(C(CSc2n[nH]c(=N)s2)=O)CC1CF n1(CC(=C)C)nnnc1C(C1(CCO)CCOC1)NCC1CCCCC1 C1(C(C)NC(C=CCNC(CC=CC)=O)=O)CCN(C)C1 c1(C(=O)NC(C(C)NC(c2c(CC)sc(=N)[nH]2)=O)C)cn2cccc(F)c2n1 c1(C(C)(C)Nc2c(C)cccc2)cccc(C#N)c1 c1(OC)ccc(S(N)(=O)=O)cc1C(N1CCC(C)C1CNC(=O)CC1(O)CC1)=O C(CO)(C(=O)N1CC2COCC2O1)NC(c1c(OC)cncc1)=O CC1CN(C(C2(O)CCOCC2)=O)CCC1C(=O)N(C)OC1CCCC1 N1(C(C2C(CC)OCC2)=O)CCC(NC(=O)C=CCOC)C(C)(C)C1 C(=O)(C1=CC2(CCOC2)C1)NC1C(F)CCN(C(CCc2scc(C)n2)=O)C1 C(N=c1[nH]c(N2CCc3sc(Br)cc3C2)nc2c1CSC2)C1N(CCC)CCC1 C(=O)(CCCCCNC(N)=O)NCCC1CCN(C(Cc2nc(=N)[nH][nH]2)=O)CC1 c1(OC)ncccc1C(=O)N(CC(C)O)CCNC(=O)CN(C1CCC1)C N1(C(C(CSC)OC)=O)CC2(CCCCN2C(=O)CCc2cc(C)cc(C)c2)C1 C1(CNC(c2ccc(C)c(Cl)c2)=O)CN(C(C2CSCCS2)=O)CC(C)(C)C1 C(=O)(C(C)C(=O)NCCC1CCCN1C(c1ncc(F)cn1)=O)OC Cc1cnn(C(C)C(=O)NC2CCC(NC(C3CC3c3cccnc3)=O)C2)c1 c1(OC)ccc(O)c(C(=O)NCCN2CCN(C(c3ccco3)=O)CC2)c1 C(C(CO)N=c1nc[nH]n2c(Br)ccc12)NC(=O)C=C1CCC1 C(=O)(C(F)CC(CC)CC)N1CC2C(N(CCCC)CCCC)(CCC2)C1 c1(C2(C(=O)NCC(CNC(c3cc(C4CC4)on3)=O)OC)CCC2)ccc(C)cc1 c1(CN(c2ccnc(-c3ccccc3)n2)C)nc(Cl)ccc1Br c1(C(=O)NCC(CNC(C2CCS(=O)(=O)C2)=O)OC)nn(C)c(N)c1C Cc1c2c(-c3cnc(F)c(C(=O)NCC(N4CCCC4)=O)c3)cccc2nn1C c1(C(=O)NCC2CC(NC(C(CC=C)C)=O)C2)cc(O)nc(CC)n1 CCS(=O)(=O)CC(=O)N1CCC(C2CCCN2C(=O)C(C)=C2CCC2)C1 CN1CCCC1C=CC(=O)N(CC(C)(C)NC(C1C=CCCC1)=O)C N1(C(C2CC2C(F)F)=O)CCN(C(c2snc3ccccc23)=O)C2(CCC2)C1 C1(NC(=O)Cn2cccn2)CC12CCN(C(=O)CC1(CO)CCC1)C2 N1(C(CCCC(=O)NCC)=O)CCC(F)(F)C(CNC(C2CCS(=O)(=O)N2)=O)C1 c1(C(=O)NCCC2N(C(C(CC)SC)=O)CCC2)cc(C(N)=O)cc([N+](=O)[O-])c1 c1(OC)ccc(C(=O)NC(C2(O)CN(C(C3CC3C(F)(F)F)=O)C2)(C)C)cc1 Cc1occc1C(=O)NCC1CCN1C(=O)C(F)C1CCC1 C1(NC(COC(CC)CC)=O)CC2CCC1(C(=O)NCCCCCCCO)C2 c1(C(N2C(CNC(c3cccnc3)=O)COCC2)=O)ccc2c(c1)CCCO2 N1(C(C2(C)N(C)CC(OC)C2)=O)CCCc2ncccc21 C1(C)(C(N2CC(NC(c3cc(C)ncn3)=O)C3(C2)CC3)=O)CCCCNC1=O C1(NC(CC=C)=O)CN(C(c2cc(N(C)C)nc(Cl)c2)=O)CCC1O C1(NC(c2c(C)occ2)=O)CCN(C(c2ccc(-n3nnnc3C)cc2)=O)C1C C1(C(N(CCCN(C)C(C2(C)CCCN2C)=O)C)=O)CCCCN1C(N)=O c1(CNC(c2cncc(C#N)c2)c2n(C(C(=O)OC)C)nnn2)c(C)cnn1C C=CCC(CC(=O)N1CCOCC1CCO)NC(=O)Cc1cccc(O)c1 CCC(C)(CO)C(=O)N1CCCC(CCNC(=O)Cc2cnc[nH]2)CC1 C1(CC)CCN(C(=O)Cc2cncn2C)C(C(=O)NC(C)CN=[N+]=[N-])C1 Cc1ccc(C(=O)NOCC2CCNC2)c(Cl)c1O C(CC(=O)NCCCCC1CN(C(=O)C2=CS(=O)CCC2)C1)(C(F)(F)F)OC C(=O)(C(C)=Cn1ccnn1)NCC12CN(C(C(C(C=C)C)C)=O)C(CC1)CC2 c1(Cc2cc(C(=O)NCC3N(OCC)CC3)no2)ncccc1F C(=O)(C(F)CC(C)(C)NC(=O)Cc1c(C)cnn1C)NCC(CCC)C C(CN=C(NCC1(C(=O)OC)CC(C)C1)NCC)N(C(C)(C)C)CC.C1(O)CCC1 CCC(CCOC)C(=O)NC(C)(CO)C(=O)N1CC[Si](C)(C)CC1 C(CC)(CS(=O)(=O)c1ccccc1)OC.c12cc(cnc1O)CN=C1NN=C2S1 C1(C(=O)NCCC(C)NC(=O)C(C)(O)C2CC2)COC(=O)N1C c1(CN(C2CCN(C(c3ccc(C#C)cc3)=O)C2)C)cccc(F)c1C#N N1(C(C2CC(C)OC2)=O)CCC(CC(C)NC(=O)CCCN(C)C)CC1 N1(CC(=O)NCCc2nc(C)sc2C)CCS(=O)(=O)CC1c1cnn(C)c1 c1(NC(c2c(F)cc(-c3n(C)ccc3)cc2F)=O)ccc2c(c1)OC(F)(F)O2 c1(-c2cnc(NC(c3cc(I)ccc3Br)=O)s2)cc(OCCO)cc(C(F)(F)F)c1 CC1CN(C(=O)Cn2cnnn2)CCC1NC(c1cc(Cl)n(C)n1)=O CC1(C)CC(CNC(=O)C(N)=O)CN1C(c1cnn(-c2ccccc2)c1F)=O c1(CN(C)C)cc(C(=O)NC2(C)CC(NC(=O)Cc3ccsn3)C2)n(C)n1 c1(C(=O)NC2C(CNC(c3ccccc3)=O)CCCC2)[nH]nc2ncnc(O)c12 c1(C(=O)NC(C)(CNC(=O)COCC(F)F)C2CC2)ccc(-c2ccncc2)s1 C1(C(=O)NC(C(=O)NCCN(C(CC)C)C)C2(C)CC2)CC12CCOCC2 c1(-c2cn(COC)nc2)cc(C(=O)Nc2cnc(C)c(C)c2)c(F)cc1C c1(OC)cnc(NC(C2CCCN(Cc3ccc(O)cc3)C2)=O)nc1 Cc1cc(C(=O)NCC2CCCCN(C(C3CCOC(C)(C)C3)=O)C2)c(C)cn1 c1(C(N2CC3C(NC(c4c(C)nsc4C)=O)C(C3)C2)=O)c(C)oc2ccccc12 C(=O)(NN=c1[nH][nH]c(=NC2COCC2OC)s1)Cc1c(NCC)cccc1 C#CC1(O)CCCN(C(=O)CC2CCN2C(=O)CN(C)C(=O)OC)C1 CCCC(C(=O)OC)C(=O)N1CC(OC)CC1CNC(=O)COc1ccccn1 c1(OCC)ccc2cc(CN(C(C3CCSC(C)C3)=O)C3CC3)[nH]c2c1 c1(NC)c(C(N2CCCC(C3CC(NC(=O)C=CI)CCO3)C2)=O)cccc1N c1(C(=O)NCC2CC(NC(C3(OC)CC(C(F)F)C3)=O)C2)ncc(C)cn1 c1(C(=O)NCC2(C)CCN(C(CC3OCC(C)(C)C3)=O)C2)cnc2ccccn12 C1(CCN2CC(O)CC(OC)C2)Sc2ccccc2NC1=O N1(C(c2n(C=C)ncc2)=O)CCN(C(=O)C2=C(Cl)CCOC2)CC2(C)CCCC12 c1(OC)ccc(OCC(C)=CC(=O)NCC(C2CCC2)SS)cc1.C(C(N)=O)CN C(C(C)CC(=O)N(C)CCC1CCOCC1)NC(c1ccn(COC)n1)=O c1(-n2c(C)ncc2)ccnc(CC(=O)NCC2(CNC(c3cnsn3)=O)CC2)c1 C1(NC(c2cccc(N(C)C)c2)=O)CN(C(=O)CO)CCC1O Cc1nc(C2CC2)sc1C(C(=O)NC(C)CC#N)N(C1CC1)C1CC1 C(N=c1nc(O)c2ccccc2[nH]1)C12CCC(CNC(CCC)=O)(CC1)OC2 CS(=O)CCC(O)C(=O)NCCOCCNC(=O)C=Cc1cncc(F)c1 C1(CC(C)C)(C(=O)NCC2CN(C(=O)C(C)CF)C2)CCCC1 c1(C(=O)NC2C3(CCN(C(C4N(C)C(=O)CCC4)=O)C3)C2)ccc([N+](=O)[O-])cc1 FC1CCCCCC1N=c1nc(N2CCOC3(CCCC3)C2)c2c([nH]1)CCC2 N1(C(C2(C#C)CCC2)=O)CCC(N(C)C(C2CN(CC(F)(F)F)C2)=O)C(C)C1 C1(CCC(=O)NCC2C(NC(c3n(C)ncc3)=O)CCC2)CCCC(O)C1 C=CCC(C(=O)N(C)CC1CCN(C(c2c(N(C)C)c[nH]c2C)=O)C1)NC(C)=O N1(C(c2c(C)nn(C3CC3)c2)=O)CCCC(NC(=O)CC2CCOCC2)C(F)C1 CC1COc2c(C(N3CCC(C(C)NC(c4ccccc4Cl)=O)C3)=O)cccc21 C1(COC)CCN(C(C2(NC(=O)C(C)CC3CCCC3)CC(O)C2)=O)C1 Cc1ccc2c(c1)CCC(C(=O)NC1CCN(c3ncccn3)C13CCCC3)O2 C1(C(=O)NCC)CCCC(C(=O)NCC(C2CC2)NC(=O)CC(=O)NC2CC2)C1.OC c1(OC)nc(Cl)ccc1C(=O)NC1CC(CNC(=O)Cc2ccccc2)C1(C)C C1(=CCNC(Cn2ccc(C)n2)=O)CCN(C(C2(C#N)CC2C)=O)CC1 N1(C(c2nc(CNC(c3ncn(CC)n3)=O)oc2C)=O)CCOC(C)(C(C)C)C1 CC(C)CC(C(=O)N(C1CCCCCC1)C)ONC(=O)CC1CC=CC1 CC1(C)CC(CC(=O)Nc2cccc(CNC(c3ccsc3)=O)c2)CCO1 C1(CNC(C=C(C)Cl)=O)C2CC1N(C(c1cccnn1)=O)C2 c1(N(CC(COC)SC(C)=N)C)ccc(Cl)cc1 c1(C(N2CCC(CC=C)(NC(=O)C(C)C(C)C)C2)=O)cc(C#N)c(F)cc1F C12CN(C(=O)C3CC3)CC1NC2=O.c1(C2(SC)CNC2)ccc(OCF)cc1 CC1(F)CC2(CN(c3cc(NC(c4ccncc4)C)ncn3)C2)C1 C(CC(=O)N1C2CCC1CN(C(C1COC(=O)C1)=O)C2)(C(F)(F)F)OC C1(CNC(COCP(C)(C)=O)=O)CC12CCN(C(C1CCNC1=O)=O)CC2 c1(OC)c(C(=O)NCC2CCN2C(c2cc(C(C)(C)C)n(C)n2)=O)cccc1Cl CC1=C(C(=O)NCc2cc(C(=O)NCC(c3ccccn3)O)on2)SCCO1 c1(COc2c(OC)ccc(CO)c2)nc(=NC(=O)C2=COCCO2)[nH]n1C c1(OC)c(Cl)ccc(C(C)NCC2CCCN(CC(N)=O)C2)c1F c1(C(=O)NCC2CC2NC(=O)C(O)CCc2ccccc2)cc(O)nc(O)c1 C1(C)(C(=O)NC2C(CNC(Cc3cc(C)sc3)=O)CC2)CCC(=O)C1 c1(C(N2C(CCC)CCCC2)=O)sc2ccccc2c1Cl C#CCCCCCC(=O)NC(CC#C)C(=O)NC1CCCCC1CO c1(C(=O)NC2CC(NC(C3CCC3(F)F)=O)C2)cnc(CC2CC2)nc1O c1(C(N2C3CCC(NC(c4c(C)nsc4)=O)C(C3)C2)=O)cccc(P(C)(C)=O)c1 c1(C(=O)NCC2(CN(C(=O)CC3(C)CC3)C)CC2)cc[nH]c2nccc1-2 CC(CC(=O)c1ccc(F)cc1)C(=O)NC(Cc1ccccc1)CO CN1CCC(C#N)(C(=O)NC2CCCCC2CNC(=O)C2=C(Cl)CC2)CC1 c1(C(N2CCC(CNC(c3cnn(C4CC4)c3)=O)C2)=O)cccc(F)c1C(F)F N#Cc1cnc(C(=O)NC2(CNC(c3cc(C(F)(F)F)cs3)=O)CCC2)c(Cl)c1 N1(C2CCN(C(C3CN(C)C3)=O)C2)CCC(NC(=O)Cc2nccn2C)CC1 C=CCCC(C)(C)C(=O)N1CCC(CC(C)NC(=O)C#CC(C)(C)O)CC1 N1(C(C2CCN(C(=O)C(O)O)CC2O)=O)CCc2ccncc21 C1(C(N(C(C)CNC(c2cnc(C3CC3)[nH]2)=O)C)=O)CCCC2C1C2(F)F CCC(CC(=O)N(C(C)C(N1CCN(CC(C)C)CC1)=O)C)C1CCC1 C(=O)(C1=C(Cl)CCOC1)NC(CCN(C(C1C(C(C)C)CCC1)=O)C)(C)C CC1=C(C(=O)NC2(CO)CN(C(=O)C(C)(O)C(C)C)C2)CCC(C)(C)C1 Cc1c(C(N2CC3CC(NC(=O)CCC4CC4C)C(C3)C2)=O)sc2ccccc12 C(c1cnn(C)c1C)=CC(=O)N(CCOCCNC(C(n1ccc(C)n1)C)=O)C N1(C(CN(C(=O)C(F)(F)CN(C)C)C2CC2)=O)CC2(CN3C(=O)COCC3)CC1CO2 C(CCC(C)N=c1[nH]c(N2CCC(c3n[nH]c(C)n3)C2)nc(=N)[nH]1)OCCCC C(=O)(C(C)(C)CCF)NCC(C)CC(N1CC2CC2C2CC12)=O S(=O)(=O)(c1cccc(N2C3CCC2CC3)n1)N(C)Cc1nc(CC)sc1 C1(C)(CN(CCCNC(=O)C(F)(F)F)C)Cc2ccccc2C1 N1(C(c2c(CC)n(C)nc2)=O)CCC2(CC2NC(=O)CCc2cncnc2O)C1 C(=O)(C(C)CCC(C)(C)C)N1CC(C)C(CCNC(=O)CC2=NNC(=O)C2)C1 C1(NC(c2cc(C)oc2C)=O)COCCN(C(c2ccc(F)cc2Cl)=O)C1 c1(C(C)OC(CNC2(Cl)CC2(C)C)CO)nc2ccccc2s1 n1(CCN(C)C)cc(C(=O)NC2(CCNC(C3CC(C(F)F)C3)=O)CC2)nn1 N1(C(=O)C2=COCCO2)CC23CCCC2(C1)CN(C(=O)Cc1ccnc(O)c1)C3 CC1(C(=O)Cc2ccccc2)CCCN(OC(=O)CCC2CCCC2C(=O)O)C1 CCCCC(O)C(=O)NC1(CC)CCCN(C(c2scc(C)c2Br)=O)C1 CCCCC(CC(=O)NOCC(C)(C)CC)NC(C1CC2C=CC1O2)=O C(=O)(C(CN(C)C)NC(=O)CC(C)OC)N(CC(COC)O)C C1(CNC(C=CCC)=O)COCCN(C(=O)C(C)C(=O)OC(C)(C)C)C1 C(=O)(CCCC(C)(C)C)N1C(C(=O)NCCOCCOC)C=CCC1 C1(N(C)C)CC2CC1N(C(C1(N(C(=O)OC(C)(C)C)CC3CC3)CCC1)=O)C2 c1(C(=O)NC2C(C(N3CCC(=C)CC3)=O)COCC2)cc(F)ccc1C C#Cc1cncc(C(=O)NC2(C(=O)NOCCC=CCC)CC2)c1 S(=O)(=O)(c1cccc(F)c1C)N1CC2CCN(Cc3nc(OC)c(C)nc3)C2C1 c1(CCNC(=O)COCc2ccco2)ccncc1.C1(O)CCC1.C1CCNC1=O N#Cc1ccc(C(=O)NCC2CC(NC(C3CC4CCC4C3)=O)C(O)C2)cc1 C(=O)(CC1=CCOCC1)NC1CC(NC(CCc2cnn(C)n2)=O)C12CCC2 C1(CNC(C(COC)C)=O)CCC(F)(CNC(c2cc(Cl)c[nH]2)=O)CC1 c1(C(=O)NCC2CCC(NC(Cc3c(C)cnn3C)=O)C2)ccn(C)c(=O)c1 C1(CC(=O)NCC(C(=O)OC)O)N(C(=O)C(C)N(C)C)CCC1(C)C C1(C(=O)NCC)(CCCCC)CCC1.C(=O)(C(F)=CC1CC1)O.C1(=O)COCCN1 c1(Cn2c(-c3cn(CC(F)F)nn3)ccn2)ccccc1CC1CCCO1 N1(C(c2c(C)cc(C)n2C)=O)CCC2(CC1)CC2c1cn(CC2C3CCCC23)nn1 c1(OCC(=O)N(C2CCN(C(COCCOCC#C)=O)C2)C)c(C)cccc1C C1(NC(C(c2cn(C)nc2)=O)=O)CN(C(=O)C(N2CCCC2)C2CC2)CC1F c1(CC(=O)N(CCCN(C)C(c2cccc(F)c2)=O)C)c[nH]c2ccncc12 Cn1ccc(C(N2CC3CC3(NC(c3ccc(N(C)C)cn3)=O)C2)=O)cc1=O c1(C(C)C(=O)NCC2CC(NC(C3CCO3)=O)C2)cccc([N+](=O)[O-])c1 N1(C(c2sc(C)c(C3CCOCC3)n2)=O)CCC(C)(C(C)C)CC1 CC(C)(O)CC(=O)NC1CCOC(CNC(c2cn(CC(F)(F)F)cn2)=O)C1 C#CCC(CCOC)NC(C1CCCC1NC(=O)CC(C)N(C)C)=O c1(C(=O)NCc2cccc(CNC(=O)C(Cl)=CCl)c2)ccc2ccoc2c1 Cc1ccc(C(CNC(=O)Cc2cc(C)on2)NC(=O)Cc2ccns2)cc1 CC(C)C(C(C)NC(C1CCC(F)(F)C1)=O)NC(=O)Cc1nc(C2CC2)nn1C CC(CS(C)(=O)=O)C(=O)NC1COCCN(C(=O)C(C)C2CCCO2)C1 C1(CNC(C2(OC)CCOCC2)=O)CC2CCCC2N1C(=O)C(C)C1CC1 N1(C(CCC(C)SC)=O)CCC(CNC(C2CC2(C)Br)=O)C12CC2 C1(NC(CNC(N)=O)=O)CCC2CCN(C(=O)Cc3ccccc3F)C12 N1(C(c2cnc(C)o2)=O)CC(NC(=O)CN2CC(C)C2)CCC1C C1(C(N(C2CCN(C(C=CCOC)=O)CC2)C)=O)CC(COC)C12CCC2 N1(CC)CCN(C(C2CN(C(C3CC3CCOC)=O)CC(C)O2)=O)CC1C Cn1cc([N+](=O)[O-])c(C(=O)NCCNCCOC2(C#N)CC2)n1.C1C(=O)O1 N1(C(Cc2cn(CC)nn2)=O)CCC(C)C1CNC(c1ccc(C)n1C)=O C1(NC(C=C(C)C)=O)CN(C(=O)Cc2cc(F)ccc2Cl)CCC1C(F)(F)F C1(N(C(CN2CCC(N(C)C)CC2)=O)C2CCC2)CCC(=O)N2CCOCC12 c1(CC(C(N2CCN(CCCN)CC2)=O)N(C)C)ccccc1Br CC1CCN(C(=O)C(CCN(C)C)NC(c2cc(=N)[nH][nH]2)=O)CC(C)O1 CC1OCCOC1C(N1CCOC(CCNC(=O)CCCCC2CC2)C1)=O c1(CC)ccsc1C(=O)NCc1ncoc1CCNC(c1ccc(C(C)C)s1)=O N1(C(=O)OC(C)(C)C)CCC(C(=O)NCC2CC2F)C1C1CCCC1 C(N=c1cc(C)nc(N2CC3C(CO)C3C2)[nH]1)c1c(CC)cccn1 Cc1cc(CCC(N2CCOCC2CCNC(=O)CCC(C)N(C)C)=O)nn1C c1(C(=O)NCC(CCCC)NC(C2CC(C)(C)C2)=O)cccn(C)c1=O CCC(C)C(O)C(=O)NCC1(OC)CN(C(=O)CC2CCC(C)(C)CC2)C1 C=C1CC2(C1)CN(C(C1CCCC(NC(c3ncccc3F)=O)CC1)=O)C2 N1(C(C2C(CNC(=O)Nc3ccccn3)CCC2)=O)CCCc2ccccc21 c1(C(=O)NC2C3CN(C(C(C4CCC(C)CC4)CC)=O)C2C3)nc2ccccc2s1 N1(C(C(CSC)(C)C)=O)CCN(C(c2ccc(CCNC(C)=O)[nH]2)=O)C(CF)C1 CC(C)C(C)C(Cc1ccccc1)NC(c1cc(Cl)c[nH]1)=O C1(NC(C=CC=CC)=O)CS(=O)(=O)C12CCN(C(=O)C(C)CCC)CC2 c1(NC(c2ccc(CC)cc2)c2nnnn2-c2ccccc2)sc(C)c(C)c1Br C(=O)(CCC(C)(C)C#N)N1C(C(N2CCC(OC(C)=O)C2)=O)CSC1 C(CCN=C(NCC(C)(C)C(C)(F)F)NC1CCCN(c2ccccc2)C1)OC N1(C(C2(OC)CC(CF)C2)=O)CCC(C(F)CNC(C23CC(C)(C2)C3)=O)CC1 CC1CC(NC(=O)NCc2ccc(F)cc2)CN1N1CCCC(C(N)=O)C1 N1(c2c(C)c(NC(C)Cc3cnc[nH]3)ncn2)CCC(C2CCCOC2)CC1 c1(C(N(C)CC2OCCN(C(CCC(=O)NC)=O)C2)=O)cc(C)n(C)c(=O)c1 C1(NC(CCNC(C)=O)=O)CC2CC1CC2C(=O)NCCCCn1ccnc1 N1(C(C2CCC3(CC3)N2C(c2ccc(F)cc2Cl)=O)=O)CCC2(C1)CC2(F)F CCC(CC)(CO)C(=O)NC(C)C(C)NC(c1cc(C2CC2)n(C)n1)=O C12(C(=O)NCCCCCC)C3C4C1C1C2C3C41C(=O)N=c1ccn(C)[nH]1 N1(C(N2CC(F)(F)C2)=O)CCCC1(c1ccccc1)CCn1ccnc1 C1(CC(N2CCC(N(C(C3CC3F)=O)CC)CC2)=O)CCC2(CCOCC2)CO1 c1(C(=O)NCC2CC(NC(CCOCCCOC)=O)C2(C)C)ncc(F)cc1F c1(CC)nc(C)c(C(=O)N(C2C3CN(C(C4OCCC4(C)C)=O)CC23)C)o1 N1(C(c2ccno2)=O)CCC2(CC1)CCN(C(c1n[nH]c3c1CCCC3)=O)CC2 C1(CNC(c2ccc(CC)s2)=O)CCC(C)N(C(C2CCC2)=O)C1 c1(CNC(=O)NC2CCC(CCCCC)O2)nc(C)c(C)s1 C(CC(C(=O)NN(C)C)OC)OC.N12CCC(C)(C1)Cc1cn(nn1)CC2=O C(c1ccccc1)=C(CC)C(=O)NCC1CCC1NC(=O)CCC1CCCO1 c1(C=O)ncc(F)c(OC)n1.CCC(C=O)OC.C12(O)CN(C1)N1CC(C1)OC2 Cc1ccccc1C(C)CC(=O)NCC(C)NC(=O)Cn1nnnc1C c1(C(=O)NC(C2(O)CN(C(=O)C=Cc3cscn3)C2)C)ccc2nnn(C)c2c1 c1(C(N(CCN(C(C(CC=C)(C)C)=O)C)C)=O)c[nH]c2ncnc(O)c12 N1(C(C(C(C=C)C)C)=O)CCC(O)(C2(NC(=O)Cn3ncn(C)c3=O)CC2)CC1 c1(C(=O)NCC2CN(C(C3COCC(C)(C)O3)=O)C2)cc2c(cc1N)OCCO2 C(=O)(CCCC(F)(F)CO)N1CC(NC(=O)COc2cccc(F)c2)C(CO)C1 N1(C(CN(C)C(=O)C2CC2)=O)CCC(C2(NC(C3CCS3(=O)=O)=O)CC2)CC1 C1(NC(CC2C(C)C2)=O)CN(C(=O)CN2CCC(N(C)C)CC2)CC1(C)C Cn1nc(C(=O)NC2CCC(CNC(C3CC(C)(C)C3)=O)CC2)cc1O CN1CCC(C(=O)NCC2(C)CCN(C(C3(C)CCCO3)=O)CC2)S1(=O)=O C1(CNC(=O)Cc2cnco2)CCCCC1NC(=O)COC1CC(F)(F)C1 c1(C(=O)NCC(F)CNC(C23CC=CCN2CCC3)=O)cnc2[nH]ccc2n1 C1(CC(=O)NC2(CC)CCCC2)OCCC1(C)C.C12(CC1)C(=O)NC2 Cn1ncc2c1CC(C(=O)OCc1ccc(F)c(F)c1F)CC2 C1(N(CC(C)C)C(=O)CC2CCC(=O)N2)CCN(C(C2CC2(F)F)=O)CC1 C(CCNC(c1cccc(OC2CCCC2)c1)=O)(C(C)C)NC(CSCC)=O c1(C(=O)NC2CC(CC(=O)NCc3c(CC)n[nH]c3)C2(C)C)cc2occc2[nH]1 C1(N(C(C2CC(CC)C2)=O)CCF)CCCN(C(c2cccnc2C)=O)C1 c1(C(N2CCC(C)N(C(=O)CC3C=CCC3)CC2)=O)cc2ccccc2c(O)n1 C1(CCNC(=O)CCOC2CCOC2)CCN(C(C2(n3cnnn3)CC2)=O)C1 C(C)(C)(CCC(=O)N(C1CCN(C(=O)CC2CCCN(C)C2)C1)CCO)OC c1(C(=O)NC(c2c(C)c(F)ccc2)C)ccc2nc(C3=CCCC3)cn2c1 c1(CC)cc(C(=O)NCC(O)CN(C)C(c2cn(C)nc2C)=O)cc(N)c1 C1(C(=O)NCC#CCNC(Cc2n(C)ccc2)=O)CN2CCN1CC2 C1(CCNC(C2(COCC)CCCO2)=O)CCCCN1C(c1[nH]c(O)nc1C)=O c1(C(N2CC3C(C(=O)NC4(CCO)CCOC4)(CC3)C2)=O)cccc2c1CCC2 Cc1ccc(CC(C)C(=O)NCC2CCN2C(=O)CCC2CCC2)cc1 N1(CCN=C(NCCOCC=C)NC2CC(S(C)(=O)=O)C2)CCn2nccc2C1 C1(N(C(C(C)=CCC)=O)C)CCC(C(=O)NCC(=O)NC(C)(C)C)C1 c1(C(=O)OC(CC=C)C2CC2)cc2ccc(OC)cc2nc1C N1(C(CCc2scc(C)n2)=O)CCC(F)(CNC(c2cc(Cl)cn2C)=O)C1 C=C(C)CCCC(=O)C1CC1.c12ncnc(C)c1C1CCN(CC1)S2 N1(C(c2ccnc(OCC)n2)=O)CCCOC(CNC(=O)CC(C)C(C)C)C1 C(=O)(CCCn1ccnc1)N(CCC(C)NC(=O)CC1(C)CCC1)C c1(C(=O)NCCCNC(c2c[nH]nc2C(F)F)=O)cc(C2(O)COC2)on1 c1(C(=O)NCC2(F)CCN(C(C(C)OCCC=C)=O)C2)coc2c(Cl)cccc12 Cc1ccc(F)c(CNC(=O)C(C2CCN(C(c3occ4c3CCC4)=O)C2)C)c1 C1(CCC)CN(C(C2CCC2C(F)F)=O)CCN1C(c1cn(C(F)F)c(C)n1)=O C1(CC)(CC)CC(NC(c2ncncc2Cl)=O)CN1C(C1C2CCC(=O)C12)=O N1(C(c2cc(SC)oc2)=O)CCC(C)C1C(=O)NCC#CC1CC1 CC12CCOC(C(N3CCC(CNC(c4ncnc(O)c4Cl)=O)C3)=O)(C1)C2 c1(NC2CCN(C(C3(C)CCNC3=O)=O)CC2O)cc2nnc(C(F)F)n2cn1 N1(C(c2n(CC)ccn2)=O)CC(NC(C2CCCC2OC)=O)C(C)C1 CCC(C)(CC)C(=O)N1CC(CNC(c2cncs2)=O)OC(C(F)(F)F)C1 C1(C(CNC(C(C)OCC)=O)(C)C)CCN(C(=O)C(C)CC2CC2)CC1 N1(C(C(=CC2CCCC2)C)=O)CC(O)CC1(C)C(=O)NOCCCCF C(=O)(C1CCc2ccccc21)NC(COC)CC(=O)N(CC(O)CF)C CC(C)C(C(C)NC(c1ccnn1CC(F)(F)F)=O)NC(=O)CN(C)C1CC1 C1(CNC(c2c(C)ocn2)=O)CC12CCN(C(c1cc3c([nH]1)CCOC3)=O)CC2 C1(C(N(CCCCNC(C=CCN(C)CC)=O)C)=O)CN2CCCCC2CO1 N1(C(C(C)NC(C2CC(N=[N+]=[N-])C2)=O)=O)CC(C)C12CCOCC2 c1(CC(=O)NC23C(CN(C(c4cccc(OC)c4)=O)C2)C3)cc(Br)ccc1C C12(NC(C(C3(O)CN(C(CC4N(C)CCC4)=O)C3)F)=O)CCCN(CC1)C2 CCCC(C)(O)C(=O)NC1CCN(C(c2cn(C)nc2I)=O)C1 Cc1c(C(=O)NC2CCN(c3ccc(F)cc3)CC2)sc2[nH]cnc(=O)c12 C(=O)(C1=NOC(CNC(=O)Cn2ncnn2)C1)NCC(C)(C)SC N1(CC(N2CCCC(C)C2)=O)CCC2(CC1)CC2C(=O)NCC1CC2(CC2)C1 N1(C(CC(CC)CC)=O)CCC2(CC1)OC1(CO)CC2(NC(=O)C(C)C(F)F)C1 C(=O)(C#CC1CCOCC1)N1CCC(C(N2CC(C)=C(C)C2)=O)C(C)C1 C1(NC(COCCOC)=O)CCN(C(=O)CC2CCOC(C)(C)C2)CC1F C(C(C)(C)C(C)(C)C)N(C(C1CCCOC1)C(=O)NC1CCCC1)C N1(C(C2CC(OCC)C2)=O)CCC(C(C)NC(=O)CC2(C)CC2)C1 c1(C(C)O)cccc(Cl)c1F.c1(C(C)=O)ccccc1OCC(=O)Nc1cccc(Cl)c1 C(CC(C)(C)C(=O)NCC1(C)CCC(NC(C2(C(C)(F)F)CCC2)=O)C1)OC c1(C(=O)NC2C(C(N(CCOC)C)=O)CCOC2)ccc(O)nc1C c1(C(=O)NCC(CC)NC(=O)Cc2ccc(O)cn2)ccc(C)c(Cl)c1F C1(CCOC)(NC(CCC#C)=O)CCN(C(c2nc(Br)c[nH]2)=O)C1 C1(NC(C2CCN(C)C2)=O)CN(C(=O)CCC(C)(C)N(C)C)CC12CCC2 n1(CC(=O)N(CCCCCCNC(c2ccc(CC)s2)=O)C)nc(O)ccc1=O C(C(C)C(F)C(=O)Nc1cnn(C2CCCS(=O)(=O)C2)c1)OC(CCn1c(C)cc(C)n1)=O C(=O)(C(C)(C)C(C)NC(=O)CCCN(C)C(C)C)NCCn1c(C)nc(C)n1 c1(CN(C(=O)CCCN(C)C)CCNC(C2(C)C(C)C2)=O)ccc(Cl)nc1 C1(c2c(C)ncs2)CCCN(CC(O)CNCCOCC(C)C)C1 N1(C(C(C)C(C)(F)F)=O)CCC(NC(c2cncnc2)=O)C(F)(F)CC1 c1(C(=O)NCC(C2CCC2)NC(C(COC)(F)F)=O)cc(F)cc(Br)c1F C1(C(N2CCCCC(CNC(c3ccc(O)cc3)=O)C2)=O)CCCCCS1(=O)=O C=CCCC(F)(F)C(=O)NC(C)C(C)C(=O)NC1CC2CC(C1)C2 Cc1cccc2cc(C(=O)NC(CNC(c3c(Br)noc3C)=O)C(C)C)nn12 C#CCC(C)(C)C(=O)N1CCC(NC(=O)CCCCCn2cnnn2)C(F)C1 c1(NC(=O)NC(C2CCCOC2)C(=O)OC)ccc(C(F)(F)F)nc1 N1(C(c2c(C)c[nH]n2)=O)CCC2(C)CN(C(C3CCCC(C)CC3)=O)CC12 C(c1ccc(C(N)=O)o1)=CC(N1CC(O)(CN(C)C(C2COC(=O)O2)=O)C1)=O c1(C(=O)NCC(N(C)C(C2(CO)CC2)=O)C2CC2)c(N)cccc1[N+](=O)[O-] c1(N2CCC(OC)(CO)CC2)nc2c(c(=NCC(C)CC(F)(F)F)[nH]1)COC2 C(C(=O)N1CCN(C(c2ccc(OC(F)F)c(Cl)n2)=O)CC1C)(C(C)(C)C)SC C(CC(C(=O)NCC1CC(C)=NO1)NC(=O)C(C)=CC(C)(C)C)=CC C(CCCCCC(=O)N(CCCCNC(c1c(C)cc(C)oc1=O)=O)C)SC C(=O)(C(C)(F)C(=O)NCC(C)CNC(c1cn(C)nc1C)=O)OC CCC(O)C(=O)OC(C)(C)C.C12CCC(C1)C(=O)N1CC(CCO)(C1)NC2=O C1(CC(=O)NCCC2(NC(C3N(C(=O)OC)CC3)=O)CC2)CC(C)(C)CO1 C1(C(N2C(C=C)CCC2)=O)CCN(C(=O)c2cc(CO)c(C)o2)O1 C(C(C(=O)N(CCOC(C)=O)CC)C(C)C)NC(c1cnc(OC)s1)=O c1(C(N(C)CC2CN(C(c3cnc(O)o3)=O)CCO2)=O)[nH]cc2c1CCS2(=O)=O c1(NCC2(OC(C)C)CCOC2)nccc(=NC2CS(=O)(=O)CC2C)[nH]1 CCC(C(=O)N1CC(c2cc(NC(c3ccccn3)=O)on2)C1)NC(C)=O C#CC1(F)CN(C(C2(C3CCCCN3C(C3CCCN3C)=O)CC2)=O)C1 CC1CCCN(C(=O)C=Cc2cscn2)C1CNC(c1cc(Cl)c[nH]1)=O C(C(COC)C(=O)N1CC(N2CCN(C(c3cccnc3S)=O)CC2)C1)OC Cc1nc(F)ccc1CS(=O)(=O)NCC.C1(CN)(CO)CCCC1 c1(NC(=O)NCc2cccc(C(N3C=CC(CSC)C3)=O)n2)cnnc(O)c1Cl C(CC(C)(C)NC(=O)CCN(CC)CC)NC(C1C(C=C)C1)=O C1(C(C(=O)NC(CCCNC(C(CC)F)=O)C)(F)F)(OC)CCOCC1 C1(CNC(C=CSC)=O)CN(C(=O)Cc2csc(C(F)(F)F)n2)CCO1 C1(C2CCCC2)(NC(C2CC(C)CN(C(=O)C=CCF)C2)=O)CCC1 C1(OC)CC2(C1)CC(C(=O)NC1CCCN(C(=O)C(C)(C)N3CCCC3)CC1)C2 c1(C(=O)NC2(CCOC)CCN(C(C3(C)CCCO3)=O)C2)sc(C)c(C)c1C c1(OC)cccc(CC(=O)NC(C)CC(C)NC(C2CCC(C)C2)=O)c1 C(N=c1[nH]c(=NCC(CO)OC)c2sccc2[nH]1)c1ncc(CC)s1 c1(C)ccccc1.c1(C(C2CCOCC2)(CC)NCCOC)nnnn1C1COC1 C1(NC(C(C)C2CCC2)=O)CN(C(C2CCCC3(CC3)C2)=O)CC12CCOCC2 N1(C(CCCC)=O)CCC2C1CCCN2C(=O)Cn1ncc2cccnc12 CC(C)(C#N)CCC(=O)NC1(C2CC2)CCN(C(=O)Cn2cnnn2)C1 C#Cc1cc(F)c(C(=O)NCCN(C(=O)Cc2cncc3[nH]ccc23)C)cc1F Cc1ccc2[nH]nc(C(N3CC4(CCNC(=O)C=CCO)CCC3C4)=O)c2c1 N1(C(C(C)=CC2CC2)=O)CCOCC1CN(C(=O)C(C)(C)C1(O)CCOC1)C CC1CN(C(=O)COc2ccc(CF)cc2)CC(C)C1N CCS(=O)CC(=O)NCC1(OC)CN(c2ccc(COC)cn2)C1 C(=O)(CC(C)C(F)F)N(C1CC(C(=O)NC(C)CN2CCOCC2)C1)C1CC1 c1(NC(N(c2sc(F)cc2C#N)CC(C)C)=O)ccn2ccnc2c1 c1(C(N(C)CC2(NC(C34CCC3CC4)=O)CC2)=O)nccc2[nH]ccc12 C1(C(=O)NCC2CCC(NCC3CCCOC3)C2)CN2CCN1CC2 S(=O)(=O)(c1cc(C)cnc1N1CCCCC(C)(F)C1)N(C(C(C1CC1)OC)C)C C1(C(=O)NC)(C(=O)OC(C)(C)C)CCN(CC(=Cc2ccccc2)OC)CC1.OCC CC1(C)CCCC(C(=O)NC2CC(NC(C3CCOC(=O)CC3)=O)C2)CC1 c1(CN2CC(C)(NC(c3c(F)cc(OC)cc3F)=O)C2)cc(F)c(Br)cc1Cl c1(C(=O)OCc2cc[nH]c2)ccnc(N2CCCCCC2)c1 CC(CN(C)C)CCC(=O)N(C)CC1CN(C(=O)Cc2c[nH]ccc2=O)CCO1 c1(C(N2CCC(CC#C)(C(=O)NC(C)CC3CC3)C2)=O)cccc(C#C)c1C C(=O)(C1=CC2CC(C1)CC2O)C(c1ccc(Cl)c(Cl)c1)=O.C1(N)CCN1C.C(=O)C C(N=c1[nH]cnc2[nH]ccc12)C1N(C(CN(C)CC)=O)CCC1 c1(SC)nc(N2CCC(O)C(C(N3CC4(CCC4)C3C)=O)C2)ncc1F C1(NC(CCCCN(C)C)=O)CC12CCN(C(=O)CC(C)(F)F)C2 c1(C(N2CC(CCC3CC3)C2)=O)ccccc1-n1cc(CC(CO)CO)nn1 c1(C2(O)CC(C(N(C(C)CNC(=O)C(C)NC(C)(C)C)C)=O)C2)cccc(Cl)c1 c1(CC(C)N(C(C(C(CC)O)O)=O)CC)cc2ccccc2o1 N1(C(C2(C(=O)OC)CCOC2)=O)CC2(CCN2C)C1.C12(CC1)CCNC2=O S(=O)(=O)(c1ccc(=NCCCSCC(F)(F)F)[nH]c1)NC1CCC(C)(CC)CC1 c1(C(N2CC(CNC(CCSCCCC)=O)(OC)C2)=O)cc2n(n1)CC(F)C2 CCC(C)(C)C(C)CC(=O)N1CCCC(C)(C)C1CNC(=O)CSCc1ccco1 N1(C(c2cccc(-c3cc[nH]n3)c2)=O)CCC2CC1CN(C(C1(O)CCC1)=O)C2 C(C)(CCC(=O)N(C)CC1(O)CN(C(=O)CNC(=O)Nc2ccccc2)C1)SC N1(C(C(n2c(C)ncc2)C)=O)CC2CC1CN2C(C12CCC1CC2)=O Cc1ccn(C(C)C(N2CCC(C(=O)NC(c3scnc3C)C)C2)=O)n1 C1(CC)CN(C(=O)CCc2ccoc2)CCN1C(=O)Cc1ccccc1Br C1(NC(CC(CC)(F)F)=O)CN(C(c2cc3cccnc3[nH]2)=O)CC1C1CC1 N#Cc1ccc(Cl)c(NC(=O)C(=O)NC(Cc2ccccc2)C(O)C(F)F)c1 Cc1ccc(C(=O)NC2CC(CNC(=O)CCN(C)CCO)C2)c(N)c1 N1(C(C(C=C)(C)O)=O)CCC2(CC1)CC2CNC(c1conc1C1CCC1)=O O(NC(=O)CCSC1CCCCO1)C(C(=O)NCC)CNC=O.OC C1(NC(C=Cc2scc(C)n2)=O)C2CC1CN(C(=O)Cn1cc(C3CC3)nn1)C2 C1(C(N2CCC(CO)CC2)=O)CC2(CCC2N(C(C2OCCOC2C)=O)CC)C1 c1(OC)cccc(C(=O)NC2CC(O)CN(C(=O)COC(=O)N(C)C)C2)c1OC CN1CC(C(=O)NCC2(F)CN(C(c3cnnn3C)=O)C2)NC1=O C(C#CC#CCO)NC(C(C1CN(C(C2CCCCN2C)=O)C1)OC)=O C1(CNC(C(CN(CC)CC)F)=O)CCC(NC(c2ncsc2C(C)C)=O)C1 C1(F)(CNC(C=CC(C)(C)SC)=O)COCCN(C(C2CCCC(=O)N2)=O)C1 C1(NC(CCC(=O)NCCC)=O)CC2CC(C1)N(C(c1n[nH]cc1OC)=O)C2 C1(C(N2CC(O)(C(C)NC(c3n(CC)ncc3)=O)C2)=O)CCC2(CCOCC2)O1 C1(C(N2CC(O)(C3CCCN3C(C3CC(=C4CC4)C3)=O)C2)=O)CC12CCOCC2 c1(C(N2CC(C(C(=O)NC(C(C)C)c3nc[nH]n3)OC)C2)=O)c[nH]nc1C c1(C(=O)NC(CC(C)NC(C(CC#C)C)=O)C)cc(F)cc(Br)c1 C1(C(=O)N(C)CC2(O)CN(C(c3cc(Cl)ncc3N)=O)C2)(OC)CCCC(C)C1 CCC(C)C(C)C(=O)NC(C)(C)CCNC(c1cnnc(O)c1)=O c1(OC(C(=O)NC(C)CN(C)C(C23CC(F)C2C3)=O)C)ccc(C(F)(F)F)cc1 C1(COC)(Cc2cc(C(=O)NC)ncn2)CCN(C(C2(CC3CC3)CC2)=O)CC1.SC C1(SC)CC(CC(=O)NCC2(C(F)(F)F)CC2C(F)(F)F)C1 CC(CCCC(=O)N(C1CC1)CC1CCOC1)NC(c1cn(C2CC2)nn1)=O c1(OC)ncc(Cl)c(C(=O)NC(C)C(C)NC(=O)C(O)C2CCC2)c1Cl C1(NC(C(CC)C(C)C)=O)CCC12CCN(C(c1ccc(OC)c(N)n1)=O)CC2 C1(CC(=O)NC2COCC2CNC(c2ccccc2O)=O)CCCNC1=O C1(C(=O)NCC2N(C(c3c(N)cc(Cl)nn3)=O)CC2)CCC2(CC1)COCCO2 C(=O)(CCCCCN=[N+]=[N-])NCCC(C(=O)N(CC(=C)C)CC)O N1(C(C(C)C(C)(F)F)=O)CCC(NC(c2cccc3sccc23)=O)C(F)(F)CC1 N1(C(Cn2c(C)cnc2)=O)CC(O)CC1(C)C(=O)NCCC(F)(F)CO c1(C(C(=O)NCC(C)C)N(CCC#N)C(C)C)ccc(=O)n(C(C)C)n1 c1(C(=O)NC2CCCCC2N2CCNCC2)ccc(-n2cccc2)cc1 O=S(=O)(c1ccc(N2CCC(F)(F)C(F)C2)nc1)NC1CCCS1 c1(C(N(CCCn2cc(CNC=O)nn2)C)=O)ccc(-c2cnco2)cc1 c1(C(N2CC(O)(CN(C(c3c(CC)nc[nH]3)=O)C)C2)=O)ccc(N)c(N)n1 C1(CNC(C2N(C)CC2)=O)COCCN1C(c1ccc(OCCN(C)C)cc1)=O C(=O)(CCS(N)(=O)=O)N(C1CCN(C2CCN(C(C3CCOCC3)=O)C2)CC1)C C1(NC(=O)C=Cc2ncco2)CC2(CCN(C(c3cc(CO)ccn3)=O)C2)C1 C(C)(C)(CCC(=O)NCCc1ccncc1)NC(C1CC(C(=O)OC)C1)=O c1(C(=O)NC2COCCN(C(c3c(C=C)cnn3C)=O)C2)ccc(C)n(C)c1=O c1(CN2CCN(C(c3nscc3Br)C(=O)NCC=C)CC2)ccc(Cl)c(C)c1 C1(C(=O)NC2CC3(C(NC(c4c(CC)n(CC)nc4)=O)C3)C2)CN2CCN1CC2 N#CC1CCN(C(=O)N(CCO)Cc2cc(C(N)=O)no2)CC1 C1(C(N2CC(CC(C(=O)NCC3C(OCC)CC3)F)C2)=O)CC2COCC2C1 C(=O)(C1CSc2ccccc21)NCCC1=CCN(C(C2(C(=O)NC)CC2)=O)CC1 C1(N(C(=O)C=CC(F)(F)F)CC)CCN(C(=O)C(C)C2CCCO2)CC1 N1(C(c2c(C)oc(Cl)n2)=O)CC2CN(C(c3cnns3)=O)CC2C(F)(F)C1 N1(C(C(CC=C)CC(C)C)=O)CCC2(CCCN(C(=O)C(F)(F)CCC)C2)C1 N1(C(C(n2cc(C)nc2)(C)C)=O)CCSCC1CCNC(c1ncccc1N)=O C(=O)(C1CS(=O)(=O)c2ccccc21)N1CC(NC(CC2C(C)(C)C2)=O)C1 C(c1nc2ccccc2o1)=CC(=O)N(CCNC(c1c(C)cnnc1O)=O)CC C1(CNC(CC(C(CC)C)O)=O)(NC(=O)Cn2ncnn2)Cc2ccccc2C1 C(=O)(C1CC(=O)CCC1)NC1C(C(N2CCC(C)(CO)C2)=O)C2CCC1C2 C1(NC(=O)COc2cncc(CO)c2)CC2CN(C(c3cnsc3)=O)CC2C1 C1(NC(c2[nH]cc(C)c2)=O)CC2CC(C1)N(C(c1cnc(C3CCOC3)s1)=O)C2 C1(NC(c2cn(C)c(=O)n2C)=O)CC12CCN(C(=O)C#CC1CCOC1)CC2 C#CC1CN(C(C2CC=C(C)CC2)=O)CCN1C(c1cnc2sccn12)=O N1(C(CNC(CCC)=O)=O)CC(NC(=O)Cn2ccoc2=N)CC(C)(C)C1 c1(-c2ncc(CNC(c3ccsc3)C)s2)ccccc1F N1(C(c2[nH]cc(C)c2)=O)CCC(C(CO)NC(c2ncccc2N)=O)CC1 CCC(CC(=O)NC1CC(CNC(=O)C(COC)C(F)(F)F)C(O)C1)C(F)F C1(N(C)C)(CN2CC3C(C(=O)N)C3C2)Cc2ccccc2C1.c1(S)ccc(F)cc1F n1(CCC)ccnc1CN(CCNC(C1CCCSC1)=O)C(C)C CC(C)C(C)CN=c1[nH]c(=NCCOC(F)F)[nH]c2ccc(Cl)cc12 c1(C(N(C2CN(C(c3scc(C)c3)=O)CC2O)C)=O)cc2cccc(C)c2[nH]1 N1(C(C2CC(C)=C(C)CC2)=O)CCN(C(C2CC2(F)F)=O)CCC1C CCC(CC(=O)NCCCCCN(C(=O)CC1CC=CCN1C)C)OC N1(C(C2N(C(C=CCCC)=O)CC(F)C2)=O)CCS(=O)C(C)C1 C1(CC)CCN(C(C2CC(CNC(C3CC=CCC3)=O)C2)=O)CCO1 CN1CCOC(C(=O)NCC2(C)CN(C(c3ccns3)=O)CCO2)C1=O c1(CSCC)cccc(C(=O)NC2CCC2CNC(=O)C(C)CO)c1 CC(CC(=O)NC1(C2CCCN2C(=O)C(C)(C)c2cscc2Cl)CC1)C1CCCO1 Cc1nc(CNC2CC(NC(c3ocnc3-c3ccccc3)=O)C2)c(C)s1 C=C(C)CC(C(=O)NCCN1CCCCC1C)NC(=O)C(C(C)C)SCC n1(CC(=O)NCC2CC(NC(C(CCSC)O)=O)C2)cccc(C)c1=O C(C(C)(C(=O)NCCOC1CN(C(C2CCN(C)C2=O)=O)C1)OC)OC Cc1nc2c(o1)CCN(C(C1CCCCCN1C(C1CCC1)=O)=O)C2 N1(C(C(C=C)O)=O)CCC(O)(CN(C)C(C2(C)CC2(F)F)=O)CC1 C12(NC(c3ccc(O)cc3)=O)CCCC1CN(C(c1cc(=O)cc(Cl)[nH]1)=O)C2 C(=O)(C1=CCC(C)(C)CC1)NC(C(CO)NC(c1c(COC)cc[nH]1)=O)C c1(OC)ccc(N)c(C(=O)NCCC(C)NC(=O)CCOC2CCCOC2)c1 CCC(N=c1[nH]c(N2CCN(Cc3ccns3)CC2)nc2cc[nH]c12)C1CC1 c1(C(=O)NC2C(NC(=O)CCOCC(F)F)CCC2)cn2c(n1)CCCC2 Cc1ccc(C(N2CCCCC2CNC(c2cnnn2C)=O)=O)c2cccnc12 C1(NC(C2(CNC(c3cn(CC)nn3)=O)CC2)=O)CCCC(C(N)=O)C1 c1(C(C(=O)NC2C(NC(c3cc(COC)sc3)=O)CCC2)(F)F)ccc(Cl)nc1 C1(C)(C(=O)NC2C(NC(C(CC#C)C)=O)COC2)Cc2ccccc2C1 c1(C(N2CC(NC(CC=C)=O)C(C)CC2)=O)ccc2nc(O)n(C)c2c1 C1(C)(OCCNC(CC(CCC)OCC)=O)C2CC3CC(C2)CC1C3 CCCCC(CC)n1nccc1NC(=O)C(=O)NC1CCN1CCF c1(CC)cccc(C)c1C(=O)NC(C1(O)CN(C(c2nc(CC)oc2C)=O)C1)C C1(NC(c2c(CC)n(C)nc2)=O)CCCCN(C(=O)Cc2cc(CC)nn2C)C1 C1(c2nn[nH]n2)CN(C)CCN1C(=O)Nc1cc(C)n(Cc2ncccn2)n1 c1(CC(=O)NCC2N(C(C)C)C(C)(C)OC2)cc(Br)cc2c1OCC2 C(=O)(C1=CCC(C)(C)CC1)N1CCC(N(C(=O)C=Cc2ccoc2)C)CC1 C1(C(F)F)(CNC(=O)C=Cc2cocn2)CCN(C(C2CC23CCC3)=O)C1 c1(OC)c(N)c(C(=O)NC(C)(C)CNC(c2ccccn2)=O)cc(Cl)c1Br N1(C(COCCCCC)=O)CC2CC2(CNC(c2cc(C(C)(C)C)c[nH]2)=O)C1 C1(CC(=O)N(CC)Cc2ncc(Br)cn2)CCCN(C(=O)COCCO)C1 Nc1ccc([N+](=O)[O-])cc1C(N1CCC(N(C(=O)C(F)(F)F)C(=O)C=CCO)C1)=O c1(C(N(CC(CN(C(=O)C(O)CN(C)C)C)O)C)=O)noc2c1CC(F)(F)CC2 CC1CCC(O)CN1C(C1CC(N=[N+]=[N-])CN1C(c1cc(F)ccc1F)=O)=O O=S(=O)(c1cnc(NCCOc2ccc(F)cc2)c(Cl)c1)NC1CCC2CC12 c1(C(=O)NC2CCCN(C(c3ccn(C)c(=O)c3)=O)C2)c(F)cc(F)c(F)c1F N1(C(=O)Cc2nc(F)c(F)cc2F)CCCC2C1CCCN2C(=O)CC1CCC1 N1(Cc2cc(OCC)ns2)CCC(NC(=O)Cc2ccc(Cl)c(F)c2)C(C)C1 c1(C(N2CCC(CCNC(CC(C)O)=O)C2)=O)cccc(CCO)c1 C1(NC(C(c2ccccc2)C)=O)CC2(C1)CC(NCc1sccc1Br)C2 C1(CN(C(C=C(C)C)=O)C)CCCCN1C(=O)CC(C)c1ccncc1 N1(C(C2(C)CCCN2)=O)Cc2ccc(C(=O)Nc3cc(C#N)ccc3I)cc2C1 C(=O)(CCCN(C)C(C(=O)CCCn1cc(C)cn1)=O)OC.N CC1CC=C(C(=O)N(C(C)(C)CC(N2CC(=O)NCC2C(N)=O)=O)C)CC1 N1(C(C(COC)(C)C)=O)CCOC2(CCN(C(=O)Cc3sc(C)cc3C)C2)C1 C1(C)(C(=O)NC(C)CN(C)C(C2(F)CCOC2)=O)CC(c2ccccc2)=NO1 CC(CCCC(=O)NCC1C=CCC1)NC(C1(C)COC1)=O c1(C(=O)NC(CNC(C2(c3cc[nH]n3)CC2)=O)CO)cc2ncccc2[nH]1 c1(C(N2C(C(=O)Nc3cnc(F)cc3C)CC(=C)C2)=O)cc(Cl)ncc1F Cn1cc(Cl)c(C(=O)NC(C)(C(=O)NCc2ccsc2)C2CCC2)n1 c1(C(N2C(CNC(c3n[nH]cc3Cl)=O)CCC(C)C2)=O)cc2ccccn2n1 c1(C(=O)NC2CCCCN(C(c3n(CC)nc(C)c3)=O)C2)ccc(F)cc1C#N N1(C(C=CCOCCOC)=O)CC(NC(=O)C=C2CCCCC2)CC(F)C1 c1(C(=O)NC(CN(C)C(C2(c3cnccn3)CC2)=O)C)cncc(Cl)c1Cl N1(C(c2ncc(C)cc2C)=O)CC(NC(C2CC3CCC3C2)=O)C2CCCC2C1 C(=O)(CC(C)C(F)(F)F)NCCCC(C)NC(c1snc(Cl)c1Cl)=O C1(NC(CC(C)NC(=O)Cc2ccccn2)=O)CC2CCC(C1)C2O c1(NC(=O)NCC2CC(C(=O)OCC)NC(=O)C2)cn2cc(Cl)cc(Cl)c2n1 C1(N(CCC)CC2CCC(C)C2)CCN(C)CC1 N1(C(CSCC(=O)OC)=O)CCn2c(CNC(=O)C(F)n3cccn3)nnc2C1 C(CCC(C)(C)NC(C1CC1c1ccccc1)=O)NC(c1cn(C)nc1)=O N1(CCC(N2CCC(NC(C(C)(C)C)=O)C2)=O)CCCS1(=O)=O N1(C(CC(=O)OCC)=O)CCC2C1CCCN2C(c1cc(Br)cc(I)c1)=O c1(-c2cn(CCCC(N3CCOC4CC34)=O)nn2)cccc2[nH]ccc12 C1(CNC(C=CC(CC)=CC)=O)CN(C)CCN1C(=O)CC(C)(O)C=C C12(CNC(CCOC)=O)CC(NC(=O)CC(C)C(C)C)(C1)C(C)O2 N1(C(C(C(=O)OC)OC)=O)CC2(CCCC2)C1C(=O)N(C)Cc1ccns1 c1(OC)cccc2[nH]cc(CC(N3CC(NC(C4(F)CC4)=O)CC3C)=O)c12 C(c1cccc(O)c1)=CC(N1CCC(NC(c2c(CC)nc(C)o2)=O)C1)=O c1(C(=O)NCC(C2CCCC2)NC(=O)CCC2CCOC2)cncc2[nH]ccc12 C1(NC(=O)NCC2C(c3ccc(Br)cc3)(C)C2)CCCC2OCCC12 C1(OC)CN(C(=O)Cc2ccc(C)o2)CC1NC(C1CCCN1C(=O)C1CC1)=O O=C1CC(C(=O)NCCN(C2CC2)CC2CCCNC(=O)C2)=NN1 c1(OC)cccc(-c2ccc(C3(C(N4CC5CC5C4C#N)=O)CC3)cn2)c1F c1(COC(=O)COCCc2ccco2)cccc(-n2cncn2)n1 c1(C(=O)NCCN(C(C2CCSC(C)C2)=O)CC)coc(C#N)c1 c1(OCC)cccc2[nH]cc(C(=O)NCC(C)NC(c3csc(C)c3C)=O)c12 N1(C(c2n(CC=C)ccn2)=O)CCCC(C2CCCN(C(=O)C(F)OC)C2)C1 Cc1ccc(-c2cnc(NCC3CC4CCC3O4)c(O)c2)c(C)n1 C(=O)(C(O)CC[S+](C)C)N1CC(C)(NC(c2c(COCC)cc[nH]2)=O)C1 c1(CCC(=O)NCC2C(NC(CC3(OC)CC3)=O)C2)nc(C)c(C)[nH]1 c1(C(N2C(C(N(CCCOCC)C)=O)CCC23CC3)=O)ccc(C#N)cc1C C(=O)(C(C)(C)C(F)(F)F)N1CCCC(CNC(C2C3(CC(OCC)C3)C2)=O)C1 C1(NC(CSCC)=O)CN(C(c2cc(OC)cc(Cl)c2F)=O)CC12CCC2 c1(C(=O)NC(CCOC)CNC(c2cccnc2)=O)c(C)cc(Cl)cc1N C1(NC2CCN(C(=O)C(=O)NCC3CCC(C)CC3)C2)C2C3CCC(C3)C12 C1(CC(=O)NC2(C(COC)O)CC2)COC(=O)C1 C(=O)(CC1CS(=O)(=O)c2ccccc21)NC(CNC(C1(CC)CC1)=O)CO C1(NC(C)=O)CN(C(=O)Cc2ccc(C#N)cc2)C2(CCOCC2)C1 C1(NC(=O)OC(C)(C)C)CC12CCC(C(=O)NCc1n[nH]cc1C1CC1)CC2 N=c1cc(C(=O)NC2CCC(NC(=O)Cn3cccn3)C2)c(Br)c[nH]1 C1(NC(CN(CCOC)C)=O)CC12CCN(C(c1csc(C(C)C)n1)=O)CC2 c1(C(=O)NCC(=O)N(CCNC(C(CC)N2CCCC2=O)=O)C)ccccc1C N(C1CCCc2cc(CNC(=O)CC3CCC(O)C3)ccc21)C(CC(=C)C)=O c1(OC)cc(SC)ccc1C(=O)NC(CNC(=O)C(C)(C)CF)CC(F)(F)F C1(CNC(CCC2CC(NC(C3CCC(NC)CC3)=O)C2)=O)CC2C(C1)C2(F)F c1(CCC)ncoc1C(=O)NC(C)(C)CCNC(=O)C(C1CCOC1)OC C1(C(=O)NCCCOC=C)CCCC(NC(=O)C(CCSC)OC)C1 C1(NC(c2cnc(C3CC3)nc2)=O)CN(C(C2CC2F)=O)CC2(CCC2)C1 C(=O)(C(C)CN(C)N1CCOC2(CCCN(c3cccc(C)c3)C2)C1)OC C1(O)(CNC(c2c(C)noc2C)=O)CCCN(C(C2CC(CF)C2)=O)C1 C1(CNC(C2N(CC)CC2)=O)CC2(CCOCC2)CN1C(=O)CC1CC(=O)C1 N1(C(CN(CCC)C)=O)CCN(C(c2ccc(C)n2C)=O)CC1CC Cc1cccc(O)c1C(=O)NC1CC1CNC(c1cc(C)n(C2CC2)n1)=O N1(C(COC(C)(C)C)=O)CC(CNC(C2(c3ccsc3)CC2)=O)C(O)C1 c1(NC(=O)NCC2CC(O)(CC#C)C2)cc(CN)ccc1OC(F)F.C(C)(C)(C)O C1(C(N(CC(=C)C)C)=O)CC12CCN(C(c1ccnc(OC)n1)=O)CC2 N1(C(c2cn(C)nn2)C(=O)NCCSC)CCC2OCCC2C1 c1(C(=O)NCC2(CNc3nc(C)nc(O)c3)CC2)nc2nccc(C)n2n1 CC1(C)CCC(CC(=O)NCC(C(C)(C)C)NC(=O)C2=COCC2)C1 c1(OC)cc(OC)c(CCN(CC(=O)O)C)cc1C(=O)OC C12(C(=O)NC3C4CN(C(c5c(C=C)cnn5C)=O)CC43)CCCC1CC(=O)C2 C1(O)(CNC(=O)CCC2CCOC2)CCN(C(=O)Cc2c(Cl)cccc2Cl)CC1 C(=O)(C(COC)CC(C)C)NC1C(CN(C(CCCCC#C)=O)C)CCC1 C1(N(C(C(F)=CC)=O)C)CCC2CN(C(c3cc(S(=O)(=O)NC)co3)=O)CC12 N1(C(C2(CCN(C)C)CC2)=O)CC2CCC1C1CN(c3nnco3)CC21 CCC1=C(C(=O)NCCCCN(C(=O)CCOc2ccccc2)C)CCCO1 C=CC1(CC(N2CCCC(NC(=O)CNC(=O)NC3CC3)C2)=O)CCCCC1 c1(C(=O)NCCC(C)N(C)C(c2ccns2)=O)csc(-c2ncc[nH]2)n1 N1(C(C2C(CC)CCN2C(=O)CCS(C)(=O)=O)=O)CCCC2CC1C2(C)C C(C1=NOC2CN(C(c3c[nH]nc3OC(C)C)=O)CC12)NC(CCC(=C)Cl)=O c1(N(C)C)nc2c(c(=NC3CCN(C(C4CC4c4cn(C)cn4)=O)C3)[nH]1)SCC2 N1(c2nccc(C)n2)CC(NC(=O)C(N2CC3CNC(=O)C23)=O)CC(F)C1 Brc1ccc2c(c1)OCCN2Cc1cnc2n1CCC2 C(=O)(CC(C)(C)CC(=O)NC1CN(C(=O)C2=C(C)CCC2)CC1C(F)F)OCC C1(C(=O)NCC2CN(Cc3ccccc3)CCO2)CCOCC12CCCCC2 C(=O)(CC(C)CC(C)C)NC(CCC=C)C(=O)NC(C)(C)CCCF C1(CN(C)C(c2cccc(CNC(C3CC(N(C)C)C3)=O)c2)=O)CC2C=CC1C2 O=C(C(O)C(F)F)NC1CC(NC(=O)C(Cc2cccnc2)C2CCCC2)C1 C(C(C)(C)C#CC(=O)NC1(CO)CC2CCCC12)NC(Cc1nc(C)oc1)=O C(CCC(C)(C)C(=O)N(C)Cc1nccn1C)NC(CC(CC)CC)=O C1(C(=O)NC(CCC)C(=O)N2CCCC2)CCCCCN1C(=O)CN1CCSCC1 C1(CSC)CCN(C(=O)C(C2(O)CCCCC2)NC(=O)CSC(F)F)CC1 C(=O)(CC(C)(C)C(F)F)NCC(CC)NC(C1(c2ccccn2)CC1)=O c1(CC(=O)N(CC(C)NC(=O)CCCF)CC)cc(C)cc(Br)c1 Cc1ncn(C)c(=O)c1C(=O)NCC#CCNC(C1CC2CCC1O2)=O c1(CCC(=O)NC2CN(C(C(C)(C)OC)=O)CC2O)ccc(F)c2ccccc12 c12cc(ccc1O)NC2=O.C(=O)(C(C)(CC)CO)N1CC2C(SCC)C2C1.C(C)(C)O C1(NC(c2n(CCCC)nnn2)c2nc(CO)cs2)CCC(C)(C)CC1 c1(C(=O)NC(C2CCCN(C(C3CC(C#N)C3)=O)C2)C)cnc2c(c1)CCC2 N1(c2nc(C)c(C#N)cc2)CCc2ccccc2C(NC(C2(N=[N+]=[N-])CC2)=O)C1 N#Cc1ccc(SCC(=O)NCc2ccnnc2O)cc1.C12CN(CC1O)C2 C=CC1(C(N2CCC(C(F)F)CC2)=O)CCN(C(c2ccnc(C)c2)=O)CC1 C(=O)(C1CCc2snnc21)N(CCCNC(C(C)O)=O)C1CC1 C(=O)(CCCCC(=O)N1CCCC1CCNC(C1(C)CC1(Cl)Cl)=O)OC C1(N(CCO)CC2CC2)CCN(C(n2nnnc2C(c2cc(C)on2)OC)=O)CC1 N1(C(c2c(COC(C)=O)cccn2)=O)CCCC12CCN(C(C1CC(F)C1)=O)C2 CC(CNC(=O)CN1CCSCC1)C(=O)N1CC=CCC1 C1(C(=O)NCCCN(C(CCCCC)=O)C(C)C)CC2C=CCC(C1)C2 c1(C(N2CCN(C(c3cc(CCC)oc3C)=O)CC2)=O)ccc(S(C)(=O)=O)cc1 C1(NC(c2ccn(CC)n2)=O)CC2CC1N(C(c1cscc1OC)=O)C2 N1(C(=O)OC(C)(C)C)CCC1CCCNC(CCCC1CCCO1)=O C=CCC(C)(C)C(=O)N1CCC(CNCc2cc(O)ccc2O)C1 c1(C2(C(=O)NC(c3nc(CC)[nH]n3)C)CC2)nnc2n1CCCC2 CC(C)(O)C#CC(=O)N1CCC(CNC(=O)CC2CC2)C1(C)C c1(C(=O)NC(C2CN(C(c3cc(O)ccc3O)=O)C2)C)[nH]nc([N+](=O)[O-])c1Cl c1(C(=O)NC23CCN(C(C=Cc4nc(C)sc4)=O)CC2C3)cc(N)c(Cl)c(O)c1 C1(F)(C(=O)Nc2c(C(C)C)scc2)COC(C)(C)C1 N1(C(C(CC=CC)CC)=O)CC(O)(C2(CNC(=O)Cc3cccc(SC)c3)CC2)C1 c1(COC(C(C)C(C)c2ccccc2Cl)=O)cn2ccccc2n1 c1(C(C)C)ncc(C(=O)N(C(C)CNC(=O)C(C)C2CC2)C)s1 n1(CC(=O)NCC2N(C(COCC(=O)OC)=O)C3C(C2)C3)ncc(O)nc1=O N1(C(C=C(C)C2CCCCC2)=O)CC(NC(=O)CCc2nccs2)CC(C)(C)C1 Nc1c(C(N2CC(NC(=O)COC3CCCCC3)C2)=O)cnn1CCO C1(C(N(C)CC#N)=O)CCC2(CN(C(=O)CCc3ccn(C)c3)C2)O1 CCC(C)C(C)N=c1[nH]c(N(CC(c2ccccc2Cl)OC)C)nc(=NC)[nH]1 C1(CNC(C=CC(CC)=CC)=O)CN(C(=O)CNC(C2CCCC2)=O)CC1C C1(C2CCN(C(=O)C(C)(C)C(C)(C)O)CC2)(NC(C(C=CCCC)O)=O)CC1 N1(C(CC=C)=O)CCN(C(c2nccc(C(F)(F)F)n2)=O)C(C2CC2)C1 c1(C(=O)NC2C3CN(C(CCSCCCC)=O)C(C3)C2)cc(F)c(F)c(F)c1 c1(C(=O)NC23CC(NC(C4C5CCC(F)(F)C45)=O)(C2)C3)cnc2[nH]cnc2c1 CC1COC(C)(C)CN1C(C1CCC2(CC2)N1C(c1cocn1)=O)=O c1(C(=O)NCC2COCCN(C(c3cc(C)ns3)=O)C2)ccnn2ccnc12 CC(C)C(C(=O)N1CCC(N(C(=O)C2=CCSC2)C)CC1)n1ncc(N)n1 S(=O)(=O)(c1cccnc1NCc1ccc(C#N)o1)NCC1(OC(C)C)CCC1 N1(C(CCNC(c2nc(CCC)oc2)=O)=O)CCC(CF)CC1 C=CC(C)(O)CC(=O)N(CC(=O)NCc1ccc2c(c1)CC2)CC1CC1 c1(OCCN(C)C)cccc(CNC(=O)CN2C(=O)CCC2=O)c1 CC1(C)COCC(C(N2CC(CNC(c3nn[nH]c3Cl)=O)C(F)(F)C2)=O)O1 c1(CCC)nc2cc(C(N3CC(N(C(=O)CCCCSC)C)C3)=O)cc(C)c2[nH]1 C1(C2CC2)(NC(C=CC=CCC)=O)CCN(C(C2CCC2CF)=O)C1 c1(C(=O)NCC(CC=C)NC(=O)C(c2ccc(C)o2)C)cccc(CCO)c1 C1(CCNC(=O)CSC(F)F)CCCC(NC(=O)C2CC2)C1.C12CC(C1)NC2=O Cc1cn(C)cc1C(=O)NCCCN1CCN(C(C2(CN(C)C)CC2)=O)CC1 CN1CC(CNC(=O)CC2CCCN(C(C3C4CCC(F)C34)=O)C2)CC1=O N1(C(c2cc(CCC)ncc2)=O)CCCCCC1CNC(=O)COC1(C)CCC1 O=C(Cc1ccc([N+](=O)[O-])c(O)c1)N=c1cc[nH]cc1CCN1CCOCC1 Cc1ccc([N+](=O)[O-])cc1CN(C=O)CC(N1CC(c2ccc(Br)c(F)c2)C1)=O CS(=O)(=O)c1ccc(N(C)Cc2csc(-c3ccsc3)n2)cc1 CC1(C)OCc2cc(C(c3nnnn3C)NCc3cnc(C(N)=O)nc3)nn2C1 C(C(F)(F)CCC(=O)N(CCC1CC1)CC1CC1)n1cc(C(C)NC)nn1 c1(CNC(CC(C)NC(N)=O)=O)cccc(NC(=O)C(c2ccccc2Cl)O)c1 N1(C(C2CCN(C(CC(C)C3CC3)=O)CC2)=O)CCC12CCC(O)CC2 C(c1ccncc1)=CC(=O)NCCNC(CCOCCOCC)=O Cc1ccc(C(C)C(=O)N(C2CC2)CC2CN(C(=O)CC(C)c3ccccc3)C2)o1 C(CC(O)C(=O)NCC(=C1CN(C(C2CN(C)C(=O)N2)=O)C1)F)SC C1(NC(CS(N)(=O)=O)=O)CC2CCC(C1)N2C(c1ccsc1S(N)(=O)=O)=O CC1N(C(c2cc(CNC(C3(C#N)CC(=O)C3)=O)[nH]n2)=O)CCC1(C)C CC1CN2CCN1C(C(N1CCCCC1CNC(=O)Cc1ccccc1F)=O)C2 c1(C(N2C3(CN(C(CC(CC)C)=O)C3)CC2)=O)cccc([Si](C)(C)C)c1 C(=O)(C1=NOC2COCC12)NC(CC(N1CCC(N)C(O)C1)=O)=O N1(C(C(CCCOC)C)=O)CC2(CCCCN2C(c2snnc2C)=O)C1 C(C)(CCC(=O)NCC(C)CNC(c1cc(C)nn1Cc1ccccc1)=O)OC C1(N(C(CCCN(C)C)=O)C)CN(C(C2C(Cl)(Cl)C23CC3)=O)CC12CC2 c12cc(sc1C)NC(=O)C2(F)F.C1(CN(C)C)CC(NC(C2CCSC2)=O)C1 NS(=O)(=O)c1ccc(C(=O)NC2CCN(C(C3COCCO3)=O)C2)cc1 C1(NC(C2SCCCS2)=O)CCC12CN(C(=O)C(c1ccccc1F)O)C2 CC(C)C(C(=O)NCC1CCN(C(C2(C)CC3CC3C2)=O)C1)N(C)C c1(C(=O)OC(C)(C)C)ccc2c(n1)CCC2.CCCC1=CC(=O)OC(=O)NCC1 N1(C(c2n[nH]c3c2CC(C)CC3)=O)CC2CCN(C(=O)COC(F)F)CC(C2)C1 N1(C(c2ccc(C)c(O)c2)=O)CCCN(C(c2cnc(Cl)s2)=O)CC1C c1(C(=O)NCC(C)CNC(=O)C=Cc2cncc(F)c2)cc(=O)n2ccsc2n1 C1(NC(COC(CC)C)=O)CCN(C(c2ccc(NC(C)=O)cn2)=O)CC1F CCC1C(=O)Nc2ccc(C(N3CC(CNC(c4csc(CO)n4)=O)C3)=O)cc21 N1(C(c2cccc(C#N)c2)C(=O)NC(C)C)CCN2CC(F)(F)CC2C1 CC1(C)CC(CC(=O)NCCC(F)(F)F)CN1C(=O)C=CC(F)F C1(NC(C2(OCC)CC2)=O)CC1C1CCN(C(C2CCCN2CC)=O)CC1 C(CC(C(=O)N1CCC(CNC(N)=O)CC1)NC(=O)CC1CCC(=O)CC1)OC O=C1CCN(C(c2cc(CNC(C3(CC4CCC4)CC3)=O)no2)=O)CCN1 C(CCCCC(=O)NCCCN(C(=O)CCN1C(=O)CCC1=O)C1CC1)SC N1(C(C2(CC#C)CCC2)=O)CC2CC(NC(=O)COCCOCC)C1C2 C1(O)(CN(C(=O)C(F)n2ccnc2)C)CN(C(=O)CCc2cncs2)C1 N1(C(c2c(CNC(c3cnn4c3CCC4)=O)ccs2)=O)CCC2CCC(O)C1C2 c1(C(=O)NC(CNC(c2c(OC)cncn2)=O)C)cc(Br)cc2c1OCC2 c1(CNC(c2cccc(C(F)(F)F)c2Cl)C)ccc(F)c(F)c1O C(c1ccccc1F)=CC(=O)NCC1CCC1NC(=O)CC(F)(F)F N1(C(C(C)N(C)C)=O)CCC(O)(CNC(c2cn(C3CCCCC3)cn2)=O)C1 C1(NC(=O)CCn2ccnn2)CN(C(=O)Cn2ncnn2)CC12CCC2 c1(CCC(=O)NC(C)C(=O)NC(c2nccs2)C)ccn(C)n1 c1(C(=O)NC2(CNC(c3cn(CCC=C)nn3)=O)CCCC2)ccc(C)cc1C c1(OC)nc(C(=O)NCC2CN(C(=O)C=CC(C)C)C3CC23)cc(O)n1 c1(C(=O)NCCC2(O)CN(C(C3(CC)CC3(F)F)=O)C2)cc2[nH]nc(C)c2cn1 C1(O)(OCC)CCN(C(C2(C(=O)CCNC(C3CCC3CO)=O)CCC2)=O)C1 Cc1nc(C)c(CCC(=O)NCC(C)(C)CC2CC2)c(O)n1.C(=O)CCCC(F)F N1(C(C2CC(C)=C(C)CC2)=O)CCC(NC(C2CN(C)C2)=O)C(C)(C)C1 O=C(C(O)C1=CCCCC1)NC1CC(C(N2CCCC23CCNC3=O)=O)C1 Cc1ccc(C)c(C(=O)NC2CC3CC(NC(=O)CC(C)N(C)C)CC3C2)c1C N1(C(c2c(C)noc2C(C)C)=O)CCCC2CN(C(c3occc3F)=O)CCC12 c1(C(=O)NCC2(O)CC(NC(C3CC(=C)C3)=O)C2)sc2ccc(C)cc2c1C c1(C(=O)NC2CCC(C(N3CCC(F)(F)CC3)=O)C2)nnc(O)nc1O C1(CNC(C2(CCCC)CCC2)=O)C(CNC(C23CC(F)(C2)C3)=O)C1(F)F C1(C(=O)NC(CC)C)CC(C)CCN(C(=O)C(C2CCOCC2)C)C1 Nc1cc(Cl)cc(Cl)c1C(N1CC2CCC1CN2C(C1CCCC12CC2)=O)=O N1(C(=O)CC2(O)CCC2)CC2CCC2(CC(=O)NC2CCC=CCCC2)C1 CC(C)(C(c1nnnn1CC(F)F)NCCC(N)=O)c1ccccc1 c1(OC)cnccc1C(=O)NCCCCNC(C1CCC2(CC2)C1)=O c1ccc2oc3c(c2c1)CCCCC3.O=CN=c1ccc(Cl)n[nH]1 C1(NC(c2cccnc2O)=O)CC2CC1N(C(C1(N3CCCC3)CC1)=O)C2 C1(CC(N2CCC(c3cn(CCCC)nn3)C2)=O)CCN(C)CC1 N#Cc1ccc(C(N2CCCCC2C(O)C(F)F)=O)cc1[N+](=O)[O-] c1(C(=O)NC2CN(C(C(C)CF)=O)CC(C)(C)C2)c2c(nn1C)CCSC2 C1(C(N(C(CSC)C)C)=O)CN(C(=O)CC2CSCCO2)CC1C(C)C C1(CNC(c2scc(OC)c2)=O)CCN(C(c2cnc(C(F)F)s2)=O)CC1C c1(C(=O)OC)cnn(C)c1S(=O)(=O)NCCc1cccc(N)c1 CS(=O)C=CC(=O)NCC1(CNC(=O)CNC(C2CCCCC2)=O)CC(F)(F)C1 n1(C(c2ccccc2)C(=O)OCC)nnc2c(N3CCC(OC)C(C)C3)ncnc12 C=CCC(C(=O)N1CC(NC(=O)CCc2ccc(Cl)c(F)c2)C(C)C1)C(C)(C)C c1(C(=O)NCCCN(C(C2CC(C#N)(OC)C2)=O)C)c[nH]c(=O)c2ccnn12 C1(NC(C(c2cccnc2)N(C)C)=O)CC2(CCCN(C(C3(C)CSC3)=O)C2)C1 CC1(CC(=O)NC2CC(CNC(c3c[nH]cc3C3CC3)=O)C2)CCCO1 C1(CNC(C(C)O)=O)CC2CC(C1)N(C(c1ccccc1OCC#N)=O)C2 N1(C(c2cc(C(C)=O)c(C)o2)=O)CCCN(C(=O)C=CCN2CCCCC2)CCC1 c1(OC)ccc(C(=O)NC2CC(C)N(C(C3CCCC(=O)N3)=O)C2)nc1Cl N1(C(Cc2cc(C(C)(C)C)sc2)=O)CCN(C(=O)Cn2nccc2N)CC(O)C1 c1(N(C(c2cc(Br)c(C)o2)C(=O)NC(CC)C)CC)cc(C)ccc1[N+](=O)[O-] C(=O)(CC(CCC(=O)NNC(=O)NC1CCCC1)C(F)(F)F)OC C1(C)(C(=O)OCc2onc(CN(CCCC(=O)OC(C)(C)C)C)n2)CC2CCC1C2 CC1(C)CC(CNC(C2CC(C(C)(C)C)C2)=O)N(C(C2CCOC2(C)C)=O)C1 C(=O)(C(C)S(C)(=O)=O)NCC(CC=C)NC(c1cnc(C)o1)=O c1(C(N2CCCC(C(C)NC(c3csnn3)=O)C2)=O)cc(S(N)(=O)=O)cs1 N1(C(CCC(=C)C)=O)CCC(NC(=O)C(C)OCCc2ccccc2)CC(O)C1 O=C1OCC2CN(C(c3ccc(-n4ccc(O)n4)cc3)=O)CCC12 CC1(C)CCCOC1C(=O)NC1C2CC3C1C3C2C(N1C2CSCC1C2)=O C(=O)(CCC(=O)NC1CCCCC1CNC(c1ncc(OC)cn1)=O)OC C1(NC(C2CCC2)=O)CN(C(c2ccc(CO)o2)=O)Cc2nccn2C1 C(=O)(CCCS(C)(=O)=O)NC1(C)CN(C(=O)CC2(C(F)(F)F)CCC2)C1 c1(NC(C23C(CN(C(=O)CCCc4ccccc4)C2)C3)=O)cc(Br)c(F)cc1F CC1CCCCCCN1C(=O)C(CN(C)C)NC(=O)C(C)(C)n1cnnn1 C(=O)(C(C)(C)C(C)O)N1CCC(C)(C(=O)NC(C)Cc2cnccn2)C1 N(C(=NCC(F)(F)C(C)(C)O)NCC(C)(C)CC(=O)N(C)C)C(C)C c1(C(N2CCC(NC(COCCCC#C)=O)C(CC)C2)=O)ncnc2ccsc12 C1(NC(C2CC2C(=O)Nc2ccc(Cl)cc2)=O)CN(C(=O)C2=CCCC2)CC1(F)F N(C1CN(C(=O)Cc2cccc(Cl)c2Cl)Cc2ccccc21)C(CNC=O)=O C(=O)(C#CC1CCCCC1)NCC(CNC(c1c(CC)con1)=O)CO C1(C(=O)NCC(c2ccccc2)NC(c2snnc2C)=O)(COC)CCCCC1 CCC(C)C(=O)N(C)CCOCCN(C)C(c1cc(Br)no1)=O CC1CCC(NC(=O)C(C)(C)c2cnn(C)c2)CN1C(c1cnco1)=O N1(C(c2c(CNC(c3ccc(CC)[nH]3)=O)nnn2C)=O)CC23CCC2(COC3)C1 C1(F)(CNC(c2n(CC=C)ccc2)=O)CCC(NC(=O)CCc2nncn2C)C1 C1(C)(CNC(C=Cc2n(C)cnc2)=O)COCCN(C(C2CCNC(=O)C2)=O)C1 c1(CC)nc(C(C)OOC(F)(F)F)n(-c2ccc(C(=O)O)cc2)n1 N12CCC(C)(C1)C2=O.c1(C(=O)NC(CC)CSC)ccsc1C(F)F c1(C(=O)NC2(CO)CN(C(c3cnc(CC(C)(C)C)o3)=O)C2)ccc(CF)cc1 c1(C(=O)NC2CCN(C(C3CC4C=CC3C4)=O)CC2)ccn2ncnc2c1 C=CC(C)C(=O)NC(CN(C)C)C(=O)N1CCC(CF)C1 Cc1ncc2n1CCC(C(=O)NCC1CN(C(=O)COCCO)CCC1(C)C)C2 O=C1CN(CCOCCc2ccccc2)C(=O)N1SCCCCc1ccccc1 Cc1nc(SCC(=O)NCCC(C)NC(=O)CNC(c2cnoc2C)=O)cs1 CC1CC(NC(c2cnn(C3CC3(F)F)c2)=O)CN1C(=O)C=CI N1(C(C(C2CCC2)OCC)=O)CCC(COCC)(NC(C2(CF)CC2)=O)C1.CF c1(C(N2C(CC)CN(C(C3C(F)(F)C34CC4)=O)CC2)=O)cn2ccc(C)cc2n1 C1(O)(COC)CCN(C(=O)C(C2CCCO2)NC(=O)C=C(C)C)C1 Nc1cc(C(N2CCC(NC(c3cnc4n3CCC4)=O)C(F)C2)=O)cc(O)c1Cl c1(C(=O)NCC2CC2CNC(C2CCCC2O)=O)cc(C(F)F)no1 Cc1ccc2c(c1)C(=O)N(CC(=O)NCCOCCNC(=O)C(C)C(C)O)C2=O N1(C(Cc2cc(C)no2)=O)CCC(F)C(NC(c2ccc(C(F)F)c(Cl)c2)=O)C1 C1(CNC(Cc2ccc(C)cc2)=O)CN2CCCCC2CN1C(c1cn[nH]c1)=O N1(C(C(C=C)(C)C)=O)CCC(NC(C2(C)CC(OC)CN2C)=O)C(C)C1 n1(CC(=O)NCCC2CCCN(C(c3cc(CCO)on3)=O)C2)ncccc1=O C=CCC(CNC(=O)CC(Cl)Cl)C(=O)NC(CO)CCC(C)C C1(CNC(CC=CCNC(C2(CC)CCC2)=O)=O)C=CCOC1 C1(C(N(C(C)CNC(c2cccc(C(C)(C)C)c2)=O)C)=O)CCC2(C1)CC2(F)F N1(C(C=CCOC)=O)CCCCC12CC(NC(c1ccc(SC3CC3)cc1)=O)C2 c1(C(=O)NC2CC(NC(=O)CSC(F)F)C2)cccc(-n2ccnn2)c1 n1(CC)cnc2[nH]c(=NC3COc4ccc(Br)cc43)[nH]c(=NC(C)CCOC)c12 c1(C(N2C(C(C)(C)NC(C(CCCC)C)=O)CCC2)=O)cc2sccc2cn1 c1(C(=O)NCC(C)N(C)C(c2c[nH]nc2C(F)(F)F)=O)cccc(C2CCC2)c1 N1(C(C=CCCC)=O)CCN(C(=O)C(CC(C)C)NC(=O)OC(C)C)CCC1C C=CCC(C(=O)NCc1cncc(OC)n1)NC(=O)Cn1[nH]cnc1=N Cc1c(C(N2CCN(Cc3ncco3)CC2C)=O)sc2ccccc12 C1(C(N(C2CN(C(C(n3ccc(C)n3)C)=O)C2)C)=O)CCCN(CC(F)F)C1 N1(C(C2CCN(C)C(=O)C2)=O)CCC2(CCCN2C(=O)C(Cl)=CCl)CC1 C1(C(=O)NC(CCC)(C)CC)CCC2(CC2)N1C(c1c[nH]nc1C)=O Cc1cc(F)cc(CN2CCC(F)(C(=O)Nc3cc(N(C)C)ccc3F)CC2)c1O N1(C(c2ccc(SC)cc2)=O)CCC2CCC(NC(=O)Cc3cnn(C)c3C)C12 c1(NC(C(C)NCC#CC)=O)ccc(S(=O)(=O)N(C)C)cc1Br C1(C(=O)NC(C)Cc2nnc(CO)s2)COCC(C)O1 Cc1ccc(CN2CCN(C(C3CCCCN3S(C)(=O)=O)=O)CC2)c(C)c1 C(=O)(C1=CCCOCC1)NCCN(C(C12OC(C)C(C1)C2)=O)CC1CC1 c1(C(=O)NC2(CC)CCN(C(=O)C=C(C)C(F)F)C2)cc(OC)cc2c1OCC2 CCC(C)(C)C(O)C(=O)NC1(C(N2CCN(CC(C)O)CC2)=O)CCCC1 N1(C(c2ccc(OC)cc2)=O)CCC(O)(C(N2CCOCC2C(F)(F)F)=O)CC1 C(=O)(C(F)CCC(C)(C)C)NC1C(F)CCN(C(C(C)CN(C)C)=O)C1 C1(OC)CC(CO)N(C(=O)COC2(C)CN(C(=O)C=C3CCC(C)CC3)C2)C1 CCC(C(O)C(C)C)NC(C1CCN(c2ccccc2Cl)C1)=O Cc1ccc(F)c(C(N2CC(NC(c3ccc(Cl)s3)=O)CC(F)(F)C2)=O)c1O c1(OC)ccc(C(=O)NCCc2n[nH]cc2C(=O)N(C)CCc2ncon2)cc1 c1(NC(C2C3(CN(C(CCOC)=O)C3)C2)=O)noc2ccc(Br)cc12 CCC(CO)C(=O)N1CC(=C(F)CNC(C2(CCF)CCC2)=O)C1 C=C(C)C(C)(C)C(=O)NC(CNC(c1cnc(-c2cccs2)o1)=O)C(C)C(C)C c1(C(N2CCCC(N(C(=O)CN3CCSCC3)CC)C2)=O)cc2c(ccn2C)[nH]1 N1(C(c2c(C)cn(C)n2)=O)CCN(C(c2ncn3cc(Cl)ccc23)=O)CC(O)C1 C(=O)(C#CC1CCOCC1)N1CC(O)(C(C)NC(C2(C)CCCC2(F)F)=O)C1 c1(C(=O)NCCN(C(c2cc3n(c2)CCCC3)=O)CC)c(N)cccc1[N+](=O)[O-] c1(C(=O)NC2C(NC(C3C(C)(C)C3C(F)F)=O)CC2)ncc(Cl)cc1O CCC(CC(=O)N1CC(CCCC(=O)N(CCCOC(C)C)C)C1)C1CC1 Cc1nc(C(=O)NCCCCn2cc(C3CCCC(O)C3)nn2)sc1C Cc1cccc(Br)c1C(C(=O)NCC1CC2CC1CC2=O)NC(=O)C(F)N(C)C C1(C(=O)Nc2scc(CC(=O)N(c3cn[nH]c3)CC)n2)CCOCC1(C)C CC1CCCN(C(=O)C(=O)NCC=CCNC(=O)CCc2csc(=N)[nH]2)C1 c1(OC)cc(N(C)CC2(C)CN(C(=O)OC(C)(C)C)C2)c(SC)cc1OC C1(C)(C(=O)NC(CC=C)CO)CCCN1C(=O)CCCCN(C)C S(=O)(=O)(c1cccnc1NCCCCC1CCCC1)NC(c1ncc(C)o1)C C(CC(=O)N1C(C)C(=O)C1CC)(CC(C)C)NC(C(COCC)C)=O.OC C1(C2CC2)(C(=O)NC(CCCC)CC)CN(C(=O)C(CC2CC2)OC)C1 n1(CC)ccc2c(C(=O)C(C)=O)cc(C)nc12.c1(CN(C(=O)CO)C)ncc(C)o1 n1(CC)nc(C)c(=NC(=O)c2cccc(NC(=O)C(F)(F)F)c2)[nH]1 N1(C(c2c(C)[nH]nc2Cl)=O)CC2(C1)CN(C(C1CC=CCC1)=O)CCO2 c1(N(CC(Cl)Cl)C)nc(N2CCC(Cc3ccccc3)C2)c2sccc2n1 CCCCN=C1NCC2CCN1C2.c1(NCC2CC2)nc(-c2ccccc2)cs1 c1(C(N2CCC(C3N(C(CC(=C)C)=O)CCCC3)C2)=O)cccc2[nH]c(=N)oc12 c1(C(=O)NCC2N(C(c3c(C)nc(C)o3)=O)CCCC2)cncc(C)c1Cl C=CCC(C(=O)N1C(CNC(C2(CN(C)C)CCC2)=O)CC2CC12)C(C)C C1(C(=O)NCCN(C)C)CC12CCN(C(=O)C(c1ccccc1)O)CC2 C1(N(C(=O)C(C)OC(C(C)(C)C)=O)CC(=O)NC(CC)C)COC(=O)N1 c1(C(N2CCC(OCCOCC(=O)NC3CCCC3)C2)=O)ncnc(O)c1F N1(C(COC)=O)CC2CCC1C1CN(C(=O)CC3(OC(C)C)CCCC3)CC21 N1(CC(=O)N(CC(C)(C)NC(=O)C(C)C(F)F)CCSC)CCCCC1C.CO c1(CC2(CCNC(C3(N(C)C)CCC3)=O)CC2)ncnc2c1COC2 C(C(=O)NC1CCC(F)(F)CC1)(C(C)CC(C)(C)C)N(CCC=C)CC S(=O)(=O)(c1ccc(=NCCSC2CCCOC2)[nH]c1)NC(CCC=C)CO c1(C(C(=O)NC2CCOC2)N(CCF)CC)cccc(C(F)(F)F)c1F c1(C(=O)NCC(CNC(C2C(C(C)C)C2)=O)(C)C)ccccc1CCC(F)(F)F C1(NC(=O)C=Cc2ccc(Cl)cc2)CCN(C(c2ccc(Cl)o2)=O)CC12CCC2 C(=O)(CCCCC(F)F)N1CCC(CNC(C2C(CC)CCC2)=O)C1(C)C N1(C(CCC(=O)NCCC)=O)CCC(C(=O)NCCCc2cncnc2)C1(C)C c1(C(N2C(C)(C(=O)NCCC(CCC)O)CCC2)=O)cc(C)cc(O)n1 C(CC(=O)N(C1CCC1)C(C)C)(C(F)(F)F)NC(Cn1ncc(CC)c1)=O CS(=O)(=O)c1nccc(NC(=O)CCC(=O)N2CCCC2)n1 Cc1cn2cc(C(=O)NCC3CCCC3NC(C3CN(C)C3)=O)cc(C)c2n1 c1(N(C)C)ccccc1C(N1CC(OCC(=O)NC2CC(C(=O)N(C)C)C2)C1)=O Cc1cnc2cccc(C(=O)NCC=CCNC(=O)C(C)OC(C)(C)C)n12 C1(CCC)CCCCN1C(c1cncnc1)=O.c12ccc(cn1)NC2 N1(C(C(CC)(F)F)=O)CCC(NC(=O)CCCSC)C(O)C1 N1(C(C(C)SC)=O)CCC(F)(NC(=O)C(C)NC(=O)NC2CCCC2)C1 c1(SC)cccc(Br)c1CC(=O)NCC(C)(CC(C)C)NC(=O)C(C)O CC1(C)CCOC1C(=O)NC1(C(=O)NC2(C)CCSC2)CCOCC1 CCCCC(O)C(=O)NC1CN(C(c2cc(N)ccc2SC)=O)CC1F c1(C(CNC(=O)C(C)(N(C)C)N(C)C)NC(CC2CC(C)C2)=O)cccc(Cl)c1 Cc1ccc([N+](=O)[O-])c(C(=O)NCC(CNC(c2cnsc2)=O)CO)c1C CCCCC(F)C(=O)N1CCCCCC1C(=O)NC1CCNC(=O)C1 CC1(C)CC(C)(C(N2CCCCC(F)(F)C2)=O)CN1C(=O)C1=NOCC1 Cc1nccc(C(C)Nc2cc(N3CCC(C)(CO)C3)ncn2)n1 C12(C(N3CCN(CCN(C)C(C4(C5CC5)CC4)=O)CC3)=O)CCCN1CC(O)C2 C(C)(CC(C)(C)CO)NC(C1N(C(C(C)C2(O)CCC2)=O)CCSC1)=O N1(C(c2cc(C)nc(O)n2)=O)CCC2CCCN(C(=O)CCN3CCCC3)C2C1 C(=O)(CCCC(=O)N1CC2CC2(NC(=O)C(C)OCC(F)(F)F)C1)OCC N1(C(c2ccc(C(=O)NC3CCCCC3)cc2)C(=O)NC)CCC2(C1)CC(F)(F)C2 c1(CC)cc(C(N2CCN(C(=O)CC(O)CN(C)C)CC2C)=O)ccc1OC c1(CNC(Cc2cccc(OC)c2)C(C)C)cc(C)c(F)c(F)c1 CCS(=O)c1ccccc1C(=O)NC(CCN(C)C(c1cc(Cl)cs1)=O)C(C)C N1(CCNC(N(C(C2CCCOC2)C)CCOCCO)=O)CCCCC1C Cc1nc(Br)c(C(N2CCC(CF)(NC(=O)C(C)C3CC3)C2)=O)s1 N1(C(c2c(OC)oc(C)n2)=O)CCC(O)(CN(C)C(c2cnc(C#N)s2)=O)CC1 CC1CN(C(=O)COc2cccnc2)CC(CNC(c2ccnc(O)c2F)=O)O1 Cc1cnc(F)cc1C(=O)NC(C)CCCCN C(CCCCC(=O)NCc1cnc(C)o1)N(C(C(CC)COC)=O)C c1(NC(C2N(C(c3nc(COCC)sc3)=O)CCC2)=O)ccccc1C S(=O)(=O)(c1ccc(NC(c2ccc(SC)cc2)C)cc1Br)NC(CC(=O)NC)C C=CC1(C(N2CCOC(CNC(=O)C(C)(C)c3cccs3)C2)=O)CCCCC1 C1(NC(c2cc(OC)ncn2)=O)CCN(C(=O)CSCC(=O)N(C)C)C1(C)C C(c1ccc(Cl)nc1)=CC(=O)N(C)CC1CCCN1C(=O)CC1CCCCO1 c1(OC)cc(COCC(=O)NCC2(O)CCN(C(c3cncs3)=O)C2)ccn1 c1(CC)ccc2cc(C(=O)NCC3CC3CNC(c3csc(C#N)c3)=O)[nH]c2c1 CCC(C)C(O)C(C)C(=O)N1CCCC1C1(C(=O)NCc2cc(C)ncn2)CC1 Cc1cccn(CC(N2CCC(NC(c3ccc(C(C)C)o3)=O)C(O)C2)=O)c1=O c1(C(c2nnnn2CCCSC)NCCCC=CC)ccc(Br)cc1OC CC#CCCCC(C(=O)NCCC#N)N(C)CCN1CCOCC1 c1(C(N2C(C3CCN(C(C(CC)SC)=O)CC3)CCCC2)=O)cc(Cl)c(C)cn1 c1(C(=O)NCC(CC)(C)NC(c2n[nH]cc2C2CC2)=O)cccc(COC)c1C CC(C)CCCCC(=O)N1CC(NC(C2C3CN(CC(F)(F)F)CC23)=O)C(C)C1 c1(Cn2c(C(=O)Nc3ccc(CC(=O)NC)cc3)ccc2)cc(F)cc(F)c1 C(CNC(c1cccnc1C)=O)(C(C)C(C)C)NC(Cn1ncc(C)c1)=O N1(C(CC2CC(=O)NC2=O)=O)C2CCC1C(CNC(c1cc(F)c[nH]1)=O)C2 c1(C(=O)O)sccc1C#N.c1(C2CC(OC(C(C)S)=O)C2)ccccc1 CC1C(NC(c2cnccc2Cl)=O)CC2CCC1N2C(c1ncc(Cl)s1)=O C(=O)(CC(CNC(=O)CC(C)n1ccnc1)C1CCC1)N1CC(C)(CC)C1 C1(NC(Cc2c(C)non2)=O)CC2CC(C1)N(C(c1cc3c(s1)CCC3=O)=O)C2 N1(C(c2c(CC)nn[nH]2)=O)CC(NC(=O)C(C)CC#N)C(C)C1 c1(CC(C)NC(C2CCN(C(c3ccc(C)s3)=O)C2)=O)cc(Cl)ccc1Cl C1(C(=O)NC(CNC(c2n(CCC)nc(C)c2)=O)C(C)(C)C)CC2(C1)CC(C)C2 c1(C(=O)NCC(=O)NC)ccc2c(c1)CN(Cc1cccc(OC)c1F)CC2 C=CCN=c1[nH]cc(C(=O)NC2CN(C(=O)COCC(F)F)CC2C)s1 C1(C(N(CCCCNC(C(C)OCC2CC2)=O)C)=O)CCC(=O)N1C c1(OCC)nc(C(=O)NCC(CNC2(C)CCCC2)OC)ncc1C CCC(Cc1ccccc1)CC(=O)N1CC(N(C)C(C2COC(C)(C)CO2)=O)C1 C1(CNC(CCCN(C(C)=O)C)=O)CC2(CC2)CN1C(=O)COCC1CCCO1 C1(NC(=O)CSCCNC(c2sccc2Cl)=O)CCCN2CCCC12 C(=O)(CCCC(C)(F)F)N1C(C(C)C)CN(C(C2CC=CCC2)=O)CC1 C1(NC(C(CC)(O)c2ccccc2)=O)CCN(C(=O)C2=NOCC2)CC1(C)C C1(C)(C(N(CC(C)(C)CNC(c2csc3cncn23)=O)C)=O)CCCNS1(=O)=O C1(CNC(CSCCN(C)C)=O)CN(C(c2conc2C(F)(F)F)=O)C2CC12 c1(CN2C(C)(C(N3CCCC(C(=O)OC)CC3)=O)CC2)cccc2nccnc12 N1(C(C2C(CC)C2)=O)CCC(C2(O)CN(C(c3cc4c(s3)CCCC4)=O)C2)CC1 C=CCCC(F)(F)C(=O)NCC(O)C(=O)NC(CC1CCCC1)CO c1(C(N2CCC(COC)(NC(C3C=CCC3)=O)C2)=O)ccc(Cl)c(Br)c1 C=CC1(NC(=O)C(CNC(=O)C(O)C2CCC2)N(C)C)CCC1 C1(CN(c2n(CC)c(C3COC(C)(C)OC3)nn2)C)CS(=O)(=O)CC1C C1(C(=O)NCCNC(=O)CC2CCC2)CCCN(C(=O)Cn2ncnn2)C1 C12(C(=O)NCC3N(C(C(N4CCSCC4)C)=O)CC3)CCCC1(C(N)=O)C2 N1(C(C(CO)NC(C(C)C)=O)=O)CCC(CO)(CNC(=O)CCS(C)=O)CC1 c1(OCC)ccc(C(=O)NCCNC(c2cncc(C(N)=O)c2)=O)cc1Cl Cn1c(C(=O)NCC(C2CCCCC2)NC(=O)C(F)C2CC2)cc(Cl)c1Cl N1(C(=O)CCn2cc(COC3CCOC3)nn2)CC2CC(C1)C1CCCCN1C2 C1(C(C)C)CN(C(=O)CCF)CCC1NC(c1nocc1Cl)=O C1(OCC)CCCCC1N=c1[nH]c(=NCC(C)(C)S(C)(=O)=O)c2ccccc2[nH]1 n1(CCC)nc(C)c(C(=O)NCCCNC(c2nnn(C)c2CC)=O)c1C c1(C(N2C(CCC(=O)NCCCc3ccncc3)CCC2)=O)ccc(F)nc1F c1(C(=O)NC2C(CNC(C=CC)=O)CCC2)sccc1C#N c1(C(=O)NC2CCC(NC(CCC(=O)NC)=O)CC2)c(F)ccc(Cl)c1N c1(CNC(=O)C(O)C2CN(C(=O)CC3CCCSC3)C2)ncccn1 C1(CCNC(=O)COC2CCCC2)CCCN(C(c2ccsc2)=O)CC1 C(CCN=C(NC1CC(N(C)C)C1)NC1CCCC(C(=O)OC)C1)OC C(=O)(C1CN2CCc3ccccc3C12)N1C(C)CN(C(C2(CO)COC2)=O)CC1 N1(C(C(c2cnn(C)c2)C)=O)CC2CC(O)C1C2NC(c1snc(O)c1Cl)=O CCCC(C)CC(=O)N1CCCC(CNC(C2(C(F)(F)F)CCO2)=O)C1 N1(C(c2cnc(C)nc2)=O)CC2(C1)CN(C(C1CC1(C)Br)=O)C2 O=C(C1=COCCC1)NC1CC(F)CN(C(c2cc(O)nc(O)n2)=O)C1 N1(C(C(CCN(C)C)N(C)C)=O)CC(N(C)C(c2cnccc2Cl)=O)C2(CC2)C1 c1(CC)nc(C)c(C(=O)NC(C2CCCC(C)C2)CC)o1 c1(CC(N2CC=C(CNC(C)=O)CC2)=O)ccc2c(c1)COCC2 Cc1c(Cl)cnn1CC(=O)NC1CC1CNC(=O)CCCc1cncs1 N1(C(C(C(C)O)N(C)C)=O)CC2CC(C1)C2NC(C1CCCO1)=O C1(C(=O)NC2CCC(OC)C2)COCCN(C(=O)COC2CC2)C1 c1(NC(C(=O)NC2CCCN(C(=O)OCC)C2)=O)cccc(C#N)c1Br C1(OC)CC(NC(c2c[nH]nc2C2CCCO2)=O)CN(C(c2occc2C)=O)C1 C(=O)(C1=CC2CCCCCC12)NCCN(C(CSCCCC)=O)C1CC1 C(=O)(C(CN)C(C)(C)C)N(C)CCN(C(=O)COCCCF)C c1(C(=O)NC(C(=O)NCC(C)OC(F)F)CCF)cc2ccccc2[nH]1 N1(C(c2nc3c(s2)CCC3)C)CCN(C)CC1c1ccccc1C(F)(F)F N1(C(C(c2cccc(C)c2)=O)=O)CCc2ccccc2C(NC(C(C)(C)C)=O)C1 c1(NC(=O)CC2(CNC(=O)Cn3cnnn3)CC2)cncc(F)c1 c1(C(N2CC(NC(C=C(COC)C)=O)C(C)(C)C2)=O)cc(N)c(C)c([N+](=O)[O-])c1 C=CCCCCC(=O)N1CCCC1(C(=O)NC)CCc1ccccc1 N1(CCC(=O)NC2(CNC(C3CCCO3)=O)CCCC2)CCCCC1=O CCS(=O)(=O)c1cccc(C(=O)N=c2ccc(-c3ccccn3)n[nH]2)c1 C(=O)(C(O)CC(N)=O)N1CC(C(N2C(CC)(CC)CC2)=O)C(C(C)C)C1 N1(c2ncc(C(=O)OC)nc2)CCCC2(NC(C3(C)CCC(=O)N3)=O)CC2C1 c1(C(N2CCC(C(C)NC(C3(CO)CCC3)=O)CC2)=O)ccc([N+](=O)[O-])cc1F N1(C(CC(C=C)C)=O)CCN(C(=O)COc2cccc(C(N)=O)c2)CC(C)(C)C1 C(CN(C)N1CC(C(N)=O)N(C)CC1)Cc1ccc(OC)cc1.OC c1(C(=O)NC2C(NC(C(CC(C)(C)C)OC)=O)CC2)cccc2nn(C)cc12 c1(CC(=O)N(CCN(C(=O)CCc2cccn2C)CC)CC)cc(F)ccc1Cl c1(C(N2CCCC2C2(C(=O)NCc3cccc(O)n3)CC2)=O)cc(O)ncc1F CCCCC(C)C(=O)N(C1(C(=O)OC)CC1)C(C1CCCC1)C1CCC1 c1(C(=O)NCC2N(C(C3CCC(=O)NC3)=O)CCC2)c(F)cc(F)cc1Cl C=CCC(CNC(c1nonc1N)=O)C(=O)NCc1ccns1 CN1C(=O)CC(C(N2CCCC(CN(C(=O)CC3CC=CC3)C)C2)=O)NC1=O CCC(CCCC(=O)N1CCC(SCC)CC1)NC(=O)CC(=O)OC(C)(C)C c1(CC(C)NCC2(OCC)CS(=O)(=O)C2)ccc(Cl)cc1Cl N1(C(c2n(C)ncc2)=O)CCC(C2CC2)(CNC(C2CC(=O)N(C3CC3)C2)=O)C1 C1(NC(=O)C(F)F)CCN(C(=O)Cc2cnn(Cc3ccccc3)c2)CC1CO O=S(=O)(c1cccnc1)N1CC2(CC(NCc3c(F)cc(Cl)cc3Cl)C2)C1 CCCCCCCCCC(=O)N1CCN(C(=O)CN(C)CCC)CCC1C CC1CC(C(=O)NC(C)(C)CNC(c2cc(-c3cnn(C)c3)[nH]n2)=O)=NO1 c1(NC(=O)NC2CCN(CC#N)C2)ccc(C(F)(F)F)nc1 c1(C(=O)NCC(C)NC(C2CCC(=O)O2)=O)cnn2cccc(Cl)c12 c1(C(=O)NCCOCCOCCF)cscc1C(=O)O N1(C(C2C(Cl)(C(=O)OCC)C2)=O)CC2CN(C(=O)CCF)CC2C1 c1(C(C(=O)NCCCN(C)C(C2CCCC2CF)=O)(C)C)ccc(Cl)cn1 c1(CNC(C(C)C)=O)cn(C2COCC2CNC(=O)COC(F)(F)F)nn1 C(=O)(CC(C(F)(F)F)N(C)C1CC1)NCC(CC=C)NC(c1ccn(C)c1)=O Cc1nc2c(F)cccc2cc1C(=O)NC1(C2CN(C(C3CCCO3)=O)C2)CC1 N1(C(C2(CC#C)CCCC2)=O)CCCCC(CNC(=O)CC2CC=CCC2)C1 Cc1ccn2ncc(C(N3CC4(C3)CN(C(=O)CC3CCC3(F)F)C4)=O)c2n1 c1(CC)cc(C(=O)NCCN(C(=O)CCC2CCC(O)CC2)C)nn1C C(=O)(C1=NOC(CC2(O)COC2)C1)NCC1CCCN(C(Cc2c(C)scc2)=O)C1 c1(C(N(CCC(C)(F)F)C)=O)ccc(C2CC2)cc1 CC(C)(C)C(CC(=O)NCC1OCCC1(C)C)NC(=O)CSCC(F)F N1(C(c2c(=O)ccn(C)c2)=O)CC(CNC(C2CC3CC2C3)=O)CC12CCC2 CCC(C)C(CC(=O)NCC(C)(C)N(C)C)NC(c1ccnc(C2CC2)c1)=O c1(C(C)=O)cc(C(=O)NC2CCC2CNC(c2ccon2)=O)n(C)c1 c1(CNC(CC(CC)NC(c2ccc(Cl)s2)=O)=O)cc(F)ccc1F C(N=c1[nH]c(=NCCCn2cc(Br)cn2)[nH]c2c1CSC2)C1(OC)CCCCC1 c1(C(N2CCN(C(C3CCC(CC)CC3)=O)C3C2C3)=O)cc(O)c(O)c(O)c1 CN1N=C(C(=O)N2CCC(F)(CNC(c3cccc4c3OCC4)=O)C2)CCC1=O CS(C)(=O)=NCC(=O)N1CC2CC1C2NC(c1nc(C2CC2)ncc1Br)=O O=C(N=c1cc[nH]cc1O)C1CC=CCC1NCc1nc(-c2ccccc2)no1 C1(NC(CC(CC)C2CCC2)=O)C2CC1CN(C(=O)CC1(C)CCS(=O)(=O)N1)C2 c1(C(=O)NCC2CC(O)(CCNC(C(CC)=CC)=O)C2)cccc(NC(C)C)c1 c1(CCCC)ncc(C(=O)NCC(c2ccccc2)NC(=O)C(O)CN(C)C)s1 Cc1c(C(N2CC(CNC(c3ccc(C(N)=O)cn3)=O)C(C)C2)=O)nnn1C c1(CCC(N2CCC(F)(CNC(C3(N(C)C)CC3)=O)C2)=O)ccc(Cl)c(F)c1 CC(C(C)C(=O)N(C)Cc1nccs1)NC(=O)CCC1CCCOC1 CCCCCC(C)CC(=O)N1CC(N(C)C)(CNC(=O)CC(C)CC(=O)OC)C1 C12(NC(Cc3nc(C(C)C)sc3)=O)CCN(C(c3ccc(F)cc3Cl)=O)CC1C2 Cc1cc(O)ccc1N(C(=O)CC=CCNC(=O)C=CC(C)(C)C)C CC1CCc2sc(C(N3CCCCC3CNC(=O)Cc3cnnn3C)=O)cc2C1 N1(C(c2cc(OC)n[nH]2)=O)CCOC(CCNC(=O)C=CC=C(Cl)Cl)C1.C1CO1 C1(C(=O)NC(C)CNC(c2coc(Cl)n2)=O)CCCCC1OCc1ccccc1 N1(C(CC(C=C)C)=O)CCC2CCC(NC(c3cc(CC)cc(Cl)c3)=O)C1C2 N1(C(=O)Cc2cc(Br)ccc2F)CC2CN(C(C3(C4CC4)CC3)=O)CC2C1 C(F)(F)(C(F)(F)F)c1cc(NCC(=O)N(C)Cc2ccncc2)no1 c1(CC(=O)N(C(C)CCNC(=O)C#CC2CCC2)C)cc2ccccc2oc1=O N1(C(C2CC(CC)OCC2)=O)CCCC(C)C1CNC(c1cc(C)ccc1N)=O c1(C(=O)NC2CC(CCNC(CC=C)=O)C2)cnn(C(C)C)n1 N1(C(CN2CC(C)C2)=O)CC(NC(=O)C=Cc2ccc(C(N)=O)cc2)C(C)(C)C1 c1(C(N2C(C)(C(=O)Nc3c(OCC)c(F)ccc3)CC2)=O)cc(C)cc2[nH]ccc12 C1(NC(Cc2cccc(C)c2Cl)=O)COC2(C1)CN(C(C1CC3C=CC1O3)=O)C2 c1(C(=O)NC(CCCC)CO)cc(-c2cnc(C#N)c(F)c2)c2cn[nH]c2c1 C12(NC(C(C)C3CCCC3)=O)CCCN(C(=O)C(c3ccccn3)O)CC1C2 c1(CC)ccc(C(=O)NCCC2CC(NC(c3cnccc3C(F)F)=O)C2)cc1 c1(C2(NC(=O)NCCN(C3(C(N)=O)CCOC3)C)CCC2)ccc(Br)cn1 C=CCCCC(C)(C)CNC(C1CC(=O)CN1C(C1CCC(=O)N(C)C1)=O)=O C1(NC2C(CC)CC2)CCC(C(=O)OC)C1 c1(C(=O)NCC(CC)NC(=O)C(CC(C)C)OC)[nH]c2cc(F)ccc2c1C N1(C(c2nc(CNC(C=CC(C)(C)SC)=O)oc2)=O)CCn2ncc(C)c2C1 CC1CCN(C(c2c(F)cncc2Cl)=O)CC1CNC(C1(c2cccnc2)CC1)=O C1(C(=O)NC2(CNC(C=CC(C)=O)=O)CCC2)CNC(=O)CC12CCC2 C1(CNC(CCNC(C)=O)=O)CC2CC2N1C(c1ccsc1C)=O CN1CCC(C(=O)NCC2(C(=O)O)CC3(CC3)C2)S1(=O)=O C1(C)(NC(C(C)O)=O)CCN(C(=O)CN2CCC(N(C)C)C2)CC1 N1(C(C(CO)N(C)C)=O)CC2CC1C2NC(=O)C(c1cccc(Cl)c1)(F)F C(C)(CNC(=O)CN(C)C(C1(OC)CCCC1)=O)(CO)OC c1(C(N2CCCC(CCC)(NC(c3coc(Cl)c3)=O)C2)=O)cccc2nncn12 N1(C(c2cc(NC(=O)OC(C)(C)C)ncn2)=O)CCC(C2CC2(F)F)C1 c1(CCNC(c2nnnn2C2CCCC2)CCOC)ccc(OC)c(OC)c1 C1(CNC(C2CCC2)=O)CC2(CCN(C(C3OC4CCC3CC4)=O)CC2)CO1 C(=O)(C1=C(C)OCCS1)NCCCC(C)NC(C(C)OCCC=C)=O c1(CC)nc(C)c(C(=O)NCCCN(C(=O)CN2CC3CC3C2)CCSC)o1.C1(S)CC1 N1(C(c2ccc(CC)s2)=O)CC(C2CCN(C(C3(c4ccsc4)CC3)=O)CC2)C1 N1(C(c2ccc(OCC=C)c(OC)c2)C)CCc2nccc(N)c2C1 c1(C(=O)NC(C)(C)CNC(=O)CC2(O)CCCCCC2)ccc(P(C)(C)=O)s1 C(=O)(CCCCC(=O)OCC)c1c(Cn2cc(C(C=C)(C)O)nn2)c(F)ccc1 c1(C(=O)NCC(C)N(C(=O)C(C)n2cncn2)C)cc(S(N)(=O)=O)c(Cl)cc1Cl C1(NC(c2c(C)cco2)=O)CCN(C(c2cnc(S)n2C2CC2)=O)CC1F c1(CN(C(=O)OC(CCc2ccc(C(C)=O)s2)=O)C2CC2)ccc(F)cc1 Cc1cc(CNC(=O)C(C2CCCCC2)O)oc1C(=O)NC1(CCF)CCC1 c1(C(=O)NCC(O)CNC(C2CCC(C(F)(F)F)C2)=O)cc(F)cc2ccncc12 C(=O)(CC(O)C(C)C)N1CC(OCCC)C(NCc2ccc(C(=O)OC)cc2)C1 N12CCC3(CC1)OCCc1sc(cc13)C2=O.c1(CCSCC(C)=O)cccs1 c1(C(=O)NC(CCCCNC(C2CC(SC)C2)=O)C)cncc2ncn(C)c12 N1(C(C(c2cn(C)nc2)=O)=O)CCC2(CC(NC(=O)CN3CCC(O)C3)C2)C1 N1(C(CCC=CC(C)C)=O)CC2CCN(C(C3CN(C)CCO3)=O)CC2C1 C1(NC(c2cnn(CCC)c2C)=O)CN(C(=O)C(C)(O)CCC)CCC12CCC2 N1(C(c2c(C)nccc2Cl)=O)CCCN(C(=O)Cc2csc(S)n2)C(C(C)C)C1 Cc1ccc(S(=O)(=O)NCCC(=O)NCc2cccc(-n3cncn3)c2)c(F)c1 CC1(CNC(c2cccnc2)=O)COCCN(C(C2CCCS(=O)(=O)C2)=O)C1 c1(C(=O)NCC(C2CCC2)NC(=O)CCc2cc[nH]n2)ccc(Cl)c(Cl)c1 C1(CNC(=O)CC2CCC(=O)O2)CC2CCC1N(C(c1c[nH]cc1Br)=O)C2 CN1CCCC1CCC(=O)NCCOC1CCN(C(=O)CC2CC=CC2)C1 N1(C(C(C(=O)OC)C)=O)CCCC(O)(C(=O)NCCC2(COC)CCC2)C1 O=C(C1=CCCCC1)NC(CNC(=O)C=C1CCOCC1)C1CC1 C(=O)(C(CC(C)SC)N1CCCC(C)(CCC)C1)NCC(=C)C C(=O)(C(F)(CNC(=O)C1=CCCCCC1)C(C)C)NCc1onc(CC)n1 c1(C(=O)NCC(CCOC)NC(C2CN(C)C2)=O)cc2c(s1)CCCC2 c1(NC(C(C)NC(=O)NC(C2COCCO2)C)=O)ccc(F)cc1 C1(COC(C2(C(C)=O)CC2)=O)CCCC2(CCC2)O1 C1(F)(CNC(c2cnc(C(C)(C)C)[nH]2)=O)CCC(NC(C2CCCCO2)=O)C1 C(=O)(C1(C)CC(C(C)C)c2ccccc21)NCc1c(C(=O)OC)cccc1F C(C)(N=c1nc2sccc2c(N2CCC(CCF)CC2)[nH]1)c1c(C)noc1C N1(C(CC2(OC)CCC2)=O)CCCC(NC(c2cc(C(N)=O)[nH]n2)=O)CC1 CC1CSCCN1C(=O)NCCC1(C)OCCO1 N1(C(C2(CCOC)CC2)=O)CCCC(O)(CNC(c2cccc(N)c2F)=O)C1 c1(NCC)ccc(OC(F)F)c(F)c1.C(CC(=O)N(CC(C)C)C1CC1)(OCC)OCC C(=O)(CCC(=O)N(C)C)N(C1CCN(C(c2cccc(C(C)(F)F)c2)=O)C1)CC CC1(C#CC(=O)NCCC2(C)CCN(C(c3cccc(F)c3O)=O)C2)CCCO1 C(=O)(C(C)C(=O)N(C1CCN(C(=O)CN(C)C(N)=O)CC1)CCO)OC C1(C(=O)NC(C#C)CO)CCn2cncc2C1 c1(CC2CN(C(C(C)Oc3ccccc3)=O)C(C)C2)ccccc1[N+](=O)[O-] C=C(Cl)CCC(=O)N1CC2CC1C2NC(=O)Cc1csc(C2CC2)n1 c1(NCC2N(C)CCN(c3ccc(C(F)(F)F)cn3)C2)csc2ccc(Cl)cc12 c1(COC(C2CCCC(CN)O2)=O)nc2ccccn2c(=O)c1Br C1(OC)CCN(C(C2(CCNC(=O)C(O)C(C)(C)C)CC2)=O)CC1C Cc1cc(N)cc(C(N2CCC(OCCO)CC2)=O)c1F c1(C(N2CC3CC(OCC)C3C2)=O)[nH]nc2c1CCC2(C)C N1(C(CCCn2cc(C3N(C)CCC3)nn2)=O)CCC12CCN(C)C2 C(C1=CCN(C(c2c(C(C)C)n[nH]c2C)=O)CC1)NC(C(C(C)C)SC)=O N1(C(C)=O)CCCC1CNC(C12CC(C)(C1)C2)=O C(=O)(C1=COCCC1)NC(C(=O)N(C)Cc1cc(C)nn1C)(C)CO C(c1cccc([N+](=O)[O-])c1)=CC(=O)NC1CC1C(=O)NCc1cccc(O)c1 c1(C(N2CC(CNC(COCC#C)=O)OCC2)=O)cnc2[nH]c(C)nc2c1 C(CCCCC(=O)NCC1CN(C(=O)C(C)NC=O)CCO1)OC C1(NC(c2ccc(C(N)=O)cn2)=O)CCCCN(C(c2ccnn2CCF)=O)C1 N1(C(c2c(C)scc2)=O)CCC(N(C)C(c2ccc(C(F)(F)F)s2)=O)C(C)C1 C(=O)(C(CC(C)(C)C)NC(=O)C=CC1CCCCC1)N(C1C(C)COCC1)C C1(OC)CC2CC(OC)CC12.c1(C(=O)NCn2cc(C)nn2)ccc(C2CCC2)cn1 CN=S(C)(=O)c1ccc(C(=O)NCC(C)N(C)C(c2ocnc2C)=O)cc1 C1(NC(C(CC)OC)=O)CCCCN(C(=O)C(C)(C)C(=O)c2ccccc2)C1 c1(CN2C(C(C)C(N)=O)CCC2)ccc(F)nc1 C1(NC(C2CCN(CC)C2)=O)(CC)CCCN(C(c2ccn(C(C)C)c2C)=O)C1 N1(C(c2n(C)ncc2)=O)CCN(C2CN(C(=O)CCC3NC(=O)NC3=O)C2)CC1 C1(C)(CNC(Cc2nc(C)oc2)=O)CCCN1C(=O)CC1CCCCC1 Cc1nc(C(=O)N(C(C)CNC(c2c(-c3ccccn3)noc2C)=O)C)c(C)o1 C1(NC(CSC)=O)CCSC12CN(C(=O)C(C)Cc1ccc(F)cc1)C2 C=CCCC(C(=O)NC1(CNC(=O)C2=CCCOC2)CC1)c1ccccc1 c1(C(=O)NCCC2OCCN(C(C3C(C)(C)CCC3)=O)C2)cc(Cl)cc(Cl)c1F FC1(F)CC12CCC(NCCN1CCC(C3OCCO3)CC1)CC2 N1(C(c2n(C)nnc2CNC(=O)CCNC(=O)C2CC2)=O)Cc2ccc(O)cc2C1 c1(OC)c(Cl)cc(NC(=O)Nc2cn(C)nc2C(F)(F)F)cc1Cl c1(COC)cc(NC(=O)CNC(C)C(c2cccc(O)c2)O)ccc1F c1(C(N(C2CCN(C(=O)C(c3ccccc3)O)C2)C)=O)ccc(C(F)F)c(Cl)c1 N1(C(C(C)CC2CCC2)=O)CC2(CCCC2)C1C(N1CCN(CCO)C(=O)C1)=O C(C(O)C(=O)NCC1CCCS1)NC(c1cc(Cl)n[nH]1)=O C1(CNC(c2c(C)ccnn2)=O)CN(C(c2coc(CO)c2)=O)CCC1C C1(C(=O)NC(CC(C)(C)C)c2ccc(F)cc2)CCCC(F)(F)C1 C1(C(=O)NC2(CC=C)CCOC2)CCCN(C(=O)C(CC2CCC2)OC)CC1 c1(C(=O)NCC2N(C(C=CCOCCOC)=O)CCOC2)coc2c(C)cccc12 c1(N2CC(OCCNC(c3c(OC)cc(O)nc3)=O)C2)c(Cl)nc(SC)nc1Cl C1(C(N2C(C(=O)NCC(N(C)C)C3CC3)CCC2)=O)CCCC(=O)C1 N1(C(c2c(CC)non2)=O)CCN(C(=O)COc2ccc(C(C)C)cc2)C(C)C1 Cc1csc(CNC(C2CC2CNC(C2CCC2)=O)=O)c1 N1(C(C=CCSC)=O)CC2CCN(C(c3ccc(Br)c(OC)c3)=O)CC2C1 N1(C(c2cc(Cl)nn2C)C(=O)NCCOC)CCN(C)C2CC12 N1(C(C2CCN(C(c3c(C)nns3)=O)C(C)C2)=O)CCC12CCCOCC2 N1(C(CC=CC=C)=O)CC(C)(C)CC1C(N1CC(C(=O)OC)(OC)C1)=O N1(C(CCSCCOCC)=O)CCC2CC12CNC(=O)Cn1cc(CO)nn1 CCC(CNC(C1CC1(F)Cl)=O)(CC)NC(c1cncn1C)=O C1(NC(Cc2cc(OC)no2)=O)CC12CCN(C(C1CC1F)=O)CC2 c1(NC(C(=O)NC(C)CCCOc2cccnc2)=O)cnc2ccnn2c1 Cn1cc(SC=CC(=O)N2CC(C(CCCO)NC(=O)CC3CC34CC4)C2)cn1 CC(C)(CC(=O)NC1CCC1NC(c1c[nH]nc1C(C)(F)F)=O)CC(F)F C=C(C)CC(C)C(=O)N1CCCC(CNC(=O)CCCOc2ccccc2F)C1 c1(C(N2CC(NC(C(C)OC)=O)C(CO)CC2)=O)c(O)ccc2ccccc12 c1(NC(=O)NCC2C(C#N)CCC2)ccnc(Cl)c1Br c1(N2C(C(=O)NC3(N(CC)CC)COC3)CCC2)cc(C(F)(F)F)nc(Cl)n1 N1(C(COCC=C)=O)CCCC(F)(CNC(C2(C)COC(=O)C2)=O)C1 c1(C(=O)NC2CCN(C(C3(F)C(C)OCC3)=O)CC2)c(C(F)(F)F)cc[nH]c1=N C(C(C)(C)C(=O)NC1CCOCC1NC(=O)CC1CNC(=O)O1)SC N1(C(c2c(SCC)n(C)nc2)=O)CC2CCN(C(=O)Cc3cc(C)no3)C2C1 CCN=C(NCC(=O)N(C)OCC)NC(c1ccc(Br)cc1)CF N1(C(c2c(C)scc2)=O)CCC(O)(CCNC(C2C(C)C2C)=O)C1 c1(C(N(CC(CNC(C2(C=C)CCC2)=O)(C)C)C)=O)ccc(O)c(Cl)n1 C1(CNC(c2c(C)scc2)=O)CC2CCC1N(C(=O)COCCOCCO)C2 c1(C(N2CCC(O)(C(C)C)C2)C(=O)NC2COC2)cccc2sccc12 c1(C(=O)NCC(CN(C(CC(=O)OCC)=O)C)C)cc2n(n1)CCN(C)C2 C1(C(=O)NCC(C)CNC(c2ccnn2C)=O)CCCCC1C C(=O)(C(C)(CNC(=O)CSC(F)F)CC)NC(CCC)C(=O)N(C)C C(c1ccncc1)=CC(=O)NC1C(NC(C2N(C)CCC2)=O)CCC1 c1(CNCC2N(C(C3CC(O)C3)=O)CCOC2)ccc2c(c1)Cc1ccccc1-2 C(=O)(CCCCCCNC(C1CC1COC)=O)NCC(=O)NCCC Cc1cn(CC(=O)NC2CCN(C(c3cnc(S)nc3)=O)C2C)c2ccccc12 c1(C(=O)NCCCCN(C)C(C2CC=CCC2)=O)cncnc1-c1ccccc1 C1(NC(C2C(CCOC)C2)=O)CCN(C(=O)Cc2c(F)cccc2Cl)C1(C)C C(=O)(C1=CCC(C)CC1)NCCOCCCNC(c1c(C)cccc1)=O c1(C(=O)NCC(CC(=O)NC2CC2CF)OC)c[nH]nc1-c1ccoc1 c1(OC)cc(C(=O)NCC2(NC(c3ccc(C)[nH]3)=O)CCCCC2C)ccc1F Cc1c(NC(C2(CC3(C#N)CCOC3)CC2)=O)cccc1Cl N1(C(=O)OC(C)(C)C)CCC(NC(=O)CC2CC2(C)C)C(C)(C)C1 CCCC(Cl)C(=O)N1CCC(N2CCNCC2)CC1 C1(S(C)(=O)=O)(C(N2CC(C(C)NC(C(CC=C)OC)=O)OCC2)=O)CCC1 Nc1ccc(C(N2C3CCC(C3)C2CNC(c2cc(Cl)no2)=O)=O)cc1F N1(C(C2(C)C3Cc4ccccc4C23)=O)CC2(CC(Cn3ccnc3CO)CO2)C1 c1(OC)cc(O)ncc1C(N1CCC(NC(=O)C=Cc2cc[nH]n2)C1(C)C)=O Cc1ccnc(C)c1C(N1CC=CC1C(=O)N(CCC1CCCC(C)(C)C1)C1CC1)=O c1(C(N2CC(C)C(NC(C3(c4cccnc4)CCC3)=O)C2)=O)cnc2n1CCC2 C1(CC(=O)NC(CO)CCCNC(=O)C(F)CC2CCOC2)CCCCC1(F)F Cc1cc(F)c(NC(=O)C(=O)NCC(C)CSc2ccccc2)c(I)c1 CCC1=NOC(CC(N2CCN(C3CN(C(=O)Cn4nnc(=N)[nH]4)C3)CC2)=O)C1 C1(C#N)(CNC(C2CCCCC2)C#C)CC2CCC1CC2 Cc1c(NC(C2CC2c2cccnc2)=O)n[nH]c1C1CC1 C1(CNC(CC2CCC(C)C2)=O)COCCN1C(c1cccc(C(F)F)n1)=O C(=O)(CC1=NN(C)C(=O)C1)CCOC.N12CCCC(C1C)CNc1ccnc2n1 CC#CCCC(=O)NC1CCC(CNC(C2CCN2C(C)(C)C)=O)CC1 C#CCCCCCCC(=O)NCC(O)CN(C)C(c1ccc(P(C)(C)=O)s1)=O C1(NC(C=CC(CC)=CC)=O)CC2(C1)CC(NC(=O)C(N1CCSCC1)C)C2 C1(CC=C)(C(=O)N(CCCN(c2nccc(-n3ccnc3)n2)C)C)CCOCC1 Cc1ccc(F)nc1C(N1CC2(CC2C(N2CC3CCC2C3)=O)C1)=O N1(C(=O)CC2CCCCCCC2)CCC2CCN(C(=O)CCc3nncs3)C2C1 C(=O)(CS(=O)(=O)CC(C)C)N1CCC(OCCNC(c2n[nH]c(C)c2C)=O)C1 Cc1csc2c(N3CCC(C(=O)NCC(=O)NC4CCCC45CC5)C3)ncnc12 C1(NC(=O)CC2CC2)CCN(C(c2cnc(C3CC3)nc2O)=O)CCC1CO Cc1cc(C)c(C(N2CCC(NC(c3nncn3C)=O)C(F)C2)=O)c(=O)o1 C(=O)(C(O)C(F)(F)F)NCCN(CCOC)C(c1cc(C(C)(C)C)n[nH]1)=O N1(C(=O)CCc2cccnc2Cl)CC(CNC(=O)C(O)CC2CC2)C2(CC2)C1 c1(OC)ccccc1C(N1CCC(C(CO)NC(c2[nH]c(C)cc2C)=O)CC1)=O N1(C(C=CC)=O)CCC2(CC1)CCN(C(=O)C(c1ccn(C)n1)C)C2 N1(C(CNC(CCCC)=O)=O)CCN(C(c2csc(CC)n2)=O)CC1C1CCC1 Cc1nc(N)cnc1C(=O)NCC1CCCCN1C(c1cc(C(C)C)n(C)n1)=O c1(SC)cc(C(N2CC3(CCN(C(C4(C(N)=O)CC4)=O)C3)C2)=O)c(Cl)cc1Cl CCC(CC(=O)NCCN1CCN(C(C2CCCCNC2=O)=O)CC1)C(C)C N1(C(C2CN(C(COCCCC)=O)CC23CC3)=O)CCN2CCCCC1C2 CC1(C)CC(CNC(c2ccsn2)=O)CN1C(c1coc(O)n1)=O Cc1ccc(C(N2CCCC2C2CCN(C(c3csc(Cl)c3)=O)C2)=O)nc1 C1(CC(N2CCC(CNC(C3(C4CCC4)CC3)=O)C2)=O)CCC2(CC1)CC2 c1(C(N2CCC(C(C)NC(c3n[nH]cc3Cl)=O)C2)=O)ncsc1S(N)(=O)=O n1(CCCOC)nc(-c2ccccn2)nc1C(C)Cn1ccnc1 c1(C(=O)NCC2(COC)CN(C(c3nc(C)nn3C)=O)C2)cnn(C)c1N C1(C(=O)NCCC2(O)CCN(C(c3n(CC#N)ncc3)=O)C2)CCC(F)(F)CC1 CN1N=CC(CC(=O)NCC(C)(C)C(=O)NCC2CC(C)(O)C2)C1=O C(=O)(CCCCCNCCOc1cc(C)on1)NCC1N(C(C=CC)=O)CC1 C1(NC(=O)C=Cc2cccs2)CS(=O)(=O)CC1NC(=O)C(F)(F)c1ccncc1 c1(CC)ccc(OC)cc1.N12CCCC1CC(=O)NC1(CC1)CNC(=O)C=CC2 c1(C(=O)NC2C(NC(CNS(N)(=O)=O)=O)CCC2)ncn2ccccc12 Cc1cc(Cl)ccc1C(=O)NC1CN(C(c2cc(Cl)on2)=O)CCC1C c1(C(=O)NC2CCN(C(C3C(CN(C)C)C3)=O)C2)cccc2c1OCC2 C(CNC(C1CCCC(O)C1)=O)(C(C)(C)C)NC(c1[nH]cc(C(C)=O)c1)=O C(=O)(CN=c1[nH]c(=NCC2CCCCO2)c2[nH]ccc2[nH]1)N1CCN(C)CC1 C(=O)(C(C)(C)CC(=O)NCC1CCN1C(=O)CCCCc1cnc[nH]1)OC c1(C(N(C(C2CCOC2)CNC(=O)CC(=O)OC(C)(C)C)C)=O)ccc(F)cc1Cl CON1CCC(C(N2CCC(O)(C(C)NC(=O)C(=CC3CCCC3)C)C2)=O)CC1 Cc1cc(C=CC(=O)NC(C)CN(C)C(C2CCC3(CC2)CC3)=O)c[nH]c1=N c1(OC)cc(=O)n(C)cc1C(=O)NCC1(C)CCCN1C(=O)C=C1CCN(C)C1 N1(C(c2c(NC(C)=O)c[nH]c2C)=O)CC2CN(C(=O)CC(C)(C)O)CC2(C)C1 C(C)(C)(CC(=O)NCc1nc(CNC(C2CC(C)CO2)=O)cs1)OC c1(NC(CCNC(C(=Cc2cnc[nH]2)C)=O)C)nc(Cl)nc2c1ncn2C(C)C O=C(C1=C(Cl)CCOC1)N1CCCCC1C1CCN(Cc2ccnc(Cl)c2F)C1 CC(O)(CNC(c1coc(CNC(=O)C=C2CCCCC2)n1)=O)C(F)F c1(C(N2CCN(C(C3(C)CCC(=O)N3)=O)CC2CF)=O)ccc(F)c(Cl)c1F C1(C(=O)NC(C)(C)COCCCNC(C2CCSC2)=O)CCCOC1 C=Cn1nccc1C(=O)NC1CCN(C(=O)CCCOCC)C1C(C)C Cc1cccnc1C(N)C(N1CCOC(CF)C1)=O c1(OC)coc(C(N2CCC(C(C)(C)NC(C3NC(=O)C4CC34)=O)C2)=O)cc1=O C=C(Cl)C(C)(C)C(=O)N1CCCC(N(C(=O)C(F)(F)C(C)O)CCC)C1 c1(OC)cc(Br)ccc1CC(=O)NC1CN(Cc2cc(Br)ncc2F)CC1C#N C1(CC)CCC2CN(CCC(c3ccccc3)O)CC12 Cc1ccc(C(=O)NCCOC2CCN(C(C3CC(=O)CS3)=O)C2)n1C c1(C(=O)NCCN(C(CC=C)=O)CCCN(C)C)cc(Cl)cc([N+](=O)[O-])c1O c1(C(=O)NCC(n2cc(C3CCC3)nn2)C)nc(O)nc(O)c1F C1(NC(CCC#C)=O)CC2CC(C1)N(C(=O)C(CC(F)F)c1ccccc1)C2 Cc1cc(C#N)cnc1C(N1CCC(C2CCCN2C(=O)C=C2CCC2)CC1)=O N1(C(C2CCC(CC)O2)=O)CCCC(C)C1CCNc1ncc(F)cn1 CC(CS(C)=O)C(=O)NCCC1(NC(=O)CCOCc2ccccc2)CC1 Cc1nc(C(C)(C)C)sc1C(=O)NC1CCN(c2ncc(Cl)cn2)C1C c1(C(=O)NCC2CCC(F)(CNC(C3(C)CCC(=O)C3)=O)C2)cnn2c1CCC2 N1(C(C)C(=O)NC(CC(=O)Nc2ccco2)C2CC2)CCC(O)CC1 c1(C(c2nnnn2C)NC2CC(C)C2)cccc(C2CC2)c1F c1(C(=O)NCc2c(C(N(C3CC(SC)C3)C)=O)cco2)ccc2c[nH]nc2c1 N1(C(C)=O)CCCC(NC(=O)CCS(=O)(=O)Nc2cnn(C)c2)CCC1 CN1C(=O)CCC1CC(=O)NCC1(F)CC(CNC(=O)Cc2ccccc2Cl)C1 C(CC(C)N=c1[nH]c(=NCc2cnn(CCF)c2)[nH]c2c1CCCC2)OC C(C(C)(CC(C)C)NC(=O)COC1CCC1)NC(c1cc(C(C)=O)sc1C)=O C1(CNC(C(CCC#C)O)=O)CN(C(=O)CCNC(=O)CO)CC12CCOCC2 C12(NC(C(CC=C)C)=O)CCCC1(F)CN(C(c1cc(OC)cc(OC)c1)=O)C2 Cc1occc1CC(=O)NC1CCN(C(C2(C)CSC2)=O)C1 c1(C2N(C(C3C(P(C)(C)=O)CCC3)=O)CCC2)ccc2cnccc2c1 c1(CC)nc2sc(C)cn2c1C(=O)NC1CCCN(C(=O)C2=CCCCO2)C1 CC1(NC(C2CC2c2ccncc2F)=O)CCC(NC(c2nn[nH]c2Cl)=O)CC1 Cc1c(F)cc(C(=O)NC(C)Cn2cc(C(C3CCCCC3)C)nn2)c(F)c1N C1(C(=O)NCc2c(C)nc[nH]2)CSCCN1C(=O)CO N1(C(C(C)OCC2CC2)=O)CCC(O)(CCNC(C2(N=[N+]=[N-])CC2)=O)C1 C1(C(N2C(C(C)(C)NC(=O)Cn3ccnn3)CCC2)=O)CC(F)C(=O)N1 c1(C(=O)NCCOCCNC(C2C3CCC23)=O)c[nH]c2cc(F)c(F)cc12 N1(C(c2nc(CNC(=O)CCCCC#N)sc2)=O)CCC2(OCC)CC2C1 c1(C(=O)NCc2ccc(N(CCCC)C)cc2)cc(C)c(CC)nc1O C(=O)(C1CCCn2ccnc21)N1C(c2cc(CC)no2)CCCC1.C1CCCO1 c1(C(=O)NC(C)CCCCNC(C2CC(C)(C)CO2)=O)ncnc2c1CCC2 N1(C(COC)=O)CCOC(CCCNC(=O)C(C)(C(C)C)C2CCCCC2)C1 c1(C(C)C)cccc(CN(C)C(=O)NCC(C2CC(F)(F)C2)O)n1 C1(C(=O)NCCCCN(C)C(c2c[nH]c(C#N)c2)=O)C2CC2C2CC12 Cc1ccc(F)c(C(N2CCC(O)C(NC(C3CC3C(F)(F)F)=O)C2)=O)c1 c1(C(=O)NC2CN(C(C3(SC)CC3)=O)CC(C)C2)cc(N(C)C)ccc1[N+](=O)[O-] C(CCC(C)C)(C(=O)N1CCNC(=O)CC1C)NC(Cc1cc(C)n(C)n1)=O C(CCC(O)C(=O)NCC(C)CN=[N+]=[N-])NC(Cn1c(C)nnn1)=O C(CC1=CCCCC1)NC(C1CC(=O)NCC1)c1nnnn1C1CCCC1 C(=O)(CCS(C)(=O)=O)N1CCC(N(CC(C)C)C(=O)Cc2cccs2)CC1 Cc1cnc2n1CCN(C(=O)N(c1cccc(NC(=O)OC(C)(C)C)c1)C)C2 c1(-c2nnc(C(=O)NC(C(=O)OC)Cc3ccc(Cl)cc3I)o2)cccc(Cl)c1Br C1(C)(CNC(c2c(CC(C)C)onc2)=O)CCN(C(c2ccc[nH]2)=O)C1 N1(C(c2[nH]cc(CC)c2)=O)CCN(C)CC1CNC(C1CCCCC12CC2)=O C1(NC(CCN(C(CC)CC)C)=O)CN(C(c2cc(=O)cc[nH]2)=O)CC1C N1(C(C)=O)CCC(CC(=O)NCC(C)(C)CNC(C2(OC)CCCOC2)=O)CC1 C1(C(N(C)CC2CC(=C3CC3)C2)=O)CC(O)(CNC(=O)C(c2cccn2C)=O)C1 c1(CN2C(C(=O)NCC3COC3)CC3CC32)cc(Br)c(F)cc1F C#CC1CCN1C(C1COC(CNC(=O)CCc2cn(C)nn2)C1)=O c1(C(C)=O)cnc(C(=O)NCC2(C)CCC(NC(=O)C=Cc3cccs3)C2)cn1 N1(C(C2C(C)C2)=O)CC(NC(c2ccc(-c3nnc(S)o3)cc2)=O)CCC1C.C1(S)CC1 Cc1noc(C)c1CC(C)NS(=O)(=O)CCCC1CCC1 c1(CC)noc(COCC(=O)NC2CCN(C(=O)C(C)NC=O)C2)n1 N1(C(C(C(CC)CC)C)=O)CC(C)CN(C(c2ccc(OC)nc2)=O)CC1C C1(C)(C(=O)NCC2N(C(C3CCN(CC)C3)=O)CCC2)CNC(=O)N1 c1(C(C(=O)NCCOC)N(C)Cc2ncccc2Br)ccc2c(c1)N(C)CC2 C1(CCCCNC(C=CC)=O)CCN(C(c2cnn(C3CCCC3)c2C)=O)CC1 C1(C(N2C(CN(C)C(c3nn(C)cc3N)=O)CCC2)=O)CC12CC(F)(F)C2 c1(C(N2CC(NC(C3C(CC)C3)=O)C(OC)C2)=O)cccc2c1CCCCN2 c1(C(N2CCC(C(N(CC(=O)N(C)C)CC)=O)C2)=O)cnc(O)c(C)c1 c1(C(=O)NC2CCN(C(c3c(CC)c[nH]c3)=O)CC2CC)cc(C)c(F)cc1Cl c1(C(=O)NCC2CC(NC(Cn3c(C)ccn3)=O)C2)ccc2cccc(O)c2c1 N1(C(c2ccn(CC)n2)=O)CC2CC1C2NC(c1nc(-c2cccs2)oc1C)=O C(=O)(C(C)(C)CN(C)C(c1ccns1)=O)NC(c1ccsc1)C C(=O)(C(C)(C)C)NC1CC(CC(=O)N(CCN(CCCC)C)CC)C1 c1(C(=O)NC2CC(C)(CC)N(C(=O)CCC(C)C)C2)cc(=O)c(OC)cn1C C1(NC(c2c(C)oc(C(C)C)n2)=O)COCCN(C(C2(C#N)CC2(C)C)=O)C1 c1(C(N2CCC2Cc2ccccc2)=O)cnn(CC2CC(C(=O)NC3CC3)C2)c1 N1(C(COCCC=C)=O)CCCC(C(=O)NCc2cnc(C(C)C)[nH]2)C1CC C1(NC(CCOCC)=O)CC2CC1CN(C(c1c(C)cc(Cl)nc1N)=O)C2 c1(OC)cccc(C(=O)N(C(C)CNC(C2CCC(C)C2)=O)C)c1 C1(NC(C(CCOC)OC)=O)CC12CCN(C(=O)C1=CC3C=CC1C3)CC2 c1(C(N2CCN(CC3CN(C(CC(C)F)=O)C3)CC2)=O)cc(C2CC2)nc(O)c1 N1(C(C(CC)SC)=O)CCCCC1CCNC(=O)CSc1nnnn1C C12(NC(CCC=CC)=O)CC1CN(C(=O)COc1ccccc1O)C2 CCCC(C)CCCC(=O)N1CCN(C(=O)C2=CCOCC2)CC1 C(CC1=CCN(C(=O)C(F)(Cl)c2ccccc2)CC1)NC(C1CC(COC)C1)=O N1(C(=O)Cc2cccnc2O)CCC2CN(C(c3ccoc3Cl)=O)C2C1 CC1=C(C(=O)NC2CCC2CNC(C23CC2C3)=O)CCO1 C1(C(=O)Nc2cn(CC(C)C)nc2)CC2(CCN(C(=O)C(F)C(C)(F)F)C2)C1 C1(NC(CCN(C)C)=O)CCN(C(c2csc(Cc3ccccc3)n2)=O)CC1F N1(C(C(C)C)=O)CC(N(C)C(c2ccc(NS(=O)(=O)C(F)F)cc2)=O)C2(CC2)C1 C=C(Cl)CC(C(=O)NC1(CF)CCC1)NC(c1cc2n(n1)CCO2)=O CC1CCN(C(c2ncn(C)n2)=O)CC1CNC(c1ccsc1-n1cnnn1)=O C(=O)(C(=O)N(CCn1cnnc1)CC)N(C1CC1)CC C1(CNC(CNS(CC)(=O)=O)=O)CCN(C(c2cc3c(s2)CCC3)=O)C12CCC2 C1(=O)CC(=O)N1.CC(CCNC(=O)CC1(CSCC(C)(C)C)CC1)N(C)C N1(C(C=C(C)C)=O)CCC2(CC1)CC(C)N(C(c1ncoc1C)=O)C2 N1(C(C2N(CC(C)C)CCC2)=O)CCC(NC(c2cc(O)nn2C)=O)C(C)C1 Cc1nc2nccc(N3CC(CO)(NC(c4cc(C)oc4C)=O)C3)n2n1 C(CC(C(C)(C)C)NC(=O)COC1CCC(C)CC1)N(C(c1cnc(C)s1)=O)C C12CC3CN(CC13)C(=O)CCC(=O)N2.c1(CC)ccc(C2(C(=O)OC)CC2)cc1 S(=O)(=O)(c1ccc(OC)cc1C)NCCC(=O)NC1C(OC)C(C)(C)C1 N1(C(C(Cc2ncn(C)c2)O)=O)CCC2(CCCN2C(C2(C3CC3)CCC2)=O)C1 Cc1ccc2cc(C(N3CC(C)(NC(=O)CN(C)C(=O)C4CC4)C3)=O)ccc2c1 N1(C(C2C(SC)CCC2)=O)CC=CC(NC(=O)C(C)(C)CC2CC2)C1 C(=O)(C(=O)N=S(C)(C)=O)N1C(CN(C(C(c2ccc(O)cc2)C)=O)C)COCC1 c1(N2CCC(SCC)CC2)ccncc1S(=O)(=O)NC(c1ccc(F)c(F)c1)C C1(CC(=O)NCC(CC)NC(c2c(C)nn(C)c2F)=O)CCCC(C)(C)C1 c1(C(=O)NCC(CC(=O)N(C(C)CS(C)=O)C)(C)C)cncc2[nH]ccc12 Cc1ccc(Br)nc1C(N1CCN(C2CC2)CC1)C(=O)Nc1cn[nH]c1 c1(C2C(CC(N3CCC(CCn4cc(C(=O)O)nn4)CC3)=O)C2)cccc(Cl)c1 C1(NC(=O)C(C2CCOCC2)O)CC2CCC1CC2NC(C1(C(F)(F)F)CC1)=O C(=O)(C(CC(C)(C)C)NC(C1CCOC1(C)C)=O)NCC(C(C)C)C C1(C(N(CCn2ncc(C)c2)C)=O)C2CCC(C2)C1NC(=O)C=CCC1CCC1 N(C1CC2CCCc3cccc1c32)S(CC(C)C1CC1)(=O)=O CCCCCS(=O)(=O)CC(=O)N1CCC(CNC(=O)Cc2cnn(C)c2)C(C)C1 C1(C)(C(=O)NCC2C(C(=O)NCC3(COC)CC3)CC2)C=CCC1 c1(C(=O)NCC(C2CCN(C(C3CCCO3)=O)CC2)C)nccc2ccn(C)c12 C1(CC(N2CC(CCO)(NC(C(C)NC(=O)NC)=O)C2)=O)CCCCN1C C1(C2CC2)(NC(C(CC)NC(C2CCCSC2C)=O)=O)CCOC1 N1(C(C(CC#N)NC(=O)OC(C)(C)C)=O)CCC2(CC(C(F)F)=NO2)C1 C1(NC(C2C(NC(C(CN(C)C)N(C)C)=O)CCOC2)=O)CCC(=O)N(C)C1 c1(CC(=O)NC(C2CCN(C(c3cc(Cl)no3)=O)C2)C)ccc(S(C)(=O)=O)o1 c1(OC)ccnc(CN2CC(c3cccc(C)c3)(O)C2)n1 N1(C(C=C(CCC)C)=O)CCCCC1CN(C(=O)CCc1ccon1)C CC(C)CC(C)C(=O)NC1CC1CNC(c1cc(C(F)(F)F)c(F)cn1)=O C1(CNC(C(CC)COC)=O)CN(C)CCN1C(=O)C(c1ccc(C)o1)C N1(C(C(C)OC2CCCC2)=O)CCC2(NC(=O)C(C)(C)N3CCCC3)CCCC12 c1(C2N(C(C(c3ccc(F)nc3Cl)(C)C)=O)CCC2)nc2ccccc2[nH]1 C(C1(C)OCCc2sccc21)NC(=NCCc1cn(C)nc1)NCC1CC1 C1(CNC(C2CC(=C(F)F)C2)=O)CCCCN1C(C1CCC(F)(F)C1)=O n1(CC)nnc(C)c1C(=O)NC(C1CCN(C(C2(C(C)C)CCCO2)=O)CC1)C C1(NC(C=C(C)C)=O)CC2CN(C(=O)C=Cc3ccncn3)CC12 Cc1cncc(C=CC(=O)NC2CN(C(c3c(C)ncn3C)=O)CC2C)c1 C1(CNC(C2CC(C)(NC(c3c(C)snc3)=O)C2)=O)CC(O)C(O)C1 Cc1cc(=O)n(C)cc1C(=O)NCC1CCN1C(=O)CN1CCCNC1=O CS(=O)(=O)CCCCCCCC(=O)NC(c1ccc(Cl)s1)C(=O)O c1(NCc2ccc([Si](C)(C)C)cc2)c(Cl)cc(F)c2ncccc12 c1(C(=O)NC(CC#C)C(=O)NCCCN2CCOCC2)ccnc(C)c1N N1(C(CC2(C=C)CCC2)=O)CC(C2CCCN(C(=O)C(O)CN(C)C)C2)C1 C1(NC(c2c(C)cccc2C)=O)CC2CC1CN(C(C1(C)CC3(CCC3)C1)=O)C2 C12(NC(=O)OC(C)(C)C)CC(C(N3CCC(SCCCCO)C3)=O)(C1)OC2(C)C N#Cc1cccc(-c2cc(C(=O)OCCC3OCCO3)no2)c1 CCC(C)(C)C(C)CC(=O)N1CC2(C1)CN(C(c1cc3n(n1)CCO3)=O)C2 C#CC1CCCC(NC(C2CCN(C(c3ncnc(O)c3F)=O)C2)=O)C1 C1(C(NOCCCC=C)=O)CN(C(C23CC(C#N)(C2)C3)=O)CC1(F)F CC(C)(Cc1cnn[nH]1)C(=O)N(CCO)CCNC(c1cccnc1OC1CC1)=O c1(NC)cncc(C(N2CC(C(N3CCC(CCO)CC3)=O)(SC)C2)=O)c1 c1(CN2CC3CN(C(c4scc(C(C)C)n4)=O)CC3C2)cnc2ccccc2n1 N1(C(C(COC)NC(CCCOCC=C)=O)=O)CCC(COC)C(C)C1 c1(C(=O)NCC2C(NC(CCc3ccn(C)c3)=O)C2)c(C2CC2)cccc1F c1(C(=O)NCC2OCC(CNC(C3CC(CC)C3)=O)C2)cc(OC)ccc1Cl Cn1nnc(CNC(C2CC2Cl)=O)c1C(=O)NC1CNC(=O)C1 c1(SCONC(C2C3CN(C(Cn4c(C)ncc4)=O)CC32)=O)ccc(F)cc1F c1(C(=O)NCC(CNC(Cc2c(C)nc[nH]2)=O)C)ccc(CO)cn1 Cc1c(F)ccc(C(=O)NCC(C)(C)CN(C(=O)C(C)(C)CN(C)C)C)c1F CCCCC(CNC(=O)C=CSc1ccccc1)NC(c1coc(C(C)C)n1)=O C(=O)(C(F)(F)CNC(C1(NC(C2C=CCCC2)=O)CCCCC1)=O)OC c1(C(N2C3CN(C(CC4(C#N)CC4)=O)C(CC3)C2)=O)ccn2c(O)nnc2c1 N1(CC=C)CCC2(CCCN(C(C3CNC(=O)CC3(C)C)=O)C2)C1 C1(NC(C(C)CC2CC2)=O)CCCC(NC(=O)CSCc2ccccn2)C1 CC(C)CCN=C(NCc1ccc(C(C)O)cc1)NCC1CN(C(C)C)CCO1 N1(C(C(=O)NCC(CNC(C)=O)CO)C)C(=O)c2ccccc2C1=O C(=O)(C1=CCC(C)CC1)NCC1OCCCN(C(C2(COC)CC2)=O)C1 CC1CCC(C)(C=CC(N2CCN(c3cccc([N+](=O)[O-])c3)CC2)=O)C1(C)C C1(C(=O)NC2(C(=O)NCC3CCCS3)CC(F)C2)(OC)CCOCC1 N1(C(C(C)NC(C)=O)=O)CCC(CNC(=O)CN2CC(=O)N(C)C2=O)C(C)C1 CC1CCC2(CC1)CCN2C(=O)CCC1CCN(C(C2(CO)CCC2)=O)C1 c1(C(N2CCC(CNC(C(C)S(N)(=O)=O)=O)C2)=O)ccc(Br)cc1[N+](=O)[O-] c1(OC)ccc(CNC2C=CC(C(N3CCCC3C)=O)C2)c2cccnc12 N1(C(C2CCN(C(C3(C)C(C)C3)=O)CC2O)=O)CCC2(CC1)COC(=O)N2 Cc1cc(C#N)ccc1C(=O)NC1CC1NC(C1CS(=O)(=O)CC(=O)N1)=O CC1C(NC(=O)CCc2ccncc2)CC2CCC1N2C(c1ccnc(Cl)c1)=O c1(C(=O)NC2(CO)CN(C(C(C(C)OC)O)=O)C2)ccc2ncc(OC)nc2c1 c1(OCC)ccccc1C(=O)NC1CN(C(c2occc2C)=O)CC1C N1(C(C=CC(C)(C)SC)=O)CC2(C1)CN(C(=O)CNC(c1cn[nH]c1)=O)CCO2 c1(C(N(CC(C)(C)NC(c2ccc(CN(C)C)o2)=O)C)=O)cnc2n1CCOC2 c1(NC(N2CCC(C(=O)NC3CC3c3cccnc3)C2)=O)cc2scc(Cl)c2[nH]1 N1(C(C2(Oc3ccccc3)CC2)=O)CCC(O)C(c2ccccc2)C1 N1(C(c2c[nH]nc2C)C(=O)NCCOC)Cc2cc(OC)ccc2OC(C)(C)C1 C1(OC)CN(C)C(C)(C(N2CCCC(CNC(c3cc(Cl)cn3C)=O)CC2)=O)C1 n1(CC(C)C)cc(S(=O)(=O)NCc2nc3cnccc3s2)cn1 Cc1ccccc1C(C)CC(=O)NCC1CCN1CCCc1cccnc1 c1(NC(C(N2CCC(NS(C)(=O)=O)C2)c2cccs2)=O)ccccc1C c1(CCC)nc(C(=O)N(CCN(C)C(C2CCCN2C(=O)NC)=O)C(C)C)co1 CCCCC(O)C(=O)N1CCCC(NC(=O)Cc2csc(C)n2)C1C C1(CC(=O)NCc2ccccc2)CCCC1NC(c1nc(CO)cs1)=O CCC(C)C(O)CC(=O)NCC1CCCN1C(c1cnc(C(N)=O)s1)=O N1(C(C2(C#C)CCC2)=O)CCC(CO)C(NC(c2ncccc2NC(C)=O)=O)C1 c1(NC(C2CCC(NC(c3nn(C(C)C)nc3C)=O)C2)=O)nc[nH]c2nccc1-2 Cc1cc(C)c2nc(N3CCC(NC(c4ccnn4CCF)=O)C(F)C3)sc2c1 CC(C)CC(C)(C)C(=O)NCC1CCN(C(=O)CN2C(C)CCC2C)C1 Cc1cccc(NC(C23CC(CN2C(=O)Cc2cccnc2C)C3)=O)c1C c1(C(N(c2nc(C#C)c(F)cn2)C)=O)c(Br)cc2ccccc2c1F Cc1cc(C(N2CCOC(CC(=O)NC3CC3c3ccn(C)n3)C2)=O)ccn1 C1(C(=O)N(C2CC(NC(C3CCOCC3)=O)C2)C)(CC)CCOC1 N1(C(C=CCNC(C(CCCC)=O)=O)=O)CCCC2NC(=O)CC12 C(c1ccccc1)=C(CC)C(=O)NCC(C)NC(=O)CCc1ncc(F)cn1 N1(C(c2ncc(N)nc2)=O)CCOCC(CNC(C2CC2C(N)=O)=O)C1 c1(C(C(=O)NC(CN(C(C2CC3(CC3)C2)=O)CC)C)C)ccc(C)s1 C(C(CC(C)C)NC(C12CCCC1C2)=O)NC(c1cc(C)on1)=O c1(C(=O)NC2C(C)CN(C(c3ccccc3)=O)C2)ccc(F)c2cccnc12 CC(C)C(CNC(=O)CCc1cn[nH]c1)NC(=O)COc1ccccc1 O(NC(=O)C(CCSC)NC(c1cc(C)c(C)o1)=O)CCCC#C C1(CNC(C2=CCN(C)C2)=O)CN(C(C2CCCCC(=O)N2)=O)CCC1(F)F c1(OC)cccc(C(N2CCC23CCC3)C(=O)NC(C)C)c1Br Cc1cnc(C(=O)NCC2C3CC2N(C(c2ccc(C4CC4)cn2)=O)C3)c(F)c1 Cc1cccc(CC(=O)NCC(CC(C)C)NC(c2ccc(F)cc2)=O)c1 N1(c2ncnc(Nc3c(OC)ccc(SC)c3)c2C)CCC(C2CC2)C1CO c1(C(=O)NC2CN(Cc3cccc(Cl)c3)CC2F)ccc2cccc(Br)c2n1 CC(C)C(CNC(c1ncoc1-c1ccco1)=O)C(=O)O N1(C(C(CCOC)NC(c2cc(C)nc(O)n2)=O)=O)CC2CCC1CC2 CC1CN(C)C(C)CN1C(C1CN(CCF)CCC1O)=O Cc1cc(NC(C2(C)CN(C(=O)CSc3ccccc3)C2)=O)c([N+](=O)[O-])cc1C c1(OCC(=O)NCC(CN(C)C(C2COCCO2)=O)O)ccc(C#N)cc1Cl n1(CC)nnnc1C(C1CCCC1O)(C)NCCC(C)F C12(NC(CC)=O)CC3CCC(C1C2)N3C(c1nn(-c2ccccc2)cc1OC)=O c1(C2(C(C)NC(=O)CC3(NC(N)=O)CCC3)CC2)ccc(Br)cc1F C(=O)(C(C)C(O)C(C)C)N1CC(C=C)(CC(=O)NCC(C)(O)COC)C1 N1(C(=O)OC(C)(C)C)CC2CCCC2(NC(C2COCC2(C)C)=O)C1 c1(CCC(=O)NC(CNC(CC2CC(=C)C2)=O)(C)Cn2cccn2)ccc(C)cc1 C1(C(=O)NC(C(F)OC)=O)CCC2(CCOCC2)C1 N1(C(C2C3CN(C(CC(C)(C)C)=O)CC32)=O)CCS(=O)(=O)C2CCCC12 N1(C(c2cc(I)ccc2Cl)=O)CC(N=c2ncc3cc(F)cc(Br)c3[nH]2)C1 Cc1c(C(=O)NC(C)CC(C)NC(C23CC(F)(C2)C3)=O)[nH]c2c(C)cccc12 C(CC(=O)NCCCCC1CN(C(=O)COC2COC2)C1)NC(C1C(C)C1)=O CC(C)CCCCCC(=O)NCCC(N1CCCC1CN=[N+]=[N-])=O c1(C(N2C(C(=O)NCC3CCC(O)CC3)CCCC2)=O)cc(O)cc(F)c1F Cc1ccncc1CNC(c1cn(C(C)(C)C)nn1)c1nnnn1CCCF C1(C(=O)Nc2c(O)ncc(C)c2)CC2C=CC1N(C(=O)CCc1cccs1)C2 N1(C(C(CC(C)(C)C)O)=O)CCC2CN(C(=O)CS(=O)(=O)NC)CC2C1 C1(CNC(CC2(OCC)CCC2)=O)CC2CCC1N(C(=O)CC#N)C2 CC1CCC(C(=O)NCCOC(C)(C)C)C1.c1(CC(=O)NCCOC)cn(C)nn1 c1(C(=O)NCCCN(C(CSC)=O)CCO)cc2c(=O)n(C)c(=O)n(C)c2s1 N1(C(C(CCC(C)C)F)=O)Cc2n[nH]cc2C1C(=O)NCCNC(N)=O CON(CCC(=O)Nc1c(C)noc1C1CC1)C(=O)C1SCC=C1C Cc1ccc2snc(C(=O)NCC(C)N(C)C(C3CC(N(C)C)C3)=O)c2c1 N1(C(C(CC=CC)CC)=O)CCCC2C(NC(c3sccc3CC)=O)C(C)(C)C12 C=CCC(C(=O)OC)NC(=O)C(COCC)NC(c1ccn(C)c1C)=O C(=O)(C(O)CC(C)(C)C)NC(CN(C(=O)CN)CC)C.C(=O)(C(C)(C)C)NC(C)=O c1(C(=O)NC2C3CN(C(c4n(C)nc(CC)c4Cl)=O)C2C3)coc2c1CCCC2 C12(C(=O)NC(CC)CN(C)C(c3cc(C(N)=O)no3)=O)CCC(C)(C1)OC2 n1(C(C)C)cc(C(c2nnnn2C(C)(C)C)NCCC2CCCC2)cn1 c1(C(=O)NCC(C)NC(C2C(OCC)C2)=O)c[nH]c2cc(C)ccc12 N1(C(=O)NC2CCC(C)N(C(=O)CCNC(=O)CO)C2)CCc2sccc2C1 CCCCS(=O)(=O)NCC(=O)N(CCCN(C)CC1CCC(O)CC1)C N1(C(c2coc(Cl)c2)=O)CCN(C(=O)Cc2sc(O)nc2O)C(CCO)C1 c1(C(=O)NCCOCCN(C(c2cccc(C)c2)=O)C)cccc(Cl)c1Cl C1(=C(C)C(=O)Nc2cccnc2Cl)N=C(c2ccncc2)NC1=O C(=O)(C(C)(O)CC(F)(F)F)N(CCCNC(C(C1CC1)OC)=O)C1CC1 c1(C(=O)NCC2C(C)CCN(C(=O)CS(C)(=O)=O)C2)cnc2c(Cl)cccn12 Nc1cc(C(=O)NCC2CCC2NC(C2CCSCC2)=O)ccc1-n1cncn1 Cc1cncc([N+](=O)[O-])c1NC(=O)Nc1ccc(CSCSC)c(F)c1 N1(C(CC(C)C)=O)CC2CC1C2NC(=O)C(C)Oc1ccccc1F C(=O)(C1=COCCO1)N(CC(C(C)C)NC(=O)CCC(=O)c1cccc(Cl)c1)C n1(CC(=O)NC2(C3CCN3C(c3cnc4n3CCS4)=O)CC2)cc(F)ccc1=O CC(F)(F)CCC(=O)N1CCN(C(c2cnn(CCF)c2)=O)C(CO)C1 c1(C(N(CC(CC)NC(=O)C(C)OC(C)(C)C)C)=O)nnc(C)cc1O C(CO)(C(=O)NCc1ccn(C)c1)NC(C(C)=C1CC1)=O n1(C(=O)NCC(CC)(CC)NC(=O)CSCC(C)C)ccc(=O)cc1C C1(C)(C(=O)NCC(c2ccccc2)NC(CSCCOC)=O)CCN(C)C1=O c1(C(C(=O)NCC(C)N(c2nnc(CC)s2)C)C2CC2)ccccc1OC N1(C(=O)OC(C)(C)C)CCCC(CNC2CC2C(=O)Nc2cc(F)n[nH]2)C1 N1(C(C)=O)CCc2cccc(C(=O)NC3(c4ccc(Br)c(Cl)c4)CCC3)c2C1 C1(C(=O)OC)CC(C2CC2)=NO1.c12cc(sc1C)CNC(=O)NC2 c1(C(=O)NC2CCCCN(C(c3cncc(C)c3C)=O)C2)cc2ccncc2[nH]1 C(c1cccc(Br)c1)=CC(=O)NC(CNC(C=COCC)=O)CO CC1(C)COCCN(C(C2COCCC2NC(=O)C=Cc2ccco2)=O)C1 Cc1sc(-c2ccco2)nc1C(=O)N(CC(C)NC(=O)C=CCO)C N1(C(C2(C)CCN(C(=O)COc3ccsn3)C2)=O)Cc2cccnc2C1 c1(C(=O)NC23CC(NC(COC)=O)(C2)C3)ccc(Br)cc1O c1(CNC(c2ccccc2)C(C)C)c(Br)cnn1C.c12csc(n1)S2 C(=O)(C#CC1(C)CCCO1)NCc1nc(CNC(c2c(C)cc(C)nc2)=O)sc1 C1(CN(C)C(c2cc[nH]n2)=O)CN(C(c2cn(C3CC3)nn2)=O)CCO1.NC c1(CC(=O)NC(CNC(C2(CC=C)CCC2)=O)CO)cnc(C2CC2)[nH]1 c1(C(C(N2C(C(=O)OCC)CC2)=O)=O)cn(CC(=O)NCCC)c2ccccc12 C1(C(=O)NCCN(C(c2c(CCC)n[nH]c2)=O)C2CC2)CCCCN1C(C)C C1(OC)CN(C(c2cnc(C(C)C)o2)=O)CC1NC(C1(c2cc[nH]n2)CC1)=O N1(C(=O)CCc2cncnc2)CCC(C2CCCN(C(C3CC(O)C3)=O)C2)C1 Cc1ccc(C(=O)NCC2(F)CC(NC(C3(CCN(C)C)CC3)=O)C2)cc1C C1(NC(c2ccc(C)o2)=O)CCN(C(=O)Cc2ccccc2SCCO)CC1C c1(C(N2CC(NC(C(F)=CC)=O)C(C)C2)=O)cn2c(n1)CC(C)CC2 C1(C2CC2)(CNC(C(C=C)(C)CC)=O)CCN(C(=O)COCC(C)C)C1 CC1CN(C(=O)CCS(C)(=O)=O)CCN1C(c1ccnc(OC(F)F)c1)=O C1(NC(=O)NCC(c2ccc(O)cc2)O)CCCN(c2ccncc2)C1 C(C(CC)CC)(c1ccc(C(F)(F)F)s1)N(CC)CC1(c2ccc(F)cc2)CC1 N1(C(C(C(CC)CC)C)=O)CCC2CN(C(=O)CC(C)C)CCC2C1 CCC(CC)C(C)C(=O)NCC1(C)CCN(C(=O)C(C)n2cccc2)CC1 c1(C(=O)Nc2nc(C3CC3)cs2)ccc(S(=O)(=O)Cc2ccc(Br)cc2)cc1 Cc1ccc(NC(C2OCCC2NC(c2ccc(C)c(C#N)c2)=O)=O)c(C)c1C C1(C(N(C(CC)CNC(=O)Cc2ncoc2C)C)=O)N(C(C)=O)CC12CCCC2 c1(OCC)cccc(C(=O)NC2CC(NC(=O)CC3(CO)CCCCC3)C2)c1N S(=O)(=O)(c1ccc(NCc2cnc(-n3cccn3)s2)cc1Cl)N1CC(C)=C(C)C1 N1(C(CC(=C=C)C)=O)CC2(CCCN(C(=O)C(F)(F)CCC=C)C2)C1 C(CCO)(C(F)(F)F)NC(N1CCN(c2cc(N3CCOCC3)ncn2)CC1)=O c1(OC)ccc(Cl)cc1C=CC(=O)NCC(C)N(C)C(C1CCOC1)=O C(c1c(Cl)cccc1Cl)=C(C(CNC(CCCCNC(=O)OCC)=O)=O)C N1(C(C2OCC(C)(C)C2)=O)CC(NC(=O)COCCN(C)C)CC(O)C1 c1(NC(c2ccc(CN(C(N(C)C)=O)N(C)C)cc2)C)cc(=O)cc[nH]1 C(CCc1cn[nH]c1)(C(=O)N1CCC1C(F)F)NC(=O)OC(C)(C)C C1(NC(C=CC(=O)NC2CC2)=O)CCC2CC1CN2C(=O)C1=CCCC1 c1(C(=O)NCCC23CCC2CN(C(=O)C(Cl)=CCl)C3)cc2ccccn2n1 CC(C)(C)CC(O)C(=O)N1CC(O)CC1CC(=O)NCC1(O)CCSC1 N1(C(c2cccc(OC)c2)=O)CCC2(NC(=O)CCC3CC3(C)C)CCCC12 Cc1nc(CO)ncc1NC(=O)CCCC1(NC(=O)CN2CCCCCC2)CCC1 C(=O)(C(C)(C)C(N)=O)NC(CCOC)CNC(=O)C(c1ccccc1)C1CC1 CC1(C)CC(CC(=O)NCC23CCN(CC2)C3)N(C(c2ncncc2Cl)=O)C1 CC1(C(=O)NCC2CCN2C(=O)Cc2csc(Cl)n2)CCc2ccccc2C1 C1(C(N2C(CNC(CCCCCSC)=O)CCC2)=O)Cc2ccncc2C1 c1(C(=O)NC(CNC(C(CC#C)(C)C)=O)C2CCC2)ncn2c1COCC2 c1(C(=O)NC2CC(NC(C3CCN(C)C3)=O)C2)c[nH]c2cccnc12 C1(NC(c2c(CCNC(C(C)(C)N=[N+]=[N-])=O)n[nH]c2)=O)CCc2nncn2C1 c1(C(=O)NS(=O)(=O)CCCNC2C(C(=O)OC)C2)ccncc1C(F)(F)F N1(C(CSCC=C)=O)CCCCCC1C(=O)NC(c1ncc(C)[nH]1)C C12(CNC(C3CCCC(=O)N3)=O)CCC(CC1)N2C(c1cc2n(c1)CCC2)=O C(CCC1CC1)(C(=O)N1CCC(O)C1)NC(C(CC)C1CCC(=O)N1)=O C(=O)(CS(=O)(=O)CCO)NC(C1CCCCC1)CNC(c1n(CC)nnc1C)=O N1(C(c2nc(COC)oc2)=O)CCCC(NC(C2CCCC2Br)=O)C1 N1(C(C(c2ccoc2)NC(C(CCC)NC(C)=O)=O)=O)CC2C3C=CC(C3)C2C1 c1(C(=O)NCC(CCCC)NC(=O)C(C)(C)CN(C)C)cc(O)ccc1C C1(CC=C)(NC(c2[nH]nc(C(F)(F)F)c2C(C)C)=O)CCN(C(C2(C)CC2)=O)C1 c1(C(=O)NC(C2CCCC2)CNC(CN(C)C2CC2)=O)ccc(O)c(CO)c1 C1(C(N2CC(CC(C)NC(c3ccncc3)=O)C2)=O)CCC2(CCOCC2)O1 c1(C(N2CCC(N(C(=O)C(C)SC(C)C)CC)C2)=O)cccc(C(F)F)c1 c1(CC(=O)NCC2(NC(COC3(C)CC3)=O)CCOC2)cc(F)ccc1F n1(CC)nc(-c2ccc(COC)cc2)nc1C(C)Oc1cccc(OC)c1 N1(C(Cc2c(C)noc2Cl)=O)CCCC2(NC(=O)Cc3cccs3)CC2C1 C1(C#N)(C(=O)NC2CC3(CN(C(C4N(CC)CCC4)=O)C3)C2)CC2CCC1CC2 N1(C(C2(C#N)CC2)=O)CC(C(=O)NCC2CCCC23CC3)C2(CCC2)C1 Cc1cc(=NCC(C)CN2CCOCC2)[nH]c(N2CCN(Cc3cccs3)CC2)n1 c1(CC(N2CC(C)(NC(c3cc(C)nc(O)n3)=O)C2)=O)oc2ccccc2c1C C1(C(N(CC(C)CNC2(C(O)CO)CC2)C)=O)CCC(=O)C1 c1(C(COCCO)N(C(C)=O)C(=O)NC(C)(C)C)cc(C)cc(Br)c1 Cc1[nH]nc(C(=O)NC2(C(N3CC(n4cnnc4)C3)=O)CC2(C)C)c1Cl C1(CC)CCN(C(=O)C=C(C)C2CCN2C(=O)C(C)OCCOC)CC1 CCS(=O)(=O)CC(=O)N1CCCC1CCNC(C1CCN(C(=O)N(C)C)CC1)=O C=Cn1nccc1C(=O)NC1CCC(CNC(=O)CCC=CC)C1 n1(CC)cc(C(=O)N(CCNC(C2CCC(C(=O)OC)C2)=O)C2CC2)c(C2CC2)n1 c1(SCC)cnc(O)c(C(N2CC(N(C)C(c3nc(O)c(C)s3)=O)C2)=O)c1 c1(CCC(N2C(CNC(C(COC)O)=O)CC3(CC3)C2)=O)csc2ccccc12 CC(C)CCOC1(CCC(=O)N2CCC2CC(=O)N(C)C)CCC1.C1C(=O)N1 C(=O)(C1=NN(C)C(=O)CC1)NC(CC)(C)CNC(C12CCOC(C)(C1)C2)=O N1(CCNC(C(C(C)OC)O)=O)CCCN(C(c2nocc2C(C)C)=O)CC1 Cc1ncc(C(=O)NC2CCCCN(C(c3ccnc(O)c3)=O)C2)c(C(C)C)n1 N1(C(C(=O)NC2CC2)=O)CC(C(=O)NOCC2CCCC2)CC12CCC2 c1(C(=O)NCCn2cc(CCO)nn2)ccc([N+](=O)[O-])cc1F N1(C(CC(=O)NCC#C)=O)CCC(C)C1CNC(=O)CSc1ccc(C)cc1 c1(C(=O)NC(C(C)C)CCN(C(=O)C(C)CN(C)C)C)ccnc2ccsc12 C(=O)(C(F)(F)C(O)C1CC1)N1CC(CC(C)NC(C2OCC2(C)C)=O)C1 N1(C(c2c(C)ncc(N)c2)=O)C2CCC1CC(N(C)C(C1CCCC(C)C1)=O)C2 c1(C(N(CCCNC(C2CC3CC2C3)=O)C(C)C)=O)cc2n(n1)CCCO2 Cn1ncc2cc(C(=O)NCC3C4CN(C(C5CCS(=O)(=O)N5)=O)CC34)cnc12 Cc1c(C(N2CC(NC(C3(C)CNC(=O)C3)=O)C(F)C2)=O)ccc(F)c1F c1(CCCN(C2CCN(C(CN(S(CC)(=O)=O)C)=O)C2)C)ccccc1C C12(C(=O)OCC)CCC(C(=O)NCCN(C(=O)C(C)CCOC)C)(CC1)CC2 Cc1cc(C(N2CCC(C)(CNC(=O)CCC3CCOC3)C2)=O)nn1C1CC1 C1(C(CNC(CN(S(CC)(=O)=O)C)=O)C)CCN(C(C2C(C)C2C)=O)CC1 CC1CC(N=c2[nH]c(N3CCC=C(Cl)C3)nc3c2CCCCC3)CC(C)(C)C1 c1(CC)cc(C(=O)NCC2CCC(CCNC(=O)C(C3CCC3)OC)C2)n(C)n1 c1(OC)ccc(CN2CC3CC3(C(=O)N(c3ccccc3)C)C2)c(Br)c1OC CCCCC(O)C(=O)N1CCCC(O)(CNC(=O)C=C2CCC2)C1 Cc1nc(O)nc(O)c1CC(=O)NC1CCCC1NC(=O)C(C(C)(C)C)C1CC1 N1(C(c2cc(C)sc2)=O)CCCC1C1CCCN1C(C1C(O)C(=O)N(C)C1C)=O C1(C2CC2)(C(=O)NC2CCCN(C(c3c(NCC)cccn3)=O)C2C)CCOCC1 N1(C(CC(CC)(F)F)=O)CC2OCCN(C(c3cnc4[nH]nnc4c3)=O)C2C1 C1(CNC(c2cc(O)ncn2)=O)CC2(CC(NC(C34CSCC3C4)=O)C2)C1 N1(C(c2c(C)cc(CC)o2)=O)CC2CCCC2(C(=O)NC2(C)CC(O)(CO)C2)C1 C(=O)(C(F)C(C)CNC(c1cnc(O)cc1C)=O)NC(c1cn(CC)nc1)C C(=O)(C(CC)CC(F)(F)F)NCC1(C)CCN(C(C(CSC)O)=O)CC1 CN1C(=O)OCC1NC(C1CC1c1cn(CCCCCCC2CC2)nn1)=O C1(COC)(CNC(c2cnns2)=O)CCN(C(C2(C(C)(F)F)CC2)=O)C1 c1(C(N(C(C)CNC(c2ncccc2C(F)F)=O)C)=O)c(F)cccc1C#N N1(C(c2n(C(C)C)ccn2)=O)CC(C(=O)NC2CCC3(CCC3)C2)CC(C)(C)C1 C1(OC)CCC(C)(C(=O)NC2CCCN(C(C3CCCN3C=O)=O)C2C)CC1 c1(C(C(=O)OC)N(C)C(c2ccccc2Cl)=O)ccc(F)cc1F.C1C(C)CN1 c1(OC)cccc(CCN(CC(C)C)C(C)C)c1F N=c1[nH]ccc(C(=O)NC2CCC(CNC(=O)CC(O)C3CCCC3)C2)c1Cl C1(C(=O)O)CC2CCCCC2N(C(CCCC2CC2)C(=O)NC)C1 c1(CNC(C(C)OCCOCC#C)=O)ccc(C(=O)N(CCCCC)C2CC2)o1 CCC(C)CCCC(=O)N1CC(C)C1C(N1CC2(C1)CN(C(C)=O)C2)=O CCCS(=O)(=O)CC(=O)NC12CCCN(C(c3c(C)cc(C)cc3O)=O)CC1C2 C12(C(N3CCC(C(C)NC(c4cc(=O)cc[nH]4)=O)C3)=O)CCCCC1OCC2 C(=O)(C#CC1CCCOC1)N1CCCCC(NC(c2ccc([N+](=O)[O-])o2)=O)C1 c1(-c2n(CC)c(N3CCCC(c4nnc(S)n4C)C3)nn2)ncc(C)cc1F c1(C(N(CC(O)CN(C)C(c2cc(C(F)F)no2)=O)C)=O)n[nH]c2c1CCOC2 N1(C(C2CC(C)C2)=O)CCN(C(=O)CCC(=O)c2ccccc2)CC(C)(C)C1 c1(C(N2C(C)CC(NC(=O)C=Cc3cnccn3)C2)=O)cc(F)cc(Br)c1O C1(CNC(c2nc(CNC(CC=C)=O)oc2)=O)CCC(C#N)C1 C1(CNC(Cc2cnc(C)s2)=O)(CO)CCN(C(c2sccc2C)=O)C1 c1(NCC2(OCC)CCCSC2)cc(NCC(F)(F)Br)nc(-c2ccccc2)n1 c1(C(N(C2CN(C(c3cnc4n3CCOC4)=O)C2)C)=O)c[nH]c2ccc(F)cc12 C1(CNC(CC2CCN(C)C2)=O)CCCCCN1C(c1ccc(C(N)=O)[nH]1)=O N1(C(CC=CC)=O)CCCC2(C1)CN(C(C1CCCN1C)=O)CCO2 C(CCCCCNC(=O)Cc1ccc(O)cn1)NC(C(C)CC1CCCCC1)=O O=C1CCC2(CC1)C(c1nc(CCC(F)(F)F)nn1CCOCF)C2 c1(OC)ccc(C(=O)NC2CCN(C(=O)OCC3(F)CCC3)C2C(C)C)cc1 c1(OC)cc(OC)c(CN2CC(F)(F)CCC2C)c(Cl)c1 c1(CC)ccc(F)c(C(=O)NC2(CF)CCN(C(=O)CCCN(C)C(=O)OC)C2)c1 CCCCS(=O)(=O)NC(C)C(=O)NCC(C)N(C(CNC(=O)CCOCCF)=O)C c1(N(C)C)cc(N2CCC(C(N(C(c3cccs3)C)C)=O)C2)nc(Cl)n1 C1(CN(C2CCSCC2)C(C2CCCCC2)=O)CCCCN1CCO C(=O)(C1=NOC(C)C1)N1CCC(C)(CC(=O)NCc2nnc(C)n2C)C1 N1(C(C=CCCC(C)C)=O)CC2C(NC(C3CC(=O)N(C(C)C4CC4)C3)=O)C2C1 CS(=O)(=O)C1CC(CNC(=O)C(=O)NC2CC3(CCCC3)C2)C1 c1(C(=O)NCC2CN(C(C3CN(CCC)C(=O)C3)=O)C(C)C2)cc(Cl)ccc1F c1(CC(=O)NCC(CNC(C(C)NC(=O)NC)=O)OC)cccc(F)c1F CC(C)CS(=O)(=O)CC(=O)NC1CS(=O)(=O)CC1N(C(=O)C(C1CCCCC1)=O)C CC(C)(C)C(CNC(c1csc(O)n1)=O)C(=O)NCC12CCC(CO1)C2 N=c1ccc(C(=O)NC2(CCNC(=O)Cc3cc(C(F)F)on3)CC2)c[nH]1 C(N=c1nc(N2CCC(OCCF)C2)c2c([nH]1)CCCCC2)C1(P(C)(C)=O)CC1 CCCC(C)(O)C(=O)N1CCC(C(=O)NCCc2cccc(O)n2)C1 c1(CN2CCC(C(N3CCc4c(nc(C)o4)C3)=O)C2)c(F)c(F)c(F)c(F)c1F C(=O)(CCCC(=O)OC)NCC1C(C(=O)NC(COCCCC)C)CCCC1 C1(NC(Cc2ccn(C(C)C)n2)=O)CC2(C1)CN(C(=O)CCN1CCCC1=O)C2 c1(C(=O)NC2CC(N(C(C(CC)O)=O)C)C2)cc(OC)cc2c1CCC2 C1(C#N)(C(=O)NCC(C)NC(=O)Cn2nnc(=N)[nH]2)CC1C(F)(F)F c1(-n2c(CC(O)C3CCC3)nc(CCCC)n2)nc2ccccc2[nH]1 c1(C(=O)NCCC2(C(=O)NC3CCCC3F)CCC2)cc[n+]([O-])cc1 c1(OC)ccc(F)c(CC(N2CC(CNC(c3cc(CO)[nH]n3)=O)C(O)C2)=O)c1 N1(C(C2CCSCC2)C(=O)NCSc2ccc(OC)cc2)CCCC(C)(O)CC1 N1(C(Cc2onc(C)n2)=O)CCCC(N(C(=O)CC2CC2(C)C)C)CC1 C1(F)(CNC(=O)Cn2cccn2)CCC(NC(c2cc[nH]c2C(F)F)=O)C1 N1(C(=O)CCC2CCCC2)CCN(C(C2CCCCS2)=O)C(C2CCC2)C1 N1(C(c2c(C#C)c[nH]n2)=O)CCOC(C)(CNC(c2cc(C3CC3)cs2)=O)C1 c1(C(=O)NCc2ccc(CNC(C(C)(C)SC)=O)cc2)cncc(Cl)c1C c1(C(=O)OC)ccc(C(F)(F)F)nc1NC(C12CCCC(C1)OC2)=O C1(NC(c2c(C)cco2)=O)CCC2CCN(C(C3CCCC34CC4)=O)C1C2 N1(C(C=CC2(C)COC2)=O)CCC2(CC1)CC2CNC(C1CC2SCC(C1)C2)=O C1(NC(CC(=O)NCC#C)=O)CCC2CN(c3cncc(Cl)n3)CC2C1 C(C(C)(C(=O)NC1CCC(C(=O)N(C)CC2CCCC2(C)C)C1)OC)OC N1(C(c2c(C)noc2C(F)(F)F)=O)CC(CNC(c2cscn2)=O)CC(C)(C)C1 Cc1nc2ccnn2c(C)c1CCC(=O)NCC1CN(C(C2CC2C(N)=O)=O)C1 C(=O)(C(F)(F)C(C)(C)O)N1CCC(C)C(NC(=O)C(O)Cc2cnn(C)c2)C1 c1(C(=O)NC(C)Cc2ccccn2)c(CNC(C2(C)CS(=O)(=O)C2)=O)nnn1C C#CC1CCN(C(C2CC2NC(=O)Cn2cc(-c3ccccc3)cn2)=O)CC1 c1(C(=O)Nc2scc(CC(=O)NCCN3CCC(C)CC3)n2)cnn2ccncc12 Cc1oc(CNC(C2(O)CC2)=O)nc1C(=O)NC1CCOC1C C1(NC(C(C=C)(C)C)=O)CC(C(=O)NCCNS(N)(=O)=O)=CC1O c1(C(C)NC(c2cn(Cc3onc(C)n3)nc2)=O)c(Cl)ccc(F)c1Cl O(N(C)C(=O)CN=c1nc2c(cnn2C)c(N2CC3CCOC3C2)[nH]1)CC N1(C(C2CC(C)N2C(C2CCc3n[nH]cc3C2)=O)=O)CCC(C)C(C)(C)C1 N1(C(c2ccc(C)cc2)C(=O)NCCC(=O)OCC)CC(C)C(F)(F)C1 CC1CCC(CC(=O)NCC(=O)NCc2ccnn2CCF)O1 N1(C(CCCC#C)=O)CC2CCC(C3(CNC(C)=O)N=N3)(C2)C1 c1(NC(C2(C)CCN(C(Cn3ncn(C)c3=O)=O)C2)=O)ccc(O)c(F)c1 N1(C(C=CCOC)=O)CC(CNC(=O)Cc2nc(C)no2)CC(C)C1 C=C1CC2(C1)CC(C(=O)NCCCOCCNC(=O)C(C1CCOCC1)C)C2 C1(C2CN(C(=O)C(O)Cc3ccc(Cl)cc3)C2)(NC(=O)CC2CCC2(F)F)CC1 C1(C(=O)NC(CC)CNC(=O)Cc2cccs2)CC=C(C)CC1 C1(F)(CNC(CC2CC(OCC)C2)=O)CCCN(C(=O)Cc2ncoc2C)CC1 CCCCC(O)C(=O)NCC1CCN1C(=O)COc1ccc(Cl)c(CC)c1 c1(C(N2CCC(C)(CNC(C3(CF)COC3)=O)C2)=O)cccc(Br)c1F C(=O)(C1CCCn2cnnc21)N(CC(O)CNC(=O)CCc1cccnc1Cl)C c1(CC(N2CCC(N(CCC)C(C34CCC3C4)=O)CC2)=O)cnc(Cl)cc1C C1(CCCNC(c2cc(Br)n[nH]2)=O)CCCCN1C(c1cn[nH]c1)=O Cc1c(CNC(C2CC(C)(F)C2)=O)sc2cncn12 N1(C(=O)C2CC2)C(=O)NC(c2ccc(OC(F)F)nc2F)C2=C1CN(CC)C2=O C1(C(F)(F)F)(C(=O)NCC2N(C(C(c3ccnn3C)C)=O)CC=C2)CC=CCO1 O=[N+]([O-])c1cnn(-c2nnc(NC(c3cnccc3F)=O)s2)c1 c1(C(=O)NC2(C)CCN(C(c3cccn(C)c3=O)=O)C2)cc(Cl)c(F)c(Cl)c1 c1(C(=O)OC)ncc(NC(C23CCC2CN(S(=O)(=O)CCCCl)C3)=O)cc1Cl C1(C)(CC(=O)NCC2(NC(C(CC=CCC)C)=O)CC2)CCS(=O)(=O)N1 C1(=O)CC(C(F)(F)F)N1.N1(CC(=O)NC(C)C(C)NC(=O)C2CC2)CSCC1=O C1(NC(N2CCCC(O)(Cc3n(C)ccn3)C2)=O)CCC2CCC1OC2 c1(N)ccc(O)c(CO)c1.Cc1cn(C)nc1C(=O)Nc1ccccc1C1(CO)CC1 C=C1CC2(C1)CC(C(=O)OCc1ccc(C(=O)NCCOC(C)(C)C)[nH]1)C2 C(CCCC(C)(C)C(=O)NNC(=O)c1ccc(C)s1)NC(C(CC)C)=O C(C#Cc1cn(Cc2ncoc2C(F)F)nn1)NC(C(CC(C)C)=O)=O N1(C(C(C)C2CCOC2)=O)CCC=C(CNC(=O)Cc2ccon2)C1 N1(C(CC(CC)(C)C)=O)CC2CC1CCN2C(=O)C(C)Cc1cnn(C)c1 N1(C(COCC)=O)C2CCC1CC(NC(C1CC(F)(F)CS1)=O)C2 C1(CNC(c2nc(CCCCC)sc2)=O)CN(C(=O)CCC(C)SC)CCO1 C(CS(=O)(=O)CC(=O)NCc1cnn(C)c1)OC.c12ccc(C)c(c1)NC2=O N1(C(c2n(C=C)ncc2)=O)CC(C)(C)OC2(C1)CN(C(=O)CCC(=O)NC)C2 Cc1nc2cc(CCN(C)C)c(F)cc2[nH]1.c12cn(nn1)C(C)C(=O)N1CC2C1 Cc1cc(N)n(CC(=O)NC2CC(CNC(=O)C(=O)NC3CC3)C2)n1 Cc1noc(C)c1CSCC(=O)NC(C)C(C(C)C)NC(C1CC(O)C1)=O C(=O)(C1=CC2(CCOCC2)C1)N1CC(CC)N(C(=O)CC2CSCCS2)CC1 C1(C(=O)NCCCCNC(CCC(C)(C)OC)=O)CC2CCCCN2C1 c1(OC)cnc(-c2ccc(-c3nccn3Cc3nnc(C(F)(F)F)o3)s2)nc1 N1(C(C2(S(N)(=O)=O)CCC2)=O)CCCC(C2(NC(c3cnc(O)s3)=O)CC2)C1 c1(OC)c(NC2CCN(C(=O)Cc3ccc(Cl)nc3C)C2)ncnc1C Cc1nn(C)c(C)c1C(=O)NCC(C)N(C)Cc1nc(C(F)(F)F)cs1 c1(C(=O)NCC(CO)NC(c2c(C(C)C)onc2)=O)ccc2c(c1)OCC(=O)N2 N1(C(C2(C)CCCN(C(C3CCCCC3(F)F)=O)C2)=O)CCC2(C1)CC2(F)F C#Cc1cc(C(=O)NCC2CN(C(=O)Cn3ccccc3=O)CCO2)ccc1C C1(C)(C(=O)NCC2CC(OC)CN2C(=O)C(=O)C(C)(C)C)CCCNS1(=O)=O CCC(CC(F)(F)C)C(=O)NC1CN(C(c2ccncc2C(F)(F)F)=O)CC1C C1(c2cn(C34CN(C3)C4=O)nn2)CC2(CC(=O)C2)C1.C1(C(=O)OC)CC1C(F)F C#CCC(CC(F)F)C(=O)N1CCC2(CC1)CC2C(N(C)C[Si](C)(C)C)=O Cc1ccc(CN(CCO)Cc2cccc(-n3ccc(C)n3)c2)cc1 C1(NC(=O)COC2CCCOC2)(CO)CCCN(C(c2nocc2C2CC2)=O)C1 Cc1sc(C(=O)NC2CN(C(=O)CCN3CCC(F)C3)CC2C)nc1O c1(C(=O)NCC(C)CN(C(=O)CC(C)C2CC2)C)ccc(Cn2cccn2)o1 CC1C(Cl)CCN1C(=O)CCC1CC(NC(=O)CC2CC3CC3C2)C1 C1(F)(C(=O)Sc2c(NC3CN(C(C4CCC4)=O)C3)nccc2)C2CCCCC12 N1(C(CCc2cn(C)nn2)=O)CC=CC1(C)C(=O)NC(C(O)CO)C1CC1 C1(C(=O)NC23CC(CNC(CC4C(C)OCC4)=O)(C2)C3)CN2CCC1CC2 Cc1cc(NC(C2CCCN2C(=O)Cc2nc(C)c(C)[nH]2)=O)cc(C)c1C C1(CC=C)(CNC(=O)C(C2(O)CN(C(=O)C=C3CCC3)C2)F)CCCC1 C1(C(=O)NC2CC(NC(c3n[nH]cc3C(F)(F)F)=O)C2)Cc2ccc(F)cc2O1 CC(CCNC(c1cc(CNC(C2CC3(CCCO3)C2)=O)no1)=O)C(F)(F)F C1(C)(Cc2nc(-c3cc(COCC)c(C)o3)on2)CCC(C)=C(C)C1 N1(C(=O)C=C(C)C(C)C)CC2CC1CN2CC(=O)N(c1cccc(C(C)C)c1)CC CC1=NOC(C(=O)NCC2(O)CC(NC(c3cc(C(C)(F)F)n[nH]3)=O)C2)C1 c1(C(N2CC(OC)(CNC(=O)CC3CC(C)(C)CO3)C2)=O)cc2ncccc2o1 C(=O)(C1=NOC2COCC12)N1CC2(CN(C(C3(C(=O)OCC)CC3)=O)C2)C1 C1(N(C)C(c2nn(C)cc2Cl)=O)CCCC2CN(C(C34CC(F)(C3)C4)=O)CC12 c1(COC(C(C)(C)N(C)C)=O)ccc([N+](=O)[O-])cc1Br CCC(C)C(C(=O)N(C(C)CN(c1ccnc(SC)n1)C)C)OC c1(C(=O)NCCN(CC(C)O)C(c2c(C)nc(C3CC3)o2)=O)ccc(=O)n(C)c1 C1(NC(Cc2cc(C)nn2C)=O)CC(F)CN(C(c2cncn2C(F)(F)F)=O)C1 C1(CCNC(c2ccoc2)=O)CCN(C(c2csc(-c3cccnc3)n2)=O)CC1 C=CC(C)CC(=O)OC(C(C)OCCC)=O C1(NC(c2cnc(OCC)nc2)=O)CN(C(C23CC(CC(C)O2)C3)=O)CC1(C)C c1(C(C(=O)Nc2c(CC)noc2)NC(=O)C(F)OC(F)(F)F)c(C)cccc1Br C1(NC(c2ccc(C(C)C)o2)=O)C2CC1N(C(=O)C(C)c1cc[nH]n1)C2 CCC(C)C(O)C(C)C(=O)N1CC(CNC(c2nc(C)ccc2C)=O)C(C)(C)C1 C=CCC(C(=O)NC1CCN(C(=O)CC2CCOCC2)C1CC1CC1)C(C)C c1(CC(=O)NC2CC(NC(CN(C)C3CC3)=O)C2)cc(C(F)(F)F)ccc1Cl c1(C(N(C2CCC(C)C2)CCO)=O)ncc2c(F)cccn12 c1(SCC=C)nnc(CCO)n1N.c1(-n2ncc(SCC)n2)ccc(F)cc1 c1(OC)ccc(-c2nc(C3CCCN(C(C)=O)C3)n(CC(C)C)n2)nc1 c1(C(N2CCC(c3nncn3C)C2)C(=O)NC(C(=O)OC)C)ccc(F)cc1 c1(OC(C)C(N2CCC(NC(=O)Cc3ccnc(F)c3)C2)=O)ccc(F)cn1 C1(C(=O)NC2(CO)CN(C(CC3(CO)CC(C)(C)C3)=O)C2)CC12CCCCC2 c1(NC)nn(C)cc1C(=O)NCCNC(c1cc(C(=O)OC)no1)=O CC1CCCCC1C(=O)N(CC(O)CN(C(=O)CN1CCC(C(N)=O)CC1)C)C Cc1nc(CC(=O)N(C)CC2CCN(C(C3CCCCC3)=O)CC2)[nH]c1C c1(C(C(=O)NC)N(C)Cc2nnc(C(C)(C)C)o2)ccc(C)cc1 N1(C(c2cc(C)c(C)o2)=O)CCN(C(=O)C=CCCc2ccccc2)C(C)C1C C(CC1CC1)(C(=O)N(C1CCC2CC12)C)OC(C)C(=O)NCCOCC1CC1 N(S(=O)(=O)N1CCC(C)CC1)CC(N1CC(C)OC(C)C1)C C(=O)(C(F)C(F)(F)F)NCC=C1CCN(C(C2(C#N)CCCO2)=O)CC1 c1(C(C(=O)NC(CN(C(CNC(C(CC)C)=O)=O)CC)C)C)ccc(F)cc1 C(C(=O)NOCCCCF)(c1ccoc1)NC(=O)CCCC1CCCC1 c1(CC(=O)N(CCNC(C2(C#C)CCCC2)=O)C)ccc(OC)cc1OC N1(C(c2cc(C)cc(Cl)n2)=O)CC(F)C(N=c2ncnc3[nH][nH]c(I)c2-3)C1 c1(C(C)(C)C)ccc(C(=O)NC2CCC(CNC(c3c[nH]c(=N)o3)=O)CC2)nc1 N1(Cc2cc(C)sc2)CCC(C(=O)N(CCCCC#N)CCN2CCCC2)CC1 C1(C(N2C(C(C)NC(c3cc(C)oc3)=O)CCCC2)=O)CC(S(C)(=O)=O)C1 C(C(=O)N(C1CC1)Cc1cccnc1C)(C(C)(C)C)N1CCCC(CCC)CC1 C=CCCC(C)(C)C(=O)N1CC(CN(C)C(c2csc(C(C)C)n2)=O)C2(CC2)C1 C1(CNC(C2CCC3CC3C2)=O)CC2(CC2)CN1C(C12CC(C1)C2)=O c12ccc(cc1)Oc1cc(ncn1)N1CCC(C1)NC2=O.c1(COC)c[nH]c(Br)c1 C(=O)(CCS(N)(=O)=O)NC1(C(N2CCCC(CN(C)C(N)=O)C2)=O)CCCCC1 c1(C(=O)NCCC2C(C)CN(C(C3CCCN3C=O)=O)C2)ncnc(O)c1Br C(=O)(CCCCCN(C)C)NCC(CNC(c1ccc(-c2ccc(C)o2)s1)=O)O c1(C(=O)NC(C(N2CCN(C(=O)NC)CC2)=O)CCC2CC2)ccc(O)c(F)c1 N1(c2ccc(C#N)cc2Cl)CCOCC2(COCC3CCCCN23)C1 c1(CC(=O)NCC2(CNC(CSC)=O)CCCCC2)ccnc(F)c1F c1(CNC(c2cc(-c3ccccc3)cs2)=O)cccc2c1CNC2 N1(C(c2ccc(OC)s2)=O)CCC(C2CCN(C(=O)Cc3ccn(C)n3)C2)C1 c1(C(=O)OC)ccc(Oc2ccccc2NC(c2ccn(C)n2)=O)cc1 C1(C(N(CC(C(C)C)OC)C)=O)(CO)CCN(C(=O)C(C)Cn2ccnc2)C1 C(=O)(C1CCCCc2ccccc21)N1CCC(C(C)NC(=O)C2=CCSC2)CC1 C1(NC(c2cc(CC)cc(F)c2)=O)CC12CCN(C(c1conc1C)=O)CC2 C1(C(F)(F)F)(COC)CN(C2CCC(Oc3ccncc3)C2)CCO1 N1(C(C(C(C)C)CO)=O)CCC2(CC1)CCN(C(=O)CCc1ccc(F)nc1)C2 N1(C(=O)COC2CN(C(C3(F)CC=CCC3)=O)C2)CCN2CCC1C2 Cc1sncc1C(N1CCC(N(C)C(c2cc(C3CC3)no2)=O)C1)=O C1(C(C2CCN(C)C2)=O)C=CCCC1C(=O)NC1CC1.N1(CC(=O)OC)CCCC1=O N1(C(c2cc(C(C)C)nn2C)=O)CCCC(O)(CCNC(C2(C)CCOC2)=O)C1 c12ccc(F)c(c1)Cn1cc(nn1)C(C1CC1)C1CN(C1)C2=O.C1(CO)CC1 c1(C(N2CC(CNC(C=CC)=O)C3C2C3)=O)cc2ncccc2cc1Cl C1(NC(C(F)=CC)=O)CCCN(C(c2ccc(C)c(N)c2)=O)C1C c1(C(=O)NCC(C2CCC2)NC(c2cnn(CC)n2)=O)c(C)cnnc1O N1(CC(=O)NC2CC(NC(CN(C(=O)OC)C)=O)C2)CCCCCC1=O C1(NC(=O)OC(C)(C)C)COCC2(CCN(OC)C2)O1.C123CC1CCC2C(=O)N3 c1(-n2ccc(C(=O)NC3CN(C(COC)=O)CC3C)n2)ccc(Cl)cc1Cl C1(CC)C(C(=O)NC2CCCC2OC)CCN1C(c1oc(C)nc1C)=O C1(C(F)(F)F)(C(N(C2CCN(C(=O)Cn3cc(Cl)cn3)C2)C)=O)CCCCO1 CC(CCCCNC(=O)CC1CCCN1C)NC(=O)CSc1n[nH]c(O)n1 c1(OC)ccccc1NC(=O)C(N1CCCC1Cc1ccsc1)C1CC1(C)Br C(C(=O)O)(C1=CCC=CC1)C(NNC(Cc1c(OC)cc(Br)cc1)=O)=O Cc1ccc(C#N)cc1NC(=O)C(C1CCCO1)NC(=O)CC1C(C)(C)C1(C)C c1(C(N(C(C)CNC(c2cncnc2O)=O)CC)=O)cc(F)cnc1O C12(CNC(c3ccc(C)nc3N)=O)CCC(CC1)N(C(C1CSCCS1)=O)C2 c1(C(N(C2CN(C(C(C)NC(CC)=O)=O)C2)CC2CC2)=O)cc(C)ns1 Cc1cccc2ncc(C(=O)NCC3CCCCN3C(=O)CC(C)(C)C(F)F)n12 Cc1[nH]nc2c1CCC(C(N1CCN(C(c3ccc4c(c3)OCC4)=O)CC1)=O)C2 C1(O)(CNC(C(C)OCC2CC2)=O)CCCN(C(C2CC3CCC(C2)S3)=O)CC1 c1(C(N2CCC(N(C(=O)CSCC)CC#C)CC2)=O)cccc2nc(C)nn12 N1(C(c2cc(CC)[nH]n2)=O)CCC(O)(C(C)CNC(c2ocnc2C)=O)C1 C1(CNC(=O)Cn2cccnc2=O)CC2(CC2)CN1C(c1cnn2c1OCC2)=O N1(C(C(CCCCC)O)=O)CCC(N(C(=O)CC(C)OC)CC)C(F)(F)CC1 Cc1cc(O)ccc1CN(CC#N)Cc1nn[nH]n1 N1(C(C(C)N(C)CC)=O)CCC(NC(C2(NC(c3nscc3C)=O)CC2)=O)CC1 c1(C(=O)OC2C(C)(C)CCC2)cc(F)cc([N+](=O)[O-])c1 N1(C(c2n(CC)ncc2Cl)=O)CCN(C(=O)CNS(N)(=O)=O)CC(O)C1 C(=O)(CC(F)(F)C(F)(F)F)NC(CC=C)CNC(c1cccc(C)c1N)=O CN1CCC(O)(CC(=O)NC2CN(C(=O)Cc3ccncc3Cl)CC2(C)C)CC1 CC1CN(C(=O)C(F)(F)c2cscc2Br)CC1NC(=O)C(C)(C)F N1(C(c2c(C)cnnc2)=O)CC(F)(F)CC1(C)CNC(=O)C(c1ccnn1C)O Cc1cc(C(F)(F)C(=O)NCC(C)NC(=O)C(C)N(C)C)cnc1Cl N1(CCC)C(=O)NC(c2ccc(F)c(F)c2)C(C(=O)OCCOC)=C1C c1(CC)cc(C)ccc1NC(=O)CCCSC(C)(C)C N1(C(C(F)=CC)=O)CCC(C(C)(O)CNC(c2ccnc(C(F)F)c2)=O)CC1 CCCC(CNC(=O)C(O)CC(C)C)C(=O)NC(c1nn(C)cc1O)C c1(C(=O)OC)sc(=NCC2CCCC(NC(C3(O)CCC(C)CC3)=O)C2)[nH]c1Cl C(CN=c1[nH]c(=NCCSC)[nH]c2cc[nH]c12)=CCCC.c1ccccc1C#N c1(C(=O)NC2CC(NC(C3N(CC)CC3)=O)C2)cc2nnn(C)c2s1 C12(C(N3CC(C)C(CO)CC3)=O)CCC(CN(C(=O)CC(C)(C)C3CC3)C1)C2 N1(C(CC(C)C2CC2)=O)CC2(CCC(NC(C3CCC(C)(C)O3)=O)CC2)C1 O=C(CN=c1cc[nH]cc1)N1CC2CCCC2(CNC(C2(Cl)CC2(F)F)=O)C1 c1(OC)cccc2c1OC(c1nc(C(C)N)no1)C2 c1(N)cc(C(N2CC(N(C(=O)C(CC)n3nccc3C)C)C2)=O)[nH]n1.C(=O)OCC c1(C(=O)NC2CCC(NC(Cc3onc(C)n3)=O)C2)cccn(C(C)(C)C)c1=O Cc1nc(C(=O)NCC2CN(C(=O)C(C)(C)C3CC3)CC2C)cc(O)n1 C#CC1(N(C(COOC(F)F)C(=O)NC(C)(C)C)C)CCCCCC1 CC1CCN(CC(c2cn(C)nc2C(F)F)=O)CC1C Cc1ccnc(C(N2CCOC(CC(=O)NCC(C)C(C)O)C2)=O)c1F C1(NC(=O)CCCF)CCC2(CC1)CCN(C(C13CC1COC31CCC1)=O)CC2 c1(C(=O)NC2CCCN(C(C(C(C)C)OC)=O)C2)cc2ccc(Cl)cc2c(=O)o1 C1(CC(N)=O)(C(=O)NC23CC(CNC(=O)C=Cc4cc[nH]n4)(C2)C3)CCCC1 c1(C(C(=O)NC2C=CCN(C(C3(SC)CCC3)=O)C2)(C)C)cc(Cl)ccc1F n1(CC)nc(C(=O)NCC2(CNC(c3snc(C)c3N)=O)CCCCC2)cc1O N1(C(c2c(OCC)cco2)C(=O)NCCSC)CCCC(N=[N+]=[N-])C1 CCCCCC(O)C(=O)NCC(C)CNC(=O)CCCCO N1(C(CCOC(C)=O)=O)CCCC2(CCCN2C(C2CC(C)C2)=O)C1 C1(O)(C(C)NC(CNC(CC(C)C)=O)=O)CCN(C(C2CC2(Cl)Cl)=O)C1 N1(C(C2CC(C)(N)C2)=O)CCCc2cc(NC(=O)C(F)(F)F)ccc21 N1(C(C=Cc2n(CC)ccn2)=O)CCC(C)CC1CNC(c1c[nH]c(C#N)c1)=O c1(NC(C=CC(C)NC(=O)C(=O)N(C)C)=O)cc(F)ccc1N1CCOCC1 CCCC(C)CC(=O)NC1CC1NC(c1cccc(OCCOC)c1)=O c1(C2C(C(N(C3CCC(NC(=O)COC4CC=CC4)C3)C)=O)C2)ccccc1F CCCCC(CC)CCC(=O)NC(C1CCCC1)CNC(=O)CCn1ccnn1 O=C(CCCCCNC(c1ccc(=N)[nH]n1)=O)NCc1ccc(O)cc1F c1(C(=O)NCC(CNC(c2cc(CC)ncc2)=O)F)cc2ccc(Cl)cc2s1 c1(C(CNC(N(c2ccccc2)CC)=O)C)snnc1C C1(C(=O)NCC2C(NC(c3nccn4ccnc34)=O)CC2)CCCCC(F)(F)C1 CC1(C)CC(C(N2CCC(NC(=O)CC3=CCOCC3)C(O)C2)=O)CC(C)(C)O1 c1(COC(c2ccc(F)c(I)c2)=O)ccc(C(F)F)c(Br)c1 C1(NC(CC(C)c2ccco2)=O)CN(C(=O)CC2CCCC2)CC12CC2 CCC(C)(C(=O)N1CCC(NC(=O)COc2ccc(F)cc2Cl)C(O)C1)C(N)=O CC1C(C(=O)N(CCC(O)CO)C)CCCN1C(=O)C1=CCCOC1 Cc1c(NCCCSCC(C)(C)C)ncnc1N1CCN(C)C(c2ccccc2)C1 C(N=c1[nH]c(=NCC2CCOCC2)c2[nH]ccc2[nH]1)C1(Br)C(F)(F)C1 N1(C(C(N2CCOCC2)C)=O)CCC(C2CCCC2C(=O)O)CC1 c1(NC(C2C3CC2N(C(c2cc4sccn4c2)=O)C3)=O)cc2ccccc2[nH]1 C1(C(=O)NC2CCN(C(CSCCCC)=O)C2C2CC2)CCC2(CC1)CC2CO O=C(C1=NOC2COCC12)NCC1CN(C(C23CC(CO2)C3)=O)CCO1 C1(CC=C)(NC(C2CCC(F)(F)C2)=O)CCCN(C(=O)C(O)C(F)F)C1 C1(C(=O)NCC2C(C)(C)CCN2C(=O)C=CC2CCC2)CCC2(CC1)CC2(F)F c1(C(C2CCCC2)CN2CCCC(c3ccc(C)cc3)C2)nnc2n1CCCC2 CCCC(C(=O)N1CC(N(C)C(C2CC3CC2CC3(F)F)=O)C1)C(C)C C1(CNC(Cc2cc(C(C)C)no2)=O)CC(NC(=O)C(C2CC2)C2CC2)C1(C)C C1(NC(C2(C(=O)N(C)C)CCC2)=O)CC2CC1CN(C(C1(CC)CC1)=O)C2 N1(C(C2CC(C(F)(F)F)CN(C=O)C2)=O)CCC2(CCCNC2=O)CC1.CO N1(C(C2(F)CC(C(=O)OC)C2)=O)CC(CNC(=O)CN2CC3CC3C2)C(C)C1 S(=O)(=O)(c1cc(-c2ccccc2)[nH]c1C)NCC(C(=O)OC)C CCC(CC)(CCNC(c1cc(COC)cs1)=O)NC(c1oc(C)cc1C)=O Cc1ccc(F)cc1C(=O)NC1CC2CCC1N2C(C1CC1c1ccco1)=O c1(C(=O)NCC(COC)S(C)(=O)=O)cc(Br)cc(I)c1N C1(NC(C2C(C)C2)=O)CC1C1CCCN(C(C2CCC([N+](=O)[O-])CC2)=O)C1 c1(CNC(=O)OC(C)(C)C)ccc(Cl)c(C)c1.C1(C2CC2)C(=O)N1 C(c1nc(C)c(C)[nH]1)=CC(=O)NCCC1(O)CCN(C(C2C(C=C)CC2)=O)C1 C(=O)(C1=CC(O)C(NC(=O)CCCC2CCCC2)C1)NCC1CCC(=O)NC1=O C1(c2nnnn2CCCC2CC2)(C(C2CC2)NC2C(CO)C2)CCSC1 N1(C(C(n2cc(C)nc2)(C)C)=O)CCC(NC(=O)C2=COCCC2)C(CO)CC1 c1(OC)cc(OC)c(C(=O)NC(C)CN(C(=O)C(C)c2cncs2)C)c(F)c1 C1(C(=O)NCC(C)(O)C2CCCC2)CCCCN(C(=O)CCCCC2CC2)C1 c1(C(C(=O)NC(CC)CNC(C2CC(C)(F)C2)=O)N(C)C)ccc(Cl)cc1 c1(C(N2CC(O)(CNC(c3cnc(CC)[nH]3)=O)C2)=O)ccc2nn[nH]c2n1 c1(OC)nccc(C(=O)NC2CCCC2CNC(C2(OC)CCC2)=O)n1 C1(C(=O)NC(C2(OC)CCC2)C)C2CCN(C(c3cc(O)cc(F)c3)=O)CC12 C1(OCCCNC(C(CC)n2ccnc2)=O)CCN(C(C2(C)C=CCC2)=O)CC1 c1(CN2CCN(C(C(C)n3cncn3)=O)CC2C#N)cccc2ccncc12 C1(OC)CN(C(c2ccc(C)n2C)=O)CC1NC(=O)C(C)NC(N)=O C(CC(=O)Nc1cc(C(C)(C)C)cc(O)c1)(C(F)(F)F)c1cccc(OC)c1 C1(CC(=O)NC2CC(OCC(=O)NCCCOCCC)C2)CSCCO1 C1(NC(C2C(C=C)C2)=O)CCC(N(C(=O)COCCC)C)C1 c1(CC)cc(C(=O)N(CC(C)NC(=O)CCOCCF)CC)ccc1Cl O=S(=O)(c1ccc(Cn2cc(Br)cn2)cc1)Nc1cccc2c1COC2 c1(CCN=C(NC2(C)C(C)(C)C2)NC2CC2)c[nH]c2cc(Cl)cc(Cl)c12 c1(C(N2CCC(C(=O)NCCC(C)(C)O)CC2)=O)cc(I)c(F)cc1F CCCC(C#N)C(=O)NC1CN(C(c2cc(Br)ncc2OC)=O)CC1C N1(C(c2n(C(C)C)ncc2)=O)C2CCC1(CNC(=O)CCn1ccnn1)CC2 c1(C(=O)NCC(CN(C)C(c2cnsc2)=O)O)ccc(OC(F)(F)F)cc1F N1(C(c2c(C)con2)=O)CCCN(C(c2cccc(C(=O)N(C)C)c2)=O)CC1C N1(C(C(c2cccc(C)c2)O)=O)CC2(CC(NC(=O)CCc3cc[nH]n3)C2)C1 C1(O)(C(=O)NCC2CCN(C(=O)CCc3nccs3)C2)CN2CCC1CC2 Cc1ccc(O)c(CN2CCC(F)(C(=O)NCc3cccc(F)c3)C2)c1 CC1=C(C(=O)NCc2nc(C(=O)NCC3(CCO)CC3)c(C)o2)COCC1 C1(C(=O)NC(CCC)C(N2CCCC3(CC3)C2)=O)CC2(CCC2O)C1 c1(C(C)NC(C(C=C)O)=O)ccc(CNC(c2csc(CC)c2)=O)cc1 C1(NC(c2cc(CCOC)on2)=O)CC(F)CN(C(C2CCCC(F)(F)C2)=O)C1 c1(N2CCC(C(C)NC(=O)C(c3ccc(Cl)c(Cl)c3)C)CC2)nc(Cl)ncc1Cl Cc1nc(C(=O)NC2CCC(CNC(c3ccccc3N(C)C)=O)C2)c(C)o1 N1(C(C(N)=O)=O)CC2(C(=O)NCC3COC(=O)C3)CC1CCO2 c1(NC(C(N2CC(CC)OC(C)C2)=O)=O)ccc(S(C)(=O)=O)nc1 C1(CCCNC(C(c2ccccc2)C)=O)CCCN1C(c1cc(C(N)=O)[nH]n1)=O Cc1nn(CC(=O)NCC2(C)CCCN(C(C34C=CC(CC3)C4)=O)C2)c(C)c1C C1(C(=O)NC23COC(CNC(C4(F)CCCCC4)=O)(C2)C3)C2(CCC2)C12CCC2 C1(NC(C(CCOC)(C)C)=O)CN(C(C2CC2(Cl)Cl)=O)C2(CCOCC2)C1 N#Cc1ccc(Cc2noc(C3CC(OC(F)F)C3)n2)cc1 C1(CC(=O)NC(C2CCCC2)C)CCCN1C(=O)CCc1cnn(C)c1 c1(CN(CC(O)CNC(=O)CCC2CC2CC2CC2)C)ncn2ccccc12 CC(C)(C(=O)NC1CCC1NC(C1COC(=O)N1)=O)c1ccsc1 C(CCS(C)(=O)=O)(C(=O)NC(C)(C)CN(C)C(C1CC1C(C)(F)F)=O)OC N1(C(c2c(C)nc(C(N3CCCC(C(C)C)CC3)=O)o2)=O)CCCC(N)C1C.CC C1(OC)CN(C(C2CCCCN2C)=O)CC1C(=O)NC(C1(OC)CCC1)C c1(C(C(=O)NCC2(F)CC(CNC(CC(C)SC)=O)C2)=O)ccc(F)cc1 N1(C(C2CN(C(COCC#C)=O)C2)=O)CC2(CO)CC2(CO)C1.C1CC(=O)N1 CC1(C)CC(CC(=O)NC2(C)CC3(CC3)C2)N(C(=O)C2=COCCC2)C1 c1(C(N2CC(N(C)C(c3cc4sccc4n3C)=O)C2)=O)ccc([N+](=O)[O-])cc1F C(=O)(C(F)(CNC(c1nonc1CC)=O)C(C)C)NCC(CCC)(C)O C1(NC(=O)NC(C23COC(C2)C3)C)CCC2C3C=CC(C3)C12 C(CC)(C(=O)N1CCC(N(C(=O)CCN(C(CC)CC)C)CCOC)C1)OCC C1(NC(C2(C)CC2(F)F)=O)CCCCN(C(C2CC3(C2)CC(O)C3)=O)C1 c1(-c2c(OCC)cc(C(C)=O)cc2)ccc(Br)c(C)c1C C1(C(C)NC(c2csc(-c3cnc[nH]3)n2)=O)CCCN(C(=O)COC2(C)CCC2)C1 C(=O)(CS(N)(=O)=O)NC(C)CNC(=O)C(c1cscc1Br)N(C)C c1(CC)nc[nH]c1C(N1CC(O)(CN(C(=O)C(n2cc(C)cn2)C)C)C1)=O C1(NC(C2CC2F)=O)CC2CCC1N(C(c1cccc3oncc13)=O)C2 c1(C(=O)NCC2(F)CC(CNC(c3c(C)nncc3)=O)C2)cc([N+](=O)[O-])oc1C CCC(C)C(O)C(C)C(=O)NC(CC(=O)NC(C)(CO)C(F)(F)F)C(F)F CC(C)C(C(=O)NCc1ccc(C#N)o1)C(C)NC(C1CS(=O)C1)=O Cc1ccc(C)n1-c1cn(CC(c2nc(C(=O)O)cs2)N(C)C)nn1 n1(CC)nc(C(N2CCC(C(=O)NC3CCCC(COC)C3)C2)=O)cc1O Cc1cccc(OCC(c2cn(C3CCOCC3)nc2C)=O)c1C Cc1cc(NC(=O)C(CC2CCOCC2)NC(=O)CC2CSCCO2)cnc1Cl c1(NC(c2cccc(C)n2)C)ncccc1S(=O)(=O)N1CC2CCC2(C)C1 Cc1ccc(N2CCN(C(=O)C(=O)NC3CCCC3(F)F)CC2)cc1N N1(C(C(=O)NCC23CC(F)(CO2)C3)=O)CCC(C2CC2)C1 c1(C(N2C(C)CC(NC(C(NOC)=O)=O)C2)=O)cc([N+](=O)[O-])c[nH]1 Cc1cc(C)n(CC(=O)NC2CN(C(=O)CC(C)C)C3CC23)c(=O)n1 CCCCCC(C)CC(=O)N1CCC2CN(C(c3cc4c(s3)CCC4)=O)C2C1 C1(C(=O)NC(C)CC2CCC2)CN(C(C2CCN2C)=O)CC12CC2 C1(C(N(C)CC2C(NC(c3c(C)onc3)=O)CCC2)=O)OCC2CCCC12 C1(C(=O)NCCCCCCNC(c2c(C)noc2C(C)C)=O)CCCS(=O)(=O)N1 N1(S(CC2(C(=O)OC)CCOCC2)(=O)=O)CCC12CCOC(C)(C)C2 C1(N(C)C(=O)NC2(CC3CC3c3ccncc3)CC2)COCC1(C)C CCCC(O)CC(=O)NCCCC(C)NC(c1ccc(C#N)o1)=O c1(C2(N(CC(N3CCCC34CC4)=O)C)CCC2)ccc(Br)nc1 C1(C(N(C2CCN(C(=O)CCCc3ccsc3)C2)CC)=O)CC2(CCCCO2)C1 Cc1cnc(N)c(C(=O)NCC2CCN(C(c3cnc(C4CC4)s3)=O)CC2C)c1 C(=O)(C1CCCc2nnn(C)c21)N1C(CNC(C(C)Cc2cnn(C)c2)=O)CC1 C(=O)(CC(C(F)F)NC(=O)C(F)C(C)(F)F)NC(C(=O)N(CC)CC)C N1(C(C(CC)C#N)=O)CCC2(CC1)CC(CNC(=O)COCC1CCCO1)C2 S(=O)(=O)(c1c[nH]ccc1=NCC1CCCCO1)N(CC(CC)OC)C CC1CC(NC(C2(C)CCOCC2)=O)CN1C(c1ncncc1F)=O N1(C(C2(CC)CCCC2O)=O)CCCN(C(=O)C(=O)Nc2ccc(C)cc2)CC1 c1(C(N(CCCCCNC(CCOC(C)C)=O)C(C)C)=O)cc(F)ccc1O C(=O)(CC(O)C(C)CC)NCC(=C)CCNC(c1ccccc1CO)=O c1(N2C(C(=O)N=c3[nH]nc(Cl)cc3Br)CC(OC)C2)ncnc2cccc(F)c12 c1(C(N(CC(C)NC(=O)C(O)CN2CCCC2)CC)=O)cc(Cl)c(Cl)s1 c1(C(=O)NCCCC(C)NC(C(C(=C)Cl)(C)C)=O)cc2ccc(O)nc2s1 c1(NC2CC(C)N(Cc3ccccc3)CC2)cccc2cccc(Br)c12 c1(C(=O)NCC2C3CN(C(C4(C)CCC4)=O)C2C3)ccc(S(=O)(=O)N2CCC2)o1 C(=O)(CCN1C(=O)CSc2ccccc21)Nc1nnc(CCC(=O)OC)s1 N1(C(C(CC)C(C)(F)F)=O)CCCC2(C1)CN(C(c1c[nH]c(C#N)c1)=O)CCO2 C1(NC(C(C)OCC#C)=O)CN(C(c2cccc(CN(C)C)c2)=O)CCC1F N1(C(CSCCN(C)C)=O)CCC(C(C)(C)CNC(C2CNC(=O)C2)=O)CC1 S(=O)(=O)(c1ccc(Br)c([N+](=O)[O-])c1)NCCc1ncn(C)c(=O)c1 C1(CC)CCCN(C(c2cn(C)c(C)n2)=O)C1C(=O)NCC(=O)NCC1CC1 C=CCC(CC)C(=O)NC12CCC(C1)N(C(c1cccc(NC)n1)=O)C2 O=C(C#CC1CCC1)N1C(C(=O)NC(c2ccc(F)cc2)CO)CC2CC12 c1(C(C(=O)Nc2scc(CCOC)n2)N(N(C)C)C)nc(NC(C)=O)ccc1C CCC(CC(=O)N1CCC(CN(C)C(c2ccnc(C(F)F)c2)=O)C1)SC C1(N(C(CC=CCCCCC)=O)C)C=CCCC1C(=O)NC(C1CCC1)C Cc1[nH]c(C(=O)NCC(C)CNC(=O)CC(C)n2cc(Br)cn2)c(C)c1C CCC(C)CC(=O)NC1CCC1CNC(C1CC(CC(C)(C)C)C1)=O C1(CNC(Cn2nnc(C)n2)=O)CC(C(F)(F)F)CN1C(C1(C)CC1(F)F)=O C12(C(=O)Oc3c(CC#N)cccc3)COC(C)(CN1Cc1ccccc1)C2 N1(C(C(F)=CC)=O)CC(NC(c2cocc2C)=O)CC12CCOC2 C1(C(N2C3(C)CC3CC2)=O)CC2C=CC1N(C(c1cnn[nH]1)=O)C2 C(c1cc(F)cc(F)c1)=CC(N1C(C(=O)Nc2c(C)ccc(I)c2C)CC1)=O C1(c2n(CC(C)C)c(N(C)C(C)C)nn2)CNC(=O)CC12CCC2.C1(C)(O)CCC1 C(=O)(C(C)CC(C)C)NCC12CC(NC(c3c(C)oc(-c4ccsc4)n3)=O)(C1)C2 C1(NC(CCSC)=O)CCN(CCNC(c2csc(-c3nc[nH]n3)n2)=O)CC1 C1(O)(C(=O)NCC2(CNC(=O)C(O)CC3CC3)CCOCC2)CCCCCC1 N1(C(CCC=C(C)C)=O)CC2CC1CN(C(=O)CCC(C)O)C2 c1(OCC)ccc(C(C2CCCCC2)NCc2ncc(Cl)n2C)cc1 C(=O)(C1CCCc2nn[nH]c21)NC1CC2(CCN(C(C3COC(=O)O3)=O)CC2)C1 c1(C(=O)NC2CCC2NC(c2cn(CCF)nn2)=O)ccc2c(c1)C(=O)NC2=O C(C(C)(C)CC(=O)NC(c1ccco1)C)OC.C12(CC1)CC(=O)NC2 N1(C(C2CCC(C)(CC)O2)=O)CCCC(NC(c2cc(Br)co2)=O)CC1 c1(SC)ccc(Cl)c(C(N2CC=CC(NC(C3CC(C(F)F)C3)=O)C2)=O)c1 CCC(CC)C(C)C(=O)N1CCN(C(=O)C2=CCCOC2)CC1c1ccncc1 C=CCC(C(=O)NC(CNC(=O)CN1CCN(C)C1=O)CO)c1ccccc1 c1(OC)ccc(F)c(C(=O)NC(C)CNC(c2cc(C)ncn2)=O)c1OC Cc1ccc2cccc(NC(=O)CSCCC(=O)Oc3ccc4nsnc4c3)c2n1 C(CCCC(C)(C)C)(C(=O)NCCn1cncn1)N1CCC(OC)C(C)(C)C1 CC(N=c1[nH]c(=NCC(C)C2CC2)c2cccc(F)c2[nH]1)c1ccc(Cl)c(F)c1 N1(C(c2occ(C)c2C)=O)CC2(CCC2NC(C2CC3C=CC2C3)=O)C1 C(=O)(C1CCc2cccc(OC)c21)NC(CCN(C(CC(=C)C)=O)C)C(C)(C)C c1(C(N(CCCN(C(=O)C=Cc2ccc(=N)[nH]c2)C)C)=O)ccc(N)c(O)c1 c1(C(N2CCC(C)C(NC(C(C)O)=O)C2C)=O)ccc(Br)c2cn[nH]c12 C#CC1(C(=O)NCCC2CC(CC)C2)CN(C(=O)Cc2cn(C)cn2)C1 c1(CNC(C2CCN(C(c3n(CC#C)cnn3)=O)CC2)=O)ncc(F)cc1F C1(NC(c2c(COC)nn(C)c2)=O)C2CC3CN(C(=O)C(C4CC4)SC)C1C3C2 c1(C(=O)NC(C)(C)CNC(c2ccc(Cl)o2)=O)nnn2c1CCCC2 N1(C(c2c(SCC)cccn2)=O)C(C)C2CC1C2NC(c1cnc(CC)[nH]1)=O c1(C(N(CC(C)NC(c2cccc(OC(C)(C)C)c2)=O)C)=O)cncn(C)c1=O CCCC(C)(C)C(=O)NC1CC1CNC(c1ccnc(OC(F)(F)F)c1)=O c1(CCC(=O)NCC(CCCCC)CO)nc(O)c2ccccc2n1 c1(CN2CC(NC(c3cc(Cl)nc(Cl)c3)=O)C(F)C2)cccc2cc[nH]c12 C1(NC(c2c(OC)cccn2)=O)CC(C)CN(C(c2cnc(Cl)c(N)c2)=O)C1 c1(C(N(C(CNC(COCCN(C)C)=O)C)C)=O)ccc(Cl)c(N2CCCC2)n1 Cc1nc2cc(C(=O)NCC(C)N(C)C(C3CC3F)=O)[nH]c2s1 c1(NC(CN2CC(CC)C(F)C2)=O)ccc2c(c1)CCO2 C12(C(N3CC(NC(c4cc(C(N)=O)cc(C)c4)=O)C3)=O)CCOC1CCOC2 N1(C(CCCCSC)=O)CCCC1C1CCCCN1C(=O)Cc1cc(C)on1 C12(C(=O)NCCc3ncc[nH]3)CCN(C(c3cc4ncccc4[nH]3)=O)CCC1C2 C1(NC(Cc2c(C)ccc(C)c2)=O)CCC(O)CN(C(C2CC(C)(C)CO2)=O)C1 c1(C(C2CN(C(c3c(C)occ3C(F)(F)F)=O)C2)=O)cc(F)ccc1C(F)(F)F Cc1nsc2ncc(C(=O)NCC=CCNC(=O)C(=C3CCCCC3)F)cc12 N1(C(C(C)OCC=C)=O)CCN(C(=O)CCC2CCCO2)CC1c1cn[nH]c1 c1(C(N2CCC(NC(C3CCSC3)=O)C(O)C2)=O)ccc2c(O)nnc(O)c2c1 Cc1nccc(CCC(=O)N2CC(N(C)Cc3cn(C)nc3C(F)F)C2)n1 c1(CC(N2CCC(N(C(C(CCC)OCC)=O)CC)C2)=O)cccc(F)c1O c1(NC(CNC(c2nc(C)nc(O)c2)=O)C)ncc([N+](=O)[O-])cc1C#N c1(N(CCC(C2CC2)NC(=O)OC(C)(C)C)C)ccc(N=[N+]=[N-])cc1 CC(F)(C(=O)N1CCN(C(=O)CNC(c2cnc(Cl)c(Cl)c2)=O)CC1)C(F)(F)F N1(C(=O)C=Cc2cnco2)CCC2(CCCN(C(c3[nH]cc4c3CCC4)=O)C2)C1 N1(C(C=COCC)=O)CCCC2CN(C(C3(C)COCCO3)=O)CCC12 N1(C(CCCC)=O)CC2CCC2(CNC(c2cc(-c3c(C)n[nH]c3C)on2)=O)C1 C(=O)(C(C)C(=O)c1ccccc1Cl)N1CCC1c1cn(CCF)nn1 C1(C)(CNC(C#CC2(C)CC2)=O)CN(C(c2ncccc2Cl)=O)C(C)(C)C1 Cc1nc2cc(C(=O)NCCC(C)N(C(=O)CC3CCCO3)C)ccc2n1C CC1(C)CCC(C(N2C3CC2CN(C(C2CCCCS2)=O)C3)=O)CO1 N1(C(C(C=CC)O)=O)CC(NC(c2cnn(CCC(C)C)c2C)=O)CC(F)C1 c1(C(=O)NCC(C)N(c2nnc(C3CCCC3)s2)C)csc(CO)n1 Nc1ccc(Cl)cc1C(=O)NCCC1CCCN(C(C2CC=CCO2)=O)C1 N1(C(=O)C(O)Cc2ccc(Cl)cc2)CC2CCCC2(NC(C23CC(F)(C2)C3)=O)C1 C(=O)(C1CCc2c[nH]nc21)NC(C(C)C)CCNC(c1cc2c(ncn2C)s1)=O CCCCC(CC(=O)NCCC(C)N1CCC1)NC(c1cncc2[nH]ccc12)=O C12(O)CN(C1)C(=O)OC(C)(C)CN(C)C(=O)C2F.C1(OC(C)(C)C)CCCC1 C1(C(N2CCC(C)(NC(c3cnc(Cl)s3)=O)C2)=O)CC2CCCCCC12 c1(CSC)cccc(C(=O)NC(C)CCCCNC(=O)CC2CC2C)c1 CC(C(=O)NCCN1CCC(NC(=O)CCS(C)=O)CC1)C(C)(C)O C(=O)(CCCCc1ccccc1)OC.c12ccc(o1)C(=O)COC2=O Cc1cc(C)n(CC(=O)NCC(C(C)C)NC(=O)CCCc2cnn[nH]2)c(=O)n1 c1(SC)nc(C(N2CCC(O)(CCNC(c3ccco3)=O)C2)=O)c2ccccn12 c1(C(=O)NC2C(NC(C(C)(C)N3CCC3)=O)C2)sc2cccc(Cl)c2c1Cl CC(C)(C)C(CNC(c1ccnc(-n2ccnc2)c1)=O)NC(C12CCC1C2)=O c1(OC)cnc(NC(c2cnc(Cl)c(Cl)c2)c2nnnn2C)cc1N(C)C CC1(C)CC(NC(C2CCS(=O)(=O)C2)=O)CCN(C(=O)COCCCF)C1 N1(C(C(CC)F)=O)CC(NC(c2cnc(S)[nH]2)=O)CC12CCC2 c1(CC(=O)NCCC(C)(C)CO)c(C(C)(C)C)cccc1CN c1(C(C)NCc2cn(CC3CC(=O)N(C)C3=O)nn2)ccc(F)cc1Cl CC1(C(=O)NCCC(C)(C)NC(=O)COc2ccc(F)cc2)CCS(=O)(=O)CC1 c1(C(N(C2C3CN(C(C(CC)C(C)O)=O)CC32)C)=O)ccc2c(c1F)CCC2 C(C#Cc1cn(-c2ccc(F)nc2)nn1)NC(=O)NC1CCS(=O)(=O)C1 N1(C(c2[nH]c(=NC)sc2)=O)CCCC(C)C1NC(=O)CNC(=O)OC(C)C C1(C(C)NC(c2ccc(N)cn2)=O)CCCCN1C(=O)CSCC(F)(F)F c1(SC)cc(F)ccc1C(=O)NC(C)CCCCNC(C1CN(C)CCO1)=O CC12CSCC1CN(C(c1ccc(CNC(c3cc[nH]n3)=O)cc1)=O)C2 C1(NC(C=CC=CC)=O)CCN(C(c2c[nH]nc2CCOC)=O)C1C Nc1ccc(C(=O)CCC(=O)NCCC(O)CNC(=O)CCc2cn[nH]c2)cc1 C(C)(CCC(=O)NC1CCCN(C(=O)CSc2nnnn2C2CC2)C1)SC C12(CNC(c3c(C)nn(C)c3)=O)CCCC1CCN2C(c1nccn1C)=O c1(C2(C(N3CC(NC(c4csnn4)=O)(CO)C3)=O)CCC2)ccccc1F N1(CNC(c2cn(CCNC(=O)CC3CSCCO3)nn2)=O)CC(=O)CCC1=O Cn1cc(Cl)cc1-c1noc(CCNC(=O)OC(C)(C)C)n1 CCCCC(C(=O)NC1(CNC(=O)C(F)=CC2CC2)CCC1)C(C)C Cn1ccc(S(=O)(=O)N2CC3(CC(C(=O)Nc4ccc(F)nc4F)C3)C2)n1 Cc1ncc(C(=O)NCC#CCNC(=O)Cc2cnn(C3CC3)c2)c(=N)[nH]1 C(=O)(CCCC(=O)OC)N(CCCN(C(C(C(=O)NC)C)=O)C)C C1(NC(c2nc(CCC)oc2)=O)CN(C(=O)C(CC)SC)CC12CC2 c1(C(C(=O)NCC)NC(COC(C)C)C2CC2)ccc(OC)c(OCC)c1.C(C)(C)O S(=O)(=O)(c1cc(C(C)(C)C)cc(O)c1)N(C)Cc1cc(C)on1 Cc1cc(Cl)c(C(=O)NC2CCC(NC(=O)Cc3nccs3)CC2)s1 CC1(NC(=O)CCC2CCCCO2)CC(C(=O)NCC2C3CCCC23)C1 CCC(C)(CNC(=O)C(C)n1cncn1)C(=O)N(C)Cc1nncs1 c1(C2Cn3c(nnn3)C(c3nc(Cl)cs3)N2)cccc(F)c1C.C1(CC)CCCO1 N1(C(CCNC(=O)NC)=O)CCC(NC(=O)Cc2cccs2)C1C(C)(C)C N1(C(C2N(CC)CC2)=O)CC(NC(=O)CCc2c(C)noc2Cl)CC12CCC2 N1(C(c2ccc(C#C)o2)=O)CCC(C)(C)C(C(=O)NCC2(SC)CC2)C1 c1(C(N(C)CC2(CNC(C3(CC)COC3)=O)CC2)=O)cc([N+](=O)[O-])cc(C)n1 CCCC(O)C(=O)NCC(F)CNC(c1ccc(-c2cnn(C)c2)cc1)=O C1(C(=O)NCc2c(OCC(C)C)cccc2)CCN(CC(C)O)CC1C C1(C)(CNC(CNS(NC)(=O)=O)=O)CC(F)(F)CN1C(=O)C1=C(Cl)CCC1 c1(CC(=O)NCCNC(=O)C(=O)NCC2CC2)ccc2c(c1)CCCC2 Cn1cc(NC(=O)NC(CO)CF)c(Cc2ccccc2)n1 CN1CCCCC1C(N1CC(C)(NC(=O)CCc2cccc(F)c2)C1)=O C1(CC(=O)NCC(=C)CO)COCCN1C(=O)CC1(OCC)CC1 c1(C(=O)NCC(CC)NC(=O)Cc2cscn2)cccc(OCF)c1 N1(C(c2cn(C(C)C)nn2)=O)CC(C)N(C(=O)C(C)CC#N)CC1C Cc1[nH]ccc1C(=O)N(C(C)CNC(C(C)C(O)COCc1ccccc1)=O)C N1(C(C(C)OC)=O)CC2CCCC2(NC(=O)Cc2c[nH]c(=N)nc2O)C1 C1(C(N2CC(C#C)(C(=O)NCC(O)C3CC3)C2)=O)CC(C(C)C)=NO1 N1(C(c2cnc(C(C)C)[nH]2)=O)CCC(N(C)C(C2CNC(=O)O2)=O)C(C)C1 c1(CN2C(CNC(=O)Nc3cccc(CC)c3)CCC2)c[nH]c2cc(C)ccc12 C1(NC(Cc2scc(C)c2)=O)CCN(C(=O)CS(=O)(=O)N2CCOCC2)C12CC2 N1(C(CSCC#C)=O)CCCC2(CCC(NC(=O)C(C)(C)C3CCCCC3)C2)C1 C1(CNC(c2cc(OC)c(Cl)s2)=O)CCC(C)CN1C(=O)CN1CC=CC1 c1(C(N2CCN(C(C)=O)CC2)=O)ccc(S(=O)(=O)NC(C)Cn2ccnc2)cc1 c1(C(=O)NCC2OCC(C(=O)NCC(=O)NCCC)C2)cccc(O)n1 c1(C(N2CCC(CN(C(=O)C#CC3CC3)C)C2)=O)cncc2c1CCNC2=O c1(CNC(=NCC=C)NCC(C)C(F)(F)F)nnc2n1CCOC2 c1(C(N2CCC(CNC(C3CC=CC3)=O)C2)=O)cccc2c1OCCO2 CC1CC(C(=O)NCC2(O)CC(NC(=O)CCCn3ccnc3)C2)CC(C)O1 c1(OCC)ncc(NC(C2(CCNC(c3cnc(Cl)n3C)=O)CC2)=O)cn1 N1(Cc2ncc(OC)nc2)CCC2(CC2C(=O)Nc2ccnn2C(C)C)C1 c1(CCC(=O)NCC2(O)CC(NC(C(CSC)C)=O)C2)cccnc1Cl c1(-c2nc(-c3scc(C)n3)nn2CCS(N)(=O)=O)ccc([N+](=O)[O-])cc1 c1(C(=O)NCC(=O)N(CC(=O)NC2(C(=O)NC)CC2)C2CC2)cc(C)n(C)n1 C1(F)(C(=O)NC(c2ccsc2)C)CCCN(C(=O)C(F)=CC2CC2)C1 CC(C)(CC(=O)NC1(CNC(=O)C(c2cc(F)cc(F)c2)O)CCC1)C(F)(F)F c1(C(=O)NCC2N(C(C#C)=O)CCC2)nc(SC)ncc1Cl CCC(C)CC(=O)C(=O)N(C(C(=O)NC1(c2cc[nH]n2)CC1)C1CC1)C N1(C(Cc2c(C)n(C)nc2)=O)CCC2(CC2)CC1C(=O)NCCc1cc[nH]n1 c1(C(N2CCNCC2CC)=O)c(C(=O)OCC)cc([N+](=O)[O-])cc1Br C(=O)(C(C)S(N)(=O)=O)N1C(CN(C(CS(CC)=O)=O)C2CC2)CCC1 N1(C(c2cn(CC)nn2)=O)CCc2ccccc2C(NC(=O)C(C)C2CC2)C1 N1(C(CCCCc2ccc(C)cc2)=O)CC2CC(C(=O)N(C)C)C(CBr)C2C1 CC(O)C(=O)NNC(=O)C1CCOC1(C)C C(=O)(CC1CCOc2ccccc21)N(CCNC(C1C(C)C1)=O)CC1CC1 N1(C(c2cnc(C(F)F)nc2)=O)CCC2CN(CC3CCC4(CC3)CC4)CC12 C1(C(=O)NCC2(C)CCN(C(CC34CC(C)(OC3)C4)=O)C2)CC2(C1)CC1(CC1)C2 c1(CNC(=NCC)NCC2COC(=O)O2)cc(C)cc(Br)c1 N1(C(CC(CCC)CC)=O)CCCC2CN(C(C3CC4(CCOCC4)C3)=O)CC12 C12(NC(CC3(CS(C)(=O)=O)CC3)=O)CCN(C(c3cc(O)ncn3)=O)CC1C2 c1(C(=O)NCC2CCC(NC(c3cccc(CC)n3)=O)C2)ccc2c(c1)OCCO2 C1(C(=O)NCCOC2CCN(C(CSCCN(C)C)=O)C2)OCC2CCCC12 N1(CC)CCCC(NC(c2cnc(C3CCNCC3)[nH]2)=O)C1 N1(C(CCCCC(C)C)=O)CCCCC12CC(NC(C1CCCCC1(C)C)=O)C2 N1(C(C=C(CC)C)=O)CC(NC(c2cnoc2-c2ccccc2)=O)C(O)C1 C#CCC(CC(F)F)C(=O)NCC1CCCN1C(=O)C(C)CC CC1OCCN(C(=O)CCCN2CCCCC2)C1C(N1CCCC(C)CC1)=O Cc1ccc2c(c1)C(NC1CCCC1C#N)CCC2 C1(NC(=O)CCCc2cccc(Cl)n2)CN(C(c2cnc[nH]2)=O)CCC12CCC2 C1(C)(OC)CCN(C(C2CC(NC(=O)Cn3cnccc3=O)C2)=O)CC1 c1(OC)cc(C(N2CC(C(=O)NCC3CCCOC3)C(F)C2)=O)ncn1 C1(CNC(c2cc(CC#C)ncc2)=O)CCCC2CN(C(=O)C(C)(C)C#C)CC12 c1(C(N2CC3(N(C(C4(CC)CC4)=O)CC3)C2)=O)[nH]nc2ccncc12 Cc1cc(C(=O)NC(C)(C)CN(C)C(C2CCCC(C)C2)=O)cc(Cl)c1 S(=O)(=O)(c1ccc(NC(CO)C2(C)CC2)c(C#N)c1)NCC(C1CCCCC1)C c1(CCNC(=O)C(N2CCCC(NC(C3CC4CC3C4)=O)C2)=O)ccc(F)nc1 N1(C(C2(C)CCOC2)=O)CCOC2CN(C(=O)CCC3CCCCCC3)CC2C1 C1(F)(C(=O)NCC(C2CCCC2)NC(CNC(CNC(C)=O)=O)=O)C2CCCCC12 C1(CNC(c2ccc(C)nn2)=O)CN(C(C2(Cl)CC2)=O)CCC12CCC2 C1(OC)CC2(C1)CC(SCC(N1CC(N(C(=O)C(C)n3cccn3)C)C1)=O)C2 C1(CCOC)(NC(c2cc(C)sc2C)=O)CCN(C(=O)Cc2csc(C)n2)C1 c1(C(=O)OC)cccc(F)c1C(N1CC2(C1)CN(C(C1(C)CCC(C)C1)=O)C2)=O C=CC(C)CC(=O)N(C1CCC(NC(c2ccc(OC(C)C)nc2)=O)CC1)C C(=O)(CC(C)CC(C)C)NCCN(CCC)C(C12CSCC1C2(F)F)=O C(=O)(CC1COc2ccccc21)NC1CC(NC(C(C)C#N)=O)C1 N1(C(C2(CC)CC2)=O)CCOC(C)(CNC(C2CC2C(C)(F)F)=O)C1 C1(C(=O)NC2(CNC(=O)Cc3sccc3Cl)CCCCC2)CCC([N+](=O)[O-])CC1 c1(C(N2CCC(N(C(=O)CCCC(C)(F)F)C)C2)=O)cnc([N+](=O)[O-])n1C c1(OC(C)C(=O)NC2CCC(n3cccc3)CC2)ccc(Cl)cc1Cl N1(Cc2c(OC)ccc(OC)c2)CC2CN(C(c3csc(C)n3)=O)CC2C1 C#CC1(C(=O)NCC(=O)N(C)O)CN(C(=O)Cn2nc(C)nc2C)C1 N1(C(CC=CCC)=O)CCC2(CC1)CC2C(N1CCC(C)C1(C)C)=O NS(=O)(=O)C1(C(=O)NC2CC2NC(C2(Oc3ccccc3)CC2)=O)CCC1 CSC1=C(C(=O)N2CC3(NC(=O)CSC4CCCCO4)CCC2CC3)CCCC1 C1(NC(c2ocnc2C(F)F)=O)CN(C(c2c(F)cccc2Cl)=O)CCC1CO c1(CC(=O)NCC2(CCNC(CC3CC(=C)C3)=O)CC2)coc2cc(C)ccc12 C1(C(N(C)CC2(NC(c3csc(=N)[nH]3)=O)CC2)=O)CCC(C(C)(C)C)CC1 c1(C(=O)NCCOC2CCN(C(C(C)N(C(C)=O)C)=O)C2)nn(C)c2c1CCC2 C1(CNC(c2cnn(-c3cccnc3)c2)=O)CCN(Cc2ccc(Br)s2)C1 N1(C(CCN(C(CCNC(=O)OCC)=O)C(C)C)=O)CC2CC1CS2=O C(CN=C(NCC1CCOC1)NCC1CCCCS1)C1(O)CCCC1 c1(COC)n[nH]c(=NCC2(F)CCN(C(=O)CC3CS(=O)(=O)C3)CC2)s1 c1(SCNC(C(c2[nH]nnc2C)N(C(C)COC)CC)=O)ccccc1OC c1(C(N(C2C(C)CCN(C(=O)CSC3CC3)C2)C)=O)ncn2cccnc12 Cc1cn2c(n1)CC(C(=O)N(C1CCCCC1N(C(=O)C(O)CN(C)C)C)C)C2 C(CCCC(=O)NC1(CN(C(=O)C(C)CCc2ccccc2F)C)CC1)OCC N1(C(c2ccc(OC)c(N)c2)=O)CC2CCC1C1CN(C(C3CC3C#N)=O)CC21 C1(C(=O)OC)CCC2(CCN(C(C3CCCC3(C)C)C(=O)NC3CC3)CC2)O1 N1(C(c2cc(CCNC(c3ccnc(SC)n3)=O)on2)=O)CCC(SCC)CC1 C(C)(C(CO)NC(c1cc(-c2ccco2)no1)=O)NC(C1C(OCC)C1)=O CCC(C)CC(C(=O)NCc1cnccc1OC)NC(c1nnc(S)n1C)=O Cc1c(C(=O)NC(C)C(C)NC(c2ccn(CCF)n2)=O)c(C(F)F)nn1C c1(C(=O)NC2(C)CC(C(=O)NCC(c3cccnc3)C)C2)ccc(F)cn1 c1(CC)n[nH]c(CC)c1CC(=O)NCC(F)CNC(=O)CCc1cc(C)no1 n1(CC(=O)NCC(CNC(c2ccc(O)cn2)=O)OC)nc(C)ccc1=O N1(C2CN(C(C3CCC(OC)C3)=O)C2)CCN(C(=O)Cc2cnsc2)CC1 C1(NC(c2c(C)coc2)=O)(CNC(c2cc(CO)c(C)o2)=O)CCCCC1C c1(NC(=O)NC(CCC#C)C(=O)OC)c(Br)cc(Cl)c2sccc12 C1(NC(C(C)C)=O)(CO)CCN(C(c2cccc(Oc3cccc(F)c3)c2)=O)C1 C1(NC(C2CCN(C(C(C)N3CCCC3)=O)CC2)=O)CC12CCN(C)CC2 N1(CC)CCCCC1C(=O)NC(COCC)C(=O)NCC1(C(=O)OC)CC1 C1(NC(C(C)OC)=O)COC2CN(C(c3c[nH]c(=N)nc3C)=O)CC12 N1(C(c2cnc(C)s2)=O)CC(C(=O)NC(C(O)CO)C2CC2)C(C2CC2)C1 N1(C(c2c(C)cnnc2)=O)CC2C(C1C(=O)Nc1c(Cl)cnc(Cl)c1Cl)C2(C)C CCCCC(C(=O)NC1CCCCC1)N1CCC(C(=O)NCC)(OC)CC1 C(=O)(C1=CCC(C)CC1)NC(C1(O)CCN(C(c2occc2CN(C)C)=O)C1)C C(=O)(CS(=O)(=O)CC)N1CCC(N(C(=O)COCC(C)(C)C)CC#C)CC1 Cc1cc(C(N2CCN(C(=O)OC(C)(C)C)C(CO)C2)=O)cc(Cl)c1 c1(C(N2CC(C)(CNC(c3c(C)nc(C)s3)=O)OCC2)=O)cc(C#N)ccc1O c1(CN2CC3N(C(c4ccc(OC)nn4)=O)C3C2)ccc(Br)c(C)c1 c1(C(NC(=NC)NCCCn2ccc(C3CC3)n2)C)ccc(F)cc1 n1(CC)ncc2cc(C(N3CCC4CN(C(=O)C(C)CO)CC4C3)=O)c(C)nc12 C1(C(N2CC(C)C(NC(=O)CCc3ccc(Cl)s3)C2)=O)CC12CCOCC2 c1(C(=O)NCC2N(C(C(CC)C)=O)CCCC2)cc(C#N)c(SC)nc1O CC(C)C(C(=O)NCCOCCN(C)C)NC(C1CCCC1)=O C1(N(C(CC)=O)C)CCC(CC)CC1.C12CC(C1)OOCCNC(=O)C2 c1(C(=O)NC2CC(NC(C(C)Cc3cccnc3)=O)C2)nccnc1C(N)=O C(=O)(C(CO)C(C)(C)C)Nc1c(F)ccc(C(=O)OC)c1 C1(C)(CNC(CCCCOC)=O)CC(F)(F)CN1C(=O)CCC(C)OC C#CCC(C)C(=O)N(CCCCN(C)C(c1cn(C)nc1SC)=O)C CCC(CC)(C(=O)N1CC(CNC(c2cnco2)=O)C(F)(F)C1)OC CC1CN(C(c2cnc(S)n2C)=O)CC(CCNC(c2cccc(N(C)C)c2)=O)O1 N1(C(CN(CCOC)C)=O)CC2CC2(CNC(C23CCC(CC2)C3)=O)C1 N1(C(C2CCC(C)CC2)=O)CCc2c(NC(=O)C3=CC(O)CCC3)cccc2C1 N1(C(c2cnc(COC)s2)=O)CCC2(C1)CN(C(c1ccc(CO)c(F)c1)=O)C2 C1(C)(C(=O)NC(C2CCOC2C)CC)CCCN1C(=O)CCc1cnco1 C1(C)(COCC)CC(F)(F)CN1C(=O)CNC(C)=O.C1(NC(C2(C)CC2)=O)(OC)CC1 Cc1ccc2c(c1)C(N(c1ccnc(F)c1C)C1CC1)CCCO2 C1(C(=O)NC(CCN(C(=O)CSC(F)F)C)c2cccs2)CC2CCCCC12 Cc1cnc(Cl)n1CC(=O)Nc1cccc(C(N)=O)c1 C1(OC)CN(C(=O)COO)CCC1NCc1ccccc1.C(=O)(C(C)CC(C)C)O N1(CC(=O)Nc2cccc(SC)c2)CCC(O)(Cc2ccc(C)c(F)c2)CC1 C1(CNC(c2scc(C(=O)OC)c2)=O)CN(C(C23CC(C#N)(C2)C3)=O)CCC1C C1(C)(C(=O)NC2CN(C(C(CC)N(C(=O)CSC)C)=O)C2)CC(C)=NO1 C1(NC(C(C)S(C)(=O)=O)=O)CC2(CCN(C(c3ccc(O)c(F)c3)=O)C2)C1 C1(CC(=O)NCC2CCN(C(c3cc(CC)c(CC)o3)=O)C2)CCCCC1(C)C c1(C(N(CCCN(C(=O)C(F)(F)C(F)F)C)C)=O)ccc2nc(CO)[nH]c2c1 O=C1COC2CCN(c3nnnn3Cc3nnn4c3CSCC4)CC2N1 c1(C(C(=O)NC2C(CNC(C(C3CCOC3)OCC)=O)C2)=O)ccc(Cl)s1 N1(C(c2cccc(C)n2)C(=O)O)CCC(C)(C2CC2)C1.C12CCC(CC1)CO2 C1(NC(c2cncc(Cl)c2Cl)=O)CC(C(F)(F)F)CN(Cc2ccccc2I)C1 C1(CNC(=O)C2=NOCC2)CCN(C(=O)CCN2C(=O)CNC2=O)CCC1(F)F c1(NCC)ccccc1C(=O)NCC1(CCc2ccc(Cl)cc2)CC1 Cc1cc(C(C)C(=O)NCC(O)CNC(c2cc(C3CCC3)on2)=O)cc(F)c1 CN1CCC(C)(C(N2CC3CC(CNC(=O)CCC4CCCC4)C3C2)=O)CC1 C(=O)(CCS(=O)(=O)N(C)C)NC1CC(CNC(C(CO)OC)=O)C1 CCCCC(CC)C(=O)N1CCC(CO)C(NC(=O)CCOC)C1 N1(C(c2ccc(S(C)=O)cc2)=O)CC(C2CCCN(C(=O)C3=CCC3)C2)C1 c1(NC(C(=O)NC(CNC(c2cc(C(C)=O)on2)=O)CO)=O)ccc(F)cc1 c1(C(N2C(C(N(CC(C3CC3)OC)C)=O)CCCC2)=O)cnc2n1CCC2 c1(C(=O)NCCC2CSCCN2C(=O)CC2C=CCC2)cnccc1Br C(CCCCCCO)NC(C1N(C(Cc2cccc(C)c2)=O)CSC1)=O N1(C(C=CCOCCOC)=O)C2CCC1C(F)C(NC(c1[nH]nc(OC)c1Cl)=O)C2 C(=O)(C1COc2ccccc21)NCCC(C)(C)NC(c1cccc(C)c1F)=O CN1CCC(C(=O)NCc2cc(C(=O)NCCC(O)C3CCCC3)no2)CC1 CC1CC(CNC(c2cnc(Cl)s2)=O)CN(C(=O)CC2CC(=O)NC2=O)C1 c1(NC(C(CCNC(c2cnn(C(C)C)n2)=O)O)=O)cccc(Cl)c1O c1(N(C2CCN(CC)C2)C)nc(=NCC2COCCO2)[nH]c2c1CCCC2 C1(C(N2CCCC(C(N)=O)C2)=O)(CC)CCN(C(C2CCC3(CC3)C2)=O)C1 c1(CC(=O)Oc2c(C)n[nH]c2C)ccc(S(=O)(=O)OC(F)F)cc1 c1(OC(C)C)cccc(CNC(C2CN(C(C3C4COCC34)=O)C2)=O)c1 C1(C(N2CCC(CNC(c3c(CCC)occ3)=O)C2)=O)Cc2cc(C)ccc2S1 N1(C(C2C(=C)C2)=O)CCC2CN(C(c3cc(F)ccc3C3CC3)=O)CC2C1 c1(NC(=O)OC)cccc(-c2nnc(N3CCCC3C)n2C2CCCC2)c1 c1(NC)ccc(C(=O)NCCC(CNC(=O)C(C)CO)OC)nc1 C(CCSC)(C(=O)N1CCCC1CNC(N)=O)NC(c1c(CCC)nco1)=O C1(NC(c2ccc(CC)c(F)c2)=O)CC1C1CCN(C(=O)C(C)(O)C2CC2)CC1 CC1CCN(C(=O)COC(F)(F)F)C1c1cn(C(c2ccncc2)C)nn1 C#CCC(C)(C)C(=O)N1CCN(C(C)CNC(C2(O)CC(=C)C2)=O)CC1 CC(C)C(O)C(=O)N1CCCC(N2CCN(C(=O)CCc3cnn(C)c3)CC2)C1 N1(C(C(C(C)C)NC(COC)=O)=O)CCC2(CC1)CC(C)N(C(=O)C(C)O)C2 CC1CCCn2c(C(N3CC(CNC(c4cccc(F)c4)=O)C(C)C3)=O)cnc21 c1(OC)cc(C(C(=O)NCC2CCCO2)N(CC(C)(C)C)C)cc(C(F)(F)F)c1 C12(C(=O)OC)CC(C(=O)OC)(C1)C2.C1(C2CCC2)C(C)NC(=O)NCC(=O)N1 C1(O)(CNC(=O)NCC(CC)(C)CC)CC2CCC1C2 c1(CS(C)(=O)=O)nc(C(=O)NC2(CCNC(C3(CO)CCC3)=O)CC2)cs1 C(CC1CC1)(CC(=O)N1CCOC(CF)C1)NC(C1CCCO1)=O N1(c2c(C)c(NC3CC3C3CC4(CCCC4)CO3)ncn2)CCC2(CC1)CC2(F)F c1(C(N2CC(C(C(=O)N(CCCCCO)C)O)C2)=O)cccc(F)c1 Cc1ccc(C)c(CNC(C2(F)CCN(C(C3CN(C4CCC4)C3)=O)C2)=O)n1 C1(CNC(COC(CC)C)=O)CN(C(=O)C(F)CC2CCC2)CCC1CO C1(C2CN(C(=O)C=CC(=O)NC3CC3)C2)(NC(C(CC=C)C)=O)CC1 C1(OC)CC2CC(C1)N(c1cc(F)cc(F)n1)C2 C1(NC(c2c(OCC)scc2)=O)CC2CC1N(C(c1ncc(F)cc1F)=O)C2.OCC CCC(C)(C)C(O)C(=O)N1CC2CN(C(c3cc(Br)c(Cl)s3)=O)CC2C1 C=Cc1cnn(C)c1C(=O)NC(CNC(c1cnn(CCC)c1C)=O)CCOC c1(C(C(=O)NC2CC(CNC(C3CC(C(C)C)C3)=O)C2)(F)F)cccc(Cl)c1 C(=O)(C(C)C(O)CCCCC)NC1CC2CN(C(C(CC=C)(C)C)=O)C(C1)C2 C1(C(N2CC(NC(CCC=C(C)C)=O)C2)=O)CCS(=O)(=O)C1(C)C C1(O)(C(C)NC(=O)C(F)=CCCF)CN(C(c2coc(C3CCC3)n2)=O)C1 C(=O)(C1COc2ccccc21)NC(C1CCCN1C(=O)CCC(F)F)(C)C N1(C(C(=O)NCC)=O)CCC(C2(NC(c3cncn3C(F)(F)F)=O)CC2)CC1 Cc1cnc2cccc(C(=O)NCC3(NC(C4CC5(C)CC4CO5)=O)CCC3)n12 CCCCCC(C)CC(=O)N1CC(N(C)C(C2(c3ccc(F)cn3)CC2)=O)C1 N1(C(c2cnc(C(C)C)[nH]2)C(=O)NCCCC)CCC(c2ncccc2Cl)CC1 C#Cc1cnc(C(=O)NC(C2(O)CN(C(=O)Cc3cccnc3O)C2)C)c(C)c1 CCCN=c1ncc(CN2C(C(N3CCC(C)(C)C3)=O)CC3CC23)c[nH]1 C(=O)(C(CCC(C)(C)C)NCCC12CCC(CC1)CC2)N(CCCOCCO)C N1(C(c2cc(C)c(C)nc2)=O)CCN(C(=O)CC2CCCCC2O)CCC1C CC(O)CCCCCC(=O)N1CC(C)(NC(c2ccc(NC(N)=O)cc2)=O)C1 C1(NC(CC(=O)N(C)C)=O)COC2(CCN(C(c3cncc4nc[nH]c34)=O)C2)C1 N(C1c2ccccc2C2CC1C2)C(c1c2ccccc2nn1C)C C12CN(Cc3nccn3C1)C(=O)N2.N1(C2CN(C(=O)OC)C2)CCOCC1 c1(OC)nn(C)cc1C(=O)NC(C)CC(C)NC(C1CC(=O)N(C(C)(C)C)C1)=O C1(C(C)Nc2cccc(C3CC(=O)C3)c2)CCCCN1C(=O)CC1CCCC1 c1(C(=O)NC2C(OC)CN(S(=O)(=O)CCCCl)CC2)nc2ncccn2n1 c1(C(N2C(CN(C(=O)CCC3CCC3)C)COCC2)=O)cc(F)ccc1C(F)F CC1(C)OCCc2cc(C(=O)Nc3ccc(Oc4ccncc4)cc3)ccc21 N1(C(Cn2nc(C)oc2=O)=O)CCC(CNc2nccc(C)n2)C(C)C1 Cc1cccc(C(O)C(=O)NC(CNC(=O)Cc2ccc(F)cc2)C2CC2)c1F C1(CC(=O)NCC(CCCC)O)N(C(=O)C(F)CC2CCOC2)CCC1(C)C c12cccc(c1)NC(=O)C2OCC.CCCC(C)N(C)CCNC1CC1 S(=O)(=O)(c1ccc(N2CCC3(CCCC(C(=O)O)O3)CC2)c([N+](=O)[O-])c1)N(C)C C1(NC(C(C)(C)OCC)=O)CC2(C1)CC(NC(C1CCC3(CC1)CC3)=O)C2 N1(C(c2cccc(OC)c2)C(=O)NC2CC2)CCCC(C)(O)C1 O=C1COc2ccc(S(=O)(=O)NC3CCC(NC(c4ccno4)=O)C3)cc2N1 O=C1CC(C(N2CC3CC(NC(C4CC5(CC5)CO4)=O)C3C2)=O)Cn2ncnc2N1 CCCCC(C(=O)NC1(C)CC(C(=O)NCC2CCC(C)(C)O2)C1)C(C)C C1(C(N(C2CCCCC2)CC=C)=O)CC(=O)NC(c2cnn(C)c2)C1 c1(C(N(C(CNC(C2C(C=C)C2)=O)C)C)=O)csc(C2CCCCC2)n1 C(CC(=O)N1CC(C)CC1CC)(C(F)F)NC(CCC=CCC=C)=O Cc1cc(N)cnc1C(N1CCC(C)C1CC(=O)Nc1ccc(O)cc1O)=O c1(C(=O)NCC(CC)NC(C2(C)CCCS2(=O)=O)=O)nccc2ccncc12 C12(C(N(CC(CN(C(=O)CCCc3ccncc3)C)O)C)=O)CCC(F)(CC1)C2 c1(C(N2CC(F)(CNC(CCCC(C)C)=O)C2)=O)cc2c(=O)ccn(C)c2s1 C(=O)(C1CCCc2nnn(C)c21)NC1CN(C(c2ccn(C)c2)=O)CC2(C1)CC2 N1(CC(=O)NCC=CCC(=O)N(CCOC)C2CC2)CC(=O)NC1=O Cc1cc(C(N2CC(O)(c3cn(C(C)C(=O)OC4CC4)nn3)C2)=O)cc(N)c1 C12(C(=O)OC)C3C4C1C1C2C3C41CO.C12CCCCCC1NC2=O C(=O)(C(C)(C)C1CC1)NC(C)(C)C.n12ccc(n1)C(=O)NCCN(C)C(=O)C2C N1(C(c2c(CC)oc(C)c2)=O)CCN(C(=O)Cn2ccc(C)cc2=O)C(CO)C1 c1(OC)cccc(C(N2CCCC2(C)CNC(=O)CC2CSCCS2)=O)c1 C(=O)(C(C)C(O)C(C)CC)NC1(CC(N2CCC(C(=O)NC)CC2)=O)CCC1 C#Cc1c[nH]nc1C(=O)NCc1cncc(C(=O)N(CC(N2CCCC2)C)C)c1 Cc1cc(-n2cc(C)c(C3CCN3C(C3CN(c4nncs4)C3)=O)n2)cc(C)c1 C1(NC(Cc2n(C)cc(I)c2)=O)Cc2cc(Br)ccc2OC1 c1(C(CC)=O)cncc(C(=O)N(C)CCNC(c2sc(OCC)nc2Cl)=O)c1 C1(NC(C(C)SCCCC)=O)CCCCN(C(=O)C=Cc2cccc(CO)c2)C1 Cc1ccc(-n2cc(CN3CCCC3NC(c3nn(C)cc3N)=O)nn2)cc1Cl N1(C(CC2C(C)CCCC2)=O)Cc2occ(NC(=O)CN3CCNC3=O)c2C1 CN1CCC(C(N2CC3CC3(C(=O)NCC(=O)OCCO)C2)=O)CC1=O c1(CC(=O)NC(CC)CNC(C2CC2C)=O)coc2cc(C(C)C)ccc12 N1(C(c2c(C)[nH]c(C#N)c2)=O)CCC2(CC2)CC1C(N1CCCC(O)(CO)C1)=O CC(C)C(CO)C(=O)NC(C)CC(C)NC(=O)C(C)CCNC(=O)OC(C)(C)C C(=O)(CCCC(F)(F)F)NC(C1CCCN(C(=O)CC2CCCOCC2)C1)C c1(OCC2OCCN(C(C(C)C)=O)C2)cccc(Cl)c1N1CCCCC1 C#CCC(C)(CNC(=O)CN(C(c1ccnnc1)=O)C1CC1)CO C1(C(=O)NCCCCCN(C(=O)CCSCc2ncccn2)C)CC2CCC1C2 CC1(C)CC(NC(=O)C(C)(O)C2CCCCC2)CN1C(=O)CCNS(C)(=O)=O C#CC1CN(C(=O)CC)CCN1C(C1C2CC(=O)CC12)=O N1(C(CCNC(C)=O)=O)CC(NC(C2CCC(C)(C)O2)=O)CC12CCCOC2 C1(C(=O)NCC(C2CCC2)NC(c2cncnc2)=O)OCC2CCCC12 N1(C(C2C(CC)C2)=O)CCN(C(c2cccc(F)c2F)=O)CCC1C c1(C(=O)NCCC2CCCN(C(=O)CCc3ncc[nH]3)C2)cc2ccnn2cn1 N1(C(C2C(NC(COCC(C)C)=O)CCO2)=O)CCS(=O)CC1C N1(C(Cc2n(C)ccc2)=O)CC2ON=C(CNC(=O)Cc3ccc(Cl)cc3)C2C1 c1(C(N2CCCC(CNC(CC(CC)OC)=O)C2)=O)c(N)sc(C)c1C c1(OCC)cc(C(N2C(CNC(=O)CC3CCCO3)CC3CC23)=O)ccc1[N+](=O)[O-] C(=O)(C1=CCCCO1)NC(C1CCN(C(c2cnc(C)[nH]2)=O)C1)C N1(C(C2C(C)=C2)=O)CCC2(CC1)CN(C(C1CC1F)=O)CC2CO N1(C(C=CCOC)=O)CC(NC(c2cccc(-n3cncn3)n2)=O)C2(CCC2)C1 c1(C(N2CCC3(NC(CCCC#C)=O)C(CC2)C3)=O)nsc2ccc(C)cc12 Cc1ccc(C(=O)NCC2(C)CN(C(=O)C(C)n3cncn3)C2)c(N)n1 CC1=CC(NC(=O)C(CC2CCOCC2)NC(=O)C(C)C#N)CCC1 c1(OC)cc(C(N2CC3CC2C3NC(=O)CCNC(N)=O)=O)cnc1O C1(CCc2ccccc2)(CNC(N2CC(C(=O)OC)C2)=O)CCOCC1 S(=O)(=O)(c1ccc(Cl)cc1)Nc1ccc(OC2CCS(=O)(=O)C2)cc1 N1(C(=O)CCc2ccon2)CCN(C2CC(NC(C3(O)COC3)=O)C2)CC1 c1(C(C)CC(=O)NCCC2(CNC(=O)C=Cc3cn[nH]c3)CC2)ccc(F)cc1 C(CO)(C(=O)Nc1cn(Cc2ccccc2)nn1)NC(CN(CC)CC)=O c1(C(=O)NCc2cn(Cc3cccnc3)nn2)cccc([N+](=O)[O-])c1Cl C(=O)(C(O)(C(F)(F)F)c1ccccc1)NCC1CCCCN(C(CCC=C)=O)C1 N1(C(c2oc(CC)c(C)c2)=O)CCCC(C(=O)NC2CN(C(N)=O)C2)CC1 C(C(C)C(F)C(=O)NC(CCO)C(F)F)NC(C(CC)(C)C)=O N1CCC2CCN(C(=O)C(c3ccc(F)c(C)c3)=O)C2C1.CO CCC(CNC(=O)C(C)C(C)n1cccn1)(CC)NC(c1ccc(CO)s1)=O c1(C=O)cc(C(N(N2CC(N(C)C(C3CC3c3cccnc3)=O)C2)C)C2CC2)nn1C.OC c1(C(=O)NCC(CC=C)NC(C2(CCOC)CC2)=O)ccc2cc(Cl)ccc2n1 N1(C(c2ccc(N)c(F)c2)=O)CCCC(O)(CNC(c2ccoc2)=O)CC1 CC1(c2ccccc2)CN(C(C(=O)NCCC#N)c2ccoc2)CCO1 c1(C(=O)NC(CCNC(c2c(C)cccc2C)=O)C)ccc(C#N)cc1O O=S(=O)(c1cncc(Br)c1Cl)NCc1csc2c(F)cccc12 C12CN(CC(C)(C)C1)C(=O)N2.C(=O)(C(C)(C)NC(=O)OC)OCC C=C(C)CCC(=O)NC(C)CCN(C)C(c1ccccc1C1CCC1)=O CN1CCN(c2cc(CNC(C3(CCO)CC3)=O)ccn2)CC1 CC#CCC(C(=O)NCCc1cnn[nH]1)NC(c1cncc(OC)n1)=O N1(C(C)C)CC(CNC(N2CCC(O)(Cc3cccc(F)c3)C2)=O)CC1=O c1(C(=O)NC2(CNC(c3c(OC)scc3)=O)CCOCC2)ccc2cc[nH]c2n1 C1(CNC(=O)CCSCC(F)(F)F)CC2(CCN(C(=O)C(O)C3CC3)CC2)CO1 Cc1[nH]c(C)c(C(=O)NCC2(O)CC(C(=O)NCC3(O)CCC3)C2)c1C c1(CNC(c2cccc(C#C)c2)c2nnnn2CC2CC2)ccc(F)c(C)c1F C1(C(N2CCC(NC(Cc3nnc(C)o3)=O)(CO)C2)=O)CCn2c(C)cnc2C1 N1(C(c2ccc(OC)s2)=O)CCN(C(=O)COCc2nc(C)no2)C2CC12 C(=O)(C(F)C(=O)NCC1CCN(C(=O)C(SC)C2CC2)CC1)OCC C(=O)(CCCS(C)(=O)=O)N1CCC(CCCCNC(c2c(C)nns2)=O)CC1 C(=O)(C1=CCN(C(c2ccc(O)cc2)=O)C1)NCCC(C)CO c1(OCC(=O)NC2C(NC(c3cc(C)no3)=O)C2)c(F)cccc1F N1(C(c2onc(OC)c2Br)=O)CC(NC(c2nnn(C)n2)=O)CC(C)C1 C1(CC(N)=O)CCCN(C(=O)CN2CCC(N(C3CCCC3)S(C)(=O)=O)CC2)C1 CC(C)C(O)C(=O)NCCC1(C(N2CCC(n3cccn3)C2)=O)CC1 N12CCN(C3CS(=O)(=O)CC13)C(=O)C1N(CCC1)C2=O.CCC(=O)OC(C)(C)C C1(C(=O)NCC(C)CC(=O)NC2(c3ccccn3)CC2)Cc2nccn2C1 C1(NC(c2n(Cc3nnn(C)n3)nnn2)(C)CCBr)CC2CCC1O2 N1(Cc2cc(OCC)ns2)CC2(CCC(C(=O)Nc3cc(F)c(F)c(F)c3)O2)C1 CC1(C(N2CCC(CCNC(=O)Cc3cnns3)CC2)=O)CC=CCC1 N1(C(c2nn(C)c(O)c2)=O)CCCC2C(NC(c3ncccc3Cl)=O)C(C)(C)C12 c1(COC2CCN(N(C(F)(F)C(F)(F)F)C)C2)cccc(C#N)n1.c1(O)ccccc1 N1(C(COC(CC)(C)C)=O)CCN(C(=O)CN(C)C(=O)OC(C)(C)C)C(CO)C1 c1(C2C(C(=O)NCCOCCNC(C3C(C)(C(=O)OC)C3)=O)C2)cccc(Cl)c1 c1(OCC2CCCCO2)cccnc1SCC(N1CC(COC(C)C)C(C)C1)=O CC1CC(C)N(C(c2cn[nH]c2)=O)CCN1C(=O)C=C1CCSCC1 C=CC(C)C(=O)NC1CCN(CCCNC(=O)C(c2ccn(C)c2)C)C1 N#Cc1ccc(C(=O)NC2(CC(N3CCn4nccc4C3)=O)CCC2)cc1F C1(CN(C(C2(SC)CC2)=O)C)CC(F)CN1C(c1cc(C)no1)=O C1(C(C)(C)C)(CNC(c2ccc(F)s2)=O)CCN(C(=O)C=CC2CCOCC2)C1 N1(C(CC(n2ccc(C)n2)C)=O)CC(C2CN(C(C3CC(C(F)F)C3)=O)C2)C1 C(=O)(C1=C2CCN=C2NC=C1)N1CC(NC(C2CCCCC2)=O)CC12CCC2 C1(CNC(CCP(C)(C)=O)=O)CC2CCC1N(C(C1(N3CCCC3)CC1)=O)C2 c1(C(N(CC(O)CNC(=O)CCn2ccccc2=O)C)=O)cccc(C#N)c1 CC1(F)CN(C(=O)C(c2ccc(Cl)c(Cl)c2)O)CCN(C(C2CC(O)C2)=O)C1 c1(COC(C2CCCN(Cc3ccccc3)C2)=O)ccc(C(F)(F)F)cn1 C1(C(=O)NCC(C)OC(F)F)CCN(C(=O)C2(C)CCCC2O)O1 N1(C(c2ccnn2C(F)F)=O)CCC2(CC1)CN(S(=O)(=O)CCCl)CCO2 N1(C(C2C(C)(C)OCC2)=O)CCN(C(=O)C(O)CC(F)F)C(CO)C1 Cc1ccc(C(=O)NC2CN(C(=O)CCOC3CCCOC3)CC2F)c(O)n1 C#CCC(C(=O)NC(C)CCNC(=O)CCc1ccc(OCC)cc1)C1CC1 C(=O)(C1=CCN(C(=O)CCOC(C)C)C1)NCc1c(C)nccn1 C(Cc1ccccc1F)(N=c1[nH]nc(SC(F)F)s1)OCC O=[N+]([O-])c1cccc2ccnc(NC3CCC4(CC3)C(F)(F)C4(F)F)c12 O=C1NC(CNC(=O)C(C2CCCO2)NC(=O)CC2CCCCC2)CO1 CCC(CC)CCC(=O)N1CCC(F)(CNC(=O)CC2CCCC2O)C1 Cc1ccc(C(=O)NCc2ccc(CNC(=O)C3=C(Cl)CC3)cc2F)c(Cl)c1 c1(C(=O)NCCC(C)N(C)C(C2CCC(F)C2)=O)ccc2nnn(O)c2c1 N1(C(c2ccc(C#N)[nH]2)=O)CCN(C(c2csc(CO)n2)=O)C2CCCCC12 N1(C(C(C)(C)c2nccs2)=O)CCC(C2CCN(C(C3CCCOC3)=O)CC2)C1 N=c1[nH]ccc(C(N2CCC(NC(C3CC4CCC3C4)=O)C2)=O)c1[N+](=O)[O-] C1(NC(=O)CCOC2COC2)COC2(CCN(C(=O)C=CBr)C2)C1 CC12CN(C(c3nonc3N)=O)CC1CN(C(C1CCCCC13CCC3)=O)C2 C(=O)(CCCCCN=[N+]=[N-])N1CC(C)C(C2CC2)C1 C1(C(=O)NCC(C2CC(C)(C)C2)O)CCCN(C(c2cccc(O)n2)=O)C1 c1(C(=O)NC2(C)CC(NC(=O)CN3CC4CCC3C4)C2)cccc(O)c1Cl C1(NC(CSCCCC)=O)CC2CCC1(C(=O)NCC(C)(C)C1(O)CCC1)C2 c1(C(=O)NCCOCCN(C(=O)CC2COC(=O)C2)C)ccc(Cl)c(O)c1 N1(C(C(C)CO)=O)C2CCCC1CN(C(c1csc(-c3ccccc3)c1)=O)C2 C1(NC(CCC(=C)C)=O)CCSC12CN(C(=O)CCc1ccc(C)nc1)C2 c1(C(=O)NCCSCC(=O)NCCC2CCCC3CC23)cc(O)cc(F)c1 c1(C(C)(C)C)nnc2cc(N3CC(NC(C4(Br)CC4)=O)CC4(CCC4)C3)ncn12 N1(C(C2CCC(C(C)C)CC2)=O)CC2CCC(C1)N2C(=O)Cc1cncn1C c1(C(=O)NCC(C(C)C)NC(C2CCCCS2)=O)cc2c(nn1)CCCO2 CC1CC(CC(=O)Nc2cc(F)ncn2)C(C)O1 CCCC(C)CCCC(=O)NCCC1CCCN(C(=O)C=Cc2csc(C)n2)C1 C(=O)(C1(C)OC(=O)c2ccccc21)NC1C(C)CN(C(C2(N(C)C)CC2)=O)C1 C(CC(C(=O)Nc1ccc(CCF)cc1)NC(=O)CC1CCC1)=CC C1(=CC(=O)NCC2(O)CN(C(C(OC)OC)=O)C2)CCC(C(C)(C)C)CC1 CC1OC2(C)CC1(C(N1CCCC1CNC(c1cccc(Br)c1Cl)=O)=O)C2 C=CCC(CC)C(=O)N(C(C)(C(=O)N1CC(N(C)C)C1)C1CC1)C N(C1CN(C(c2cnn(CCO)c2)=O)Cc2ccccc21)C(C(CCCC)F)=O n1(CC(=O)NCC(CNC(c2n(CC)nnc2C)=O)(C)C)ncc2cccnc12 c1(C(=O)NC2(CC=C)CN(C(=O)C(F)(F)c3ccccc3)C2)cc(C)ccc1F C1(NC(c2cnn(C(F)(F)F)c2)=O)CC2(C1)CN(C(c1csc([N+](=O)[O-])c1)=O)C2 c1(CCNC(=O)Nc2c(C(CC)(F)F)cccc2)ccc(C#N)c(C)n1 N1(C(CC(CC(=O)OC)C)=O)CCC2C1CCCN2C(c1cc(Cl)ccn1)=O c1(OC)ccc(CC(=O)N(CC(C)(C)NC(C2CC(C)(O)C2)=O)C)c(Cl)c1 Cc1ccnc(C(N2CCC(NC(c3cnc(-c4ncccn4)s3)=O)C2)=O)c1 c1(OC)cc(C)ccc1Nc1cc(C)nc(NC(c2cnon2)=O)n1 N1(C(=O)CCc2ccc(F)cc2)CCC2CCN(C(=O)CC3C=CCCC3)C2C1 c1(C2(CN(CCCNC(=O)CCc3nc[nH]n3)CC)CC2)ccc(O)cc1 CC(O)C(C(=O)N(C)CC1CCN(C(C2CC(OC)C2)=O)C1)NC(N)=O C(=O)(C1=CCCN(C(C2CCC(=O)N2)=O)C1)NC(C)CS(N)(=O)=O C1(C(=O)NCC(=C)CC)CNC(=O)CN1C(=O)CC1COCC(C)O1 N1(C(C2C=CC(C(=O)OC)C2)=O)C2CCCC1CC(NC(C1CCCCC1)=O)C2 N1(C(C(CC)CNC(C)=O)=O)CCCC(C)(NC(=O)C(=O)OC(C)(C)C)C1 N1(C(C(C)(C)C(N)=O)=O)CC2C3CCC(C2C1)N(C(c1ccnnc1)=O)C3 N1(C(C(C(=O)OCC)F)=O)CCN(C(=O)C(=O)CC(C)C)C2COCC12 c1(C(N2CCC(CN(c3ccnc4ncnn34)C)C2)=O)cc2cc(Cl)ccc2o1 C(C)(CNC(=O)CCN1CCOCC1=O)(CC(C)C)NC(CCSCC)=O C1(C(=O)OC)N(C(c2cc(C(F)(F)F)ccc2F)=O)CC12CCC2 CC1CC(OC(=O)CC2CCCCC2=O)CCO1 c1(C(=O)Nc2cncc(Cl)c2)cn2c(n1)CCN(C(C1CC(O)C1)=O)CC2 CC(C)(C)CCC(=O)NC1(CNC(C2CCC3(CCC3)O2)=O)CCCC1 c1(OC)cc(Cl)ccc1CNC1CC(C(=O)Nc2c(F)cccc2F)C1 N1(C(c2cc(C(=O)OC)sn2)=O)CCC2(NC(c3cccc(CO)n3)=O)CC2C1 c1(C(=O)NC(C)CCNC(C23CCC(CO)(CC2)C3)=O)ccc(Cl)c(O)c1N c1(C(=O)NCC2CN(C(C3CCO3)=O)CC2O)c[nH]c2c(Cl)cccc12 CCCC(C(C)CC)NCC(C)(C)CC C(=O)(C(C)(C)CS(N)(=O)=O)N(CCCCNC(c1nsc2ccccc12)=O)C C1(NC(COCCCC)=O)CCN(C(c2cnc(CC)[nH]2)=O)C1C1CC1 C1(CC(=O)NC2CCN(C(c3cnn(C(F)F)c3)=O)CC2)CCCOCC1 CC1=NOC(C(N2CC(C(N)=O)(CNC(=O)C(C3CCCCC3)=O)C2)=O)C1 c1(NC)cncc(C(=O)NCC(C2CC2)NC(C2CCCN2C(C)=O)=O)c1 c1(C(N(C2CCN(C(=O)CC3CCOCC3)C2)CC)=O)cc(N)nc(Cl)c1 C(C(F)(F)C(=O)NC1(COC)CCCCC1)OC.C12CCCCC1NC2=O Cn1cnnc1C1CCCC1C(=O)NCCN1CCC(NC(C2(CF)CC2)=O)C1 c1(C(N(C)CC2CCN(C(C(C)(C)SC)=O)C2)=O)ccc2cnc(C)n2c1 CC1(C)CCC(C(N2CC(C)(CCC(=O)NCC(F)C(C)(C)O)C2)=O)C1 c1(C(=O)NCCCC(C)NC(=O)CN(C)CCO)c(F)ccc(F)c1F CC1=C(C(=O)NC(C)C(C)(C)NC(C2CC3(CC3)CO2)=O)CCS1(=O)=O c1(C(=O)NCC2N(C(CN(C)C)=O)CC2)cc(NS(C)(=O)=O)ccc1Cl c1(OC)ccc(C(=O)N(C2CCCC(N(C)C(c3[nH]c(O)nc3C)=O)C2)C)cn1 C=CC1(C(=O)NCc2cscn2)CCN(C(=O)CC2CCC(O)C2)C1 C(=O)(C(=O)C(C)(C)C)NCCC(C)N(C)C(c1ccnc(Cl)c1F)=O c1(C(=O)NC2CCC(CNC(C=CCOC)=O)C2)c[nH]c(=O)c2ccncc12 N1(C(c2cc(OC)ns2)=O)CCN(C(c2ncc(C(F)F)cc2F)=O)C(CF)C1 C1(C(N2CC(CC(C)NC(C=C(CC)C)=O)C2)=O)CC12CCC(F)(F)CC2 C1(CC=C)(NC(=O)Cc2ccoc2)CCN(C(c2cnn(C)c2COC)=O)C1 C1(N(C(C(C(CC)C)NC2CC(C(=O)OC)C2)=O)CC)CCCCCCC1O N1(C(C2CN(S(N)(=O)=O)C2)=O)CC2CC1CCC2NC(C1(C(F)(F)F)CC1)=O CC1CCC(Nc2cccc(NC(N)=O)c2)CS1(=O)=O c1(C(=O)NCC(CC)NC(=O)C(C)(C)NC(=O)C(F)(F)F)cc(C)c[nH]1 c1(N(C)CC)cc(N2CCOC(C(C)(C)C)C2)nc(CO)n1.N1(CC)CCOCC1 C1(CC)CCCN(CCC(=O)N(C(C)CCNC(c2nc(C)nn2C)=O)C)C1 N1(C(C(C2(O)CCC2)NC(C(C(C)C)C#N)=O)=O)CCC2CN(C)CC2C1 c1(C(C(N2CC(N(C(=O)CCOC3CCCOC3)C)C2)=O)O)ccc(F)cc1 c1(C(N2C(CNC(CC(=C)Br)=O)COCC2)=O)cncc2c(F)cccc12 C1(NC(c2c(C)n(C3CC3)nc2)=O)CN(C(C2CC(C)CCO2)=O)CC(F)(F)C1 n1(CCCOC)nnnc1C(c1csc(C(C)C)n1)N(CCN1CC=CC1)C1CC1 C(=O)(C1Cc2c(Cl)cccc21)NC1CCN(C(c2c(CN(C)C)cco2)=O)C1 CC1(C)CN(C(=O)CCCc2cccnc2)C(CNC(=O)CC2C=CCC2)CO1 C1(COC)COCC1n1cc(C(=O)NCCCNC(C2(C)CC2(F)Cl)=O)nn1 C1(C(=O)NC(CCNC(C(C2CCCCC2)OC)=O)C)CN(S(N)(=O)=O)C1 C12(C(N(CCC(=O)N(C)CC3CCN(C)CC3)C(C)C)=O)CCC(C1)OC2C c1(C(CC)OC(=O)CSCC(=O)OC)ccc(Sc2nccn2C(C)C)cc1 C(=O)(C(C)(C)CNC(C12CCC(C(=O)O)C1C2)=O)OC N1(C(CCC#C)=O)CCC2CC2(NC(c2sc(C3CCCC3)nc2C)=O)CC1 c1(C(=O)NCC2OCCC(NC(CC3(CSC)CC3)=O)C2)cccc2cncn12 C(=O)(CCC(C)NC(=O)CC1CSC1)NCC(C1CC1)OC N1(C(C2CC3CCC3C2)=O)CCC2OCCN(C(c3cn[nH]c3)=O)C2C1 c1(C(C)C)cccc(NC(=O)C(C2CCCC2)NC(=O)C#CC2CC2)c1 N1(C(C)=O)CCCc2cc(NC(C3(Cl)CC3(F)F)=O)ccc21 C1(CCC)CCC(C(N2CC(NC(=O)CNC(=O)OC)C(C(F)F)C2)=O)CC1 N1(C(C(C2(C)CC2)NC(c2cc(C)c(F)cn2)=O)=O)CCN(C)CC(C)C1 C1(C)(OC)CCN(C(C2(CNC(=O)CC3CCN(C)C3=O)CCC2)=O)CC1 C(=O)(C(C)CC(N)=O)NCCN(C1CCCC1)C(CC1CC(SC)C1)=O C(=O)(C(CNC(c1cc(C)c(C)s1)=O)(CC)CC)NCC1CCC(OC)C1 C1(C(=O)OCC)C2COC(C(=O)NC3CCC(NC(C4CCSCC4)=O)C3)CC12 CC1CC(=O)CCC1C(=O)N(C(C)CNC(C1(c2ccncc2)CCC1)=O)C C1(C(=O)NCC2CC(CNC(c3cc(C(C)C)no3)=O)OC2)CCC=CCCC1 c1(OC)ccc(C(N2CCC2CNC(C2(CF)CC2(F)F)=O)=O)cc1N Nc1ccc(C(=O)NCC2CC3CCC2N3C(=O)C(F)=C2CCCC2)nc1N C1(C(=O)N(C2(CC)CCC2)C)COCC1C(N1CCC(c2nn[nH]n2)C1)=O Cc1cnc(C(N2CC(CNC(=O)CCn3cnccc3=O)CC2C)=O)cc1C C1(n2cc(SCC3(C)CC3(Cl)Cl)nn2)CCCN(C(c2cc(N)ccn2)=O)C1 Cc1cc(C(=O)NCc2cccc(CN(C(=O)Cc3ccco3)C)c2)cc(N)c1 Cc1c(C(=O)NCC2CN(C(=O)CC3CCCCC3O)CCO2)cccc1C#N N1(C(c2cnc(N(C)C)s2)=O)CC2(CCN(C(=O)C(C)(C)C)C2)C1 c1(C(=O)NC2(CNC(C3C(C)SCCC3)=O)CCCC2)cnn(C)c1C#N c1(C(=O)NC2CC(N(C(=O)C(c3ccccc3)F)C)C2)ncccc1Br C=CC(C)(O)C(=O)N(CC(C)CNC(=O)C(CC1CCCC1)CC)C C1(C(=O)NCC=CCNC(c2nc(C(=O)OC)sc2)=O)OC2CCC1C2 c1(OCCCC)ccc(C=CC(=O)NCCSc2ccns2)cc1 c1(OC)ccc(Br)c(F)c1CN1CC(C(=O)Nc2cccc(N)c2)CC(F)C1 N1(C(CC(=C)C)=O)CCC2(CO)CN(C(=O)C(C)(C)n3cc(Cl)cn3)CC2C1 N1(CCN(C(Cn2ncc(C)c2)=O)C)CCN(C(=O)C(F)C2CCCC2)CC1 CC(C)C(C)(O)C(=O)N1CC(CNC(c2ccc(Cl)s2)=O)C(F)(F)C1 CC(N=c1nn[nH]n1-c1ccccc1)c1cccc(Oc2ccccc2)c1 C1(CNC(=O)CC2CCN2C(c2ccn(CCF)n2)=O)(CO)CC2CC2C1 C(=O)(C(C)(C)CCNC(c1cnn(C)c1)=O)NCC(=O)N(C)C NC(=O)CCCCC(=O)NC1CCCCN(C(=O)C=CC=C(Cl)Cl)C1 CC1(CNC(C2CC3(CC3)C2)=O)CN(C(c2ccnc(Cl)c2N)=O)CCO1 CC(C)CC(C)C(=O)NCC1CN(C(c2ncncc2F)=O)CC(C(F)(F)F)O1 CC#CCCC(=O)NCC1CCCC(NC(C2CCCN2CCC(C)C)=O)C1 N#CCS(=O)c1ccc(C(N2CCC2CNC(=O)C(=O)NCC2CC2)=O)cc1 Cc1ccc(O)c(C(=O)OCc2ccc(=N)[nH]c2Cl)c1 C1(CNC(CCC)=O)CC2CN(C(=O)Cc3ncc(C)s3)CC12 CCC(CO)(C(=O)NCC1(C(=O)NCc2cccnc2)CC=CC1)OC C1(NC(=O)CCc2ccccc2F)COC2(CCN(C(c3coc(Cl)c3)=O)C2)C1 c1(NC(C2(c3nc(COC)on3)CC2)=O)cc2c(cc1N)OCCO2 Cc1cnccc1C=CC(=O)NC1(C2CN(C(c3csc(C(F)F)n3)=O)C2)CC1 c1(C(=O)NC(CCOC)Cc2ccco2)cnc(Cl)cn1 C(C)(C(=O)NCC(C(=O)N(C)Cc1ccoc1)N(C)C)(C1(C)CC1)OC N1(C(Cc2c(C)n[nH]c2C)=O)CCC2(CCCN(C)C2=O)C1 c1(NC(C(=O)NCCC(COCCC(=O)NC)O)=O)cccc(F)c1F C1(CCC)(C(N2CC(O)(C(C)NC(c3cncc(F)c3)=O)C2)=O)CCNC1=O c1(OC)ccc(F)c(C(=O)N(C)CCNC(C2(CSC)CC2)=O)c1Cl C1(CC(N2CCC(N3CCCC3)C2)=O)CCN(C(c2cc(CO)[nH]n2)=O)CC1 CC(Cc1ccco1)C(=O)N(CCCNC(C1(C(F)F)CCCO1)=O)C1CC1 C(=O)(N=S1(=O)CCNCC1)NC1CCCN(c2c(C)cc(Br)cc2)C1=O N1(C(C2(C)CC2)=O)CCC2(C1)CN(C(=O)C=C1CCOc3ccccc31)CCO2 C1(C(=O)NCCN(CCOC)C(c2cscc2C(N)=O)=O)CS(=O)(=O)C1 c1(CNC(COCC2CC2CNC(c2coc(C3CC3)c2)=O)=O)n[nH]cc1C(N)=O C#CCC(CC(=O)N(CCCCO)C)NC(c1cc(C)c(N)cn1)=O Cc1cnnc(O)c1C(N1CCC(F)(CNC(=O)CC(C)F)C1)=O CN1N=C(C(=O)NC2CN(C(=O)Cn3cnc4c3CCCC4)CC2F)CCC1=O c1(C(=O)NCC(C)(C2CC2)NC(=O)C=Cc2cccs2)cc(O)ccc1F N1(C(=O)C(C)N(C(c2ccccc2)CCC)CC)CCCCC1CCc1ccco1 c1(C(=O)NC2CCC(CCC(=O)NC3(CC#C)CC3)C2)ccc(O)nc1 N1(CC)CC(C)N(C(=O)CCN(C(=O)Cn2cccnc2=O)C)CC1C c1(CC)ncc(Cl)c(C(=O)N(C)CC2CCCCN2C(=O)C(F)C2CCCC2)n1 c1(OC)nc2ccc(C(N3CC(NC(c4cc(SC)ccc4Cl)=O)C3)=O)cc2[nH]1 c1(C(=O)NCC2N(C(C3ON=C(C)C3)=O)CCCC2C)[nH]cc2c1CCCC2 c1(-c2nc(NC(c3cc[nH]n3)=O)sc2)cccc(Br)n1 c1(OC)ccc2cccc(C(=O)OCC3CCN(C)C3=O)c2c1 N1(C(CCCCCOCC)=O)Cc2ccccc2C1CNC(=O)C(C)=CC1CC1 C(=O)(CC(C(F)(F)F)N1CCOCC1)NCCC1(C)CCN(C(CC(=C)C)=O)C1 Cc1cccnc1CC(=O)NCCC1CCN(C(C2CCC(O)C2)=O)CC1 N1(C(c2ccc(C(=O)NC3CC(C4CC4)C3)cn2)=O)CC2CCC(C1)O2 n1(CC)nnc(C)c1CNC(=O)C(C)=CCNC(C1(O)CCCC1)=O C(C(=O)NCC1(C(F)(F)F)CCCCC1)(C(C)C)NC(C)=O N1(C(c2cn(CC)nn2)=O)CCC(F)C(NC(c2ccc(Cl)cc2F)=O)C1 N1(C(Cc2scc(C)c2)=O)CCN(C(c2nnc(O)nc2O)=O)CC1CC(F)F c1(CC(C)NC(C2CCC23CCCO3)=O)ccc(F)c(F)c1 Cc1sc2ccccc2c1NC(C12CC1CN(C(c1ccco1)=O)C2)=O c1(C(=O)NC2C(NC(C(C)N(C(C)=O)C)=O)CCC2)ccc(CC(C)C)cc1F C1(CC(N2CC(NC(c3cccs3)=O)C2)=O)CCCS(=O)(=O)C1 N1(C(CN(C(Cc2n(C)ccn2)=O)CC2CC2)=O)CCC(NC(=O)C2CC2)CC1 N1(C(CCCN(CCC)CCC)=O)CC2(CCN(C(=O)CC(C)NC(N)=O)CC2)C1 CC(C)CCCCC(=O)NC1CC2(C1)CC2C(=O)NCC1CCCN1C c1(C(=O)NC2CC3N(C(C4(OC)CCC4)=O)C(CC3)C2)cnn2c1C(C)CCC2 C(=O)(CC(C)(C(F)(F)F)N(C)C)N(CC(O)CNC(=O)CN1C(=O)CCC1=O)C C1(C(=O)NCc2cncc(C)n2)C2CCC(C2)N1C(=O)CCc1ccccc1Cl C1(NC(C2CC3C=CC2O3)=O)CCN(C(c2ccc(Br)s2)=O)C12CC2 C1(NC(C2C(C)CCO2)=O)CCCC(C(=O)NC2CC3CCC2C3)C1 C1(C(CNC(CCOC)=O)NC(C2CCSCC2)=O)CCCCC1 c1(C(N(C2CCN(C(C3(CC)CCC3)=O)C2)C)=O)cc(Cl)ccc1N CCCCCC(CC)C(=O)N1CCC2(CC(NC(=O)C(F)C(C)C)C2)C1 c1(C(=O)NC2CCC3(CN(C(C4CN(C)C4)=O)C3)C2)sc2ccccc2c1Cl CCCC(C)CC(=O)N(C1CCN(C(=O)Cc2cc(F)ccc2O)C1)CC C1(N(C(c2csc(-c3ccccc3)n2)C(=O)NCCCF)CC)CCN(C)CC1 c1(C(N(C2CCN(C(CCCOCC=C)=O)C2)CC)=O)cc(Cl)c(Cl)[nH]1 N1(C(C2CCC(CC)O2)=O)CCC(NC(c2ccc(CO)s2)=O)C(CO)CC1 C1(CNC(C(C2(OC)CCCC2)(F)F)=O)CN(C(C23CCC2C3)=O)C2(CCC2)C1 c1(C(=O)NC2CCC(CCNC(CC(=C)C)=O)C2)c[nH]c2cc(OC)ccc12 Cc1cc(C(=O)N(C2CC(C#N)C2)CC(=O)NCC(c2ncc[nH]2)C)ccc1O O=C1NCCCCC1C(N1CCC12CN(C(C1CCCC13CC3)=O)C2)=O CC1CC(CNC(c2ccc(Cl)o2)=O)CCN1C(C1CCOC1C(F)(F)F)=O c1(CC(=O)NCC2CCN(C(CC(CC)(F)F)=O)C2)coc2cc(OC)ccc12 c1(OCC(=O)NCC(C(C)C)NC(c2occc2COC)=O)ccccc1C#N Cc1cccc(C(=O)NCC2(F)CCN(C(C3(O)CC3)=O)C2)c1F c1(CC(=O)NC2C=CCN(C(c3ccsc3Cl)=O)C2)cccc(C(F)F)c1 CC1CN(C(C2CCS(=O)CC2)=O)CC1CNC(C1CN(S(C)(=O)=O)C1)=O C=CC1(C(=O)OCc2cc(O)c(O)c(O)c2)CCN(C(=O)OC(C)(C)C)CC1 CCCC(CCNC(=O)C(C)(CSC)NC(=O)C(C)c1ccco1)CCC N1(C(c2ccc(SC)s2)=O)CC2CC2(CNC(C2CC(C)(C(N)=O)C2)=O)C1 c1(C(C(=O)NC2CC(NCC3CC3)C2)N(CC)CC)cnn(CC2(C)CCCS2)c1 C1(C(=O)NC(CC)C(N)=O)CCC2(CCN(C(=O)CCc3cccnc3)CC2)C1 c1(CC(C(=O)NC2CCCC2)NC(c2cnsc2)=O)ccc(O)cc1 O=C(NNc1ccc(-c2nn[nH]n2)cc1F)C1CCN(c2nccs2)CC1 N1(Cc2cc(C(=O)OC)sc2C)CCc2ccccc21.C12CCCC1NC2=O c1(CC(=O)NCCN(C(c2c(OCC)nsc2)=O)CC2CC2)cncnc1O c1(CC(=O)OC)ccc(CNC(=O)N(C2CCCN(C)C2)c2cnn(C)c2)cc1 CCCCCC(=O)NC1CC(NC(=O)COCP(C)(C)=O)C(O)C1 CN1C(=O)C(O)C(C(=O)Nc2ccc(Cl)cc2CC#N)C1c1ccccc1 C1(CC(C)C)(C(=O)NCC(C)CNC(c2sccc2Cl)=O)CCNC1=O Cc1cc(C(=O)NC2CCN(C(c3cnc(O)n3C)=O)C2)nn1CCO C(=O)(C(C)N=c1cc[nH]cc1)NCC1CC(NC(c2c(Cl)cn(CC)n2)=O)C1 c1(N(CC)CC2CCN(C(c3nnn(C)n3)=O)CC2)ncc([N+](=O)[O-])cc1C#N CS(=O)c1ccc(CC(=O)NC(CNC(c2ocnc2C2CC2)=O)C2CC2)cc1 c1(CCC)[nH]nc(C(=O)N(CC(C)NC(c2ccc(Cl)c(N)c2)=O)C)c1[N+](=O)[O-] O=C(CC1OCc2ncccc21)NCC12CC(CO1)N(C(C13CC(F)(C1)C3)=O)C2 N1(C(c2ccc(COC)o2)=O)CC(NC(c2cc(C#N)oc2C)=O)CC12CCC2 c1(CC)cccc(C(=O)NCCN(C)C(C2(C3CCCO3)CC2)=O)c1C c1(NC(N2CC(CC(C(=O)NCC3C(CC)C3)F)C2)=O)ccccc1S N1(CC)CCOC(C(=O)N(CCC(=O)NCC(N2CCCC2)C)C(C)C)C1 N1(C(c2cnc(OC)c(Cl)c2)=O)CC2(CCCN(C(=O)C(C)C3CC3)C2)C1 C1(C(=O)N(C)CC2CN(C(=O)C(F)OC)CCO2)(OC)CCOCC1 CC(C)(CC(=O)NCc1ccc(CCNC(c2coc(CO)c2)=O)cc1)C(F)F CC(C)C(C(=O)NC1CCN(C(c2conc2C2CCC2)=O)C12CC2)C(C)C c1(N2CCC(SC)CC2)nc2ccccc2nc1N1CCC(S(C)(=O)=O)C1 N1(CC(=O)Nc2n(C)ccn2)CCC2CCNC2C1 C(CC#CC)(C(=O)N(C1CCCCCC1)C)NC(C1CC(C#C)(O)C1)=O c1(C(CO)NC(C(COCC)NC(=O)Cc2nccn2C)=O)cccc(C)c1 c1(C(N2CCOCC(O)C2)C(=O)NC(CC)C)noc2ccc(Br)cc12 CC1(C)C(C(=O)NCc2ccsc2)CCN1C(=O)Cc1ccc(O)c(Cl)c1 C1(C(=O)NC(CC=C)CNC(c2nc(O)sc2C)=O)CC12CC(C)(C)C2 C(=O)(C1=C(Cl)CCOC1)N1C2(CCC1)NC2.C#Cc1nccnc1C(=O)OCC N1(C(c2c(OC)scc2)=O)CC2CC1CN(C(=O)C(C)(C)OC)C2 N1(C(COCC=C)=O)CCC(C=C)(C(=O)N(C2CCCC(C)C2)CC)C1 c1(O)ccc(-c2ccc(CNC(C3(Br)CC3)=O)nc2)cc1F.CCCOCCCl C(C)(CO)(C(=O)N1CC(N(C)CCO)C1)NC(C(C)=CC=C)=O c1(OC)nc(N2CCN(C)C(CNC(C3CCCC(C)O3)=O)C2)nc(C)c1F C1(C(=O)NCc2cc(OC)no2)CCN(C(=O)C(C)OC)C12CCC2 C(=O)(C(C(C)C)OC)NC1(CCC(=O)N(C(C=C)C)C)CCCC1 Cc1nc(O)ccc1C(=O)NC(C)CNC(=O)C(CO)c1ccccc1 c1(OCC)ccc(CNC2CC3(CCC3)C2O)cc1C(F)(F)F C1(C(=O)NC2CN(C(CCCOC)=O)CC2C)CC(c2cnn(C)c2)=NO1 Cc1cc(NC(C2CN(Cc3ccc(Cl)nc3)CCC2(F)F)=O)ncc1Cl N1(C(c2c(CC)noc2)=O)CC2CC(NC(c3cnn(C(C)C)c3C)=O)C2C1 C1(NC(=O)NCc2cc(C(=O)OCC)[nH]c2)CC(C)SC(C)C1 Cc1ncc(C(N2CCC(CNC(c3cc(C(F)F)cs3)=O)C(C)C2)=O)c(C)n1 C(=O)(C(C(=O)NCC(C)CNC(=O)C(c1ccc(F)cn1)(F)F)C(C)C)OCC C(C(CC(C)C)C(=O)NCC(C)CC(=O)N1CC(c2ccccc2)C1)OC Nc1ccc(Cl)c(C(=O)NCC2CN(C(=O)CCCCF)C2)c1 n1(CC)cc(C(=O)NC2(C)CC(NC(c3cc(C(N)=O)c[nH]3)=O)C2)c(C)n1 CCC(C)CCCC(=O)N(CCCNC(C1CC2CCCC(C1)C2)=O)C1CC1 N1(C(c2cn(CC#N)nn2)=O)CC(F)(F)CC1CNC(=O)CC1NC(=O)NC1=O S(=O)(=O)(c1cnc(N(C)CCc2ccns2)c(Cl)c1)NC(COC)COC CCS(=O)(=O)c1cccnc1CN.C(=O)(COCCOC)N1CCC1 C1(NC(c2cc(C)c(O)cc2)=O)COC2C(NC(C3COC(C)C3)=O)COC12 N1(C(c2c(CC)ncnc2)=O)CCN(C)CC1C(N1CC2CC1(CO)C2)=O Cc1cc(C(N2CC(c3cn(CCCF)nn3)C(C)C2)=O)c(C)o1 C1(CCC)CCN(C(=O)COONC(=O)COCCOC)CC1.CC c1(OC)ncc(Cl)cc1C(=O)NC(c1ccc(Br)nc1)C(C)(C)C N1(c2cc(C(=O)OC)ncn2)CCC(NC(c2cccnc2C(F)F)=O)C(C)C1 C1(C(N(CC(C)N(C(CC(C)C)=O)C)C)=O)CCC(F)CC1 N1(C(C2N(C(C)C)CCC2)=O)CCC(CC(C)NC(=O)COC(F)(F)F)CC1 C(=O)(CC(O)(C(F)(F)F)c1ncco1)N1CC(NC(=O)C=CCF)C(C2CC2)C1 N1(C(c2cnc(CC)o2)=O)CCC(F)(F)C(CNC(C2CC3C=CC2CC3)=O)C1 C1(CC=C)(NC(=O)C=CS(C)=O)CCCN(C(=O)C(O)C2CCCC2)C1 C1(C(=O)NCCCC)CCCCC1(C)NC(C1CC(N=[N+]=[N-])C1)=O c1(C(N2CCC(N(C(=O)CC(F)(F)F)C)C2)=O)cc(Br)c(F)c(F)c1F c1(CCn2cc(-c3cc(C)on3)nn2)cccc(Cl)c1F Cc1cncc(C(=O)N(C2CCCN(C(=O)NC3CC(C4CC4)C3)CC2)C)c1C N1(C(c2nc(CCC)oc2)=O)C2CCC(C2)C1C(=O)NC1CC2(CCCC2)C1 CCCCCC(CC)C(=O)NCC(C(=O)NCCOC1CC1)C(C)C CC(C)(CC(=O)N1CC2CCC1CN2C(C1(S(C)(=O)=O)CC1)=O)CC(F)(F)F N1(C(C2(CC)COC2)=O)CCC(NC(c2cc(C)c(C)nc2O)=O)C(CO)CC1 N1(C(CC(=C)CCNC(=O)CC(CC)SCC)=O)CCN(C(=O)CC(F)(F)F)CC1 N1(C(C=CCN(C)CC)=O)C2CCC1C1CC1(NC(=O)CCc1ccccc1)C2 C#Cc1cccc(C(=O)N(C2CCC(NC(=O)CC3=CCCC3)C2)C)c1C CCC(CC(=O)NCc1cnc[nH]1)N(C)C(c1ccc(NC)cc1)=O N1(C(C(CCNC(C2CCC2C)=O)OC)=O)CC(=O)NC(C)C1 Cc1nn(C)c(NC(C2C3CCC(C3)C2NC(c2cc(Cl)ncc2Br)=O)=O)c1Cl N1(C(c2cncc(Cl)c2)=O)CCCN(CCNC(=O)C(F)(F)C2CC2)CC1 CCC(C(=O)NC1CC(SCC(=O)OCn2cccn2)C1)c1cccnc1 N1(C(c2c(C#N)ccs2)=O)CC2(CCCC2)C1C(=O)NCC(=O)NC(N)=O c1(OC2CCN(C(C(=O)NCC(CC=C)C)=O)CC2)cc(Cl)ccc1Cl S(=O)(=O)(c1c[nH]c2ncccc12)N1CCC(n2cc(S(C)(=O)=O)nn2)C1 C12(NC(C(c3ccc(N(C)C)cc3)C)=O)CC(C1)N(C(c1ccnnc1S)=O)C2 CCCC(C(O)C(=O)N1CCC(F)(C#N)C1)NC(=O)CC(C)CC N12CCCC(CC1)C(=O)N(N1CCC(CC3CC3)CC1)C(C)CC2.CS C12(CC(F)(F)C1)NC(=O)C(CC)N(C)C2.C(C)(C)(C)NC(=O)OC c1(C(=O)NC2CC(CNC(C(C)SC(C)C)=O)CC2O)ncsc1S(N)(=O)=O OC1CCC2(CCCC2)C1CNCC1CCCc2nccn21 Cc1c(Cl)ccc(Cl)c1N(C=O)Cc1cc(-c2ncccn2)nn1C c1(NC(c2nncs2)CC)cc(Br)ccc1S(=O)(=O)N1CCn2nc(C)cc2C1 N1(C(C(C)Cc2ccccc2)=O)CC(NC(c2cc(N)c(F)cn2)=O)C2CC2C1 C(c1ccnn1C)=CC(=O)N(C)CC1CCN(C(COCC(=O)NC)=O)C1 c1(C(N2CC(NC(CCCCCSC)=O)C(C)C2)=O)cc(F)cc2cnccc12 C#Cc1cc(C(=O)NC(CC(C)CC)C(=O)NC2CCC3(CC2)N=N3)ccc1C C1(C(N(C)CC2CN(C(c3coc(O)n3)=O)C2)=O)CC12CCOC2 C(=O)(C1=C(C)CCC1)N1CC(C(=O)NCC(C(CC)C)C)OCC1 C12(NC(=O)C=CCO)CCC(CN(C(=O)Cc3ccc(Cl)cc3Br)C1)C2 CC(C)CCCCC(=O)N1CC2CCC(C1)N2C(=O)Cn1ncn(C)c1=O Cc1cnc(N2CC3(CCC(C(=O)Nc4ccccc4)O3)C2)c([N+](=O)[O-])c1 N1(C(c2c(C(C)C)[nH]cc2)=O)CCC(C2CCCN(C(=O)C3=C(Cl)CC3)C2)CC1 C1(NC(c2n(C(C)C)cnc2)=O)CCCCCN(C(C2CCCNS2(=O)=O)=O)C1 c1(NC(c2ccccc2)=O)cc(CNC(C2CCCCC2)C(=O)O)ccc1F C(=O)(C(CC)CC)NC1C(C(N(CCC#C)CCO)=O)CC1 Cc1cnc2n1CCC(C(=O)N(C1CN(C(C3CC34CCSCC4)=O)C1)C)C2 C1(NC(CCC(=O)NCC)=O)CC1C1CCCN(C(c2c[nH]nc2C)=O)C1 C12(NC(C3C(CCC)C3)=O)CC(C(=O)NCCCc3ccsc3)(C1)C2 N1(C(c2coc(Cl)c2)=O)CCC2(CCCCN(C(c3nncn3C3CC3)=O)C2)C1 C1(C(C)(C)C)(CO)CCN(Cc2ccccc2)C1.C1(=O)CO1 Cn1nc(C(N2CCC(CCC(=O)NCCC3COC(C)(C)C3)C2)=O)cc1Cl Cc1cnc(CNC(C2(CCF)CCC2)=O)[nH]1.C12CCC(C1)NC(=O)CC2 N1(C(C2(OC)CCSC2)=O)CC2CCC(C1)C2NC(c1ccnc2ccnn12)=O CC(C)C1=NOC(C(=O)NCc2ccoc2C(=O)NCc2ccoc2)C1 N1(C(c2n(C)ncc2)=O)CC(NC(=O)Cc2cc(-c3ccco3)on2)C(F)C1 C#CC1(C(N2CCC(OCCCCC)C2)=O)CCCC1 C1(NC(c2cc(C)n[nH]2)=O)CCC(C)(C)CC1CNC(=O)CN(C)C(=O)C1CC1 c1(OCC)cccc(Cn2c(N3CCC=C(C)C3)nnc2C2CCOC2)c1 Cc1cc(F)ccc1C(=O)N(C1(C(=O)NCC2CC(C)(C)CO2)CCC1)C1CC1 CN(CCCC(=O)NC12CC1CN(C(=O)C#CC1CCC1)C2)N=O N1(C(c2cccnc2O)=O)CCC(CO)(NC(C2(F)CCOC2)=O)CC1 C(N=c1nc(O)c(Br)c[nH]1)C1N(C(COc2c(C)n(C)nc2)=O)CCCC1 c1(NC(=O)CCn2cc(-c3nccs3)nn2)cccc(F)c1 CC(C)(CCNC(C1CCSC1)=O)C(=O)Nc1ccc(F)c(F)c1 c1(CNC(C2C(C)C2)=O)cccc(C(=O)N(C)CCN2CCOC2=O)n1 c1(C(N2C(CCNC(c3n[nH]c(CC)c3C)=O)CCCC2)=O)ccc(N)c(F)n1 Cc1nn(CC(=O)NCC2(C)CN(C(=O)C3=CCSC3)CCO2)c(C)c1Cl Cc1cc(NCC(C2CC2)NC(=O)CC(O)C(C)C)c(Br)cc1[N+](=O)[O-] CC1CN(C(C2CCCC(O)C2)=O)CC1NC(c1cc(-c2ccccc2)co1)=O CC(=O)CCCC(=O)N1CCC(O)(CCNC(C2CN3CCN2CC3)=O)C1 Cc1nc(C(N2CC3(CCN(C(=O)Cc4csnn4)C3)C2)=O)c2ccnc-2[nH]1 c1(CC(CNC(=O)CC2CCCNCC2)OC)cccc(Cl)c1 Cc1n[nH]c(C)c1C(=O)NCC1CCCN1C(c1cccc(CC(F)(F)F)c1)=O N1(C(C(COC)O)=O)CCC2CCN(C(c3cc(OC4CC4)ncc3Cl)=O)CC12 C1(C(=O)NC2C(NC(CC3(COCC)CC3)=O)C2)CC2CC2C1 CS(=O)(=O)c1ccc(CC(=O)NC2CCN(C(c3cc(C4CC4)on3)=O)C2)cc1 C1(NC(CCC(=C)C)=O)CCC(C)(CNC(=O)C(c2ccc(F)cc2)OC)CC1 C12(C(N(CC(C)NC(c3ccccc3CC#N)=O)C)=O)CC(C1)C(C)(C)O2 c1(OC)cc(C)ccc1C(=O)NC1CCN(C(=O)CCCC(C)=O)C1C(C)C c1(C(=O)NCC2CCCN(C(CC(CC)SC)=O)C2)cccn2c(CO)nnc12 c1(C(=O)NCC(=O)NC(C)CNC(c2coc(Cl)n2)=O)ccccc1CC#N c1(N(C(=O)CN2CCC(NC=O)CC2)C)ccc(Br)cc1F c1(C(=O)NC2C(NC(c3ccc(C(F)F)c(F)c3)=O)CCC2)ccc(O)c(Cl)n1 C(=O)(CCCC(C)=O)N(C(CC)C(=O)NCC(c1ccccc1C)C1CC1)C Cc1nn(CC(=O)NC2CCC(N(C(=O)C=CCF)C)C2)c(=O)n1C c1(C(=O)NCCCN(C(=O)C=Cc2cn[nH]c2)C(C)C)cc(CS(C)(=O)=O)on1 N1(C(c2nc(OC)oc2)=O)CCCC12CCN(C(=O)CSc1nncn1C1CC1)C2 N1(C(CNC(CC)=O)=O)CC(NC(C2CS(=O)(=O)CCO2)=O)CC2(CC2)C1 N1(C(C(CC)C(C)O)=O)CC2CC(NC(=O)C(F)C3CCOC3)CC2C1 Cc1cnc(C(N2C(C(N3CCCC3C(O)CO)=O)CC2C)=O)c(C)c1 c1(C(=O)OCC)ccc(CNC(C2(C)CC2(C)C)c2nnnn2C(C)C)[nH]1 C1(NC(Cc2c(C)noc2Cl)=O)CCCCN(C(=O)C(C)(O)c2ccccn2)C1 C1(C(=O)NCC(C)CN(C(=O)Cc2ccc(O)cn2)C)CC1C1CC1C N1(C(=O)NC(CCC(=O)NC)=O)CCC(C2CC2)C1C(N1CC2C=CC1C2)=O c1(C(C)N(CCCCO)C(CSc2ccncc2)=O)ccc(C#N)cc1F N1(CC2CC=CC2)CCC2(CCOCC2)CC1 c1(C(N2CC(F)(C(=O)NC(C3CCOC3)C)C2)=O)cc(C#N)ccc1Br N1(C(Cc2c(C)n[nH]c2C)=O)CCCCC(NC(c2ccncc2Br)=O)C1 N1(C(C2CC(C)N(C)C2)=O)CCC2(C=C(C(=O)N3CC(NC(N)=O)C3)C2)C1 N1(C(C2(C)N(C)CCC2)=O)CC2CCN(C(c3cn(CC4CC4)nn3)=O)C(C2)C1 CN1CC(C(N2CC(C3CN(C(=O)CC4(C5CC5)CC4)CCO3)C2)=O)CCC1=O c1(C(N(CCCN)C2CC2)=O)cc(F)cnc1O.CC1(OCC(=O)C(=O)N)CCC1 c1(C(=O)OCC)c(NC(C2CCCN2C(c2ccc(N(C)C)s2)=O)=O)ncn1C S(=O)(=O)(c1cccc(F)c1)NCC(N1CCN(C(c2ncn(C)c2)=O)C2C1C2)=O N1(C(C23OC(C)C(C2)C3)=O)CC2(CC(NC(c3n[nH]c4c3CCSC4)=O)CO2)C1 C(=O)(C#CC1CCCCO1)NCC(C)(C1CC1)NC(c1cc(CSC)c(C)s1)=O C(=O)(C1CCSc2ccccc21)N(C1CCN(c2ncccc2[N+](=O)[O-])C1)CC CC(C)C(CO)CCNC(C1CC(C)N1C(=O)COCCCN(C)C)=O N1(C(=O)Cc2ccc(O)c(O)c2)CCC2CN(c3ncnc4cc[nH]c34)CCC12 C12(C(N3CC4C(CNC(C5CCC(=O)NC5)=O)C4C3)=O)CCC(CC1=O)C2 C1(C)(C(=O)NCC(C)(C)NC(C(CC)n2ccnc2)=O)CCC(=O)N(C)C1 N1(C(C(COC(C)C)NC(C)=O)=O)CC=CC(NC(C2(C)CS(=O)(=O)C2)=O)C1 C(=O)(C(C)(C)CCCO)NCC1C(NC(C2(COCC)CC2)=O)C1 N1(C(C2CN(C(C)C)C(=O)C2)=O)CCCN(C(C2CC(CF)C2)=O)C(C)C1 c1(-c2c(NCC)cco2)cc2nc[nH]c2cn1.c12cc(no1)C(=O)NC2.C(=O)OCC CCCCC(C)(C)NC(=O)C(COCC)NC(c1nc(O)sc1C)=O c1(C(N2C(C(=O)NCC3(OC)CC3)COCC2)=O)cc(C)c2ccccc2n1 C1(C(=O)NCC(C)CN(C(=O)Cn2ncn(C)c2=O)C)CCC2(CCC2)CC1 C(=O)(C(C)CC(N)=O)NCC1C(NC(C(C(C)C)OCC(C)C)=O)C1 C1(c2ccn(C(C)C)n2)CN(C(=O)C(=O)NC2CN(C3CCCC3)C2)CCO1 CC1(C)COC(CCC(=O)NC2C3CN(C(=O)CCC4CCCC4)CC23)C1 N1(C(c2c(OC)c(C)cs2)=O)CC(C)C(NC(c2cc(O)nc(O)n2)=O)C(C)C1 C(=O)(C(C)(C)C(O)C(C)C)N(CC(=O)OCC)C.C1(=O)CN1CC(C)C c1(C(C)NC(C)CN=[N+]=[N-])cc(F)ccc1C(N1CCCC1)=O CC(C)CN=C(NCc1ncn(C)n1)NCC1C(F)(F)C12CCCC2 N#Cc1cccc(C(N2CC3C(NC(=O)CC45COCC(C4)C5)C3C2)=O)c1 Cc1coc2c(C(N3CCCC(CCNC(=O)C(C)CC(F)F)C3)=O)cccc12 C1(CCNC(CN(C(=O)CC2OCCC2C)CC#C)=O)OCCC1C N1(C(C(C)(C)C)=O)CCN(C(C2CCC(=O)O2)=O)C(CC(F)F)C1 CCC(CC(=O)N1CCCC1(C)C(=O)N(C)Cc1ncc(C)o1)CC(C)C c1(C(=O)NC(CNC(C2ON=C(C)C2)=O)(C)C)cccnc1CN1CCOCC1 c1(C(N2C(CNC(C3CS(=O)(=O)C3)=O)COCC2)=O)cccn(C2CCC2)c1=O N1(C(c2ccc(CC)cc2)=O)CCN(C(=O)C2=NNC(=O)C2)CC1CC(F)(F)F C(=O)(C(C)N1CC(C)C1)NCC(=O)NCC(=O)N(C(CC)C)C C12(NC(CCCOCCC)=O)CCCC1N(c1ncccc1C(=O)OC)CC2 C1(O)(C(=O)NC(C)CNC(=O)Cn2cnnc2O)CC(F)(F)C1 C1(NC(C=C(CCC)C)=O)CC2(C1)CC2NC(c1ccc(C2CC2)nc1)=O C12(C(=O)NC3C(CNC(c4ccnc(Cl)c4Cl)=O)CCCC3)COC(CCO1)C2 N1(C(c2cc(CC)c(C)s2)=O)CCC(O)(CNC(=O)C(F)CC2CC2)CC1 c1(CCNC(N(C(c2ccncc2)C)C)=O)csc(-c2ncccn2)n1 CC1CN(c2ccccc2NC(c2cccc(N(C)C)c2)C)CC(C)O1 C(=O)(C(CC1CC1)NC(c1cnc(CC)o1)=O)NCC(COCC)O C(=O)(CCC(C)(C)NC(c1cnc(Cl)s1)=O)N(C1C(C)CC1)C N1(C(c2c(C)noc2)=O)CCN(CCCCCNC(=O)CNC=O)CC1 c1(C(c2nnnn2CC)NC(C(COCC)C)C)cc(-c2ccccc2)nn1C C1(CCC)CN(C(c2cn(C3CC3)nn2)=O)CCN1C(=O)CCN1CCC(F)C1 c1(C(=O)NCC2(OCC)CN(C(=O)C(F)C3CCC3)C2)ccc(NC)nc1C c1(CC)ccc(CC(=O)NCC2CCC(NC(=O)CC(F)(F)F)C2)cc1 c1(C(=O)NC(C)C(C)(C)NC(=O)Cc2ccc(F)c(Cl)c2)cc([N+](=O)[O-])n[nH]1 c1(N2C(CCNC(C(C)(C)C)=O)CCCC2)ncnc2c(Br)c[nH]c12 CC(C)CC(C)CNC(=O)NC(C(F)(F)F)C1CCC1 c1(NC(C2C(C(=O)Nc3c(C(=O)NC)cccc3)C2)=O)cnc(O)nc1O Cc1ccc(CC(N2CCCC2(C)CNC(C2CCC(=O)N(C)C2)=O)=O)cc1F CN1CCC(C)(C(N2CCC(CC(N3CCC(CC(C)(C)C)C3)=O)C2)=O)C1 CC1CCC(CC(=O)NC(CCN(C)C)C(=O)NCCC(=O)NO)OC1 N1(C(=O)CCC2CCOCC2)CCCC(CNC(C2CC23CC3(F)F)=O)C1 C1(CC(=O)NC)CN(C(=O)CC(F)(F)c2ccccc2)CCN1C(=O)C1CC1 O=C(C1=COCCC1)NC(Cc1cc[nH]n1)C(=O)NCCc1cocn1 N1(C(Cn2cc(C(N)=O)nn2)=O)CCC(CCN(C)C)C(F)(F)C1 CC1(C#N)CCN(C(C2C3CCC(C3)C2NC(=O)C(C)(F)c2ccon2)=O)C1 N1(C(=O)CSc2n[nH]c3ccccc23)C2CC3C4CC(C3C2O)C1C4O C=CC(CC)C(=O)NC1CCN(c2ccnc(C3CC3)n2)C1C Cc1nn(CC(N2CC(F)(CNC(=O)C(C)(C)n3cccn3)C2)=O)c(=O)o1 C1(C(c2n(CCCOC)nnn2)NCCn2cnnc2)CC2(C1)CC(F)(F)C2 n1(CC)cnc2nc(N3CC4CC3CO4)nc(NCCC3(C)CCCO3)c12 C1(CNC(C(CC)C)=O)CCN(C(c2ccc(F)c(Br)c2)=O)C12CC2 C1(CN(C(C2CC(C3CC3)C2)=O)CC)CCN(C(=O)CCc2nccs2)CC1 c1(C(=O)NC2C(CNC(C3=CCC(C)CC3)=O)C2)ccc2nc(O)n(C)c2c1 c1(OC)ccc(-c2cn(C3CC(C(=O)NC4CCCCC4C)C3)nn2)cc1OC c1(C(N2CCN(C3CC(C)(C)OC3=O)CC2)=O)cnc2c(c1)CCCO2 C1(CNC(=O)C2CC2)CC(O)CN1C(c1cc(-c2cccs2)on1)=O Cc1ncc(CC(N2CCCC2C(C)(C)NC(=O)C(O)Cn2cncn2)=O)s1 c1(C(=O)NCC2C(NC(C(C3CC3)OC)=O)CC2)ccc2nonc2c1 C(=O)(C(CC(C)(C)C)OC)N(CCN(CCOC)C)CC1CC1OC C1(CNC(C2CCC(COC)C2)=O)CC2(C1)CN(C(=O)C(F)=C(C)C)C2 N1(CC(=O)N(CC#C)CC=C)CC(NC(c2c(C)cccc2F)=O)CCC1C c1ccc(NC(=S)NCc2csc(N3CCOCC3)n2)cc1 N1(C(C=CS(C)(=O)=O)=O)CC(NC(=O)Cc2ccc(Cl)s2)CC2(CC2)C1 CC(C)(C(=O)NC)N1CCCCC1.C12=CCOCC(=O)N(C1)C2.N1(CCN)CCCC1 Cn1cc(C(=O)NC2CC(CNC(C3CC34CC4)=O)C2)c2cccc(Cl)c12 C1(S(N)(=O)=O)(C(=O)NC2CC(C)(NC(CSc3n(C(C)(C)C)ccn3)=O)C2)CC1 N1(C(C2CCN(C(c3cc(CC)[nH]n3)=O)C2)=O)CCC(C)(CCO)CC1 c1(C(N2CC3CCC(O)CC23)C(=O)NC(CC)(C)C)ccc2ccccc2c1 N1(C(C(CC)N(C)C)=O)CCn2ncc(CNC)c2C1 c1(CC(=O)NCC2C(NC(C3(C)ON=C(C)C3)=O)COC2)cccc2nsnc12 c1(C(N2CC(OCCNC(=O)CCCCC3CC3)C2)=O)cc[nH]c2nccc1-2 C1(CC(=O)N(CCOCCNC(C=CC=CC)=O)C)C=CC(OC)C1 N1(C(C(C(C)C)OC)=O)CC(C)N(C(c2cc(Cl)nn2C)=O)CC1C N1(C(c2cc(SC)oc2C)=O)CC2CCN(C(C3C4CCC3CC4)=O)CCC2C1 c1(C(N2CCC(CCC)(NC(C3CCCCO3)=O)C2)=O)cc(O)nc(C)n1 CCC(CC)C(C(=O)NCC(CC1CC1)C(=O)NCC1CC(F)C1)OC CCCCC(O)CC(=O)NC1CCCC1CNC(c1ccc(CO)c(F)c1)=O C1(C(=O)NCCC2CCCN(C(=O)OC)C2)CCCC(C)(C)O1.C12(CC1)C(=O)N2 c1(C(=O)NCC2C(NC(c3c(C)nc(C4CCC4)o3)=O)C2)cn(C)c(=O)cn1 N1(C(c2cc(CC)on2)=O)CC2(CCN(C(c3ccc(C)cc3I)=O)CC2)C1 CCCC(O)(CCC)CC(=O)NC(CCN(C)C(c1cnc(C)s1)=O)C(C)(C)C N1(C(C(C2CCC(=O)N2)C)=O)CCCN(C(=O)C(N)=O)CCC1 CS(=O)(=O)CCCCNC(C1(C2CCC2)CCC1)=O c1(C(=O)NCC(CC)NC(=O)CC2CCN(C)CC2)ccc(C)nc1C(C)C C(=O)(C1CCCc2scnc21)N1CCOCC(CNC(C=CSC)=O)C1 C(CC(=O)Nn1cncn1)N(CCCO)C(C1(C)CCC1)=O c1(C(N(CCN(C(C(c2ccc(C)o2)C)=O)C)C)=O)scc(C)c1Cl Cc1ccc(C=CC(=O)NC(CNC(=O)CCC(=O)c2ccc(Cl)s2)CO)s1 C1(C(N2CC(NC(c3c(CC)con3)=O)C(O)C2)=O)CCOCC12CCCCC2 N1(C(C(CC(=O)OC)(C)C)=O)CCC2C1CCCN2C(=O)C(F)CC(C)C C(=O)(C(C)CNC(=O)C(Cn1cccn1)NC(=O)CCC1CC(C)C1)OC C1(C(=O)NCC(CNC(c2c[nH]nc2C(F)(F)F)=O)O)CCCCC12CCC2 C#Cc1cc(F)c(C(N2CC(NC(=O)C(F)=CC3CC3)C(C(F)F)C2)=O)cc1F c1(CNC(=O)NC(CC(C)=O)Cc2ccccc2)ccc(OC(F)(F)F)cc1F c1(C(=O)NCCC(CNC(CC(=C)C)=O)O)ccc(Cl)cn1 N1(CCNC(C(=O)NCCCC(C(=O)OC(C)C)O)=O)C(=O)NC(C)(C)C1=O Cc1cc(Cl)cc(CNCC(C(C)(F)F)c2ccccc2)c1O C#CC1COCCN1C(c1occc1CNC(C1C(C)(C)C1(C)C)=O)=O C(=O)(CN=c1cc[nH]cc1)C(C(c1cn(C)nn1)NC(CSCC=C)=O)=O.NC N1(C(C2(C(C)NC(=O)CC3CCC3)CC2)=O)CCN(C)C(C2CC2)C1 Cc1ccc(F)nc1C(=O)NCCn1cc(CC2(CO)CCC2)nn1 C(=O)(C(C)CCC(C)(C)C)N(C1CN(C(c2nnn(C)n2)=O)C1)C Cc1nc2ccc(C(N3CCC4(NC(=O)CC5(C#N)CC5)CC4C3)=O)cc2[nH]1 c1(C(=O)NCC2N(C(C(CC=C)N(C)C)=O)CCC2)c[nH]c2ccncc12 C(=O)(C(Cc1ccco1)N(C)N1CCN(C(C)C2CC2)C(=O)C1)OCC C1(CNC(C(c2ccccc2F)C)=O)CN(c2ccnc(Cl)n2)CC(C)(C)O1 Cc1ccc(C(=O)C(=O)NC(C)CC(C)NC(=O)C(F)n2cccn2)cc1 c1(C(=O)NCCC(C)NC(c2ccc(Cl)nc2O)=O)ccc2oc(O)nc2n1 N1(C(Cc2c(C)nn(C)c2)=O)CCC2(CC1)CC2NC(c1nc(=O)n(C)[nH]1)=O c1(CN(C2CCCC2)C)cc2cccc(-c3ccccc3OC(F)F)c2s1 C1(O)(CNC(C(C)(Cl)Cl)=O)CCCN(C(=O)C(F)n2cccn2)C1 C1(CC(=O)NCCCOCCNC(c2c(CC)nc[nH]2)=O)CC2CCC1O2 C=C(C)C(C)(C)C(=O)NC(CNC(C1C2CCC1(c1ncco1)C2)=O)C(C)C c1(C(N2CCCC(C(C)NC(Cc3c(C)non3)=O)C2)=O)cn(C)c(=O)nc1O N1(C(Cc2ccc(CC)cc2)=O)CCCC(CO)(NC(=O)CCC#N)C1 C(CC1=CCN(C(C2CC3(CCC3)CO2)=O)CC1)NC(CC(C)C(F)F)=O c1(OC)cc(C(N2CC(F)(CNC(=O)C(F)(F)COC)C2)=O)cnc1O c1(OC)ccc(F)c(F)c1C(N1CCC1NC(C)=O)=O.N12CCN(CC1)CC2=O c1(N2CCC(N(CC)CC)C2)cc(C)c(S(=O)(=O)N(C)C)cn1.C(CC#N)N CC(C)C(C(=O)N(C)CCOCCNC(=O)Cc1nc(=N)[nH][nH]1)C1CCC1 C1(C(N2CC3(CC(NC(C4CCC(=O)O4)=O)C3)C2)=O)CCc2nccn2C1 N1(C(=O)COCCC2OCCO2)CC2CCN(C(c3cccc(F)c3)=O)C2C1 C1(CC)(NC(C2COC3(CCC3)C2)=O)CCCN(C(=O)CCNC(C)=O)C1 Cc1ccc(C(=O)NCC2CC3(CC3)CN2C(=O)C(C)S(N)(=O)=O)cc1C CCC(O)C(C)(C)C(=O)N1CCN(CC2(NC(=O)C(C)c3ccco3)CC2)CC1 c1(C(C)CC(=O)NCC(CNC(=O)CC2CC=CC2)CO)ccc2c(c1)OCO2 N1(C(=O)C=Cc2cnccn2)CC2(C(N3CC(O)(C4CC4)C3)=O)CC1CCO2 C=CCCCC(C(=O)Nc1csc2ccccc12)N(C(C)C(=O)OC)C c1(C(c2nnnn2C(C)C)NC2C(CC)OCC2)cc(OC)c(CC2CC2)o1 c1(NC2CCN(C(C(CC)c3ccccc3)=O)C2)cccc(C)c1 c1(CC(C)NC(=O)C(c2cccnc2)NC(C2CC2(F)Cl)=O)nccn1C c1(C(=O)NC(CN(C(=O)CCC2CCOCC2)CC)C)coc2c1COC2 c1(C(N2C(CC)CN(C(=O)C(C)CC#N)CC2)=O)ccc2cnc(C)n2c1 S(=O)(=O)(c1cnc(NC2CCN(C(C)(C)C)C2)cc1C)NC(COC)(C)CO c1(CC(=O)NCCC(CCNC(CC(C)C(F)F)=O)C)ccc2c(c1)CCCO2 N1(C(c2n(CC)ncc2)=O)CC2CCCC2(C(=O)NOCCN(C)C)C1 C1(NC(C2(CNC(c3cc(CC)[nH]n3)=O)CC(C)(C)C2)=O)CC2(C1)CN(C)C2 C1(C(=O)NC(C)(CNC(c2ccc(CO)s2)=O)CO)COc2cc(F)ccc2C1 C1(NC(=O)Cc2ccc(Cl)s2)CC2CC(C1)N(C(=O)CCOC1COC1)C2 N1(C(CC(=C)C)=O)Cc2ccnn2CC(NC(=O)CCc2nc(CCC)no2)C1 C1(C(=O)NC2N(C(c3cccc(CC)n3)=O)CC2C)CCCCCC1CO S(=O)(=O)(c1cnc2ccsc2c1)N1Cc2c(nn(C)c2C(N)=O)CC1 C1(NC(C(C)OC(C)C)=O)C=CCN(C(C2(c3ccc(F)cn3)CC2)=O)C1 c1(C(=O)NCC(CN(C(=O)CCc2ccc(Cl)s2)CC)(C)C)cnn(C)c1C#N c1(N(C)CC2CCCS2)nc(=NCCn2ncc(Br)n2)[nH]c2ccccc12 CCCC(C(=O)NCC(CC(C)C)NC(=O)C=CCN1CCOCC1)OC C1(C(COC)C)CCN(C(=O)CC2CC(NC(c3ccc(COC)o3)=O)C2)CC1 N1(C(C2(CC#C)CCOC2)=O)CCCCC1CN(C)C(c1cncnc1)=O CCC(C)CC(C)(c1nnnn1C1CCCCC1)NC(c1cccnc1)CCO C(=O)(C(F)C(C)(C)O)N1CC(C(=O)NCC(c2ccnn2C)C)OCC1 N1(C(c2cc(C#N)no2)=O)CCCCCC1CNC(=O)CCC1CCC(=O)N1 N1(C(c2cnc(SC)s2)=O)CCN(C(=O)CC(F)(F)F)CC1C1CCC1 Cc1ccc2cc(OCc3nnnn3-c3ccc([N+](=O)[O-])cc3)ccc2c1 Cc1cnc(C(N2CCCC(O)(CCNC(=O)CCCCN(C)C)C2)=O)cc1C CCCCC(C(=O)N1CCN(C(c2ccc(C(=O)OC)nc2)=O)C(C)C1)N(C)C N1(C(C(C(CC)C)NC(=O)COCCOCC)=O)CCn2nc(C)cc2C1 C(=O)(C(C)(C)CC(C)(C)C)N(CC(=O)N(CCC(C)C)C)C1CCC1 c1(CC)occ(C)c1C(=O)NCC(C)NC(C1CCOC(C)C1)=O c1(C(C(N2C(CNC(=O)CC3(CO)CC3)CCC2)=O)O)cccc(Br)c1 Cc1c(C(=O)NC(C)C(CO)NC(C2CC3CCC2C3)=O)sc2nccn12 c1(-c2nc(C(C)C)nn2C2CCSCC2)cn2cc[nH]c(=O)c2n1 Cc1cc2c(cc1C)C(C(=O)N1CC3CCN(C(C4CC(O)C4)=O)CC3C1)CO2 CC1(C)C(NC(c2cnccc2Cl)=O)C2CCCN(C(C3CCC(=O)N3)=O)C12 CCCCC(C(=O)NCC(C(C)C)NC(c1ccccc1SCC)=O)N(C)C C1(C(=O)NC2CCN(Cc3n(C)ccn3)C2)CCC([N+](=O)[O-])CC1 c1(C(=O)NCC2CN(C(CCCNC(C)=O)=O)CC2C)c(C)cnnc1O N1(C=O)CCCC(C2CCN(CC(=O)OC)C2)C1.C=C(C)C(=O)NCCNC(=O)C(C)C c1(OC)ccccc1C(C)COc1cccc(-n2cnnn2)c1 C12(C(N3CC(N(C)CC)C3)=O)CC(CO1)N(C(=O)C(n1cc(C)cn1)C)C2 c1(N2CCC(C(C)NC(=O)CN3CCC(C)C3)CC2)ncnc2c1nnn2C1CC1 S(=O)(=O)(c1ccc(N=C2OC(=O)N2)cc1)NC(C)(C(F)(F)F)C1CC1 c1(OC)c(CNCC2CCN2C(=O)OC)cccc1CC(C)(C)C N1(CCNC(C2CC(=C3CC3)C2)=O)CCCCCC1.c12cc(no1)C(=O)NC2 CC(C)C(C(C)NC(C1(C)CSC1)=O)NC(=O)CSc1nnc(-c2ccco2)o1 c1(C(CCC2CC2)NC(C(=O)NCCN(CC)CC)C)ccc(F)cc1.C(=O)(N)N c1(C(N2CCC(NC(C(CC)N(C)C)=O)CC2)=O)ccc(Cl)c2c1OCCO2 c1(C(=O)OCC)cccnc1NCC1CCC(NC(C2CC(C(C)C)C2)=O)C1 C1(OC)(CNC(C2CCCN2C(c2cc(Cl)no2)=O)=O)CCC(C)C1 C(=O)(C1SCCc2sccc21)N1CCN(C(c2sccc2F)=O)CC(C)(F)C1 N1(C(c2c(C)nn(C)c2Cl)=O)CCc2sc(CNC(=O)Cc3cc[nH]n3)nc2C1 C1(NC(c2cncnc2)=O)CN(C(=O)Cn2cccn2)CCC1CO C(=O)(C(CC)c1ccccc1)NC1(CCCCNC(CCSCCC)=O)CC1 c1(C(C)OC(C(COC)CC2CCCC2)=O)nc2ccccc2o1 Cc1cc(O)ncc1NC(=O)C(CNC(c1cccc(O)n1)=O)CC1CCCC1 Cc1c(C(=O)NCCOCC(=O)N(C2CC2)CC2CCCCO2)cncc1F CC(C)(C)CC(O)C(=O)N1CCC(CCC(=O)NCC2(c3ccon3)CC2)C1 c1(C(c2nnnn2CCCF)NCCC2(C)COCCO2)cc(S(C)(=O)=O)co1 n1(CC)cc(Cl)c(C(=O)NCCNC(C2CN(C)C2)=O)n1 C1(CNC(c2n(C)cc(Cl)c2)=O)CN(C(=O)C2=C(Cl)CC2)CCC1(F)F C(=O)(CCC(F)(F)CN=[N+]=[N-])N1C(C)(C)CC(NC(=O)COCC(F)(F)F)C1 C(=O)(C(C)S(=O)(=O)C(C)C)NC(CCCNC(C(C)(C)NC(C)=O)=O)(C)C CC(C)(C)C(C(=O)N1CC(NC(C2(CF)CC2)=O)C(C(F)F)C1)c1ccccc1 N1(C(N2C(c3ccc(OC)cc3)CCC2)=O)CCC(C#N)(CO)CC1 C(=O)(CC(C(F)(F)F)NC(C1(NC2CC2C(=O)O)CCC1)=O)NC C1(NC(CN2CCC(OC)C2)=O)CCN(C(=O)Cn2nccc2C)CC1F c1(OC)ncc(Cl)cc1C(=O)NCCC1CCN(C(=O)C(C)(C)N(C)C)CC1 N1(C(c2scc(C)c2)=O)CCC2CCN(C(=O)CS(=O)(=O)NCC3CC3)C2C1 N1(C(c2c(C)nc(O)cc2)=O)CC(C)CN(C(C2CCCCCN2C)=O)CC1C C(=O)(CC(CC(=O)O)c1ccccc1)NC(c1ccc(F)cn1)(C)C c1(C(N2C(C)CC(NC(CCC(C)=O)=O)C2)=O)ccc(C)c(-c2cnn(C)c2)c1 N1(C(c2ccn(C)c2)=O)CC2CCOC2(CNC(C2CC2c2cccs2)=O)C1 N1(C(C(c2cn(C)nc2)N(C)C)=O)CCCC1C1CCCN1C(=O)NCCCl C1(F)(C(=O)NCC2CC(C(=O)NCC3(OCC)CCC3)C2)CCCCCC1 CCCC(C(=O)OC)C(=O)NCC(CC)NC(=O)C(c1cccc(Cl)c1F)(C)C Cc1cnc(C(=O)N(CC(N2CCN(C(C3(C)CCOC3)=O)CC2)=O)C)cn1 S(=O)(=O)(C1CCN(C(=O)NCC2CCC(C)SC2)C1)NC(=O)OC(C)(C)C N1(CCNC(CCC2CC(NC(C(C)OCOC)=O)C2)=O)CC2CC2C1 C1(CNC(c2cccc(Cl)c2F)=O)CN(C(=O)Cc2ccccn2)CCCO1 C(=O)(CCS(N)(=O)=O)NC1C(C(=O)NC(c2nc(C)sc2)C)COC1 C=CCC(CC=C)C(=O)N1CCCN(CCNC(C2CCCC(OC)C2)=O)CC1 C(CC(C)C)(C(=O)N1CCOCC(NC(=O)CCCc2cc[nH]n2)C1)OC C(=O)(C1=CCCN(C(=O)COC2CC=CC2)C1)N1C(CCC)CSCC1 C(=O)(CC(O)CC(C)(C)C)NCC1N(C(=O)Nc2c(C)cccc2)C2C(C1)C2 C1(C(N2CC(OC)(CNC(c3cccc(=O)o3)=O)C2)=O)CC(O)C12CCC2 C1(CC(NOCCCC#C)=O)C2CCCC2N1C(c1ccc(CC)s1)=O Fc1ccc(C2CN(CC=CCOc3ccccc3)CCO2)cc1 c1(C(N2CCC(CNC(C3CC3C3CCCO3)=O)C23CC3)=O)cnc2ccnn2c1 CC1(C(=O)NCC(C2CCCC2)NC(=O)COc2cccnc2)CC=CCC1 N1(C(c2nc(N(C)C)oc2)=O)CCC2CCCC12C(=O)NCC1(C)CC1(C)C N1(C(c2c(C)oc(C(C)C)c2)=O)CCN(C(=O)CN2C(C)CCC2C)C(CO)C1 N1(C(C(c2ccccc2F)C)=O)CCN(CCNC(C2(C(N)=O)CCC2)=O)CC1 C(C(C)C(F)(F)F)N(CCCC1(C)CN(C(C=CCC)=O)C1)C CCC(CC)C(C(=O)NC1CC(C)CN(C(c2ccccc2O)=O)C1)OC C(CCC(C)(C)NC(C1CCCCN1C(C)C)=O)NC(CCc1onc(C)n1)=O C#CC1(NC(C2(C(C)NC(C3CCN(OC)CC3)=O)CC2)=O)CCCOC1 Cc1cc(CCC(=O)NC2(CNC(C34CCC(CO3)C4)=O)CCOC2)c(C)s1 C1(c2n(CC(=C)C)nnn2)(NCC(c2ccccc2Br)C)CCCSCC1 C1(C(=O)NC(CCC)(C)CC)CN(C(C2CC2C(F)F)=O)C2(CCC2)C1 N1(C(C2CC3C=CC2O3)C(=O)NC2CCOC2)CCC2(CCC2)CC1 c1(CS(=O)(=O)NC(C2(C(F)(F)F)CC2)=O)cccc(Cl)c1 C1(NC(C(C)C)=O)CCCCC1NC(c1csc(-c2cnccn2)n1)=O c1(C(C(=O)N(CCc2ccccc2)CC2CCC2)O)ccccc1I Cc1ccnc(C)c1C(N1CCCC(CNC(c2nccnc2C(N)=O)=O)C1)=O Cc1occ(C(F)(F)F)c1C(N1CCCC(CCN)C1)=O N1(C(CNC(CCC)=O)=O)CCC(CNC(c2sccc2Cl)=O)CC1 C1(CC)C(CNC(C2(N(C)C)CC2)=O)CCN1C(=O)CCn1ccnn1 C(=O)(C1CCc2cccnc21)N(CCCNC(c1n[nH]c(C)c1Br)=O)C1CC1 CCC(C)(CNC(=O)CNC(=O)CO)NC(=O)CCCOC(C)=O n1(CC(=O)NCCC2CCN(C(C(C)(CO)OC)=O)C2)cnc([N+](=O)[O-])n1 C(=O)(CC1=CCCCC1)N(C1CCC(CNC(C2CC2Cl)=O)CC1)C c1(OCC)c(-c2nc(NC(=O)C(C)Sc3ncco3)cs2)c(C)nn1C C(=O)(C1=CCCC(C)(C)C1)NC(C(C)C)CCN(C(=O)C#CC1(C)COC1)C c1(CC2N(C(c3cn(CC4CC4)nn3)C(=O)NCC)CCCC2)ccc(C#N)cc1 C1(C)(C(=O)NCC(CC)(CC)NC(=O)Cc2ccccc2F)CC(C2CC2)=NO1 c1(C(=O)NCC(CC)NC(=O)C(c2ccccc2)O)nn(C)cc1[N+](=O)[O-] CC(C)(C)C(=O)NCC(=O)NCCNC(=O)CC1CSC1 O=C(C1=CS(=O)CCC1)NC1CCCC1CNC(c1ccnnc1Cl)=O C1(O)(CNC(c2ccc(COCC)o2)=O)CCN(C(C2CC2C(=O)OC)=O)CC1 c1(COCC)nc(C)c(C(N2CCC(C)(NC(c3ncsc3C)=O)C2)=O)s1 c1(CC)ccc(Cl)c(C(=O)NC2(C(=O)O)CC2C)c1 CC1CCC(Cl)=C(C(=O)NC2(CNC(c3nc(Cl)c(=O)[nH]c3N)=O)CC2)C1 CC1CCN(C(c2ncccc2C(F)(F)F)=O)CC1NC(=O)CCSCC(N)=O N1(c2cc(C)nc(N3CCCC(C(C)(F)F)C3)n2)CCCC2(CCCO2)C1 c1(CN(C2CCCN(C(c3c(CC)cccc3)=O)C2)C)ccncc1[N+](=O)[O-] C1(CCNC(C=CC=CC)=O)CN(C(=O)C=CC2(C)COC2)CC(C)O1 C1(NC(CCC=C)=O)CCCCC12CCCN(C(=O)C(C)n1ccnn1)C2 C=CCCCCCCC(=O)N1CC(NC(c2c(C)nc3sccn23)=O)CC(C)C1 C(Cc1ccccc1F)(CN=C(NC(C)C)N1CCc2cccc(C)c2C1)OC CC(CC(F)F)C(=O)N1CC=CC1CNC(=O)CCc1ccccn1 c1(OC)ccc(F)c(C(N2CCN(C(c3cc(Br)c(C)s3)=O)C(CO)C2)=O)c1 Cc1ncc(N)cc1C(N1CC=CC1CNC(=O)CCc1cnco1)=O N1(C(c2cc(CCCCC)no2)=O)CCN(C(=O)CCC2CCC2)C(COC)C1 N1(C(C2(Cl)C(C(C)=O)C2)=O)CC(C(=O)N(CCCCO)C2CCCC2)C2(CC2)C1 C1(OC)(OC)CC(C(=O)NCCN2CC(C)(CCCC(=O)O)C2)C1 N1(Cc2nc(=N)[nH][nH]2)CCC(O)(C(N2CCCC2Cc2ccccn2)=O)CC1 C(C(CO)(CO)NC(C1CNC(=O)N1)=O)N(C)C(c1cncc(-n2ccnc2)n1)=O CN1N=C(C(=O)N2CCOC(C(=O)NCCc3cccc(Cl)c3)C2)CCC1=O CCC(C)C(CC(=O)NCc1cnnc(C)c1C)NC(=O)CC1CC(OC)C1 c1(C(C)(C)C)n[nH]c(=NCC2CC(CNC(C34CC3COC4(C)C)=O)CO2)o1 C(=O)(C1COc2ccc(Cl)cc21)N1CCC(CCOC)(NC(=O)CN2CCC2)C1 N1(C(C2CC(C)=C(C)CC2)=O)CCC(C2CC2)(NC(c2cccc(F)c2Cl)=O)C1 c1(NC(COCC)=O)cccc(C(C2(C)CCNCC2)C)c1 C(CC(C)(C)C)(C(=O)NC(C1CCN(C(C2(C(F)F)CCC2)=O)C1)(C)C)OC c1(N(C)Cc2cn(CC)nc2)nc(=NCC2CC2(C)C)[nH]c2ccccc12 c1(OCC)ccc(OCC(N2CCC2C(=O)NC2CCC(SC)C2)=O)cc1 C1(C(C)C)CN(C(=O)CCCCN(C)C)CCN1C(c1c[nH]ccc1=O)=O CCC(O)C(C)(C)C(=O)NC1CCC1CNC(=O)CCc1cnco1 N1(C(C)=O)CC(C)(C(=O)NC2CN(Cc3cn[nH]c3)C2)C1 c1(OC)ccc2c(c1)CC(C(=O)NC1CC3(C1)CN(C(=O)C(C)OC)C3)O2 c1(C(=O)OCC)sc2ccccc2c1C(=O)OC(C1CC(OC)C1)CC c1(CN2C(CNC(C(C)(C)C)=O)CCC2)c(F)c(F)cc(F)c1F O=C(CCCCCn1cc(-c2cc[nH]n2)nn1)NCCC1=COCCO1 C1(C#CC(=O)N(C)CC2CCCN2C(=O)C(N2CCN(C)CC2)C)(CC)CC1 c1(C(=O)NCC2C3CN(C(C(C4CC4)OCC)=O)CC32)cc(Br)cc(F)c1C C(=O)(CCCCC(C)C)N(C1CN(C)NC1=O)CCC c1(N)ccc(CC(=O)N(C)C)cc1.c1(C(=O)NC2(C(=O)OCC)CC2)csc(Cl)n1 C1(NC(CN(C(C)C)C)=O)CCCC(NC(c2nnn(C)n2)=O)C1 C1(NC(=O)CCC(F)F)CC2(CCN(C(=O)C(O)CC(F)F)CC2)C1 CCCCCCN(C)CCNC(=O)C=C(C)CNC(C1(C)CC(C)C1)=O C(CC(C)(C)C(=O)N1CC(C)(NC(=O)CNC(=O)OCc2ccccc2)C1)SC C(=O)(C(O)C(C)c1ccccc1F)OCCOCCOCCOC CCC(CC(=O)N(C)C(c1ccc(C)cc1)C)C(C)(C)C CS(C)(=O)=Nc1cccc(C(=O)NC2CC3(C2)CN(C(=O)C(O)C(F)(F)F)C3)c1 C1(NC(c2c(C)scc2)=O)CC2CCC1N2C(C1CC(=O)N(C)C1)=O c1(C(N2C(C)CC(NC(Cn3c(C)ccn3)=O)C2)=O)c[nH]c(C#N)c1C c1(C(=O)NCCN(C(C2=CC(C)(CC)C2)=O)C)cc2cn[nH]c2cn1 C#CCCCCCCC(=O)N1CCC(N(C(c2conc2C(C)C)=O)CC)C1 Cc1cn(C)c2nc(N3CCC4(CCCC4=O)CC3)ncc12 c1(OC)ccc2nc(N3C4CCC3CC(O)(C(Cl)(Cl)Cl)C4)sc2n1 C1(C(=O)NC(CCCNC(C(C2CCCC2)OC)=O)C)CCCC(F)C1 N=c1[nH][nH]c(C(=O)NCSN2CC3CC3(C(N)=O)C2)c1Br Cc1cc(N(C)C)ccc1C(=O)NC1CCN(C(=O)CC2CCCC2)C1 C1(C(N2CC(CC(C(=O)N(CC(O)CO)CC)F)C2)=O)CN(C)CCN1C c1(OCC)ccc(F)cc1-c1cccc(CC(=O)OC(CC)CO)n1 c1(C(=O)NCC2N(C(C(C)NC(C)=O)=O)CCC2)cc2nccc(Cl)c2s1 C1(NC(C(CSC)C)=O)COCCC1C(=O)N(CC(F)F)CCO CCCC(C)C(C(=O)Nc1ccccc1Cl)N(C1CCC(OC)C1)C C1(C(=O)NC2C3CN(C(COC(C)C)=O)C2C3)CC2(CCC(F)(F)CC2)CO1 n1(CCC=C)c(N2CCN(C(C3(CC(=O)OCC)CC3)=O)CC2)nnc1CC c1(C(N2CCCN(C(C=CC)=O)CC2C)=O)cc(F)cc2nc(S)[nH]c12 c1(C(=O)NC2CC(N(C(=O)CCCN3CCCC3)C)C2)occc1F c1(C(=O)NCC(COCCCOCCOCCSCC)(C)C)ccc(C)c(Cl)c1Cl.CNC N1(C(c2n(C)ncc2)=O)CC2CS(=O)(=O)CC2(NC(=O)Cc2nc[nH]n2)C1 C(=O)(C1CCCc2c[nH]nc21)N1CC(C(C)NC(C2(CF)CC2(F)F)=O)C1 c1(C(C)=O)cccc(C(=O)N(C)CC2(O)CN(C(=O)C(C(C)C)NC(N)=O)C2)c1 N1(C(c2nc(C)c(C)s2)=O)CC(NC(=O)Cc2ccc(F)c(Cl)c2)CC(C)C1 C(N=c1[nH]c(C)cc(=NCC23CCCC2C3)[nH]1)C1(CC)CCCC1.C1(=O)N(C)O1 C#Cc1cn(C)nc1C(N1CCOC(CN(C(=O)COCC)C)C1)=O CON=CC(=O)N1CC(c2ocnc2C(=O)NC2(COC)CC2)C1.C1CC1 C(C)(C(=O)N(CC(O)CN(C)C(C1CC(CCO)C1)=O)C)NC(CC)=O c1(C(=O)NCCN(CC(C)O)C(C2C(C=C)C2)=O)cc2n(n1)CCC2 C1(C(=O)NCC(C)C(C)O)(SC)CN(C(=O)CCC2CCOC2)C1 n1(CC(=O)NCCCCC(C)NC(C2CC2F)=O)cnc2c1CCCC2 c1(C(N2CCCCC2CO)=O)ccc(OC(F)(F)F)cc1Cl c1(C(=O)NC2CCC(CNC(CC(C)CN(C)C)=O)C2)ccc(F)c(F)c1 c1(CC(N2C(CNC(=O)CCOC3CC3)CCCCC2)=O)nc2c([nH]1)CCCC2 N1(C(CS(=O)(=O)N(C)C)=O)CC2CCCC2(C(=O)NOCCC2CC2)C1 C(=O)(C(C)(C#N)CC)NCC1CC(NC(CC2ON=C(CC)C2)=O)C1 c1(C(=O)NCC(C)NC(C2(CCF)CCC2)=O)ccc(C(C)(F)F)nc1 C1(CN(C(=O)Cc2sccc2Cl)C)CN(C(=O)CNC(=O)C(C)(C)C)CCO1 N1(C(C2C(CC)CCO2)=O)CCC2(CCC2)C(NC(c2cc(SC)n(C)n2)=O)C1 N1(C(c2c(C)coc2)=O)CC(C)(C)CC1C(N1CCCC(F)C1)=O C1(CNC(CC(C)C)=O)CC2(CCN(c3ncccc3[N+](=O)[O-])CC2)CO1 C1(C)(C(=O)NC(c2cc(C(=O)OC)on2)=O)CCOCC1CO N1(C(C2CC(C)(O)C2)=O)CC2CCC1CC2NC(C1CC1c1ccccc1)=O N1(C(=O)COCC(F)(F)F)CC2(CCN(C(C3CCC4(CC4)C3)=O)CC2)C1 C1(NC(c2c(CC)onc2)=O)CCC12CCN(C(C1CC(F)C1)=O)CC2 C(=O)(C(C)(C)C(=O)NC1CCCN(C(=O)CCc2ccc(O)nc2)C1)N(C)C c1(NC(c2cc(C)nc(Cl)c2)=O)ccc2c(c1)CN(Cc1cnn(C3CC3)c1)C2 CC(C)(C#N)C(=O)NC(CNC(C1CC(=O)N(C(C)(C)C)C1)=O)C1CCC1 c1(C(F)F)cnc(-c2ccn(C3CCNCC3)n2)cn1 CC1CN(C(C2CC2[N+](=O)[O-])=O)CCN1C(=O)CC1CCCCC1 Cc1ccc(Cl)c(C(=O)NC2CC2NC(c2ccc(C(=O)N(C)C)nc2)=O)c1 N1(C(c2ccc(C)c(N)c2)=O)CCOCC(F)(CNC(=O)CN2CC=CC2)C1 CCC(CC)C(F)C(=O)N1CC(O)CC1CC(=O)NC1CCC(O)C1 c1(C2(C(=O)NCCCC(C)NC(=O)C(C)CO)CCCC2)ccccc1F c1(C(=O)NC2(c3nn[nH]n3)C(C)C2)cnc(O)[nH]1 N1(C(c2c(C)nc(C)s2)=O)CCC(NC(=O)C(C)(C)C2CCOC2)CC1C C12(C(=O)NC(CC=C)C(=O)Nc3cnc(F)nc3)CCCC1CCC2 C1(N(C)C(C2(CCF)CCC2)=O)CN(C(C2CC2[N+](=O)[O-])=O)CCC1O Cc1ccc(S(=O)(=O)N2CCCCC2)cc1NC(=O)CCCCCc1cccs1 C=CCC(CNC(c1cnnc(C)c1C)=O)C(=O)N1CCOCCC1C1CC1 c1(C(N2C(CNC(CN(CCC)C)=O)CC2)=O)csc(-c2cccs2)n1 c1(OC)cc(Cl)c(C)cc1C(=O)NC(CNC(c1occ2c1CCC2)=O)C(C)C c1(N)c(C)nn(CC(F)F)c1C.C12C=CC(C1)C2.C12CC1CC(=O)NC2=O.CSC c1(C(=O)NC2CCN(C(C(C)(C)CC3CC3)=O)C2)cccc2nc(C3CC3)[nH]c12 Cc1cc(C(N2CCC(NC(=O)COC(F)(F)F)CC=C(Cl)C2)=O)cc(N)c1Cl c1(C(=O)OC)ccc2c(c1)C(C(=O)N(CCCNC(c1cnc[nH]1)=O)C)CO2 C1(C(=O)OCCC2CC(C)OCC2)CC(C)(C)CCN1C(=O)OC(C)(C)C c1(C(C(=O)NCC(CNC(c2nnn(C(C)(C)C)n2)=O)F)O)ccc(F)cc1F C1(NC(C(CCC)N(C)C)=O)CC2C1CCN2C(=O)CC(=O)N(C)C C#CCC(C)(C)C(=O)NC(C)CNC(C1C=CCCC1)=O N1(C(C(CC)(C)CNC(c2nocc2Cl)=O)=O)CC2(CCCCC2)C1 Cc1cc(C(N)=O)ccc1C(N1CC(CNC(=O)C(CO)c2ccccc2)C1)=O C1(NC(C=C(C)C)=O)Cc2ccccc2C1NC(c1cnc2c(n1)CCCC2)=O C(C(F)(F)COC)(OC)Nc1cc(-n2nc(C)cc2C)ncn1 c1(C(C(=O)NCCCCCC)N(C)C2CC2)cc(F)c(F)c(F)c1 C(=O)(C1=CCCOC1)N1C(CCNC(CCOCC(C)C)=O)CCC1 N1(C(C2C(C)(C)OCCO2)=O)CCC2(CC1)CC2NC(=O)Cc1cc[nH]n1 CC(C)C(C(=O)NC1CCN(C(=O)C=Cc2cscn2)CC1)c1ccc(Cl)cc1 C1(C(=O)NCC(CNC(c2cnccc2C(F)F)=O)O)CCCC1C1CC1 N1(C(C2CN(C(CC3CC(=C)C3)=O)CC2(C)C)=O)CCCC2(CCCC2)C1 CC1(C)CCN(C(c2ccon2)=O)C(C(=O)NC2CCN3CCC2C3)C1 c1(SC)ccc(Cl)c(C(N2CC3CCC3(CNC(=O)CC3CCCN3C)C2)=O)c1 C1(CC(N2CCC(NC(c3cccc(N)n3)=O)C2C2CC2)=O)CN2CCC1CC2 C1(C(=O)NC2C(O)C3CCOC23)CN(C(C2(CCCF)CC2)=O)CC12CC2 N1(C(CC=CC)=O)CCN(C(c2nc(C)sc2Br)=O)CC1C c1(C(N(CC(C)NC(=O)C(O)C(F)F)CC)=O)cc(S(C)(=O)=O)cnc1O C1(CNC(CN(CC)CC)=O)C(C(=O)N(CCCO)C2CC2)C1(C)C C12(NC(CCC3CC(OC)C3)=O)COC(CNC(C3CCC(C)C3)=O)(C1)C2 c1(OC)ccc(NC(=O)C(=O)Nc2cccc(F)c2)c(C)n1 C1(CNC(C2C(C(C)C)C2)=O)CCN1C(=O)C(C)n1cncn1 c1(C(N2CCC3(C(C(=O)N=c4[nH][nH]cc4Br)C3)C2)=O)cccc2ccncc12 C(=O)(C#CC(=O)N(C(c1ccccc1)C(N)=O)C(C)=O)OC(C)(C)C(=O)OC C1(CN(C)C(c2cnc[nH]2)=O)CCCCN1C(C1(C)CCC1)=O Cc1cc2c(cc(C(=O)NCC(C)(C)CNC(C3(O)COC3)=O)n2CC2CC2)s1 C1(CC=C)(NC(C2CC(CC)C2)=O)CCN(c2nc(CC)ns2)CC1 C(C)(CNC(c1cc(Cl)cs1)=O)(CO)NC(CSCCCC)=O C(C)(N=c1[nH]cc(C#N)cc1C)C1N(C(=O)Nc2cccc(CSC)c2)CCCC1 c1(CNC(=NCCCCC)NCCNC(=O)OCC)nccc2ncccc12 c1(NC(CCNC(c2nc(CCC)sc2)=O)C)ccc([N+](=O)[O-])c(C)c1 c1(C(N2CCN(C(C=CCn3cccc(N)c3=O)=O)CC2)=O)cc(F)c(F)c(F)c1 C1(CC)CN(C(=O)Cc2ccccc2Cl)CCN1C(=O)CCNC(C)=O c1(C(=O)NCC(C)N(C(c2c(C)cc[nH]2)=O)C)c(C)nc2ccccn12 C1(CNC(c2coc3c2COC3)=O)CC2COCC2N1C(=O)Cn1cncn1 c1(CC)c(C(N2CCCC2C2CC(NC(=O)CN(C)C(N)=O)C2)=O)nnn1CC C(=O)(CC(C(F)F)c1ccccc1)NC1C2CN(C(C(CC)O)=O)C1C2 C1(C(=O)NCC2CCC(N(C)C(C3(C)CCCC3)=O)CC2)CCC2(CCC2)C1 C1(NC(c2ccc(C(C)C)nc2)=O)CCC2CN(C(=O)CNC(N)=O)CC2C1 C1(C(C)(C)C)OCCC1CNCC1(F)CCNC1 CC1CCN(C(=O)Cc2ccon2)CC1CNC(C1CCCCC1(F)F)=O N1(C(C(CCOC)(C)C)=O)CC(C)C(NC(=O)CC2COCCOC2)C(C)C1 N1(C(Cc2cc(C)nn2C)=O)CCCCC(C(=O)NCC(CO)C(C)C)C1 Cc1nn(CC(=O)N(CC(C)(C)CNC(C2SCCC2C)=O)C)c(C)c1C Cc1noc(C)c1C=CC(=O)NC(C)CCNC(=O)C(C)Cc1cnn(C)c1 Cn1cccc(C(=O)NCC(CC2CC2)C(=O)NCC2CCCC2(C)C)c1=O C12(C(N(C(C=C)C3CC3)C)=O)CCN(C(=O)CC3C(C)(C)C3(C)C)CCC1C2 n1(CC)nc(C(=O)NC(C)C(C)NC(c2coc(C(C)(C)C)n2)=O)cc1O c1(CN(CCCC)C(=O)NC(C)CSc2cccc(Br)n2)ccc(F)cc1 Cc1cc(C)c(CC(N2CCOC(C(C)NC(=O)C=CCO)C2)=O)s1 CC(C)(CC(F)F)C(=O)NC1CCC1C(N1CCc2sccc2C1)=O c1(C(N(CC2CCN(C(CCCCC#C)=O)C2)CC)=O)c(O)ccc(Cl)c1F CC1CC(NC(=O)C=CC2CCCO2)CCN1C(C1CC2CCC1C2)=O N1(C(C(C(C)(C)C)OC)=O)CCC2(C1)CN(C(=O)CCCCCC(C)C)CCO2 Cc1cncc(C)c1C(=O)NCCCCCC(=O)N1CCC(F)(CF)C1 N1(C(CCC(C)OC)=O)CC(NC(=O)CCCc2cccnc2)C2CCCCC12 CC(C)CC(C)OCCC(=O)NCCCC1CCCN1C(C1(CC2CC2)CC1)=O N1(Cc2ccc(C(=O)OC)s2)CCCCC1CN1CCNC(=O)C1 Cc1nn(C)c(C)c1C(=O)NC(C)(C)C(=O)N(C)CC1COCCO1 C1(C(=O)NCCCc2nc[nH]n2)CC(F)CN1C(=O)CCCC1CCCC1 c1(C(C(=O)NC(C(C)NC(C2(C(C)(F)F)CCC2)=O)CO)(F)F)ccccc1Cl C1(C(N(C2CCN(C(C(C)SCCCC)=O)CC2)C)=O)C2CCCCCCC12 CC(C)CC(O)C(=O)N1CCCC(CNC(=O)CC2OCCC2(C)C)CC1 C1(CC(C)NC(C2CC3(CC3)CO2)=O)CCN(C(C2CC3C=CC2O3)=O)CC1 Cc1cn2c(CC(=O)NCC(CO)NC(c3c[nH]cc(Cl)c3=O)=O)csc2n1 c1(OC)c(CN2CCCC2(C)c2ccc(C)o2)ccc(C)c1F N1(C(CN(C)C)=O)CCC(NC(C2CC2[N+](=O)[O-])=O)C(F)(F)CC1 c1(C(=O)NC(CC)CNC(C2CCOC2(C)C)=O)c(C)cc(C)cc1N C(=O)(CC(O)CNC(C1CCCCC1n1ccnc1)=O)N(c1ccc(N)cc1)C S(=O)(=O)(c1ccc(NCCC2CCC(C)C2)cc1Br)NC1CC(CC)(SC)C1 C1(C(N(C(C)C(C)(C)C)C)=O)CC2CC1CC2NC(=O)COCC(C)(C)C C(=O)(CCCC(=O)COC(c1cnn(-c2ccccc2F)c1N)=O)OC C1(NC(C2CC(F)(F)C2)=O)C=CCN(C(c2cn(C3CC3)cn2)=O)C1 C1(C(=O)NCC2(CC(=O)NC(C3CCOCC3)C#C)CC2)CC2CC1CC2=O N1(C(c2c(C3CC3)[nH]c(=N)s2)=O)CC2CC(NC(C3CCSCC3)=O)CC2C1 c1(C(N(CCNC(C2C3CCCC23)=O)C2CC2)=O)ccc(-c2ccco2)nn1 c1(CCN(C(=O)C=CC(=O)NC2(CCCS(C)(=O)=O)CC2)C)cccs1 C1(CNC(C2ON=C(C)C2)=O)CCC(C)(C)CN1C(=O)CCc1ccc(F)cc1 N12CC=CC1CC2=O.C1(NC(CN(CCC)C)=O)CCC(C(N)=O)C1 CC1(C)C2C1C(=O)N2.c1(C2(NC(=O)CCCn3cncn3)CC2)ccccc1 C1(NC(c2scc(OC)c2)=O)CC(NC(c2cccc(=O)n2C)=O)C12CCC2 c1(C(=O)OC)cnc(NC(=O)CC2CCCN2Cc2nc(C)ncc2Br)nc1Cl c1(CC(=O)N(CC(CC)NC(c2nc(C)ns2)=O)C)cccc(SC)c1 c1(CC(=O)NC(CNC(CSCCOC)=O)(C)CO)cccc(OC)c1F c1(C(N2CCC(CNC(c3c(C)ccn3C)=O)C2)=O)nc(C2CC2)ncc1Cl N1(C(C2(OC)CCSC2)=O)CCCC(NC(c2cc(C(C)(F)F)n[nH]2)=O)C1 N1(C(c2c(C)cc(F)s2)=O)CCC(NC(c2cc(C(C)(C)C)ccn2)=O)C12CC2 CC1CN(C(c2cc(O)nn2C)=O)CC(C(=O)NCC2(C)CSC2)O1 c1(C(C)=O)cc(C(=O)NCC23CC(NC(C4CCOC4C)=O)(C2)C3)c(C)o1 Cc1cnncc1C(=O)N(CC(=O)N(C)CC1(C#N)CC1)C c1(C(N2CCC(N(C(C3CCCC(O)C3)=O)CC)C2)=O)cc[nH]c2nccc1-2 CC1OCCC1C(=O)N(C1CCCC1)CCNC(C1(C)CC1)=O c1(C(=O)NCCC2N(C(c3n(C)nnc3)=O)CCC2)cc2ccc(F)cc2[nH]1 C1(C(N2CC(CC)N(C(C34CC(C)(C3)OC4C)=O)CC2)=O)CN=C2N=CNN2C1 C(=O)(CCCCCN(C(=O)C1CC1)C1CC1)N(C)Cc1c(C)n[nH]c1C c1(C(=O)NC2CC(C)N(C(=O)C=CCOc3ccccc3)C2)ccnn(C)c1=O C1(NC(C2CCCS2)=O)CN(C(C2CCCS(=O)(=O)C2)=O)C2(CCOC2)C1 c1(NC(C2(C)CN(C(C34CCC(OC)C3C4)=O)C2)=O)n[nH]c2ccc(F)cc12 C1(CNC(CC2N(C(CC3(N(C)C)CCC3)=O)CC2)=O)CCCC2(CC2)C1 CCC(C)(O)C(=O)NC1C2CN(C(c3ccc(C4CCC4)nc3)=O)CC12 c12ccc(cc1)C1CN(C1)C2.C(=O)(C(C)C(=O)O)OC.c12cn(nn1)CC21CCC1 C12(CNC(C=CC=CC)=O)CCC(CC1NC(c1cc(CC)ccn1)=O)C2 C(=O)(C(C)CC(C)C(C)=O)N1C(C(C)NC(c2cc(CCC)[nH]n2)=O)CCCC1 C1(C(N2CC(NC(=O)CO)C2)=O)CCCC(=O)N1C.Cc1cc(CNC)n(C)n1 C1(C(=O)NCC(C)N(C(CN(CCC#C)C)=O)C)(CF)CCOCC1 C1(CNC(c2ccoc2)C)CCN(C(=O)OC(C)(C)C)C2C1C2(F)F CC1(C#CC(=O)N2CCC(Nc3ncc([N+](=O)[O-])cn3)C(F)(F)CC2)CCCO1 S(=O)(=O)(CCCCCl)NC1CC(N(CC(=O)OCC)Cc2cccc(Cl)c2)C1 O=C1CC2(COC2)C(=O)N1CC(O)Cn1ccnc1 C(=O)(CC(O)CC(C)(C)C)NC(CCN(C(c1c(SC(C)C)cccc1)=O)C)C c1(NC(C2CC2NCc2ccc3n[nH]cc3c2)=O)ccc2c(Cl)ccnc2c1 Cc1nc2cncc(C(N3CCC4(C3)CN(C(=O)C(C)CC(F)(F)F)C4)=O)c2[nH]1 c1(OC)cc(C(=O)Nc2c(Cl)ccnc2Br)cnc1-c1cnc(F)cc1C CCCCCC(=O)N1CCN(C(c2ncc(-c3ccc(F)cc3)o2)C)CC1 N1(C(CCC)=O)CCC2(CCCN2C(c2c(C)csc2Cl)=O)C1 N1(C(c2cnnc(O)c2)=O)C2CCC1CC(NC(C1(F)CCOCC1)=O)C2 c1(C(=O)NC2CN(C(c3csc(Cl)c3)=O)CC2O)cccc2nc(O)ccc12 N1(CC(N2CCN(C(C3(C)C(C)C3)=O)CC2C2CC2)=O)CCCCCCC1=O c1(OC)ccc(S(N)(=O)=O)cc1NC(C1CC1C1CCNC1)=O C(=O)(C(O)C(C)(C)C)NCCCN(C)C(c1c[nH]cc1-c1cccc(Br)c1)=O c1(C(=O)NC2CC(CNC(=O)CCCF)CC2O)cc(Cl)cc(Cl)c1 CC1CN(C(=O)Cc2nc(=N)[nH][nH]2)CC(C)N(C(c2cc(O)ncn2)=O)C1 C1(CNC(C2(CC#C)CC2)=O)CC(OC)CN1C(=O)CC.c1ccncc1Br c1(OC)cc(C(=O)NCCCN(C)C(c2cnc(S)nc2)=O)sc1Cl N1(C(C(CC(C)(C)C)OC)=O)CCCC12CCCN(C(=O)C=C(C)C(C)(C)C)C2 C1(C(N(c2cnn(C)c2)CC)=O)CN(C(C2CN3CCC2CC3)=O)C(C)(C)C1 c1(CC)cc(Cl)ccc1NC(=O)C(O)C1CN(C(C2(CF)CC2)=O)C1 C1(CNC(c2n(CC)cnn2)=O)CC2(CCN(C(C3CCS(=O)(=O)C3)=O)C2)CO1 c1(COC(c2c(C)nc(-c3ccccc3Cl)s2)=O)cccc2c[nH]nc12 N1(C(C(C)=C(C)C)=O)CCN(C(=O)CCc2ccoc2)CC1CO C1(C(N2CC(C(C)NC(=O)Cc3n[nH]cc3Br)C2)=O)CCCCN1N=O c1(COC)nn(C)cc1C(N1CCC(N(C)C(c2cc(C(N)=O)cs2)=O)C1)=O C(=O)(C(C1=CCCCC1)N1CCCC(Nc2ccccc2F)C1)NC(C(=C)C)=O C12(NC(C(C)c3cccs3)=O)CCCC1N(C(=O)CC1CCC(C(F)(F)F)O1)CC2 CC1CCC(C(=O)NCCCS(N)(=O)=O)N1C(=O)C=Cc1cocn1 c1(C(N(C2CC(NC(=O)CCN3CCCC3)C2)C)=O)cc(F)c(Cl)cc1Cl N1(C(C(CC)OCC)=O)C2CCC1C(C)C(NC(=O)Cc1cnccn1)C2 Cn1cc(Cl)cc1C(=O)N(CCC(=O)NCC(=O)NCCO)CC1CC1 c1(OC(C(=O)N(C2(C)CC2)C)(C)C)ccc(Br)cc1.C12CCCN(C1)C2=O C1(NC(Cc2c(C)n(C)cn2)=O)CN(C(c2ncoc2C(C)C)=O)CC1N=[N+]=[N-] Cc1cc(C(=O)NC2C3CC2N(C(c2ccnc(O)c2)=O)C3C)ncc1F c1(C(C)C)ncc(C(=O)N(CCC(C)NC(=O)CC(=O)NC2CC2)C)s1 Cn1nncc1C(=O)NCCC=C1CN(C(=O)CNC(C2CCC2)=O)C1 C1(CNC(c2ccc(OC)s2)=O)CC2CC2N1C(=O)Cc1ccccc1Br CC(C)(C)CCCONC(=O)CN(C)CC=Cc1ccccc1 c1(C(=O)NC(C)CNC(=O)C=CC(c2cnn(C)c2)=O)cncc2c(F)cccc12 Cc1sc(C)c(C(=O)NCC2CC(O)CN2C(C2CCCN2C)=O)c1C#N c1(C(N2CC(CCCC=C)N(C(=O)C=C(C)Cl)CC2)=O)cccc2scnc12.C(C)(=O)O C=C(CNC(C1CC1(F)F)=O)CCNC(c1nocc1C)=O S(=O)(=O)(c1ccc(NC2CCC(O)CC2)c(Br)c1)N(CC)Cc1ccnn1C c1(C(N(CCOCCNC(c2c(NC)cnnc2)=O)C)=O)cccc(CC)c1F C(=O)(C1=CC(O)C(Nc2cc(C)ccc2F)CCC1)OCC C1(CC)(NC(c2csc(C(C)OC)n2)=O)CCN(C(c2cscc2C)=O)CC1 O=C1CC(C(N2CCC(OCC(N3CCC(CF)C3)=O)C2)=O)CC(=O)N1 c1(C(C(=O)NC(CC)C)N(C)Cc2ccc(F)cc2)cccc(OCCCC)c1 c1(NCCC)nc(N(C)CC2CC2(F)F)nc2c1ncn2C c1(C(=O)NCCC2N(C(C(C)SC(F)(F)F)=O)CCC2)cc(N)c(F)c(F)c1Cl C1(c2cn(C3CN(CC(C)Oc4c(C)cncc4)C3)nn2)(CO)COCCN1C Cc1nn(C)c(C(N2CCN(C(c3nnsc3C)=O)C(C3CC3)C2)=O)c1Cl C1(C(N2CCN(C)CC2)C)CCC2(CCC2)O1.C12CCN(C1)CC(=O)N2 N1(C(C2(C(=O)OC)CC2)=O)CCC2CN(C(c3cnc(Cl)cc3C)=O)CC2C1 n1(CC(=O)NC(C(=O)N(C(C(C)SC)C)C)Cc2cn[nH]c2)cnc(C#N)n1 C1(CC(=O)NCC2C(NC(C(C)(C)OC)=O)CC2)CCCC(C2CC2)O1 c1(OC)cc(Cl)c(C(=O)NC(C)CCN(C)C(C2(OC)CCC2)=O)cc1Cl C1(NC(C2(CCC=C)CC2)=O)CCCC12CN(C(c1cscc1Cl)=O)C2 C1(C(=O)NC(C)CCN(C(=O)CCc2cnn(C)c2)C)COC2(CCC2)C1 C1(C)(COC)CC(NC(=O)CC2CC3(CC3)C2)CN1C(=O)Cn1cnnc1 C(CCN=c1[nH]nc(O)s1)NC(c1c(C)cno1)=O C(=O)(C(F)C(F)(F)F)N1CC(SCCNC(c2n(C(C)C)ccn2)=O)C(C)C1 c1(C(=O)NCCn2cc(I)c(C(F)(F)F)n2)ccc(C(=O)O)c(F)c1 C1(C(=O)NCCCC2OCCN(C(c3cc(C)oc3)=O)C2)OCC2CCCCC12 C1(C(=O)NC(c2ccc(C)cc2)CNC(C(CCC)F)=O)CC(=O)NC1(C)C N1C(NCC(C)C)=NCCNC(=O)C2(CC2)CC1.c1(COC)cccc(Cl)c1 C1(C(=O)NCC(CC=C)NC(=O)CN(C)C)CN(C)C(=O)CCO1 C(=O)(CC(C)P(C)(C)=O)NC1C(C)CN(C(C2(C(C)(C)O)CC2)=O)C1 c1(C(C(=O)NCC2(F)CN(C(C3(CC)CCCO3)=O)C2)O)ccc(Br)cc1 C1(C(=O)O)CCN(Cc2cn(Cc3ccc(-n4cc(Br)cn4)cc3)nn2)C2(CC2)C1 c1(C(N2CC=CC(NC(C(C)CC3CCCCC3)=O)C2)=O)nc(Cl)cc(N)c1Cl C1(C(N(CCCOC)CCO)=O)COCC1NC(=O)CCC1(C#N)CCC1 c1(C(=O)NCC2CC(NS(CCCC)(=O)=O)C2)cnc2ccoc2c1 c1(C(=O)NC2(c3cn(C)nn3)CCNC2)cc(F)c(F)cc1NC(N)=O N1(C(c2c(C)n(CC(C)C)nc2)=O)CCN(C(=O)CCC2CC2)CC1CO C(=O)(CP(=O)(C(C)C)C(C)C)N(CCC(C(C)C)NC(C1C(CCOC)C1)=O)C C(CC(C)(C)C)(C(=O)NCCCC(O)C(=O)NC)NC(c1cnn(C=C)c1N)=O c1(C(N(C)CC2CCCCN2C(=O)CCCc2ccsc2)=O)cc(Cl)nnc1Cl c1(CCNC(C2SCCS2)=O)cc(F)ccc1Br c1(C(=O)Nc2cnoc2CNC(CN(CCC)C)=O)csc(C(C)OC)n1 CC(C)(CNC(=O)CONC(C1CC2(C1)CC(O)C2)=O)C1=CCCC1 c1(Cc2ccccc2)cn(C2CCCc3cncn32)nn1 c1(C(=O)NCC(C)NC(CCc2c(OCC)cccc2)=O)ccc(C)n(C)c1=O C(=O)(C(C)(C)C(C)C)N(C(C)CN(C)C)Cc1ccc(OC)cc1.C1C(O)CN1 C(CCN=c1[nH]c(=N)[nH]c(=NCC23COCCN2C(=O)OC3)[nH]1)OCC c1(C(N2CCC(C(N(C)Cc3c(C)n[nH]c3)=O)(CF)C2)=O)ncn2c1CCC2 Cc1ccc(F)c(CC(=O)NCC(C)NC(c2ccc(OCCO)cc2)=O)c1 CC1(CNC(C2C3CN(C(C4C(C)(C)C4(C)C)=O)CC23)=O)CCOCC1 C1(C(=O)NCC(C2CCCC2)OC)CN(C(=O)CSC2CC2)CCC1(C)C N1(C(C2(CCCC)CCC2)=O)CCOCC(C(=O)N(C(C)COC)CC)C1 C1(N(C(C(C)=NOCC#N)=O)C)CCCCN(C(=O)C=CC2CCCCCC2)C1 c1(C(N(C2CCC(NC(CN(c3cnccn3)C)=O)C2)C)=O)cncc(O)c1 C1(C(N(CC(=O)OC)C)=O)(CC)CCCN(C(C2(OC)CCOC2)=O)C1 CC1CCC(C(=O)NC2C(=O)OCC2(C)C)CN1C(c1cccnc1O)=O N1(C(C(CC)CC)=O)CCN(C)CC1CNC(=O)C(c1ccc(Cl)cc1)CO C1(C(=O)Nc2c(CC)noc2)CC(NC(=O)C(C#N)CC)CCO1 c1(C(N2CCC(NC(C3CC(=O)N3)=O)C2)=O)cc2cc(F)ccc2s1 CN1CC(C)(C(=O)NC2CCCCC2C(N2CCN(C(=O)CO)CC2)=O)CC1=O N1(C(c2cc(NC(C)=O)ncc2)=O)CCN(CCc2ccccc2F)CC1C c1(N(C2CC3CC2CN3)C(c2scc(CC)n2)=O)cc(F)c(F)cc1Br C1(CNC(c2cn(CCC)nn2)=O)CN(C(=O)C(C(C)C)OCC)CCC1(F)F c1(SC(C2(C)CC2(F)Cl)=O)ccc(Cc2cn(CCN3CCSCC3)nn2)cc1 Cc1ncccc1C(=O)NCCOCCN(C(=O)C(C)N(C(C)C)C(C)C)C N1(C(c2ccc(N)nc2)=O)CCCC(O)(CNc2csnn2)CC1.CC(C)(C)O Cc1cc(CC(N2CCC(NC(c3sncc3C)=O)CC2C2CC2)=O)cc(F)c1 N1(C(CC2(OC)CCC2)=O)CCC(CCCNC(=O)Cn2cc(C)cn2)CC1 c1(C(N(C)CC2CCCN(C(C(C)C)=O)C2)=O)c2c(cc3c1CCC3)CCC2 C1(C(=O)NCCCN(C(c2ncsc2Br)=O)CC)CC2CCC1O2 N1(C(C(C=CC)O)=O)CCC(NC(=O)Cn2nc(C)nc2C)C(CO)CC1 C=C(C)CC(C(=O)Nc1cnn(COC)c1C)NC(C1CCCN1C1CC1)=O C(=O)(C1=CC(C)(CC)C1)NCC1N(C(CC)=O)CCCC1 c1(NCc2ccnc(C)n2)[nH]c(=NCCCCn2cnnc2)nc2ncn(C)c12 c1(C(=O)NC2CCN(C(C(N3CCOCC3)C)=O)C2)ccc(N(C)C)cc1 C=CC(C)(O)CC(=O)NCC1CC(C)CCN1C(=O)Cc1sccc1C C1(CC(=O)N(C(C)CCNC(c2cnn[nH]2)=O)C)(CO)CCCCC1 c1(CC(=O)N(C(CNC(c2c(CC)nccc2)=O)C)C)cnn2c1CCCC2 c1(C(N2CC(C)N(C(=O)Cc3cc[nH]c(=N)c3)CC2)=O)ccc2nnnn2c1 Cc1ccccc1C1=NOC(C(N2CC=CC2CNC(C2CCC2)=O)=O)C1 N1(C(c2nc(N(C)C)oc2)=O)CCN(C(c2csnn2)=O)C(c2cn[nH]c2)C1 c1(NCc2snc(OC)c2Br)cnc(N2CCC(CO)C2)nc1C N1(C(CCOC(C)C)=O)CCC(CCNC(c2ccc(=N)[nH]n2)=O)CC1 Cc1cc(C(=O)NCCC(C)N(C)C(c2ncn(C(C)(C)C)n2)=O)n(C)n1 Cc1cccc(-c2cn(C(C)C(=O)NC(c3ccccn3)CF)nn2)c1 C(=O)(C1=CCCC1)N(C1CCN(C(C2CNC(=O)N2)=O)C1)CC N1(C(CC(CC)C)=O)CCC2(CCCN2C(c2ccc(F)c(N)c2)=O)CC1 c1(C2(C#N)CC2)cccc(-c2cnc(CNCC(c3ccc(Cl)cc3)O)nc2)c1 N1(C(c2c(CC)n(CC)nc2)=O)CC(CNC(C2(C)CCCC2)=O)CC12CCC2 c1(C(N2CC3C(NC(c4ccnc(OC)n4)=O)C3C2)=O)nccc(Cl)c1O C(CNC(=O)C(c1cnn(C)c1)O)(CCCC)NC(COCCC=C)=O c1(C(=O)NC2CC(C(N3CCC(c4ccccc4)C3)=O)C2)ccc(O)c(O)c1 C1(CC(=O)NCCCCCN(C)C(c2cn(C3CC3)nn2)=O)CCCCC1(F)F C(CC)(CC(C)O)NC(C(Cn1cccn1)NC(C(CC)OCC)=O)=O C1(NC(CCCCC=CC)=O)CN(C(=O)Cc2cc(COC)on2)CC(C)(C)C1 c1(C(c2n(CC(=C)C)nnn2)NC(C)CSCOC(C)(C)C)ccc2occc2c1 c1(NC(=O)CC2CC3COCC23)cccc2cccnc12 C1(NC(C(C)=C2CCCC2)=O)CN(C(=O)CC2CCN(CC(C)C)C2)CC1C c1(C(N(CCNC(C2(OCC)CCOC2)=O)C2CC2)=O)nc(C)sc1C N1(C(COC(C)C)=O)CCCC(C(C)(C)C(=O)NC2(CCF)CCC2)C1 c1(CC(=O)NC2CN(C(C3C(CCC)C3)=O)CC2O)cc(Cl)ccc1OCC N1(C(C2C=CCC2)=O)CC23CCCCC2(C1)CN(C(C1(C(F)F)CCCO1)=O)C3 C(=O)(C(CN(C)C)N(C)C)NCCN(C(=O)C(F)C1CCCC1)CC CCC(C)(C(=O)NCCCN(CCO)C(C1CCC(C)(C)C1)=O)C(N)=O c1(SC)ccc(C=CC(=O)NCC(F)CNC(C2(C)C(C)(C)C2(C)C)=O)cc1 c1(CC(=O)N(CCNC(C2N(CC)CCC2)=O)C2CC2)ccc(OC)cc1Cl c1(NC)cc(Cl)ccc1C(=O)NC1CC(CNC(=O)CC2CCCC2O)C1 c1(C(N2CC(C)(NC(C3CN(C4CCC4)C3)=O)C2)=O)cc(Cl)c(F)cc1Cl CC1(C)CC(C)(CNC(=O)C2=CCCCO2)CN1C(c1ccc(C(N)=O)cn1)=O N1(C(=O)Cc2cc(Cl)ccc2O)CCCC2(C1)CN(C(=O)CC1CCC1)C2 Cc1[nH]c2ncccc2c1C(=O)NC(CO)C(C)NC(C1CC(F)C(=O)N1)=O C1(CC(=O)N(CCCN(CC)CC)C)CC(C(=O)Nc2cnc(C)s2)C1(C)C N#Cc1nnc2ccccc2c1N1CCC(C(=O)NCc2cc(=O)cc[nH]2)C1 Cc1nc(C(N2CC=C(CNC(=O)CCS(C)=O)CC2)=O)ccc1Br Cc1ccnc(C(C)(C)C(=O)NCC2CCC(NC(c3cn(C)c(O)n3)=O)C2)c1 C=CCCC(C(=O)NCCc1noc(CC)n1)NC(C1CC1C1(C)COC1)=O c1(NC(N)=O)coc(C(C)(C)NC(C(C)NC(=O)OC(C)(C)C)=O)n1.COCO c1(C(N2CCC(CCNC(C(C)SCCCC)=O)C2)=O)ccc(Cl)c(OC)c1F N1(C(c2cc(C)cc(O)c2)=O)CC(C)(C)OCC1CNC(=O)CCC1CCOC1 c1(N2CCCC(OC)CC2)nc2cc[nH]c2c(=NC(C)Cn2nccc2C)[nH]1 n1(CC)nc(C)c(C(=O)NCC2(NC(C3CCC(C)S3)=O)CCOCC2)c1C Cc1nc2ccc(C(N3CC4(CCCCN4C(=O)C4=CCCC4)C3)=O)cc2s1 c1(CC)cc(C(N2CC3C(NC(C4C(C(=O)OCC)C4C)=O)C3C2)=O)ccn1 c1(C(N2C(CNC(COCCCC)=O)C(C)(C)CC2)=O)ccc([N+](=O)[O-])cn1 N12CC3CC1(C3)NC(=O)C1CCCC(C1)NC(=O)C1(CC1)CC2=O.CCOC.N(C)C N1(C(C(=O)NC(C)C)=O)CCCC(C2(NC(c3cccc(O)c3Cl)=O)CC2)C1 C1(C(=O)NC2CC(C)CN(C(c3csc(O)n3)=O)C2)CC2COCC(C1)C2 N1(C(CCN(C)CC)=O)CCCCC1C1CCN(C(=O)CCC2CCC2)C1 C1(C(=O)NCc2cn(C(C)C)nc2)CC=CC(NC(C2(C#N)CC2(C)C)=O)C1 C(C1CCCC1)=CC(=O)NC1(CC(=O)NCCC2CC=CCC2)CCC1 C(=O)(CCC(=O)N1CCC(CCCNC(c2cn(CCO)nn2)=O)C1)OC CC(C(=O)N(CCCCC(=O)N(C1CCCC(O)C1)C)C)S(C)(=O)=O C(=O)(C1CCCc2ccnn21)N1CC(CNC(=O)CC2CCCO2)OCCC1 C1(c2cn(CC3CCC(C(N(C4CCC4C#N)C)=O)C3)nn2)Cc2nccn2C1 C1(C(=O)NC2C3CC2N(C(c2cccc(OC(F)F)c2)=O)C3)CC2CC1C1CC21 C(=O)(C1CCc2cccc(=O)n21)N1CCC(C)(NC(C2CCCC2(F)F)=O)CC1 C1(CNC(Cn2c(C)ccn2)=O)CC(C)CCN1C(=O)C(C)Cn1cccn1 c1(OC(C)C2(C(F)(F)F)N=N2)ccc(Cl)cc1CC1CC2CCC1O2 c1(OC)ncc(C(N2CCCC2C(C)(C)CNC(=O)COC)=O)cc1C(=O)OC C1(CNC(c2c(CC)scc2)=O)CCN(C(c2cccc(C)n2)=O)CC1(F)F C1(C(C)(C)O)CN(C(C23CCCC2C3)=O)C1.C1(C(=O)NC)(CCO)CC1 c1(NC(C2(C)CCN(C(CCc3cccc(C)n3)=O)C2)=O)cc(Cl)ccc1I n1(CC(N2CCC(N(C(C3CCC(N(C)C)CC3)=O)C)C2)=O)cccc(N)c1=O C(CC(C)C)(C(=O)NCC(C(C)C)NC(c1cc(Cl)ccc1O)=O)OC C1(C(N(CCN(C(C#CC(C)C)=O)C)C)=O)C2Cc3ccc(Cl)cc3C12 CC1(C)CCCN(C(=O)CCCn2cncn2)C1CNC(C1CCCOC1)=O C(C(CC1CC1)C(=O)N1CCC(C(=O)NC)CC1)NC(C1C(=C)C1)=O n1(CC#C)cnnc1C(=O)NCC1(CC(=O)NC2CNC(=O)C2)CC1 N1(C(C(CC)CC)=O)CCC(C(=O)NC2CC(C)(CO)C2)C(O)C1 N1(C(c2ccc(CC)cc2F)=O)CC2COCC(C1)C2NC(=O)CCN(C)CC N1(C(C(C(C)C)NS(C)(=O)=O)=O)CCN(C)CC1CNC(=O)CNS(C)(=O)=O C(CCCC(=O)N(C1CCCC12CC2)C(C)C)NC(CC1ON=C(C)C1)=O C(C(=O)NC1CCN(C(c2ccc(C)c(Br)c2)=O)C1C)(C(C)(C)C)OC C(=O)(C1CCCc2scnc21)NC1CC(F)(CNC(CCCC(CC)C)=O)C1 C1(C(N2CCC(N(C(=O)CNC=O)CC)C2)=O)CCC(F)(F)CC1(C)C C(=O)(C(CC)CCCC)N(CC(C)O)CCNC(c1ccc(C#C)cc1)=O C1(NC(c2sccc2Cl)=O)COC2(CCN(C(=O)C(c3ccc(F)cc3)F)C2)C1 C1(CCNC(CN(C(CC=CC)=O)CC(C)C)=O)CCCCC1O N#Cc1ccc(C(=O)NCC2CCCC2C(=O)NCC2(CCO)CC2)s1 N1(C(c2cccc(N)c2N)=O)CCCC(C2CC2NC(C2CCC(=O)N2)=O)C1 N(C1CCc2ccccc21)(C(CCC=C)C(=O)OC(C)(C)C)C(=O)NCCCC C#CCCCCCC(=O)NCCC(O)CNC(C12CCC(CF)(C1)OC2)=O C12(CNC(CCCCSC)=O)CCCCC1N(C(=O)CCCCCOC(C)C)CC2 C1(NC(Cn2ncc(C)cc2=O)=O)CCCC12CN(C(c1n[nH]c(C)c1O)=O)C2 C1(C)(NC(CC)=O)CCCN(C(c2csc(CN3CCCC3=O)n2)=O)C1 N1(C(CN(CC)CC)=O)CCC(CN(C)C(c2cnc(C(C)C)o2)=O)CC1 C12(C(=O)NC(CN(C(=O)CC3(COC)CC3)CC)C)CC1COC2(C)C C=CC(CC)CC(=O)N1CC2C(CNC(c3nn(C)cc3C)=O)C2C1 N1(C(C(C(C)C)(C)O)=O)CCS(=O)(=O)C(CCNC(=O)C2=CCC(C)CC2)C1 C1(C(N(CCCCCCC)C)=O)CC2CCC1N2C(=O)C(C)CCN(C)C c1(C(N)=O)ccccc1C(N1C(CNC(C2CCCS2(=O)=O)=O)CC2CC12)=O C1(C(N2CC(NS(CC(=O)OCC)(=O)=O)(CF)C2)=O)CCCC12CCC2 C(C(=O)NCCCS(C)=O)(C(C)(C)C)NC(CC(C)c1ccco1)=O N1(C(C(C)C2CC2)=O)CCC(O)(CN(C(=O)Cn2ccc(Br)n2)C)C1 c1(C(N2CCC(O)(CNC(CN(C)C)=O)C2)=O)c(F)cc(Br)cc1F c1(CC(=O)NC(C)(CNC(C2(C(F)(F)F)CCC2)=O)C2CCC2)cccnc1Cl N1(C(COC2(C)CCC2)=O)CC(CC(=O)NC2CCCCCC2F)CC1(C)C C(C(C)(C)C#CC(=O)NC1CC12CCOCC2)NC(CS(CC)(=O)=O)=O N1(C(C(C)N(C(C)=O)C2CC2)=O)CCC2(CC1)COC(C)C2 c1(CC)nc(C)c(C(=O)N(C2CCCCC2N(C)C(C2CCC(C)(C)C2)=O)C)o1 Cc1c(C(=O)NC(C)(CNC(=O)C(C)Sc2ccccc2)CO)cccc1Cl c1(C(=O)NC(CC(=O)NCc2ncon2)Cc2cccs2)ccnc(Cl)c1Cl C(=O)(C(C)C(F)(F)F)NC1CCCC1.c1(SCC)cc(C)c(C(N2CCCC2)=O)o1 FC(F)CCN=C(NCc1ccccc1)NC1CCCC(F)C1 N1(C(C2CC(C)C2)=O)C(C(=O)NC2CCSCC2)C2CCCC12 C1(CNC(COC2(C)CCCC2)=O)C2CCC(C2)N1C(C1CC2CC1CC2O)=O C1(C#N)(C(N(CCCCNC(=O)CSCCC#N)C)=O)CCCOC1 c1(SC)ccc(Cl)c(C(=O)N(C(C)CCNC(C2(c3ccncc3)CC2)=O)C)c1 c1(C(C)C(N2CCCC(C(N3CC(O)CC3(C)C)=O)C2)=O)ccc2c(c1)CCN2 C1(CNC(=O)NCC(n2cc([N+](=O)[O-])cn2)(C)C)CCC(F)(F)C(=O)N1 C(=O)(C1=CCCC1(C)C)NC1CCCN(C(c2c(N)cn(C)n2)=O)CC1 c1(C(N(C2CCN(C(C(C)N(C)C)=O)C2)C)=O)cc2ccnn2cn1 N1(C(C(N2CCC(C)C2)=O)=O)CC(OC(C)CC2CC2)CCC1=O Cc1cc(CNC(c2cc(F)c[nH]2)=O)oc1C(=O)NCC1CC1(F)F NC1CCc2cc(NCc3ccn(C4CC4)n3)ccc2C1 CCC(CC(C)C)C(=O)NC1COCC1CNC(=O)CCc1nnc(C2CC2)o1 C1(C2CCN(C(C3CNC(=O)CC3(C)C)=O)C2)(NC(c2c(CC)nco2)=O)CC1 c1(CC)cccc(C)c1NCc1ccc(N2CCC(C)CC2)c(F)c1 Cc1cc(C(N2CCCC2C=CC(N2CC(O)(CCO)C2)=O)=O)cc(F)c1 C1(C)(C(=O)NC2CCN(C(c3cnc(C(C)=O)s3)=O)C2C)CCCCNC1=O C(=O)(CC(C)C(C)(C)C)NCCCCCNC(c1ccn(C(C)C)n1)=O CC1(C)CCC(NC(=O)CSC2CC2)C(CNC(=O)CCCS(C)(=O)=O)C1 c1(NCc2n(CCC)ccn2)cc(N(C)Cc2cnn(C)c2Br)nc(C)n1 c1(C(N2CC(CCCNC(C3N(CC)CC3)=O)OCC2)=O)cc([N+](=O)[O-])cn1C C#CC1CN(C(C2CC(N(C)C)C2)=O)CCN1C(c1n[nH]cc1C)=O C(=O)(C1=CC2CCC(C1)C2)NC(=O)CC(C(F)F)n1cccn1 c1(C(=O)NCC2N(C(CC(COC)C)=O)CCC2)cc(F)ccc1O c1(C(=O)NCC2CCC(NC(c3ccc(Cl)nn3)=O)CC2)ccc2sncc2c1 Cc1ccc2c(c1)CCN2C(=O)CC1(C)CCN1C(=O)NC1CC(O)C1 c1(C(N(C)CC2(NC(c3ccnn3C(C)(C)C)=O)CCC2)=O)cc(O)nn1C c1(CC(=O)OC)cc(C)nc(NCCCCCNC(=O)CCn2cc(C)cn2)n1 CC1C(C(=O)Nc2ccc(C(=O)Nc3n[nH]c(C4CCCC4)n3)s2)CCN1C c1(C(N2CC(C(NOCC(=O)OC)=O)OCC2)=O)ccc(C)c(OC)c1 N1(C(COCC)=O)CCCC2(NC(C3COCCC3(F)F)=O)CCCC12 C1(COC)CC(O)CN1C(C1COCCN1C(=O)Cn1nc(C)oc1=O)=O c1(C(N2C(C(=O)NC3CC3)CCC2)=O)cncc2c1CCC2.C12CCCC1N2 Cc1cc(C(=O)NC(C)CC(C)NC(=O)CCc2cnc[nH]2)cc(C)c1O Cn1ncc(C(=O)NC2CC(F)(CNC(=O)CCOC3COC3)C2)c1C1CC1 N12CC(CC1(C)C)SCC2=O.C(=O)C(CC)CC.N12CCC(C1)C2=O.CCCN C1(C)(CC)CC(NC(=O)C(C)(C)NC(=O)Cc2cnc(C)s2)C1 C1(C(=O)NCCN(C)C(C2CNC(=O)C2)=O)CC(C2CC2)C1 C=CC1(C(N2CCCC(NC(=O)Cc3nccs3)CC2)=O)CCOCC1 C12(C(=O)OC)CCC(CN(C(CSCC(=O)OC)=O)CCSC)(CC1)C2 Cc1cc(=NCC(C(F)(F)F)N(C)C)[nH]cc1S(=O)(=O)N1CCCCC(C)C1 c1(NC(CC(CC=C)CC)=O)ccc2cc(C(=O)O)ccc2c1 c1(OC)cc(Br)cc(CN2CCNCC2C(=O)Nc2nc(C)cs2)c1O c1(CC#N)cccc(C(N2CC(C3CN(C(=O)Cn4nccn4)CCO3)C2)=O)c1 c1(NC(C)=O)ccc(C(N2CCCC(NCc3ccc(C)nc3)C2)=O)c(Cl)c1 c1(C(=O)NC(C(C)NC(CC(CCC)O)=O)(C)C)ccc([N+](=O)[O-])cc1Br CC1(NCCC2(I)CC2)CC1(c1nnnn1C1CCCCC1)OC N1(C2C(=O)NC3C2C3)CC(C(F)(F)F)C(C)(C)C1.c1(C(=O)NC)ccccc1Cl N1(C(CC(CC)C)=O)CCN(C(=O)Cc2ccc(F)cc2C)C(c2cn[nH]c2)C1 N1(S(CCCCC)(=O)=O)CCC2(CCC2)CC1C(=O)OC C1(O)(C(=O)NCCC(C)NC(C(CC=C)CC)=O)CN2CCC1CC2 Cc1ccc(CC(=O)NC(CNC(=O)C(C)SC(C)C)CO)cc1C N1(C(N(C)CC2CCSC2)=O)CCn2ncc(CNC(=O)CSC)c2C1 C1(N(C(CCc2ncc(C)[nH]2)=O)CCO)CCN(C(=O)C(O)c2ccco2)CC1 Cc1nc(CC(N2CCCCC2CCN(C(=O)C=CC(C)(C)C)C)=O)[nH]c1C c1(CNC(C(N2CC(C)CC(CCC(=O)OC)C2)=O)=O)coc2ccc(C)cc12 c1(Nc2c(C(C)=O)cccn2)ccc(Sc2ccncc2)c(F)c1 C(=O)(C(F)(F)C(O)CC)N(CC1CCN(C(C2(C(CC)(F)F)CC2)=O)C1)CC C=CCC(CNC(c1cnnc(C)c1C)=O)C(=O)NCC1(CCO)CC1 N=c1nc2c(C(=O)NC3CC(O)CN(C(=O)Cc4cn[nH]c4)C3)cccn2[nH]1 c1(CNC(c2cnc(C)s2)c2nnnn2CCCF)nc2ccccc2n1C C1(C(=O)OC2CC(C)OC2=O)COC2COCC2O1 C1(CC(=O)NCC2CC2NC(c2cc(C(N)=O)co2)=O)CCCOC1 c12[nH]c3nccnc3c1[nH]oc2=O.c1(C(=O)NCC)ccc(C)nc1 CC(C)CC(C)C(=O)N1CCC(Nc2ccc(NC(C3CCCO3)=O)cn2)C1 CC1C(C(N2CCN(C(c3n[nH]cc3C(C)(C)C)=O)CC2)=O)CCN1C Cc1cn2ccc(C(=O)NCC(C(C)C)NC(=O)CNC(=O)C(F)(F)F)cc2n1 n1(CC(=O)N(C)CCN(C)C(C23CC2C3)=O)nnc2ccccc12 c1(CC)ccc(-c2nc(C(n3cncn3)(C)C)nn2C(C)C(C)C)cc1 Cc1nc(CC(N2CCC2CNC(=O)C(N2CCOC2=O)C)=O)n[nH]1 C12(CNC(=O)CCCC(C)=O)CCCN(C1)C(=O)CN2.S(=O)(=O)(CCC)NC CN(NS(=O)(=O)c1ccc2sccc2c1)C(=O)Cc1ccccc1 c1(CC)cc(C(=O)NC2CC2CNC(C2(O)CC2)=O)oc1CC CC(C)CC(C)CC(C)NC(c1cccc(N2CCCCC2)c1)=O C#CC1CN(C(C2CC2C2CCCC2)=O)CCN1C(c1cnn(C)c(=O)c1)=O c1(SCC)cccc(C(=O)NC(CNC(=O)CC2CCS(=O)(=O)C2)C(C)(C)C)c1 c1(C(=O)OC)coc(C(=O)NCCCCCN(C(=O)C(C2CC2)SC)C)c1 N1(C(C2CCC(C)(CC)O2)=O)CCC2(CCC2)C(CNC(c2csc(C)n2)=O)C1 N1(C(C2OCCN(CC)C2)=O)CCN(C(c2c(C)cc(C)oc2=O)=O)CC(O)C1 c1(C(=O)NCC2(COC)CCCN2C(=O)CC(F)F)coc2ccc(C)cc12 C1(CCOC)CN(C(=O)CC2CCCCN2C)CCN1C(=O)CC1(CO)CC1.OC c1(N2C(C(C)C)CN(C(C3CNC(=O)C3)=O)CC2)nccc(S(C)(=O)=O)n1 C(=O)(CCC1=CCCCC1)N1CC(S(=O)(=O)N2CCN(C)CC2)C1 CCC(C)CCCC(=O)NC1CCCC(NC(C2(CC3CC3)CCCC2)=O)C1 c1(CC(=O)NCC(CC=C)NC(=O)CNC(=O)Cn2ccnn2)ncccc1C n1(CCC)nc(C)cc1C(=O)NCC(C)(C)NC(=O)C(c1cncc(F)c1)C CC1CN(C(=O)C2=CC(C)(C)C2)CC(CCNC(c2cccc(C#N)c2)=O)O1 c1(C(=O)NC2(CC)CN(C(=O)CC3(C)CC3)C2)ccc(Cl)cc1Cl CC1(CO)CN(C(C2C3CN(C(c4c(O)ccc(F)c4Br)=O)CC23)=O)CCC1O CCC(F)(F)CC(=O)NCC1CN(C(C2CC(C)OC2C)=O)CC1C CC1C(C)(C)CNC(=O)N1.c1(C(=O)NCc2ccco2)ccc(CN)nc1 C1(C(=O)NC2CC(C(C)NC(=O)Cn3cccc3)C2)CC2(C1)OCCO2 Cc1c(C(N2CCC(C(=O)NC(C)(C)C)C2)C(=O)NC(C)(C)C)cccc1O c1(NC(C2N(C(Cc3scc(C)c3)=O)CCC2(C)C)=O)ccc2ncccc2c1 c1(OCC(=O)NCCC2CN(C(C3CC34CC4)=O)C2)cc(Br)ccc1F CC1=C(C)CC(C(=O)NCC(O)CC(=O)NCC2(CO)CCCO2)CC1 C1(OC)(CNC(c2cc(C3CCCCC3)on2)=O)CCN(C(=O)C(C)C)CC1 C1(OC(C)(C)C)CC2C1CCN2CCNc1nc(-c2c(F)cccc2F)cs1 c1(SC)ccc(C(=O)NCC(C)(C2CCC2)NC(c2ccnn2CCF)=O)s1 CCC(C)C(O)C(=O)NC1(C(=O)NCC(=O)N2CCCO2)CCSC1 C1(NC(c2ncsc2Cc2ccccc2)=O)CCCN(C(=O)C(F)C2CCC2)C1 N1(C(C(C)N(C)C(c2cccnn2)=O)=O)CC(O)(C(F)F)C1 C(CN=c1[nH]c(N2CCOC(NC(C)C)C2)nc2c1CSC2)(C(C)C)OC C1(C(CC)NC(=O)CNC(=O)COCCOC)CC=CCC1 C[S+](C)CCC(O)C(=O)N1CCOCC(C)(CNC(=O)C=C2CCOCC2)C1 C1(NC(CCC)=O)CN(C(=O)CC2CCOC2=O)CCC12CCC2 c1(C(=O)NCC(CNC(C2(C(N)=O)CC2)=O)F)ccc(C#CC2CC2)cc1 Cc1cc(C)n(C)c(=O)c1C(=O)NCC1CC(NC(C2CCC(C#N)C2)=O)C1 Cc1cc(C(N2CCN(C3CCCN(C(C4CC4C)=O)C3)CC2)=O)oc1Br C1(C(N2CCC(O)(CCNC(C3(Cl)CC3)=O)C2)=O)CCC(F)(F)CC1 c1(C(=O)NC2CN(C(C3C(CC)C3)=O)CC2CC2CC2)cc(N)ccc1C CN1CCOC(C(=O)NCC(CO)NC(=O)CCc2cncnc2)C1 Cc1cc(CNC(c2cnccn2)=O)oc1C(=O)NC1CC(C(N)=O)C1 N1(C(C2(C#C)CCCC2)=O)CCC2CN(C(c3ccc(F)c(SC)c3)=O)C2C1 c1(C(=O)NC2CC(CNC(c3ccoc3Cl)=O)C2)cc2sc(F)cc2[nH]1 C(=O)(CC1=CCOCC1)N1CCC(C(=O)NCCOCCC(C)C)C1C C(=O)(C1=C(Cl)CCCC1)NC(CC(=C)Cl)C(=O)NCC1(C(N)=O)CC1 C1(NC(c2nccc(C)c2)=O)CN(C(c2ccncc2O)=O)CC12CCOCC2 N1(CCNC(CC2(CNC(=O)CCn3cccn3)CC2)=O)CCC2CC12 c1(NC(C(CCC)OC)=O)ccc(NC(c2ccn(C(C)(C)C)c2)=O)cc1C N1(C(=O)C(Cl)=CCl)CCN(C(c2ccc3c[nH]nc3n2)=O)C2CCCCC2C1 C=C1CCCN(C(C)C(=O)NC(=O)NCC)CC1 n1(CC(=O)NC(CCCCNC(COCC#C)=O)C)nc(C(F)F)c2c1CCC2 C(=O)(CC(C(C)C)NC(c1cccc(C)c1C)=O)NCc1n(CC)cnc1 C(=O)(C1CCCc2nccn21)N(CC(C)(C)NC(=O)C=C1CN2CCC1CC2)C Cc1cccc(C(=O)NC(C)CC(C)NC(c2c(F)cnn2C(C)C)=O)c1 C(=O)(C(F)C(C)CNC(C1CC2(CC(=O)C2)C1)=O)NC(CCC)CO Cc1cncc(C)c1C(N1CC(NC(c2cccc(Cl)c2O)=O)C(C)C1)=O CCS(=O)(=O)c1ccccc1-c1cnc(OC)c(C(N2CC3(CCC3)C2)=O)c1 CC1(C)CCC(CC(=O)NC2(CC=CC(=O)NCC3(C)CC=CCC3)CCC2)O1 C1(C(=O)NC2CN(C(C)C)C(=O)C2)C(C2CC2)CCN1C(=O)C1=CCCOCC1 CCCC(CC)CCC(=O)N1CCC(C(N2CCCNC(=O)C2)=O)(CC)C1 c1(OC)ccccc1OC1CN(C(=O)CC(C)(C)C)C1 N1(N2CCC(NC)C2)CC(F)(F)CC1CO.c1(C)ccc(CC(=O)O)s1 N12CC3CC1CC3Nc1ncccc1C2=O.C(=O)(C=C(C)C(=O)O)OCC Cc1cc(Cl)cc2[nH]c(C(=O)N(C3CCN(C(c4csc(CO)n4)=O)C3)C)cc12 N1(C(COC)=O)C2CCC1CN(C(c1sc(NC3CC3)nc1C)=O)C2 N1(C(=O)CSCC(F)(F)F)CC(C2CCCN(C(=O)CC3CC3)C2)C1.c1cccs1 C1(NC(C2(COC)CC(=O)C2)=O)CCN(C(C2NC(=O)OC2C)=O)CC1F c1(C(=O)NCC2(CNC(C3(Cl)C(C)(C)C3)=O)CC2)ncn2c1CCC2 c1(C(N(C(CN(C(Cn2c(C)csc2=O)=O)C)C)C)=O)cc2c(ccn2C)s1 C1(NC(C(n2cc(-c3cnccc3Br)nn2)C)=O)CC2CC3C(C2)C13 C1(OC)CC2(CCC(C(=O)NCC3(O)CCN(C(C4C5CCCC45)=O)C3)CC2)C1 CC1(C)CCCCC1CC(=O)NC1CC2CC1CN2C(=O)C=Cc1ccoc1 C1(CCCCNCC(=C)C)CCCN(C(C2(C3CCCCO3)CC2)C)C1 C(=O)(CC(C(C)C)C(C)C)N1CC(CNC(C=CC)=O)C(c2cncn2C)C1 C=CC(C)CC(=O)NCCCC(C)NC(c1cccc(CN2CCCC2)c1)=O C1(NC(c2ccccc2)CC)CCN(c2ccncn2)C1 Cn1cnc(N2CC(O)(CCNC(=O)C=CSCc3ccco3)C2)cc1=O C1(CNC(Cc2c(C)ocn2)=O)CCCC2CN(C(=O)CCCS(C)(=O)=O)CC12 C(=O)(N=c1cc(COC)n(C)[nH]1)C1C2CN(C(CC(CC)O)=O)C1C2 c1(C(=O)NC(C2CCN(C(CCC(C)OC)=O)C2)(C)C)nccn2c(C)nnc12 Cc1cc(F)c(C(N2CCOCC2CC(=O)Nc2ncc(Br)cc2I)=O)c(Br)c1 C1(N(C(c2ccc(OC)s2)=O)C)CCCC2CN(C(C3CC(F)(F)C3)=O)CC12 C(CCCCCC(=O)N1CC2(C(=O)NCc3ncc[nH]3)CC1CO2)NC(C)=O CCCC(C(=O)N1CCCC1CSC)NC(=O)C(=Cc1ccco1)C N1(C(C(CCC)C)=O)CC2CCC(Nc3ncnc4ccc(Cl)cc34)CC2C1 c1(C(N(CCNC(=O)CC2CCC(C)CC2)CC)=O)cccc(=O)n1C N1(CC(=O)NCC2C(CNC(C3(C=C)CCC3)=O)C2)Cc2ccccc2C1=O C(=O)(CS(=O)C(F)(F)F)N(CC(C)CNC(=O)C1=NOCC1)C N1(C(C2C(COC)C2)=O)CC2(COC(CNC(=O)CCN3CCCS3(=O)=O)C2)C1 c1(N(C2CCN(C(C3=C(C)CC3)=O)C2)C)ncnc(C(F)F)c1Br c1(-c2c(C(N3C(C)CCC3C)=O)cc(Cl)cn2)nc2c(s1)CCC2 N1(C(CCCn2cc(C(C=C)(C)O)nn2)=O)CC(C)C(O)C1.c1(N)ccccc1 NS(=O)(=O)CCCCCC(=O)NC1CC(NC(=O)CCCn2cccn2)C1 c1(C(=O)NC2CN(c3ncc4sccc4n3)CC2F)csc2ccccc12 Fc1ccc(OCC2CCCO2)c(CN2CCC2c2ccccc2)c1 C(=O)(C(F)(CN)CC(=O)OCCCc1ccc(Cl)cc1OC)OC C(=O)(C(C)S(C)(=O)=O)NCC1(SC)CN(C(c2cncc(NC(CC)=O)c2)=O)C1 c1(C(c2n(CCOC)nnn2)NC2CCCSC2)ccc(CNS(C)(=O)=O)cc1 N1(C(c2ccc(C(=O)OC)s2)=O)CCC(NC(c2cnn(C)c2C)=O)C1C c1(SC)ccsc1C(=O)NC(C)C(C)NC(=O)CC(C)C N1(C(Cn2cc(C(C)(C)OC)nn2)=O)CCCC(Cn2cc(CC(C)O)nn2)C1 CC(CC(C)(C)C)C(=O)NC1CC12CCN(C(c1ccc(Cl)cc1F)=O)C2 C(CCCCCCCCC)(c1n(CC=C)nnn1)NCC(c1cccc(F)c1)(C)C CCCCC(C)C(=O)N1CCOC(CCCNC(c2snnc2CC)=O)C1 c1(C(N2CCC(CCNC(C3(Cl)CCCCC3)=O)CC2)=O)ccc2cccnn12 N1(C(c2n(C(C)C)ccc2)=O)CC(NC(c2c(Cl)csc2Cl)=O)CC(C)(C)C1 N1(C(c2c(C)cccn2)=O)CC2(CCC(NC(C3CC3CN(C)C)=O)CC2)C1 C#CCC(C)(C(=O)NCP(C)(=O)OCC)NC(=O)CCCCCSC C1(O)(CNC(C2C3CCC23)=O)CCCN(C(c2ccccn2)=O)C1 c1(OC)ncccc1NC(N1CCCC(CCCCSC)C1)=O N1(CC(=O)N(CCNC(CC)=O)CCOC)CC2CC(C1)C2 C=CCC(C(=O)N1CC=CC(NC(=O)Cc2cnc(C)s2)C1)OC CC1CCC(NC(=O)Cc2ccc(Cl)c(F)c2)CN1C(=O)CC1(C)CCCC1 C(=O)(C(C(C)C)C(C)C)NCC(CNC(c1nc(C(=O)OC)sc1)=O)OC Cc1cnccc1C(N1CC2C(CNC(c3cnc[nH]3)=O)C2C1)=O C1(C(N(CCC)CCNC(=O)CC2CCC3(CC3)CO2)=O)CCC2CC1C2(C)C N1(C(C(C(C)C)SC)=O)CC2(CCCC(CNC(=O)C(C)Cc3cnco3)O2)C1 c1(C(=O)NCC(CNC(CC(CC)C2CC2)=O)CO)cc(N(C)C)cc(F)c1 c1(OC)ccc(C(N2CCCN(C(C3CCCS3)=O)CC2)=O)cc1[N+](=O)[O-] C1(CCOC)(NC(C2CCC(=O)N2C)=O)CCN(C(c2sc(CO)nc2C)=O)C1 N1(C(CC)=O)CCCC(C(=O)NCC2C3CN(C(c4c(C)ncn4O)=O)CC23)C1 CCC(CC(=O)N(C)CCN(C)C(c1cnn(CC(F)(F)F)n1)=O)CC(N)=O N1(C(C(CC#C)O)=O)CC2CC(NC(c3cc(C4CC4)ccn3)=O)C1C2 c1(OCCC(=O)NC2CCC(CNC(C=C(C)C(F)F)=O)C2)cccc(C)c1C N1(C(c2noc(CC)c2C)=O)CCN(C(=O)Cc2ccccc2Cl)CC1C Cc1cc(F)ccc1C(N1CC(N(C)C(C2CC2C)=O)C(C)(C)C1)=O C(=O)(CCCCCCCC1CC1)NC(C(C)C)(C)CNC(=O)CN(C)C1CC1 N1(C(CS(CC)=O)=O)CCCC2(NC(=O)COc3cc(C)ccc3C)CC2C1 C(C(COC)C(=O)N1CC(O)(CCNC(C2SC3C=CC2C3)=O)C1)OC C1(Nc2ccc(C#C)s2)CC2(C1)CC(C(=O)N(C(C)C)Cc1ccccc1I)C2 C(N=c1cc(C)[nH]c(=NCCOc2ccccc2OC)[nH]1)C1(C)N=C(C)SC1 c1(CC)nnc(CNC(C2CCN2C(=O)C(C)n2ccnn2)=O)o1 N1(C(C2(C(=O)OC)CC2)=O)C2CCC1CC(NC(c1cc(Cl)sc1Cl)=O)C2 CC1NC(C(=O)Nc2nnnn2Cc2ccccc2)=NN(c2ccccc2)C1=O c1(C(=O)NCC2CN(C(c3c(CC)n(C)nc3)=O)CC2C)cc(C)c(F)c(C)c1 c1(OCCC(=O)NC2CCC(NC(c3c(CC)nco3)=O)C2)cccc(C)c1 N1(C(C(C)SC(F)(F)F)=O)CCCN(CCNC(C2(S(C)(=O)=O)CCC2)=O)CC1 N1(CCNC(c2c(CC)cno2)=O)CCCN(C(=O)CC2(C)CCCO2)CC1 C1(NC(C2(N(C(c3cnn(CC)c3C)=O)C3CC3)CCC2)=O)CCCC(O)CC1 c1(C(N2CCC(F)(CNC(=O)CC3CNC(=O)C3)C2)=O)cc(F)cc2nc[nH]c12 Cc1nc(C=CC(=O)NCC(C)(C)CNC(c2ncn(C)n2)=O)[nH]c1C N1(CCCNC(=O)NCC(=O)NCC2CC(C(=O)OC)C2)CCOCC1.OCC N1(C(c2c(C(C)C)ccc(Br)c2)=O)CC2(CCCN2C(=O)C#CC2CC2)C1 C1(C(N(c2c(C)c(Cl)ncn2)C2CCCOC2)=O)CCN(CP(C)(C)=O)CC1 N1(C(C(n2cc(CCN(CC)CC)nn2)C)=O)CCC(C#N)(CCC#N)CC1 C1(NC(C(C2CC2)OC)=O)CC2CC(C1)N(c1ccnc(Cl)n1)C2 Cc1ccc(Cl)cc1C(=O)N(C1CN(C(C2(c3ccc(Cl)cc3)CCC2)=O)C1)C CN1CCC(NC(=O)CSCc2ocnc2)C1.C1(C(=O)N)(CO)CCCO1 C1(NC(C2C(C(=O)OCC)C2)=O)CCOCC1NC(=O)CC1(C)CCCCC1 Cc1ccc2oc(C(N3CC4(CCCN(C(C5CC(C)CO5)=O)C4)C3)=O)cc2n1 C(=O)(C(F)(F)C(C)O)NCc1c(C(NOCC=CC)=O)c[nH]n1 C1(CC(C)C)CCN(C(C2CC23CC(NC(c2ccnnc2)=O)C3)=O)CC1 c1(CC)c(C)cc(C)nc1N1CCCC(NC(c2cnn(CCCOC)c2)=O)C1 N1(C(c2ccn(CC)c2C)=O)CC2(CC(NC(C3CCS(=O)CC3)=O)CO2)C1 CCN=C(NCC(c1ccco1)N1CCCC1)N1CCC2C(C1)C2(F)F C1(=O)CC(C)C(C)(C)N1.C(=O)(C(O)Cc1cnc[nH]1)NC(C)C=CC(=O)N(C)C Cc1cccc(C)c1CNC(N1CC(NC(=O)CCCCCO)C1)=O Cc1cc2sc(C(=O)NCC(C)CNC(c3c(C)cccc3Cl)=O)cc2s1 N1(C(c2cccc(OC)c2F)=O)CCN(C(c2cncc(N)c2C)=O)C2CCC12 N1(C(C(F)=CC)=O)CC(C)(C)CC1CNC(C1(c2cccc(Cl)c2F)CC1)=O C1(CNC(C(CC)N(C)C)=O)CCN(C(c2c(C)nn(C)c2C)=O)C12CCC2 C(C)(C1=NOC(F)C1)NC(C1CC=CC(OC)C1)=O Cc1ccc(Br)c(C(N2CCC(C(N3CCC(CO)C(O)C3)=O)C(O)C2)=O)c1F c1(C(N(C(C)CNC(=O)Cc2ccon2)C)=O)cc2scc(Br)c2[nH]1 N1(C(C=CC(C)NC(c2cc(C(C)C)no2)=O)=O)CC2CCC(C2)C1 C1(C)(CNC(C(CSC)O)=O)CN(C(c2cc(C(F)(F)F)n(C)n2)=O)C(C)(C)C1 C1(CC)COC(C)(C)CN1S(=O)(=O)CCc1cccc(F)c1 C1(COC)(NC(c2cnncc2C)=O)CCN(C(=O)CN(C)C)C1 C(=O)(CCCCC(F)F)N1CC2CC(N)C2C1.c1(C(=O)OCC)cncc(C=O)c1 c1(N2C(C(=O)NC(C(=O)OC)C(C)O)CCC2)nc(C(F)(F)F)c2sccc2n1 C(=O)(CC(C)CN(C)C)NCC=CC(=O)N(CC)Cc1cccnc1 Cc1ncc2n1CCC(C(=O)NC1CCCCC1NC(c1ccc(Cl)[nH]1)=O)C2 C12(NC(Cc3c(C)ncs3)=O)CCOC(CNC(C3CCCS3)=O)(C1)C2 Cc1ncncc1C(N1CC(CNC(c2cc(Br)sn2)=O)CC1C)=O N1(C(c2c(CCC)[nH]cc2)=O)CCCC(NC(c2cn(C)cn2)=O)C1 C(=O)(C(C(C)C)SC)NCC(CC)NC(c1cc(CC2CC(O)(CO)C2)on1)=O N1(C(C(C)CC#N)=O)CCC2(CCN(C(=O)C(C)(C)C(N)=O)C2)C1 CC(C)(C)CS(=O)(=O)CC(=O)NC(CNC(C1(S(N)(=O)=O)CCC1)=O)C(C)(C)C c1(C(=O)NCC(C2CCC2)NC(=O)CC2CCCC23CC3)cc(F)c(F)c(F)c1 c1(OC)ccc2c(c1)C(C(=O)NC(c1ccc(F)cc1Cl)C(C)C)CCC2 N1(C(CC2(C(=O)OC)CC2)=O)CCCC(N(C)C(C2CC2(Cl)Cl)=O)C1 C1(CNC(c2n(COC)ncc2)=O)CCN(C(c2cc3c(s2)CCC3)=O)CC1O Cc1cc(CCC(=O)NC2CC(CCNC(C3CCS3(=O)=O)=O)C2)n[nH]1 CC1(C)C2CCC1(C(N1CCC(C)(NC(c3ccn(C(F)F)n3)=O)C1)=O)CC2 C1(NCC2(N3CCCC3C(=O)NCC)CCC2)CCCCCC1 c1(C(=O)NC(C2CCN(C(CC(C)O)=O)CC2)C)ccn(C(C)(C)C)c(=O)c1 c1(C(N2CCCC(NC(=O)C3=CCC3)C2)=O)ccnc2cc(F)cnc12 c1(C(COCC)N(C(c2ccc(Cl)c(Cl)c2)CC)C=O)cc(Cl)cc(Cl)c1 c1(C(N2CC(O)(CNC(CC3CC(CC)C3)=O)C2)=O)c(O)ccc(F)c1C c1(C(=O)NC2C(NC(C(=C(C)C3CC3)F)=O)C2)nc(-c2ccccc2)oc1C C1(F)(C(=O)NC2CC(CCNC(C=CCCC=C(C)C)=O)C2)CC2(CCC2)C1 C1(C(N(CCC)CCO)=O)CN(C(=O)CC2CC3(CC3)C2)CC1C1CC1 N(C(=NCCCCl)NC1CCCC(C)C1)CC(=O)NC(CC)(C)C Cc1nc2c(C(=O)Nc3cc4n(n3)CCC4)cccc2o1 C(=O)(C(C)CCC(C)(C)C)N1CC2(N(C(Cc3cc(C)cc(F)c3)=O)CCC2)C1 c1(CNc2n(CC(=C)C)nnn2)nn(C)cc1Cl N1(C(C=CC(CC)C)=O)CCC(C(=O)NCC2CC(O)C(O)C2)CC1C1CC1 C1(CC(=O)NC(C2CCOCC2)C#C)CC(NC(=O)C=CCCC)C1(C)C N1(C(C(C)(C2CC2)OC)=O)CC2CCC1(CNC(C1(F)CCC(F)(F)CC1)=O)CC2 C(C(CC(C)C)C(=O)N1CC(F)(C(=O)NCC2(CO)CCCCC2)C1)OC c1(C(=O)NC23CC(CNC(C4(COC)CCOCC4)=O)(C2)C3)ccc(=O)n(C)n1 C1(O)(CNC(N)=O)CCC(F)(F)CC1.c12ccc(cc1)C=CC(=O)N2 C1(C(=O)NCCCOCC)CCN(C(=O)CC2CCCCC2)C1C N1(C(c2cnc(CCC)s2)=O)CCN(C(C2C=C2C)=O)C2(CCC2)C1 N1(C(c2c(SC)snn2)=O)CCCC(O)(CNC(=O)C(F)C(C)C)C1 c1(CN2C(C(=O)Nc3c(C(=O)OC)ncs3)CC2)cc2cc(Br)ccc2s1 N1(C(C(CC#C)C2CC2)=O)CC(C(=O)NCCc2nc[nH]n2)CC1(C)C c1(-c2cc(C(N(C(CNC(C3C(C)C3)=O)C)C)=O)no2)ccccc1Br N1(C(CC(C)(C)C)=O)CC2CCN(C(c3cc(Cl)c(Cl)s3)=O)C2C1 C1(CC)CN(C(=O)C(=Cc2c[nH]cn2)F)CCN1C(=O)C1=CCN(C)C1 c1(CC)cc(NC(C2CC(F)CN2C(=O)CN2CCN(C)CC2)=O)cc(F)c1 C#CCC(C)(CC)C(=O)NCC1CC(NC(c2cccc(C)c2)=O)C1 N1(C(C)=O)CC2(C=C(C(=O)N3CCC4CC4C3)CO2)C1.c12ccc([nH]1)C2=O N1(C(C(CCSC)O)=O)CCC2CN(C(=O)Cc3nocc3C)CCC12 C1(CC(C(=O)Nc2cccc(CO)c2)O)CCCN(CC(F)F)C1 CC(C)CCCCC(=O)N1CC(NC(c2ccc3ocnc3c2)=O)C(C)C1 C1(C(=O)NC(c2c(C)cccc2)C)CN(C(C2CCCC2F)=O)C(C)(C)C1 N1(C(CCCCC)=O)CCN(C(=O)CSc2nnnn2C)C(CC2CC2)C1 N1(C(C(=O)NCC(=C)C)C(C2CCCCC2)OCC)CCC(CN(C)C)C1(C)C CCCS(=O)(=O)C(C)C(=O)N1CCCC1(C)CNC(=O)CCc1ncc[nH]1 N1(C(c2c(C)cccc2C)=O)CC(CNC(C2(C#N)CC2(C)C)=O)C2(CCC2)C1 N1(C(CC)=O)CCc2cc(C(N3CCC3CNC(=O)CC(C)SCC)=O)ccc21 C(=O)(C1CCCc2ncccc21)N1C(CNC(C(C)CCO)=O)CC(F)(F)C1 Cc1[nH]nc2c1CCC(C(=O)NCC#CCNCCN(S(C)(=O)=O)C(C)C)C2 N1(C(C2(C)CCCO2)=O)CCC2(CCN(C(C3CCCC(=O)N3)=O)C2)C1 C1(N(C(C2CC(Cl)(Cl)C2)=O)CC)CCN(C(=O)CC2CCCCO2)CC1 CCCS(=O)(=O)CC(=O)N1CCCC1C1(C(=O)NCc2ocnc2C)CC1 n1(CC(=O)NC(CC)CNC(C2COC(=O)N2)=O)cc(S(N)(=O)=O)cn1 C1(NC(c2[nH]cc(CC)c2)=O)CCC(C)(CNC(=O)C=Cc2sccc2C)CC1 c1(C(=O)N=c2ccn(-c3ncccc3F)[nH]2)cc(F)c(F)c(F)c1F c1(N(C)CCF)nc(N(C)Cc2csc(C(F)(F)F)n2)c2c(n1)COC2 N1(C(C(c2ccc(C)s2)C)=O)CC2CC2(NC(c2cnn(CCO)c2)=O)C1 c1(CC(C2CCCOC2)OC(CC(=O)NC(C)(C)C)=O)nccc2ncccc12 C(=O)(CC(C(F)(F)F)SCC)NCC1CC(NC(CCC=C)=O)CC1O c1(C(N2CC(CNC(CSCCC)=O)C(O)C2)=O)ccc(N)c(Cl)c1 C1(CC(=O)NC(C2CCCCC2)C)CCCN1C(c1cc(C(C)(C)C)c[nH]1)=O N1(c2nnc(COCC)s2)CCC2(CC1)CC2C(=O)NC(c1ccncc1Cl)C C12(C(N3CC(O)(CN(C(C(C(C)C)SCC)=O)C)C3)=O)CCC(C#N)(CC1)CC2 CC(C)CCCC(C)C(=O)NCC1(CC(=O)N(C)CC2CC2C)CC1 c1(C(N2C3C(Nc4nc(SC)nc(C)c4)C(CC3)C2)=O)sc2cncn2c1C C1(C(C)C)CCN(C(C2COC(=O)N2)=O)C(C(=O)NC(C2CSC2)C)C1 C1(=CC(=O)NCC(C)(Cn2cccn2)NC(C2CSC2)=O)CN2CCC1CC2 C1(CNC(CCOCCC)=O)CC(C(C)C)CCN1C(=O)C(CC)NC(C)=O O=S(CCc1nc(-c2c(F)ccc(F)c2Cl)no1)CC(F)(F)F c1(CCC(=O)N(C2CCN(c3ccncc3)C2)C)nc(Br)cs1 CC1(C)CCCOC1C(N1CCCC(CCNC(C2CCC=CCCC2)=O)C1)=O c1(OC)cc(C#N)ccc1C(=O)NCC(C)(C)OCCNC(C1C2CCCC12)=O c1(C(=O)NC2C3CN(S(CC(=O)OCC)(=O)=O)CC32)cc2c(F)cccc2[nH]1 C1(C(N2CCC(CC(=O)N(C)CC3CCOC3)CC2)=O)CCC(C2CC2)C1 C12(CCNC(CN3CCN(C)CC3)=O)CCC(C1)N(C(C1CCC(C)CC1)=O)C2 Cc1coc(C(=O)N(C)CC2CCCN2C(=O)Cc2cccc(C(N)=O)c2)c1C N1(C(C(CC)C)=O)CCCC(CCCCNC(=O)Cc2ccc(C(C)=O)cc2)C1 C(=O)(C(O)C(C)OC)NCCC1CC(C(=O)NCC2(C(=O)OC)CC2)C1 Cc1cnc(NC2CCC(NC(=O)CC3CCCC3(F)F)CC2)nc1C c1(C(N2CC(O)(C(C(=O)NC(CCC)CC)F)C2)=O)cncc2[nH]ccc12 C(=O)(CC1CC(=O)c2ccccc21)N(C)CC1CCCN(C(C=CCC)=O)C1 c1(N(C2(C#N)CCNC2)C(C(C)C)=O)ncnc2cccc(F)c12 c1(C(CNC(CCOCC#C)=O)NC(C2(O)CCSCC2)=O)cccc(Cl)c1Cl n1(Cc2ccoc2C(=O)NC(C)CSC)ccnc1C(=O)OCC N1(C(CC2CCCN(CCn3ccc(C)n3)C2)=O)CCOC(C)(C)C1C N1(C(c2ccc(C)n2C)=O)CC(O)C(O)C1CNC(=O)CCC1CC1 C1(CNC(CN(C2CCSC2)C)=O)CCC(C)(C)CN1C(c1cnn(C)c1N)=O C(=O)(CCCCNC(=O)C(C)C1(O)CCC1)NCCCOCC(C)C CCCCN=C(NCCn1ncc2ccccc2c1=O)N1CCC2(CCCC2)C1 CC(F)(F)C(Cl)CNC(=O)C(Cc1cn[nH]c1)NC(=O)COCCCF N1(C(c2nc(C(C)C)oc2)=O)CC2CC1CC2CNC(c1cc(O)cs1)=O c1(SC(C(=O)NC2CCC(CNC(C(C)NC(N)=O)=O)C2)C)ccccc1 c1(CNC2C(C(=O)NCc3ccc(C(=O)OC)cc3)CCC2)ccc(O)c(I)c1 Nc1nc(Br)ccc1C(=O)NCC1CCN(C(=O)CN2CC=CC2)CC1O Cn1ccnc1C(=O)NCc1n[nH]cc1C(=O)NCC1CC(CO)CO1 N1(C(COC2(C#C)COC2)=O)CC2CCC2(CC(N2CC(C(=O)NC)C2)=O)C1 N1(C(C2(CC=C)CCC2)=O)CC(CNC(c2cc(CC)no2)=O)C(C)C1 c1(C(=O)NC2C(CNC(C(C)(C)c3cnsc3)=O)C2)cc(Cl)c(F)cc1Cl c1(OC)ccc(S(=O)(=O)N(C)C)c(NC(C2CC(=O)C2C(C)(C)C)=O)c1 N1(C(C=CC)=O)CC2(CCCCN(C(C3CCOC(C)(C)C3)=O)C2)C1 N1(C(=O)CC2CC3(C2)CN(Cc2cccc(F)c2F)C3)CCC2COCC2C1 N1(C2CN(S(C(C)C)(=O)=O)C2)CCC(O)C(O)C1 N1(C(C2N(C(C)=O)CCCC2)=O)CCCC2(NC(C3SCCS3)=O)CC2C1 c1(N2CCN(C(c3ccc(C)cc3O)=O)C3C2C3)ncc2[nH]ccc2n1 CCC(CC)(C(=O)NC1CN(C(=O)CC(C)(C)C)CC1c1ccccc1F)OC C(=O)(C1CC(=O)Nc2ccccc21)N(C1CCCN(C(c2ccc(=N)[nH]n2)=O)C1)C CN1CC(C(=O)NCCOCCN(C)C(c2cnc(Cl)cn2)=O)C(C(F)(F)F)C1 S(=O)(=O)(c1cc2sc(=NCCCCCCCC#N)[nH]c2s1)NC(CCC=C)CO c1(C(=O)NC2C(C)N(C(C3CCC3(F)F)=O)CC2)cc2c(s1)CCOC2 c1(C(=O)OC)cc(S(=O)(=O)Oc2cccc(OC(C3CCCCO3)=O)c2)ccc1C C1(NC(C(CCC)NC(N)=O)=O)CCN(C(=O)CCN2CCCCC2=O)C1(C)C Cc1nc2cccc(C(=O)NC(C)CC(C)NC(=O)CN3CC(C)(C)C3)n2n1 C1(C(=O)NCC(C)OC(F)F)CCC(C)N(C(=O)C(C)c2ccco2)C1 n1(CC)cc(CCNC(=O)C(c2cccs2)NC(C2CCC(=O)O2)=O)cn1 Cc1cc(CCNC(=O)CC=CCNC(=O)C(C)CN2CCCC2)nn1C c1(C(N2C(C)CCC(CNC(CCOCC)=O)C2)=O)ccc(C)c2ccccc12 N1(C(C(CCC)O)=O)CCCC2(NC(C3CCc4ccccc4C3)=O)CC2C1 c1(OC)ccnc(C(=O)NCC2CCN2C(C2CCC3CC3CC2)=O)c1OC Cc1cc(C=CC(=O)NCC(CO)NC(C2CC(C(C)(C)C)=NO2)=O)c[nH]c1=N CCCC(C)(CC)C(=O)NC1COCCN(C(C2CCCC2O)=O)C1 c1(N2CCC(CCCC)C2)cc(N2CCC(CCC(N)=O)C2)nc(C)n1 CC1(C)C2CCC1(CC(=O)NCC1CCCN(C(c3cc(Cl)no3)=O)CC1)CC2 c1(C(N(C(CCNC(C2(CCOC)CCC2)=O)C)C)=O)csc(C(F)F)n1 N1(C(C2(C(=O)O)C(C)OCC2)=O)CCc2nnc(-c3ccccc3)cc2C1 C1(N(C(C(CCC)O)=O)C2CCN(C)C2)CNCCOC1C(=O)OC.C(C)(C)(C)O N1(C(c2ccc(CCC)s2)=O)CC(C)CCC1CNC(c1cccn1CC)=O C(=O)(C(C)(C)COCCN(C)C)NCC(C)CF Cc1ncc(C(N2CC3C(C(F)(F)F)C3C2)C(=O)NCCC#N)cn1 Cn1ncc2cc(C(=O)NC3CC(NC(=O)C(O)CN4CCOCC4)C3)sc12 c1(C(=O)NC2CC(C(=O)NCC3CCC(C)C3)CC2O)cnn(C)c1C#N C1(C(=O)NC(CC2CCN(C(C(COC)C)=O)CC2)C)CCCC12CCOCC2 C1(NC(C(C=CC)O)=O)C2CC3C1C3C2C(=O)NCC=CC=CC C1(C(=O)NC(CC(C)NC(C2CCCOCC2)=O)C)CC2CCC1CC2 c1(C(C)NC(N2CC(c3ccc(C)cc3)(O)C2)=O)ccc(F)c(F)c1 C(=O)(C(CC)CC(F)F)NCC1(CO)CCN(C(C2(C(=O)OCC)CC2)=O)CC1 N1(C(C2C(C)(C)CC2)=O)CC2CCC1C(NC(=O)CSCC#N)C2 C1(NC(C2C3CCCCC23)=O)CCCN(C(C2CC23CCCCC3)=O)CC1 N12CC3CCCC(C1)(C3(F)F)NC2=O.C1(CC(C)C)CCC(C(=O)OC)CC1 c1(C(=O)OC)cc(=NCc2ccc(C#N)cc2)cc[nH]1 N1(C(CC2CC(N(C)C)C2)=O)CCC(C)(CNC(C2CCSC2)=O)C1 N1(C(COCCN(C)C)=O)CCC2(CCCN2C(C2CC(=O)OC2(C)C)=O)C1 C(C(CO)(CO)NC(=O)CCNC(N)=O)N(C(C(=Cc1ccco1)C)=O)C Cc1nc(C(N2CCSCC2CCNC(=O)CC2(OC)CCOCC2)=O)nn1C c1(C(N2CCC(CNC(C(COC)O)=O)C2)=O)c[nH]c2cc(C)ccc12 N1(CC(C2CCCC2)OC)CCC(C(=O)NC2CCCCC2)C1 C1(O)(CNC(C2(C#N)CC2)=O)CN(C(=O)Cc2nc(C3CC3)cs2)C1 CC1CC2CN(C(=O)C(=O)NC3CC3C3CC3)CC2N1C(=O)Cc1ccccc1 c1(C(C)C)ccccc1OCC(N1CCC(O)(CN2C(C(C)NC)CCC2)C1)=O N1(C(C2C(C=C)OCCC2)=O)CC(CNC(=O)CCOCC2CC2)CC(C)(C)C1 N1(C(Cc2c(C)n(C)cn2)=O)CC2(CCCC2)C1C(=O)NCc1cnns1 CC1CCCN1CCNC(C1CCC(CNC(=O)OC(C)(C)C)C1)=O.C(C(C)(C)C)O CN1CCC(Cc2ccccc2)(NC(=O)NC2CCCC2n2ccnn2)C1 n1(CCC)c(CN2CC3CCOCC(C3)C2)nc2sc3c(c2c1=O)CCCCC3 N1(C(C(C)C#N)=O)CCN(CCNC(c2ccnn2CC2CCC2)=O)CC1 c1(C(=O)NC(CC)CNC(=O)C(C)(C)C#N)cc2cc(OC)ccc2n1C N1(C(C(=O)NCCCO)=O)CCCC1.C(CCCO)C1(C(=O)NCCCN)CC1 N1(C(CC2CC(CC)C2)=O)CCCCC(CC(=O)NCC(N2CC=CC2)=O)C1 CC1(C#CC(=O)NC2CN(C(=O)Cn3ccc(C(F)(F)F)n3)C(C)(C)C2)COC1 C1(CNC(C(C)(C)SC)=O)CCC2CN(C(=O)CN(c3ccccc3)C)CC12 CCC(C)(C(=O)NCC1CN(C(C2CCCC2)=O)CC(C)(C)O1)C(N)=O c1(C(=O)NC2CC(N(C)C(C3CCCCNC3=O)=O)C2)nccc2c1CNC2=O C1(NC(COC)=O)CN(C(c2cccnc2-n2nccn2)=O)CC1N=[N+]=[N-] N1(C(C=C(C)C)=O)CCN(C(=O)Cc2cc(C)ccc2C)C(C)C1C c1(C(N2C(C)CN(C(C3COCCO3)=O)CC2)=O)cccc2nn[nH]c12 C1(NC(COC)=O)CC2CCC1N(C(=O)CNS(=O)(=O)C1CC1)C2 c1(C(N2CCC(CC=C)(NC(=O)CO)C2)=O)nc(Br)c2c(F)cccn12 C1(NC(CC2(N(C(CN3C(C)CCC3C)=O)C)CC2)=O)CCCCC12CC2 C1(NC(C(C)OCC#C)=O)CN(C(c2ccccc2COC)=O)CC1F N1(C(Cc2nc(=N)[nH][nH]2)=O)CC(NC(C2CCC(=O)NC2)=O)C(C(F)F)C1 O=C(CCCCc1ccc(Cl)s1)NC(c1ccccc1CC(F)(F)F)C(=O)O C1(C(N(CC(C)(C)CNC(c2ccc(CO)cn2)=O)C)=O)CC12CCCOC2 N1(C(C=CCN(C(=O)Cc2cnn(C)c2)C)=O)CCC(C)(O)C(O)C1 Cc1ccc(COCC(=O)NCC(CO)NC(=O)CC2(C)CC2)cc1 N1(C(c2c(C)ccn2C)=O)CCN(C(=O)CC2CCCCCCC2)C(C2CC2)C1 C12(C(=O)NC)CC(C=O)(C1)OC21CCOCC1.N1(CS(C)=O)CC(OC)CC1=O Cc1cn2ccc(C(N3CC(C)(NC(C4SC5C=CC4CC5)=O)C3)=O)cc2n1 c1(C(N2CCCCC2C2(C(=O)OCC)CC2)=O)onc(OCC)c1Br c1(C(C)NC(c2ncoc2CNC(c2sccc2C2CC2)=O)=O)cccnc1O c1(C(=O)NC2CN(C(C(CCCC)C)=O)C(C)CC2)ccc2c(n1)CCC2=O c1(C(N(C2CN(C(C=Cc3scc(C)n3)=O)CC2F)C)=O)cc(Cl)cc(C)c1C C1(NC(COCC=C)=O)CCC(OC2CCN(C(=O)COCC)C2)CC1 c1(C(N2CC(C=C)(CC(=O)NCCC3OCCC3C)C2)=O)ncc(C)cc1F c1(C(=O)NC(CNC(CCCOCC=C)=O)CCOC)ccc(C)c([N+](=O)[O-])c1 c1(CC)cccc(C(=O)NC23CC(CNC(c4sncc4C)=O)(C2)C3)c1 Cc1cccc(C(C)C(=O)NCCOCCN(C)C(c2nc(Cl)c(Cl)s2)=O)c1 C1(C(=O)NC(C=C)C2CCC2)CC1C1CN(C(=O)CN=[N+]=[N-])C1 C(=O)(C1Cc2c(Cl)cccc21)NCC1N(C(C(C(CC)O)C)=O)CC2(CC2)C1 c1(C2(C(=O)NCCC(=O)NCC=CCSC)CC2)ccncc1 Cn1nc2c(c1NC(C1C=CCN1Cc1cccc(C(F)(F)F)n1)=O)CCCC2 CC1CN(C(c2cnc(Cl)cc2Cl)=O)CCC1CNC(=O)CN1CCC1 c1(-c2scc(NC(C(c3n(C)ncc3)N)=O)n2)ccc(Cl)cc1 Cc1nn(CC(=O)NC2CC3CC(C2)N(C(=O)C(C#N)C(C)(C)C)C3)cc1[N+](=O)[O-] Cc1ccc2c[nH]nc2c1NC(C1CCCN(Cc2cc(Br)cs2)C1)=O C1(O)(CCNC(CC(CC)SC)=O)CCCN(C(c2ccc(N)cc2OC)=O)C1 C1(N(C)C(c2ccnn2CC#N)=O)CCC(NC(=O)CN2C(=O)CNC2=O)CC1 C(=O)(C(CC(F)F)Nc1nccnc1N)NCC(C(C)C)C CCC(C#N)C(=O)N1CC(C(C)NC(c2c(Br)nnn2C)=O)C1 c1(C(N(CCC)CCNC(=O)CC(C)(C)C)=O)cncc2c1CCNC2=O S(=O)(=O)(c1ccc(NC2CCCN(C3CC3)C2)c(Br)c1)NCC(C)F Cc1cc(C(=O)NCC2CCN2CC=C(Cl)Cl)sc1C C1(NC(C(C)=C2CCCC2)=O)CC(F)CN(C(c2cnc(S)n2C)=O)C1 C(C(C(=O)N1CC(F)(COCc2nnnn2C)C1)n1cc(C2CC2)nn1)OCC N1(C(c2c(CCNC(=O)CCC3CCCO3)n[nH]c2)=O)CC23CCC2(COC3)C1 c1(C(N2CC(C(C(=O)NC34CCCC3C4)OC)C2)=O)ncn2ccccc12 CC(C)CC(C)C(=O)N(C1CN(C(=O)Cn2cnnc2O)CCC1O)C N1(C(C(C(=O)OC)c2ccccc2)=O)CC(C)CN(C(=O)C(C)CC(C)C)CC1C CCC(CCC(=O)NCCC[Si](C)(C)C)NC(C1C2CCC(F)C12)=O Cc1nn(C)cc1CC(C(=O)O)NC(c1ccc(OC(F)(F)Cl)cc1)=O c1(C(=O)NC2(CC(=O)NCc3ccc(Cl)o3)CC2)cnc(CO)cn1 CC(N=c1[nH]c(Cl)ncc1[N+](=O)[O-])C1CCN(C(c2c[nH]nc2C2CC2)=O)CC1 c1(OC)ccc(F)c2c1CN(C(c1cc3ccccc3cn1)=O)CC2 c1(N(C(c2c(N)ccc(C)c2F)=O)C(C)C)ccc2oc(=O)ccc2c1 c1(C(=O)NC2CN(C(c3ncsc3C(F)(F)F)=O)C2)ncc2n1CCCC2 c1(C(=O)NCC2CN(C(C=CCC)=O)CC2C(F)(F)F)cc(P(C)(C)=O)cs1 c1(NC(N2C3CN(Cc4n(C(C)(C)C)ncc4)CC32)=O)cc2cc(Cl)ccc2s1 c1(OC)cc2c(C(=O)NCCN(CC(C)O)C(C3CC4CC4C3)=O)c[nH]c2cc1Cl Cn1cc(C=CC(=O)NCC(C)(C)C(=O)NCCn2ccnn2)cn1 c1(C(N2C(CNC(C3(C)CC(=CC)C3)=O)CC2)=O)cc(F)cc([N+](=O)[O-])c1Br Cc1sc(C)c2sc(C(=O)NC3CCCC3NC(=O)Cc3nncn3C)cc12 C(=O)(C(C)C(=O)OC)N1CC(CCNC(c2ccc(CN(C)C)s2)=O)(OC)C1 C1(C(C)C)CN(C(=O)C=CC(=O)N(C)C)CCC1NC(=O)CC1(C2CC2)CC1 c1(OCCC)ccccc1C(=O)NCCC1(O)CCN(C(=O)CC(Cl)Cl)C1 CC1(C)Oc2cc(C(N3CCC(c4ccccc4)(CO)CC3)=O)cnc2NC1=O C(CC(CC)C(=O)N(C1CCCC(C)C1)CCNC(C1CC(C)(C)CO1)=O)=CC c1(C(=O)NC(C2CCN(C(=O)CC3CNC(=O)O3)CC2)C)ccc(C#N)cc1F Cc1ccc(C(=O)NCCC2=CCN(C(=O)C3=COCC3)CC2)c(=O)n1C C(=O)(C(CC1CCCC1)C(C)C)N1CC(CNC(Cc2c(C)n[nH]c2)=O)OCC1 C(N=c1[nH]c(=N)[nH]c(=NCC2CCC23CCC3)[nH]1)C1N(C(=O)OC)CC2(CC2)C1 Cc1cncc(C(=O)NC2CCN(C(c3ccsn3)=O)CC2F)c1C C(=O)(CCS(=O)(=O)CC(C)C)NC1CCN(C(C(CC=C)C)=O)C12CCCC2 Cc1c(C(N2CCN(CCN(C)C(C3CCO3)=O)CC2)=O)cnn1CCC(C)C c1(OC)ccc(CNC(C2(C)CCCN2Cc2ccc(F)cc2O)=O)c(C)c1C N1(C(CCC(C)NC(C2CCC(CO)CC2)=O)=O)CC2(CCC2)OCC1C C(=O)(C1CCCc2nccn21)N(CC(C)(C)CNC(c1ccc(F)cc1N)=O)C C1(C(N2CC3(CC(NC(C4(CCCC)CCC4)=O)C3)C2)=O)CC2(C1)CC21CCC1 Cc1ccc(C(=O)NCC2CCN(CCCN3CCCCC3)C2)cc1 c1(C(N2C(C(C)NC(C3CC3C(C)(C)C)=O)CCC2)=O)ccc(-c2ccco2)o1 c1(CNCCN(c2cc(C)cc(F)c2)C(C2CC(Br)C2)=O)cccc2cc[nH]c12 c1(OC)cc(C(N2CCC(O)(CNC(c3ccnnc3)=O)C2)=O)ccc1F c1(C(N2CCC(C)(N(S(CC)(=O)=O)C)C2)=O)ccc(C)cc1SC.C1C(=O)N1 Cc1cc(C(=O)NC(C)CCNC(c2nnn3c2CSCC3)=O)cc(=O)n1C c1(OC)cc(C(=O)NC2CC(C)CN(C(c3ccc[nH]3)=O)C2)ccc1Br C#CCCCCCC(=O)NCC1C=CCN1C(=O)C(C)Cc1ccccc1Cl O=C(CCCCCNC(=O)CCc1nc(O)n[nH]1)Nc1ccc(CCO)cc1 C(=O)(CCCC(=O)NC1CC1)N1CC(C)C(NC(=O)CC2CCCSC2)C1 C1(CNC(Cc2c(C)ncs2)=O)CC2(CC2)CN1C(c1ccc(C(N)=O)cc1)=O c1(CNC(C2CCCN(C(C(COC)OC)=O)C2C)=O)cccc2c1OCC2 c1(N(C)CC)ccc(C(=O)NCC(C)NC(C2CC2c2cncn2C)=O)cc1 c1(C(=O)NC2CCN(C(CCCOCC=C)=O)CC2)ccc2ccsc2c1 c1(C(N2CC(CNC(C3C(CC)CCC3)=O)C2)=O)cccc(Br)c1 Cn1nc(C(N2CC3CC2C3C(=O)NCC#CC2CC2)=O)cc1C#N c1(C(=O)NC(c2nocc2C(N2CCN(C)CC2)=O)C)ncccc1F CCCCCC(C)(C)C(=O)NC1CCOC(C(=O)N(CC(C)COC)C)C1 CN1CC(O)(CN(C(=O)C(C2CCC2)NC(=O)C=CC2CCOC2)C)C1 c1(CC)oc2ccccc2c1CNCc1cc(Cl)ccc1OC(F)F C1(CCCC)CCCN1C(=O)CC(C)N(C(=O)CCN1CCOCC1)C c1(OCC)ccc2cc(C(=O)NCCNC(C34CC3CCC4(F)F)=O)ncc2c1 c1(C(=O)NC2CCCN(c3cc(C(=O)OC)ncn3)CC2)cc2ccncc2s1 CC1(C)C(C(=O)NCCC2NC(=O)NC2=O)CCN1C(c1n[nH]c(=N)[nH]1)=O CC1CCC(C(N2CC3CC3(NC(=O)COCCN(C)C)C2)=O)CC1 c1(C(N2CC(C(N)=O)(CNC(=O)C(c3cncn3C)O)C2)=O)cccn(O)c1=O N1(C(C(C)OCCC=C)=O)CCC(C(C)(C)Cn2cc(CSC)nn2)CC1 c1(NC2CCCN(CCCO)C2)[nH]c(=NCc2ccsc2)nc2sccc12 C1(C(N(CC(C)(C)NC(=O)CCn2cnnn2)C)=O)CCC2(CC2)C1 N1(C(c2cnc(C)n2C)=O)CCN(C(C2C=CCC2)=O)C(C)C1 Cc1ccc(N2CCCC2)c(C(=O)NC(C)CNC(c2ccc(=O)oc2)=O)c1 CCCC(C)(O)C(=O)N1CC2CCC2(CNC(c2ncc(Cl)cc2Cl)=O)C1 N1(C(C2C(C=C)CC2)=O)CCC(NC(=O)CCCC)C12CCC2 N1(C(C2(C(F)(F)F)CC(=C)C2)=O)CC(CO)C2(C1)CN(C(=O)CCNC(C)=O)C2 C(C(F)(F)C(=O)NC(C1CCN(C(=O)C(=C2CCCCC2)F)C1)C)OC C(=O)(C1CCc2ccccc21)NC1C(C2N(Cc3n(CCOC)ncn3)CCC2)C1 c1(C(=O)NC(CCNC(C=C(CCC)C)=O)C)cc(C)c(Br)cc1Cl c1(-c2nc(C(C)O)nn2Cc2ccc(Cl)cc2Cl)cnc(O)n(C2CC2)c1=O c1(SC)cccc(C)c1.C(C(O)C(=O)C(C1(CN)CC1)=O)SC CN1c2ccccc2CC1C(=O)N(C1CC1)CC1CCN(C2CCCCCC2)C1 C(C)(CNC(c1ncc(Br)cc1F)=O)(CC(C)C)NC(CSC)=O N1(C(C(COC)(C)O)=O)CC(C(=O)N(C)CC2CC2C)CC1(C)C CCC(O)C(F)(F)C(=O)N(C1CC1)CC1CCCN1C(C1CC1CC)=O C(=O)(C1=C(C)C(C)(C(=O)NC2CCCN(CC(C)(C)O)C2)C1)OCC C(=O)(C1COCc2ccccc21)NCCCC(C)(C)NC(Cc1cc(C)[nH]n1)=O c1(C(C)C)ccc(C(=O)NCC2CCN(C(C3(C)CCN(C)C3)=O)C2)nc1 N1(C(C(CC#C)C2CC2)=O)CCC2(CC(NC(C3(C4CCCO4)CCC3)=O)C2)C1 c1(C(=O)NCC2(c3ccccc3)CC(NC(C3C(C)=C3)=O)C2)ccc(C)cc1 c1(SC)c(C(=O)NCC(C)N(C(=O)CCC2CC2)C)ccc2c1OC(F)(F)O2 C1(NC(c2c(C)nsc2)=O)CN(C(c2cc(C3CC3)oc2C2CC2)=O)CC1F CCCC(C)(C)CC(=O)N1CC(O)(C(F)C(=O)Nc2cccc(CCO)c2)C1 C(=O)(C1=C(Cl)CCOC1)NCC1COCCN(C(c2c(C)scc2)=O)C1 c1(C(N)=O)ncn(CC(=O)NCCNC(=O)CCn2ccnc2C2CC2)n1 C1(OC)CC(C(=O)NOC2CCCCC2)C1(C)C.C12CC(C1(C)C)NC(=O)CO2 CCCCC(C)C(=O)N1CCC(CN(C(c2cc(C3CC3)on2)=O)CC)C1 C(=O)(C1CCc2cccc(=O)n21)NCC=CCNC(CC1(C)OCCO1)=O N1(C(CC(CC)OC)=O)CCC2(NC(c3ccc(C(F)F)cc3Cl)=O)CCCC12 CC1CCc2[nH]c(=NCCCOc3ncccn3)[nH]c(=NCC(Cl)=CCl)c2C1 CC1(C)CCCc2c1n[nH]c2C(=O)NC1CC(NC(=O)C(F)F)C12CCC2 C1(C(=O)NC(CNC(C2N(C)CCC2)=O)(C)C2CC2)COc2cc(O)ccc2C1 Cc1ncc(Br)c(C(=O)NCC2CC2NC(C2CCC3CC3CC2)=O)n1 C1(C(N(C2CCCN(C(Cc3c(C)noc3)=O)C2)C)=O)CC1C1CCOCC1 c1(CNC(C2CCCC2N2CCCC2)=O)nnc2c(=O)[nH]ccn12 C1(N(C(CSC)=O)CC2CC2)CCCN(C(=O)C(C(C)C)NC(N)=O)C1 n1(CC(=O)NCC(C)(CNC(c2cncc(C)c2)=O)OC)ccccc1=O c1(-c2c(C(=O)Nc3ncn(CC)c3)scn2)ccc(SC)cc1 CC1CC(CNC(c2csc(C(F)F)n2)=O)CN1C(c1nnsc1C(F)F)=O c1(C(N2CC(F)(C(=O)Nc3c(OC)ncnc3)C2)=O)cc(C)ccc1O C1(NC(c2c(C)cncc2)=O)CN(C(c2ccc(C(C)O)cc2)=O)CCC1O c1(C(N2CC(n3cc(CC4(CO)OCCO4)nn3)C2)=O)c(F)cc(F)c(F)c1Br c1(C(=O)NCC(c2cccc(C#N)c2)O)cc2ccc(Br)c(F)c2[nH]1 Cc1ccc(C#N)cc1C(=O)NCC1CC(NC(C2CC3CCC(C2)C3)=O)C1 CC(C)C(=O)C(=O)N(CC(=O)NCC(O)C1(Cl)CC1)C1CC1 S(=O)(=O)(c1ccc(NC(c2ccccn2)COC)cc1Cl)N(CCCCO)C C=C1CCC(C(=O)NC(C)CN(C(=O)CNC(=O)CC)C)CC1 C#Cc1ccc(C(N2CCOC(CN(C)C(C3CC(C)=NO3)=O)C2)=O)c(F)c1 Cc1cccc2oc(N3CC4CC(NC(C5(S(C)(=O)=O)CC5)=O)CC4C3)nc12 N1(C(C2CNC(=O)N2)=O)CCCCC(CNC(c2n[nH]cc2C2CCC2)=O)C1 O=C1CC(C(=O)NCCC2CCCN2C(C2COC3CC2C3)=O)=NN1 C1(C(N2C(C)CC(NC(C(C)C3CC3)=O)C2)=O)CCCCC12OCCO2 Cc1cc2ccccc2n1CC1CC2CCC(C1)N2CCC(=O)NC(C)(C)C C1(C(=O)Nc2ccc(CC)o2)(CC)CCCN1C(=O)C=Cc1ccc(C(N)=O)o1 CC1(CNC(=O)Cn2cc(COCC3CCCCC3)nn2)CCCC1(F)F N1(C(c2nn(CC)c(O)c2)=O)CCN(C)C(C(=O)NCC2CC23CCC3)C1 c1(N(C(c2scnc2C)C(=O)Nc2ccc(F)cc2)CCC)cc(C)cc(F)c1 C12OCCC1C(=O)NC2.c1(OC(=O)COCC2CCC2CO)ccccn1 C12C(CCCN1C(c1cc(C)ncn1)=O)C(=O)N2.N(C)(CCSC)CC CCCCC(CC)C(=O)NN(C(c1cccc(CC2CN(C3CC3)C2)n1)=O)C N1(C(c2cn(C(C)(C)C)nc2)C(=O)NCC(F)F)CCCC(F)C1 C(=O)(CS(=O)(=O)CCO)NCCC1(O)CCN(C(CCSC)=O)C1 c1(C(N2CC(CCNC(c3cnc(N(C)C)s3)=O)C2)=O)cccc2cncn12 c1(C(N2CCCC2Cc2ccccn2)=O)cnc(-c2ccsc2)s1 CN1CCC(C(=O)NC2(C3CCCO3)CC2)(NC(C2CC2Cl)=O)C1 C1(C(=O)NCC2(NC(C)=O)CCC2)C2CSCC1CN(C(C1CC1(F)F)=O)C2 N1(Cc2nc(-c3cc(C(=O)OC)sc3)sc2)CC(CO)CC(SC)C1 Cc1c(CNC2CCn3c(cnc3C)C2)sc2ccc(Cl)cc12 c1(CNC2(c3n(CCCCCC)nnn3)CC(C)C2)cnc(OC)c(C)c1 c1(C(N(CCCNC(C(C)(C)OC(C)=O)=O)CCO)=O)ccc(C(C)C)nc1C C1(CNC(C2C(CCOC)C2)=O)CN(C)CCN1C(=O)COCCCCC C1(C(=O)NCC2N(C(C=Cc3c(C)n(C)nc3)=O)CC2)CNC(=O)CC1(C)C C(CCCCCN(C)C(c1ncsc1Br)=O)NC(C1CCC(C)S1)=O Cc1cc(CC(N2CC(=C(F)CNC(=O)Cc3cn[nH]c3)C2)=O)c(O)nc1C C=CC(O)(C(=O)N1CC(CNC(c2cnc3ccoc3c2)=O)C1)C(F)(F)F C1(CNC(c2cnc(CC)o2)=O)(CO)CCN(C(=O)C(C2CCCCC2)C)C1 C1(SC)CCCC1C(N1CC(C(C)NC(c2cnsc2C)=O)C1)=O c1(CC)cccnc1NC(=O)NCC(C)(O)CNC(=O)C(C)(C)C1CCCCO1 c1(C(C(=O)N(CC(C)(C)CNC(C2SCCS2)=O)CC)C)ccccc1OC c1(CC(N2CCCC(N(C(=O)COCC(F)F)CC)C2)=O)ccc(Cl)c(Cl)c1 S(=O)(=O)(c1nc[nH]c1[N+](=O)[O-])NC(CCC)(CCC)CCC N1(C(C2(C)CCCC2)=O)C(C(=O)NCCCCN2CCC2)CCC12CC2 CC1CCCC1(C(=O)NC1CC=CC1)NC(c1ccc[nH]1)=O c1(OCC=C)ccc(C(=O)NCC2(CF)CC2(F)F)cc1OC c1(C(=O)NC2C(NC(C3C(C=C)OCC3)=O)CCC2)nccc2[nH]ccc12 CC(C)CCC(C(=O)N1CC2(CC2)CC1C)NC(=O)COC1CCC1 Cc1nc2cc(C(=O)NC3(CS(C)(=N)=O)COC3)ccc2o1 Cc1cc(Cl)c(Cl)cc1C(N1CC2CN(C(C3(C)CC3C)=O)C2C1)=O c1(CN(CCC)Cc2nc(=O)n(-c3ccccc3)[nH]2)ccc(F)c(C)c1 C=CC(CCC)CC(=O)NC(C(=O)NOCCCN(C)C)C1CCCC1 C1(CC(=O)NC2(CCCNC(CCOCCCOC)=O)CC2)CC2C=CC1CC2 c1(NCCc2ncn(CC)c2)cc(Cl)c(Br)cc1[N+](=O)[O-] CN1C(=O)c2ccccc2C1C(=O)N1CC2CC(NC(c3occc3F)=O)C1C2 C1(C(=O)NC2C3CN(C(C=C(C)Cl)=O)CC2CC3)CC12CCc1ccccc12 C12(C(=O)NCCSC3CC3)COC(C1)C2.c1(NC(C)C(=O)N(C)C)n[nH]c(CO)c1C C1(O)(CC(=O)NCCN(C(C(C)CC2CCC2)=O)CC2CC2)COC(C)(C)C1 C(C(C(=O)NC1CCC1(C)C)C(C)(C)C)NC(c1n(C)ncc1C#N)=O CCCCCC(O)C(=O)NCC1CCN(C(c2ccc3c(c2)NCC3)=O)C(C)C1 c1(C(=O)NCC2C(F)(F)CCN(C(c3cc(C)oc3)=O)C2)cc2cccnc2s1 Cc1ccc(OC)c(OC)c1.C1(C=O)(C(N(C2CC2)C)=O)CCC1.C1(C=O)CC1.C1CC1 C(CC(O)CNC(=O)CCOC1CN(C(=O)C(F)F)C1)OC C1(NC(C(C2CN(C(C(C3CC(C)(C)C3)OC)=O)C2)O)=O)CC(C)(CO)C1 C#Cc1cccc(CC(=O)NC2CN(C(=O)COC3COC3)CC2OC)c1 c1(C(N2CC3C(C(N4CCC(N(C)C)C4)=O)(C3)C2)=O)ccc(Br)c(Cl)c1F c1(C(N=c2cc(OC)[nH][nH]2)=O)cccc([Si](C)(C)C)c1.c12ccc(cn1)[nH]c2=O C1(C(=O)NCC2(CCC)CC2)CN(C(C23CSCC2C3)=O)CC1(C)C c1(C(=O)NC(C2(C(N3CCC(N4CC=CC4)C3)=O)CC2)C)cc(C)c(C)cc1C C(=O)(CC(C)C(F)F)NCC(CCCC)NC(=O)CC1OCCC1C c1(NC(C2(CC)CN(C(=O)CCC3CCC(=O)C3)C2)=O)ccc(OC)cc1C C12(C(=O)NC3CN(C(C(C)CN4CCOCC4)=O)C3)CCCCC1NC(=O)C2 Cc1n[nH]c(C)c1CC(C)C(=O)NC(C)(C)CCNC(=O)C=CC1CCCO1 C(=O)(C(COC)C(F)(F)F)N1C(CNC(C(CCC)O)=O)CC(C(F)(F)F)C1 N1(C(C2(CO)CN(C(C=CC3(C)COC3)=O)C2)=O)CCCCC(CO)C1 Cc1cccc(C(N2CCCC(N(C)C(C3CCCC34CC4)=O)C2)=O)c1F N1(C(CSC(C)C)=O)CCN(C(C2CCCSC2C)=O)CC(C)C1 c1(NC(=O)NCC2(CC(=O)OC)CCCCC2)ccc2c(n1)OCC(=O)N2 c1(C(=O)NC2CC(F)(CNC(C3(C=C)CCCCC3)=O)C2)c(F)ccc(O)c1F C(=O)(CS(=O)(=O)c1ccccc1F)N(CCNC(C(C)C)=O)Cc1ccccc1 c1(CNC(C=C(CC)C)=O)ccc(C(=O)NCCCc2ncco2)nc1 c1(C(N2CC(N(C(C(CC)C)=O)C)C2)=O)ccc(=NCCOC(C)C)[nH]c1 N1(C(c2c(C)nns2)=O)CCC2C(CCCN2C(c2ccnnc2S)=O)C1 C1(C)(CC(=O)NC(C)C(C)NC(c2cnns2)=O)CCCO1 O=C(C1OCCn2ccnc21)NC1(CO)CCN(C(c2ccccn2)=O)C1 c1(C(=O)NCC2C3CN(C(c4n(C)nc(Cl)c4)=O)CC32)cnn2ccn(C)c12 C(CCNC(C1(C)CCC(=O)C1)=O)(C(=O)NCCNS(=O)(=O)C1CC1)OC C1(NC(C(C)NC(N)=O)=O)CCOC12CCN(C(c1cc(Cl)ncc1F)=O)CC2 C1(CNC(CC(CC)O)=O)CCCCN(C(c2cc(C)c[nH]2)=O)C1 c1(CN2C(C)CN(C(=O)Nc3ccccc3)CC2)cc2c(cc1Br)OCCO2 N1(C(COC2(C)CCC2)=O)CCOC(C(=O)NC2CCOCC2(C)C)CC1 N1(C(=O)NCC)CCCCC1c1ncccc1Cl.n1(CC=O)cc(C(=O)O)nn1 C(C(C)(O)CC(=O)N1CCC(C(=O)Nc2cnccc2CO)C1C(C)C)OC C1(NC(C2(CS(C)(=O)=O)CCC2)=O)CN(C(c2c(Cl)csc2Cl)=O)CCC1CO CN1CCN(CC(=O)NC2C=CC(CNC(C3CC=CCO3)=O)C2)CC1 c1(C(N2CCC(C(C)NC(C3C(C(=O)OC)C3)=O)CC2)=O)ccc(C)cc1F C12(CNC(C3N(C)CCOC3)=O)CC(C1)C(NC(=O)CN1C(=O)CNC1=O)CO2 Cc1cc(CNC(C2CCN(Cc3cnc(CCCl)s3)CC2O)=O)cc(C)n1 c1(C(=O)NC2CC(C)(CC)N(C(=O)Cc3cc(C)no3)C2)ccc(F)c(N)c1F C(=O)(C(F)C(C)C)NCC(CN(C(c1c(CCC)n[nH]c1)=O)C)C CN1CCCC(CNC(c2coc(CNC(C3CC3F)=O)n2)=O)C1 N1(C(C2(C)CN(C(C(CC)C#N)=O)C2)=O)Cc2cccc(C#N)c2C1 n1(CC)cnc(C(N2CC(C(C)NC(=O)CCn3ccc(C)n3)C2)=O)n1 C(c1cc(Cl)ccc1Cl)=CC(N1CCCC2(NC(c3c(C)onc3)=O)C1C2)=O C=CCCCCC(=O)NC1(C)CCN(C(C2CC23CCSCC3)=O)C1 C=CCC(C)(C)C(=O)NCc1csc(C(=O)NCCN2CCCCCC2)c1 CCC(C)C(C(=O)NCCCN(C(C12CC(CC(C)O1)C2)=O)C(C)C)NC(C)=O c1(C(=O)NC2C(CC)CN(C(C3CC=CC3)=O)CC2)cc(=O)c2ccccc2o1 c1(OC)nc(C)c(C(=O)NC2(C)CN(C(c3ccn(CCF)n3)=O)C2)s1 Cc1c(C(N2CC(CC(C)NC(=O)C(C)CF)C2)=O)cnn1CC(F)F c1(C(N(C2CCC(NC(=O)C(C)(O)C3CC3)CC2)C)=O)cccc(C2(C)CC2)c1 CC(C)C(CNC(C1CC(OCc2ccccc2)C1)=O)NC(=O)C(C)(C)O C1(NC(c2cncnc2)=O)CN(C(=O)COc2cccnc2)CC(F)(F)C1 C1(NC(C2CN(C)C2)=O)CN(C(c2cncc(-n3ccnc3)n2)=O)CC12CCC2 N1(C(C(CCCC)O)=O)CC2CCC(C1)N2c1cc(C)nc(C(C)CC)n1 C1(c2ncn(C)n2)CCCCN1C(=O)N(CC(c1ccc(Br)cc1)(C)C)CCO C1(NC(CC(CC)O)=O)CCCCN(CCOc2cc(C)cc(C)c2)C1 c1(CN(C(=O)NC(C2CC(F)(F)C2)CC)C2CC2)cn(C)nn1 C1(CNC(=O)CC2CCSCC2)CC2(CCN(C(C34CC(C3)C4)=O)C2)CO1 c1(CC(N2CCC(NC(C3CCCC3)=O)C2)=O)ccc2c(c1)CCCO2 C(C(C(C)(C)C)NC(=O)C(C1CC1)C1CC1)NC(c1c(C)[nH]cc1)=O Cc1c(C(=O)N(C2CC2C(=O)N(C2(C)CC2)C)C)[nH]ccc1=O N1(C(C2N(CC)CCC2)=O)CCC2(CC1)CC2C(=O)NCC1(CO)CC1 N1(C(C2CC(=C)C2)=O)CCC(C)(C)C(C(N2CCN(C(C)C)C(=O)C2)=O)C1 Cc1[nH]nc2c(C(N3CCC(NC(C4CCCOC4)=O)C(F)C3)=O)cccc12 C(CCCC(=O)NC1(C(=O)NCC2COC(C)(C)C2)CCOCC1)N(C)C CC1OC2(CNC(c3cnccc3C(F)F)=O)CC1(NC(c1ccnnc1)=O)C2 C1(NCC)CC(C)N(C(c2csc(Cl)c2OC(Cc2c(CCC)con2)=O)=O)C1 n1(CCC(=O)NC2CCN(C(C3(C(N)=O)CC3)=O)CC2)ccc2cccnc12 n1(CC)ccc2nc(N3CCC(NC(C4CC4(C)C)=O)C(O)C3)ncc12 N1(C(C(CC)(CC)CO)=O)CC2(C1)CN(C(=O)C(CO)OC)CC2CO N1(C(=O)NC(C)C(c2ccccc2)N(C)C)CCCN(CC(O)C(F)(F)F)CC1 C(C(=O)N)(C1=NOCC1)C(C)(C)C.C1(OC)C(C(=O)O)C1C(F)(F)F C(=O)(CCCCC(N)=O)NCC(C)CN(C)C(C1CC2CC1CC2O)=O N1(C(C2=C(C)CC2)=O)CCCC(O)(CNC(=O)CCn2ccc(C)n2)CC1 C1(C(=O)NC2CC(CNC(C3(C#N)CCCO3)=O)C2)CC1C1CCCCC1 C1(N(CC(C)C)CCc2ncc(CC)s2)CCN(CC)CC1 c1(-c2cc(F)c(OCCCC(=O)OC)c(F)c2)c[nH]c2ccc(Br)cc12 c1(C(N2CCC(NC(c3nc(CC)sc3)=O)C(F)C2)=O)c(C)ccc(C)c1C c1(C(=O)NCC(CC(F)(F)F)NC(C(CSC)C)=O)nc2ccccc2[nH]c1=O C(C(O)CN(CN1CCOC(c2ccccc2Cl)C1)OC)OC c1(OC)cc(C(=O)NC(C2CCN(C(c3ccccc3F)=O)C2)C)ccc1Cl C(=O)(CCCCCN=[N+]=[N-])NCCCC(C(=O)O)NC(N1CC(C)(C)C1)=O N1(C(CCCCC#C)=O)CCCC12CCN(C(=O)C(CO)N(C)C)C2 N1(C(CCCOCCC)=O)CCC(NC(=O)C(CC)SC)C12CC2 c1(C(=O)NCCC2(OC)CN(C(c3snc(O)c3Cl)=O)C2)ccc2ccnn2c1 c1(CC)ccc(C(=O)N(C)CCNC(=O)C(Cc2ccccc2)OC)c(C)n1 c1(OC)cc(Br)ccc1CN1CCC2(CC1)CC2.C12CC1CNC2=O c1(C(=O)NCC2CN(C(C3C(C)=CCS3)=O)CC2O)cc(C)n(C2CC2)c1C c1(CSC(C)C(=O)NC(C2(C)CN(C(=O)COCCF)C2)=O)cccc(F)c1 C1(C)(NC(CC2CC(NC(C(CC3CC3)OC)=O)C2)=O)CCC(C)C1 C1(NC(C=Cc2cn(C)nc2)=O)CN(C(=O)Cn2cnnc2O)C2(CCC2)C1 c1(NC(CCC)CCO)ncccc1S(=O)(=O)NCc1cc(Br)ccc1N(C)C N1(C(C=CCC)=O)CCCN(C(=O)C(O)Cc2ccc(Cl)cc2)CCC1 c1(C(=O)NC2CC(CNC(C(C(C)C)(C)O)=O)OCC2)ccc2c(c1)CC(=O)N2 CC(C)(O)C(F)C(=O)Nc1cccc(CNC(C2CC2(Cl)Cl)=O)c1 Cc1cn2ccc(C(=O)NC(C)C(C)NC(c3cc(Cl)cnc3O)=O)cc2n1 c1(OC)ccc(C(N2CCCC(C(=O)Nc3cnc(C)cc3C)CC2)=O)c(F)c1 C(CCC(=O)NO)NC(C(C1CCCN(C(=O)CC2NC(=O)NC2=O)C1)C)=O c1(C(C)N(C)C(C2CC(C(C)(C)O)C2)=O)ccc(F)c(F)c1 c12c(C)noc1C(C(=O)O)OC2=O.c1(CNC(C(CC)SC)=O)ccccc1SC n1(N2CCC(c3nccc(C)n3)CC2)ncc2ccc([N+](=O)[O-])cc12 n1(CCC)ccc(=NC(=O)C2(C)CCCN(C(c3cnc(C4CC4)o3)=O)C2)[nH]1 Cc1noc2cc(C(N3CCN(C(=O)CC4CCOC4)CC4(CC4)C3)=O)ccc12 c1(C(N2CCC(NC(C(CCC#C)O)=O)C2)=O)cc(Br)cc(C)c1C c1(C(NOCC(=C)C)=O)ccc2c(n1)CN(C(C1CCC(OC)CC1)=O)CC2 c1(C(N(CC(C)N(C(Cn2c(C)nnn2)=O)C)C)=O)ccc(O)c(CO)c1 C(=O)(C(O)C(C)(C)C)NCc1cccc(NC(COCCC=C)=O)c1 c1(C(C(F)(F)F)OC(C=CCOC)=O)ccccc1F C(CCCCC(=O)NC1CCN(CCF)C1)NC(C(CCC)OCC)=O C1(NC(CC(CCC)O)=O)CN(C(c2cc(C(N)=O)cc(F)c2)=O)CCC1(C)C c1(CN2CCC(C(C(=O)OC)C)C(OC)C2)c(C)cc(C)nc1OC N1(C(COCC)=O)CCC(C2CC2)C1C(=O)Nc1ccc(C)cc1C C1(NC(=O)Cn2cnnc2)COCCC1NC(=O)C1CC1 c1(C(=O)NCc2nnc(C3CCN(C(C(F)OC)=O)CC3)s2)cc(CO)c(C)o1 N1(C(c2cc(SCC)no2)=O)CCN(C(=O)CNC(=O)C(CC)CC)CC1 N1(C(=O)Nc2ccc(C)s2)CCC(c2ccc(Br)cn2)CC1 CC1CN(C(=O)COc2ccc(Cl)cc2)CC1CCNC(C1CC=CC1)=O N1(C(C(CC#C)CC#C)=O)CCC2CN(C(=O)CCN(C)CC)CC2C1 CN(Cc1nccn1-c1ccccc1)N1CC(CCO)C(O)C1 C1(CNC(c2c(CCC)occ2)=O)COCCN(C(c2cscc2C)=O)C1 Cc1ccc(CN2CCC(NC(=O)Cc3cccc(C)n3)C2)c(Br)c1 CC(CC(=O)Nc1cnsc1)NC(c1csc(O)n1)=O CCCCCCC(F)C(=O)N1CCOCC(CNC(c2ccc(C)cc2C)=O)C1 N1(c2cc(COC)ncn2)CCC(O)(C(=O)N(CC(C2CCCC2)C)C)CC1 c1(C(N2CC3C(C(=O)NCc4cnc(C)nc4)C3C2)=O)ccc(Br)cc1O c1(C(Cc2nc[nH]n2)NCC(CC)SC)cccc(Br)c1 CCC(CC(C)C)C(=O)NCC1CCN(C(C23CC(CN2C2CC2)C3)=O)C1(C)C N1(C(C(CC(F)F)N(C(Cc2c(C#C)cccc2)=O)C)=O)CC2(COC(C)C2)C1 CC(C(CO)NC(c1cc(-c2cccnc2)no1)=O)NC(C1CC=CC1)=O N1(C(=O)C=Cc2ccc(F)cc2)CC2CCCCC2(NC(C2CCCS2)=O)C1 c1(C(=O)NCC(CNC(C2C(C)CN(C)C2)=O)(C)C)coc2cc(O)ccc12 C(CCC(=O)N1CCC(N(C(C2CCCS2)=O)CC)C1)OCC=C.SCC C1(N(CC(C)C)C(C2CC2(C)C)=O)CCN(C(c2ccc(O)nc2)=O)CC1 n1(CC)ncc(I)c1C(=O)NC(c1ccc(Br)cc1)CC(C)O c1(C(=O)NC2(CNC(C34CC(C(C)(C)C)(C3)C4)=O)CCOC2)cnc(O)c(F)c1 C(C(CNC(=O)CCC1CCC(=O)NC1)C(F)(F)F)NC(CC(=O)N(C)C)=O N1(C(C(C)n2ccnc2)=O)CC2CC(NC(=O)COCc3ccncc3)C(C2)C1 c1(C(C(N2C(CN(C(CCC)=O)C)CCC2)=O)C)c(C)n[nH]c1C Cc1ncc(NC(=O)C(C)CN(C)C(c2ccccn2)=O)cc1C#N C1(C(=O)NC2C(C(=O)NCC(N)=O)CCOC2)CCCC12CCC2 C(C)(C(=O)N(C)CC1CCCN1C(c1cn(C2CC2)nn1)=O)(C1CC1)OC C(=O)(C(C)CC(F)(F)F)N(C(CN(C(Cc1c(C)nn(CC)c1C)=O)C)C)C C1(c2cncnc2)(COC(C(CNC(=O)OC(C)(C)C)F)=O)CCOCC1 C1(CC)C(C(=O)NCCCCCOC)CCN1C(c1ccnn1CC)=O CCC(C)(C)C(C)CC(=O)NCC(c1ccc(F)c(F)c1)NC(=O)CCC(F)(F)F CCC(CC(=O)NC(CNC(C1CCN(C2CC2)C1=O)=O)C(C)C)C1CCC1 c1(C(=O)NCC2CCN(C(COCc3ccc(C)cc3)=O)C2)cc(N)c(Cl)cn1 C(=O)(C(C)(C)C(=O)N1CCCC(CC(=O)Nc2cc(Cl)ccc2C(N)=O)C1)OC CC(C)CCCC(=O)N1CCCCC1COC1(Oc2ccccc2F)CC1 c1(C(N2CC(CNS(=O)(=O)CBr)C2)=O)cccc(SC(F)F)c1 Cc1cc(CCC(=O)N(CCCCNC(=O)C(=C2CCCCC2)F)C)cc(C)c1 C(=O)(CCCn1cc(C2CC2C(=O)O)nn1)NCC1(SC)CC1 C1(C(=O)NC2CN(C(C(C)N(C)C)=O)C2)CC2(C1)CC2F C#Cc1ccc(C2CC2C(=O)NCC2(O)CN(C(C3(C(=O)NC)CC3)=O)C2)cc1 C1(C(N2C(c3cccc(C)c3)CCC2)=O)CC2CN(C(C3CC3(F)Cl)=O)CC2C1 C1(NC(c2ccc(CC)c(Cl)c2)=O)CCC2(CCCN(C(=O)CC(F)(F)F)C2)C1 C=CCC(CNC(C1(c2ccccc2)CC1)=O)C(=O)NCC(C)OC C1(C(=O)NC2CCCC2N(C)C)(CC)CCN(C(=O)COCC(C)(C)C)CC1 CC(CC(F)F)CS(=O)(=O)NCc1cn(CC(F)(F)F)c(=O)nc1O CC(O)C(F)(F)C(=O)NC1CCCC1NC(c1csc(-c2cnn(CCO)c2)n1)=O N1(N2C3CCN(C(C=CC(=O)OCC)=O)C3CC2)CC2CC(C1)CS(=O)(=O)C2.OCC N1(C(c2ccc(OC)cc2)=O)CCC2CC1CN2C(=O)CCCC(C)=O c1(C(=O)NC(CN(C(C2CC(F)C(=O)N2)=O)CC)C)cc2c(cc1N)CCCC2 C1(CC(=O)NCCCCSCC)CCCN(C(=O)CC(=O)OC(C)(C)C)CC1 C12(CNC(NC3CCN(CC)C3)=NCC3CCCN3CC)COC(C1)C(O)C2 CC1(c2cccc(F)c2)CN(C2CCC(O)CC2)CC1CO C(C)(C)(CC(C)N=c1[nH]c(N2CC3CCC(C2)O3)nc2ccc(Cl)cc12)OC C(=O)(C1=CCCCC1)NC(C1CCN(C(C2(C)CC(C)(C)C2)=O)CC1)C(C)C CCCCC(C)CCC(=O)NCC1CCCC(N(C)C(c2ocnc2CC)=O)C1 C1(CN(C)C(C2CC2(C)Br)=O)CN(C(c2cccc(=O)o2)=O)CCO1 N1(C(C2C(C(=O)OC)CC2)=O)CCCC(CCNC(c2ccnc(S)c2)=O)CC1 c1(-c2nc(CCSC)nn2CC(F)(F)F)ccnc(Br)c1F Cc1nc(C#N)ccc1C(N1CCC(NC(C2CC23CC3)=O)C(C)C1)=O c1(CC)cccc(C(=O)NC2CCN(C(C3CN(CC)CCO3)=O)C2CC)c1F Cc1cc(CC(=O)NC(C)C(C)NC(c2cnnc(O)c2)=O)no1 N12CC3(C1)CN(CCO3)C(=O)CNC(=O)C=CC2=O.c1(NC2CC2)nccs1 c1(C(=O)NCCCC(C)NC(C2OCCN(C)C2=O)=O)ncn2c1CCCC2 c1(C(N2CCC(C)(CNC(=O)Cn3nnnc3C3CC3)C2)=O)cc(F)ccc1F N1(C(c2c(S(C)(=O)=O)scc2)=O)CC(CO)C2(C1)CN(C(=O)CC1CSC1)C2 CCCS(=O)(=O)C(C)C(=O)N1C2CCC1C(NC(c1cc3nc(C)sc3[nH]1)=O)C2 CS(=O)(=O)C1CC(n2cc(CNC(C(C)(C)C(F)(F)F)=O)nn2)C1 C(=O)(C(C)C(C)NC(=O)Cc1ncccc1F)NCc1nnn(CC)n1 C1(CC(=O)N(C)C(=O)OC(C)(C)C)CCC(O)C1.c12ccc([nH]1)CNC(=O)NC2 C(=O)(C(F)CC(C)(C)C)N(CC(N1CCOC(CCF)C1)=O)CCC c1(C(=O)N(O)Cc2cccc(F)c2Cl)ccc2c(c1)OCC2 N1(C(c2c(C)scc2)=O)CCN(C(=O)Cc2cc(F)cc(F)c2)C2CC12 c1(NC(CC2CC(NC(c3nccc(C)c3)=O)C2)=O)cc(F)c(F)c(F)c1Br Cc1cc(=NC(CC(C)C)c2nc[nH]n2)[nH]c(CNCCCN(C)CCO)n1 CN=c1nc(N2CC3CC3C2)[nH]c(=NCC(F)F)[nH]1.C1CO1.C(=O)N CCCC(C(=O)N1CCC(N(C(c2ocnc2CC)=O)CC)CC1)C(C)C c1(CC)cccc(-c2cccc(OCc3cccc(C)c3)n2)c1 C12(CNC(CCNC(N)=O)=O)CN(C(=O)CCn3cccn3)CC1(CC(N)=O)C2 C1(NC(=O)C(=O)NCC(c2cccs2)O)CCN(CC(F)(F)F)CC1 C12(C(CNC(c3n[nH]cc3Cl)=O)NC(Cc3ccc(C)s3)=O)CCC(CC1)C2 C(=O)(C#CC1(CC)CC1)N1CC(CCNC(c2cc(C(C)=O)oc2C)=O)C(C)C1 C1(NC(CCCC(N)=O)=O)CN(C(C2CC=CC2)=O)CC(F)(F)C1 C1(C(=O)NC(c2ccc(O)cc2)C)CCCCN(C(c2noc(C3CC3)n2)=O)C1 C(CC(=O)N(C)CC1CCN(C)CC1)(C(C)OC)NC(C(C)=C(CC)C)=O C1(CC(=O)NCC(CNC(COC)=O)OC)CC(F)(F)C1 c12cccc(n1)NC2=O.N1(CCOC(CSC(C)(C)C)=O)CCCS1(=O)=O c1(C(N2CC3(CCN3C(=O)C=Cc3cccc(Cl)c3)C2)=O)nnc(O)nc1O N1(C(c2cc(CC)ncc2)=O)CC2CCC1C1CN(C(=O)C=CBr)CC21 C1(NC(C2C(=C)C2)=O)CC2CCC1CN(C(c1c(C(F)(F)F)cc[nH]c1=N)=O)C2 N1(C(=O)Nc2c(C)cc(I)cc2)CC(C(=O)O)C2(CCC2)C1 C1(CC(=O)N(CC(CC)NC(=O)Cc2sc(S)nc2C)CC)CCS(=O)(=O)C1 c1(C(=O)NCC(CNC(=O)CC(C)SC)OC)cnc(O)c(C(C)=NO)c1 c1(CCC)cc(-c2nc(C(C)CC)nn2Cc2ncc(CC)o2)ccc1Br c1(C(N(CCCN(C(CC(CC)C)=O)C)C)=O)nc(C)ccc1C c1(OC)ccc(C(C)(C)CNCCC2CCCCN2C2CC2)cc1 c1(CC(=O)NCC2(F)CC(CNC(C(NOC)=O)=O)C2)cc(C)ccc1C C1(NC(C(C)Cc2cnc[nH]2)=O)CN(C(c2ccccc2F)=O)CC2(CCC2)C1 O=C(O)C#CC(=O)NC1CCN(C(=O)CCc2ccsc2)CC1 Cc1cc(C(N2CC(N(C)C(c3cncc(C4CC4)c3)=O)C(F)C2)=O)c(O)nn1 N1(C(C2CC3CC3N2C(=O)CCN2CCCCC2)=O)CCS(=O)(=O)CC1 N1(C(Cc2cn(CC)nn2)=O)CC(NC(C23CCCC2C3)=O)C(C)C1 n1(CC)nc(C(N2CC(NC(c3cc(C)sn3)=O)C2)=O)c2c1CCOC2 N1(COC)CC(NC(C2CCCN2C(c2cc(CCO)on2)=O)=O)CC1=O C#Cc1cccc(C(N2CC(NC(=O)CC3CCCN(CC)C3)C(O)C2)=O)c1F C=CC(C)(CC)C(=O)N1CC(CNC(c2cn(C(C)(C)C)nc2C)=O)C(C)(C)C1 c1(C(=O)NC(CC(C)NC(=O)CCc2cccc(O)n2)C)cc2c(s1)COCC2 c1(SC)nc(N2CC(NC(c3cc(F)cc(Cl)c3)=O)CC(C)C2)cc(C)n1 c1(OC)ccc(C(=O)NCCN(C(=O)CC(C)SC2CN(C(N)=O)C2)C)cn1 c1(N(CCOC)C)nnc(N2C3CCC2CC3)n1CCSCC(F)(F)Cl N1(C(C(c2ccccc2F)OC)=O)CC=CC(NC(=O)C=C2CCN(C)CC2)C1 C(=O)(C1=C(Cl)CCC1)NCCCCCCN(C(CC(c1cccc(F)c1)C)=O)C N1(C(c2ccc(C(N)=O)[nH]2)=O)CC(O)CCC1C(=O)NCC1CC=CCC1 Cc1nc(CC(=O)NCC(C2CCC2)NC(=O)Cc2cscn2)oc1C N1(C(CCC(C)=O)=O)CCCC(F)(CNC(c2c(Cl)csc2Cl)=O)C1 N1(C(c2c(C)cn(C)c2)=O)CCN(C(=O)CN2CCOC2=O)CC1C(C)(C)C C1(OC)CCCC(NC(C2CCCC2NC(C2COCCN2C2CC2)=O)=O)C1 CCCS(=O)(=O)C(C)C(=O)NC(C)(C)CCNC(c1scc2c1OCCO2)=O N1(C(c2nc(OC)oc2)=O)CCC2(C1)CN(C(c1c(C)n[nH]c1C)=O)CC(C)O2 C(c1cocn1)=CC(=O)NC1CCCC1CNC(=O)C(F)C1CCC1 c1(CNC(C2C(C)C(=O)C2)=O)ccccc1CN(C(=O)COCCCF)C C1(N(C(C(c2cccs2)SC)=O)C)CCCN(C(=O)CC2(C(F)(F)F)CC2)C1 N1(C(C2CCN(C(CCNC(C)=O)=O)CC2O)=O)CC(C)N(C)C(C)C1 C(=O)(C1=CCCSC1)N(CCNC(=O)CCOc1ccc(F)c(Cl)c1)C1CC1 N1(CCC)CCC(c2cn(C3CN(C(c4cc(C)co4)=O)CC3O)nn2)CC1 c12cc(ccc1OC)CNC(=O)C2N(C)C.C1(CSC)CC12CC2(F)F N1(C(C2CN(S(=O)(=O)C(F)F)C2)=O)CC2(CC(NCc3cc(Cl)ccc3O)C2)C1 CCC(C#N)C(=O)NC1CCCC(CC(=O)NCCCn2nccn2)C1 c12ccc(F)c(n1)C(C(=O)N(C)C)N2C1CCCCC1.C1(NC(C)=O)CCCC1 Cc1ccc(C=CC(=O)NCc2c[nH]nc2C(=O)NC(c2nccn2C)C)o1 C1(C)(N(C)CC)CCN(C(=O)CC2CCCN(C(=O)C(C)C3CCCC3)C2)C1 C1(C(=O)NCCCCCNC(C(C)(C)c2cccs2)=O)CCCC(C2CC2)O1 c1(NC(=O)C2=CCCCO2)ccc2cnccc2c1.C12CCCN(CC1F)C2=O C=CC1CN(c2ccc(S(=O)(=O)NC(C)C(OC)OC)s2)CC1O CC1CN(C(C2(S(C)(=O)=O)CCC2)=O)CC1(C)CNC(=O)CN(C)C1CC1 C1(NC(C(CN(CC)CC)F)=O)CCN(C(=O)Cn2ncnn2)C(C)C1 C1(CNC(c2cn(C(C)C)nc2)=O)COCCN1C(c1cccc(Br)c1)=O Cc1cc(C(=O)NCC2(NC(C3C(C)(C)C3(C)C)=O)CCCCC2C)nc(O)n1 Nc1cc(C(=O)N(CCCNC(=O)CC2CC2C2CC2)C2CC2)ccc1Cl CC1CC1C1CC1COC(=O)C(F)CC1CCOC1 N1(C(C2C(C)C2)=O)CCOCC1CNC(C1(C(C)(C)O)CCC1)=O C1(C(N2CCC(OC)C2)=O)CCN(C(=O)C(C)C)CC1C N1(C(C2C(C(N)=O)C2)=O)CCCC(CO)(NC(C2CC3CCC2CC3)=O)C1 C1(NC(c2cc(C)ncc2)=O)CCCC(C(=O)NOC2CCN(C)CC2)CC1 CC1CC=C(C(=O)NCCC2(CNC(C3CCSC(C)C3)=O)CC2)CC1 c1(CCC(=O)NCC2(NC(COCC=C)=O)CCCC2)ccccc1CC CC1CCC(NC(c2coc(C3CC3)n2)=O)CN1C(=O)CC1OCCO1 N1(C(C2(COC)C=CCC2)=O)CCOC2(CCCN(c3ncnc(C)c3Br)C2)C1 Cc1cc(C(N2CCOCC2CNC(=O)CSCC(C)C)=O)c(N)c(Cl)n1 c1(OC)c(F)ccc(F)c1C(N1CCN(C(C2CC2C2CCCC2)=O)C(C)C1)=O c1(CNN(C2CCN(C)CC2)CCOC)ccc(C)cc1.C1(C=O)CC(O)CN1C c1(OC)c(C)cc(C(N2CCC(NC(c3scnc3Cl)=O)C2)=O)cc1C c1(-n2c(-c3ccc(Cl)nc3)nc(C(C)SCC)n2)ccc2c(=O)[nH]ccc2c1 N1(C(c2cc(CC)sn2)=O)CCCOC(CNC(c2nccnc2C(N)=O)=O)C1 C(=O)(CCCC(F)F)N1C(C(C)NC(C(n2ccc(C)n2)C)=O)CCC1 N1(C(C(CC)OC)=O)CCCC(C)(C)C1CNC(C1CC2C=CC1CC2)=O CC(C)C(O)C(=O)NC1CN(C(=O)C(C)(C)CF)CC1C c1(C(N2C(C(=O)NC(CCC)CCC)CCC2C(C)C)=O)cnn2c1CCC2 c1(CSCC)ccccc1C(=O)N(CC(O)CN(C(=O)C(C)n1cccn1)C)C C=CCC(CC)C(=O)NCC1(F)CCC(NC(c2nc(CC)sc2N)=O)C1 C1(C(=O)NC2CC(CCn3cc(CCSCCO)nn3)C2)C2CCC(C2)S1(=O)=O N1(C(C(C)N(C(CC2CC(=C)C2)=O)CCC)=O)CC(F)(F)C1C1CC1 Cc1c(C(N2CC3(CC3C(=O)Nc3cncnc3Cl)C2)=O)cccc1[N+](=O)[O-] C1(CNC(CCN(C)CC)=O)CN(C(=O)C=CCN2CCCC2)CCO1 c1(C(C(N2CCC(CNC(COC(CC)C)=O)C2)=O)C)ccc(F)cc1 C1(NC(C(C)CF)=O)CCC(N(C)C(C2(c3ccc(CO)cc3)CCC2)=O)CC1 C(=O)(CC(CC)C1CC1)NCC1C(CC(=O)NC(C=C)COC)C1 N1(C(C(C)S)=O)CCn2cc(C(=O)NCC#N)nc2C1 c1(C(N2CC(OCC(=O)NCC(CN(C)C)(C)C)C2)=O)cc(Cl)c(F)cc1F c1(C(=O)NC2CC(C)(NC(=O)CC(=O)NCC3CC3)C2)cnn2c1OCC(F)C2 C(CCCCCCO)NC(C1(CCNC(c2cc(OC)ns2)=O)CC1)=O S(=O)(=O)(c1[nH]c(=NCCC(N)=O)ccc1Br)NCc1cccc(N(C)C)c1 N1(C(c2c(Cl)cn(C)n2)=O)CCC2(CCCN(C(=O)CCc3ncnn3C)C2)C1 c1(CCCC(=O)NCC2OCC(CC(=O)O)C2)ccc(F)c(F)c1F C(=O)(CCN(OC)C(=O)Cc1ccccn1)N(C(C)COC)CC=C N1(CCC)CCCC(C(=O)NC2(CF)CCN(C(c3nncn3CC)=O)C2)C1 CC(C(C)NC(=O)N(C)Cc1ccc(Cl)s1)S(C)(=O)=O c1(C(=O)NC(C2CCCN2C(c2nc(O)sc2C)=O)C)c(Cl)nsc1Cl C(=O)(C(C)(C)CCOC)NCC1N(C(c2ccc(OCCCC)cc2)=O)CC1 c1(-c2cccc(C(C)=O)c2)cccc2cc(C(=O)NCC3CCCOC3)sc12 Nc1cc(F)c(CC(=O)NCC2CC2NC(C2(n3nccn3)CC2)=O)cc1F C1(C(N2CC3(C2)CN(C(c2ncc(Cl)nc2Cl)=O)C3)=O)CCC(C2CCCO2)O1 c1(C(=O)NCC2CC3(CN(C(CC(CC)C)=O)C3)C2)cc2cc(Cl)cnc2o1 c1(C(=O)NC(CCO)C2CCC2)cc(Oc2ccccc2Cl)ccn1 C1(NC(C(n2ccc(C)n2)C)=O)CN(C(c2csc(C(F)F)n2)=O)CCC1O N1(c2nc(C)c(F)cn2)CCC2(CC1)CC(C(=O)N=c1cco[nH]1)CO2 Cc1cc(C(=O)NCc2csc(CNC(C3(F)CCCOC3)=O)n2)ccn1 C1(NC(c2cnc(OC)nc2)=O)CN(C(C2(c3ccsc3)CC2)=O)CCC1CO N1(C(c2c(C)ocn2)=O)CC(NC(=O)Cc2ccc3c(c2)OCO3)CC(C)(C)C1 N1(C(C(n2ccc(C)n2)C)=O)CCCC(CN(C)C(c2c(Cl)cnn2C)=O)C1 c1(OC)cncc(C(=O)NC2CCC2CNC(=O)CCCC2CCOCC2)c1C CCN=C(NCc1nn(C)cc1Br)NNC(C1CCCN1C1CCCCC1)=O N1(CC2CCC(=O)O2)CCCC2(CCCCC2)CC1 N1(C(C(C)C)=O)CCCCC1C1CCCN1C(c1c[nH]c(=O)c2ccnn12)=O C1(C(=O)NCCNC(c2cc(F)cnc2O)=O)CC2(CCCCO2)C1 C=CC(CC)CC(=O)NC(c1ccccc1)CNC(=O)C(C1CC1)OC NS(=O)(=O)c1cc(-c2ccc(CN3CCSC3)cc2)c(F)cc1Cl CCC(C)(C)C(O)C(=O)NC(c1ccccc1)CNC(c1ccc(N)cc1C)=O C1(C(=O)NC2(C)CC(NC(=O)C(C3CCC(=O)CC3)F)C2)CCC(F)(F)C1 C(C(C(=O)NCC(C)OC(F)F)C(C)(C)C)NC(C1C(C(C)C)CCO1)=O C1(NC(C2C(NC(C=C(C)C(F)F)=O)COC2)=O)CCN2CCC1C2 C(CC(CC)(CC)NC(C1CC2CC2C1)=O)NC(C(C=C)O)=O Cc1cn2c(n1)C(C(=O)N1CCC(CN(C(=O)C(C(C)C)C(C)C)C)C1)CCC2 c1(CN2CCN(C(C)=O)CC2)ccc(NS(=O)(=O)NCc2ccccc2)cc1 C1(C)(C(=O)NCC2(C)CCCN(CC3CCCO3)C2)CC2CCC(C1)S2 C(N=c1[nH]cnc2cccnc12)C1CCC(NC(c2n[nH]c(CC)c2Cl)=O)C1 N1(C(c2c(Br)cc(OC)s2)=O)CC2CCC2(CNC(C2(SC)CC2)=O)C1 c1(C(N2C(C)CC(NC(c3cc(C)n(C)n3)=O)C2)=O)cccc(F)c1Br C1(C)(NCC)CCN(C(=O)NC2C(NC(CCCOC)=O)C2)C1.c1(OO)ccc(Cl)cc1 C(=O)(C(CC1CCC1)NC(=O)C=C(C)C)N(CC(C1CC1)OCC)C C(CC(=O)N1CCCCC1CCO)(C(F)(F)F)NC(C1(C)COC(=O)N1)=O CCCCC(O)C(=O)NC(CNC(=O)Cc1ccc(F)c(F)c1)CC(C)OC N(C=CC(=O)C(F)(F)F)C(CC1CCN(C(C(c2cccc(O)c2)C)=O)CC1)=O C=C1Cn2c(C(=O)NCC(C)NC(C3(CSC)CCC3)=O)nnc2S1 CC1CCCN(C(=O)C(=O)NC2CN(C)CC2C(F)(F)F)C1.C12(O)CN(C1)C2C c1(C(N2CC(C(C)NC(Cc3c(C)ccc(C)c3)=O)C2)=O)ccc(N)c(Cl)c1O C=C1CC2(C1)CC(C(N1CCCC1CNC(c1ccc(NC(=O)NC)cc1)=O)=O)C2 N1(C(c2c(NC)cccc2)=O)CC(C(=O)NC(CCO)C(C)(C)C)C2(CCC2)C1 CC1CCN(C(=O)Cc2cc(Br)cs2)CC1CNC(=O)CC1OCCO1 Cc1cn2cccc(C(=O)N(C)CCN(C(=O)CCNC(=O)CO)C)c2n1 N1(C(C(CCCCC)O)=O)CC2CN(Cc3cc(OC)cc([N+](=O)[O-])c3)CC2(C)C1 N1(C(C(CCC)C(C)C)=O)CCC2(CNC(c3cccnc3C)=O)CCCCC12 C1(C(N2CC(O)(C(C(=O)NCC(C)O)F)C2)=O)CSCC(=O)N1 CC(C)CC(C(=O)N1CC(F)C(F)C1)ONC(c1ccccc1)=O CC1CC(NC(=O)OC(C)(C)C)CCN1C(c1cnc(N)c(N)c1)=O Cc1onc(Br)c1C(N1CCC(NC(c2nnn(C)c2C)=O)C1)=O C1(NC(c2c(C)scn2)=O)CCN(C(c2cccc(F)n2)=O)C1(C)C c1(C(=O)NC(C)C(C)NC(=O)Cc2ccccc2O)cccnc1O c1(C(=O)NCCOCCC(=O)N(C(C)C(C)C)CC)cc(F)c[nH]1 C1(C(N2CC(C)(NC(c3ccsc3)=O)C2)=O)COc2ccc(F)cc2C1 Cc1ccnc(C(N2CCC2(C)CC(=O)NCC(C)(O)CCO)=O)c1N N1(C(C(=O)N)c2ccco2)CCC2NC(=O)NCC2C1.C(=O)(CCNC(C)=O)OC c1(C(CN(C(=O)C(CNC(=O)CC2(O)CCCC2)N(C)C)C)O)ccccc1 Cc1ncncc1C(N1CCC(NC(=O)COC2CCN(C)CC2)C1C)=O c1(C(N2CC(CNC(C3C(SC)CCC3)=O)C2)=O)nc2n(c1Cl)CCCC2 c1(C(=O)NCCC(=O)NCC2CN(C(COCCOC)=O)C2)ccc(F)c(F)c1 c1(C(=O)NC2C(NC(C(CC=C)CC=C)=O)C2)cnc2c(c1)CCCC2 n1(C(C)C)cc(NC(=O)C(=O)NC2CC3CC3C2)c(C(N)=O)n1 c1(C(=O)NC(CC)(CNC(c2cc(C)n(C(C)C)n2)=O)CC)c(C)cccc1Cl N1(C(C(C2CCC(=O)N2)C)=O)CC(C(=O)NOC2CCOC2)C(C2CC2)C1 C1(NC(Cn2ncc(C)c2)=O)CCC(O)CN(C(c2ccn3nccc3n2)=O)C1 CC1(C(N2CCCC2C(=O)NCCCC2CCCCC2)=O)CC1(F)F N1(C(c2c(CC)cno2)=O)CCN(C(=O)CC2CCCOCC2)CC1CCOC N1(C(C=C(C)Cl)=O)C2CCC1CN(C(c1nn(-c3ccc(F)cc3)cc1C)=O)C2 c1(C(=O)NCC2(NC(C3C4OC(C)(C)OC43)=O)CC2)ccc(Cl)c(N)c1Cl c1(C(=O)NCc2cn(CC(C)NC(=O)C(C)CF)nn2)cccc(CN(C)C)n1 C1(C(N(CCCO)CC#C)=O)CCC(C(C)C)N1C(C1CN(C(C)C)C1)=O Cc1nc2cc(C(=O)NCCC3CCN(C(C4CCCN4C(C)C)=O)C3)[nH]c2s1 CN1CCN(C(C2CCC(NC(=O)CC3CCOC3)CC2)=O)CC1(C)C N1(C(C(CNC(C(C)CC#N)=O)N(C)C)=O)CCC(C)(C#N)C1 c1(SC)cc(NCC2CCN(C(=O)CC3CC=CCC3)CC2C)nc(SC)n1 c1(C(CCO)NC(CNCCSCCOC)=O)ccccc1Cl N1(C(C=CS(C)=O)=O)CCC2(CCC(CNC(c3coc(CO)c3)=O)CC2)CC1 c1(C(=O)NCC2CCCCN2Cc2cccc(Cl)c2F)nccc2[nH]ccc12 c1(C(N2CC(CC(C)NC(c3n(CCOCC)ncc3)=O)C2)=O)ccncc1C Cc1cccc(C)c1C1(C(=O)NC2CN(C(=O)CC3CC(C)C3)CC2C)CC1 c1(C(N2C(C3(NC(C(C)O)=O)CC3)CCCC2)=O)ccc2occc2n1 N1(C(C(N)=O)=O)CCCCC2C1CCCN2C(c1ccc(N)c([N+](=O)[O-])c1)=O C1(C(=O)NCC(C)CNC(=O)C=Cc2ccco2)CCCCN1C(N)=O C(=O)(C1=CC2(CCOC2)C1)N1CCC(C)C1C(=O)NCC1C(C)(C)C1(C)C c1(CNC(C2(SC)CCC2)=O)ccc(CNC(=O)CC2C(=O)NN=C2C)cc1 c1(C(c2nnnn2C2CC2)Nc2cc(C)c(Cl)cc2)ncc2ccccn12 C1(CC(=O)NCC(C)NC(C2(C=C)CCC2)=O)CC(C)(C)C(=O)N1 Cc1ccn2ncc(C(=O)NC3CCC(C)N(C(=O)CC4=CCCCC4)C3)c2n1 C#Cc1cccc(C(N2CCC(CC(=O)N(C)CCCCCC)CC2)=O)c1.C(C)(=O)N c1(C(=O)NC2CC(CO)N(C(=O)CC3(O)CC3)C2)cc(Cl)ccc1C(F)F C(CCC(C)CC(=O)NCCC(O)CNC(c1cn(C2CC2)cn1)=O)=C(C)C c1(C(N2CCN(C(CC(=C)C)=O)C(C)CC2)=O)cnc2nc(Cl)ccc2c1 c1(OCC)cnc(C(=O)NCCCC(C)NC(=O)CN(C)C(=O)OC)cn1 c1(NC(C2C3(CN(C(CC(C)C)=O)C3)C2)=O)cn2nc(Cl)ccc2n1 C(C(C)C)(C(O)C(=O)NC1CCN(C(C2CSCN2C(C)=O)=O)C1)OC CC1CCN(C(=O)C(C)Cn2ccnc2)CCN1C(=O)CC1CC2CC2C1 c1(C(N2CCC(N3C(C(N)=O)CC(O)C3)CC2)=O)cc(Br)cc(F)c1F c1(NC(C2CCC(NC(CC)=O)CC2)=O)cc(Cl)ccc1Br n1(CCSC)nnnc1C(c1n[nH]cc1C)NCC1CCCC1 N1(C(C=Cc2ccc(OCC)cc2)=O)CC2(CC(NC(=O)CNC(N)=O)CO2)C1 c1(CC)cc(C(=O)NCc2nocc2C(N2CCC2(C)COC)=O)no1 c1(C(C)C)noc(CCC(=O)NCC2CC(NC(=O)C=CCN3CCCC3)C2)n1 CC1CCCN(C(=O)CN(C(=O)C=CCONc2ccccc2)CC2CC2)C1CO.O c1(C(=O)NC2CN(C(CC(C)C)=O)CC(F)(F)C2)cc2n[nH]cc2cc1Cl CCCCC(C(=O)N1CCCC1C(C)NC(c1cccc(C)n1)=O)N(C)C C1(C)(CCNC(Cc2nc(NC=O)sc2)=O)CCN(C(C23CC(C#N)(C2)C3)=O)C1 N1(C(CC2CC(C)C2)=O)CCCC2(CC(NC(c3cc(O)nc(Cl)c3)=O)C2)C1 CC(CCNC(c1cnoc1C1CC1)=O)CCNC(c1cccnc1)=O C(CC(C)(C)NC(=O)CCN1CCCC1)=CC(=O)NC1(C(C)O)CCC1 c1(C(=O)NC2(CO)CN(C(Cc3c(C)cccc3)=O)C2)cccc(Cl)c1F c1(C(N)=O)ccc(Cl)c(C(=O)NCC(C2CCOC2)NC(=O)C#CC2CC2)c1 C1(C(C)(C)CNC(=O)Cc2cccnc2)CCCCN1C(c1ccnc(O)c1)=O N1(C(C(=O)NCCC(=C)CNC(=O)C(C)(Cl)Cl)=O)CCC(C)CC1 CC1(C(=O)NC2CN(C(c3cnc(-c4cccs4)o3)=O)C2)CCCCC1(F)F C1(C(=O)NCC(CNC(c2c(C)ccc(C)c2)=O)CO)CCC(F)(F)CC1(C)C c1(C(=O)NCCNC(C(C)CNC(=O)OC(C)(C)C)=O)ncnc2c1CCCC2 C1(C(=O)NCC(C(C)C)NC(CCC#C)=O)CCC=CCCC1 c1(OC)cccc(NC(C2CC2NC(c2cc(Br)cc(F)c2O)=O)=O)c1C#N c1(NC(C2CC(F)CN2C(c2ccnc(Br)c2F)=O)=O)ccc2ncccc2c1 N1(C(C(CC)C#N)=O)CC2OCCN(C(c3cccs3)=O)C2C1 C(=O)(CP(C)(C)=O)N1C(Cc2cn(CC(C)O)nn2)CCC1 O=C(CCCCn1ccnn1)NCC1CCCN1C(c1c(O)noc1C)=O N1(C(Cn2cc[n+](C)c2)=O)CC(OC)C(NC(c2csc(CC(F)F)n2)=O)C1 N1(C(c2cc(C)n(CC#C)c2C)=O)CC2CC1CN(C(c1ccn(CC)n1)=O)C2 C(CCCOC)(C(=O)NC(c1cscn1)C)NC(C(C(=O)OC)OC)=O C1(NC(=O)NCC2CCCOCC2)CC12CCOCC2 Cc1cc(=NC(C)c2nnc(CO)s2)[nH]c(=NCC2CC(F)(F)C(=O)N2)[nH]1 CCC(C)C(O)C(=O)NCC1=CCN(S(=O)(=O)CC2CCOC2)CC1 c1(C(N2CC(N(C(C3CCCCC3NC)=O)C)C2)=O)ccc(Br)c(Cl)c1.CN N1(C(C(CCOC)OC)=O)CC2(CC(C(=O)N(C(C)CO)C)CO2)C1 C1(C(=O)NCCc2cccc(OC)c2)CC12CCN(C1CCOC1(C)C)CC2 c1(SCC(=O)NC2C(N(C(C=CSC)=O)C)CCCC2)ccccc1[N+](=O)[O-] C1(NC(CC(=C=C)C)=O)CCN(C(=O)C(C)NC(C)=O)CC(C)(C)C1 N1(C(CSC)=O)CCC2(CCC(NC(=O)COC3CCN(C)CC3)C2)CC1 C1(CC(N2CC(O)(CCNC(c3cc(OCC)n[nH]3)=O)C2)=O)CCN(C)CC1 C1(C(=O)Nc2c(C)cc(O)nc2)C2CCCC2CN1C(c1ccc(Cl)s1)=O CCCC(CC)C(=O)N1CCCC(CC)(NC(=O)CC(F)(F)F)C1 C(=O)(C1=CCCC1(C)C)NC1CCCC(NC(C(C)Cc2ccc(Cl)cc2)=O)C1 c1(C(=O)NC(CNC(C23CCC(OC)C2C3)=O)(C)CO)ccc2c(c1)nnn2C C1(NC(c2ccccc2)=O)CCN(Cc2cn(-c3cccnc3)nn2)CC1 c1(NC(=O)C=CCN2CCOCC2)cnc(O)c(F)c1.c12ncccc1C(=O)N2 Cc1ccc(F)c(CNCCS(=O)CC(F)(F)F)c1 C(=O)(C(C)CC(=O)NCC1CC1CC(=O)N1CC(C(N)=O)C1)OC N1(C(C(C=C)OC)=O)CC(C2CCCN(C(c3[nH]nnc3C3CC3)=O)C2)C1 C1(C)(C(=O)NCCN(C)C(c2ccc(CO)c(F)c2)=O)CCNC(=O)C1 c1(NC(c2ccc(CNC(c3ccc(F)c(O)c3)=O)cc2)=O)nc(Cl)c(Cl)cc1Cl C1(C(=O)NCC(C)CNC(c2cc(C(F)(F)F)n[nH]2)=O)C(F)(F)C12CC2 N1(C(C2(C)C(CC)CCC2)=O)CC(CN(C(=O)Cc2cncn2C)C)C2(CC2)C1 C1(CNC(c2cnn(CCF)c2)=O)CC2(CCC2)CN1C(=O)CCC(F)(F)F c1(C(N2CCC(CC=C)(NC(C3CCSC3)=O)C2)=O)c(C)nc(C2CC2)nc1O c1(C(=O)NC(CC=C)CNC(c2ccc(Br)o2)=O)nc(C2CC2)ncc1Cl N1(C(C(CCSC)O)=O)CCC2CN(C(c3nn(C)c(C)c3Cl)=O)C2C1 CC(C)CCC(=O)C(=O)NC1(C)CC(C(=O)N(C)Cc2cnn[nH]2)C1 C1(C(N(C)Cc2cc(C)on2)=O)CCCCN(C(=O)COCCN(C)C)C1 CC1CN(C(c2cc(Cl)nnc2O)=O)C(C)CN1C(c1csc2ccncc12)=O c1(C(=O)NC2(CN(C(c3c(C)ccc(OC)c3)=O)C)CC2)ccc(C#N)cc1C C1(NC(CCNC(CC(C)C)=O)=O)CCC(NC(=O)C(F)(F)N2CCCC2)CC1 c1(C(N(C(C(=O)NCC2OCC(C)C2)C)C)=O)cn(C)ccc1=O N1(C(C(C)N=c2[nH]ncs2)=O)CCCC12CCN(C(c1c[nH]cc(Cl)c1=O)=O)CC2 N1(C(CCNC(C)C)=O)CCc2nc(C(N3CCCC(F)(F)C3)=O)ccc2C1 N1(C(C2(C(C)C)COC2)=O)C2CCC1CN(C(=O)CN1CCC(C)(C)C1)CC2 Cc1cc(C(N2CCC(NC(=O)CC3(N4CCCC4)CC3)C2(C)C)=O)cc(O)c1 C#Cc1cncc(C(=O)NC(C)(C(=O)NCc2ccc(OC)o2)C2CCC2)c1 c1(N(C)CC2CCN(C(=O)CC3(C)CCCO3)C2)nc2ccc(O)cc2s1 C(CC(C)C)(C(=O)N1CC2CC2C1C(=O)NCC1CC(C#N)C1)OC c1(C(=O)NCC(CN(C(=O)CSC2CC2)CC)(C)C)cc(C)c(Cl)s1 n1(CC)cc(C(N2CC3C(CNC(C4(C)CC(=O)N(C)C4)=O)C3C2)=O)cn1.CC N=c1nc(NC(N2CCC(c3nnc(S)n3-c3ccccc3)CC2)=O)cc[nH]1 Cc1noc(C)c1-c1cncc(F)c1.c1(C2C(=O)N2)ccc(N(C)C)cc1 CC(CN=[N+]=[N-])NC(=O)CCOCCCNC(=O)C(C)N1CCCC1 C1(NC(C(C)SC)=O)CC2CCC(C1)N2C(c1c(C(F)(F)F)coc1C)=O c1(CNC(c2cc(C)n(C)c2)=O)n[nH]c2c1CN(C(C1(N(C)C)CCC1)=O)CC2 C1(NC(CCCNC(C(C)C2CC2)=O)=O)CC(C)(C)C12CC2 Cc1cc(C(=O)NCC(C)(C)CNC(=O)C=Cc2cscn2)c(F)c(Br)c1 C#Cc1ccccc1CC(=O)NC(C(=O)N1CCC(C)(F)C1)C(C)(C)O C1(CNC2(C(N3C(C(=O)OCC)CC(O)C3)=O)CCCCC2)Cc2nccn2C1 C1(CC(N2CC(OCC(=O)NCC(CC)C)C2)=O)CCC=N1 C1(C(N(CC#C)C(C)C)=O)CCC(NC(c2coc(C)n2)=O)CC1 C1(C(=O)OCC)C2CC1CN(CC(C#N)C1CCOC1)C2 N1(C(C(C2C=CCN2C(c2cc(F)cc(F)c2)=O)C)=O)CC2CCCN2CC1C C=CCC(C(=O)NCC1(CC(=O)OC)CCC1)C(C)C C(=O)(C1=NN(C)C(=O)CC1)N1CC2CCC(NC(C(CCOC)(C)C)=O)(C1)C2 CC1(C(=O)NC(C2CCCC2)CO)CCN(C(C2CC3C=CC2O3)=O)C1 c1(C(=O)NCCN(C(C2(COC(C)C)CC2)=O)C)ccnc(C(F)(F)F)c1 Cc1nn(C)c(C)c1OCC(=O)NCC(O)CCNC(c1csc(S)n1)=O C1(NC(c2cocc2Br)=O)CN(C(=O)CCF)C2(CCCCCC2)C1 C1(CC#C)CCCN(C(c2cc(Br)co2)C(=O)NCc2ccccc2Cl)CC1 c1(C(N(C(C)CNC(c2ccco2)=O)C)=O)cccc(Cl)c1O C(=O)(NNC(=O)CN1CCCCC1c1ccccc1F)c1ccc(C)cc1 C1(NC(C(C)N(CC)CC)=O)CC2CCCC(C1)N2C(=O)Cn1cc(Br)cn1 c1(C(N(C2CCCCC2)CCNCc2cnn(CC)n2)=O)ccc(CF)cc1 N1(C(c2c(OC)nsc2)=O)CCCCC1C1CCCN(C(=O)CCCSC)C1 Cc1c(N(C)CCN2CCOCC2)ncnc1N1CCC(CC2CN(C)C2)C1 C#CC1(NC(=O)CC2(C)CCN(C(=O)C(C)(O)C3CC3)C2)CCC(C)(C)C1 C1(C(C(=O)NCCCC(=O)OCC)N2CCC2c2cccc(Cl)c2)CCC(C)(C)C1 C(=O)(CCC(=O)c1cccc(N)c1)N(CCCNC(C1C(SC)CCC1)=O)C c1(C(N2CCC(N(c3ncncc3F)C)C2)=O)ccc(Cl)cc1 c1(C(N(CCN(C(c2c[nH]c(Br)c2)=O)CC)CC)=O)cc(O)n(CC)n1 c1(SC)cnn2c1CN(S(=O)(=O)Cc1ccc(C)o1)CC2 CCCCC(O)C(C)C(=O)NCCc1cn(C2COCC2C(F)F)nn1 c1(NC(C2N(C(CC3ON=C(CC)C3)=O)CCOC2)=O)nnccc1C C1(CNC(C2CC(CNC(COC(CC)C)=O)C2)=O)CC(C)(C)CO1 N1(CC(=O)N(C)CC2CCN(C(c3[nH]nnc3C3CC3)=O)C2)CCCCCC1=O N1(C(CC(CC)(C)C)=O)CCCCCC(N=c2ccc(C(F)(F)F)n[nH]2)C1 C1(O)(c2cncs2)CCOCC1.C12(CC(F)(F)C1)c1cn(nn1)C(C)C2=O C1(C(N2C(CC(=O)NCCn3cnnn3)CC2)=O)CC2(COCCO2)C1 CC(CC(C)(C)C)C(=O)NC(C1CCCN1c1ncc(I)cn1)(C)C CCCC(C)CC(=O)N1C2CCC1(CNC(c1coc(Cl)n1)=O)CC2 C1(C(F)(F)F)(C(N(CC(O)CNC(=O)C(C)(C)CN(C)C)C)=O)CC2(CCC2)C1 c1(C(C(=O)NC2CCOC2)N(C)Cc2ccccc2CO)cc(Cl)cc(Cl)c1 C1(C(N2CC3C(C(=O)NCC(C)(O)CO)C3C2)=O)CC(=O)CC(=O)N1 c1(C(N(CCC(=O)N(CCCCC)C)CCO)=O)csc(=N)[nH]1 c1(NC(=O)OC)ccc2c(c1)CCN(C(C1CCCC13CC3)=O)C2C CC(C(C)C(=O)NCCn1cc(CO)nn1)NC(=O)C=Cc1ccccc1 CC(C)(C)CC(=O)COC(c1cccc(OC(F)(F)F)c1)=O N1(C(C2(COC)COC2)=O)CCOC(C(=O)N(C2CCCNC2=O)C)CC1 c1(C(c2n(C(CC)C)nnn2)NC(C)(C)CSC)nnn(C)c1C C1(NC(=O)COCC2CCC2)CCN(C(=O)C=Cc2ccsc2)CC1O C1(C(N2CCC(N(C)C(c3cccnc3C(F)F)=O)C2)=O)C2CCC1(C)C2(C)C CC1(C)CC(NC(c2coc(CO)c2)=O)CN(C(C2(C#N)CC2C(F)(F)F)=O)C1 S(=O)(=O)(c1ccsc1C(=O)NC1CCCC12CN(C(c1ccc[nH]1)=O)C2)NC C1(NC(c2cccc(NC(N)=O)c2)=O)CC2(C1)CN(C(C1CCC(=O)O1)=O)C2 C1(CNC(c2c(CC)c[nH]n2)=O)CC(OC)CN1C(c1ccnc(C(C)C)n1)=O c1(C(=O)NC2COCCN(c3nc(C)nc(O)c3C)C2)ccc2ncncc2c1 c1(SC)cc(N2CCC(NC(=O)C(c3cccnc3)C)CC2)nc(SC)n1 c1(-c2nc(NC(C(C3CCC3)OC)=O)sc2)ccc(C)cc1 Cc1cc(NC(C2CCC=CCC2)=O)nc(Br)c1 C1(NC(c2ccc(CC)[nH]2)=O)CN(C(=O)CSC(C)C)Cc2nccn2C1 C1(CC(=O)NC(C)(C)CF)CCCN1C(N)=O C(=O)(C1=CC2(CCOCC2)C1)NC(C)(CNC(C1(C2CC2)CCC1)=O)CO c1(OCCC)cccc(S(=O)(=O)N2CC3(CCN3Cc3ccc(F)nc3F)C2)c1 N1(CC)CC(C)N(C(=O)CCN(C)C(C2(OC)CCCC2)=O)CC1C N1(C(C2CCN(C(C)=O)C2)=O)CCC2C(NC(c3ccoc3)=O)C2C1 c1(OC)cccc(F)c1C(=O)Nc1cnc(N2CCOC(CO)C2)nc1 C1(NC(c2cc(COC)no2)=O)CC2CCC1CN2C(=O)CC(F)(F)C(F)F N1(C(CC(C)OC)=O)CC(SC)C(NC(=O)CSc2nncs2)C1 c1(C(=O)NC(CNC(C(C)(C(C)C)NC(C)=O)=O)CO)oc(S(N)(=O)=O)cc1C c1(NCC=CCNC(c2c(C)nc(CC(C)C)o2)=O)cc(C)nc2ncnn12 C1(CNC(c2c(CC)ocn2)=O)C2CN(C(c3ccnc(OC)c3)=O)CC12 C(=O)(C(CCF)NC(c1ccc(F)cc1)=O)N(CC(=O)OC(C)(C)C)CC N1(CC)CCCOC(CNC(=O)COC2CCOC2)C1 N1(C(c2cc(C(N)=O)sc2)=O)CC2CC1CN2C(=O)C(C1CCCO1)C1CC1 c1(OCc2onc(COC)n2)cccc(OCc2noc(C3CC3)n2)c1 CCCC(C)CNC(C1(NC(c2cc(CO)[nH]n2)=O)CC1)=O c1(OCC(N2CC(O)(C(C)NC(C(C(C)C)C)=O)C2)=O)cc(F)ccc1F CCCCCCC(F)C(=O)NC(C)CNC(c1sc(CC)nc1C)=O n1(CC(N2CC(C)(NC(C3N(C(CCC)=O)CCC3)=O)C2)=O)ncc(C#N)c1N c1(NC(c2c(C)con2)c2nnnn2C(C)C)cc(S(=O)(=O)N(C)C)ccc1Cl N#Cc1cccc(F)c1CC(N1CC(NC(C2CCCO2)=O)CC(F)C1)=O n1(CCSC)nnnc1C(c1cnc(C2CC2)o1)NC1CC(C(N)=O)C1 S(=O)(=O)(c1ccc(=NCCN(C2CCN(C)CC2)C)[nH]c1)NC(CC)C1CCC1 c1(C(=O)NCC(C)(O)CNC(C2CC2c2ccccn2)=O)ccc(CO)nc1 Cc1ccc(NC2CCOC(c3ccccc3)C2)nc1 Cc1cc(C(=O)NCC(C)N(C(=O)C2=COCC2)C)sc1-c1ccc(Cl)cc1 C1(NC(C(C)O)=O)CCC2(CCN(C(c3cnsc3)=O)CC2)C1 C=C1COCCN(C(=O)NC(C)C(=O)NC2CC2)C1 C1(C(=O)NC2CCN(C(COCC)=O)C2C(C)(C)C)CC12CCC(F)(F)CC2 C1(C(=O)NCC(c2ccsc2)C)CCC(C(C)(C)C)O1 CCC(CC(=O)Nc1ccc(O)cc1)NC(=O)CC1CCCC(=O)N1 c1(C(=O)NCC2CC3CN(C(CSCCC)=O)CC32)coc(S(=O)(=O)NC)c1 C1(C(=O)NCCC(CC)(CC)NC(c2nc(Cl)ccc2N)=O)CN2CCCN1CC2 N1(C(Cc2c(C)nc[nH]2)=O)CC2CC(NC(=O)CCn3cnnn3)CC1C2 N(C1c2ccccc2CC1C)C(Cc1ccc(OC)cc1Br)=O C(c1ccccc1F)=CC(=O)NCCCN(C)C(c1cn(C)nn1)=O C1(CNC(C(C)OCCC#C)=O)CCCN(C(=O)Cn2cnc(C#N)n2)CC1 N1(C(c2c(C)ccs2)=O)CCN(C(=O)CNS(=O)(=O)C2CC2)C(CC(F)F)C1 C1(N(C(=O)C=CC2CCCC2)C)CCCCC1NC(c1cncc(C2CC2)c1)=O c1(C(=O)NCC(C)C(=O)NC2CCOCC2F)ccc(C#N)s1 Cc1cc(CN(C)C(C2(CCNC(c3[nH]ccc3C)=O)CC2)=O)cc(F)c1 C12(CNC(C3N(C(=O)OCC)CCC3)=O)CCCC1(CO)C2 CN1CCCC(CNC(=O)C(CC2CCCO2)NC(C2C(C)(C)C2(C)C)=O)C1 Nc1cncnc1C(=O)NCC1(CO)CCN(C(c2ccccn2)=O)C1 c1(C(N2CC(CO)C3(CC3)C2)C(=O)NC(C)(C)C)ccc2ncccc2n1 N1(C(c2ccnn2CC(F)F)C(=O)NCCOC)CCC12CCN(C)C2 CC(C(=O)NC(=O)N(C)CCN(C(c1cccs1)=O)C1CC1)N(C)C CN1CCCC1(C)C(N1CC2C(CNC(c3cncc(C4CC4)n3)=O)C2C1)=O c1(C(C)NC(c2cccnc2Br)C)ccc(F)c(I)c1 C1(NCCOC(C(=O)NCC)C)CC(C(=O)ON(C)C)=NO1 N1(C(C)=O)CCC2CN(C(c3cncc(C4CCOCC4)c3)=O)C2C1.C(F)(F)F C1(CC)CCCN(C(=O)CN2CCOCC2)C1C(=O)N(C)Cc1ccccc1C C1(N(C)C(c2snnc2C2CC2)=O)CCCCC1NC(=O)CCCn1cncn1 Cc1nc(N)cnc1C(=O)NC1CCOCC1NC(=O)CCn1cccn1 CC1CN(C(=O)CNc2nccs2)CCCN1C(C1CC2(CCC2=O)C1)=O c1(CN2CCCC(C(=O)NS(=O)(=O)CC3CCC3)C2)cc([N+](=O)[O-])c(O)cc1O c1(CCC(=O)NC(C2CCOC2)CNC(C=CC(CC)C)=O)nc(C2CC2)no1 C(=O)(C(CCOC(=O)Cc1ccsn1)SC1CC(=C)C1)N(C)CCO c1(CC)cc(C)ccc1NC(C1C(C)CCN1C(c1cnc(C)n1C)=O)=O N1(C(C(C=C)OC)=O)CC(NC(C2CCCOCC2)=O)CC(C)C1 CC(N=c1nc2scnc2c(NCC(CO)C2CC2)[nH]1)c1cc(F)c(F)cc1F C1(NC(Cc2ccc(C)c(Cl)c2)=O)CCC2(CCCN(C(c3cncs3)=O)C2)C1 c1(OCC=C)ccc([N+](=O)[O-])c(C(=O)OC)c1.C1(CC)CNC(=O)N1 C1(NC(c2c(C)c[nH]n2)=O)C2CC(NC(=O)CC3CCCC3C)CC12 c1(C(C)C)ccc(CC(=O)NC2CC(NC(C34CC(C)C3C4)=O)C(O)C2)cc1F C(=O)(C(CCC(C)C)NC(=O)CC1CCSC1)NCCOCC C1(NC(CCC(=O)OC)=O)CN(C(C2CC23CCCCC3)=O)CC(C)(C)C1 C1(CNC(c2nn[nH]c2Cl)=O)CN(C(=O)Cc2cnsc2)CCO1 C1(C(N(CC(COC)C)C)=O)CCN(C(c2cc(OC)cs2)=O)C1(C)C c1(C(=O)NCC2CCC(F)(CNC(c3c(C)n[nH]c3)=O)C2)cccc(F)c1F N1(C(c2c(OC)cc3c(c2)OCO3)=O)CCc2ccc(F)cc2C1C Cc1cc(F)c(N)cc1C(=O)NC(C(C)NC(c1ccc(Cl)c(F)c1)=O)C(C)C c1(CC)nnc(N(CC(C)CNC(=O)C=CC2CCOC2)C)o1 C1(C2CCN(C(=O)C3CC3)C2)CCCCN1C(=O)CC1CCCC1 C1(C)(NC(CCNC(=O)NC)=O)CCN(C(C2CCCCC2)=O)CC1 c1(C(N2CC(C)(NC(=O)CCc3csc(=N)[nH]3)C2)=O)cccn2nnnc12 N1(C(Cc2ccc(OCC)nc2OC)C)C(=O)NC(C2CCCO2)C1=O c1(C(C)C)ccc(C(=O)NCCCN(C(=O)CC2CSC2)C(C)C)cn1 C(=O)(CC1OCc2ccccc21)NC1CC(CNC(c2ccc(C)c(C)c2)=O)C1 Cn1cc(C(=O)NCC2CCCCN2C(c2ccnn2CC#N)=O)c(O)nc1=O C(=O)(C(C)(C)C(=O)NC(CC(F)F)C(=O)NC1C(O)C2CCOC12)N(C)C O=[SH](=O)CCN(CCS(=O)(=O)NCC(F)(F)F)C(CO)CCF S(=O)(=O)(c1ccc(NCc2cc(Cl)ccn2)nc1)NC(c1n[nH]c(=N)s1)C S(=O)(=O)(c1ccc(F)c(F)c1)NC12CC(NC(c3cc(C(F)(F)F)c[nH]3)=O)(C1)C2 C12(NC(c3ccoc3C(F)(F)F)=O)CCC(C1)N(C(C1CC=CCC1)=O)C2 CCC(C(=O)NCC1CCCCN1C(c1cc(F)ccc1F)=O)C(C)O c1(C(=O)NCC(C)SC)cc(=NC(=O)CNC(=O)C(C)(C)C)[nH]n1C N1(C(C(C(CC)O)(F)F)=O)Cc2ccccc2C(NC(=O)COC2CCCC2)C1 c1(C(=O)NCC(c2ccccc2)NC(CCOC)=O)ccc(SC(F)(F)F)nc1 c1(C(=O)NC(CC(C)NC(c2ccccc2O)=O)C)ccc2c(c1)OC(C)(C)O2 c1(OC)ccc(C(=O)N(C2CC(NC(c3c(C(C)C)cccc3C)=O)C2)C)c(O)c1 c1(CCNC(C(COC)NC(=O)C(C)CC2CC2)=O)cn(C)nc1C N1(C(C2CC(NC(c3c(C)oc(CO)c3)=O)C2)=O)CCC(C#N)CC1 CC(C)C(C(=O)NC12CC(CNC(=O)C(C)CC3CCCCC3)(C1)C2)N(C)C c1(C(=O)NC(CC#C)C(=O)N(C(C)CSC)C)cc(C)ccc1F c1(CC(C(N2C(CNC(C(C)=C(CC)C)=O)CCC2)=O)C)cccc(Cl)c1 C1(C(=O)NCC2N(C(C3C(C)CC3)=O)CCC2)CC(C)(C)CO1 C1(C(=O)NCCC(N)=O)CCCC2CN(C(c3cc4cc(C)[nH]c4nc3)=O)CC12 N1(C(C(C(CC)C)O)=O)CC2CCC1C(NC(c1[nH]ccc1C)=O)C2 CCC(C)CCCCC(=O)NC1CCC(CNC(c2cncc(CO)c2)=O)CC1 CCCC(C)CC(=O)N1CCN(C(c2cc(COC)cn2C)=O)CC1COC CC1=C(C(=O)N2CCC(NC(C3CCS(=O)CC3)=O)C(CO)C2)CCC1 C=CCCC(C(=O)NCCC(C)F)NC(=O)CCC(CC)OC c1(NCC(CCCC)NC(=O)CC2(CSC)CC2)nc(C)nc2c(C)csc12 Cn1cc(C(F)=CC(=O)NCCC2CCN(C(C3CC4(CC4)C3)=O)C2)cn1 CC1(C)CN(C(c2ccc(C(F)F)c(Cl)c2)=O)CC1CNC(=O)C1=CCCCC1 N1(C(C(C)OC)=O)CCC(C)C(NC(C2CC3(C2)CC3(F)F)=O)C1 c1(C(N(CC(F)F)CC#C)=O)ccc(CNC(=O)C(F)CC2CCOC2)s1 N1(C(C(C(C)O)N)=O)CC2CCCC2C1C CC1(C)CC1(C)CNC(c1csc(O)n1)c1nnnn1C(C)(C)C C1(CC)CN(C(=O)OC(C)(C)C)C2(CCC2)C1.N1(C(CCN(C)C2CC2)C)CCOCC1 c1(C(CNC2(COC)CC(=O)C2)CO)ccc(OC)c(OC)c1 N1(C(CC2(C=C)CN(C(=O)CC(Cl)Cl)C2)=O)CCOCC(O)C1 c1(C(N2C(C)CN(C(CCCC#C)=O)C(C)C2)=O)c[nH]c2cccc(F)c12 C1(NC(CCCOC(C)=O)=O)CC2CCC1(NC(c1cc(C)n(CCO)n1)=O)C2 N1(c2n(CC(=C)C)c(-c3cc(O)nn3C)nn2)CC(C)OC2(CCCOC2)C1 CS(C)(=O)=Nc1ccc(C(=O)NCCOCCCNc2sccc2C#N)cc1 c1(C(=O)NCC(O)COc2ccccc2)ccc(CO)c(Cl)c1.C12CC(C1)NC2 c1(C(N(CC(C)NC(=O)C(O)C(C)c2ccccc2F)C)=O)ccc(F)cc1N N1(C(c2cccc(Cl)c2C)CC)CC2CCC(C1)N2Cc1ccccc1F C(=O)(C(C)(C)CCCNC(=O)C(C1CC1)OCC)NC(CC#C)CO c1(C(=O)NC(CNC(C(C(C)C)OC)=O)(C)CO)cnc2sc(C)cn12 Cn1cc([N+](=O)[O-])cc1C(N1CC2CCC(C1)C2NC(c1cscn1)=O)=O c1(CC)ccc(CC)c(NC(C23CC(CO2)N(C(=O)CNC(=O)OC)C3)=O)c1 C(CC(C)CC)(C(=O)NCC(CC)CC)NC(C1CC(O)(CC#C)C1)=O c1(C(N2C(C(=O)NCC(=O)OC)CCC2)C(=O)OC)c(Cl)c(C)nn1C Cc1ccc(NC(C2CCOC2CNC(c2nonc2N)=O)=O)c(C)c1O CCCC(C)NC(CC)(C)c1nccs1.C(=O)(CN1CC1)OC N1(C(C(C)SCCCC)=O)CCCC(NCCN(C)C(c2coc(CO)c2)=O)C1 C(=O)(CC(C)CC(F)(F)F)NC(CCN(C(C1CC(C)(C(=O)OC)C1)=O)C)C C1(N(C(c2sccc2Cl)=O)CC)CCCN(C(c2cc(Cl)cs2)=O)CC1 c1(C(=O)NC2CCN(C(C3C(C)C3C)=O)CC2F)nn2cccnc2c1Br C=C(Cl)C(C)(C)C(=O)NCC1(COC)CCN(C(c2ccncc2O)=O)CC1 c1(CN2CC(NC(C(CC)F)=O)CC(C)(C)C2)nc(O)c2c(C)c(C)sc2n1 N1(C(CCOCCNC(c2ccc(C(C)=O)[nH]2)=O)=O)CCOCCC1C1CC1 C1(CNC(=O)NC(CC)C(=O)NC)CN(C(=O)OC(C)(C)C)CC12CCC2 C1(CCCNC(C(C)C2CCC2)=O)CCN(C(=O)C=Cc2cn[nH]c2)CC1 CN1CCCC2C1CCN2C(=O)NCC1COCCN1C c1(OCC)nccc(C(=O)NN2S(=O)(=O)CCC(=O)N3CC(C3)C2)c1F.CC.NC c1(OC)cccc(C(N2CCN(C(=O)C(CO)C(C)C)CC2C(C)C)=O)c1F CCC1CN(CC)CCN(CC(C)O)C1=O.C(=O)(C=COCC)NCC C(=O)(C1=C(C)CCCC1)N.CCCC(C)C(=O)NC(C)Cn1cc(C)nn1 N1(C(c2c(C)cncc2)=O)CCN(C(c2cnn(C3CC3(F)F)c2)=O)C2CCC12 O=S(=O)(c1cccs1)NCC1(O)CCCN(Cc2cc(Cl)ccc2Cl)C1 N1(C(C2CC2F)=O)CCN(C(=O)CC2(CO)CCCC2)C(c2ccc(Cl)cc2)C1 c1(C(N(CCNC(C(n2ccc(C(F)(F)F)n2)C)=O)C)=O)ccc(S(C)(=O)=O)o1 C1(C)(C(=O)OCCN(C(=O)OC)C)CN(C(=O)OC(C)(C)C)CC1(F)F Cc1cc(Br)cc(C)c1C(=O)NCC1CC(NC(=O)Nc2cccc(Cl)c2Cl)C1 Cc1nc(C(=O)NCC2CC23CCS(=O)(=O)CC3)ccc1[N+](=O)[O-] Cc1nnc2n1C(C(=O)N1CC(CNC(=O)CCc3cccc(CO)c3)C1)CC2 N1(C(c2c(C)nc(SC(F)(F)F)s2)=O)CCN(C(C2CC3CC3C2)=O)CC(O)C1 N1(C(C2CN(C(=O)NC)C2)=O)CCC(C)C1CNC(=O)Cc1ccc(OC)nc1 CC1Cc2ccccc2N1C(=O)COCO.N12CC(C3CC3)C(F)(C1)COC2=O c1(CCC(C)NC(=O)NCCNC=O)ccccn1.c1(CC)cccs1 C(=O)(C1CCc2c[nH]nc21)N(CCNC(=O)C(F)(F)CC(C)C)CC C(=O)(C(C)(C)CN(C(=O)CCn1cccn1)C)NCCc1cc(C)on1 c1(C(=O)NCC(C2CCCC2)NC(=O)CC2(O)CCOC2)cc(Cl)c(Cl)s1 c1(C(N2CC(NC(C(C)OCC#C)=O)CC3(C2)CC3)=O)cccc2c1COCC2 c1(C(N(CCC)CCNC(=O)CCCc2ncc(C)o2)=O)ccc(C)c(F)c1F c1(C(N2CC(C=C)C(NC(=O)CCc3cnc[nH]3)C2)=O)cncc2[nH]ccc12 Cc1cccc(C)c1C(=O)NCCC12CCC(C1)N(C(c1ccnc(O)c1)=O)C2 CN1CC2(CCN(C(C3C4CC3N(Cc3ccc(Br)cn3)C4)=O)CC2)C1 C(=O)(CC(C)(C)CC(F)F)N1C2CC(CNC(C(C)OCCCC)=O)C1CC2 C1(NC(c2cnc3ncccn23)=O)CCC2CN(c3nnco3)CC2C1 Cc1cc(=NC(=O)C(=O)NC2CC23CC(NC(=O)CC2CCC2)C3)[nH]o1 CC1CCN(C(c2cnn(CCF)c2)=O)CCN1C(=O)C(F)CC(C)(C)C c1(CC)cc(C(=O)N(C2CCN(C(=O)C(C)NS(C)(=O)=O)C2)CCO)c(C)o1 Nc1c(F)ccc(Cl)c1C(N1CCOCC(CNC(=O)C=CC(N)=O)C1)=O C1(C(=O)NCC(C(=O)NCC(C)OCCO)O)CCC(=O)CC1 C1(C(=O)NCCCCNC(c2n[nH]c3cccnc23)=O)C2CCC3C(C2)CC13 C1(C2(C)CC2)(C(N(CCCCNC(C(CC2CCC2)OC)=O)C)=O)CC1 c1(C(=O)NCC2C(NC(C(C(CC)O)C)=O)CCCC2)c(C)cc(=O)n(C)c1C c1(CCNC(C=C(C)CNC(=O)CC(C)N(C)C)=O)cnc(C)s1 C12(C(N(CC(=C)C)C)=O)CCN(C(=O)CC=C(C)C)CCC1C2 C=CC(C)(CC)C(=O)NCCC1CC(F)(F)CN1C(=O)C=CC(C)(C)C CN=c1nc(C(=O)NCC2CCN(C(c3cc(C)nc(C)c3)=O)C2)cc(C)[nH]1 CCCCS(=O)(=O)CC(=O)NC1CC1CNC(c1cc(OC)n(C)n1)=O C1(NC(CCOC2CN(C(C(C(=O)OC)C)=O)C2)=O)CCC(=O)N(C)C1 c1(C(C)C)ccc(S(=O)(=O)NCC2CC(n3ccnc3)C2)s1 C=CCC(CC=C)C(=O)N1CCC(NC(=O)CCCF)C(CC)C1 C(CNC(=O)Cc1c(C)n[nH]c1C)(C(=O)NOCCC(C)O)OCC N1(C(C2CC(C#N)(OC)C2)=O)CCC(C)C(NC(=O)Cc2cnco2)C1C Cc1ccc2oc(C(=O)N(CC(C)(C(C)C)NC(=O)O)CC3CC34CC4)cc2n1 N1(CCCSCCNC(=O)CNc2cccnc2)CCCC1=O.C(CCO)C(=O)N N1(C(C2CCCC(C)C2)=O)CCOCC(N=c2[nH]ccnc2F)C1 CC12COC(C(=O)NCCC3(O)CN(C(=O)CCCn4cncn4)C3)(C1)C2 c1(OC)cccc2c1OC(C(=O)N(C1CCN(C(=O)C(C)C#N)CC1)CCO)C2 C(=O)(CCS(=O)(=O)N(C)C)NCCC1CC(NC(C=NOC)=O)C1 c1(OC)cc(CNC2(C(N3CCCC3Cc3ccccc3)=O)CCC2)cc(Br)c1 c1(C(N2C(CC(=O)NC(CC)C)CC2)=O)cn(C)c(=O)n1C c1(CC)nccn1C(C)CC(=O)NCCC1CCN(C(c2ncc[nH]2)=O)C1 c1(C(N2CC(CC(C)NC(=O)CC(O)C(C)C)C2)=O)ccc2cnccc2n1 CCC(C)(C)C(O)C(=O)NCCOC(C)(C)CNC(c1nnc(S)n1C)=O c1(CC(=O)NCCN(C(c2ccc3nccn3c2)=O)CC)cc(F)c(N)cc1F Cc1nn2cccnc2c1C(=O)NC(CO)C(C)NC(=O)CN1CCCOC1=O C1(c2cn(-c3c(OCCC)cccc3)nn2)CCCN(C(=O)C2=CCCO2)CC1 CC1(C)C(NC(c2ncc(F)cc2F)=O)CCN1C(=O)CS(=O)(=O)N(C)C N1(C(C(CC)C)=O)CCN(C(c2ccc(C)c(C)n2)=O)C2(CCC2)C1 Cc1cc(CC(=O)OCC(=O)C(C)(C)C)cc(C)c1 C1(NC(c2scc(C)n2)=O)CCC(=O)NC1C1CCCO1 C1(C(=O)NC2CC(NC(C(c3ccc(C)cc3)C)=O)C2)CCOC(=O)CC1 Cc1c(C(=O)NC2CC2C(=O)Nc2ccc(C3CC3)cc2Cl)cccc1F N1(C(c2nc(C)nn2C)=O)CCC2(NC(=O)C(C)OCC(C)C)CCCC12 C(=O)(C1=C(C)OCCC1)N1C(CN(C(CC2CCC(C(C)=O)CC2)=O)C)CCC1 N1(C(C=Cc2n(C)cnc2)=O)CCC2CCC(C1)N2C(=O)CC1CCCCC1 C(CC(C(=O)N(CCCNC(c1ccn(C)n1)=O)C)NC(=O)OC(C)(C)C)SC C1(OC)CC(NC(=O)CC2CC3(CC3)CO2)N(C(=O)COCCOC)C1 c1(NC(c2cnc(-c3ccc(CO)cc3)cn2)=O)cc(F)nc(F)c1 N1(CC)CCC(C(=O)NC2CCC2NC(=O)Cn2nnc(C(C)(C)C)n2)C1 C1(CC#C)(C(=O)N(C2CCN(C(=O)CN3CCCS3(=O)=O)C2)C)CC=CCC1 N1(C(c2csc(C)c2C)=O)CCN(C(=O)C=CCO)C(COc2ccccc2)C1 N1(C(CC(n2c(CC)ncc2)C)=O)CCC2(CC1)OCCC2NC(C12CC1C2)=O C(=O)(C(C)CC(C)(C)C)NCCCCCNC(C(C(C)C)SCC)=O C(C)(CCC(C)(C)O)(c1n(CCC)nnn1)NC1(CC)CCOC1 C(=O)(CC(C)(C)NC(=O)C(C)C1(O)CCC1)NC(CCOCC)C C1(CC(=O)OC)CN(S(=O)(=O)CCCN2CCCC2)CC1(C)C c1(C(N2C(CNC(CC(C)=O)=O)CCC2)=O)cccc(Br)c1OC(F)(F)F Cc1cccc(C(O)C(=O)NC2CCCC2NC(c2sccc2F)=O)c1 C(=O)(C(C#N)=COCC)NC1(CC=C)CCN(C(c2cccc(F)c2OC)=O)C1 Cc1onc(C2CC2)c1C(=O)NCCC1CN(C(C2CCCOCC2)=O)CC1C N1(C(C(c2ccc(Cl)cc2)=O)=O)CCCC(NC(C2(C3CC3)CCCO2)=O)CC1 c1(C(C)(C)C(=O)NCc2cn(CC3CC4(CC4)C3)nn2)cccnc1F S(=O)(=O)(c1c[nH]ccc1=NC1CCCOCC1)NCc1cc(OC(C)C)ncc1 N1(C(C2(C)N(C(c3cccc(C)c3N)=O)CCC2)=O)CCC(=C(F)F)CC1 Cc1ccc(C=CCC(CCC(N2CC(n3cccn3)C2)=O)C)cc1 N1(C(CC2(C=C)CN(C(C3CC3C(N)=O)=O)C2)=O)CC2CCCCC12C N1(CC(=O)NC(CNC(c2c(C)oc(C)c2C)=O)C)C(=O)NC(C)(C2CC2)C1=O C1(NC(C(N2CC(C)OCCC2)=O)=O)CC2(C1)CC1CCC(C2)N1 C1(C(C(=O)NCCCC(=O)OC)N(CC(=O)NCCC#N)C)CCC(C)CC1 c1(CC(N2CC(CNC(C(C(C)C)OC)=O)C2)=O)nn(C)c(=O)c2ccccc12 N1(C(c2nc(Cl)sc2Cl)=O)CCC2(CCCN(C(C3CC4CCC34)=O)C2)CC1 C1(NC(C(C)=C(CC)C)=O)CCCN(C(c2cc(C(=O)OC)n(C)n2)=O)CCC1 c1(CN2CC3C(C(=O)NCCC(C)(C)O)(C3)C2)c(F)c(F)cc(F)c1F C(=O)(C(O)C(F)(F)F)NCC1(CNC(c2ccc(SC)s2)=O)CCOCC1 c1(N2CCC(CNC(Cn3c(C(F)F)cc(C)n3)=O)C2)cc2nnc(C)n2cn1 N1(C(Cc2c(C)con2)=O)CC(N(C)C(C2C(F)(F)C23CCC3)=O)C2(CC2)C1 Cn1cc(C(=O)NCC2(F)CC(NC(C3(C)CCCO3)=O)C2)c2cc(F)ccc12 c12ccc(cc1)C(C)(O)Cn1ccnc1-c1cn(nn1)-c1ccc-2s1.CCOC C1(OC(CC)(C)C)(CNCC(F)(F)COC)CC(C)(C)C1 Cc1c(-c2noc(Cc3cn(CCCN(C)C)nn3)n2)cc(C#N)n1C C=CCCC1C(=O)N1.C(C(C)(C)N(C)CC(C)(C)C)NC(=O)OC(C)(C)C CC(C)C(F)C(=O)N1CCC(C(C)CNC(=O)CN(C)C(c2ccsc2)=O)CC1 N1(C(=O)CSC2CC2)CCCC2(CCN(C(c3csnn3)=O)C2)C1 c1(C(=O)NC2C(SC)CN(C(=O)CC3CSCCS3)C2)ccc2nc(C)[nH]c2n1 N1(C(C(CCC(=O)OCC)OCC(=O)OC)=O)CCc2cc(C#N)ccc2C1 C1(C(N(CC=CC=O)C)=O)CC2(C1)CC21CC1.C1(O)(COC)CCNCC1 C1(CC#C)CCC(C(=O)N(C)CCN(c2ccncn2)C)CC1 c1(C(C)O)ccc(C(N2CC(NC(c3cc(-c4cccs4)on3)=O)C(O)C2)=O)cc1 N1(C(C(C)NC(C)=O)=O)CCOC(CNC(c2cn(CCC(C)C)nc2C)=O)C1 CCC(CC(F)(F)F)C(=O)NCC1CN(C(=O)CCc2cnc[nH]2)CC1O c1(C(N2C(C)CC(NC(C3C(C)(CC)C3)=O)C2)=O)cc(S(N)(=O)=O)co1 C1(O)(C(C)NC(C2CC(OC(F)F)C2)=O)CCN(C(=O)CNC(=O)C(C)(C)C)CC1 N1(C(C2CCC(C)N(C(c3cncn(C)c3=O)=O)C2)=O)C2CCCC1CN(C)C2 CC1(C(N2CCC(C(C)(C)C)(CNC(c3ccoc3)=O)C2)=O)CCC(F)(F)C1 C(=O)(C(C)C(C)C1CCCCC1)N(CCOCCN(C(c1onc(C)n1)=O)C)C Cc1ccnc(C(=O)NC2CCCC2CN(C)C(C2CCC(F)CC2)=O)c1F Cc1cccc(C)c1CC12CC(CNC(=O)C(=O)NC)(C1)C2 CS(=O)(=O)C(CNC(C1(O)CC1)=O)CNC(c1n[nH]c2c1CCC2)=O c1(C(N(C2CN(C(C3(C#N)CCOC3C)=O)C2)C)=O)ccc(=O)n2c1COCC2 c1(CCC(=O)N(CCNC(C2CC(SC)C2)=O)CC2CC2)c(C)n[nH]c1C Cn1cc([N+](=O)[O-])c(=NC2CCN(C(C3CCCCS3(=O)=O)=O)CC23CCC3)[nH]1 N1(C(c2cccc(C)c2O)=O)CCC(C2CC2)(CNC(C2(C)CC=CCO2)=O)C1 C(=O)(C(CC)CCOC)NC(C(N1CCC(N(C)CC)CC1)=O)CCSC N1(C(C2CC(C(=O)OCC)C2)=O)CCC(F)(C(=O)NCc2ccn(C3CC3)n2)C1 c1(OC)nccc2c1CN(C(=O)C(=O)N(c1ccc(S(C)=O)cc1)C)CC2 n1(CC(=O)N(CC(CNC(CC2CC(OC)C2)=O)C)C)sc2ccccc2c1=O C1(C(N(C(CC)CC(=O)NCCn2nc(C)nc2C)C)=O)CC2(C1)CC(C)C2 N1(C(C(COC)N(C)C)=O)CC(C)(C(=O)NCC(C)(O)CO)CC1(C)C c1(SC)ncc(Cl)c(-c2ccc(-c3nccn3CCCn3cccn3)cc2)n1 N1(C(C(C2CCN(C(C(C)(C)OC)=O)C2)C)=O)CCC(O)(CCO)CC1 N1(C(c2c(C)nc[nH]2)=O)CC2(C1)CN(C(c1nc(Cl)sc1Cl)=O)C2 O=C(CC=C(Cl)Cl)N(CCCN(C(c1ccnc(CO)c1)=O)C1CC1)C1CC1 c1(CC(N2CC(NC(C=C(COC)C)=O)C(F)CC2)=O)coc2cc(Cl)ccc12 C1(C(=O)NCC(CNC(C2(C3CC3)CC2)=O)OC)CC=CC(O)C1 CC1CN(C(C2(C)CCCOC2)=O)CC1NC(c1cccc(N)c1)=O C1(C(C(=O)NCC(CNC(c2cc(C)n(C)c2)=O)OC)O)CCCCCC1 c1(SCC(N2C(C(C)O)CCCCC2)=O)nc2c(o1)CCSC2 C1(N(C(COCCC=C)=O)C)CCCN(C(C2CC3CCC2O3)=O)C1 N1(C(CCCCC)=O)CCC(C2(NC(c3ccnc(Cl)c3F)=O)CC2)C1 CC1CCC(NC(C2(C3CCC3)CC2)=O)CN1C(c1cc(F)ccc1Br)=O c1(C(=O)NCCCc2cn(CC3(COC)CCC3)nn2)c(C)[nH]c(C(N)=O)c1C C(CC1CCOCC1)(C(=O)C=O)NC(CN(C(C)=O)CCO)=O.C(CC=C=C)N C1(NC(C2CC23CCOC3)=O)CN(C(c2cc(Br)co2)=O)CC2(CCC2)C1 c1(C(N2CCC(C)C2CNC(=O)C=Cc2ccoc2)=O)cc2ccc(Br)cn2c1 C=CCC(CNC(c1cc(C)cnc1O)=O)C(=O)N1CCC(C(C)(C)C)C1 C1(CNC(C(C)OCC)=O)CC(O)(CNC(c2cscc2OC)=O)C1 c1(C(N(CCC(C)NC(=O)Cc2cccc(Cl)c2)C)=O)cnc2[nH]cncc1-2 CN=S(C)(=O)c1ccc(C(=O)NCC2CN(C(=O)CC(F)F)CC23CCC3)cc1 N1(C(CC2(CS(C)(=O)=O)CC2)=O)CC(F)(CNC(=O)C(F)C2CCOC2)C1 c1(C(N2CCC(CCNC(C(CC(C)C)C)=O)CC2)=O)cccc2c1nnn2C S(=O)(=O)(CC(=O)NCC1CCCCC1NC(=O)CC(C)(F)F)NC(C)(C)C N1(C(C2C(NC(C3CN4CCN3CC4)=O)COC2)=O)CCC2(COC(=O)N2)C1 CC(CNC(=O)Cc1nccn1C)C(=O)NC1(CC2CC2)CCC1 N1(C(C(C)N2CCC2)=O)CC(C)(C)C(NC(=O)CSC(C)C(N)=O)C(C)(C)C1 Cc1nc(C(N2CC(OCCNC(c3ccc(=O)oc3)=O)C2)=O)c(C)o1 N1(C(CSC)=O)CC(OC(C2CSC2)=O)CC1CC(N1CCN(C(C)=O)CC1)=O Cc1c(C(N2CCC(C)(C(=O)NCc3ccc[n+]([O-])c3)CC2)=O)cncc1F c1(OC)cc(C(=O)NCCC2CCN(C(=O)C#CC(C)(C)C)C(C)C2)ccc1F Cc1cc(N)cnc1C(=O)NCC(C)N(C)C(c1ccc(C(C)(C)C)s1)=O C12(C(N(CC(C)(C)CF)C)=O)COCC1CN(C(=O)CCC1CCCCC1)C2 C1(C(N(CCSC)CC)=O)CN(C(C2COCC2(C)C)=O)CC(C)O1 Cc1ccc(Cl)c(C(N2CCN(C(=O)CCC(F)(F)F)CC2CF)=O)c1 c1(OC)ccc(-c2cnc(CC(=O)NCc3cc(I)c[nH]3)nc2)c(C)c1 c1(C(=O)NC2CC(NCCC3CCCCC3)C23CCC3)cn2c(n1)CCCC2 N1(C(CCC(=O)NC)=O)CCC2(NC(=O)CP(C)(C)=O)CCCC12 C(=O)(C(C)C(C)(C)c1ccccc1)NCC(C)N(C(c1c(C)nc[nH]1)=O)C C1(C(=O)NCC2(C)CCN(C(C(C)OCC)=O)CC2)CC1C1CCCCC1 N1(C(c2n[nH]c(C)c2Cl)=O)CC(NC(C2C(F)(F)C23CC3)=O)CC(C)(C)C1 c1(CNc2c(C(=O)NC3CC3)ncc(OC)c2)cc2c(cc1N)CCCC2 c1(OCC(=O)N(CC(C)NC(C2(C(C)C)CCC2)=O)C)ccc(F)c(Cl)c1 C(=O)(C(F)(F)CCn1cc(CN2CC3CC3C2)nn1)N(C(C)(C)C)C1CC1 c1(OCCOC)cc([N+](=O)[O-])c(-c2nc(SC)nn2-c2nccn2C)cc1OC N1(C(c2cc(C)on2)=O)CCCC(NC(C2CCC(C)(F)CC2)=O)C1C C1(CCOC)CN(C(C2C=CCC2)=O)CCN1C(c1ccc(C(N)=O)cc1)=O c1(C(CCC(=O)NCCCNC(C(C(C)SC)O)=O)=O)ccc(F)c(F)c1F N1(C(=O)CSC2CCCCO2)CCCC2C1CCN2C(c1cc(F)ccc1Br)=O N1(C(=O)Cc2cccnc2)CCn2ncc(-c3cnn4c3CCC4)c2C1 CC1(CC(=O)NCC(O)CCNC(=O)Cc2ccccc2Cl)CCCCCC1 CCCCC(C(=O)NC1CN(C(=O)C(C)CC2CCCC2)CCC1C)C(C)C c1(C(N(C2CCN(C(=O)CCc3cccn3C)C2)CC)=O)cnn(CCO)c1 N1(C(C(CC)(F)F)=O)CC(NC(=O)CCc2ccc(OC)cc2F)CC(C)(C)C1 c1(C(C)C(=O)NCC=CCNC(C23CCCC2C3)=O)cccc(C(F)(F)F)c1 N1(C(C2C=CC(NC(=O)CCC(F)(F)F)C2)=O)CC2CCC(O)C(O)C12 N1(C(N2CCCC(C(C)NC(C3CC3C(N)=O)=O)C2)=O)Cc2ccccc2C1=O Nc1cncc(C(=O)NCC2C3CN(C(C4CCCC(O)C4)=O)CC23)c1 C(C(C(C)(C)C)NC(c1c(Cl)n[nH]c1C)=O)NC(C(C)(C)NC(=O)NCC)=O CCN=c1[nH]c(C(=O)NCC2CC(F)(CNC(C3C4COCC34)=O)C2)cs1 c1(CC(=O)NC2(CNC(c3c(CC)c[nH]n3)=O)CCOC2)c[nH]c2ncccc12 N1(C(CCOCCC)=O)CC2N(C(=O)C(C(C)(C)C)C3CCC3)CCC2(C)C1 c1(C(C(=O)NCC(CC)N(C(=O)CC2CCCOC2)C)O)ccnn1C C1(N(C(CCC=C)=O)C)CCC(CNC(c2cncc(-n3cccn3)n2)=O)CC1 C1(NC(C2CCCSS2)=O)CN(c2nnc(C3CCCC3)s2)C2(CCOCC2)C1 C#CC1(O)CC(C(N2CCCCC2CNC(c2oc(SC)cc2C)=O)=O)C1 c1(C(=O)NC2C(C(N(CCN(C)C(=O)OC(C)(C)C)C)=O)C2)cccc(O)c1C C(=O)(C(CC(C)C)C(C)C)NCC1CCN(C(C(C(=C)C)(C)C)=O)CC1(F)F CN1N=CC(CC(=O)NCC(CC2CC2)C(=O)NCC2(CO)CCC2)C1=O CC1(C)CCCCC1=CC(N1CCOC(CNC(C23CCC2C3)=O)C1)=O C1(CNC(CC2(OC)CCC2)=O)CN(C(=O)CNC(=O)C(F)(F)F)CCC1C C(=O)(CCCCC(N)=O)NCCC(C(=O)N(CC(C)SC)C)O Cc1nocc1CC(N1CCC1CNC(=O)C(NC(C)=O)=Cc1cccs1)=O c1(C(=O)NC(CC=C)CNC(C2CC2CC)=O)cc([N+](=O)[O-])ncc1Br c1(C(N2CCCC(C(C)NC(=O)C(C)(F)F)C2)=O)cc2c(nc1O)CCCC2 O=C(CCCCO)NCC#CCNC(=O)CNC(=O)C(F)C1CCCC1 n1(CC)ncn(NC(=O)C2CCC=CC2NC(=O)C(C)C(=O)N(C)C)c1=O N1(C(C(CC)SC)=O)CC2(C(=O)N(C)CC3(C)CCCO3)CCC1CC2 C1(C(F)(F)F)(C(=O)NCCCCNC(c2c(C)non2)=O)CCN(C)C1 Cc1nocc1C(=O)NCC1(O)CN(C(=O)CC(=O)OCCC(C)C)C1 C1(C(N2C(C(C(=O)NC(C(=O)OC)C)(C)C)CCC2)=O)C2CCC(C2)C1C c1(NC(CCC)CCCNC(=O)CCOCCOC)ncc2ncnc-2[nH]1.OCCC O=S(=O)(c1c[nH]ccc1=NC1CCCC(C(F)(F)F)C1)NCC1(CC2CC2)CC1 C(=O)(C(C)CC(F)(F)F)N1CC2(CC(CNC(COCCCC(C)C)=O)C2)C1 C1(NC(CCc2ncn(C)c2)=O)C2CC(NC(c3scnc3C(C)(C)C)=O)CC12 c1(OC)ncc(CN2CCOC(CNC(c3conc3C)=O)C2)cc1Br C(=O)(N1CCCc2nccn21)C1(NC(C(C)n2ccnc2)=O)CCCC1 N1(C(CSCCN(C)C)=O)CCC(CNC(c2cc(C3CC3)on2)=O)C12CCC2 Cc1ccc2nc(C)c(C(=O)NC(CNC(=O)C(C)CC3CCC3)CO)n2c1 n1(NC(c2c(CNC(C(CSCC)C)=O)cccc2)=O)cnc2ccccc12 CCCC(CCC)C(=O)N1CCC(O)(C(C)NC(c2cc(C(F)F)ncn2)=O)C1 Cn1cc(C(=O)NC(C)(CNC(c2cc(C(N)=O)cs2)=O)C2CCC2)ccc1=O c1(C(N2CC(C3(NC(Cc4nc(C)[nH]n4)=O)CC3)C2)=O)cc(Br)ccc1N c1(CCC(N2CCN(C(C)=O)CC2)=O)cc(N)cc(C(F)(F)F)c1C C1(NC(c2cccc(OC)n2)=O)CCOC12CCN(C(=O)C(O)P(C)(C)=O)CC2 c1(SC)cnn(C)c1C(=O)NC(C)CC(C)NC(=O)CCC(N)=O Cc1cc(O)ncc1NC(=O)C(F)C1CC(NC(c2cc[nH]c(=N)n2)=O)C1 CC(C)CC(C(=O)NCC1(C)CC(NC(c2ccc(Cl)c(F)c2F)=O)C1)C(N)=O c1(C(N2CC(N(C(=O)COC(C)C)CCC)C2)=O)cnc2c(C)cccc2c1 c1(C(=O)NCC(C)(CO)NC(C(c2cnn(C)c2)C)=O)cn(C)nc1C(F)F Cc1ccc(C(N2CCC(CC(=O)NCCCN3CCCCC3)C2)=O)n1C CC(C)C(C(=O)N1CCC(C(=O)NCCc2nccc(O)n2)O1)C1CCC1 c1(N2C(C(=O)NCCC(F)(F)F)CCC2)nccc(Br)n1 C1(C2CC2)(N(C(=O)C(O)C2CN(C(=O)CC3CC(=O)C3)C2)C)CC1 C(=O)(C#CC1CCCO1)NC1(CNC(c2ccnc(C)c2C)=O)CCCC1 Cc1cn(C)cc1C(N1CC(NC(C2C(C(=O)O)C2(C)C)=O)C(F)C1)=O CCCCC(=O)N1CSCC1C(=O)N(C)CCc1cccs1 C1(C(N(CC(=O)OC)CC2CC2)=O)CCC(NC(=O)CCCOC(C)C)C1 C(=O)(N=c1[nH]cc(C(F)(F)F)nc1Cl)C1C(C)CN(CCCCCC)C1 C(=O)(CC1=CCOCC1)NCC1C(C(N(C(CF)CF)C)=O)C1 c1(C(N2CC(CNC(C(c3cnn(C)c3)C)=O)OCC2)=O)cc2c(ncn2C)s1 C(=O)(C1=C(C)OCCS1)NCC(CC=C)C(=O)NC1COC(C(F)F)C1 c1(CC2C(CC(=O)NC(CNC(=O)C=C(Cl)Cl)CO)C2(F)F)ccc(F)cc1 Nc1ccc(C(=O)NCC2CC(NC(=O)CCOc3cccc(F)c3)C2)nc1F Cc1cccc(C(=O)NC(C)CC2CCN(C(c3cc(C)n(C)n3)=O)CC2)c1C C1(CNC(c2cn(C)nc2)=O)CCN(C(C2CC(C(C)(C)C)C2)=O)CCC1(F)F C(=O)(C(C)(C(C)C)OC)N1CCC(CCOC)(NC(C23CSCC2C3)=O)C1 C(C(C)CC(=O)NCC1CCN(C(=O)CNC(c2ccco2)=O)CC1)OC C1(CC)COC(CC)CN1C(=O)C(=O)Nc1cccc(OCCC(=O)C2CC2)c1 CC(CCCC(=O)NCCOC(=O)C1CC1)NC(=O)CC1CCCC12CC2 C1(C(=O)NC2(CC=C)CCOC2)C2CC2CN1C(=O)CC1C(C)(C)C1(C)C C1(F)(C(=O)NCCCC2(NC(CN(C)CC)=O)CC2)CCCOC1 c1(CC)nn(C)c(NC(c2ccncc2C)=O)c1NC(C)C C1(CN(C(C=Cc2scc(C)n2)=O)CC)CN(C(=O)OC(C)(C)C)C(C)(C)CO1 c1(C(=O)NCC(CC)NC(C2CCC2CF)=O)cscc1SC N1(C(C=CCN(C)CC)=O)CC(C)CN(C(=O)CCCc2ccccn2)CC1C O=C(C1Cc2ccccc21)NC1CCN(C(c2cc[nH]c2C2CCC2)=O)CC1O c1(CNC(C2CC(=C)CN2Cc2ccc(Cl)nc2)=O)cnc(OC)c(Br)c1 c1(C(=O)NC(CC2CN(C(CCOCC)=O)C2)C)sc(C2CCCOC2)nc1C CCCCC(C(=O)N1CCC(Cn2cc(C3CC4CCCC4C3)nn2)C1)C(=O)O C(=O)(C1CCc2c[nH]nc21)NC1CCN(C(c2n(COC)ncc2)=O)CC(O)C1 c1(C(=O)NCC2C(NC(c3cn(CC)nn3)=O)CC2)ccc2c(c1)C(C)C(C)O2 C(C(C)NC(=O)CCN(C)C(C)=O)(C(C)C)NC(CN(C(=O)OC)C)=O c1(C(N2CC3CC2C3CNC(=O)C(F)(F)CO)=O)ccc2n[nH]cc2n1 CN1N=C(C(=O)N2CCC(CC(=O)NCc3cccc(Br)n3)CC2)CCC1=O N1(C(c2nc(CNC(c3cc(CCOC)on3)=O)oc2)=O)CCOCC1C1CC1 c1(NC(=O)CC2CCN(C(c3ccc([N+](=O)[O-])cc3)=O)C2)cccc2c1CCO2 N1(C(C2CC(C)C2)=O)CCC(O)(CCNC(c2cnccc2OC(C)C)=O)CC1 c1(CCNC(c2nnnn2CC2CCOCC2)C2CCCC2)ncccn1 c1(OC)ncc(C)cc1NC(C1(NC(C2(C)CC3C=CC2C3)=O)CCC1)=O N1(C(c2cccc(CC)c2O)=O)CC2(CC(NC(=O)C(C)=CC3CC3)CO2)C1 Cc1cc(C)c(NC(=O)C(N2CC(C)(C)C2CO)c2cnn(C(F)F)c2)c(C)c1 C(=O)(CCCC(N)C(C)(C)C)NCc1n(CC)cnc1Cl N1(C(C2C(CCC)CCC2)=O)CCC2CCC(NC(=O)CCCCSC)C12 CC12C3C4C1C1C2C3C41C(=O)NSc1ccco1.C12CCN(C1)CC(=O)N2 C1(C(=O)NCC=CCNC(CCC(C)C)=O)CCCc2ccccc2C1 n1(CN)ncc2c1CCCC2NCc1cccc2nsnc12 C1(NC(N(C2CC(CNC(=O)OC(C)(C)C)C2)C)=O)Cc2nccn2C1.N c1(CC)cnccc1C(N1CCC(CC)C1CNC(C1CCCC1(C)C)=O)=O C(CC(F)F)(C(=O)OC)N.C1C(=O)N1.C(=O)(CNC(=O)OCC)NC Cc1ncn(C)c(=O)c1C(=O)NC(C1CCCN1C(C1CC(C)OC(C)C1)=O)C c1(C(N(C(COC)C)C)=O)oc(Cn2cc(C(N3CCSCC3)C)nn2)cc1C C1(C(=O)NC2CCC(NC(Cc3c(C)n[nH]c3)=O)C2)CC1C1(C)COC1 N1(C(C(C(C)C)O)=O)CC2COCCC2(NC(c2ccc(O)c(C(N)=O)c2)=O)C1 C(C)(C(C(C)C)NC(=O)CC1CC2(CC2)C1)NC(Cn1ccc(C)c1)=O c1(OC)ccc(F)cc1C(=O)N(C(C)CNC(C12CC(C1)C2)=O)C Cc1nc(C(=O)N(CCCOCCN(C)C(c2sccc2Cl)=O)C)sc1C c1(C(C)CC(=O)NCCCN(C(C)C(=O)N(C)C)CCO)ccc(F)cc1 C1(NC(c2occ(C)c2)=O)CN(c2nc(C(C)(C)C)ns2)C2CCCCC12 C#Cc1c[nH]nc1C(=O)NC1CC2(C1)CC2C(N1CC(F)C(F)C1)=O C1(OCCC)CCCCC1C(N1CC(N(C)C(c2cnnn2C)=O)C(O)C1)=O C#Cc1ccc(C(=O)NC(C)CNC(c2ccc(COC)s2)=O)cc1Cl C(C(C)(C)CC(=O)NCC1CC1CC(=O)N(C1CC1)C(c1ccccc1)C)OC N1(c2cccc(S(=O)(=O)N3CCC(F)C3)n2)CCCC2(C1)OCc1ccccc12 c1(C(=O)OC)ccc(CN2CCCC2CNC(C2(c3ccccc3)CC2)=O)s1 c1(CNC(C(=O)NC2CCCC(NC(=O)OC)C2)=O)c(C)[nH]c2cccc(Br)c12 N1(C(C(C2CCC2)OC)=O)CC2(C(=O)NCC(C)(C)F)CC1CCO2 S(=O)(=O)(c1ccc(F)c(F)c1F)N1CC(C(=O)NCc2c(O)cccc2F)C1 c1(C(N2CCC(C(=O)Nc3onc(C)c3Br)C2)=O)cc(Cl)cc(Cl)c1Cl C(=O)(C1=C(C)OCCS1)N(C1CCCN(C(c2ncccc2N(C)C)=O)C1)CC C12(NC(C(C)(C)OC(C)C)=O)CC1CN(C(C1CC=CCC1C(F)(F)F)=O)C2 c1(C(=O)NCC(CC=C)NC(=O)C(c2cncn2C)O)cnc(C(F)F)cn1 C=C(C)CC(C(=O)NCc1conc1CC)NC(=O)CC12CCC(CC1)C2 CS(=O)(=O)c1cscc1C(N1CCC(C2(NC(C3CCCO3)=O)CC2)C1)=O C(=O)(C(C)NC(c1ccco1)=O)NCCN(C(=O)C(Br)=C(C)C)CCC N1(C(CCCSC)=O)CCCC(CC)C1C(=O)Nc1cccnc1C(C)C c1(CO)ccc(NC2(c3cc(Cl)ccc3F)CC2)cc1F C1(C(=O)NCCN(C(=O)Cc2csc(C)n2)CC)CCCCC(C)(C)C1 C12(CNC(c3cc(F)ccc3F)=O)CCC(CC1)N(C(=O)C(F)=CCCF)C2 N1(Cc2cn(CC)nc2)CCC2(CCN(C(=O)Cn3ccc(C)cc3=O)CC2)C1 C(=O)(CCCC(C)=O)NCC(CN(C(c1c(CC)cco1)=O)C)O c1(NC(C2OCCN(C(C(=CC3CCCC3)C)=O)C2)=O)c(CO)cccc1C N1(C(C2(CCCC)CCCCC2)=O)CC(NC(=O)CSCC(C)C)CC(F)C1 N1(C(CC)=O)CCC(C)(CNC(=O)CCc2scnc2C)C1 c1(C(=O)NCCN(C(=O)CC2CC(CO)CO2)CC)cccc(C(F)F)n1 N(C(=NCCCCl)NC1CCC(=O)NC1=O)C1(C)CN(C(=O)OC(C)(C)C)C1.C(N)(=O)N N1(CCOC)CC2(CCC(Nc3cc(OCC)cc(F)c3)C2)C1 CCCC(CC)C(=O)NC(c1ccccc1F)CNC(c1cnc(S)[nH]1)=O C(=O)(C#CC1CCOC1)NCC1C(NC(C=CC(=O)OC(C)(C)C)=O)C1 C1(NC(C=CC)=O)CN(C(C2CN(CC)CCO2)=O)CC12CCC2 N1(CCNC(=O)Nc2ccc(Oc3ccccc3Cl)nc2)CC2CCC(C1)O2 c1(CC)sccc1C(=O)NCC(C1CC1)NC(c1cc(-c2ccccc2)on1)=O C1(C(N2CC(CC(C(=O)N(C3CCC(C)C3)C3CC3)F)C2)=O)CCOCC1(C)C C(=O)(C(CO)C(F)(F)F)N(CCCC(=O)Nc1c(COC)csc1)C c1(C23CC(C(N4CCN(C(C)=O)CC4C)=O)C(C2)C3)c2cc(Br)ccc2nn1C N1(C(C(C)(O)C2CC2)=O)CCC2(CCC2)C(NC(C2CCC(F)C2)=O)C1 c1(C(=O)NC2CCC(CNC(Cc3cc(OC)no3)=O)C2)cc(F)c(F)cc1N C1(NC(COC2CN(C(C(C)(F)F)=O)C2)=O)CC2OCCCC12 CC(C)CC(O)C(C)C(=O)NC1CCC(NC(c2ccc(O)c(F)c2F)=O)CC1 c1(OC)ccc(C(N2CC(C)(C)C2C(C)C)=O)c(C(F)(F)F)c1 CC(C)(C)C(O)C(=O)N1CCC(n2cc(CNC(=O)CCC(F)F)nn2)C1 C(CCCCNC(c1[nH]nnc1C1CC1)=O)NC(=O)COC1CCCOC1 C(=O)(C(CO)C(F)(F)F)NC1CCC(CNC(C2CC3CCC(C2)C3)=O)CC1 C1(CC)CCCCC1C(=O)N(CC(C)NC(=O)C(C)(C)C1CCCCC1)C C1(C(=O)Nc2scc(-c3ccc(CC(C)C)cc3)n2)CCN(C2CC2)S1(=O)=O C(=O)(C(C)CCCc1ccccc1)N1CCC(C)(CNC(C=CCCC)=O)C1 C(C(CCN=c1[nH]c(N2CCC(CCCO)C2)nc2c1COC2)C(C)C)OC C(c1cc(Br)ccc1C1CC1)=Cc1ccc(CC=C)s1 CCCCS(=O)(=O)CC(=O)NC1C2CC1N(C(=O)Cn1cc(C(F)(F)F)nn1)C2 c1(NC(C2N(Cc3cccc(OC)c3F)C3C(C2)C3)=O)ccc2nc(O)[nH]c2c1 c1(C(N2CCC(COC)(NC(=O)CNC=O)C2)=O)coc2ccc(Br)cc12 N1(C(c2cnc(CC)o2)=O)CCCC(CC)C1C(=O)NOCC1CCCO1 C(=O)(CCCNC(c1cccnn1)=O)NCCN1C(C)CC1 N1(C(CN(CCC#C)C)=O)CCOC(C(=O)NCC2(C)C=CCCC2)CC1 Cn1cc(CCNC(=O)CC2CCN2C(=O)CCc2cccnc2)cn1 N1(C(c2scc(C)c2)=O)CC(CNC(=O)CCNC(c2ccsc2)=O)C(C)C1 c1(C(=O)NCC2(C(N3CCC(C(C)(C)C)CC3)=O)CC(=C)C2)nc2cccnc2s1 C1(C(N(C)CC2CCCN2C(c2cc[nH]c2)=O)=O)CCc2c(cnn2C)C1 c1(CC)ccc(C)c(NC(=O)C(CC2CC2)NC(C2CC(=O)C2(C)C)=O)c1 C1(=CC(N2CC(CC(C)NC(c3cccc(O)c3Cl)=O)C2)=O)CN2CCC1CC2 C1(F)(C(N(C)CC2N(C(c3c(C)cns3)=O)CCC2)=O)CCS(=O)(=O)C1 C1(C(=O)NCCN(CCCCCC)C(=O)CC(F)F)CCC(CCC)CC1 N1(C(c2cc(Br)cs2)C(=O)NCC(=C)C)CCC(CN(C)C)CC1C CC1CN(C(C2CC(C)(C)C2)=O)CC2(CCN(C(=O)C(O)c3ccsc3)C2)O1 CSC1=C(C(=O)NC(C)(C)CCNC(=O)Cc2c(C)noc2C)CCCC1 CC1(C)CC(NC(C2(C)CCCNC2=O)=O)CCN(C(=O)COC2CCCC2)C1 CC(=O)CCN=C(NCC1SCCS1)N1CCN(c2nnc(C)c(C)n2)CC1 CC(=O)CCCC(=O)NCCC1CC(NC(c2cn3c(n2)SCC3)=O)C1 C1(NC(c2cc(C(C)(F)F)ncc2)=O)CN(C(C2CC2F)=O)CC12CC2 N1(C(C(CC#C)C)=O)CCN(C(c2ccnn2C=C)=O)CC1c1ccncc1 N1(C(c2cocn2)=O)CCN(C(=O)Cc2cncnc2O)C2CCCCC2C1 N1(C(C=CC(C)C)=O)CC(NC(C23CC(CN2C2CC2)C3)=O)CC12CCCCC2 N1(C(CC2(OC)CN(C(=O)CSC(C)(C)C)C2)=O)CC2(C=CCO2)C1 C(=O)(C(C)(CNC(=O)COCCN(C)C)CC)N1CCN(CCC)CC1 N1(C(c2ccc(C#C)c(F)c2)=O)CCCC2CN(C(c3scnc3Cl)=O)CCC12 N1(c2ccnc(C)n2)CCc2sc(C(=O)NCCc3ccc(Br)cc3)cc2C1 N1(C(c2cccc(C)c2)=O)CC2CCCC2(NC(c2nc(C)nn2C)=O)C1 c1(C(=O)NC2C(CNC(C(C)NC(CC)=O)=O)CC2)cnn2c1NCCC2 c1(N2CC3N(C(C4(C)CCCOC4)=O)C(CC3)C2)nc2c(cc1C#N)CCOC2 CC1OC2(C(N3CC4CC4(NC(c4ccc5c[nH]nc5n4)=O)C3)=O)CCC1CC2 N1(C(C2CC(NC(CC(C(C)C)C)=O)C2)=O)CC(C)OC(C)(C)C1C Cc1ccc2nc(C(N3CCN(C(=O)Cc4occc4C)C(CO)C3)=O)cn2c1 C1(SCC)CCC(C(=O)NCCCCCCNC(c2nocc2C(C)C)=O)CC1 c1(C(=O)NCC(CCCC)NC(C2(S(C)(=O)=O)CCC2)=O)cc(C)c(O)c(N)c1 C1(N(CC=C)C(=O)NC2(c3ccccc3C)CCC2)CCC2COC1O2 c1(C(C)C)ncc(Cl)c(C(=O)NCCCC(C)NC(c2ncncc2F)=O)n1 c1(C(=O)NCC2CCN2C(=O)CC2C=CCC2)cccc(N2CCOC2=O)c1 CC1CCCCCCN1C(C1CC2CCC1N2C(C1(CCF)CCC1)=O)=O C1(C)(CNC(CC2N(C(CN(c3ccsc3)C)=O)CC2)=O)CC=CCC1 C1(NC(CCC#C)=O)CCN(C(C2CC(c3ccc(Cl)cc3)C2)=O)CC1F c1(C(N(CC)CC2CCN(C(=O)CC3C=CCCC3)CC2)=O)cnc(O)c(F)c1 Cc1cc(C#N)nc(Nc2cnc(Cl)cc2C(N2CCC(CO)C2)=O)n1 N1(C(c2sc(C(=O)OC)c(C)c2)=O)CCCC2CN(C(C3CCSC3)=O)CCC12 C1(C#CC(=O)NCCOC2CN(C(c3cc(C(F)F)[nH]n3)=O)C2)(CC)CC1 C1(CNC(COCCOC)=O)CN(C(C2CC2Oc2ccsc2)=O)CCCO1 c1(CC(C)NC(=O)NC(CCCC)CC)cccc2sccc12 N12CC3(CCCC3CC1=O)C2.c1(CNc2c(C)non2)ccc(Br)cc1F c1(C(N2CC(CNC(c3cccc(SC(C)(C)C)c3)=O)C2)=O)cc(F)cc(F)c1 N1(C(c2c(OC)nsc2OC)=O)CCC(CNC(C2CC2F)=O)C(F)(F)C1 C#CC1CN(C(C2CCN(C(c3cc(C)sc3C)=O)C2)=O)CCO1 c1(C(=O)OCC(=O)Nc2ccc(N(C)C)cc2)cc(Cl)cc(F)c1Br c1(C(N2CCN(C3CN(C(=O)CN4CCC4)C3)CC2)=O)ccc(O)c(CO)c1 C1(CNC(C=CC=CC)=O)CN(C(c2cc(F)c(F)cc2F)=O)CCC1(F)F CC1CC(NC(N2CCCC2)=O)CN1CC(N1CCC1c1ccsc1)=O CC1(C)OCCC1NC(C1CC(CCNC(=O)CCN2CCCC2)C1)=O C1(C(=O)OC)CCCN(C(C)C(N2CC(CO)(Nc3ccccc3OC)C2)=O)C1 O=C1NCC(C(=O)N(C2(C(=O)NC3CC3C(F)F)CCC2)C2CC2)N1 C=C(C)CCCC(=O)N1CC(CC(N2CCC(OC)C2(C)C)=O)C2(CC2)C1 N1(c2ccnc(C(C)C)n2)CCC(NC(=O)C(C)NC(c2ccco2)=O)C(C)C1 C1(CC(=O)NC(C2(O)CN(C(Cc3cn(CC)nc3)=O)C2)C)COCC(C)(C)O1 C(=O)(C(F)(CNC(c1cnn(C)c(=O)c1)=O)C(C)C)NC(CC=C)(C)C C(=O)(CCCN=[N+]=[N-])N(C1CCC(NC(=O)C(C)(C)N(C)C)CC1)C Cc1cccc(CC2(C(=O)NC(C)CNC(c3cscc3Cl)=O)CCC2)c1 C1(O)(CNC(CCSCC)=O)CCCN(C(=O)C(Cl)=CCl)CC1 c1(CC(=O)NCCCNC(C2N(CCC)CCCC2)=O)cc(F)ccc1Cl CSC1=C(C(=O)N2CCC(NC(=O)CC3CCC(O)C3)C2C)CCCC1 C1(C(N2C(C(=O)NCCC3ON=C(C)C3)CCC2)=O)CCCCC1(C)C CC1CN(C(C23CCC(C2)C3(C)C)=O)CCN1C(c1cn2c(n1)CCC2)=O N(C(=NCC1CCC2(CC2)C1)NC1CCOCC1)CC(C=C)(F)F Cc1ccc(C=CC(N2CCN(C(=O)CCCCCF)C(C3CC3)C2)=O)cc1 NS(=O)(=O)c1ccc(C(=O)NCC2CC2CNC(=O)C=Cc2cscn2)c(C)c1 C(=O)(C(C)(C)CC(=O)NC12CC1CN(C(c1ccc(C)c(Cl)c1)=O)C2)OCC C1(CNC(C2(OC)CCOCC2)=O)CCCC2(CN(C(=O)Cn3cccc3)C2)O1 c1(CNC(C2CC(F)CN(C(c3sccc3Cl)=O)C2)=O)ccc(CO)cc1F N1(CC(=O)N(C)C)CCCC(O)(C(=O)Nc2ccccc2C(F)(F)F)CC1 c1(C(N(CCN(C(=O)C(C)NC2CCC2)C(C)C)C)=O)ccc(Cl)c(O)c1 CC1(C)CCOC1C(=O)NC1CCN(C(=O)C(=O)NCC2CC2)C1 C1(C(=O)NCCCCN2CCC2)CCC(C2CC2)N1C(c1cccnc1O)=O CC(C)C(CNC(C1CCCCCC1)=O)C(=O)NCCN1CCCC1 CCC(C)(CNC(c1cc(OC)ns1)=O)C(=O)NCCN(C)C1CC1 N1(C(C2CC(NC(c3cc(C(C)=O)[nH]n3)=O)C(O)C2)=O)CCCCC(C)(C)C1 CC1CC2CN(C(=O)CCc3ncc(F)cn3)CC2N1C(C1CC2C=CC1CC2)=O N1(C(=O)NCC(CC)NC(=O)OC(C)(C)C)CC(C)(C)OC2CCCC12 C(=O)(C(C)CS(C)(=O)=O)NCC12N(C(C3CCC(CC)O3)=O)C(CC1)CC2 N1(C(C2C(=C)C2C(=O)OC)=O)CCC(C(=O)NC(C)C(=O)NCC(C)C)C1 C1(NC(C2CC3(C2)CC3(F)F)=O)CCCN(C(c2cccnc2C(F)F)=O)CC1 N1(C(C(CC=C)(C)O)=O)CC2(C=C(C(=O)NCC(C)CC(F)(F)F)CO2)C1 C1(C)(C(=O)NCC2CCN(C(CC)=O)C2)CCN(C(c2cnc(C)o2)=O)C1 O=C1NCCN(C(c2cncc(Cl)c2Cl)=O)C1c1cn(C2(CO)CC2)nn1 Cc1snc2sc(C(N3CC(C)(NC(=O)CC4COCCO4)C3)=O)cc12 C1(NC(CSCC#C)=O)CN(C(c2coc3c2CS(=O)(=O)C3)=O)C2(CCCC2)C1 c1(SCCCC)cccc(C(N2CC(O)CC2CNC(=O)CCS(C)=O)=O)c1 N1(C(CC(C(=O)OC)C)=O)CC(NC(=O)CN(C)C2CC2)C(S(C)(=O)=O)C1 c1(C(=O)NC2CC(C)N(C(c3ccc(-c4cccs4)[nH]3)=O)C2)cc2n(n1)CCO2 c1(C(N2C(CNC(C(CC)=CC)=O)CC2)=O)ccc(F)c(C(C)(C)F)c1 C1(NC(c2cnc3n2CCCC3)=O)CCC2(CC1)CN(C(=O)COCC1CC1)C2 C=CC1(C(=O)NCC2C3CN(c4ccnc(CCC(C)C)n4)CC23)CCCCC1 c1(C(=O)NC2CC(NC(C3(C)CC3(F)F)=O)C2)ccc(-c2cncnc2)cc1F C1(C(=O)OC2C(=C)OCC2)CC(=O)N(CCc2ccccc2)C1 C=CC(CCC)CC(=O)NCC12CC(NC(=O)CCNC(=O)C=CCl)(C1)C(C)O2 O=C(C1=NOCC1)NCC(C1CCOC1)NC(=O)CC1CC1 C(C(C)(C)CCO)NC(C(C1CN(C(C2OCCC2C)=O)C1)OC)=O CN1CC(NC(C23CC(CN2C(C2CCCS2)=O)C3)=O)C2(CC2)C1 C1(N(C(C2CC(C)C2)=O)C)CN(C(=O)CCC(=O)N2CCOCC2)CC1(C)C c1(C(N2CC3(CN(C(c4c(CC)c[nH]c4)=O)C3)C2)=O)cc2ccccc2[nH]1 C1(C(=O)NCC(CC2CC2)CO)(CC)CCN(C(c2cscc2C)=O)CC1 c1(C(N2CCC(N(C(C3C(C=C)CC3)=O)C)CC2)=O)ccc(C)c(F)c1 N1(C(C(CCN(C)C)O)=O)CC(NC(=O)CCc2cnc[nH]2)CC(O)C1 C1(C(N2CC(OC)C(C(=O)NC34CCCC3C4)C2)=O)CC(C2CC2)=NO1 C=C(Cl)CC(C(=O)NCc1cc(C)ns1)NC(=O)C(c1cnn(C)c1)O c1(C(=O)NC2C(NC(c3coc(Cl)c3)=O)CCOC2)cc(C2CC2)ccc1O C1(CC)CC(NC(=O)NC(c2ccc(C(C)(C)C)cc2)N2CCCC2=O)CC1O N1(Cc2c(C=C)ccs2)CCC2(CCN(Cc3cc(OC)cc(OC)c3)C2)C1 C(=O)(C1COc2ccccc21)N(C(CNC(c1c(C)nccc1)=O)C)C c1(NC(=O)NCC(C)Oc2ccccc2Br)cccc(Br)c1Cl CCC(C)CCCCC(=O)N1CCC(NC(c2cccc(F)n2)=O)C(C)(C)C1 c1(C(=O)NC2CCCN(C(CCS(C)=O)=O)C2)ccc(C(F)(F)F)nc1N Cn1nccc1C=CC(=O)NCC(C1CC1)NC(C1CC2CCCC12)=O N1(C(c2c(C)scc2)=O)CC2ON=C(CNC(COCc3cnns3)=O)C2C1 c1(C(N2CC(SC)C(NC(C3CC3[N+](=O)[O-])=O)C2)=O)cnc2cc(O)ccc2c1 C12(C(N3C(CNC(=O)C(=O)N(C)C)CC(OC)C3)=O)CCC(C(F)F)(CC1)C2 c1(OC)ccc2cc(C(=O)NC(C)CC(C)NC(=O)CC(O)CN(C)C)[nH]c2c1 N1(CCCC)CCC2(CC1)OCCc1cc(C(=O)NCCNC(C)COC)sc12 c1(N(C)C)ccc(C(=O)NCC2(NC(=O)CN3CC4CC4C3)CCOC2)cc1 C=C(C)CC(C(=O)N1CCN(C(=O)Cc2conc2C)C(CC2CC2)C1)OC C1(CNC(C(C)=CC)=O)(OC)CCN(C(c2cnc(-c3ccncc3)s2)=O)C1 C1(C(N2CC(OC)C(F)C2)=O)CCCN(Cc2cc(O)cc(F)c2)CC1 Cc1c(C(N2CC(N(C(=O)C(N3CCCC3)C3CC3)C)C2)=O)ccc(F)c1F c1(C(=O)NCC(CN(C)C(C2CCCN2C)=O)O)ccc([N+](=O)[O-])c(Cl)c1 c1(C(=O)NC(C2CCN(C(c3c(C)cncc3)=O)CC2)C)ccnc2[nH]cnc12 N1(NCc2[nH]nc(C(C)C)n2)CC2CCCN(C(c3csc4nccn34)=O)C2C1 N1(C(c2cn(CCC)nc2)=O)CC2(CCC(CNC(=O)CN(C)C)O2)C1 N1(C(C(N2CCC(O)CC2)C)=O)CCC(NC(=O)CC(O)C2CC2)CC1C C1(NC(c2n(CCSC)nnn2)c2nc[nH]n2)COc2cc(C)ccc2C1 c1(C(=O)NC2CN(C(CN(C(C)=O)C)=O)CC(C)C2)cnn2ccn(C)c12 C1(COC)CCC(C(=O)NCCN(C)C(=O)C2CC2)C1 c1(N(C(CCC(C)=O)=O)c2ncccn2)cnc2c(c1)CNCC2 c1(SC)cccc(N2CC3CC(NC(C4(S(N)(=O)=O)CC4)=O)CC3C2)c1[N+](=O)[O-] C1(CNC(C(C)OCC)=O)CCCC2CN(C(=O)Cc3nc(C)no3)CC12 Cn1cnc2cc(C(=O)NC3(C)CCC(NC(=O)C(O)C(C)(C)C)CC3)ccc12 CC(C)(CC(=O)NCCN1CCCN(C(C2CCC23CCCO3)=O)CC1)C(F)F C=CCC(C)C(=O)N(CCCN(C)C(c1cccc(OC(C)C)n1)=O)C c1(C(=O)NC2CN(C(CC=CC)=O)CC2C)cc(C2CC2)nc2c1c(O)nn2C C1(OCCOCC)CN(C(=NCCSC)NCC2COC3(CCCC3)O2)C1 CCCCC(F)C(=O)N1CCN(C(=O)CNC(c2cc(SC)c(C)o2)=O)CC1 C(=O)(CC(C)C(=O)NC1CCCC1C(N1CC(C)(C)C1C1CC1)=O)OC c1(C(C)CC(=O)NCC2(NC(=O)CN3CCC(C)C3)CCCC2)ccc(F)cc1 O=C(CCCC(F)(F)CO)NC1CCCN(C(c2cc3c(nn2)CCCO3)=O)C1 c1(NC(CCC(=O)NC(C2CN(C(=O)CC(F)(F)F)C2)C)=O)cccc(F)c1 c1(N2CCC(NC(CCCOC(C)C)=O)(CF)C2)ncnc2[nH]ccc12 N1(C(CNS(CC)(=O)=O)=O)CCN(C(=O)CNC(=O)NC)CC1CC1CC1 Cc1cc(=NC(=O)C23CCC2CN(C(c2ccc4cnc(C)n4c2)=O)C3)[nH]n1C C(=O)(C(C)(C)F)N(CCN(C(C(C)OCCC=C)=O)C)C Cc1cc(=NC2CCN(C(c3cn(C)nc3C(F)F)=O)CC2C)[nH]c(C(C)(C)C)n1 C1(F)(C(=O)NCC#CC(=O)Nc2cnn(C(F)F)c2)CC=CCC1 Cc1cc(CC(C)Nc2cc(NC(C)Cc3ccccc3F)ncn2)cc(C)c1 N1(C(C(CC)N(CC)CC)=O)CC2CC(C(=O)NCCc3cn(C)cn3)(C2)C1 C1(NC(c2c(CCC)onc2C)=O)CN(C(=O)C(F)(F)CC)CC1C1CC1 CC1CCc2c(C(=O)NC3(C)CN(C(C4CC4c4ccsc4)=O)C3)csc2C1 C=CC(C)(CC)C(=O)NCC(C)(O)CNC(c1ccccc1SCC)=O C1(NC(=O)CCC2CC2)CCOC12CCN(C(=O)C(=Cc1cccnc1)F)CC2 C(=O)(CC(=O)NC1CCN(C(c2sccc2-n2ccnn2)=O)C1)NCC C1(C(N2CC(N(C(=O)C=C3CCCC3)C)C2)=O)(C(N(C)C)C2CC2)CCCO1 C(=O)(NNC(=O)CCOCC(F)(F)F)n1cc(C(C)OCCOC)nn1 N1(C(C=CC)=O)CC2(CC(NC(=O)Cn3cc(COC)nn3)CO2)C1 C1(C(N2CC(O)(CC)C2)=O)CCC(N(C(=O)COCc2cccnc2)C)CC1 c1(C(=O)NC(C(=O)NCCS(=O)(=O)NC)C2(C)CC2)cccc(C)n1 C(=O)(CCS(N)(=O)=O)NCCC1N(C(c2c(OC)c(C)sc2)=O)CCC1 C1(c2nc(C(C)C)[nH]n2)CCCCN1C(=O)NC(CCO)c1ccco1 CC(C)(C#N)CCCC(=O)N1CCC(C(N2CCn3nccc32)=O)CC1 c1(C(N2CCN(C(c3ncc(C)cn3)=O)CC2CF)=O)ccc(C#N)cc1O C(=O)(C#CC1(C)CC1)N(C)CC1OCCN(C(c2n(CC=C)ccc2)=O)C1 c1(CN2CC(CC#N)N(C(=O)Cn3nccn3)CC2)cc(Br)cc(F)c1F C1(CC(=O)NC2CCCN(CCC)C2)CCCN(C(=O)C(=O)NC(C)C)CC1 C1(NC(C(CC2CCC2)OC)=O)CN(C(C)=O)CC1C c1(OCC2N(C(C(CC)NC(=O)C(F)(F)CN(C)C)=O)CC2)cccc(C#N)c1 c1(C(N(C2C3CN(C(C(C)NC=O)=O)CC32)C)=O)cc2nc[nH]c2cn1 C1(CC(=O)N(CC(O)CF)CC)CCN(C(=O)CCCCN(C)C)CC1 N1(NC(C(c2n(CC)cnn2)N(CC(C)C)C)=O)CCC(C#N)CC1 CC1(C)C(C)(C(N2C3CC2CN(C(c2cc([N+](=O)[O-])sn2)=O)C3)=O)C1(C)C c1(C(=O)NC(C(=O)NC2C(N(C)C)COC2)CC2CCOCC2)ccc(N)cn1 C(=O)(C1Cc2ccc(F)cc21)N(C1CCCN(C(c2c(CC)nc(C)s2)=O)C1)C c1(C(=O)NCCN(C)C(C2C3CCC2(c2ccnn2C)C3)=O)ccc2sncc2c1 Cn1cnc(C(N2CCC(CNC(c3c(C(F)F)cnn3C)=O)C2)=O)cc1=O C1(CNC(c2ncn(C(C)(C)C)n2)=O)CC(C2CC2)C1 Cc1nn2c(c1CNC(=O)C(O)CC(F)(F)F)CN(C(=O)C(C)(F)F)CC2 c1(CC)nc(Cl)c(C(=O)NC(C)CN(C(=O)CNCc2nc(C3CC3)no2)C)s1 C1(C(N(c2ccc(Cl)cc2)CCCC)=O)CCOCC1(C)C C(C)(C)(CCC(=O)NCc1ccccc1O)NC(c1ccc(CC)cc1)=O c1(NC(C2C(NC(c3c(C)n[nH]c3)=O)CCCC2)=O)c(C)cccc1F c1(NC(C(c2ccoc2)NC(Cc2c(C)n(C)cn2)=O)=O)ccc(O)cc1F c1(OC)cnc(C(=O)N(CC(C)N(C)C(C2CC2(C)C)=O)C(C)C)c(Cl)c1 N1(C(C2CCN(CC)C2)=O)CCC2(CC2C(=O)NC2(C)CC3(CCC3)C2)C1 C1(C(N(CC(=O)OC)CCC)=O)CCCC1CNC(C1OCCC1C)=O C1(C(=O)NCC2(CC(N)=O)CC2)CN(C(C2CC3CCC2C3)=O)CC12CC2 c1(NC(CCCCNC(C(c2ccccc2)OC)=O)=O)cccc(C)c1C N1(C(=O)COc2ccc(Cl)cc2Cl)CCN(C(c2ncc[nH]c2=O)=O)CC(O)C1 C(C1c2ccccc2CCN1C(c1cccn1C)=O)NC(CSCCOC)=O C12(C(N3CC(OC)C3)=O)CCN(C(C3(CO)CCCC3)=O)CC1C2 N1(C(C=CC)=O)CC(OC)C(NC(c2cn(-c3cccnc3)nn2)=O)C1 Cc1cc2ccc(C(=O)NC3CCCCC3NC(=O)C(=O)NC(C)C)cn2c1 CC1Oc2c(C(=O)NCCCNC(c3ccnc(C(C)C)n3)=O)cccc2C1C C1(NC(C(CCCC)F)=O)CC2CN(C(=O)CCc3cnco3)CC2C1 C1(C(=O)NC2CCN(C(c3ccc(CCCCC)o3)=O)C2)C2CCN1CC2 c1(C(N2C(C)(CNC(C(CC#C)C)=O)CCC2)=O)cc(OC)ccc1[N+](=O)[O-] C(C)(C)(CCC(=O)NC1C=CCCC1)NC(COCC#C)=O c1(C(=O)NC2CCCCN(C(CC(C=C)CC)=O)C2)ccsc1S(N)(=O)=O c1(NC(C)=O)cncc(C(N2CC(F)(CNC(=O)C(C)Cc3ccco3)C2)=O)c1 C(=O)(CC(C)C(C)C)NCC1(O)CCN(C(c2n(CCOC)ncc2)=O)C1 N1(C(c2ccc(OC)s2)=O)CCN(C(c2cc(F)cc(F)c2)=O)CC1C#N C1(N(C(Cc2n(C)cnc2)=O)C)CCN(C(C2CCCN(C(=O)C3CC3)C2)=O)CC1 C1(NC(c2cc(C)nc(C)c2)=O)C(C)CN(C(c2cnc(O)o2)=O)CC1C c1(C(N2CCN(C(c3ncc(F)cn3)=O)CC2)=O)ccc2nc(C3CC3)[nH]c2c1 C(=O)CCCC(F)(F)Br.N1(CCn2cc(CC(C)(C)O)nn2)CCCCC1=O c1(C(=O)NC(CC)(C)CNC(=O)C(CN(C)C)C(C)C)cn2ccnc2cn1 CC#CCCCC(=O)NCC(C)CN(C)C(c1cnc(CC)nc1C)=O C1(CNC(c2onc(CC)n2)=O)CCN(C(C23CC2COC3(C)C)=O)C1(C)C C1(C(=O)NC)(OC)CCN(C(C2CCCC2OC)=O)C1.c1(OC)cc(CO)on1 C1(C(=O)OCC)CC(=O)N(C(C(=O)C(C)C2CCCO2)=O)C1.C1(N)(C)CC1 C(=O)(C(C)(CC)C(N)=O)N1CCN(C(c2nc(COCC)sc2)=O)C(CF)C1 N1(C(c2ccnc(OC)n2)=O)CC(NC(=O)C(C)(C)CC2CC2)CCC1C c1(NC(C)=O)ccccc1C(=O)NCC1CCCN1C(=O)CNC(c1ccoc1)=O C1(CNC(C2(OC)CCSC2)=O)COCCN(C(=O)Cc2c(Cl)cnn2C)C1 C12(CNC(=O)CCCCO)CC(CO1)N(C(C1CC1Cc1ccc(F)cc1)=O)C2 C1(C)(C(=O)NCCOCCN(C(C2C(C(=O)OC)C2)=O)C)CC=C(C)CC1 Cc1cc(C(=O)NCCc2cc(C(=O)NCC3OCCC3(C)C)no2)cc(O)n1 C=CC(N=c1nc2scnc2c(NCC2(C3CC3)CC2)[nH]1)C1CC1.c1(SC)ccccc1 C1(NC(C2CCN(CC3CC3)CC2)=O)CC(CO)N(C(c2ccc(O)nc2)=O)C1 CN1C(=O)CN(CC(=O)NCC2CCN(C(=O)Cc3ccns3)C2)C1=O C(=O)(C(O)CC(F)(F)F)N1CC(OC2CCN(C(C(C(C)C)N(C)C)=O)CC2)C1 c1(C(N(C2CCCCC2)CCNC(C(C)NN2CCOCC2)=O)=O)cccnc1 C(=O)(C1=CCCCCC1)N1CCC(NC(=O)CC2CCCSC2)C(F)C1 C(=O)(C(O)C(C)(C)C)N1CC(C)CC(CNC(CCCn2ncc(C)c2)=O)C1 C=CCC(C)(C)CC(c1nnnn1C)NCC1CC1c1c(F)cccc1Cl c1(C(N2CC(NCC(=O)NCCC(=O)OC)C2)=O)nc2c(s1)CC(C)(C)CC2 N(C1c2ccccc2CC1NC(=O)CCCC1CC1)C(C(C(C)O)N(C)C)=O Cc1cc(C(=O)NCCC2CN(C(=O)C=CC3(C)COC3)CC(C)O2)nc(C)c1 C1(C(=O)NC(CCC)C2CCCC2)CN(C(c2sc(C)nc2C)=O)CCO1 C(C(CC(C)C)C(=O)NC1CCCC1(C)N(C)C)NC(c1c(C)[nH]cc1)=O Cc1nc(CC2CC2)oc1C(N1CCOC(CNC(c2cc(Cl)c[nH]2)=O)C1)=O N(C1c2ccccc2CC1NC(C1CCCC12CC2)=O)C(C(CCC)OC)=O c1(N(CCCC)CC(N)=O)nc(C)cn2nc(CC)cc12 c1(SCC)cc(C(=O)NCC2CC2CNC(C2CCCC3(CC3)C2)=O)ccc1C N1(N2C(C)CCCC2)CCN(C(N(C(C(CC)=CC)=O)C)=O)CC(C)(F)C1.C(C)=O Cc1oc(C(C)(C)C)cc1C(=O)NC1CN(C(C2CC2OC(C)(C)C)=O)CC1F c1(C(=O)NCC2CC2CNC=O)cc(C(F)F)cc(F)c1.c1(C)cscc1C1CC1 c1(C(N2CCSCC2)=O)ccc(C(N2CCCC2c2ccc(F)cc2)=O)nc1 CC1CC(C(F)(F)F)(NCc2ccccn2)CC(C)O1 C1(C)(C(=O)NCC(C)C)CC12CCN(CC(C1CCCCCN1)=O)CC2 c1(CCC(=O)NCCN(C2CCCCC2)C(C2C(C#N)C2)=O)ccccc1F Cc1cccc(C(=O)C(=O)NC(C2CCN(C(C3CC4(CC4)C3)=O)C2)C)c1 N1(C(COCC)=O)CCC2CN(C(c3cnc(O)n3CC)=O)CC2C1 Cc1ccc(C(N2CCCCC2CNC(=O)Cc2ccccc2C)=O)cc1C C(=O)(C1=CC2CCCC12)NCCC1CCCN(C(C2(C(C)C)COC2)=O)C1 N1(C(C2C(CC)CCCC2)=O)CCN(C(c2cncn(C)c2=O)=O)C(C)C1 C1(C(c2nnnn2C2CC2)N)CCC(C)CC1.CC1(C)CNC1.C1CS1.C1(CC2CC2)CC1 C1(NC(CSC)=O)CC2(CCCN(C(c3ccnc(NC4CCC4)c3)=O)C2)C1 c1(CC)cc(C(N2CCOC(C(C)NC(C3CN(CC(C)C)C3)=O)C2)=O)nn1C c1(CC)cc(F)c(C(=O)NCC(C)CNC(C2CN(C(N)=O)C2)=O)cc1F CC1(C)CN(C(=O)CC2CNC(=O)O2)CCC1C(N1CCC12CCCC2)=O CCC(F)(F)C(C)(C)C(=O)NCC(C)CNC(c1cnn2cc(C)cnc12)=O N1(C(CCCC=C)=O)CC2CCC(CNC(c3ccn(CC)n3)=O)C2C1 c1(C(N(CCNC(C2C(Cl)(Cl)C23CC3)=O)CC)=O)c(F)cc(Cl)cc1Br N1(C(Cc2c(C)nc(S)s2)=O)CCCN(C(C2CCCCS2(=O)=O)=O)C(C)C1 N1(C(C(C)OCC=C)=O)CCC2(CCCN2C(c2ccnn2CC2CC2)=O)C1 C=CCCN=C(NCc1conc1C(F)(F)F)NC1CC1C1CCOCC1 CN1C2CC(CS(=O)(=O)NCc3conc3C(C)(C)C)CCC1CC2 c1(C(N2CC(OC(CC)C(=O)OC)C(C)C2)=O)csc(=NC2CC2)[nH]1 N1(C(C(CC)(C)COC)=O)CC2CCC1C(NC(=O)Cn1cc(C#N)cn1)C2 C1(C2CCN(c3cnc(F)cn3)CC2)(NC(C2CCN(OC)CC2)=O)CC1 C1(NC(c2cc(C)c(C)nn2)=O)CCC2CC1CN2C(C1(C2CCC2)CC1)=O CCC(C)(CO)NC(=O)CC1C(NC(c2cocn2)=O)CC1O N#Cc1cc2c(nc1N1CC3(CC3)CC1C(=O)O)CS(=O)(=O)CC2 c1(CN2C3(c4nnc(C(C)C)o4)CCC3CC2)ccc2c(c1)OCC2 N1(c2c(F)cnc(C)n2)CCC2(CCCCC2NC(C2(c3cccs3)CC2)=O)C1 N1(C(C2C(C)(C)C2(F)F)=O)CC(NC(=O)CCn2cc(Br)cn2)CC1(C)C c1(-c2c(OC)nccc2)nccc(=NC(=O)C2CCCCN2C)[nH]1 C#Cc1c[nH]nc1NCCC(N1CC(CNC(=O)C2CC2)OCC1)=O CC(C)CC(C(=O)NCC1(O)CCN(C)C1)NC(=O)C(F)C(C)(F)F C(CC(=O)N1CC(N(C)C)(CO)C1)(C1CC1)SC.C1(C(=O)N)CC(CF)C1 CC(C)C(C(C)NC(=O)CN(C)C(c1cccs1)=O)NC(C1(C(N)=O)CC1)=O N1(C(c2ccc(CC)o2)=O)CC(NC(=O)CC2CCCN2C(C)C)CCC1C Cc1cc(NC(=O)C(CCF)NC(c2nccn2C(C)C)=O)cnc1O C1(CNC(c2cccc(OC)n2)=O)CC(F)(F)CN1C(C1CCC1(C)C)=O CC(C)CC(CNC(c1cccc(N(C)C)c1)=O)NC(C1CCCCC1O)=O N1(C(C=CC)=O)CCC(F)(NC(=O)C(C)OCCOCCCCCCOC)CC1 N1(CCN(C(c2c(C)nccc2)=O)C(C)C)CC(O)(C2CCCC2)C1 C(CCCCC(=O)N1CCOC(CCCNC(=O)C=Cc2ncc[nH]2)C1)OCC CN1CC(C)(C)CC1NC(C1CC(O)CCN1C(=O)CCCNC(N)=O)=O c1(OC)ccc(C(N2CCCC(NC(C3CC3C(C)(F)F)=O)CC2)=O)cc1Cl C(=O)(C(C)(C)CC(F)F)NCCC(=O)Nc1c(CC)nn(C)c1 C1(C(N(C(CN(C(c2ncn(C(C)C)n2)=O)C)C)C)=O)CCC2(CCC2)C1 C1(CNC(CCN(c2ccccc2)C)=O)CCCN1C(=O)C(c1cscn1)N(C)C Cc1nc2c(o1)CCCC2CC(=O)NC1CCN(c2ncnn3c(Br)ccc23)C1 N1(C(C2CCCO2)=O)CC2(C1)CN(C1CC1)C2.N12CCCC1NC2=O c1(NC(C)=O)ccccc1-c1noc(CC(C2CCCC(=O)N2)=O)n1 C(C(=O)OC)(C(C)C)N(C(=O)CCC1CCC(NC(c2cccnc2)=O)C1)CC C(=O)(C(F)C(C)(C)O)NCCn1cc(C(N2CC(C(=O)OC)SCC2)=O)nn1 N1(C(C2N(C)C(=O)OC2)=O)CC=C(CCNC(=O)CC2CCCOC2)CC1 C1(C(=O)NCC(C)(COC)CC)(CC)CCCN(C(c2cnc(C)nc2)=O)C1 C(=O)(C#CC1CCOC1)NC1(CNC(c2ncc(CC)cn2)=O)CCCC1 N1(c2ccc(C#N)cn2)CC(NC(C2CC3(C2)CC3(F)F)=O)C2CCCCC12 N1(CCCC)C(=O)c2ccc(C(=O)Nc3ccc(S(=O)C(F)F)cc3)cc2C1=O C(=O)(N=c1cc2ccccn2[nH]1)C1N(C(C=CC(=O)OCC)=O)CC1C c1(C(N)=O)cc(C(=O)NC2CCN(C(C3CN(C4COC4)C3)=O)C2)n[nH]1 C(C(C)(C(N)=O)NC(=O)NC1(c2ccccc2Br)CCC1)OC c1(C(=O)NCC2N(C(C3C(C(N)=O)C3)=O)CC(O)C2)cccc2nccn12 C(=O)(C(C)CC(F)F)N(CC(CC)NC(C1CS(=O)C1)=O)CC C(=O)(C1CCc2ccccc21)N1CC2C(NC(C3CCCN(C)C3)=O)C2C1 c1(NC(CSCC(=O)NCC)=O)oc(C)cc1C(=O)N(C1CCCC1C(=O)OC)C Cc1nn(C2CCCC2)c2c1C(c1ccc(F)cc1Cl)CC(=O)N2 N1(C(c2scc(C)c2)=O)CCCC(NC(=O)CC2CCCO2)C1C c1(N2CCCC(NC(c3ccc(CCC(=O)OC)cc3)=O)C2)ccc(C#N)nc1 C#CCC(C(=O)NC(C1CCCC1)CC)NC(c1cnc(OCC)nc1)=O c1(CCC)cc(C(=O)NCC2(OC)CN(C(=O)C(C(C)C)SC)C2)ccn1 c1(OC)ccc(C)c(NC(c2c(CNC(=O)C(C(C)C)OC)nnn2C)=O)c1 c1(OC)ccc(Cl)cc1C(=O)NCC1CCC1NC(=O)C1=CCCS1 C1(CC(C)(C)C)CN(C(=O)C=CC2CC2)CCC1NC(c1ccnn1CCF)=O N=c1nc(O)c(CC(N2CCCC(CCNC(=O)CC3=CCCC3)CC2)=O)c[nH]1 N1(C(COC(C)C)=O)CC2CC2(NC(C2COCC2(C)C)=O)C1 N1(C(CC(C)n2cccc2)=O)CC2(CCNC(C3CCCN3C)=O)CCC1CC2 C(=O)(CCCCC(=O)NCC1(CCNC(=O)CCCC(F)(F)F)CC1)NC N1(C(c2nccc(C)c2)=O)CCCC(C)(C)C1C(=O)NC1CCC(C2CC2)C1 C(=O)(C#CC1CCOCC1)N1C2CC(CC(NC(CC3C(C)CC3)=O)C2)C1 C(=O)(CC(C(F)F)NC(=O)CCCF)NCc1cc(CC)[nH]n1 C(=O)(CC(F)(F)C(C)C)NC1CCN(C(c2c(C)nc(=N)[nH]c2)=O)CC1CO c1(OC)ccc2nc(N3CC(CN(C)C(c4coc(Cl)n4)=O)C3)c(C#N)cc2c1 c1(OC)cccc(CN2CCC(C(=O)Nc3ncc(C)c(C)n3)C(CO)C2)c1F CCS(=O)(=O)CC(=O)N1CC(N(C2CCCC2)CC(C)C)C(C(=O)OCC)C1=O c1(OC)cccc(C(C(=O)NC2CC(NC(=O)C(C)CF)C2)OC)c1 Cc1cc(C(=O)NCC23CC(C2)C(NC(=O)C(C)C(C)C)CO3)nnc1C Cc1nn(C)c2sc(C(N3CCCC4(C3)CN(C(=O)Cc3ccns3)C4)=O)cc12 C1(C(=O)NC2CC(NC(C(OC)OC)=O)C2)OCCC12CCCCC2 c1(C(N2CCC(CNC(CCC#C)=O)CC2)=O)cc(F)ccc1F Cc1c(Cl)ccnc1CNCC1CCCO1.c1cc(N2CCN(S(C)(=O)=O)CC2)ncn1 c1(C(N2C3C(C(N4CC(C)OCC4C)=O)C(C3)C2)=O)c[nH]c2cccc(Cl)c12 Cc1cc(O)ncc1C(N1CCC(F)C(NC(=O)C2=CCCCC2)C1)=O CC1(C)CC(C(=O)NC2(c3ccccc3)CCN(C(c3cccs3)=O)C2)CCO1 C1(c2cccc(F)c2)(C(=O)NC2(CC=C)CC2)CCN(C(=O)CC(=O)OC)C1 N1(C(CC2CCN(C)C2=O)=O)CC(NC(c2cnccc2C(F)F)=O)C2(CC2)C1 C(C)(CN=c1[nH]c(N2CCn3cccc3C2)nc2cc[nH]c12)N1CCC(C)CC1 C1(CNC(c2nc(OCC)sn2)=O)CN(C(=O)CCC(C)CN(C)C)CC12CC2 C(C(C)(C(C)C)NC(=O)Cc1cnccc1OCC)NC(C=CCOC)=O C(CCN=C(NCC1CCC2(CCC2)O1)NC1CCCO1)c1ccc(F)cc1 c1(C(=O)NC2C(NC(c3nc(C)nc(O)c3)=O)COC2)c(O)nnc2c1CCC2 c1(C(=O)NCC(n2cc(-c3ccns3)nn2)C)cnn(Cc2ccccc2)c1 C(CN=C(NCC(=O)NC1CC(Cl)(Cl)C1)NC1CCS(=O)(=O)C1)SC CCC(C(=O)NCC(C)NC(c1ocnc1C)=O)OC1CCCCC1 C12(C(=O)NCC(CCOC)NC(c3ccncn3)=O)C3CCC(CC13)C2(F)F Cc1cc(N)c(C(=O)NCCC2CCC(NC(=O)C3=C(Cl)CC3)C2)cc1C C#Cc1cnc(C(N2CCCCC2CC(N2CC(C)(C(=O)OC)C2)=O)=O)c(C)c1 Cn1cc2ccc(NC(C3CC(O)CCN3Cc3ccnc(O)c3)=O)cc2n1 N1(C(C2CC(NC(c3n[nH]cc3Br)=O)C2)=O)CCC(S(=O)(=O)c2ccccc2)CC1 C(=O)(CC(C)(C)C(=O)NC1CCN(C(=O)CNC(=O)NC)CC1C)OCC C(=O)(CS(=O)CC)N(CCC(=O)NCCc1ncnn1C)CC=C c1(NCc2c(C(F)(F)F)nc[nH]2)nccc(=NCc2nc(C3CCOCC3)n[nH]2)[nH]1 c1(N(C)Cc2nc(NC(c3cn(CCC)nc3)=O)sc2)ccc(C(F)(F)F)cc1 c1(C(=O)NCC(CC=C)NC(c2cc(C(F)F)cc(F)c2)=O)ccc(N)c(F)n1 C(CC(CC)C(=O)N1CCC(N(C(=O)CN(C)S(N)(=O)=O)CCO)CC1)=CC c1(OCC)cc(C(=O)NC2(C)CCN(C(=O)COC3CCC3)C2)cc(Cl)c1O Cc1nnc(CC(=O)NCC2CCC(NC(=O)Cc3nncn3C)C2)o1 c1(C(=O)NC2(C(=O)NC(C)CN3CCCC3)CC2(C)C)csc(C#N)c1 C1(OC)CCCCN(CC(=O)NCC(C)(Cc2ccccc2)CO)C1=O C1(N(C)C(C2CCCCS2)=O)CN(C(c2csc(C(F)(F)F)n2)=O)CC12CC2 c1(OC)cccc2cc(C(N3CCCCC(NC(=O)C(C)C(C)(F)F)C3)=O)oc12 C1(CCNC(CC(C)C2CCC2)=O)CN(C(=O)CNS(N)(=O)=O)CCCO1 CC1CCCN(C(c2nc(Cl)cs2)=O)C1CNC(c1ccc(C2CCC2)cc1)=O C1(NC(C2CC(C)SCC2)=O)CC2CCC1CN(C(=O)CN1C(=O)CNC1=O)C2 Cc1ccc(C)c(F)c1-c1ccc(=NCc2cc(F)c(OC(C)C)cc2F)[nH]c1 C12(NC(C(CCOC)C)=O)COC(C1)C(NC(=O)Cc1ccc(F)c(C)c1)C2 N1(C(COC(=O)CO)=O)CCC(NC(=O)CC2CCCCC2)CC1 c1(C(=O)NCC2(O)CCN(C(C(C(=O)OC)C)=O)C2)ccc(OC)cc1F CCC(C)CCCCC(=O)Nc1ccc(Nc2cc(C3CC3)ncn2)c(C)c1 c1(C(=O)NC(C)CNC(=O)CC(c2ccc(N)cc2)C)cnc2n1CCC2 N1(C(CCN(C(C2CCC(=O)N2)=O)CC)=O)CCC(C(F)F)CC1 C(=O)(C(C)S(N)(=O)=O)N(CCCNNCCC(=O)C(=O)N)CC.C(=O)(CC(C)C)NCC c1(C(=O)NCCCNC(C2(CO)CC2)=O)cccnc1-c1ccccc1 c1(OC)cc(=NC(=O)C=CCC(C)(C)NC(=O)C(O)C2CC2)[nH]n1C c1(Cn2cc(CN(CCN(CC(=O)OC)CC)C)nn2)cnc(C2CCCO2)s1 C(C(CC)(CC)C(=O)Nc1cnc(C)c(C)c1)NC(CCC(CC)OC)=O CCC(C(=O)N(C(C)(C(=O)NCCC1CCC(=O)N1)C1CC1)C)C(C)(C)CC C1(NC(C(CSC)O)=O)CC2(CCN(C(c3cccc(SC)c3)=O)CC2)C1 C1(CC(=O)N(C(C)C)CCN(C(=O)CCCc2cccs2)C)COCC(C)(C)O1 C1(NC(C=C(CCC)C)=O)CCCC12CCN(C(C1CC(O)CN1CC)=O)CC2 C1(C(N2CC(NC(c3ccc(C4CCC4)nc3)=O)C2)=O)C2CCCCC12 c1(OC)cc(N)cc(C(=O)NCC(C)(C)CNC(C2CC2CC(C)C)=O)c1OC c1(C(=O)NCC(CCCC)NC(=O)CC2(OCC)CC2)cc(N)ccc1CC Cc1csc(=NCC(=O)NC2(CF)CN(C(C3CC4(C3)CC4(F)F)=O)C2)[nH]1 C1(NC(c2ccc(OC)cc2)=O)CCCCN(c2nnc(Cc3ccccc3)s2)C1 CS(=O)(=O)C1CCC(C(N2CCC(NC(=O)CC(F)(F)Cl)C2)=O)CC1 C1(N(C(C(=O)NCCOC)=O)CCSC)CCCN(C(=O)Cc2ccsc2Cl)C1 c1(C(=O)NCC(C2CCOC2)NC(c2cncc(OCC)c2)=O)nnc(O)nc1O C1(N(C)C(c2ccnn2CC(F)F)=O)CCCC(NC(=O)Cc2ccsn2)C1 c1(C(N2CCC3C(NC(c4cc(CC)c(C)s4)=O)C32)=O)cc(N)cnc1Cl c1(C(N2CCC(OCCNC(C(C)OC)=O)C2)=O)ccc(CC(C)C)nc1 c1(OC)ccc(CC(=O)CN(c2ccc(Oc3ccccc3Cl)cc2)CCO)cc1 Cn1cc(C(=O)NCCn2ccc(C(N3CCC(CCO)C3)=O)c2)nn1 c1(C(=O)NCC2C(CNC(C3N(C=O)CCC3)=O)C2)cc2ccccc2oc1=O c1(CNC(C2C(C)(C(C)C)C2)=O)ccccc1-n1cc(CCC2(O)CCC2)nn1 c1(CC)ccc(F)c(C(=O)NCC2CCCC(NC(c3[nH]c(C)cc3C)=O)C2)c1 Cc1cc(C(=O)NCc2ccc(C(=O)NCCCCC3CC3C)cc2)c(C)s1 c1(CNC(=O)OC(C)(C)C)cccc2c1CCN(CC1CCC3CC3CC1)C2 C1(CNC(CCCCC#C)=O)CN(C(=O)CCCCOCC)CC(C)(C)O1 N1(C(c2ccc(SC)o2)=O)CCC2CCC(NC(=O)CC3(O)CCC3)C1C2 N1(C(C2C(SC)CCC2)=O)CCC(CCNC(=O)Cc2ncc(F)cc2F)CC1 c1(CNCC(N2CCC(C)CC2)C)cnc(O)c(F)c1 CN1CCN(C(=O)Cn2nc(O)ccc2=O)C(CNC(=O)Cc2cccs2)C1 N1(C(C(C)N(C(c2cc(C)ncc2)=O)C)=O)CCn2ncc(C)c2C1 C1(NC(CCCOCCC)=O)CN(C(=O)Cn2cnc(C#N)n2)CCC1C CCCCC(CC)C(=O)NC1CCC(F)(CNC(=O)Cn2nnc(=O)[nH]2)C1 C1(C(=O)NCC(CC)NC(c2c(Cl)nn(C)c2Cl)=O)CCCNS1(=O)=O c1(OC)ccc2c(C(=O)NCC3CCN3C(=O)C3=CCSC3)ccnc2c1 Nc1ccc(Cl)cc1C(=O)NCC12CC(NC(c3c[nH]nc3C3CC3)=O)(C1)C2 C1(NC(c2cc(SC)oc2)=O)CCN(C(c2cnc(OC)c(C)n2)=O)CC1(C)C N1(C(C2(Cc3ccc(O)cc3)CC2)=O)CC2CC2(C(=O)OC)C1 c1(CNC(c2cn(C(C)C)nc2)c2nnnn2C(C)(C)C)cc(OC)c(Cl)nc1 c1(C(N(C)CC2(O)CN(C(C3C4CCCCC34)=O)C2)=O)cc2cccnc2o1 c1(CC)ccc2sc(CN(C)CCCCCCC)nc2c1 C1(C(C(=O)NCCN(C(c2c(SCC)cccn2)=O)CC)O)CCCCCCC1 Cc1cc(C#N)cnc1C(=O)NCC1CCC1NC(C1CC12CCC2)=O CC#CCC(C(=O)NOCC(C)(C)C)NC(=O)CC(=O)N(C)C c1(C(=O)Nc2nc(C)cc(C)n2)ncn2cc(-c3cncn3C)sc12 C1(F)(C(N2CC(NCc3cn(C)nc3)OCC2)=O)CCCCC1(F)F CC1(C(=O)NC2(C(=O)NC)CC2)CCCC1.C12CC1(C)CC(=O)N2.CO Cc1cccc(C(=O)NC(C(=O)N2CC(c3cccnc3)C2)C2CC2)c1F c1(C(N2CCC(N(C(C(CC)F)=O)C)CC2)=O)nc(-c2ccccc2)ncc1Cl c1(C(=O)NCCC(C)NC(C2C(SC)CCC2)=O)ccc2nc(O)cc(O)c2c1 C1(OC)CC(CNC(C2C=C(C)CS2)=O)N(C(=O)CSC2CCCC2)C1 N1(C(C2(C)C(C)(C)C2)=O)CCC(C)(CNC(c2cnn(C(F)F)c2)=O)C1 C1(F)(C(=O)NC(C2CCCC2)CNC(c2cc(SC)ncc2)=O)C(C)(C)C1(C)C c1(C(=O)NCCCCCCCn2cncn2)cc(Cl)ccc1Cl O=C1OC2C(NC(C3CCCS(=O)(=O)C3)=O)C3CCC12C3 N1(C(C2(OC)CC2)=O)CCC(CC(=O)NCC(C)CCO)CC1 c1(C(N2CC(NC(C#CC(C)(C)C)=O)C(F)CC2)=O)ccc2cncn2c1 c1(C(=O)NCCCOCC(=O)NCCN(C)C)cn(CC(N)=O)nn1 C1(C(=O)NCCN(CCCC)CCCC)CCCN(C(=O)COCC(F)F)C1 C1(COC)(NC(c2c[nH]nc2F)=O)CCN(C(=O)Cn2ncc(Br)n2)C1 c1(C(N2CCC(=CCNC(C3C(C)(C)CO3)=O)CC2)=O)cc(O)nc(C2CC2)n1 c1(OCC(=O)N(CC(C)N(C)C(C2CCCC2O)=O)C)ccsc1Cl C1(CNC(c2cc(Br)no2)=O)CC2CCC1N2C(=O)Cc1ccc(F)cc1 C1(C(=O)NC(C=C)C2CC2)CC(N=[N+]=[N-])CN1C(c1c[nH]c(C)c1)=O N1(C(CCOCCOC)=O)CCC2(CC2)CC1C(N1CC(C)N(C)C(C)C1)=O c1(NCC2(OC)CCCC2)[nH]c(=NCCS(=O)(=O)C(C)(C)C)nc2sccc12 C1(CC)CCC(C)N(C(c2conc2CNC(=O)CCCc2ncco2)=O)C1 C1(C)(C(N(CCCCNC(=O)C(C)(C)C2CCC2)C)=O)CCC(F)(F)C1 n1(CC(=O)N(C2CN(C(c3c(C)nns3)=O)CC2(C)C)C)nnc2c1CCCC2 Cc1ccc(C(C)C(=O)N2CC(CC(C)NC(c3ccsc3C(F)F)=O)C2)cc1 C(=O)(C1=CC2(CCOCC2)C1)N1C(C)(CC)CC(NC(=O)C(C)(F)F)C1 CCC(CC)(CCNC(=O)CC1OCCOC1(C)C)NC(=O)CCn1ccnc1 C(C)(N=c1[nH]c(NC2CC2C2CC2)nc2cc[nH]c12)c1scc(C)n1 C1(CNC(CCOCC(C)(C)C)=O)OCCC1C(=O)NC(C)(CO)C1CCCC1 Cc1oc(C(=O)NC2CC(CCNC(=O)CCC3CCCO3)C2)cc1CO Cc1cncnc1N1CCCC(CCNC(C2(C(C)C)CC2)=O)C1 CN1CC(C(N2CC(NC(c3ccc[n+]([O-])c3)=O)C2)=O)C(C(F)(F)F)C1 N1(CC)CC(NC(C2CC2CNC(=O)CCCc2ccccc2)=O)C(O)C1 CC#CCC(C(=O)NCCCCSC)NC(=O)CC1CCC(C#N)C1 c1(N2CCC(=CC(=O)Nc3cnn[nH]3)CC2)ccncc1[N+](=O)[O-] c1(C(=O)NC2CC(C)N(C(=O)CC3CCCOC3)CC2)cc2n(n1)CCCO2 CC(C)(C)C(O)C(=O)N1CC2(CC(NC(=O)CN3CCCCCC3)C2)C1 CC1CC1C1CC1C(N1CCC(CNC(C23CC(C)(CO2)C3)=O)CC1)=O N1(C(c2cnc(O)c(Cl)c2)=O)CCC2C1CCCN2C(C12COCC1C2)=O Cc1cc(O)ncc1C(=O)NCCN(C(=O)CC1COC2CC1C2)CC1CC1 n1(CC(=O)NC2CN(C(C3(CN(C)C)CC3)=O)CC2F)cnc([N+](=O)[O-])n1 C1(NC(=O)C=Cc2cc[nH]n2)COC2(CCN(C(=O)Cc3ccns3)C2)C1 CC1(C)CC2(CC(C(=O)NC3CC(CNC(c4cccn4C4CC4)=O)C3)C2)C1 N1(C(Cc2ccc(C)o2)=O)CCCCC1CC(=O)NC(CN(C)C)CCO Cc1cccc(C)c1C(O)C(N1CCC(C2CCCN2C(=O)CC2CC2)CC1)=O C1(NC(c2c(C)cncc2C)=O)CN(C(=O)Cn2ccccc2=O)C2(CCC2)C1 c1(C(=O)NC2C(NC(C(CC)=CC)=O)CCC2)ccc2c(c1)CCC2(C)C N1(C(CCc2cc(C)no2)=O)CC2CC2(C(N2CC(CN(C)C)C2)=O)C1 c1(NCc2c(C)noc2C)[nH]c(=NC2COCC2C2CC2)nc2c1ncn2C(C)C C1(C(N2CCCC(NC(=O)CN3CCC(O)CC3)CC2)=O)CC2(CCOCC2)C1 N12CC(C(C)C1)C2=O.c12ccc(cc1)[nH]c(=O)c2=O.C=C1CC(C(=O)NCC)C1 N1(C(C2CCN(C(C)C)C2)=O)CC2(CC(NC(C3CC=CC3)=O)c3nccn32)C1 C1(NC(COCCOCC)=O)CCCC12CCN(C(c1nn(C)cc1C)=O)CC2 Cc1ccc(COCC(=O)NC(C)C(C)NC(c2ccnn2CC(F)F)=O)cc1 C(=O)(NNCC(F)F)N(C)CC1(c2ccccc2)CCOC1 C1(NC(C2(C)CCOCC2)=O)CCC2CC1CN2C(=O)CCCCN1CCCC1 C1(OC)CC(F)CN(C(=O)C(Cc2cc[nH]n2)NC(c2ccnc(C)n2)=O)C1 C(=O)(CC1NC(=O)c2ccccc21)NCCC(C)NC(c1n[nH]cc1C1CC1)=O c1(NC2CN(C(=O)CC3CCS(=O)(=O)C3)C2)ncnc2c1CCC2 S(=O)(=O)(c1ccc(Br)cc1NCc1nc2ccccc2n1C)NC(CC)CO N1(C(c2ccc(C)c(F)c2F)=O)CCC2CCC(C1)N2C(=O)C(C)CC(C)(F)F c1(C(=O)NCC=C2CCN(C(CC(C=C)(C)O)=O)CC2)cn2nccc2nc1C c1(NC2(CNC(C(CSC)C)=O)CC2)ncnc2c1cnn2C C=CC1(CC(=O)NC2(CC3(C)CC3)CC2)CN(C(=O)CC2CC2)C1 N1(C(C=NOC)=O)CCCCC1C1CCN(C(=O)C(C)Cc2c(C)noc2C)C1 N1(C(C(C)NC(N)=O)=O)CCOCC1CNC(c1ccc(C(F)(F)F)s1)=O Cc1[nH][nH]c(=NC(=O)C23CC2CN(C(=O)Cc2cccc(O)c2)C3)c1Cl C1(C(=O)O)(Nc2cccc(-n3c(C)cc(C)n3)c2)CC2(CSC2)C1 c1(C(N2CC(N(C(C(C3CC3)SC)=O)C)C(O)C2)=O)cc(C)cc(F)c1N N1(CC(=O)N(CCCNC(c2cccc(Br)n2)=O)C)CCC(C)(O)C1 c1(CC(=O)NCC(C)NC(C(COCC)C)=O)ccc(O)c([N+](=O)[O-])c1 CC1(C(=O)NC2CCC(NC(=O)CCSC(F)(F)F)CC2)CCC12CCC2 C1(C(N2CCC(C(=O)NC(CC#CC)CO)(OC)C2)=O)CC2CC(=O)C1C2 Cc1nc(C(=O)NC(CNC(=O)C(C)Oc2ccccn2)C2CCC2)cs1 C(C(=O)N1CCCC(C)(CNC(=O)C2=COCCC2)C1)(c1ccccc1)=C(C)C N1(C(C=C(C)Cl)=O)CC(CNC(=O)C(C(C)C)N(C)C)CC12CCOCC2 N1(C(C(=O)NCCNC(C)=O)=O)CCN(C(=O)CC(C)(C)N(C)C)CC1C(F)F CC(F)CC(=O)N(C1CCCC1)CCCNC(C1CC2CC2C1)=O Cc1c(NC(=O)CC2(C)CN(C(=O)COC3(C)CCC3)C2)ccc(Br)c1F N1(C(CC(C=C)CC)=O)CC(NC(C2CCC(=O)N(C)C2)=O)CC12CCOCC2 c1(C(=O)NCC2(OC)CC2)cc(CNC(=O)C(C)n2ccnc2)[nH]n1 Cc1c(C(=O)NCCC2CCN(C(c3cc4occc4s3)=O)C2)cccc1N Cn1cnc2cccc(C(N3CC(NC(c4cccnc4S)=O)C4CC34)=O)c12 C12(C(N(CC(C)(C)NC(c3cn(CC)nc3C)=O)C)=O)CCC(F)(CC1)C2 N1(C(=O)NC(c2ccccc2)C)CCCC2(CCN2C(c2cc(Cl)ccn2)=O)C1 C1(C(N)=O)CN(C(=O)C(C2CC=CCC2)NC(=O)C=Cc2ccoc2)CC12CC2 CC(C)C(F)(CNC(C1CC(C2CC2)C1)=O)C(=O)NC1CN(C(N)=O)C1 C(CC(F)F)(C(=O)N(C)CCc1ccncc1)NC(CCC(C)OCC)=O N12CCC(CC1)NC2=O.C1(N(C)C)CC(NC(=O)CC2CC2(Cl)Cl)C1 Cn1cc(CN=C(NCC(F)F)NC2CCC2)c(C(F)F)n1 C1(NC(C=CCOC)=O)CCCCC12CCN(C(c1[nH]ccc(=O)c1C)=O)CC2 N1(C(c2cccc(C(N)=O)c2)=O)CCCC(F)(CNC(C2CCCN2C=O)=O)C1 C12(NC(C3CC(C)(F)C3)=O)CCCC1N(c1ccn3c(Br)cnc3n1)CCC2 C#Cc1ccc(CC(=O)NOCC(=O)NC(C)C(CC)CC)cc1C c1(NC(=O)CC(C)(C)COCCCC)ccc(C(=O)N(CC(C)SC)C)c(O)c1 c1(C(=O)NCCC2N(C(C(CC)C)=O)CCC2)cncc2c(OC)cccc12 c1(CC(=O)N(CC)Cc2ccnn2CC2CCCO2)ocnc1C1CC1 c1(CC(=O)NCC(CCOC)NC(C2CCC(=O)NC2)=O)cc(C(C)C)n(C)n1 C=CCCC(C(=O)O)NC(=O)Nc1ccc(SC)c(COC)c1 C1(N(C(c2cc(CC)c(CC)o2)=O)C)CCCN(C(C2CCCCO2)=O)CC1 c1(OC)c(O)cc(C(=O)NCC2CCC(CNC(c3cnsn3)=O)CC2)cc1C#N Cc1ccnnc1C(=O)NCCC(C)NC(C1(CC(C)C)CCCC1)=O C1(N(C(c2c(CCC)nns2)=O)C)CC2CC1N(C(C1CN3CCC1CC3)=O)C2 c1(N2CC3N(C(c4ccns4)=O)C3C2)ncc2cn[nH]c2n1 N1(CC(=O)NCCN(C(CC2C(C)=NNC2=O)=O)C(C)C)CCc2sccc2C1 c12ccc(cc1)CN(CCCN(C)C)C(=O)N2.Cn1cc(C2CC2)cn1 CC1(C)CC(=O)NCC1C(=O)NCCC1CN(C(c2c[nH]c(Br)c2)=O)C1 c1(C(N2CCC(C#N)(NC(CSC)=O)C2)=O)ccc2cc(O)ccc2c1 c1(CC(=O)NC(C(C)NC(c2c(C)ccnn2)=O)C)cc2ccccc2o1 c1(C(=O)NCC2N(C(C(=O)Nc3c(OC)cccc3)=O)CC2)sc(C)c(C)c1C N1(C(C2C(CNC(=O)Cc3cnsc3)CCC2)=O)CCc2nc[nH]c2C1 CC1CN(C(C2OCCC2C(C)C)=O)CCCN1C(c1cc(F)cc(F)c1)=O N1(C(=O)Nc2c(OC)cc(O)cc2O)Cc2ccc(CC3CC3)cc2C1 C=CCC(CC(F)F)C(=O)N(C)Cc1ccc(CNC(C2CCCCN2)=O)cc1 C1(C(N2CC=CC(NC(C=Cc3ncn(C)c3)=O)C2)=O)CCCC(F)(F)CC1 C(=O)(CCC(CC)CCC)N1CCC(N(C(CC(=C)C)=O)CCO)CC1 c1(CNC(C2N(C(C=C=C(C)C)=O)C(C)C2)=O)cn2cccnc2n1 c1(N(C(C)C)C(=O)NC2(CCO)CCCSC2)ccc(C(F)(F)F)cc1 C#CCCCCC(c1nnnn1C1CCCC1)Nc1ccc(C)cc1OC CCCCCCC(O)CCC(=O)NCC1CCN1C(=O)CCCCC(F)(F)F N1(C(c2c(C)c(Br)sc2)=O)CCOCC(CNC(=O)C(C)C2CC2)C1 n1(CC)c(C)cc(C)c(C(N2CCC(CN(C(=O)C(C)SC)C)C2)=O)c1=O N#CCCCCC(=O)NC1COCC1NC(=O)C(c1ccc(Cl)c(Cl)c1)O C1(NC(=O)OC(C)(C)C)CN(C(=O)COCC(=O)Nc2ccsc2)CC1C(F)F c1(OC)cnc(Cl)[nH]c1=NC1CN(C(=O)OC(C)(C)C)C(C)(CO)C1 C1(CNC(C(C)C)=O)CCCN(C(=O)C(c2cccc(CC(C)C)c2)C)C1 N1(C(C=COCC)=O)CCCC2CCN(C(=O)CCc3ccc(Cl)s3)CC12 N1(C(C2CC(CCC)C2)=O)CCC1(C)CC(=O)N(C)CC1CCCO1 C1(CC(=O)NCC(=O)N(CCN(C)C)CC2CC2)CCC2CC12 c1(SC)cc(C(=O)NC(C(=O)NCCCc2nccs2)C2CCCO2)co1 O=C(C(O)C(F)(F)F)NCC1CC2CCC1N2C(c1ccnc(CO)c1)=O N1(C(COC(C)C)=O)CCC(CNC(c2cnc(C(N)=O)s2)=O)CC1C N1(C(C(F)=C(C)C)=O)CCC=C(CNC(C2(F)CCOC2)=O)C1 C1(O)(CNC(C(C)Cc2cnco2)=O)CCN(C(C2CC3(CCC3O)C2)=O)CC1 c1(C(=O)O)cc(OC(F)(F)F)ccc1F.n12cc(cn1)C2NC1CC(C(=O)O)C1 n1(C(CNC(C(C)=C2CNC2)=O)C)cc2ccccc2n1 C1(NC(C(CCC)F)=O)CN(C(=O)CCc2nc[nH]n2)CC12CCOCC2 N1(C(CC(N2CC(O)CC(NC(COC)=O)C2)=O)C)CCCc2ccccc21 c1(CNC(C)Cc2cc(Br)ccc2Br)c(F)cc(Br)cc1Br C12(CNC(CCC#C)=O)CCCCC1CN(C(=O)C(C)(C)C1CCC1)C2 Cc1nc2sccn2c1C(=O)NC1CC(CNC(c2ccc3cncn3c2)=O)C1 C(C(CC(F)(F)F)NC(=O)C(C1CCC1)C1CCC1)NC(C(C)O)=O C1(NC(c2cncc(C)c2C)=O)CC2(CCN(C(c3cnc(S)[nH]3)=O)C2)C1 N1(C(CCCC=C)=O)CCCCC(CNC(=O)C(C)S(C)(=O)=O)C1 c1(COC)ccccc1CC(N1CCCC1CN(C(=O)C(C)CN(C)C)CC)=O N1(C(COCC)=O)CCC2(CCCN(C(=O)Cc3c(C)noc3C)C2)C1 CC1=NOC(C)(C(=O)NC2CN(C(=O)CSC(C)C)CC2C(F)F)C1 CCC(O)C(C)C(=O)NCCC1(NC(=O)CNC(c2ccc(Cl)cc2)=O)CC1 C(=O)(C(F)(F)CCN1CCCC1)NCCC1(CC(C)C)N=N1 N#Cc1cncc(C(N2CCC2CNC(C23CCC(CC2)C3)=O)=O)c1 c1(C(=O)NCC2OCC(CNC(CN(C)C3CC3)=O)C2)cccc(N)c1 C(=O)(C(Cc1ccoc1)NC(C1CCOC1)=O)NCC(C1CCCC1)OC c1(C(N2C(CC)CN(C(=O)CCCC(C)C)CC2)=O)nc(Cl)ccc1F c1(COC)cccnc1C(=O)NCC1(CC2CC2)CC1.C12CCCC(C1)NC2=O C=C(C)CCC(C)NC(=O)CCCCNC(C1(C)CCCC1O)=O C(=O)(CCC(C)(C)F)N1CCC(C2(O)CN(C(C(C)CCOc3ccccc3)=O)C2)C1 Cc1c(Br)noc1C(=O)NC1CCCCC1NC(=O)CN1CCCOC1=O C12(C(N3CC(CC(C)NC(c4ccc(OC)cc4)=O)C3)=O)CCC(CC1F)C2 c1(C(N)=O)ccc2c(C(=O)Nc3ccc(NC(c4cnc(O)[nH]4)=O)cn3)n[nH]c2c1 CCC1=NOC(C(=O)NCC2CCN(C(=O)NC(c3ccco3)C)CC2)C1 C(C1=NOC2CN(C(c3cc(C(C)C)[nH]n3)=O)CC12)NC(C(C)=C1CC1)=O C#CC1(NC(=O)CCOC2CN(C(=O)CCSCC)C2)CC2CCCC12.C(C)C N1(C(C2C(CC(C)(C)C)C2)=O)CCC(n2cc(CNC(=O)N(C)C)nn2)C1 c12ccc(cc1Cl)S(=O)(=O)NCCCCN2C.C1(CC)CC2(CCC2)CN1CC c1(C(=O)NC2CCN(C(C(CCC#C)O)=O)C2)oc2c(Cl)cccc2c1C C1(NC(c2n(CC=C)ccn2)=O)CCN(C(c2ccsc2Cl)=O)C1C C1(O)(CCNC(C(=O)N(C)C)=O)CN(C(C2COCOC2)=O)C1 C1(CC)CN(C(C2OCC3CCCC23)=O)CCN1C(=O)C(O)C(C)C N1(C(C(C(C)C)N(C(=O)OC)CC)=O)CCC(N2CC(F)(CSC)C2)C(C)CC1 C1(CNC(C(CCC)CC)=O)CCCC12CCN(C(C1(C#N)CCCC1)=O)CC2 CC1CN(C(=O)C(C)(C)C2(O)CCOC2)CCC(C(F)(F)F)O1 c1(C(N(CCCOC)C2CC2)C)nc(-c2ccc(C)s2)no1 N12CC(C1)C(C(=O)N(C)CCc1ccsc1)N(CC)CC=CC2=O.O(C)CC CCC(O)C(C)(C)C(=O)NC(C)CN(C)C(c1n[nH]c2c1COC2)=O N1(C(=O)NCC(C)(C)Oc2ccccc2Br)CCC2(CCC(O)C2)C1 N1(C(Cn2c(C(C)C)ncc2)=O)CC2C(CNC(=O)CN(C)C(C)C)C2C1 c1(C(N(CC(C)NC(c2cnc(-c3cccs3)s2)=O)C)=O)c[nH]nc1F Cc1cc(N)c(C)nc1C(N1CCC(O)(C(C)NC(c2ccn(C)n2)=O)C1)=O N1(C(C)=O)CCN(C2CC3(C2)CN(c2ccccc2)C3)CC1C c1(C(N(C2CCCN(c3ncnc(O)c3Br)C2)C)=O)cnc2[nH]ncc2c1 N1(C(CN(CCC)C)=O)CCCC1(C)CNC(=O)CC1OCCC1C c1(OC)ncnc(OC)c1C(=O)N(CCCCNC(=O)CN(C)C)C C1(NC(CCSC)=O)COCCN(C(c2ccc(OC(C)(C)C)cn2)=O)C1 CCCCCC(C)CC(=O)NC(C)CNC(c1cc(-c2cnn(C)c2)no1)=O CN=c1cc(C(=O)NCC2(CNC(C3CC(C)CCO3)=O)CC23CCC3)cc[nH]1 Cc1c[nH]c(C(=O)NC2CC(NC(=O)C(c3ccc(Cl)cc3)O)C2)c1C Cc1ncc2n1CC(C(N1CCC(CF)(NC(C3CCC3(C)C)=O)C1)=O)CC2 Cc1ncc(C(N2CC=CC2CNC(c2cn(C(C)C)cn2)=O)=O)cn1 c1(C(=O)NCC2CCN2C(=O)C(C2CCOCC2)F)cnoc1-c1cnc[nH]1 N1(C(CCCC#C)=O)CC2CCC1CN2C(=O)COC1CCCC(C)C1 C(=O)(C1CN(CC(=O)NC2CC(OCC)C2)c2ccccc21)NC(C)CCSC N1(C(C(C2CC2)OCC)=O)CC=C(C(=O)Nc2ccc(C)c(O)c2)CC1 CC(C(=O)NC1CCCN(C(c2csc(-c3cnn(C)c3)n2)=O)CC1)S(N)(=O)=O CC(CC(=O)N1CC2CC(NC(C3(n4cccn4)CC3)=O)C2C1)CC(C)(C)C N1(CCCC(=O)OCC(=O)N(C(C)C)Cc2ccco2)C(=O)NC(C)(C)C1=O Cc1c[nH]c(C(=O)NCCOCCC(=O)NCC2(C)CCOCC2)c1C C(CN=C(NCC1CCCS1)NCC1CC2CCC1CC2)c1ccnc(OC)n1 c1(OC)ccc(C(N2CCN(C(C)Cn3cc(C(C)(C)O)nn3)CC2)=O)cc1Br C(=O)(C(F)(F)C(O)C1CC1)NCC(C)CNC(c1occc1-c1ccccc1)=O CCCC(CC)C(=O)N1CC2CCC2(CNC(=O)C=Cc2nccs2)C1 C(=O)(CCCC(F)(F)F)N1CCC(OCCS)C1.c12ccc(Br)cc1C(=O)N2.CC=CCl Cc1nc2ccc(Br)cn2c1C(N1CCC(CNC(=O)C#CC2CCC2)C1)=O CCCCC(CNC(=O)C(C)N(C)C)NC(=O)Nc1sc(C)nc1C N1(C(c2c(C)cno2)=O)C2CCC(C2)C1CNC(c1ncsc1C(F)(F)F)=O C(=O)(C(F)C(C)(C)O)NC(c1ccc(F)cc1)CNC(C=C(CC)C)=O c1(C(=O)NC2CCCN(C(CC3CCN(C)C3)=O)C2)ccc2nn[nH]c2n1 c1(CN(C)Cc2csc(CC(N)=O)n2)cccc(I)c1 N1(C(c2nc(CC)oc2)=O)CCCCC1C1(NC(=O)CCc2cc(Cl)no2)CC1 c1(OCC)ncccc1C(=O)NCC(CC)NC(c1cncc(C)c1)=O Cc1ccc(CCC(N2CCC(CN(C(=O)CCC(C)(C)F)C)C2)=O)cc1C C1(NC(C2CC3C=CC2C3)=O)CC2CN(C(C34CCC(O)(CC3)CC4)=O)CC2C1 CC(C)CCCC(C)C(=O)NC1C=CCN(C(c2cncc3nnn(C)c23)=O)C1 c1(C(N2C(CNC(=O)C3=CCSC3)CC(C)(C)C2)=O)cc(Cl)c(F)cc1[N+](=O)[O-] C1(C(=O)NC(c2cn(C)nn2)C(=O)N(CC(C)C#N)CC)CCCC(C)(C)C1 C1(NC(c2c(CCC)nns2)=O)(CC)CCN(C(C2CC(C#N)C2)=O)CC1 C(CC(C)(C)C(=O)NCC1CCC1NC(c1sccc1NS(C)(=O)=O)=O)SC c1(CC(C)SC)nc(-c2cccc(Cl)c2)nn1CC1COCCO1 N1(C(c2c(C)nc(CC(C)C)o2)=O)CCN(C(=O)C=Cc2ccsc2)C2CCC12 c1(CNCCNC(C)=O)cccc2nc(C(F)(F)F)sc12 N1(C(COCCN(C)C)=O)CCCCC1C1CCN(C(C2(C#N)CC2)=O)CC1 c1(C(N2CCCC(NC(COC3(C)CCCC3)=O)CC2)=O)nccc2nn[nH]c12 C(CCSc1ccccc1C)(C(=O)NC(C(=O)O)c1nc[nH]n1)c1cn(CC)nn1 C(=O)(CS(=O)(=O)NC1CCCCC1)NCCN(C(C1C(SC)CCC1)=O)C(C)C N1(C(c2ccc(C(F)F)cc2I)=O)CC(S(=O)(=O)C2COC2)C1 C1(CC(=O)NC(C2CCCC2)CC)CCCN(C(=O)C(C)(COC)COC)CC1 C(=O)(C(CCC(C)(C)C)N(C)Cc1ccc(N(C)C)cc1)NCC c1(C(=O)NCC2N(C(C3C(SC)CCC3)=O)CCCC2)cc(Cl)ccc1N C(=O)(C1=Cc2ccccc2C1)NCCC1(C(=O)NCC(C)(O)C(F)(F)F)CC1 CC(C(=O)N1CCCCC1C1CCN(C(c2cncc(N)c2)=O)C1)C(C)(F)F N1(C(C(CNC(c2cc(C)ns2)=O)O)=O)CC(F)(F)CCC1C c1(NC(C2CCC(C)N2Cc2cc(F)ccc2O)=O)cc(C2CC2)cc(F)c1F CP(C)(=O)C1CCC(C(=O)OCC2=CCCCCC2)C1 N1(C(CN(C)C)=O)CC2CS(=O)(=O)CC2(NC(c2cnn(C3CC3)c2)=O)C1 C#CCCCC(C)C(=O)NC(C(=O)N1CC(C#N)C1)C(C)CC C1(C(F)F)(NCC(CC#C)(C)C)CNCCC1C C1(CCC)CCCCN1C(C1CC(NC(C2CC2C(F)(F)F)=O)C(O)C1)=O c1(C(N(CC(=O)NCCCC(=C)Cl)CC(C)C)=O)ccc(C)nc1 C1(C(N2CCCCC(NC(CNS(N(C)C)(=O)=O)=O)C2)=O)CCn2nncc2C1 C12(C(N(CCCNC(c3ccc(CO)cn3)=O)CC)=O)CCC(CC1=O)C2(C)C c1(C(=O)NCc2ccc(CSC)o2)ncccc1NC(=O)NC1CCOCC1 C(=O)(C(CNC(=O)C(CSC)OC)(CC)CC)NCCCCCC#C C(c1ccccn1)=CC(=O)NC1(C)CC(NC(=O)Cc2cc[nH]c2)C1 C=C(F)C1(CC(=O)NC2CC(C(=O)NCC(=O)N(C)OC)C2(C)C)CCC1 c1(CC(N2CCC(C(N(C3CC=CC3)CC)=O)C2)=O)cccc(C)c1Br O=C(CCCn1cccc1)NCC(O)CNC(=O)CCN1CCCCC1 C1(NC(NCC(F)F)=NCCN2CCCCCC2)C2CC3CC(C2)CC1C3 c1(C(=O)NCC2(F)CCN(C(CSSC)=O)CC2)cn2c(n1)CCCC2C O=C(C#CC1CCCCO1)NCC1CCN1C(=O)COc1ccc2c(c1)OCO2 N1(C(c2ccc(COC)s2)=O)CC(O)CC1CNC(C1(C)CCCCC1)=O C1(C(=O)NCC2=CCN(C(c3ccoc3)=O)CC2)CCc2nccn2C1 C(=O)(C#Cc1ccccc1)N1CC2C(C(=O)Nc3c(C)ccc(F)c3)C2C1 c1(C(=O)NC2C(CCCCNC(C=CC)=O)C2)ccnn1C1CC1 N1(C(CC2C(C)=NNC2=O)=O)CCC(NC(=O)NC(C)(C)C)C12CCC2 C1(CC=C)(NC(C2CC2(C)Br)=O)CCN(Cc2cc(OC)ncn2)CC1 N1(C(C=CCN(C(Cc2cn(C(C)C)nc2)=O)C)=O)Cc2ccc(C#N)cc2C1 Cc1cc(Br)ccc1C(N1CCCC(N(C)C(c2cn(C)cn2)=O)C1)=O C1(NC(C(CC=C)C)=O)CS(=O)(=O)C2CN(C(=O)C#CC3CC(F)(F)C3)CC12 c1(C(=O)NC(CC)CN(C(=O)CC2C=CCC2)C)cnc(S)nc1 C(CCC(=O)NC(c1cccnc1)C(=O)NC(c1cc[nH]n1)C)=CC c1(C(N2CCCC(CC=C)(NC(c3cc[nH]c3)=O)C2)=O)ccc2cccnc2c1 Cc1ccc(C(F)(F)F)cc1CN1CC(O)C(O)C1C(=O)O CCC(CC(F)(F)F)C(=O)NCC(C1CC1)N(C)C(c1cccn2nccc12)=O C1(CNC(c2c(CC)nns2)=O)CC2(CC2)CN1C(=O)CCCc1cncs1 c1(C(=O)Nc2ccc(C)cc2-n2cnnn2)cc2n(c1)CCS(=O)(=O)C2 C1(C(=O)NCCC(=O)NCC(C)C)(OC2CN(C(COC)=O)C2)CCC(C)C1 Cc1ccc(C(C(C)C)NCC(N2CC(NS(=O)(=O)C3CC3)C2)=O)cc1 c1(N(C(CN(C(=O)CN2CC3CC3C2)CC)=O)C)csc(C)n1 c1(C(=O)NC2CCN(C(c3cnc(C#N)s3)=O)CC2O)n[nH]c2c1CCOC2 N1(C(c2cnc(C)s2)=O)CCC(F)(C(=O)NCC2(C)CCCC2O)C1 CC(C)C(C)CC(=O)N1CCN(C(c2cc(O)nc(O)n2)=O)C(CF)C1 N1(C(C(CC=C)C)=O)CCC(C(=O)NCC2CN(C(C)=O)C2)(CC)CC1 N1(C(COCCOC)=O)CCCCC1CNC(C12COCC1C2)=O CC(=O)CCCC(=O)N1CCCC(NC(c2ccc(Cl)nc2N)=O)C1 C1(NC(c2onc(C)n2)=O)CCSC12CN(c1nc(C(C)(C)C)nc(C)c1C)C2 c1(C(=O)Nc2cccc(-c3cn(C)nn3)c2)c[nH]c2ccc(Cl)cc12 c1(CC(C)C(N2CCN(c3ccc(O)nc3)CC2)=O)ccccc1F N1(C(=O)Nc2cc(C)no2)CCCC(C)C1CNC1CCC(CC(F)(F)F)CC1 CCCC(C(=O)N1CCCC1C(C)NC(C1(C(F)(F)F)CC1)=O)S(N)(=O)=O N1(C(Cc2c(C)n[nH]c2C)=O)CCCC2(C1)CN(C(C1CC(C#N)C1)=O)CCO2 C1(CNC(C=CC=CC)=O)CC(C)N(C(c2nnn(-c3cccc(C)c3)c2C)=O)C1 C1(NC(c2c(CC)nco2)=O)CC2CCC1C(NC(=O)CCOC)C2 C(=O)(C1OCCc2cc(Br)ccc21)N(S(C)(=O)=O)Cc1ccc(C(=O)O)o1 C1(NC(C2C(C)=C2)=O)CN(C(c2cnc(S)n2C)=O)CC2(CCC2)C1 Fc1ccc2sc(C(N3CCOCC3)C(=O)NC3CCCC3)nc2c1 Cc1ccc(CC(=O)NCC(O)CCNC(c2ccc3c(c2)CC3)=O)c(F)c1F C(CN=c1[nH]c(=NC2CCC3(CC3)C2)c2ncccc2[nH]1)NC(COC)=O CC1(C)CN(C(=O)Cc2cnccn2)CC1CNC(C1CCC(=O)N1)=O c1(C(=O)NC(C)CC2CN(C(=O)C3=C(Cl)CCCC3)C2)coc2c1C(=O)CCC2 c1(C(=O)NCC2CN(C(C(N3CCC(C)CC3)=O)=O)C2)n[nH]c2c1COCC2 Cc1cc(C)n(CC(=O)NCc2cc(C(=O)NC3CCN(C(C)C)C3)cs2)n1 CC1OCCC1C(=O)NCC1CC(C(=O)NC(C(N)=O)C2CC2)C1 N1(C(c2scc(CNC(C(C)(CO)OC)=O)c2)=O)CC2(CCCO2)C1 C#CCC(CC#C)C(=O)N1CC(NC(=O)CCc2ccc(F)cc2)CC(C)(C)C1 C1(CNC(C2OCCN(C)C2)=O)CC12CCN(C(c1ocnc1C(F)F)=O)CC2 O=C1CC(C(=O)NCC=CCC(N2CCC(N3CC=CC3)C2)=O)CC1O Cc1ccccc1C(C)(C)C(=O)NCCCCC(C)NC(=O)C(C)C C12(CC(=O)NCC(C(C)C)NC(CCc3onc(SC)n3)=O)COC(C)(C1)C2 C1(C)(CNC(Cc2nc(C)[nH]n2)=O)CCN(C(C23CCC(CC2)C3)=O)CC1 c1(OC)ccc(C(=O)NCCN(C(=O)C(N2CCNC2=O)C)CC(C)O)s1 Cc1cccc(N)c1C(=O)N(C)CC1CCCCN1C(C1CCS(=O)(=O)C1)=O CC1(C(=O)NCC(O)CNC(=O)C(F)C2CCCC2)CC=CC1 C12(C(=O)NCCOC)CC1COC2(C)C.C12CN(CC1O)C(=O)c1cn2nn1 N1(C(C2(CC=C)CCCN2C(=O)CC2CCC(=O)N2)=O)CCOC(C)(C)C1C Cc1cc(C(=O)NCC(C2CCCC2)NC(c2ncccc2F)=O)c(Cl)cc1F C1(CNC(CC(CC)C)=O)CN(C(C2CCC(=O)N2)=O)CCC1(C)C C1(C(N(CCCN(C)C(c2sccc2Br)=O)C)=O)C(C)(C)C1(F)F c1(C(C(=O)NCC(C)(C)C(=O)NCC2C(C)C2)(F)F)cc(Cl)ccc1Cl c1(C(=O)NCCN(C(=O)CN(C)C(=O)C2CC2)C(C)C)cn2c(n1)CCC(C)C2 C1(C(=O)NC2CC3(C(C(=O)NC(CC)CCO)C3)C2)CCCCCN1C Cc1nn(C)c(C(N2CCN(C(=O)C(C)(O)C(C)C)CC2)=O)c1Cl Cc1ccc(SC(C)C(=O)N2CCCC2)c(NC(=O)CCC(C)C)c1 c1(OCC)ccsc1C(=O)N(CCNC(C1CC1[N+](=O)[O-])=O)C1CC1 c1(C(=O)NCC2N(C(c3c(C)n[nH]c3)=O)CC2)cc(Cl)ccc1N C1(NC(C(c2ccccc2)N)=O)CCN(c2ccccn2)CC1 c1(N2CCCC(OCCC)C2)nc2c(c(=NCc3nc(O)n[nH]3)[nH]1)COC2 N1(C(C2C(C)CC2C)=O)CCC(N(C)C(C2CC(Cl)(Cl)C2)=O)CC1 c1(NC(=O)NC(C(=O)OC)Cc2ncncc2OC)cccc(C(F)(F)F)c1C N1(C(Cc2cccc(C)c2)=O)CC(C(=O)NC2CCCCC2)CC(C)C1 c1(CNC(CCCSCC)=O)ccc(NC(=O)CN(C)CCOC)cc1 C1(NC(c2cccc(C)c2)=O)C2CCC(C2)C1C(=O)Nc1ncccc1Br Cc1cc(-c2noc(CCc3ccc(I)cc3)n2)c(O)nn1 C1(C)(C(=O)NCCCN(C(c2cc(CCOC)on2)=O)CC)CCCNS1(=O)=O N1(C(C=Cc2n(C)ncc2)=O)CC2CCN(C(=O)C(O)P(C)(C)=O)CC12 N1(C(c2c(CC)nc(C)[nH]2)=O)CC2CN(C(=O)C(F)CN(CC)CC)CC2C1 N1(C(C2C(OC)(OC)CC2)=O)CC2(C(N3CC(OC(F)F)C3)=O)CCC1CC2 c1(C(=O)NC(C)CCCNC(=O)Cc2cccc(O)c2)ncnc2c1OCCO2 C1(CC)CCCC1C(=O)NCCC1CC(NC(=O)COc2ccsc2)C1 c1(C(N2CC3C(C(N4CC5(CCC5)C4)=O)C3C2)=O)ccc(Br)cc1CO C1(CNC(C2CCCC(C)CC2)=O)C2CCCC1N(C(=O)Cc1ccoc1)C2 C#Cc1c[nH]nc1C(=O)NC(c1ccnn1C)C(=O)NC1COC(C(C)C)C1 C1(CNC(c2cccc([SH](C)N)c2)=O)CN(C(C2CCCC(N)C2)=O)CC12CC2 c1(CN2C(C(=O)NCC(C)C)CC(C)C2)ccc(N(C)C)c(C(F)(F)F)c1 C1(NC(C)=O)CN(C(C2CCN(CC(=O)O)CC2)=O)CC1n1cccn1 c1(C(C(=O)NCC2C(NC(c3ccncn3)=O)COC2)O)ccc(Cl)cc1F N1(C(CN(C)CC)=O)CC2CCCC2(NC(=O)C(c2ccc(Br)cc2)C)C1 c1(CC(N2CCC(NC(C=C(CC)C)=O)C2CC)=O)cnc(Cl)cc1C C(c1cc(Br)ccc1F)=CC(=O)NCc1nc(C(C)(C)C)[nH]n1 C1(C(=O)NC(C)C(=O)NC2CC2F)(CC)CCOC1 C1(F)(C(=O)NC2CN(C(C)=O)C2)CCN(C(c2ccc(F)cc2)=O)C1.C1(C)(N)CC1 c1(CC)nc(C)oc1C(N1CC(C(=O)N(C2CCOCC2)C)C1)=O N1(C(c2c(OC)ccs2)=O)Cc2ccccc2CC1CNC(C1(C(N)=O)CC1)=O c1(C(=O)NCC(CCNC(c2c(CC)non2)=O)O)cc([N+](=O)[O-])cc(C)n1 c1(OC)cccc(C)c1C(N1CCN(C(=O)CNC(=O)C(C)CO)CC1)=O Cc1snnc1C(=O)NCC(C)(C)CNC(c1cnccn1)=O C1(C(N2CCCC2CCCO)=O)CC(O)CN1C(=O)CCc1ccccc1 C1(C(=O)NCC2C(O)C(O)CN2C(=O)C(F)CC2CC2)C2CC3CC(C2)CC1C3 C(C(C)CC(=O)NCc1occc1C(=O)NC1CCS(=O)(=O)C1)OC N1(C(C(C(C)C)NCC)=O)CCN(C(C2(C)CC2)=O)CC12CC2 N1(C(C2(CC)CCCO2)=O)CCOCC(NC(=O)C=Cc2cn[nH]c2)C1 c1(-c2ccc(C(=O)NC34C(CN(c5nnc(C)o5)C3)C4)o2)cccc([N+](=O)[O-])c1 C#CCC(CC(F)F)C(=O)NCCCC(N1CC(F)(F)OC(F)(F)C1)=O c1(N2C(C)(C)C(CNC(c3ccnc(C4CC4)n3)=O)CC2)nc(Cl)nc2[nH]cnc12 c1(C(C(=O)NCC(C)NC(=O)CCn2cc(Cl)cn2)O)cc(F)c(F)cc1F Cc1c(CNC(C2CC(N(C(=O)CC3COCC(C)O3)C)C2)=O)cccc1F C1(C(=O)NCCC(C)N(C(=O)C=CC(N)=O)C)Cc2nccnc2C1 CS(=O)c1cccc(C(N2CC3C(NC(c4cc(O)ncc4F)=O)C3C2)=O)c1 c1(CC(=O)NC2C(CNC(c3c(C)ccnn3)=O)COC2)c(F)cccc1F c1(C(N(C2CCN(C(c3ccc(COC)s3)=O)C2)C)=O)n[nH]c2nccc(Cl)c12 c1(C(=O)NCC2N(C(c3n(CC)nnc3)=O)CCCC2)cccc2ncccc12 N1(C(C2CC(COC)C2)=O)CC(C2CCCN(C(C3CC4(CCC4)CO3)=O)C2)C1 C(=O)(C(C)C(O)C(C)CC)Nc1cccc(OC)c1.C1(=O)CCOCCO1 c1(C(N2C(C)CCC(NC(c3cc(CC)sn3)=O)C2)=O)cccc2c(C)[nH]nc12 c1(C(=O)NCC2C(C)CN(C(=O)C(O)C3CCC3)C2)cc2ccncc2s1 CCS(=O)(=O)c1ccccc1C(=O)N(C(C)CCNC(C1COC(=O)N1)=O)C C1(CNC(CC=C=C)=O)CC(C)N(C(C2CC(OC)C2)=O)C1 CC#CCCCC(=O)N1CCC(CC(=O)NCC(CC)C(C)(F)F)C1 N1(C(=O)OC(C)(C)C)CCOCC1CCOC(C1CC(=O)N(CCF)C1)=O c1(C(=O)NCC(C)NC(c2ccc(NC(=O)OCC)cc2)=O)ccnc(Cl)c1F CCCC(C(=O)N1CCCC1CCCNC(=O)C=C1CCCC1)N(C)C c1(C(=O)OCC#N)nc(NC(CC2(C(=O)OC)CCCCC2)=O)c(C)o1 N1(C(C2C(C)CC=CC2)=O)CCC(C2CN(C(C3CC4(CCC4)CO3)=O)C2)CC1 c1(C(=O)NCC2CN(C(CCCC#C)=O)C(C)(C)C2)ccc2ccc(C)cc2n1 C1(CC)CN(C(=O)Cc2ccc(OC(C)=O)cc2)CC1NC(=O)CCCC1CC1 c1(NC(C)=O)cccc(CC(=O)NCCCC(C)NC(=O)C(O)C(C)C)c1 C(=O)(C1COc2cc(C)c(C)cc21)NC1(NC(C(CCOC)OC)=O)CC1 c1(NC2CCCN(C(c3nc(CC)oc3)=O)C2)cc(O)nc(C)n1 C(=O)(CS(=O)(=O)Cc1cccs1)NC(CCNC(c1c(CC)cncc1)=O)C c1(C(=O)NC2C3CN(C(c4c(CC)[nH]nc4Cl)=O)CC32)c[nH]nc1S(N)(=O)=O c1(C(N2CCN(C(CS(C)(=O)=O)=O)C3(C2)CC3)=O)cc(S(N)(=O)=O)ccc1O c1(CC(N2C(CNC(C3CC(OC)(OC)C3)=O)CC2)=O)ccc(F)cc1C C12(CNC(C3OCCN(C(Cc4c(C)n[nH]c4)=O)C3)=O)CCC(C1)C(=O)N2 c1(C(=O)NC(CN2CCC(C(=O)O)CC2)C2CC2)ccc2nc(C3CC3)oc2c1 O=C(C1=NOC2(CCCN(S(=O)(=O)C3CCOCC3)C2)C1)N1CC(F)C(F)C1 Cc1ccc(F)cc1-n1nc(CC2CCOCC2)nc1CO.SC CCN=C(NCC1CC=CCO1)NCC1CCC1 Cn1ccc2c(C(=O)NCC3(F)CCCN(C(=O)CCC=CBr)C3)ncnc12 CC1CCCCC1(CNC(c1nc(C(C)(C)C)no1)=O)NC(c1nonc1N)=O C(=O)(C1CCCc2cccnc21)N1C2CC(NC(c3cn(C)nc3)=O)CC1CC2 C(=O)(C(C)(C)C(=O)NC)NC1C(N(C)C(C2CCC2c2nc[nH]n2)=O)CCCC1 C1(C(=O)NCCCCCNC(=O)COC2CC(F)(F)C2)CC2(CC2)CO1 C(=O)(C1=CC2(CCN(C(=O)C=Cc3nccs3)C2)C1)NCC(CC(=O)OC)C Cn1cc(S(C)(=N)=O)c(CNC(=O)Cc2ccc(-n3cnnc3)cc2)n1 N(C1CCOc2c(F)cccc21)c1nccc(N(C)Cc2ccc(CC)cc2)n1 c1(OC)ccc(C(N2CCC(NC(c3cc(CO)cc(F)c3)=O)C2)=O)c(F)c1F CC(CC(=O)NC1CN(C(C2C(=O)C2(C)C)C2CC2)CC(C)(C)C1)CC(F)(F)F C(=O)(CC(C)(C)CC(=O)N1CCCC2CN(C(C3CC(F)C3)=O)CC12)OCC c1(C(N2C(C)(C)C(C(=O)NCC=C(Cl)Cl)CC2)=O)cnn2ccccc12 Cc1cccnc1CNCC1CCC(C(=O)NC2CN(C(N)=O)C2)CC1 C1(C(N2CCCC(N3CCCC3)C2)C(=O)NC2CC2)CCCN(CCF)C1 N1(C(c2c(C)noc2C)=O)CC(NC(=O)C(C(C)C)n2ncc(N)n2)CC(O)C1 Cc1ccc(C(=O)NC2(CNC(=O)C(c3cnn(C)c3)C)CCOC2)cc1C#N N1(C(C2CCC(OC)CC2)=O)CCC(C)(C(N2CCCC(CCCO)C2)=O)CC1 C1(COC)(CNC(c2csc(NC=O)n2)=O)CCN(c2cc(Cl)nc(C)n2)CC1 C(CC(N)=O)(C(=O)Nc1ccc(C(N)=O)nc1CO)NC(C1C(C(=O)OC)C1)=O N1(C(CC2(C)CC2)=O)CC2(C1)CN(C(c1cc3c(cc1Cl)OCO3)=O)CCO2 Cc1ccccc1CNC(=O)C(F)C(C)C.C1=CC(=O)NC1(C)C N1(C(C=Cc2c(C)coc2C)=O)C2CCC1CN(C(C1CN(C)CCO1)=O)C2 CC1CN(C(C2CCC(O)CC2)=O)CC2(CCN(C(C3COC(C)(C)C3)=O)C2)O1 Cc1nnc2n1CC(C(=O)N(C)C)N(CC(N1CCCC1c1ccc(Br)s1)=O)C2 C12(NC(C3CCCC(OC)C3)=O)CCC(C1)N(C(c1ncc(F)cc1C)=O)C2 C1(NC(N(CCCCC=C)C)=O)CCC2(CCN(C(=O)OC(C)(C)C)C2)C1 N1(C(CCC(C)(C)F)=O)CCC2CN(C(c3cnn4c3CCCN4)=O)CC12 c1(C(N(C)C)=O)cccc(CN2CCN(C(C3(S(N)(=O)=O)CC3)=O)CC2)c1 C(=O)(C1CCCc2scnc21)N1C(CNC(c2n(C)c(Cl)cn2)=O)C(C)CC1 C1(CCOC)CN(C(=O)CNC(=O)OC)CCN1C(c1ccc(C(N)=O)nc1)=O Cc1c(C(N2CC(C)(CNC(c3ccc(Cl)c(Br)c3)=O)C2)=O)cccc1O C1(NC(=O)CNC(=O)NC2CC2)CCSC12CN(C(=O)CC=C(Cl)Cl)C2 N1(C(C2(C#N)CC2)=O)CC2(CO)CC1(C(N1CCC(CN=[N+]=[N-])C1)=O)C2 c1(C(=O)Nc2nnc(SC(F)(F)F)o2)ccc(S(=O)(=O)NC(F)C2CC2)cc1 C1(CC)CC(C(=O)N(C2CC2C2CC2)C)CCN1C(c1ccsc1C#N)=O C1(CSC)CCCN(C(c2ncccc2Br)C(=O)OC)C1 C1(C(=O)NCCC(CCC)C2CC2)CN(C(=O)CC2CC3CC3C2)CCN1C Cc1nc[nH]c1C(=O)NC1COCC1NC(=O)COCC(F)(F)F C1(C(=O)NC(C)C(=O)N(C)Cc2ccccn2)CCN(C)C1 CC1(C)CN(CCCO)S(=O)(=O)N2CC3CC4CC3C2C4C1 O=C(C1CCc2nccn21)NC1CC(CNC(C23COCC2C3)=O)C1 C1(C(=O)NC(c2ccc(F)c(F)c2)(C(=O)OC)C)CSC(c2cccs2)=N1 c1(C(=O)NCC(C)NC(C2(OCC)CCOC2)=O)ccnc(OCC)c1 c1(CC)nc2ccccn2c1Nc1nc(C(C)(C)C2CC2)n[nH]1 C(c1ccc(F)c(C)c1)=CC(=O)NC1CC(C)(NC(C(CC)n2ccnc2)=O)C1 c1(NC(C2(SC)CN(C(c3sc(O)nc3C)=O)C2)=O)ccc2ccncc2c1 C12(C(=O)NC3C(C)(C)C(C=O)C3)CCCN(CC1)C2.C1(OCCC2CC2)CCC1 Cc1c(CNC(=O)C(O)CCNC(C2(CO)CCCC2)=O)cccc1F c1(C(N(CC(CC)NC(=O)C(C(C)C)N(C)C)C)=O)c[nH]nc1S(N)(=O)=O c1(C(=O)NCCN(C(=O)C(O)c2ccco2)C)csc2cncn12 S(=O)(=O)(c1ccc(O)c(C(=O)O)c1)N1C(C(C(C)C)C(=O)O)CCCC1 c1(CC)ncc(C(=O)NC2CC(CCC(=O)N3CC(c4nncn4C)C3)C2)s1 C12(C(=O)NCC3CN(C(C4C(C)CN(C)C4)=O)C(C)(C)C3)CC3CC1C2C3(F)F C1(CC=C)(NC(c2csc(Cl)n2)=O)CCN(C(c2cc(NC)ccn2)=O)C1 C(=O)(C(N=[N+]=[N-])C(C)C)NCC(CCC)C(=O)NC1CCCC(F)(F)C1 CON(CC(C(=O)C(C)C(F)F)CCCCC)C(=O)CCC(C)C N1(C(C2(CCC)CCC2)=O)CC2CC(C(=O)NCCC#CCO)(C2)C1 c1(C(N(CC(CN(C(C=CC=CC)=O)C)O)C)=O)c(C)noc1N C1(C(N(CCCC)CCNC(C2CCC(NC)CC2)=O)=O)CCC2CCCCN12 C1(C(N2CCC(CC(=O)NC(CCSC)CO)C2)=O)CCC2(C(C)C)CC12 C(=O)(C#CC1CCOCC1)NC1(C)CC(C(N2CC3CCCC2C3)=O)C1 c1(C(=O)O)cc(CN2CCC(O)(C(=O)Nc3c(Br)ccnc3Br)C2)ccc1O C1(NC(C2C(C)CC(=O)N2)=O)CN(C(C2CC(=O)C2)=O)CC2(CC2)C1 c1(NC(c2cc3sccn3c2)=O)nc(Cl)c(Cl)cc1Cl C1(C(=O)NCC(CNC(c2ncc(OC)nc2)=O)(C)OC)CC(=O)CC12CCC2 N1(C(C2C(NC(CCc3cncc(C)c3)=O)C2)=O)CCCN(C(C)CO)CC1 c1(CC(=O)NC2(CF)CCN(C(c3c(CC)ocn3)=O)C2)cc(Cl)cc(Cl)c1 N1(C(CCOC)=O)CC(NC(=O)C(c2cncn2C)O)C(C2CC2)C1 S(=O)(=O)(c1ccc(F)cc1F)NCC(N1CCN(Cc2n(C)nnc2)C2C1C2)=O C1(NC(CN(C(=O)C2=CCCC2)CC)=O)CC(O)C12CCC2 c1(C(N(C2CCN(C(C3CC(C)=NO3)=O)C2)CC#C)=O)n[nH]c2c1CCC2 C1(CCOCC)(CNC(C2CC2C(C)NC(=O)CC2CSC2)=O)CCCCC1 Cn1nc(C(=O)NC2CCC2NC(=O)CCc2ccccc2F)nc1Br c1(CC)nc(C)c(C(=O)NCC(CNC(=O)C2=C(Cl)CC2)OC)s1 C1(NC(C2(COC)C=CCC2)=O)CCC(C)N(C(=O)C2=COCCO2)C1 n1(CCOC)cc(C(=O)NCCCC(C)NC(c2ncsc2C)=O)c(C)n1 C(=O)(C1CCc2snnc21)N1C(CNC(C2(C(=O)NC)CC2)=O)CC(O)C1 N1(C(C2C3(CC(C)OCC3)C2)=O)CCc2cccc(C(=O)NC(C)CO)c2C1 C(CCCCCNC(C1C2CCC1(c1ccco1)C2)=O)NC(c1cccs1)=O C(C(N=[N+]=[N-])C(=O)N1CCC(CCC(=O)N(C)CCO)CC1)OCC CC1(NC(=O)CC2CCS(=O)(=O)CC2)CCCN(C(=O)C=Cc2ccsc2)C1 C(N=c1[nH]c(Cl)ncc1[N+](=O)[O-])C1CN(C(CC2CC(CC)OCC2)=O)CC1(C)C C1(C(=O)NCCCN(C(=O)Cc2cccc(F)c2Cl)C)C2CC(F)(F)CC12 C1(NC(CNC(C)=O)=O)CCCN(C(c2ccc(-c3cccnc3)s2)=O)CC1 N1(C(C(CC2CCC2)NC(c2cc(C3CC3)on2)=O)=O)CCN(C2CCC2)CC1 C1(C(N2CCN(C(=O)Cc3cnns3)C(CCO)C2)=O)CCCC1C1CC1 c1(N2CCC(CC)C2)ncc(S(=O)(=O)NCC(C)NC(=O)N(C)C)cc1Cl N1(C(c2cc(CC)no2)=O)CCOC(CCCNC(=O)C(C)NC(=O)NC)C1 c1(C(=O)NCC2CC(CNC(CC=C=C)=O)OC2)csc2ccncc12 N1(C(CCCC)=O)CC(C)N(C(=O)C=Cc2ccc(C)s2)CC1C C(=O)(C(C(C)(C)C)C1CCC1)N.Cc1cc(CCC(=O)NCC(C)CCC)no1 c1(CCCC)nnc(SC)n1CCNC(=O)CCSC.c1(N)cccc(Cl)c1 c1(C(=O)NC2(CO)CCCN(C(CCC(CC)OC)=O)C2)n[nH]c2c1COCC2 CC(C)(C)CCCCC(=O)N1CC(=O)NCC1C(N1CC(CCO)C1)=O c1(C(c2nnnn2CCC2CC2)NCc2csnn2)cn(-c2ccccc2)nn1 Cc1cccn2ncc(CNC(c3cc4ccsc4cn3)=O)c12 CC1(NC(C2CN3CCC2CC3)=O)CCCN(C(c2cc(Cl)c[nH]2)=O)C1 c1(CNC(=O)NCc2cc(C3CCOCC3)no2)ccc(C(F)(F)F)cn1 N1(C(C(C)=C(CC)C)=O)CC2(CNC(C3CC3(C)COC)=O)CC1CO2 Cc1cc(F)c(CC(N2CCC(NC(C3(N(C)C)CCC3)=O)C(C)C2)=O)cc1F c1(N(CC(CN(C)C(c2cc(CC3CC3)on2)=O)O)C)cc(C(N)=O)nc(Cl)n1 c1(C(N(C)C(C2CCN(C(C(CC)(C)O)=O)C2)C2CCCO2)=O)cnc(O)c(F)c1 N1(C(CCCOC(C)C)=O)CCC2CN(C(C34CC(C)C3C4)=O)CC12 C1(NC(c2cc(O)ncn2)=O)CCCCC1CNC(c1cccc(CO)n1)=O C1(CNC(C(CCOC)NC(=O)C=CCCC(C)C)=O)Cc2nccn2C1 CC1CC(c2ccoc2)CN1S(=O)(=O)CC1COC1 Cc1csc(C(=O)NC2CC2NC(=O)CSc2ccc(O)cc2)c1C CCCCC(O)C(C)C(=O)N1CCN(C(=O)C(COCC)N=[N+]=[N-])CC1CO C1(CC)CN(C(=O)C(O)C(C)C)CCN1C(=O)CCCN(C)C(C)=O c1(OCC(=O)NCC2C(CNC(C(C)OC)=O)C2)cccc(C)c1.C(CC(C)C)O CC1=NNC(=O)C1CC(=O)N(C)CC1CCCN1C(=O)C(c1cnn(C)c1)C c1(C2(C)CC2)nc(N2CCN(C(C3CCCC(C)C3)=O)CC2)cc(Cl)n1 C(=O)(C(C)(C)CNC(C1CCN(C(c2cnc(C)s2)=O)C1C(C)C)=O)OC c1(C(=O)NC2CCN(C(Cc3nc(C)sc3)=O)CC2F)sc2nnc(S)n2c1C C(=O)(C1CSc2ccccc21)NC1(CCNC(C(=Cc2cccs2)C)=O)CC1 C1(CC(N2CCC(NC(C3(N=[N+]=[N-])CC3)=O)C(F)C2)=O)CCC2(CCC2)CO1 C12(NC(C3(COC)CC3)=O)CCC(CC1n1cc(-c3csc(C)c3)nn1)C2 c1(C(=O)NC2C3(CCN(C(CNC(N)=O)=O)CC3)C2)cccc2c(Br)n[nH]c12 C1(C(N2CC(O)(CNC(c3c(C)sc(Cl)n3)=O)C2)=O)OCC2CCCC12 C1(C(N2C(CNC(C(CCCOC)C)=O)CCCCC2)=O)CN=C2N=CNN2C1 C(=O)(C(C(C)(C)O)NC(C)=O)NCC1CC(C(=O)NCC2CC(OC)C2)C1 C(CN=C(NC1(CC2CC2)CC1)N1CCC(n2ccnn2)CC1)C(F)(F)F C1(c2onc(NCc3c(C)c(Cl)c(Cl)s3)n2)(CN)CC2CCCC2C1 C(CC(CNC(=O)C(O)c1cnc[nH]1)NC(c1csc(C(C)(F)F)n1)=O)OC CCCCCCC(C)CC(=O)N1CCCC(CO)(NC(c2nc(CC)no2)=O)C1 c1(C(=O)NC(C2CCN(C(C3CCCC3)=O)C2)C)cc2c(Cl)cccc2[nH]1 C1(O)(C(CNC(c2c(OC)c[nH]n2)=O)C)CCN(C(c2ccnnc2S)=O)C1 N1(C(c2ccc(C)cn2)=O)CCC(C)C(NC(=O)CC(C)(C)O)C1 C#CC1(O)CCCN(C(c2cccc(Br)n2)C(=O)NCCSC)C1 C#CC1CCCN1C(=O)C(c1cccs1)NC(=O)CCC(=O)C1CC1 Cc1nc2c(s1)CCCC2C(=O)N1CCC(CNC(c2cnsc2)=O)C(F)(F)C1 c1(N(C)CC2CCCO2)cc(N2CCC(C3OCCO3)C2)nc(C(F)(F)F)n1 C1(CC(=O)NCCOC(C)=O)CCCCC1NC(=O)Cc1ccc(C)s1 c1(C(=O)NCC(CC)NC(=O)COCC2CCCCO2)cc2nc(Cl)ccc2s1 N1(C(C(C)C(F)F)=O)CC(NC(c2cc(F)ccc2Br)=O)C(C2CC2)C1 C1(C(N2CCC(OC)(CNC(C3CNC(=O)C3)=O)C2)=O)CC2CCC(C1)C2 C(c1c(C)coc1C)=CC(=O)NCC(CCOC)NC(=O)CC1(C)CCCCC1 C1(C(=O)NCCOCCOCCNC(c2cnc[nH]2)=O)CN2CC3CC2(CO1)C3 CCCCC(C(=O)N1CCCC1C1CCN(C(c2nocc2Br)=O)CC1)N(C)C Cc1cnc(F)cc1C(=O)NC1CCCCN(C(C23CC2C3)=O)C1 c1(N(CC(CCC)C)C)nc(NC(C)CCn2cncn2)c2c(ncn2CC)n1 c1(OC)ccc(NC(=O)C(=O)Nc2cnsc2)c(C#N)c1 N1(C(C2C(CC)CC2)=O)CC(C(=O)NCCCS(N)(=O)=O)C(F)C1 C12(C(N(CC(C)NC(=O)Cc3ccccn3)C)=O)CCC(C1)C2(C)C c1(CC)nncn1NC(=O)C(CCC)NC(=O)C(N1CCOC1=O)C C(=O)(CCCCO)NCC(=O)N(C1CCN(C(C2CCS(=O)(=O)N2)=O)C1)C CC1=C(C)CC(C(=O)NC2CC(C(=O)NC3CCCCC34CC4)C23CCC3)CC1 CC(C(=O)NCC(C1CC1)N(C)C(c1cnnc(O)c1)=O)C(F)F N1(C(C2(COCC)CC2)=O)CCC(C(=O)NCC2CC3OC2C2CC32)=C(F)C1 Cc1nn(C)cc1C(C(=O)NC(C)(C)C)NC1(c2ccc(Cl)cc2)CCOCC1 C(CC[Si](C)(C)C)NC(N1CCC(C(=O)NCC)C1)=O C1(NC(C(CC)N(C)C)=O)CCN(C(=O)CC2CCN(OC)CC2)C12CC2 CC(C)(C)C(CNC(C1(C)CC1C(F)(F)F)=O)NC(c1cnncc1O)=O C1(C(=O)COCC)(OC)CC1.C(CCNC(C1CC1(C)N(C)C)=O)NC=O C(CC(O)C(F)(F)F)NSCC.C1CC(=O)NOCC(=O)N2CCCC12 CC1CN(C(=O)CC2CCCCC(=O)N2)CCC1n1cc(-c2ccn(C)n2)nn1 N1(C(Cc2c(C)nc[nH]2)=O)CC(C)CCC1CNC(=O)CC1(C#N)CCCCC1 C1(CN(C)C(C2COCCN2CCF)=O)CCN(C(=O)COCC(F)(F)F)CC1 c1(-c2cn(CC(=O)N(CCOCP(C)(C)=O)C3CC3)nn2)cccc(O)c1 N1(CC(=O)NC(C2CCN(C(=O)CC(C)c3ccco3)C2)(C)C)CC(=O)NC1=O N1(C(C2(SC)CC2)=O)CCN(C2CN(C(c3cnc(O)o3)=O)C2)CC1 C12(C(=O)NC(C=C)C)CC(CN(C(=O)CCS(=O)(=O)NC)C1)C2 c1(OC)ccc(CNC(c2cnn(CCF)c2)C)c(F)c1Br c1(C(N2CCCC(C(C)NC(=O)C3=CCSC3)C2)=O)c(F)cc(F)cc1F c1(C(C(=O)NC2CCOC2)N(CCCOC)C2CC2)cc(C)c(Br)c(Cl)n1 N1(C(C(CCC)C)=O)CC2(C1)CN(C(=O)C(N)=O)CC2OC c1(C(=O)NC(CCC=C)(C)c2cccc(Br)c2)ccccc1S(=O)(=O)N(C)C C1(CNC(C(COC)C)=O)CCCCN(C(=O)C(C)N(C)C)C1 N1(C(CCC)=O)CC(NC(=O)C=Cc2ccc(C(=O)O)o2)CC12CCCC2 C(=O)(C1CCc2nnc(C)n21)NC1N(C(=O)Nc2c(C)cc(O)cc2)CCC1 Cc1cc(C)c(C(N2CCCC(N(C(=O)Cn3cccn3)C)CC2)=O)c(S)n1 C1(C(N(C)CC2(O)CN(C(c3ccc(C(C)C)cc3)=O)C2)=O)CCN(C)C(C)C1 Cc1ccc(C(=O)NCC2CCN(C(=O)CCCCC(F)F)C23CC3)c(O)c1C Cc1cn2c(CC(=O)NC3CC(N(C)C(c4ccc(F)cc4F)=O)C3)csc2n1 CN(C)S(=O)(=O)NCC(=O)NCCC1CN(C(C2CCCN(S(C)(=O)=O)C2)=O)C1 c1(CC(N2C(C(C)NC(C3CCSCC3)=O)CCC2)=O)cccc(N(C)C)c1 c1(CC)cccc(C)c1C(N1CC2CC(NC(c3cnn(C4CC4)c3)=O)C1C2)=O c1(CCCC(=O)NC2C(OCC)COCC2)nc2cc(Cl)ccc2s1 Cc1cc(C#N)cnc1NC1CCCN(C(C2(F)CCCOC2)=O)C1 c1(C(N(C2CCCN(C(c3cc(C(C)(C)C)no3)=O)C2)C)=O)cc2c(s1)CCC2 c1(NC2CN(C(C(C)Cc3ccncc3)=O)C2)cnnc(Br)c1 c1(C(N(CC)CC2CCCN2C(=O)CSC(F)F)=O)cccc(CO)n1 c1(C(N(CCCNC(CCC(CC)OC)=O)C)=O)cc(N)c(N)cc1F c1(C(CNC(C(=O)NCC(C(C)C)Oc2cccc(Cl)c2)=O)N)ccc(F)cc1 C(=O)(C(C#N)C(C)C)NCC#CC(=O)N(CC(COC)C)C(C)C c1(C(=O)OC)ccc(C=CC(N2CC(C)(NC(C3CC(N(C)C)C3)=O)C2)=O)o1 CC#CCCCC(C)(c1nnnn1CC(F)F)NC(c1ccc(OC)c(OC)c1)C c1(C(=O)Nc2c(OC)ccc(O)c2)cc(-c2cccc(F)c2)cc2c[nH]nc12 C1(NC(c2cn(C3CN(C(=O)C(C)C(C)C)C3)nn2)=O)CC(=O)N(c2cnn(C)c2)C1 C1(CNC(c2ccnc(C)n2)=O)CC2(CC2)CN1C(=O)C(C1CCCCC1)F Cc1nn(C)c(C(=O)NCC2(C)CCN(C(=O)C(C)OC(C)(C)C)C2)c1Cl N1(C(CCCCOC)=O)CCC2(CC2NC(c2ccncc2F)=O)C1 CN1CCOCC1C(=O)NCCn1cc(C(=O)NCC2CC(F)C2)nn1 c1(C(=O)NC2CCN(C(C3(C)C(C)(C)C3)=O)C2)ccc(-n2cnnn2)cc1Cl C(=O)(C(C)(C)C1=CCSCC1)N(CCC(C)NC(C1CC1C(F)(F)F)=O)C C1(NC(c2cnccc2Cl)=O)CCC12CCN(C(=O)CC1CCCCO1)CC2 C1(C(=O)NC2(C)CC(NC(C3C(C)(C)OC(=O)C3)=O)C2)CCCCN1S(N)(=O)=O C(C)(C(=O)NC1CCC1C(=O)N(CC(F)F)C)OCC=C c1(C(N2CCC(NC(C3(CO)CCCO3)=O)C(F)C2)=O)cc(Cl)cc(Cl)c1Cl c1(OC)cc(CN2CC(O)CC2C(=O)NCCCc2ccncc2)ccc1Br CC1(CNC(C2CC(F)(F)C2)=O)CCCN1C(c1cn(CC(F)(F)F)cn1)=O c1(C(N)=O)ccc2c(c1)C(C(=O)NCCn1cc(Cn3nc(C)cc3C)nn1)CO2 CC1(C)CC(C(N2CCC(C(C)(C)C)C2)=O)CN(C(C2OCCC2(C)C)=O)C1 C1(C(=O)NCc2n(C)nnn2)CCCCC1(C)NC(=O)CCc1cccs1 C1(CC(N2CCN(C(C)=O)CC2)=O)CC(C)(C)CN1C(=O)CN1CCC1C CN1CCC(N(C(C2CC23CCOC3)C(=O)NC2CCOC2)C)CC1 N1(C(C2(c3ccccc3F)CC2)=O)CCN(C(C2CC3C=CC2C3)=O)CC12CC2 C(C(CC(C)C)NC(c1ccc(COC)[nH]1)=O)NC(C(C)N(CC)CC)=O Cc1[nH]nc(C(=O)NC(C(=O)N(CCCC(C)O)C)C2CCCC2)c1C C=C=CC(C)C(=O)N(CCC(=O)N(CC)CC)CC=C C1(CNC(c2cnc(SC)s2)=O)CC2CCC(C1)N2C(c1cnc(C)c(N)c1)=O c1(OC)nccc(CNC(C2CC(NC(c3csc(Cl)n3)=O)C(O)C2)=O)n1 c1(COC)ccc(NC(=O)CCN(C)C(c2cn(CCF)nn2)=O)cc1 c1(OCOC)ccc(C(=O)NC(C)C(C)NC(=O)Cn2cc(CO)nn2)cc1 C(CS(=O)(=O)CC(=O)NCC1CCC(C)N(C(=O)CSC)C1)OC C1(NC(c2cc(F)c[nH]2)=O)CCCCC12CCN(C(=O)C1=CCCC1)CC2 c1(N(CC(CN(C)C(C2CCCC2(C)C)=O)O)C)ccc(C#N)cc1[N+](=O)[O-] C(CC(=O)Nc1ccccc1Cl)(C(F)(F)F)NC(c1nn(C)c(O)c1)=O C=C(C)CC(C(=O)NCC(CC(=O)NCCC1CCOC1(C)C)C1CCC1)OC c1(-c2cc(NC(C)=O)ncc2)n[nH]c2c1CN(C(=O)Nc1cccc(Br)c1F)C2 c1(CCC(=O)NC2C(CN(S(C)(=O)=O)C(C)C3CC3)C2)cnn(-c2ccccc2)c1 C1(C(=O)NC2CC2)CC2CCC(C1)N2C(c1cnnn1C1CC1)=O c1(C(N2CC(NC(CC(CC)OC)=O)CC3(C2)CC3)=O)cc2c(C)n[nH]c2cn1 C1(CC)CCc2sc(C(=O)NCCCCCCNC(c3cocc3C)=O)cc2C1 c1(C(N2CC3CN(C(=O)CC45CCCC4C5)CC3C2)=O)ccc2nonc2c1 c1(OC)ccc2[nH]cc(CN3CC4CC3CN4C(C3CCCCC3(C)C)=O)c2c1 O=C(CCC(=O)N1CCOCC1)NCC(CO)NC(c1cn(C2CC2)nn1)=O c1(NC(=O)NC(Cn2c(CC)ncc2)C)ccc(Cl)cc1-c1ccccc1 c1(CC)cc(F)c(C(c2nnnn2C2CCOC2)NCCc2cnoc2)cc1Br S(=O)(=O)(c1cnn(C)c1)NCC(=O)NCC=CCNC(CC1C(C)=NNC1=O)=O c12ccc(cc1)S(=O)(=O)NC2=O.Cc1cnncc1NC(=O)C(=O)NC.C(CO)N Cc1cn2ccnc(C(N3CCC(NC(=O)CC(C)CC(F)(F)F)C3)=O)c2n1 C(CC(F)F)(C(=O)NC1CCCC1(C)C)N(C(c1nnn(CC)c1C)=O)C N1(C(c2c(C)nn(C)c2C)=O)CC2CCC(C1)N2C(=O)Cn1nc(C)c(Cl)c1C c1(C(=O)NCCC2N(C(C(CC)C)=O)CC(OC)C2)ccc(F)c(Cl)c1N S(=O)(=O)(c1ccc(C(C)(C)C)cc1)N1C2CN(C(C(C)(F)F)=O)CC21 C1(C(N(CC=C)C(C)C)=O)CCC(CCl)CC1.c12coc(c1)CNC2=O.C(C)(=O)N Cc1ccc(-n2nc(CC(F)(F)F)nc2C2CC2(c2ccccc2)C)c(C)c1 N1(C(c2c(C)cns2)=O)CC2CCCC(NC(c3ccnc(F)c3)=O)C2C1 N1(C(C(C2CCCC2)NC(C=C=C(C)C)=O)=O)CCC(C)(CN(C)C)CC1 c1(CN2CCC(C(=O)NCc3cccnc3)C(O)C2)cc(O)c(O)c(O)c1 c1(C(N(CCCCC(=O)NCc2ccsc2)C)=O)cc2cccnn2c1 N1(C(CCC=C=C)=O)CCC2(CCN(C(=O)C(F)(F)CCC)CC2)C1 N1(C(C2CCN(C(C3(C)C(C)CCC3)=O)CC2)=O)C2CCC1CC1(C2)N=N1 c1(CN(C2CCN(C)C2)C(c2csc(Cl)c2)=O)cccc(NC(CCC)=O)c1 c1(CC)cc(C(N2CCC(O)(CNC(=O)Cn3cccnc3=O)C2)=O)ccc1F c1(C(N(C)OCC)=O)ccc(NC(=O)Nc2ccc(OCC(C)C)cc2)cc1 N1(C(=O)CN2CCN(C(c3ccc(F)c(Cl)c3)=O)CC2)CCC(F)(CO)CC1.CCO C(N=c1nc(N2CCCCC(C)(F)C2)c2c([nH]1)CSC2)c1cc(OC(C)C)no1 C12(C(=O)NCC(CC)NC(=O)C(F)CC3CCCC3)CCC(O)(CC1)CC2 C1(CC(=O)N(CC(C)(C)NC(C(CCC)N(C)C)=O)C)OC(C)(C)OC1=O c1(Nc2scc(C(=O)N(S(=O)(=O)c3ccc(Cl)s3)CCO)n2)nccc2[nH]ccc12 CN1C(=O)CCC1CC(=O)NC1C2CN(C(=O)CNC(=O)CC(C)(C)C)CC12 C1(C2CN(C(=O)C(C)S(C)(=O)=O)C2)(NC(c2c(SC)cccn2)=O)CC1 N1(C(C(C)Oc2ccccc2Cl)=O)CCN(C(C23CC2COC3(C)C)=O)C(C)C1 N1(C(CCC#N)=O)CCOC(CCNC(=O)CCC(=O)c2cccc(F)c2)C1 N1(C(CCOCCC)=O)CCOC(CNC(=O)C#CC2CC2)C1 c1(CC)ccc(C)c(C(=O)NC2CCCC2NC(C2CC23CC(F)(F)C3)=O)c1 N1(C(c2c(OC)nsc2)=O)CCC2(C1)CN(S(=O)(=O)c1cnoc1C)CCO2 c1(C(N2CC(NC(C(=Cc3ccccn3)C)=O)C2)=O)nccc(C)c1O C(CC(=O)N1CCC(O)(Cn2cc(CCC3CCC3)nn2)C1)(C(F)F)N(C)C c1(C(=O)NCC2CCCCN2C(=O)CCn2ccnc2)ccc2c(c1)CCC=C2 c1(C(N2C3CC(NC(C4CN(C)C4)=O)C(C3)C2)=O)cc2c(cc1Cl)NC(=O)CO2 C1(c2ccc(F)cc2)(C(=O)NCC2C=CCN2C(c2ccon2)=O)CCCCC1 C1(CCNC(C2C(COC)OCC2)c2nnnn2CCCOC)CCC(SC)CC1 c1(CNC2CC(c3ccncc3F)(C(=O)OC)C2)ccc(Cl)cc1F C(CC(C(=O)N1CCC(CO)C1)OC)OCC.C1(C2C(=O)N2)CC1CC c1(OCCC(=O)N(C)CC2CCN(C(C3OCC3(C)C)=O)C2)cccc(Cl)c1Cl C(C)(C)(C(F)(F)F)SCC(=O)NCc1ocnc1-c1cn(C2C(C)CCC2)nn1 C1(N)C2CC3CN(C(=O)CCCNC(CCC(=C)C)=O)C1C3C2 c1(C(=O)OC2CCC(C(=O)OC)C2)cnc2ccoc2c1 c1(C(=O)NC2CCN(C(C(C(C)C)NC(N)=O)=O)C2)cc(N(C)C)cc(C#N)c1 c1(NC2(CNC(C3CCC(C)CC3)=O)CCOCC2)cc2nncn2cn1 c1(C(=O)NCCC2CCC(NC(CC=C)=O)C2)nccc2c1[nH]c1ccccc21 C(=O)(C1Cc2ccccc21)NC(CC=CC(=O)NC(CC=CC)CO)(C)C C(CN=c1ccnc(SC)[nH]1)c1c(OC)cccc1.C(=O)C(F)(F)CO C1(N(C(=O)CCC2CC2(C)C)C)CCN(C(=O)C=C(Cl)Cl)CC1 c1(C(=O)NC2CC(CNC(C(c3ccc(C)s3)C)=O)C2)cccc(Cl)c1F c1(C(=O)NC(c2ccc(Cl)cc2)CCO)ccc2cccc(Br)c2n1 N1(C(=O)C=CBr)CCC2CCC(NC(C3(C4CC4)CC3)=O)C1C2 C(CS(=O)(=O)C(F)(F)F)NC(c1c2cc(-c3n(SCC)ncc3)c(N)cc2oc1)=O C(=O)(CC(O)C(C)C)NC(CCOCC)C(=O)NCc1cnn(C)c1O n1(CC)c(C)nn(CC(=O)N(C(C)CNC(=O)C(CCSC)N(C)C)C)c1=O C1(C(=O)NC2CC(CCNC(=O)CNC(N3CCCC3)=O)C2)C(F)(F)C12CCC2 C1(C(N(C)CCNC(=O)CCc2nncn2C)=O)CCC(C)(F)CC1 c1(C(N2CC3(CN(C(Cc4n(C)cnc4)=O)C3)C2)=O)c(Cl)cccc1[N+](=O)[O-] N1(C(c2scc(C)n2)=O)CC(C)CC1C(=O)Nc1nc(C)cs1 CC(C)CC(O)CC(=O)N1CCN(C(C2CC23CCC3)=O)C(C(C)(C)C)C1 c1(N(c2ccccc2)C(=O)NCC2(C(=O)NC)CC2)ccc(Cl)cc1Cl Cc1nc2ccc(C(=O)NCCN(C(=O)Cn3cccn3)C)cc2s1 C(C)(CCC(=O)N(CCCCCNC(=O)CC(C)c1ccco1)C)SC C1(C(C)C)CN(C(=O)C2=C(Cl)CCC2)CCCN1C(=O)CC1COCC(C)(C)O1 C1(C(N(CC(C)CNC(C2CCCN2C)=O)C)=O)CC12CCOCC2 c1(C(=O)NC2(CF)CN(C(C(C)CN(C)C)=O)C2)ccc(CC(N)=O)cc1 c1(C(=O)NCC2CCN(C(CS(CCCC)(=O)=O)=O)C2)ccccc1C#CC1CC1 c1(C(=O)NCCN(C(CCC(C)SC)=O)C2CC2)cc2c(s1)CCOC2 C1(C(N2CC(F)(CNC(c3cc(C(F)(F)F)c[nH]3)=O)C2)=O)(OC)CCOC1 c1(C(=O)NC(C(C)NC(C2CCCN(CC)C2)=O)(C)C)ccc(F)c(C#N)c1 C1(CN(C(=O)CSc2nc[nH]n2)C)CCCN1C(=O)CCc1cncs1 C1(NC(C(CC)SC)=O)CCCC1(C)C(=O)NOCCCO C12(CNC(C(CCCC)O)=O)CCC(CN(C(C3(C)CCCN3C(C)=O)=O)C1)C2 c1(C(N2CC(NC(CCN(CC)CC)=O)C(C)C2)=O)ccc([N+](=O)[O-])s1 N1(C(c2ccc(N(C)C)nc2)=O)CC(NC(c2snc(O)c2Cl)=O)CC2(CC2)C1 c1(NC(=O)CC2CCCNC2)ccc2c(c1)CN(C(c1csc(Br)c1)=O)CC2 C(=O)(C(O)CC(F)(F)F)NCc1cccs1.C12(CCC1)C(=O)NCCS2 N1(C(c2nc(CCC)sc2)=O)CCC2(CC1)CC(NC(c1conc1C)=O)CO2 C#CC1(C(=O)NCCN2CCCC2=O)CCN(C(=O)CC2CC(C)=NO2)C1 c1(C(=O)C=Cc2ccccc2)cc(C(F)F)cc(C(F)F)c1 C1(CNC(C(c2cccc(C#N)c2)C)=O)CC2(CC2)CN1C(=O)C(C)C(C)C c1(C(=O)NC(CN(C(c2n[nH]c(C)c2F)=O)C)C)ccc2c(c1)NC(=O)C2 C1(CNC(C2(F)C(C)C2)=O)CCN(C(c2cnn(C)c2F)=O)C12CC2 Cc1nn2cc(C(=O)NCC3C(C)CCN3C(=O)C(c3ccc(Cl)s3)C)nc2s1 CC(C)C1CNC(=O)C1NC(C(C)c1cncs1)=O.n1(CN2CCOCC2)cc(C)nn1 C1(CNC(c2c(C#N)ccc(C)n2)=O)CC2(CCNCC2)C(=O)O1 Cc1c(C(=O)NC(C2(O)CN(C(c3ccc(C#N)s3)=O)C2)C)cnn1C1CC1 c1(CCC(=O)NC2CCN(Cc3ncccn3)CC2O)c[nH]c2cc(Cl)ccc12 C1(NC(c2cncc(N(C)C)n2)=O)CCC2CC1CN2C(c1ccc(Cl)cn1)=O CCC(C)(CO)C(=O)N1CC(CNC(c2nnn3c2CCC3)=O)C(C)(C)C1 N1(C(C2(NC(N)=O)CC2)=O)CCC(CCNC(=O)C=Cc2cnc[nH]2)C(F)(F)C1 N#Cc1ccccc1OCC(=O)NC1CC(O)(CNC(C2(C#N)CC2)=O)C1 c1(C(=O)NC2C3CN(C(CCOC4(C)CC4)=O)CC32)nc(Cl)ccc1Cl c1(CCC(N2C(CC(=O)NC3CCN(CCC)C3)CCC2)=O)cccnc1C c1(C(N(CC=CC(N2C(C(C)C)COCC2)=O)C)=O)cccc2[nH]ccc12 N1(C(CCC(C)c2ccccc2)=O)CC(=O)NCC1C(N1CC2CC1CN2C)=O C1(CNC(C=CC(CC)C)=O)CCN(C(=O)C(C)C2CCCC2)C1 N1(C(C(C)OCc2ccccn2)=O)CCCC(NC(=O)CNC(=O)C2CC2)C1 C(=O)(CC1COc2ccccc21)OCCN(CC(C)OC)CC N1(C(C(F)=CC)=O)CCC2(C1)CN(C(C1(OC)CS(=O)(=O)C1)=O)CCO2 C1(C)(C(=O)NCC2CCC(N(C(CSCCOC)=O)C)CC2)CC2CCC(C1)S2 c1(CC(=O)NCC2(F)CC(CNC(CCOC)=O)C2)ccccc1C C1(NC(C2(CC=C)CCC2)=O)CCC(NC(C2CCOCC2C)=O)CC1 c1(OCC)cnncc1C(=O)N(C)CCOCCNC(=O)CNC(C)=O C1(C)(C(=O)NC(CC)CNC(c2csc(-c3ccsc3)n2)=O)CCCOC1 c1(CC(=O)NC(CCCNC(COCCOC)=O)C)ccc(C(N)=O)cn1 N1(C(c2cc(C)[nH]n2)=O)CC(F)CC1CNC(C1CCN(S(C)(=O)=O)CC1)=O C(=O)(CC1COCc2ccccc21)N(C)CCNC(c1cc(Cl)cc(F)c1F)=O Cc1nc2ncccc2cc1C(=O)NCC1CC(NC(C23C=CC(CC2)C3)=O)C1 N1(C(C(C2CC=CCC2)NC(=O)CSC2CC2)=O)CCCC2(CC2)C1 CCC(CC(F)F)C(=O)N1CC(CNC(c2ccc(C(C)=O)cc2)=O)CCC1C N1(C(c2c(C(C)C)ncs2)=O)CCOCC(NC(C2(n3cnnn3)CC2)=O)C1 c1(C(=O)NCC2C(NC(CN(CC)CC)=O)CCC2)ccc2cccnc2c1O Cc1cc(C(=O)NC2COCCN(Cc3ccc(Cl)nc3Cl)C2)ccc1O CCC(CC)C(C(=O)N1CCCC1CCNC(=O)C=C(C)c1cccs1)OC Cc1ccc(C)c(C(=O)NCC(CNC(=O)C(C)Cn2ccnc2)S(C)(=O)=O)n1 C1(NC(CCc2cn(C)nc2)=O)CC12CCN(C(C1CC3CC3C1)=O)CC2 C(=O)(C1COc2ccc(F)cc21)N1CC2(C(CO)CN(C(C3C(C)(C)C3)=O)C2)C1 O=C(CC1OCc2ncccc21)NC1CC1NC(=O)C(c1cccc(Cl)c1)(F)F CN1CC(NC(=O)CCC(C)(C)NC(C2COCCN2C)=O)C(C)(C)C1 c1(OC)ccc(C(C)=CC(=O)N(C2CCN(C(=O)C3CC3)CC23CC3)C)cc1 c1(C(N(C(CNC(=O)CC2CC2(Cl)Cl)C2CC2)C)=O)cc(C2CC2)cc(F)c1 c1(C(=O)NC2CCN(C(CC)=O)C2)ccc(C(=O)NC2CCCCC2O)c(F)c1 C=CC(C)CC(=O)NCC(C1CCN(C(=O)C(C)OCCOC)CC1)O CS(=O)CCC(N)C(=O)Nc1ncc(I)c(C(F)(F)F)n1 c1(C(=O)NC2CCN(C(C3CC(NS(C)(=O)=O)C3)=O)C2)ccc(Br)c(O)c1 c1(C(=O)NC2CN(C(C(c3ccc(F)cc3)OC)=O)CC2C)ccnc(F)c1N c1(C(=O)NC(C)CNC(=O)C(C)(C)Oc2ccccc2)cccc2nc(O)oc12 C(=O)(CCC(C)(C)C)N1CCC(CN(C(=O)Cc2cnns2)C)C1 c1(CS)cc2cc(Br)ccc2o1.c12ccc(Cl)cc1CC2.C1CCS1.CO C1(C(=O)NCCC2ON=C(C)C2)CCCC(NC(c2ccc(CO)cn2)=O)CC1 CCC(C)C(O)C(C)C(=O)NC(Cn1cccn1)C(=O)NC1(CCCCO)CC1 c1(C(N2CCCC(CCNC(C3ON=C(C)C3)=O)C2)=O)cncc2c1CCCC2 c1(C2C(C(=O)NCC(CC)(C)NC(=O)Cc3csnn3)C2)ccccc1Br c1(C(=O)NCC2CCC(F)(CNC(=O)C(O)C3CC3)C2)cnc2c(c1)CCOC2 N1(C(CSCCC#N)=O)CCC2(CC1)CCN(C(=O)CCc1cc[nH]n1)CC2 c1(CC)ccc(C(=O)NCCc2n[nH]cc2C(=O)NCC2COCC2O)o1 C(=O)(C(O)CC[S+](C)C)NCC1N(C(c2c(OCC)nccc2)=O)CC2(CC2)C1 c1(C(=O)NCCN(C(c2n(C)cnc2)=O)C2CC2)c[nH]c2cccc(Br)c12 Nc1cc(F)c(CC(N2CC3CCC(C2)N3C(C2CCCC(O)C2)=O)=O)cc1F N1(C(C(=O)NCCCCCC)=O)CC(C(C)(C)C)Oc2ccccc21 C1(CC(N2CCC(NC(=O)Cc3n[nH]cc3Br)C2)=O)CC2(CCC2)CO1 c1(C(N2C(C(C)NC(CC(COC)C)=O)CCC2)=O)ccc(OC(F)F)c(F)c1 C(CN(C)C(C1CN(C)CC1C(F)(F)F)=O)(CO)(CO)NC(CC=C)=O c1(C(N(CCCN(C(CN(C(COC)=O)C)=O)C)C)=O)oc(C)cc1C C1(N(C(c2ccn(COC)n2)=O)C)CCCCC1N(C(=O)C(C)=C1CCC1)C N1(C(c2c(CC)cccn2)=O)CC(CN(C(=O)CN2CCCC2C)C)C2(CC2)C1 C(=O)(C1CCCc2c[nH]nc21)N1CCC(N(C(C(CC)CC(F)(F)F)=O)CC)C1 Cc1ccc(-n2nc(Cc3ccccc3)nc2CCCC(F)F)cc1 c1(NC(c2ccc(CO)o2)=O)cncc(-c2ccccc2)c1 CS(=O)(=O)c1ccc(CC(=O)NCC2CC3CNC(C2)C3)cc1 C1(OC)CC(NC(c2cnn(C(F)F)c2)=O)CN(C(c2cccc[n+]2[O-])=O)C1 C1(C(=O)NCC2CC(CNC(C(C)CC3CC3)=O)C2)CC1C1(C)COC1 c1(NC(c2c(-c3ccc(OC)c(F)c3)nccc2)=O)ccc(C#N)c(O)c1 CC(CCC(=O)Nc1ccccc1Cl)NC(=O)CC=C(Cl)Cl n1(CC(=O)NCCN(C(=O)CC#N)C(C)C)cc(CN2CCC2)nn1 c1(C(N2CC(NC(CSC)=O)C3C2C3)=O)c(C(F)(F)F)nn2ccccc12 C(=O)(C1=CCC(C)CC1)NC1CCN(C(CCC(=O)OCC)=O)C1 C(=O)(C(C(C)CC)NC(=O)C1=C(C)CC1)NC(CCC=C)CO c1(C(=O)NCCC2C(C)CCC2)cc(OC2CCCC2)cc(Br)c1 CS(=O)(=O)c1cncc(C(=O)NCCC2CC(NC(=O)CSCC(N)=O)C2)n1 c1(OCCC(=O)NC2C(NC(CCNC(C)=O)=O)COC2)ccccc1[N+](=O)[O-] c1(C(=O)NC2C(C)N(C(C34CCCC3C4(F)F)=O)CC2)cc2nccn2c(O)n1 C(=O)(C1OC(=O)c2ccccc21)NC1CC(OC)CN(C(=O)CCNC(N)=O)C1 CC1c2ccccc2N(C(=O)CN2CCCC3(CCCNC3)C2)C1C C1(C(=O)NCCC2(C(=O)NCCC=CCCC)CC2)CC2CC2C1 N1(C(c2cccc(OC)c2)=O)CCN(Cc2cc(F)ccc2OC)CC1C#N C1(C(=O)NC2CN(C(COC)=O)C(C)(C)C2)CC(c2ccccc2)=NO1 CC1CC(O)CCN(C(C2CCCCN2C(c2cccc(=O)n2C)=O)=O)C1 C(C(C)(C)C(=O)NC(c1ccccc1)C(=O)NCCCC(C)(F)F)OCC C1(F)(CNC(C(C)CCN(C)C)=O)CCN(C(=O)C(O)Cc2cnc[nH]2)CC1 c1(C(=O)Nc2ccc(OC)nc2)nc(C)c(COCC)s1 C1(NC(CCCCN(C(C(C)(C(C)C)OC)=O)C)=O)CCCCC12CCC2 C1(CNC(C2C(C(C)(F)F)C2)=O)(NC(c2coc(Br)n2)=O)CCOC1 c1(C(=O)NCC(CC)n2cccn2)c[nH]c2ccc([N+](=O)[O-])cc12 S(=O)(=O)(C1CCN(C(=O)NC(C)(C)C)C1)N1CCC(N2CCN(C)CC2)C1 CC1(C)CC(CNC(=O)CCC2CC(F)(F)C2)N(C(C2CC2F)=O)C1 CN1CCc2cc(C(=O)NC3CCCCC3NC(C3CC(CCF)C3)=O)ccc21 N1(C(COCCCC(C)C)=O)CC2(CCN2C(=O)CCC2CCCO2)C1 C1(CCOC)CCCCN(C(c2nonc2N)=O)C1 N1(C(C(C(C)C)C2CCC2)=O)CC(C2(NC(=O)CCc3nncs3)CC2)C1 N1(C(CCC(=C)Cl)=O)CCCC2(NC(c3ccnn3C(CC)CC)=O)CC2C1 c1(CC(=O)N(CC(C)NC(=O)CCc2cncs2)C)ccc(C#N)c(F)c1 N1(CC#C)CCC(C(N2CCC(C)C2CNC(=O)C(F)=C2CCCC2)=O)CC1 N1(C(CONC(=O)OC(C)(C)C)=O)CCC(NC(C2CCC(=O)N2)=O)C(C)(C)C1 c1(NC(=O)Nc2ncc(C#C)cn2)ccc2nccn2c1 C1(CC=C)(NC(=O)CC2CC=CCC2)CCCN(C(C2(C(=O)NC)CCC2)=O)C1 C(=O)(C(C)C(=O)NCc1occc1C(=O)N(C1CCCC1)C(C)C)OC N1(C(c2n(C=C)ncc2)=O)CCN(C(=O)Cc2cncs2)CC1CCO Cc1cnc(NCC2CCCS(=O)(=O)C2)c(S(=O)(=O)NC2CCC=CCC2)c1 C1(C(=O)NCc2c(C(N(CC(C)O)CC(C)O)=O)scc2)CCCN(C)C1 C1(CNC(C(C(C)C)SCC)=O)CN(C(=O)Cn2nc(C)oc2=O)CC(C)(C)O1 c1(C(=O)NCC(N(C(C=C(CC)C)=O)C)C2CC2)ccc(C)c([N+](=O)[O-])c1 c1(CC(=O)N(C2CCCN(C(=O)CC3(O)CCC3)C2)C)cc2ccccc2s1 Cc1ccnc2ccc(C(N3CCN(C(c4cccnc4S)=O)C4CC34)=O)cc12 C1(CNC(C(C2CC2)SC)=O)CCC(C(=O)NC2CCOC2C)CC1 c1(OCC)ccc(C(=O)NC2CC23CN(C(c2c(Br)cncc2Br)=O)C3)cc1OC c1(CN2C(C(=O)Nc3cc(C)c(O)cn3)CC2)cc(F)cc(C)c1O C(=O)(C=C1SCC(=O)N1C)N1CCOCC(C(NOC(C=C)C)=O)C1 C1(C)(CC)CC(NC(c2cn(C)nc2C)=O)CN1C(=O)CCC(C)(C)OC C1(CNC(c2cc(C(C)C)on2)=O)C(C)CCCN1C(=O)CNC(=O)NC1CC1 N1(C(C2(CC=C)CCOCC2)=O)CCC(NC(=O)Cc2ccsc2)C(C(N)=O)C1 C1(CCNC(C(n2ncc(C)c2)C)=O)CSCCN1C(=O)CSc1n[nH]c(C)n1 c1(OCC(=O)NCC2CCCN2C(=O)CC2CCCOC2)cc(F)cc(F)c1 C(=O)(C(C(C)C)S(=O)(=O)C1CCCCC1)NCCNC(c1c(CC)nccc1)=O N1(C(CSCC)=O)CCC(CNC(=O)COc2ccc(C)cn2)C(C)C1 N1(C(C(CCC)(C)CC)=O)CCCC2(CC(NC(C3CC4CCC3CC4)=O)C2)C1 N1(C(CCC2CCC(C)O2)=O)CCC(C2CN(C(=O)C3=CCCC3)C2)CC1 C(=O)(C(C)(C)C(C)O)NC1CCC(C(=O)NC(C#C)C(C)(C)C)C1 C1(O)(CCC)CCN(C(C2C3CN(C(=O)C(C)(C)OC(C)=O)CC23)=O)CC1 C1(C)(CC)CC(NC(C2(C)CC2)=O)CN1C(=O)CCc1cc(Br)cs1 CC1(NC(=O)CCNC(N)=O)CCCN(C(c2ccnc(C3CCCC3)n2)=O)C1 c1(C(N2CC(C)C(NC(=O)CC3CCCO3)C2)=O)nnc(Cl)cc1N C(=O)(CCCCOC(C)(C)C)NC(C)CCNC(=O)CC1C=CCC1 Cc1cc(C(N2CC(NC(=O)CN(C)C)C3(CC3)C2)=O)nnc1C Cc1c(N2CC(CN(C)C)C(C)C2)ncnc1N1CC(=O)NC(C(C)C)C1 Cc1cc2nc(NCCNC(c3cnn(CCO)c3C)=O)cc(=O)n2o1 C(=O)(C(O)CC(N)=O)NC(CCC(=O)NC(C(=O)OC(C)C)C)C N1(C(C2CCC(C)(C)C2)=O)CC(CNC(=O)C(C)(C)C#N)CC12CCC2 Cc1cc(C(N2CCC2CNC(c2cnn(C)c2C(F)F)=O)=O)cc(N)c1O N1(C(CNC(N)=O)=O)CCC(F)(F)C(CNC(=O)C=Cc2ccccc2)C1 C12(CNC(C3N(C)CCC3)=O)CCC1CN(C(c1ncoc1C1CCC1)=O)C2 N1(C(C2(COC)COC2)=O)CC2(C1)CN(C(=O)Cc1ccc(C)cc1)C2 C(=O)(C(CCS(C)=O)N(C)C)N1CCC(C)(NC(C=C(COC)C)=O)C1 C(C(C)(C)CC(=O)NC1(C(=O)NCC2CCCC23CC3)CC1(C)C)OC CS(=O)c1ccc(C(=O)NCC2CC2NC(=O)CNC(C2CCC2)=O)cc1 C1(CNC(C2C(C)C2C)=O)CC(F)CN1C(c1cnn(CCC2CCCC2)c1)=O c1(C(C(=O)NC(CC)CNC(=O)C#CC2CCC2)O)cc(F)c(F)cc1F N1(C(C2(N(C)C)CC2)=O)CCC(NC(=O)Cc2nn[nH]n2)CC1C(F)(F)F C1(CNC(C2CN(C(C)C)C(=O)C2)=O)CC2(C1)CN(C(=O)C(O)C(F)(F)F)C2 C1(CC(=O)NCCC=CC=C)CN(C(=O)CCCCC)CC1C c1(CCC)n[nH]cc1C(N1CC(N(C(=O)C(C)CC2CCC2)C)C1)=O N12CC(CC1C)C1CCC(O1)COC(OCC)CC2=O.C1(CO)(OC)CC1.OC.OC C(=O)(C(CC)CCOC)NCCC(=C)CNC(c1c(OC(F)F)cccc1Cl)=O CCC(C)(CC)C(=O)C(C)(C)NC=O.C12CN(C1)C(=O)NC(=O)C2 N1(C(C2(CC=C)CC2)=O)CCN(C(C2CCCN2C)=O)C(CC(=O)OCC)C1 Cc1cc(C(N2CC(CNC(=O)Cc3cn[nH]c3)OC(C)C2)=O)c2nccn2c1 Cc1nc2cc(Cl)ccc2n1CCNC(=O)C(=O)NC1CCSC2(CCC2)C1 CCC(CC)(CC(=O)OC)C(=O)N1CC(NC(=O)CCS(C)=O)C2(CC2)C1 c1(C(=O)NC2CCN(C(c3c(C)cnnc3)=O)CC2)c(Cl)cccc1Br Cc1cccc2c1NCCC2C(=O)N1CCCC(CCNS(C)(=O)=O)C1 CC1CCN(C(=O)CCCn2ccnn2)CC1CC(=O)N(C1CCCC1C)C c1(C(N2CCCC2CCNC(=O)C(F)(F)C2CC2)=O)cnn(-c2ccccc2)n1 Cc1cncnc1C(=O)NCC1(O)CCN(C(C2(n3ccnn3)CC2)=O)C1 C#CC1CCN(C(=NCCSC2(C(F)(F)F)CC2)NC(c2cccs2)C)CC1 c1(C(=O)Nc2cccc(CCC)n2)[nH]c(C)c(C(=O)NC2CSC2)c1C CC(N=c1[nH]c2ccc(Br)cc2s1)C(C1CCCCC1)NC(=O)Cc1cccs1 C(=O)(C1=CC2(CCOC2)C1)NC1(CCCNCC=CCOC)CC1 c1(C(N2C(C3(NC(C=CC)=O)CC3)CCC2)=O)cc2c(C)ccc(F)c2o1 c1(CN(C(=O)CC2CCCO2)C)cnn2c1CN(C(C1(F)CCCCC1)=O)CC2 c1(OC)ncc(C(=O)N(C2CCCN(C(=O)C(=O)NC3CC3)C2)C)nc1C c1(C(=O)NC2CCC(NC(=O)COC3CCCCC3)C2)noc2ncccc12 CCN=c1[nH]c2ccccc2s1.C1(C(=O)NCCOCC2CC2)CC2CC2C1 Cc1c(N2CCC(NC(=O)C(c3cncn3C)O)C(O)C2)ncnc1Cl C1(C(=O)NC(C2(O)CN(C(c3cc(Cl)cn3C)=O)C2)C)CCc2nnc(O)cc2C1 N1(C(C(c2ccccc2)C)=O)CCCCC1C1CCCN(C(C2(CF)CC2)=O)C1 N1(C(CC)C)CC2CCC(NC(=O)C=Cc3ccc(OC)cc3)CC2C1 CC1=CCC(CNc2nccc(N3CCC(N4CCC(CO)CC4)C3)n2)CC1 Cc1nn(CC(=O)NC2CCN(CCc3cn(CCCF)nn3)CC2)c(C)c1C CC(COCC(F)(F)F)N=c1[nH]c2c(c(=NC(C)CC#N)[nH]1)COCC2 c1(C(=O)OC(CC)C(=O)c2ccccc2)cc2cnn(C)c2nc1Cl C1(NC(C2(CNC(C(CC)OC)=O)CC(OCC)C2)=O)CC2CCC1O2 CC(C)(C)C(CNC(=O)C1=NOCC1)C(=O)N1CCC(n2cccn2)C1 C(CN=c1[nH]cnc2c(F)c(F)ccc12)N(C(C1ON=C(C(C)C)C1)=O)C1CC1 C1(NC(C=CC=CCC)=O)CC2CC(NC(=O)Cn3cc(Br)cn3)C2C1 c1(C(=O)NC)cc(=NC(=O)C2=NOC(c3ccc(C(F)(F)F)cc3)C2)[nH][nH]1 N1(C(C(n2ncc(C)c2)C)=O)CCC2CCN(C(=O)CNC=O)CC12 c1(C(=O)NCC2C(C)CCN(C(Cc3cc(C)ns3)=O)C2)cncc2ccsc12 C1(C(=O)NCC(CC)CO)CCC(NC(c2ccc(CSC)o2)=O)CC1 C(=O)(C1CCS(=O)(=O)c2ccccc21)N(C(c1ccccc1)C)CCN C1(C(N2CC(CCCCNC(C(C)NC(N)=O)=O)C2)=O)CC(C)(C)OC1(C)C c1(CC)cccc(-n2cc(-c3cc(N(CCCO)CC)c(OC)s3)nn2)c1 N12CCCCC(C1)SCc1ccc(o1)C2=O.C(=O)(CC)NCCSCC=C C12(CNC(COCC(=O)NC)=O)CC1CN(C(=O)C(F)CC1CCCC1)C2 c1(C(=O)OC)ccc(C(=O)OCC2C3CN(C(C)C)CC23)cc1F N1(CCC(=O)N(C2CCN(C(CC(CCC)O)=O)C2)C)CCCc2ccccc21 C1(NC(c2c(C)cc(CNC(=O)CC(C)C3CCCC3)o2)=O)CC(C)CC(C)C1 c1(C(=O)NC2CCC(NC(C3(COCC)CC3(F)F)=O)C2)cc(C)ccc1C N1(C(C2N(C(c3c(C#N)cc(F)cc3)=O)CC(F)C2)=O)Cc2ccc(O)cc2C1 CCC(C#N)C(=O)N1CCCC1CCNC(=O)CC1(C)CCCC1 c1(NC2C(CC(C)C)COCC2)cc(F)c2oc(O)nc2c1 C1(CSCc2cccc(C(=O)OC)c2)CC2(CCOCC2)CO1.CCS c1(OC)cc(Br)nc(NC(C2CCNC2C(C)C)=O)n1 C1(NC(=O)COc2ccccc2)C2CC3C(C2)C13C(=O)NCCCC(F)F CN1CCC(O)(C2(C(N3CCCC3CNC(=O)C3=CC4C=CC(C3)C4)=O)CC2)CC1 Cc1nn(C)cc1C(N1CCC(O)(C(=O)Nc2ccc(-n3cccc3)cc2)C1)=O c1(C(=O)NC2C(NC(CSCC=C)=O)CCCC2)cnc(C)nc1OC c1(CNC(C2N(C(C(CN(C)C)(C)C)=O)CCC2)=O)cc(F)cc([N+](=O)[O-])c1 CC1CN(C(C2CC(=C3CC3)C2)=O)CC(CCNC(=O)Cn2ncccc2=O)O1 Cc1cccc(NNC(=O)c2cccc3nsnc23)c1F C=C(Br)CC(C)(C)C(=O)NCC1CCCCN1C(=O)C(C)=C(C)CC c1(C(=O)NC2CC(CNC(C(CCC#C)O)=O)C2)ccc2c(n1)OCCO2 c1(C(=O)NCC(C)(C)CO)c(F)cncc1C1=CCC(O)CC1 Cc1cnc(N(CCCNC(c2cc(N3CCCC3)ccn2)=O)N(C)C)nc1C c1(C(N(CCCOCCNC(CCc2cnc(C)o2)=O)C)=O)cc(CO)n(C)n1 N1(C(C2C(=C)C2)=O)CCC(CNC(c2cnn(C)n2)=O)CC1C Cc1ccnnc1C(=O)NC(C)C(C(C)C)NC(c1cn(C2CCCC2)nn1)=O C1(C(=O)NCC(CN(C(=O)Cc2ccc(Cl)cc2F)C)O)CC(F)(F)C1(C)C C1(CC(=O)NC(CNC(C=CCC)=O)(C)CO)CSc2ccccc2NC1=O c1(NC(CC2(N(C(CCC(C)N(C)C)=O)C)CC2)=O)ccn2nccc2c1 CC1CN(C(=O)COc2ccc(C#N)cc2)CCCN1C(c1ccoc1)=O N#CCCCCCC(=O)NCC1CCN(C(C2CCOC2)=O)C1 C1(C(N(CCCSC)C)=O)CCCCN(C(=O)C(C)S(C)(=O)=O)C1 N1(C(COCC(=O)N(CCOC)CC)=O)CCC(C)C(NC(=O)C(N)=O)C1 C1(NC(CCOCCOC)=O)CCC2(CCN(C(C3CCC3C(=O)OC)=O)C2)C1 c1(NC(N(c2cccc(C(=O)OCC)c2)CC)=O)ncn2c1COCC2 C1(C(=O)NCC(CSC)(C)CC)COCCN(C(C2(C(N)=O)CCC2)=O)C1 C(CCC(C)CC(=O)NC1CC(NC(=O)CC2CCC3(CC2)COC3)C1)=C(C)C c1(C(=O)OCC)[nH]c(C)cc1NC(=O)NCC(CC1CC1)OC S(=O)(=O)(c1ccc(C#N)c(N2CC=CCC2)c1)NC1(C=C)CCC1 C1(CNC(CC2C(C)CCCC2)=O)CC2(CC2)CN1C(=O)CCc1cnc[nH]1 C1(CC)CC(CC(=O)N(C)CC2(CNC(c3ccccc3F)=O)CC2)CCO1 C1(N(C(c2ccc(CN(C)C)o2)=O)C)CCCN(C(c2ncncc2Cl)=O)C1 c1(C(=O)NCCCCC(CO)NC(=O)Cc2nc[nH]n2)cc2ccc(O)cc2[nH]1 C1(NC(C2C(CNC(COCCOCC)=O)CC2)=O)CCCC1(F)F C1(NC(C2CC(N(C)C)C2)=O)CN(C(=O)CC2C(CO)C2(F)F)CC12CC2 c1(-c2cn(CC(CN(CC(C)(C)C)C(=O)CO)(F)F)nn2)cccc(Cl)c1 C1(NC(C(SCc2cccc(C)c2)SC)=O)CC2(C1)CC(NCC(=O)O)C2 N1(C(CC2CN(C)C2)=O)CCOCC2(COCCN2C(c2ccc(Cl)nc2)=O)C1 c1(CC(N2CCN(C(CC(CC)C)=O)CC2CC)=O)ccc2c(c1)OC(F)(F)O2 C1(C(N2CC(O)(C(C)NC(=O)C#CC(C)(C)O)C2)=O)CCc2ncnn2C1 C1(CN(C)CCc2ncc(Br)cn2)CCN(C(C2(C)CC(C)(C)C2)=O)CC1 c1(OCC(N2CCCN(C(C(CC#C)O)=O)C(C)C2)=O)ccc([N+](=O)[O-])c(C)c1 c1(C(=O)NC)occc1SCc1cocn1.C1COC(=O)O1 C1(C(N2C(CN(c3cc(CC)ncn3)C)CCC2)=O)Cc2ccc(C)cc2S1 N1(C(C=CC)=O)CCCC2(CCCN2C(=O)C(C)COc2ccc(Cl)cc2)C1 C(=O)(C(F)C1CCCC1)NCCN(C(=O)C(C)C1CCCC1)CC C1(C(N(CCCNC(C2CC(C)=C(C)CC2)=O)C)=O)COc2ccc(F)cc2C1 N12NC=NC1=NCC1(CC1)C2.c1(N(C)C)ccc(C(N)=O)cc1 C1(NC(CCCNC(COC)=O)=O)CS(=O)(=O)CC1NC(=O)CCC1CCCC1 CC(C)C(C(C)NC(=O)CS(N)(=O)=O)NC(c1nocc1Br)=O N1(C(CCc2n(C)cnc2)=O)CC(NC(c2cn(C3COC3)nn2)=O)C(C)(C)C1 CCCCCCC(=O)N(C1CCC(NC(=O)COC(C)CC)CC1)C C1(NC(C(C)OCC)=O)CC(F)(CNC(C2(C(C)C)CC2)=O)C1 N1(CC(=O)Nc2ccc(CCC)cc2)CC2CCC(F)(C2)C1 CC1=C(C(=O)NC2CN(C(=O)COc3cc(F)cc(F)c3)C3CC23)CCCC1 C1(CNC(CCn2c(C)csc2=O)=O)CCCN(C(=O)C2=CCCO2)CC1 CCC(C#N)C(=O)N(CCCN(C(=O)CCc1ccc(Cl)s1)C)C N1(C(c2nc(OCC)sn2)=O)CC(CCNC(C2(OC)CCC2)=O)C(C)C1 N1(Cc2cc(OC)c(O)cc2)CCCC2(CCN(C(C3CCC(F)(F)C3)=O)C2)C1 N1(C(C(F)=C(C)C)=O)CCC2(CCC(NC(=O)C(C)NC=O)CC2)CC1 C(=O)(C(C)(C)C(C)NC(=O)C(C)SC)N1CC(C#N)(COC)C1 N1(C(c2c(C)onc2CO)=O)CCCCC(CNC(C2CCNC2=O)=O)C1 c1(C(N2C(CCNC(C(CC)CC)=O)CCCC2)=O)cc(F)cc(N)c1N C1(NC(c2c(C)nc(C(C)OC)s2)=O)CN(C(=O)C=CSC)C(C)(C)C1 c1(C(N2CC(NC(c3nc(COCC)sc3Br)=O)C2)C)cc2ccoc2cc1F C1(CCNC(=O)CC2CC23CC3)CN(C(=O)C(F)=CC2CC2)CCO1 Cc1ccc(SCC(N2CCC(NC(c3[nH]ccc3C)=O)C2)=O)cc1 C1(NC(C(CC=C)CC)=O)C2COCC1CN(C(c1[nH]cnc1CC)=O)C2 C12(CC(=O)NCC(C)CNC(=O)C(F)=CCCF)CCCN1CCC2 c1(C(c2nnnn2CC2CCOCC2)NCCC(C)CO)ncccc1O C#CCC(C(=O)N1CCN(C(c2cccc(O)c2)=O)CC1)C1CC1 c1(C(=O)NC(CNC(c2c(CC)onc2)=O)CC)cc(Cl)cc(C)c1C CC(CCN(C)C)C(=O)NCC12CC(CNC(C3C4COCC34)=O)(CO1)C2 N(C(=NCCC=C(C)C)NCC1COCCO1)C(c1c(OC)cccc1)C c1(OC)ccc(CC(=O)NC2CCN(C(c3cccnc3N)=O)CC2F)c(F)c1 C(=O)(C(CNC(=O)Cc1ccccc1)CC1CCCC1)N(CC)CC1(F)CCC1 Cc1ncc(C(=O)NCC2CCC(C(N3CC(O)CCC3C)=O)CC2)cc1C#N CC(N=c1[nH]c(=NC(C)CS(C)(=O)=O)[nH]c2c1COC2)C1CCCCC1 Cc1[nH]nc2c1CC(C(=O)NCCCC(C)(C)NC(=O)C(O)C(F)(F)F)CC2 Cn1ccc(C(=O)NCC2CCC(NC(=O)C=C3CCSCC3)CC2)cc1=O N1(C(CSCC#C)=O)CCN(CC(=O)NCC2CC(CF)C2)CC1 c1(OC)cccc(Cn2nnnc2C(CC(C)C)NC2(C)CCOC2=O)c1 N1(c2cc(NCC=C=C)nc(SC)n2)CCC2CC(C(=O)OC)C2C1.CC c1(C(=O)NC2CCCC(NC(CC3(C(=O)OC)CC3)=O)C2)cncc2nc[nH]c12 C(C)(C)(C(N)=O)NC(C=CC(C)NC(=O)CC1CC1(C)C)=O c1(C(N2CCN(C(CO)C3CC3)CC2)C(=O)NCC(C)C)ccnc(Cl)c1Br [N-]=[N+]=NCCCC(=O)NC1CCCCCC1NC(=O)C(c1ccc(F)c(F)c1)=O C1(NC(CCC=CC)=O)CCC2(CCN(C(c3ccnc(SCC)c3)=O)CC2)C1 C(=O)(C1=NOC(C)C1C)N(CCCC(=O)N(CC(COC)O)C)C c1(C(=O)NC2(CCO)CN(C(=O)CC3CCOC3)C2)cccc2sncc12 Cc1scc(C(=O)NC2C3CC2N(C(c2cc(C(N)=O)c[nH]2)=O)C3)c1C Cc1ccc(Br)c(CNC(c2occc2-c2ccccc2)=O)n1 C(=O)(C(C)COC(C)C)NC1CC(O)(C(C)NC(CCOCCOC)=O)C1.OCC c1(C(c2nc[nH]n2)NC(CC=C(C)C)=O)ccc([N+](=O)[O-])cc1 C(=O)(C(C)CC(F)F)NC1(CC=C)CCN(C(=O)CC2CCC(=O)N2)C1 N1(C(CCNC(=O)NC)=O)CC(F)(F)CC1CCNC(=O)CC1SC(=N)NC1=O c1(C(=O)NC2CCN(C(CN(C(C)C)C)=O)CC2)cnc2cccnc2c1 C1(CNC(C(CC)NC(C)=O)=O)CC2(CC2)CN1C(c1cc(I)ccc1OC)=O N1(C(C(N2CCNC2=O)C)=O)CC2(CCN(C(c3ccc(Cl)[nH]3)=O)CC2)C1 N1(C(c2c(C)onc2C(F)(F)F)=O)C2CCC1CN(C(=O)CN1CCC1C)CC2 N1(C(C(=O)NCCC2CC2)C2CCCC2)CCCCC(C2CCOCC2)C1 C1(C(C(=O)CC2CC2C)=O)(OC)CCCCC1.C(CCN)NC(=O)OCC c1(C(C)C(=O)NCCC2CN(C(=O)C3=COCC3)C2)c[nH]c2ccccc12 N1(C(C(C2CCCC2)NC(CNC(C)=O)=O)=O)CC2(CCNC(=O)O2)C1 S(=O)(=O)(c1cncc(Br)c1)N1CC2N(C(c3ccc(-n4ccnn4)cc3)=O)C2C1 C12CCN(C3(CC3)C1)C(=O)C2.c1(C(=O)OC)cccc(C2SCCN2C(C)=O)c1 C1(CC(=O)N(C2CCN(C(CCOCCC)=O)C2)C)C(=O)NN=C1C C=CCC(F)(F)C(=O)N1CC(NC(=O)Cc2nn(C)cc2Br)CC(C)C1 N1(C(c2c(C)noc2C)=O)CC2CN(C(C3CC(C)OC(C)C3)=O)CC2C1 Cc1nc2ccc(C(C)(C)C)cc2n1C.C1(C(=O)N)CCN(C(=O)C2CC2)C1 C1(NC(c2ccc(CC)s2)=O)CC2(C1)CC(C(N1CC3CC1CS3)=O)C2 N1(C(c2c(C)cc(C(N)=O)cc2)=O)CCC(CNC(C2CCCO2)=O)C(F)(F)C1 c1(C(N(CC(C)NC(C2CC(n3cnnc3)C2)=O)C)=O)cc(C#N)on1 CCCCC(CNC(=O)C(C1CCC(=O)N1)C)NC(C1C=CC1C(=O)OC)=O C1(CNC(C2C(CC)OCC2)=O)CC2CN(C(C3C=CC=CC=C3)=O)CC12 c1(C(=O)NC(CC)CNC(c2cnc[nH]2)=O)ccnc(C(C)(F)F)c1 c1(C(N(CCCNC(C2(C)CCCC2C)=O)CC)=O)cnn2c1CCCC2 Clc1nc2c[nH]c(=NCc3cccc4c3CCC4)cc2[nH]1 O(NC(=O)C(C)C(C)NC(=O)C(C)(C)CCF)CCCOCC CC1CCN(C(c2ncoc2-c2ccco2)=O)C(C)C1NC(=O)C=Cc1ncc[nH]1 CCC(O)(C(=O)N(C(CNC(c1ccc(C)nc1)=O)C1CC1)C)c1ccccc1 O=C(CC(O)CNC(c1cnc(C2CC2)o1)=O)NCC(c1ccccc1)O CCCCCCC(=O)NCC1COCCN1C(=O)C=CSC C1(C(N2CCC(C(N(CCN(C)C)CC)=O)(CC)C2)=O)C2CCC(C2)C1C C1(NC(C2CC(=C)C2)=O)CC(F)(CNC(C2CC(SC)C2)=O)C1 C1(CC(=O)Nc2cnc(C)s2)CCCCN1C(c1ccccc1-c1nn[nH]n1)=O C(=O)(C(C)(F)C(=O)NC(CNC(=O)CS(=O)(=O)Cc1cccs1)C(C)C)OC C12CCCCC1NC2=O.C(=O)(CC1(CO)CC1)NC(C1(CC2CC2)CC1)C N1(C(c2c(CNC(C3(CC)CC3)=O)[nH]cc2)=O)Cc2ccnn2CC1C C1(N(C)C)CCCN(C(C2(NC(=O)CNc3ccccc3)CCN(C)C2)=O)CC1 c1(C(N2CCC(C)C(NC(=O)Cc3ccno3)C2)=O)c(N)cc(F)cc1F C(C)(C)(CCCNC(c1cc(CO)on1)=O)NC(C(c1ccc(F)cc1)SC)=O N(C1CCc2sc(Cl)cc21)C(c1cc(C)cc(C)c1)c1nnnn1C1(C)CC1 C1(C(=O)NC(C(O)CO)C2CC2)CN(C(C2(O)CCCCC2)=O)CC12CCC2 C=CCCN=C(NCc1cccc(C(C)C)n1)NC(c1ccn(C)n1)C S(=O)(=O)(c1ccc(C(=O)NC2CC(CNC(=O)C3=COCCC3)C2)cn1)N(C)C C1(N(C)C(c2nccn2C)=O)CN(C(c2cc(N)cc(O)c2)=O)CC1(C)C S(=O)(=O)(c1ccc2c(c1)C(=O)C(=O)N2)C(C)C.n12c(C)cc(c1C)C=CC(C)CC2 Cc1c(C(=O)NC2CC(CNC(=O)C=CCO)CC2O)sc2cccc(F)c12 C1(NC(CCCCCCSC)=O)CC2CCCC(C1)N2C(c1ncncc1F)=O c1(C(N(C(C)CNC(c2ccc(CCO)cc2)=O)CC)=O)cnc(=N)[nH]c1 CCCC(C)CCN=c1cc[nH]cc1S(=O)Cc1ccc(C(C)(C)C)cc1 n1(CCC(=O)NCC2(C(N)=O)CN(C(=O)Cc3cc[nH]c3)C2)cc[nH]c(=O)c1=O C1(CNC(C2CN(c3cccc(C)c3)C(=O)C2)=O)(CO)CCCC12CCC2 c1(NC(C(CC2CCC2)NC(C(CCCOC)C)=O)=O)cccc([N+](=O)[O-])c1 n1(CCN(C(C)C)CC)ccc(=NC(=O)Nc2ccc(Br)s2)[nH]1 CC(C)C(C(=O)NCCNC(C1CSCCS1)=O)S(=O)(=O)C1CCCCC1 O=C(CC1OCCc2ccsc21)NCC1(CNC(c2ncc(C(F)F)s2)=O)CC1 C(c1ccnn1C)=CC(=O)N(C)CC1(NC(c2c(OC)scc2)=O)CC1 N1(C(c2c(CC=C)cccc2)=O)CC2CCCC(C1)N2C(C1CC(C)(C)CO1)=O CCCCCCC(C)C(=O)NC1(C)CCN(C(c2cnc(OC)nc2C)=O)CC1 C1(C(=O)NC2CC(CNC(CCc3n(C)ncc3)=O)C2)CCc2nnnn2C1 C(CN=c1[nH]cnc2c1COC2)N(C(C1C(CC)OCC1)=O)CC S(=O)(=O)(CC(=O)NCC1(F)CC(CNC(=O)C(c2cccc(F)c2)C)C1)NC C1(CNC(CC2CC(C)C2)=O)CCC(N(C)C(c2sccc2C(C)(C)C)=O)CC1 C1(=CC(=O)N(CCC(C)(C)NC(Cc2cc(C)on2)=O)C)CCN(C)CC1 N1(C(CCNC(c2cn(CC=C)nn2)=O)=O)CCCC(CO)C1 c1(C(=O)NCC2CC(NC(C(C(CC)C)C)=O)C2)cc([N+](=O)[O-])cnc1C c1(C(=O)NCC(C(=O)NC(CN(CCC)CC)C)N(C)C)cc[nH]c(=NC)c1 c1(C(N2C(CNC(CC(C)C(F)F)=O)CC(F)(F)C2)=O)cc2ccc(F)cc2s1 Cc1cnc(Cl)[nH]c1=NC1CC2CN(C(=O)Cc3ccc(F)cc3Cl)CC2C1 CN(C1CCN(C(=O)OC(C)(C)C)CC1)N1CC(N(C)C2CC2)C2(CCOCC2)C1 N1(C(c2cc(C)cc(C(F)F)c2)=O)CCC(NC(=O)C=CC2CCC2)C(C)(C)C1 Cc1cc(C)c(C(=O)N(C2CCN(C(=O)CC(C)CF)CC2)CCO)cc1C C(CN=C(NCC1CC=CCC1)NC1CC1NC(=O)COC(F)F)NS(C)(=O)=O C(=O)(C=C1SCC(=O)N1C)NC1C(CNC(CN(CCC#C)C)=O)CCC1 c1(C(N2CC(C(F)(F)F)OC(C)(C)C2)C(=O)NCC=C)sc([N+](=O)[O-])cc1Cl C=CCC(C(=O)N1CCC(C)(NC(c2cc(C(C)(F)F)n[nH]2)=O)C1)NC(C)=O Cc1nc2ncnn2cc1C(=O)NC1CN(C(c2cnns2)=O)C2CCCCC12 c1(N2CCC(COC)C2)nc(N2CCN(C)C(=O)C2)c2ccccc2n1 c1(C(=O)NC2CCN(C(C(N3C(=O)CCC3=O)CC)=O)C2)sccc1S(N)(=O)=O n1(CC)ncc(C(N2CC(NC(=O)COC3CCCCC3)C(CO)C2)=O)c1C N1(C(CC2N(Cc3c(OC)ccc(Br)c3)CCC2)=O)CCc2ccc(F)cc2C1 Cc1cc(Br)c2c(c1)CN(N1CCCC(C(=O)OCC(F)F)C1)CC2 c1(C(=O)NC(C(C)C)CNC(C2(O)CCC2)=O)cc(CO)ccc1Cl C#CCCCCCC(=O)NCC(=O)N(CC(C)C(C)(C)C)CC.C(COC)N n1(CC)c(C)cc(C(N2CC(NC(c3ccc(C4CC4)nc3)=O)C3CC23)=O)c1C Cc1c(Br)ccc(S(=O)(=O)N2CCCN(CCS(C)(=O)=O)CC2)c1F c1(CN2CCC(NC(=O)C3CC3)C2)cn2c(Br)cccc2n1 Cc1ccc(I)c(NC(C2CN(Cc3ccc(O)cc3Br)CC(F)(F)C2)=O)c1 c1(COC(C2CC2Cc2ccc(Cl)cc2Cl)=O)cc2cc(F)ccc2o1 Cc1nc(CC(=O)NCCNC(=O)CCCc2ncc(C)o2)c(C)s1 C1(C(F)(F)F)(C(=O)NCC(C2CC2)SCC)CCCCC1 Cc1cccc(C(O)C(=O)NC2CC(F)CN(C(=O)C=Cc3cnc[nH]3)C2)c1F c1(NC(C2CC2C(N2CCN(c3ccccc3F)CC2)=O)=O)cnnc(Cl)c1Br C1(CNC(c2n(C)ncc2)=O)CCCCN1C(=O)CCc1ccco1 C(=O)(C(CC)(CC)OC)N1C(C(C)NC(C=CCN(C)CC)=O)CCC1 C1(NC(C2(COC)CC(=O)C2)=O)CCN(C(=O)C(Cl)=CCl)CC1C c1(C(C(=O)NCC2C(NC(C(C)(C)OC)=O)CCC2)OC)ccc(OC)cc1 C1(C(=O)NCC(CN(C(CCOCCC)=O)C)(C)C)CC12CCC(F)(F)CC2 C1(NC(=O)NC(C)CN2CCCCCC2)CC2(CCC(C)(C)C2)C1 c1(C(=O)NC(C2CCCN(C(=O)Cc3ccnn3C)C2)C)cccc2c1CCC2 C1(NC(CCC=C)=O)CC(OC)CN(C(c2c(C(F)(F)Cl)n[nH]c2C)=O)C1 C1(C(=O)NC(C2CCN(C(c3cccc(C)c3)=O)CC2)CO)CC2(C1)CC2(F)F C1(NC(CC(CC)O)=O)CN(C(=O)COC(C)CC)CCC1CO CCCC(C(=O)NOCC(=O)OC)NC(c1c(Cl)cnn1C)=O c1(C(=O)NC2C(NC(c3nc(N(C)C)oc3)=O)CC2)cc(Cl)sc1Cl c1(N2CCC(NC(=O)NCc3cc(-c4ccc(O)cc4)[nH]n3)C2)ccc(Br)cn1 c1(C(N2CCOCC(NC(CC=C)=O)C2)=O)c(C)nc(C(C)C)nc1O N1(C(C(CCC#C)NC(=O)OC(C)(C)C)=O)CCN(C(C)C)CC1(C)CC Cc1cc(C(N2CCC(CN(C)C(c3cc[nH]n3)=O)C2)=O)cc([N+](=O)[O-])c1Cl Cc1ccnc(C(C)NC(=O)CC2(C)CCN2C(C2C3CCCCC23)=O)n1 C(CNC(c1cc(Br)sc1C)=O)(C(C)(C)C)NC(CC1(NC(C)=O)CC1)=O c1(C(c2ccc(C(N(OC)C(C)C)=O)o2)OC)ccc(F)c(F)c1.N1CCCC1 C1(C(=O)NC(C)CNC(=O)Cc2cc(C(F)(F)F)no2)CCCS1(=O)=O c1(C(=O)NC2C(CNC(C3(CC#C)CCCC3)=O)CC2)c[nH]cc(F)c1=O N1(C(C(C)OC)=O)CC(CNC(c2ocnc2C)=O)CC12CCC2 C(=O)(C(O)CCC(F)(F)F)NC(C1CC2(CCOCC2)CO1)C C(CCCC(C)NC(=O)Cn1nnnc1C1CC1)NC(C1C(C(=O)OC)C=C1)=O C(=O)(C(C(C)(C)C)C1CCC(F)(F)CC1)NCCN(C(=O)C(F)C(C)(C)O)CCC Cc1cn2c(C(=O)NC(C3CCN(C(C4CCC(=O)C(C)C4)=O)C3)C)cnc2s1 N=c1nc2c(c[nH]1)CC(C(N1CCCN(C(c3ccsc3)=O)CC1CO)=O)CC2 N1(C(C)C)C(=O)CCC1C(=O)NCCC(C)NC(C1CC1c1ccc(Cl)nc1)=O c1(CN(C(=O)CSS(C)(=O)=O)CCNC(C2C(C=C)C2)=O)ccc(Cl)nc1 C(=O)(C#CC(C)(C)CNC(=O)CC1CCC(O)C1)NCCc1c(C)nccn1 c1(C(=O)OCC(CCCC(=O)OC(C)(C)C)=O)cc2n(n1)CCCNC2=O c12ccc(O)c(c1)C(=O)N(C1CC1)CCCO2.c1(C(=O)O)ccc(C(F)F)cn1 C1(C#N)(C(N2CC(CCNC(C(C)CSc3ccccc3)=O)C2)=O)CCOCC1 N1(C(c2cc(C)nn2C)=O)CCN(C(C2(CO)CC2)=O)CC1CC#N c1(OC)ncc(Cl)c(C(=O)NCC2CCN(C(=O)Cc3nc[nH]n3)CC2C)c1Cl N1(C(c2ccn(COC)n2)=O)CCCN(C(C2CCCN2C=O)=O)C(C)C1 S(=O)(=O)(c1ccc(F)c(F)c1F)N1CCC(C#N)(NC(C2CCN(C)C2)=O)C1 C1(C(=O)NC(C2CCN(C(=O)OC(C)(C)C)CC2)C)CCCC(C(=O)O)O1 CC1CCCC(CCN(C(C2CCCN(C(=O)Cc3cnoc3)C2)=O)C2CC2)C1 C1(C)(CC(=O)OC)CCCN1C(=O)NCc1ccccc1-c1cn[nH]c1 S(=O)(=O)(c1ccc(Cl)cc1)N1C(C(N2CCC(O)CC2)=O)CCC1 c1(CC(=O)NCC2(CC=C)CNCCO2)cc(F)c(C)cc1F N1(C(C(C(C)C)(C)C)=O)CC2(CCOCC2)C1c1cn(Cc2cccc(Cl)c2)nn1 CC1(C)C=CC(NC(=O)COCCNC(c2cc(N)cc(F)c2)=O)CC1 N1(C(CC2(C)CC2)=O)CC2CC(C1)N2C(C1CCC(C(N)=O)O1)=O C(=O)(C1CCCn2cnnc21)NC(CNC(Cn1ncc(C#C)c1)=O)C1CC1 N1(C(c2cc(OCC)ncc2)=O)CCC2(CCCC2NC(=O)CNS(C)(=O)=O)C1 CCC(CC(F)(F)F)C(=O)NCCC1CN(C(=O)CC2CC3CC3C2)CC(C)O1 C1(N(C(=O)CCC2CCCN(C)C2)C)CC2CCC(C1)N2CC1CCOC1 CC1OC(C)CC1C(N1CCN(C(=O)Cc2cn(CC3CCOC3=O)nn2)CC1)=O CCS(=O)(=O)CC(=O)N1CCCCC(NC(=O)CCc2ccnc(C)n2)C1 C1(CNC(CC(CCC)O)=O)CN(C(=O)C=CC=C(Cl)Cl)CC2(CCC2)O1 N#Cc1cc(C(=O)N=c2nc(CCOc3ccccc3)[nH]s2)ccc1O c1(C(=O)NC2C(CNC(c3cc[nH]n3)=O)C2)ccnn1C1CCCCC1 C=CC(C)(C)CC(=O)NCC(C(=O)NC(CC)C(=O)N(C)C)c1ccccc1 N1(C(C(C)NC(CC)=O)=O)CCC(CNC(c2ccc(Br)o2)=O)C1(C)C CCCC(C)(C)CC(=O)NC1CCCC(NC(=O)COCCSC)CC1 N1(C(C(C2CCCO2)NC(CC(=O)NCC)=O)=O)CCC(C)(CC(=O)OC)C1 N1(C(C2C=CC(NCc3ccn(CC)n3)C2)=O)CCC2(CC1)CC2(F)F c1(C(N2C(C)CC(NC(=O)CC3CCOC3(C)C)CC2)=O)cn2c(n1)CCCC2 N1(C(C2(CC)CCCNS2(=O)=O)=O)CCN(C(=O)Cc2ccc(Cl)s2)CC(O)C1 C(=O)(CCC(C)S(C)(=O)=O)NC1CCC2CN(C(COCCC#C)=O)CC21 C1(NC(=O)CCOC)CC(F)(F)CC1NC(C1CCC1)=O.c1(N)ncc(F)cn1 CC1CCCC(C(=O)NCCCC(N2CCC(N=[N+]=[N-])C2)=O)CC1 c1(C(=O)NC2CCC(CCC(N3C(COC)CC(O)C3)=O)C2)n[nH]cc1[N+](=O)[O-] c1(C(N2C3CC(NC(C(C)(C)CF)=O)C2CC3)=O)sccc1S(N)(=O)=O C=CC1(CC(=O)NC2CCN(C(C)=O)C2C)CN(C(=O)COC)C1 c1(-c2ccc(OC)c(OC)c2)ccc2c(O)c(C(=O)O)cc(CO)c2n1 C#Cc1cc(C(=O)NC(CNC(=O)C(CC(C)C)OC)CC)cc(N)c1 c1(CC(=O)NCC23N(C(CN4CC(C)C4)=O)CC(C2)C3)ccc(S(N)(=O)=O)cc1 c1(CC(=O)NCC(C2CCCCC2)NC(CCOC)=O)sc(C)cc1C C1(C(=O)NC(COC)CO)COC(CNC(=O)CCC=CC(C)C)C1 C1(NC(COCC(=O)NC)=O)(CO)CCCN(C(=O)C=CSC)C1 C1(C(=O)OCC)CC2(C1)CN(CCCC1CC(C(C)(C)C)C1)C2 C#CC1CCN(C(C23CC2CN(C(c2cnc(C)s2)=O)C3)=O)C1 C=CCCC(O)CNC(C1(C(C)C)CCN(C(=O)CCCC2CC2)C1)=O c1(C(C(=O)NCC(C)CNC(c2cc(C3CC3)[nH]n2)=O)OC)ccc(F)cc1 c1(OC)ccc(OC)c(C2CC(S(=O)(=O)OC(C3CCCC3OC)=O)C2)c1 N1(C(C(CCC)NC(=O)Cn2ccc(C)n2)=O)CC2(CC(N(C)C)C2)C1 C1(NC(C=CC(C)(C)C)=O)CN(C(c2ccc(C(O)CF)cc2)=O)CC1(C)C c1(C(=O)NCC2(COC)CCN(C(=O)C(F)OC)C2)ncc(OC)nc1OC N1(C(C(=O)NCCOC)=O)CCC(CO)C(NC(c2oc(Br)nc2C)=O)C1 CC(CC(C)(C)C)C(F)C(=O)N1CC(CCNC(=O)C=Cc2cocn2)C1 Cc1ccc(Cl)c(N=c2scc(-c3ccc(Cl)s3)n2CCC(C)C)c1Cl c1(CNC(C2CCN(C(C3CCC(=O)C3)=O)C2)=O)ccc(O)c(F)c1 c1(C(N2CCC(OCCCO)CC2)C(=O)NCC(F)F)ccc(C2CC2)cc1 C(=O)(C1=Cc2ccccc2C1)N1CC2(CC(CC(C)(C)C)=O)CC1(CNCC1CC(O)C1)C2 C(CC(Cc1cn[nH]c1)C1CC1)NC(c1cc(C(=O)O)co1)=O c1(C(CNC(CCC)=O)NC(=O)COC2CCOCC2)ccc(Br)c(C)c1 C(=O)(CCC(C)NC(C1CC1C(C)NC(=O)Cc1ccc(O)cc1)=O)OC O=C1NC(=O)C(CCNC(=O)CC2(NC(C3CC(=C4CCC4)C3)=O)CC2)N1 N1(C(CCC(=O)NCCCOC)=O)C(C)C2CC1C2NC(c1ccncc1Cl)=O C(=O)(C(F)C(=O)N1CCSCC1C(N1CCCC1CC1CCC1)=O)OC C(=O)(C(CC(=O)N1CCC(CCN2CCCO2)C1)C(C)=O)OCC CN1CCCC(C(=O)NC2CCC(Cn3cc(CCNC(N)=O)nn3)CC2)C1 N1(C(CCc2c(C)noc2Cl)=O)CCCC2(NC(c3cc(C)n(C)c3)=O)CC2C1 Cc1cc(-c2cccc(C(=O)NOCCOc3ccccc3)c2)ccc1C#N C12(NC(=O)C=CC(F)(F)F)CCCC1CN(C(c1cccc3[nH]ccc13)=O)C2 N1(C(c2cc[nH]n2)=O)CCC2CN(C(c3ccoc3C(F)(F)F)=O)CC2C1 c1(OC)ccnc(C(N2CC(NC(C3CCCCO3)=O)CCC2C)=O)c1N CC1=C(C)CC(C)(C(=O)NCCC2CSCCN2C(=O)COC2CCCC2)CC1 N1(C(C(N2C(=O)CCC2=O)C)=O)CCC2CCN(C(=O)Cc3ccnn3C)CC12 C1(C(N2CC(C3(O)CCCC3)C2)=O)CN(C(C2CCCOCC2)=O)CC1(F)F N1(C(C(COC)O)=O)CCC(NC(=O)C(c2ccccc2)=O)CC1C C1(NC(CC=CC)=O)CCC(C(=O)NCCN2CCC(O)CC2)CC1 CC(C)(F)CC(=O)N1CCC(CNC(=O)Cn2ccccc2=O)C1 C(=O)(C1CCCn2cnnc21)N1CCC2CN(C(c3c(C)sc(O)n3)=O)CC21 C1(C(N2CCCC(NC(Cc3n(C)ccc3)=O)CC2)=O)CS(=O)(=O)CC12CCC2 N1(C(c2cccnc2)=O)CC2(CC(C(=O)NCC3(Sc4ccno4)CC3)CO2)C1 c1(C(C(N2C(CNC(c3c(CC)occ3)=O)C=CC2)=O)C)ccc(Cl)c(Cl)c1 O=C(CC(C(F)F)NC(C1CC12CCCC2)=O)NC12CCN(CC1)CC2 Cc1c(C(=O)NC(CNC(=O)CNC(N)=O)C2CC2)cnc2c(Cl)cccc12 CC1(C)CN(C(=O)C=CC2CCC2)C(CNC(C2CC2(F)F)=O)CO1 c1(C(N2CCN(C(C3C(C)C3(F)F)=O)CC2)=O)nnc(O)cc1O Cc1[nH]nc(C(=O)NC(C2CCN(C(C3CCCCC3F)=O)CC2)C)c1C Nc1c(C(N2CCC(NC(C3CCc4nccn4C3)=O)C2)=O)nc(O)nc1O N1(C(CCC2CC(OC)C2)=O)CC2CC(C1)N(C(=O)C(C)SCCN(C)C)C2 C(=O)(C(C)C(C)c1ccc(F)cc1)NCC(C)CNC(C1CCCO1)=O N1(C(=O)OC(C)(C)C)CCc2ccncc2C1C.Cc1cccc2c1NC2=O C1(COCCNC(c2c(C)[nH]nc2Cl)=O)CN(c2ncc(Cl)cn2)CCS1(=O)=O c1(C(=O)NC(C)CNC(=O)CC2CC(=O)NC2=O)c(Br)c2ccccc2n1C C1(COC)(CNC(c2ccc(C3CC3)s2)=O)CCN(C(C2(C)C=CCCC2)=O)C1 C1(C(=O)NC2CN(C(C3C(C)(C)C3(F)F)=O)CC23CC3)=CNC2=CC=CC=C1C2 N1(C(C2N(C(C(C)C)=O)CCC2)=O)CCC(C2(NC(=O)CN3CC(C)C3)CC2)C1 N1(C(c2ccc(C(C)=O)[nH]2)=O)CC(CNC(c2ccc(C)o2)=O)CC(C)(C)C1 C1(CC(=O)NC(C#C)C)(NC(=O)CCNC(=O)COC)CCC1 N1(C(c2c(CC)csc2)=O)CCCC(c2cn(CCC(C)(C)C)nn2)C1 CCS(=O)(=O)C=CC(=O)N1CC(C(C)NC(c2csc3ccccc23)=O)C1 c1(C(C)C(=O)NC2CC(CNC(=O)CC3CCCSC3)C2)ccc2c(c1)OCO2 C(=O)(C(O)CC12CC(C1)C2)NCCN(C(=O)Cc1ccoc1)CC C(CC(C(C)C)NC(=O)C(C)SCCN=[N+]=[N-])N(C(c1c(OCC)ccs1)=O)C C1(C(N2CC(NC(C3N(S(C)(=O)=O)CC3)=O)(CO)C2)=O)CCN(C)C1=O N1(C(CC2C(C)(C)C2)=O)CCOCC2(COCCN2C(c2snc(Cl)c2Cl)=O)C1 c1(NC(CC2N(C(c3c(C)nccn3)=O)CCOC2)=O)c(C=O)c(C)nn1C C1(NC(C2(CC)CCN(C(c3cc(OC)ccn3)=O)C2)=O)CCC(O)C(O)C1 c1(C(=O)OC)scc(-c2ccc(C)cc2)c1NC(=O)Cc1ccns1 c1(C(N(C2CCCN(C(C3CNC(=O)C3)=O)C2)C)=O)cnc(C(F)(F)F)cn1 c1(CC)cnccc1C(N1CC(OC)CC1CF)C(=O)NC(C)C(=O)OC c1(CNCC(=O)NCc2c[nH]c(=NC3CC3)cn2)ccc([N+](=O)[O-])cc1F Cc1nc(O)ccc1C(N1CCC(O)(C(C)NC(=O)CN(C)C(N)=O)C1)=O Nc1cc(C(N2CCCC(NC(C34CCCN(CC3)C4)=O)CC2)=O)ncc1F c1(C(=O)NC(C2C(CNC(C(C3CCCC3)OCC)=O)C2)=O)ccc(O)c(C)c1C C(CCCC(=O)NCC1CN(C(=O)C(=O)NCC(F)F)C2CC12)SC N1(C(CCCN(C(C)C)C)=O)CCCC2(C1)CN(C(=O)CCS(C)=O)CCO2 N=c1c(C(N2CC3CC(NC(C4(Br)CC4)=O)C3C2)=O)c[nH]c2ccccc12 C1(O)(CNC(CCN(C(C)=O)C)=O)CCCN(C(C2CC2(C)C(F)(F)F)=O)CC1 N1(C(c2ccc(CC)cc2)C(=O)O)CCC2(COC(C)(C)C2)C1 N1(C(C=CCC)=O)CC2CCC1C1CN(C(c3cccc(N)c3F)=O)CC21 c1(NC2CN(C(C)C)CC2C)nc2c(c(=NCC3OCCOC3(C)C)[nH]1)CSC2 C1(C)(C(=O)NC2CC3(CN(C(CCC)=O)C3)C2)Oc2ccccc2NC1=O c1(N(C(C(N)C2CCC2)=O)C2CC2c2ccccc2)ccc(F)cc1 C12(NC(CNC(CCC)=O)=O)CCC(CNC(c3cnsc3)=O)(C1)OC2 c1(OC)c(F)ccc(F)c1C(N1C2CN(c3nccc(Br)n3)CC12)=O c1(CC(C(=O)N(CCC(C)NC(c2c(CC)cno2)=O)C)C)ccccc1C C(C(C(C)C(C)C)NC(c1ccoc1C)=O)NC(c1scc(C)c1Br)=O Cc1[nH]nc2ncc(C(=O)NC(CNC(=O)CS(=O)(=O)N(C)C)C(C)C)cc12 c1(C(N2C(CNC(C3C(C)OCCO3)=O)CC2)=O)ccc(N)c(N)n1 CN1CC=C(CC(=O)NC2CN(C(c3c(F)cc(O)cc3F)=O)CC2F)CC1 c1(C(=O)OC)ccc(NC(C2CCN2C(=O)CCCC2CCCC2)=O)c(OC)c1 C12COC3(C1)CN(C3)C(=O)CNC(=O)CO2.c1(OCCOCC)ccccc1F C1(NC(CCc2cc(C)no2)=O)(CO)CCCN(C(=O)CC2CCOC2(C)C)C1 C1(C(=O)NC(c2ccccc2)CC=C)CN(C(=O)CCC)CCO1 C1(NC(c2c(C)n(CC(F)F)nc2)=O)CCN(C(C2OC(C)CC2C)=O)CC1C CC1CCC(NC(c2cc(O)nc(Cl)c2)=O)CN1C(=O)CC1C(C)(C)C1(C)C C1(COC)(CNC(C2CSCCS2)=O)CCN(C(=O)C(C)(O)COC)C1 C(=O)(CS(=O)(=O)CC(C)C)NC(CNC(C(C(=O)NC)(C)C)=O)(C)CO N1(C(C(CCC)OC)=O)CC2CCC1CN2C(=O)CCc1cn(C)cn1 C1(C(=O)NCC(CNC(c2ccc(C(C)C)o2)=O)OC)CCCCS1 C#C[Si](C)(C)CCCNC(=O)NCC1CC1(F)F N1(C(C2C(C(=O)NC(C)C(=O)O)C2)=O)CCOC(C2CCCCC2)CC1 C1(C(=O)NCC2CN(Cc3csc(-c4ccccc4)n3)C2)CN2CCN1CC2 C1(C(=O)NC2(C)CC(C(=O)NCCC=CC=C)C2)CN(C)CCN1C CC1CC(CC(=O)NCc2nc[nH]n2)CN1C(c1csc(C#N)c1)=O c1(C(N2CCC(CNC(CC(C)(F)F)=O)C2)=O)ccc(F)cc1Br C1(N(C(C2CCCN(CCC)C2)=O)C)CC2CCC(C1)N2C(=O)COCC1CC1 c1(OC)ccccc1C(=O)C(=O)NCCN(C(c1cnn(CCF)c1)=O)C(C)C N1(C(CCc2ccc(C)o2)=O)CC2CCC1C2NC(c1cncc(N)n1)=O CC(CS(=O)C(F)(F)F)NC(=O)C(=O)NC1CCC(C(=O)O)CC1 N(C(=NCC(C)C1CC1)N1CCC(NC(=O)C(C)(C)C)C1)CCOC N1(c2nnn(C)n2)CC2CCC1C(NC(C1CCCCC1C1CC1)=O)C2 CCCCC(C)C(=O)N1CC2C(CNC(C3CC4CCC(C3)S4)=O)C2C1 c1(C(N2C(C)CC(NC(CC(C)C)=O)C2)=O)ncnc(O)c1Cl C12CCC(CC1)N(C)C(=O)C1CN2C1.C1(C(=O)ON(C)C)(CNC(C)=O)CC1 C(CCCCNC(=O)Cn1ccc(C(F)F)n1)N(C(=O)COC1CC1)C O(NC(=O)CC(CC1CC1)NC(=O)C=Cc1cnn(C)c1)CC=C c1(C(C(=O)NCCCC)N(c2ccc(F)cc2)C)cc(F)nc(F)c1F c1(C(=O)NC(CCN(C(C(C(C)C)N(C)C)=O)C)C)cccc2nncn12 c1(C(=O)NCC2CC(NC(C(C)C3CCCO3)=O)C2)ccccc1-c1cn[nH]c1 C(C(C)(O)C(C)(C)C)CC(=O)N(C(c1n(CCOC)ncc1)=O)C.C(C)(C)(C)OC=O c1(C(=O)NC2CCC(CNC(C3C(C)(CC)C3)=O)C2)cc2oc(C)cc2[nH]1 N1(c2ncc(C)c(O)n2)CCC(NC(=O)CC(C)(C)C2CCCO2)CC(C)(C)C1 N1(C(CC)=O)CC(CN(C(=O)CCCF)C)C2(CC2)C1 CS(=O)(=O)c1ccc(F)c(-c2cn(CC(N3CCC(C4CCC4)C3)=O)nn2)c1 S(=O)(=O)(c1ccc(N(C)C)c(F)c1)NCC(CO)N(C)C.C1C(F)(F)C(=O)N1 c1(C(N2C(C(=O)OCC)CC(O)C2)=O)ccc(N2CC(C)(OC)C2)c([N+](=O)[O-])c1 c1(OC)ccc(C(=O)N(C)CCN(C(=O)C(O)P(C)(C)=O)C(C)C)c(Cl)n1 C1(C(=O)NCc2occ(C)c2)CCC=CC1NC(=O)CCCF C1(NC(Cc2cc(COC)on2)=O)CCN(C(=O)Cn2nnc(=N)[nH]2)CC1C C1(CC(=O)NCC(C)CNC(C2CCOC2=O)=O)OCCC1C C1(C(=O)NC2(C)CN(C(Cc3c(C)noc3C)=O)C2)Cc2ccccc2C(=O)O1 C(=O)(CN=c1cc[nH]cc1)NC1CCC(NC(C(CC)=CCCC)=O)C1 c1(NC(CCc2ccc(C(=O)Nc3scc(C)c3C)[nH]2)=O)ccn2cnnc2c1 C=CCC(C(=O)N1CC(COC)(NC(c2cc(C3CCC3)no2)=O)C1)OC c12ccc(cc1)OC2C.C1(C(=O)NCC(=O)N(CCSC)CC)CCOC1.C1CO1 CC(C)C(C(=O)N1CCCCC1Cc1cn(Cc2ccno2)nn1)C1CCC(=O)N1 C(=O)(C1=Cc2ccc(Cl)cc2OC1)N1C2CN(C(C(C)=CC)=O)CC1CC2 c1(C(=O)NCC2CCCC(CNC(C3CCO3)=O)C2)c(F)cc(F)cc1F c1(C(=O)NCC2C(C)CCN2C(=O)CCCc2ccsc2)ccc2c(n1)CCC2 C1(C(=O)NC(c2nnc(O)o2)C)CCC(O)CN1C(c1cc(Cl)c[nH]1)=O c1(NC2(C(=O)NCC(=O)OC)CC2)ccc2c(Cl)ncnn12 N1(CC(C)NC(=O)C(C)CF)CCN(C(C2(C(=O)C3CC3)CC2)=O)CC1 C1(CCC(=O)NCC2CCCN(C(C3C(C#N)C3)=O)C2)CCc2ccccc2C1 c1(CC(=O)NCC2(C)CCN(C(C3(CC)COC3)=O)C2)c(O)ncnc1O CCC(C)CCC(=O)NCCN(C(C1CCC12CCCO2)=O)Cc1ccccc1 c1(CC(=O)NCCOCCCNC(=O)C=CCF)ccc2c(c1)OCCCO2 C(=O)(C(N=[N+]=[N-])C(C)C)NCC(C(=O)N(CC(C)OC)C)C N1(C(C(C(=O)OCC)F)=O)CCC2CCN(C(=O)C(C)O)CC12 C1(C(=O)NC(CC)CC(C)O)(CC)CCCN(C(C2CC(OC(C)=O)C2)=O)C1 C1(C)(C(=O)NC2CC(CNC(c3c(SC)cccn3)=O)C2)CCN(C)CC1 c1(NC(C2(CC=C)CC2)=O)ccc(NC(C2CCCCS2(=O)=O)=O)cc1C C1(C#N)(C(=O)NC2CC(O)(CNC(c3cn(C(C)(C)C)nc3)=O)C2)CC2CC2C1 N1(CCN(CC(F)F)C)CCN(C(C2CC3CC3C2)=O)CC1.N1CC1 CC(C)(C)C(CNC(C1CCC(O)C1)=O)C(=O)NCC1CC12CC2 c1(C(N2C(CCOC)CN(C(=O)C(C)CSC)CC2)=O)cc2ccccc2nn1 N1(C(COC(C(N2CCC(C)C2)=O)=O)=O)CCC(OC2CCC2)CC1 c12ccc(Cl)nc1CNC(=O)N2.C1(CC)CC(NC(=O)C(O)C2CC2)CCO1 c1(NC(C(=O)NCc2ccc(C(OCC)OCC)cc2)=O)coc(S(C)(=O)=O)c1 C1(NC(c2ccc(C)nn2)=O)CC2(C1)CC(NC(=O)Cc1cnsc1)C2 N1(CC(N2CC3C(C)C3C2)=O)CCN(C(=O)C(C)(C)N(C)C)CC1=O c1(C(=O)OC(C)C)ccc(OC(=O)NC2CC(CF)C2)cc1 c1(C(=O)NC23CC(NC(CC4CCN(OC)CC4)=O)(C2)C3)ccc2c(n1)CCO2 C(=O)(CC(C)C(C)C)NCC(Cc1ccccc1)NC(c1oc(CC)c(C)c1)=O C=C(Cl)CC(C(=O)N(CC(C)(CC)OC)C)NC(C1CCCN1C)=O Cn1nc(C(=O)NC2CCC23CN(C(C2COC(=O)O2)=O)C3)ccc1=O Cc1ccc(N(C)C(C)C)c(C(=O)NC2CC(CNC(C3CC34CC4)=O)CC2O)c1 CC1CN(C(=O)CC(C)n2cc(Br)cn2)CCCN1C(=O)Cn1cccc1 N1(CC)CCCC(C(N2CC3CC3(C(=O)NC3(C)CC(F)(F)C3)C2)=O)C1 C(=O)(C(C)(C)C)N(C(CC)CNC(=O)Cc1ccnn1CC(C)C)CC C(c1ccncc1)=CC(=O)NCC1(C(=O)NC2CCCCCCC2)CC=CC1 Cc1ccc2nc(NC(=O)CNC(C3CCCN(C(=O)C4CC4)C3)C)sc2c1 C1(NC(C2C3COCC23)=O)CN(C(C2CCCOC2)=O)CC12CCC2 CC1(C(=O)NCC(CO)NC(c2cc[nH]c2C2CCCC2)=O)CCCNC1=O C1(Cc2ccc(CN3CCCC3)cc2)CCC12CN(C(c1ccc(CN)[nH]1)=O)C2 C1(C(N2C(C(C)NC(=O)COCC(F)(F)F)CCC2)=O)CC(=O)NC1(C)C c1(C(N2CC(C(C)(C)O)(CNC(c3cnc(C)[nH]3)=O)C2)=O)c([N+](=O)[O-])cnn1C Cc1cc(C(=O)NC(N2CC(Cc3cnc(CC(C)(C)C)s3)C2)=O)ccc1N Cc1ccccc1C(=O)NCc1csc(CNC(=O)C(O)C(F)F)n1 N1(C(C(C2CCN(CC)C2)=O)C)CCN(c2cnn(C)c2)C(=O)C1=O N1(C(C(C(CC)C)OC)=O)CCC(C2CC2)(CNC(=O)C(C)(C)CO)C1 c1(C(=O)NCc2ocnc2C(N2CCC2CO)=O)cc(Cl)cnc1O.C(COC)OC c1(NC(N2CC(NCCN3CCN(C)CC3)C2)=O)ccc(I)c(F)c1F c1(C(N(C)Cc2scc(C)n2)=O)ccc(CNC(=O)C(F)CC2CCOC2)cc1 C1(C(N(C2CCN(C(=O)C3=C(C)CCCC3)CC2)CC)=O)CC12CCC(=O)CC2 c1(C(=O)Nc2c(OCC)cc(C#N)cc2)cncc2cnccc12 N1(C(CCCCCSC)=O)CCN(C(=O)CC2CC(OC(F)F)C2)CC(CO)C1 C1(CNC(CCN(C(CC)CC)C)=O)COC(C)(C)CN1C(C1CC2CC2C1)=O c1(C(C(=O)N(CCC(C)NC(C2COCC2C(F)(F)F)=O)C)O)ccccc1Cl CCCC(C)(C)C(=O)N1CC(O)(CCNC(=O)C(C)Oc2cccnc2)C1 c1(C(N(C2CCN(C(c3c[nH]cc(F)c3=O)=O)CC2)C)=O)cc(O)c(O)c(O)c1 C1(CN(C(C2CC(CN(C)C)C2)=O)C)C2CN(C(c3cc(Cl)cn3C)=O)CC12 N1(C(CCOC)=O)CCCC(NC(c2sccc2CON(C)C)=O)C1 N1(C(CCCN(C)C(c2ccccc2CC#N)=O)=O)CCC(C)(O)C1 Cc1cccc2[nH]c(C(=O)NC3CCCN(Cc4c[nH]c5ncccc45)C3)cc12 CC(C)(C)C(CNC(C1CCCC1O)=O)C(=O)NCc1cnn(CCF)c1 n1(CC)cc(C(=O)NC(CC(=O)NC(C)(CC)CO)C2CC2)c(C)n1 C(c1ccc(SC)s1)=CC(=O)N(CC(C)NC(=O)CCn1cnnn1)CC C(=O)(CCC(N)=O)N(CC(=O)NCCN(C)C)C(C)C Cc1cc([N+](=O)[O-])c(C(=O)NC2CCC(F)(CNC(=O)C(C)O)C2)cc1Cl N(C1CCCc2c1cnn2C)CCN(C(CCN1CCCC(N(C)C)C1)=O)C C1(CNC(C(CCF)NC(=O)CCCC2CCCO2)=O)CC2OC1C1CC21 N1(C(CC2N(C(C(CC)CO)=O)C3C2CCC3)=O)CCc2ccc(C)cc21 c1(NC(C2=C(C)OCC2)=O)ccc2c(c1)CCN(C(=O)C(C)(C)C(F)(F)F)C2 CCC(CCC(=O)NCc1cc(C)ncn1)NC(=O)C(C)NC(=O)NC N1(C(C2N(C(COCCC(C)C)=O)C(C)C2)=O)CCCC(O)(C2CC2)C1 c1(C(N2CCC(O)(C(C)NC(=O)C=CBr)C2)=O)ccc(N)c(O)c1 C(=O)(C(C(C)NC(=O)C(O)CC1CCC1)C(C)C)NCC1(C(=O)OC)CC1 C(c1ccc2ncccc2c1)=CC(=O)NC1CCCC1NC(=O)CC1CCOC1 c1(C(=O)NC(CC)CNC(=O)CCCc2ccsc2)cccc(S(C)(=O)=O)c1 C=C(C)CC(C(=O)NC1CCC(=O)NC1)NC(c1cn(C2CC2)cn1)=O N1(C(N2CCN(C3CC3)CC2)=O)CCC(F)(C(=O)NC2CC2)C1 c1(OCC(=O)N(C2CCCN(C(CCC3C(C)C3)=O)C2)C)cc(F)ccc1F C1(OC)CN(C(=O)COCCc2cccc(F)c2)CC1CNC(C1CC=CC1)=O C(=O)(C(C)n1ccnn1)N(CC(C)N(C(=O)Cc1cscn1)C)C c1(OCC2CN(C(C(CC)N(C)C)=O)C(=O)C2)ccc(S(=O)(=O)C(F)(F)F)cc1 c1(CN2CCOCC(NC(c3cccc(O)c3)=O)C2)cc2cccnc2[nH]1 c1(CC)ccc(C=CC(=O)NC(C)CN(C)C(c2ccnn2CC)=O)o1 n1(CC)nc(C)cc1C(N1CCC1CNC(C1(n2ccnn2)CC1)=O)=O c1(C(=O)NCC(C)(CO)NC(c2ccc3c(c2)COC3)=O)ccc2nn[nH]c2n1 CCC(CNC(=O)COC)(CC)C(=O)NC(c1cc(C)on1)C C#CCCN=C(NCc1nc(C2CC2)n[nH]1)NC(C)CCS(C)(=O)=O N1(CC(=O)NC2C(NC(C3(CCC)CC3)=O)CCOC2)C(=O)NC(C)(C)C1=O CC1CN(S(=O)(=O)CCNC(=O)N(C)CCc2ccccc2)CC(C)O1 O(NC(=O)CN(C(=O)C(C)NC1CCOC1)C)CCC#C CC1CCN(c2nnc(CO)n2Cc2csc(-c3ccsc3)n2)CC1C c1(C(=O)NCCN(C(=O)C(O)CC2CC2)CC)ccc(C(C)C)cn1 C1(C(=O)NCC2(N(C)C)CC2)CCN(C(=O)C(=O)C2CCCC2)C12CC2 N1(C(CCC)=O)CC2CCCC2(CNC(c2ccc(-c3ccco3)nc2)=O)C1 Cc1ccc2c(N(C(C)(C)CN(C)C)C)nccc2n1 C1(NC(c2cnc(C(C)C)[nH]2)=O)CC2(NC(C3CC(C)(C)CO3)=O)COC1C2 S(=O)(=O)(c1ccccc1C#N)N1CC2(OCCN(C(CC(C(=O)O)NC)=O)C2)C1 c1(CC)cc(C(N2CCCC(NC(=O)CCC(CC)OC)C2C)=O)ccc1F N1(C(C(C)OC)=O)CC2CC(C1)C2NC(=O)C(CC(C)C)n1ccc(C2CC2)n1 C(=O)(CC(C)(C(F)(F)F)N(C)C)N1CCC(NC(c2c(Cl)cc(CC)c(C)n2)=O)C1 C1(C(=O)NC(CNC(C(CC#C)O)=O)CO)CCCC2(CC2)C1 c1(C(=O)NCC(CNC(c2cc(COC)[nH]n2)=O)C)c(C)ccc(F)c1O c1(C(N2CCCCC(CNC(c3ccsn3)=O)C2)=O)cc2cccnc2o1 C1(NC(CCC(=O)OC)=O)CCC2(CC1)CCN(C(c1ccc(OC)s1)=O)CC2 O=C(CSCc1nc2ccc(Br)cc2o1)NN=c1[nH]c(Cl)c(Cl)nc1Cl C12(NC(N3CC(C4(C=C)N=N4)C(F)C3)=O)CC1COC21CCC1 CC1CN(C(=O)CCN(C(=O)CC2CCC(=O)C2)CCO)CCS1=O N1(C(C23CC(C(=O)NC4CC(N=[N+]=[N-])C4)(C2)C3)=O)CCC(C2CCOC2)C1 c1(C(N2CCCC(C(C)C(=O)Nc3ccc(C(C)C)s3)C2)=O)ccn(C)c(=O)c1 C12(NC(CNS(N)(=O)=O)=O)CCC(F)(F)CC1CN(C(=O)CC1CC13CC3)C2 N1(C(c2ccc(CC)[nH]2)=O)CCC(C(N2CCNC(=O)C2)=O)C1C(C)C N1(CCNC(c2c[nH]nc2CNC(=O)C(F)CC2CCOC2)=O)CCCCC1=O N1(C(c2cc(OCC)no2)=O)CCC(NC(=O)CCc2cncnc2)C(CO)C1 c1(C(=O)Nc2c(O)ccc(C)c2)n[nH]c2c1CN(C(=O)CC1CCN(C)CC1)C2 N1(C(c2c(CC)onc2)=O)CCC(N(CC(C)C)C(c2cc(C)c[nH]2)=O)CC1 C1(NC(C2N(C(c3c(CC)cns3)=O)C(C)C2)=O)CCCN(O)C1=O c1(COC)ccc(C(=O)NCC2CCCC2NC(C23CC(C)C2C3)=O)o1 CC(C)(C)C(C#N)C(=O)N1CCSCC1C(=O)NCCCCN1CCC1 c1(C(N2CCC(C)(NC(C(CCSC)O)=O)C2)=O)cc(C2CC2)cnc1Cl C1(NC(CC(C)(C)C)=O)CC(F)CN(C(c2ccc(O)c(F)c2)=O)C1 C12(CNC(CN(C3CCC3)C)=O)CCC(Nc3ncc(I)cn3)(CO1)C2 N1(C(c2cscc2Br)=O)CCC(CNC(C2(F)CC=CC2)=O)CC1 N#Cc1ccc(CN2CC(NC(=O)Cc3cc[nH]n3)C(C#N)C2)c([N+](=O)[O-])c1 CCS(=O)(=O)CC(=O)NCC1CC2CC1CN2C(=O)CCN1CCN(C)CC1 c1(CNC(C2CC2COCn2ccnn2)=O)oc2ccccc2c1NC(=O)OCC N1(C(CCC(C)C)=O)CCC(C)C(N(C(=O)CCCc2ccc(F)cc2)C)C1 C1(OC(c2c(C)con2)c2nnnn2CSc2ccccc2)CC(C)OC(C)C1 N12CCCCC(C1)C2=O.c1(NC(C2C(C)C2c2ccccc2)=O)ncc(Br)cn1 N1(C(c2ccccc2OC(F)(F)F)C(=O)NCCCCCC)CCN(CC)CC1 c1(NC(CCC=C)(c2nnnn2CCC2(C)CC2)C2CC2)cnc2ncccn12 N1(C(c2ncc(C)s2)=O)CCCCC12CCCN(C(=O)C(Cl)(Cl)Cl)C2 c1(OC)ccc(Cl)cc1CC(=O)N(C(C)CN(C(=O)Cc1cccs1)C)C CC1=C(C)CC(C(=O)NCCC(O)C(N2CC3CC3C3CC23)=O)CC1 Cc1ccccc1SCC(=O)N(C1CCSC1)CC1CCCN1C(C1CC1F)=O C(=O)(CCCCCC#N)N1CC(CC(C)NC(C2(C)N(C)CC(OC)C2)=O)C1 CCC(CC(=O)NC1CC(O)CN(C(C2CC2F)=O)C1)CC(F)(F)F Cc1ncc(C(=O)NCC(C)(C)CNC(C2CC(CF)C2)=O)cn1 c1(CCCN2CCN(C(C(C=C)(C)C)=O)C(C)C2)ccc([N+](=O)[O-])cc1 C1(NC(C(C)(F)F)=O)CN(C(=O)C=CC2CCCCCC2)C2(CCCOC2)C1 C1(CCC)CCCC1C(=O)N(C)CCOCCNC(=O)CCN1CCC(F)C1 c1(CC(=O)NCC2CCN(C(=O)CCC=CBr)CC2)ccc(F)cc1Cl C1(CC)(NC(=O)C(C)O)CN(C(=O)C(C)(F)c2ccccc2)C1 c1(C(N2CC(CNC(C(N3CCOCC3=O)C)=O)C2)=O)ccc2[nH]ccc2c1F N1(C(=O)Nc2cccc(CC)c2)CCC(NC(=O)CC(C)C(F)F)C(CC)C1 C1(C(=O)NCCCCNC(Cc2n(C)cnc2)=O)CCCC(C)(C)O1 c1(C(CNC(CCN(C(C)=O)C)=O)(C)NC(C2CC2(F)F)=O)ccccc1 C(=O)(C1=NN(CC)C(=O)CC1)NC(CC)(CNC(C1CC2CCCCC12)=O)CC c1(COC)cc(C(=O)NC2CCCC2(C)CNC(C2(CO)CCCO2)=O)n(C)c1 c1(CCC)ccccc1C(=O)NC1CCN(C(c2cc(CC)oc2C)=O)C1C C(CCC(C)(C)C(=O)Nc1ccc(NC(c2n[nH]cc2Cl)=O)cc1C)OC N1(CC(=O)NCCOCCNC(C(C)c2cccs2)=O)C(=O)NC(C)(C)C1=O C(=O)(C1CCCc2ccnn21)NC1(CF)CCN(C(C(C)C2CC2)=O)C1 C1(CN(C(=O)Cc2cocn2)C)CCCN(C(c2cnc(=N)[nH]c2)=O)C1 CCCC(C)(CC)C(=O)N1CC(CC(C)NC(=O)C(C(C)CC)OC)C1 C=C(Cl)C(C)(C)C(=O)NC(CNC(=O)Cc1csc(C(C)OCC)n1)CC c1(NC(C(CC2CCC2)NC(C2CC3(CCC3)C2)=O)=O)ccc(CCO)cc1 c1(C(N2CC3CCC(CNC(C(COC)C)=O)(C2)C3)=O)cnc([N+](=O)[O-])cc1C C1(NC(=O)CCC2CCCN2C(=O)CCc2nc[nH]n2)CC2(C1)CC(O)C2 CC(C)CC(CNC(=O)CCn1cccn1)C(=O)N1CCCC1(C)C(C)(C)C C(c1cc(Cl)c2c(c1)OCCO2)=CCCN1CCCC(N(c2ccc(Br)cc2)C)C1 c1(C(C(N2CCCC(CN(C(CC)=O)C)C2)=O)C)ccc(OC)c(OC)c1 c1(OC)cccc(C2CC2C(=O)NCCO)c1.N12CCC(CC1)NC(=O)CC2.OC N1(c2ccnc(CC)n2)CCC2(CNC(=O)CSSC)CCCCC12 N1(C(C(C)OCC=C)=O)CCN(C(=O)Nc2cccnc2)CC1 Cc1cc(C(=O)N(c2cccc(Cl)c2)CCCO)c([N+](=O)[O-])c(O)n1 N1(C(C2N=C(C)SC2)=O)CC(F)(F)CC1(C)CNC(c1cn(C(C)C)cn1)=O C(=O)(CCC(C)(C)O)N(C1CCN(C(=O)C(CC(F)F)C2CC2)CC1)CCOC N1(C(c2c(CC)oc(C)c2)=O)CC(NC(c2cnc(C(C)OC)s2)=O)CC(O)C1 C1(CC(=O)NCC(CNC(C2(CC)CCCCC2)=O)O)COCC(C)(C)O1 CCCCC(CC)C(=O)N(CC(O)CNC(c1cc(-c2csc(=N)[nH]2)c[nH]1)=O)C C1(NC(c2ncn(C)n2)=O)CCSC12CN(C(=O)CC1CCC(C)(C)C1)C2 C(=O)(C(F)(F)CC1CCCO1)NCC1(C(C)NC(Cc2nc(CC)sc2)=O)CC1 CC(c1ccccc1C)=CC(N1CC(NC(c2[nH]nnc2C)=O)CCC1C)=O N1(CC(C)NC(=O)C(O)Cc2ccccn2)CCN(C(C2(O)CCC2)=O)CC1 Cc1cnccc1C=CC(=O)NC1CCCC(NC(=O)C(C)OCC(C)C)C1 C1(NC(c2n(C(C)C)ncc2)=O)CCC(N(C(=O)CC2CCN(C)C2)C)CC1 c1(-c2c(C(=O)NC3C(NC(C=CC(=O)N(C)C)=O)C3)noc2)ccccc1F N1(C(=O)OC(C)(C)C)CC(C(=O)NCCCOc2cncc(C#N)n2)C2(CC2)C1 C=CCCC(C(=O)N(C)CCSC)NC(c1cocn1)=O C1(NC(C(CC(CC)C)=O)=O)COC2(CCN(C(C3(OC)CCC3)=O)CC2)C1 Nc1nc(Br)ccc1C(=O)N(O)Cc1cn(-c2cc(F)ccc2Cl)nn1 C1(NC(CC(C)(C)O)=O)CCC2(CC1)CN(C(c1n[nH]c3c1CCC3)=O)C2 c1(C(C)NC(c2n(CCCSC)nnn2)c2ccc(CO)s2)cn(C)nc1C C(C(=O)NCCSCC(N1CCC2CC12)=O)(C(C)C)OC c1(OC)nccc(C(=O)NC2CN(C(=O)C(C)OCC3CCCO3)C2)c1F N1(C(c2n(C=C)ncc2)=O)CC2ON=C(CNC(c3cc(C)ccc3C)=O)C2C1 N1(C(C(CCCC)=O)=O)CCC(C)(C)C(C(=O)NCCC(O)C(F)(F)F)C1 CCC(C)(COC)CN=c1cc(NCc2cnc(Cl)c(C)c2)nc(C(F)(F)F)[nH]1 C1(CC)(CC)CC(C(=O)NC(c2cn(CC(C)O)nn2)C)C1 c1(C(N(C2CCC(NC(COCCC#C)=O)C2)C)=O)ccc(P(C)(C)=O)cn1 n1(CC(N2CCC(NC(C3N(C)CC(F)C3)=O)CC2)=O)ccc2cc(F)ccc12 Cc1nc(C(F)(F)F)oc1C(N1CC=CC(NC(=O)Cn2cc(C#N)cn2)C1)=O c1(C2(NC(=O)NCCOC3C(C(C)C)(CC)C3)CC2)nccc2ccccc12 C1(NC(CC2OCC(C)(C)C2)=O)CC2CC(C1)N(c1nnco1)C2 N1(C(c2cc(C)sn2)=O)CCC2(NC(=O)C=Cc3ccoc3)CC2C1 Cc1nc2cc(Cl)cc(C(=O)NC3CN(C(c4ccoc4)=O)CC3C(F)F)c2[nH]1 c1(C(N(CCOCCCN(C(c2c(C)nccc2)=O)C)C)=O)cccc(O)c1Cl Cc1noc(C)c1CN(C(=O)C(C(C)C)NC(=O)C1CC1)C.C1(=O)CCCCN1 C1(CN=c2cc(C)nc[nH]2)CCC2(CCOCC2)CO1.c12ccc(N)cc1CN2C c1(CN2C(C(=O)NCCCOC)CCCC2)c(OC)cc(OC)cc1F C(=O)(C1=NOCC1)NCC(CNC(c1c(CC)nc[nH]1)=O)O Cc1ccc(NC(C2CC(O)CN2C(c2ccc(O)nc2)=O)=O)c(C(C)C)n1 C1(CC(=O)NCc2nc(C(=O)NCC(CC3CC3)CO)co2)CC=CCC1 C(C(C)C(=O)NCCC1CC(NC(C2(Cc3ccccc3)CCCC2)=O)C1)OC Cc1cc[nH]c(=N)c1C(=O)NC1C2CN(C(C3CC4CCC(C3)C4)=O)CC12 CCC(C)(O)C(=O)NC(C12CCC(CC1)C2)CNC(c1c[nH]cc1Br)=O c1(CNC(C2(C#C)CN(C(=O)CCc3cncnc3)C2)=O)cnc(F)c(C)c1 N1(C(C=CCCC)=O)CCCC2(CNC(c3cc(OC)cnn3)=O)CCCC12 Cc1c(Br)cnn1CC(=O)N(C(C)CCNC(c1ccc(N)cn1)=O)C c1(C(=O)NC2CN(C(Cc3scc(C)n3)=O)C2)ccc(Cl)cc1F c1(CC)[nH]nc(C(=O)NCC(C(C)C)NC(=O)C(C(C)C)SC)c1[N+](=O)[O-] n1(CC)nc(C(N2CCC(NC(c3ncccc3OC)=O)CC2)=O)cc1C1CC1 c1(C(=O)NC2CCC(NC(C3CN(C)C3)=O)CC2)cc(S(N)(=O)=O)co1 C(=O)(C(C)CC(C)(C)C)NCC1C2N(C(c3scc(C(C)=O)c3)=O)C(CC2)C1 c1(C(N2C3CCN(C(c4cc(C(C)C)no4)=O)C3CC2)=O)ccc2c(c1)OCCO2 Cc1coc(C=CC(=O)NCC23COC(CC4CCCN4C(C4CCC4)=O)(C2)C3)n1 N1(C(C2COC3(CCC3)C2)=O)CCCC(O)(CC2(C)CCCC2)CC1.CC1C(=O)N1 N1(C(C2(COC)CC2)=O)CCCCC(NC(=O)CC(C(F)F)c2ccccc2)C1 CCCS(=O)(=O)CC(=O)OCC(=O)Oc1ccc(Br)cc1F C1(N(CC(C)OC(F)F)C(=O)CC2CCC(C)C2)CC2C=CC1C2 c1(C(N(C)CC2N(C(c3ccnc(C)c3N)=O)CCC2)=O)cccc(S(C)=O)c1 C1(C)(CNC(CCC=CCC=C)=O)CCC(NC(c2ccsc2Cl)=O)CC1 C1(NC(C2CC(C(F)(F)F)(OC)C2)=O)CCN(C(C2(O)CCC2)=O)CC1F N1(C(C(=O)NC(COC)C)C(C2CCC2)OC)CC2CC1CCC2CO C1(C(=O)NCC(CC)NC(C2(N3CCCC3)CC2)=O)CCC2(CCC2)OC1 C(=O)(C(CC(N)=O)NC(C1CC(c2ccccc2)C1)=O)N1CCC(=C)C1 N1(C(C(C)C2CCC2)=O)CCC(NC(C2(S(C)(=O)=O)CC2)=O)C(CO)CC1 CC(C(C)(C)C(=O)NC1CC2C(C1)C2(F)F)NC(c1n[nH]cc1Cl)=O Cc1ncc(Br)cc1NC(C1CC1C(=O)Nc1cnc(C#N)cn1)=O N1(C(C(C)O)=O)C2CCC1CC(CNC(=O)C(c1ccc(F)c(F)c1)(C)C)C2 C(C(C(=O)N(C)CCC1CCCN1C)C(C)C)NC(c1c(OC)ccs1)=O c1(C(=O)NC2CCC(C(=O)NCC(C)(C)C)C2)ccnc2[nH]cnc12 c1(C(=O)NCC2(NC(CN3CCN(C)C(=O)C3)=O)CCC2)cc2c(ccn2C)[nH]1 C1(O)(CNC(C2CCCC2)=O)CCCN(C(=O)CCCn2ccnc2)C1 N1(C(c2c(C)c(I)nn2C)C(=O)NCCSC)CCC(O)CC1(C)C C1(CNC(C(C)n2cccn2)=O)CN(C(=O)CC(C)(C)CN(C)C)CC1(C)C CC1=C(C(=O)NCC(C)(C)CN(C)C(c2coc3c2CCCC3)=O)SCCO1 CC(C)(C)CCCC(=O)N1CCN(C(C2C=CCC2)=O)C(C2CCC2)C1 c1(C(=O)NC(c2ccccc2)CNC(C(C)(C)F)=O)ccn2ccsc12 N1(C(CCOc2ccc(CC)cc2)=O)CCC2CN(C(=O)C(F)=C(C)C)CC2C1 C1(NC(=O)COCC2CCC2)CCN(C(c2ncncc2Cl)=O)CCC1CO CC1OCCC1CN(C)C(c1c[nH]nc1CNC(c1ccoc1Cl)=O)=O c1(N2CC3(c4cccc(OC)c4)C(C2)CCCO3)nc2ccc(N)cc2s1 c1(C(=O)NC2C=CC(C(=O)NCC3CC3[N+](=O)[O-])C2)cnc(Cl)s1 N1(C(C(CC=CC)CC)=O)CC2CC(NC(c3n[nH]c(=N)s3)=O)C(C2)C1 c1(C(=O)NCC2(C)CCCN2C(=O)CCc2ccsc2)cccc(F)c1O c1(C(C)NC(C2CCC3(CC3)C2)c2nnnn2C(C)C)csc2c(Cl)cccc12 CCC(C)CC(C(=O)N1CC2C(C(=O)OC)C2C1)NC(=O)CCN1CCCCC1 c1(C(=O)NC(CN(C)C(c2cc(C3CC3)[nH]n2)=O)(C)C)ccc(N)c(F)n1 c1(OC)cc(OC)c(-c2nc(-c3ccn(C)n3)nn2Cc2ccsc2)c(OC)c1 c1(C(N2CCCCC(NC(C3OCC(C)(C)C3)=O)C2)=O)ncc2ccccn12 C1(C(=O)NCC(C)(C)NC(C2CC(C)CC(C)C2)=O)Cc2cc(F)ccc2O1 Cc1cccn2cc(C(N3CC4CCCC(C3)N4C(=O)C3=CCCC3C)=O)cc12 Cc1cc(C(=O)NCC2CCC(NC(C3Cc4nccn4C3)=O)C2)cc(N)c1O c1(C(=O)NCC23CC2CN(C(c2cnns2)=O)C3)cnc2sccn12 C1(C)(CNC(c2n(CCC)nc(C)c2)=O)CCCN(C(C23CC(C)C2C3)=O)C1 c1(C(N(CCCNC(=O)C=Cc2ccoc2)CC)=O)ncc(C(F)(F)F)cc1Cl CCCC(C)(C)CN=c1[nH]c(=NC2CCCCC2OC)[nH]c2c1SCC2 O=C1CC(CC(=O)N(C2CCCN(C(C3(F)CCCCC3)=O)C2)CCF)CCCN1 c1(N)cn(C)nc1SC.C1(CN(C(=O)NCC(c2cnc[nH]2)C)C)CCCC1 c1(C(=O)OC)nc(CNC(=O)N(CC(=O)NC(C)(C)C)C)cs1.N(C)C1CC1 Nc1cc(C(=O)NC(CNC(=O)CC2(N3CCCC3)CC2)C2CC2)cc(F)c1O C1(=CC(=O)NCC(C)(C2CCC2)NC(C2CCCSC2)=O)CCCCCC1(F)F c1(NCC(C2CCC2)OC)nccc(=NCC2CCC=CCC2)[nH]1 Nc1cncc(C(=O)NCC2(F)CC(NC(C3CCS(=O)(=O)N3)=O)C2)c1 c1(C(=O)NC2CCCN(C(C)C)C2)cc(F)cc2c(Br)ccnc12 c1(C(N2CC(C)CC(NC(C(C(CC)C)O)=O)C2)=O)ccc2ccoc2c1 c1(C(=O)NCC2(C(=O)NC)CCCO2)cc(CN2CCCC2CC(=O)OC)on1 N(C(=NCc1ccc(Cl)nc1)NCC(F)(F)CO)CC1C(C)C1 C1(CNC(CC(C)O)=O)CCCCC1C(=O)NCCNC(C1CCCC1)=O n1(CC)cc(C(N2CC(C)(NC(=O)C(O)CC3CC3)C2)=O)c(C(C)(C)C)n1 N1(C(C2CCN(S(C)(=O)=O)C2)=O)CCN(Cc2ccccc2)C(C)(C)C1 C=C(C)CCCC(=O)N1CC(N(C(=O)C2=CCCSC2)C)C(O)C1 N1(C(=O)Cc2csnn2)CCC2C(CCCN2C(c2c(F)ccc(F)c2O)=O)C1 C(CCC(=O)NC(C1CCN(C(=O)Cc2cnn(C)c2)C1)(C)C)NS(C)(=O)=O C1(NC(C(C2CCN(C(c3csnn3)=O)CC2)C)=O)CC2CC1CC21CC1 c1(CC(=O)N(CCOCCN(C(=O)Cn2nnc(=N)[nH]2)C)C)ccsc1Br c1(C(=O)OC(=O)OCC23OCC(COC)(C2)C3)c(C2CC2)nc2sccn12 C(=O)(C(C)(C)C(C)(C)O)NCC1C(NC(c2cn(CC)nc2C)=O)CC1 CC(C)C(C(C)NC(=O)C=Cc1ccccn1)NC(c1ncncc1Cl)=O N(C1CC(O)c2ccccc21)C(C(N1Cc2c(ccc(C(N)=O)c2)C1)=O)=O CC1(C)CC(CNC(=O)C(C2CCCCC2)NC(=O)COC2(C)CCCC2)CO1 Cc1cncc(C(=O)NC(Cc2cn[nH]c2)C(=O)NCC(CO)N(C)C)c1 CCC(CC)C(C)C(=O)N(C)CC1COCCN1C(c1ccc(S(C)(=O)=O)o1)=O C(=O)(CCCCCF)NCC1CN(C(c2cccc(OC(C)C)c2)=O)C(C)C1 CC1(C)COC(CC(=O)NCCCN(C2CCCC2)C(=O)C=Cc2cncs2)C1 c1(-c2cc(OC)c(Br)cc2)n[nH]c2c1CN(C(=O)C(C)n1cncn1)CC2 N(C(=NCCC=C(C)C)NCC(F)C1CCC1)CC1(OCC)CCCOC1 C(=O)(CCCCCn1cc(C2CCN(C)C2)nn1)NCC(=O)OCC c1(C(=O)NC(CC=C)CNC(C2(C)CCCC2)=O)ccc(C)c(S(N)(=O)=O)c1 C(=O)(CCP(C)(C)=O)NCc1cccc(CN(C(CCC=C)=O)C)c1 N1(C(c2c(C)cc(F)cn2)=O)CC2CCC1C(CNC(C1CCCC(=O)C1)=O)C2 n1(CC)nc(C(=O)NCC(C)(C)NC(C23CCC(C2)C3)=O)c(Cl)c1Br CC1(C)CCCC(NC(N2CCOCC2c2ncno2)=O)C1 C1(CNC(C=CC=CCC)=O)C(CC)CCN1C(C1OCCC1(C)C)=O N1(C(C2N(C(C3C=CCS3)=O)CCC(CC)C2)=O)CCc2nc(C)[nH]c2C1 C1(Nc2ncc(C(=O)OCC)cn2)CC2CCC(C1)N2C(=O)CC1CC(SC)C1 C12(NC(=O)CCF)CCOCC1CN(C(c1noc3ccc(Cl)cc13)=O)C2 CCC(C)CC(=O)N1CC(CN(C(=O)C(c2ccc(SC)cc2)(C)C)C)C1 N1(C(C=C(CC)C)=O)CCC(CCOC)(NC(=O)C(C)C)C1 Cc1cc(C)n(CCC(=O)NC2CC(CNC(c3ncc(C)cn3)=O)C2(C)C)n1 C1(CC(=O)NC2C(OC(C)(C)C)CC2)CCN(C(C2(c3ccno3)CC2)=O)C1 C12CN(CCC1CO)C2=O.n1(CC)nnc(C)c1C(=O)N.n1(C2CC2)ccc(CO)n1 C1(C(=O)NCC2(F)CCN(C(c3c(C)nn(C)c3Cl)=O)C2)CCc2cncn2C1 C12N(CCC1(C)C)C2=O.c1(NC(=O)NC(COCC)C)cccc(C)c1 N1(C(C=CC)=O)CCC2CCC(NC(c3ccc(F)cc3[N+](=O)[O-])=O)C1C2 n1(CCC(=O)NCC2(O)CC(NC(C(CCC)C)=O)C2)cc([N+](=O)[O-])cn1 C=CC(CC)CC(=O)NCC1(N(C2CC2)C(C)=O)CCCC1 c1(C(=O)NC(C(C(C)C)C)CNC(C23CC(CO2)C3)=O)ccnc2c1CCC2 N1(C(CC=C)=O)CCC(C2(O)CCN(C(c3cc(Br)ccc3N)=O)C2)CC1 O=C(N1CC2OC(=O)OC2CO1)NCc1ccc(Br)c(F)c1F c1(SC(C(=O)NCC(CC)NC(=O)CSc2ccccc2)C)nncn1C1CC1 C1(NC(c2ccc(COC)[nH]2)=O)CCC(NC(C2(S(N)(=O)=O)CC2)=O)CC1 c1(CNCc2cn(CC(=O)NC(C3CCCCC3)(CC)C)nn2)cccc(C)c1 C1(NC(C(COC)OC)=O)CCCCN(C(C2CCC(C3CC3)C2)=O)C1 C1(C(=O)NCCn2cc(CNC(C(C)OCC=C)=O)nn2)CCN(C)C1CC C(=O)(NNc1cc(C#N)ccc1Br)NCC1N(C(COC)=O)CCC1 CON1CC(C(=O)NC(C)(CNC(c2cn(C)nn2)=O)C2CC2)CC1=O c1(C(=O)NCCN2CC(C)OCC2C)ccc(S(C)(=N)=O)cc1 C(C)(N=c1[nH]c2c(c(=NCc3cscc3Cl)[nH]1)CCCCC2)c1nc(CC)[nH]n1 C1(C(N2C(CC(=O)OC)CC2)=O)C(C2CC2)CCN1C(c1ccc(OC)s1)=O c1(C(=O)NCCN2CCN(C(Cc3c(C)ccs3)=O)CC2)ccccc1S(C)=O Cn1ccc2[nH]c(C(=O)NCCC3(CNC(C4CC(C(F)F)C4)=O)CC3)cc12 c1(CC(=O)NCCCNC(=O)C=CC(F)(F)F)cccnc1S.C1COCCS1 C1(NC(C2C(C)(C)COCC2)=O)CCC2(CC1)CN(C(c1cnc[nH]1)=O)CCO2 c1(CNC(c2cc(C)nn2C)c2n(CCOC)nnn2)cnc2ncccn12 C(=O)(C1=NNC(=O)CC1)N(C)CCN(c1cccs1)C(=O)C(c1ccccc1)=O C1(C(N2CC3(CN(C(C=CCC)=O)C3)C2)=O)CCc2ccc(F)cc2O1 c1(C(N2CCC3(NC(C(=O)NCC)=O)C(CC2)C3)=O)sc2cccnc2c1N CC1CCN(C(C2CCC2)=O)CC1N(C(=O)COc1ccc(Br)cc1)C n1(CC)nc(-c2cncc(F)c2)nc1CCCOC(=O)NCCc1ccccc1 c1(NCC2CC(C)C2)ncoc1C1CN(C(C2CCCO2)=O)C1 C(C(=O)N1CCC(CNC2CCN(c3nccc(SC)n3)C2)CC1)(C(C)C)OC Cc1cccc(C)c1S(=O)(=O)Oc1ccc2oc(=O)n(C)c2c1 C1(C(C)C)CN(C(=O)COCP(C)(C)=O)CCN1C(=O)Cc1nccn1C n1(CC)nccc1C=CC(=O)NCCC(C)CCNC(C1CC1C(N)=O)=O CC1CN(C(C2(C)CC2C)=O)CC(C(=O)NCC2CC2Cl)O1 C1(O)(CC(=O)NCC(c2ccccc2)CNC(C2CC2F)=O)CCOC1 N1(C(C(CC)(C)CC)=O)CC2CCC1C(NC(c1ccc(C)c(C(C)=O)c1)=O)C2 CC1CC(C)(C(=O)NCC(=O)NCC(=O)NCC2CC23CCC3)C1 Cc1ncc2c(n1)CCCC2NC(c1coc([Si](C)(C)C)c1)=O N1(C(c2cncc(C)c2)=O)CC2(CCCC2)C1C(N1CCC2(CC(F)C2)C1)=O c1(NC(C2CN(C(C3CN(C(C)=O)C3)=O)CC(F)C2)=O)coc2ccccc12 c1(C(=O)NCC(C(C)C)NC(c2c(CSC)cccn2)=O)cc(Cl)c(F)cc1F N1(C(C)=O)CC2CCCC(C1)N2C(C1CN(C(C(C)(C)C)=O)CCS1(=O)=O)=O c1(C(N2CC(F)(CNC(c3cc(F)ccc3Cl)=O)C2)=O)cc(F)cc2nn[nH]c12 N1(C(C2C(=C)C2)=O)CCC2(CCCN2C(c2cccc(SCCC)c2)=O)C1 n1(CC)cnc2c(NCCN3CCC(C)C3)nc(N3CC4C(C3)C4(F)F)nc12 C1(C)(C(=O)NC(C)CNC(c2cc(C(F)F)[nH]n2)=O)CCNC1=O C1(OC)CC(CNC(c2cc(CO)c(C)o2)=O)N(C(=O)CC2CCCO2)C1 N1(C2CCCC(CC)C2)CC2CC(NC(=O)Cc3[nH]cnc3C)CC1C2 C1(C2N(C(C)=O)CCC2)CCN(C(c2c[nH]cc2C(C)C)=O)CC1 Cc1cc(N)cnc1C(=O)NC(CC1CC1)C(=O)N(C)CC1CC1(C)C C(CCCC(=O)NCc1ncoc1C1CN(C(=O)CCCC2CCCO2)C1)OC c1(C(N2CCCC(NC(C(C)(C)CC3CC3)=O)C2)=O)cn2cc(Cl)cnc2n1 CC1CN(C(=O)CCC2CCCCN2C(=O)C=CC(F)F)CC1O c1(C(N2CCC(COC)C2)=O)cc(N2CCCC2)nc(Cl)c1 c1(N2CCC(N3CC(C)(C)C3)C2)nccc(N2CCOC(CC(=O)N3CC3)C2)n1 c1(C(=O)NCCC2CCN(C(CCOCCN(C)C)=O)C2)ccc2ccoc2c1 C1(COC)CN(C(c2cc(C)on2)=O)CCN1C(c1cc(C)ccc1I)=O N1(CCCCn2cncn2)CCCC(n2nccn2)C1 c1(C(=O)NCC2OCC(CNC(C(CSC)C)=O)C2)ccc(C(C)(C)C)cn1 N1(C(C(=O)N(C(c2ccc(C)s2)C2CCC2)CC)=O)CCNC(=O)C1C N1(C(c2ccn(C)c2)=O)CCCC(CCNC(c2c[nH]c(=O)cn2)=O)CC1 CC1COCCC1N(C(=O)CN(C(=O)CCc1cnoc1)C1CC1)C N1(C(c2cnc(CC)s2)=O)C(CNC(C23CCC(C)C2C3)=O)CC2CCCC12 C1(CNC(Cc2nnc(C)s2)=O)CN(C(c2sc(Cl)cc2Cl)=O)CCC1C Fc1cc(C23CCCC2C3)c2nn[nH]c2c1 c1(C(=O)NCC2CCCCN(C(=O)C(F)CC3CCC3)C2)cccc([N+](=O)[O-])c1 Cc1noc(Cl)c1CC(=O)NCC12CC1CN(C(=O)C(=O)N(C)C)C2 c1(CC(=O)NC2CN(C(c3cc(C)n(C)c3C)=O)CC2O)cccc([N+](=O)[O-])c1 C(CNC(=O)C(C)(C)CF)(C(C)(C)C)NC(CCC(=O)OC)=O C(=O)(CC(CC)C(C)C)NCC(CC)N(C)C(c1c(C)nn(C)c1C)=O C=CCCCC(C)N=c1[nH]c(N(C)Cc2cccc(C(F)F)c2)nc2ccsc12 C(C(COC)CC(=O)N(C1CCN(C(c2cc(C)n(C)c2)=O)CC1)CCO)OC C(=O)(C(CC)C(F)(F)F)OC.C1(CCC)C(=O)OC(CC=C)CC(=O)N1 c1(C(N(C2CC(NC(c3c(C)c(C4CC4)on3)=O)C2)C)=O)cccc2c1COC2 CC1CC(=O)CCC1C(=O)NCC1(NC(c2cncnc2)=O)CCOCC1 C1(CNC(c2cn(CC=C)nn2)=O)CCCC(NC(c2cnnn2C=C)=O)C1 C1(C2(O)CN(C(C3CC(Cl)(Cl)C3)=O)C2)(CNC(=O)Cc2ccc(Cl)cn2)CC1 C(=O)(C(C)C(C)C)NCCOC.CCCCCN(C(=O)CCOCCS)C c1(CNc2cncc(C(N)=O)c2)ccc(-c2cccc3ncnn23)c2cc[nH]c12 N1(C(C)=O)CCC2(CC1)OC1(C)CC2(NC(=O)CCc2ccc(C)c(C)c2)C1 C1(C(N2CC(NC(c3cc(C(C)=O)oc3)=O)C(F)C2)=O)CC2C(C1)C2(C)C N1(C(c2c[nH]c(=NC)s2)=O)CCC(O)(CNC(c2ccnnc2S)=O)CC1 c1(C(=O)NC(C2CCN(C(C(CC)OCC)=O)CC2)C)ccc([N+](=O)[O-])c(N)n1 c1(CCNC(C2C(=C)C2)=O)ccc(CNC(c2sccc2OC)=O)cc1 N1(C(C(=O)N)c2ccco2)CCCC(CCF)C1.C1(C(CCCF)=O)CCCO1 N1(C(C=CC(C)C)=O)CCC2C(C(=O)NCC34CCCC3OCC4)C2C1 C1(CNC(CCCOCCNS(CCOCC)(=O)=O)=O)CCn2ccnc2C1 N1(C(C2=C(C)CCCC2)=O)CCC(NC(=O)Cc2c[nH]ccc2=O)C2(CCC2)C1 C12(C(=O)NCC3N(C(C(C)NC(N)=O)=O)C4CCC3C4)CCC(CC1)C(C)O2 C1(NC(c2nnc(C(C)C)s2)=O)C(C)CCN(C(C2CCC(=O)N(C)C2)=O)C1C c1(SC)nc(C)cc(=NC(C)C2CN(C(C3(OC)CCC3)=O)CCO2)[nH]1 C1(N(C(CCCc2scc(C)n2)=O)C)CN(C(C2OCCC2C)=O)CC12CC2 c1(OC)cc(C(=O)NCC(C2CCOC2)NC(c2cnn(CCF)c2)=O)sn1 c1(NC(C2C(NC(c3ccc(F)nc3)=O)C2)=O)ccnc(Cl)c1 c1(C(N(CCCC(=O)NC(CO)C2(C)CC2)C)=O)cccc2c[nH]nc12 CCC(C)(C#N)C(=O)NCC(=O)NCC(=O)NCC1CCOC(C)C1 c1(NC(C2CC2CNC(COCCCOC)=O)=O)[nH]c(=N)ccc1C c1(C(=O)NCC2N(C(CC(CC)C)=O)CC(O)C2O)cnc2c(ccn2C)c1 O=C(C1=CS(=O)CCC1)NC1(CO)CCCN(C(c2cccn3ncnc23)=O)C1 c1(C(N(CCNC(C(C(C)C)OC)=O)C)=O)cc2c(F)cc(F)cc2[nH]1 Cc1oc(CO)cc1C(N1CCCCC1C(=O)N(CC(C)CO)C)=O N1(C(c2n[nH]c(=N)[nH]2)=O)C2CC=C(C(=O)NC(CO)CCF)C1CC2 C(CC(O)C(=O)NCc1ncccc1CNC(=O)CCn1cccn1)SC N1(C(c2cc(CC)on2)=O)CCC(CNC(=O)C(C)Cc2ccccc2)C12CC2 C1(O)(CNC(c2cn(CC=C)nn2)=O)CCCN(C(C2CCC3(CC2)CC3)=O)C1 C(=O)(CCC1=CCc2ccccc21)NC1CC(N(C(C(CCC)C#N)=O)C)C1 N1(C(Cc2cnc(C)s2)=O)CCN(C(=O)COCC(C)C)CC1c1cccnc1 C(=O)(C(C)C(F)(F)F)NC1C=CC(CC(=O)NC2(c3nc(C)on3)CC2)C1 C1(CNC(C(C(=O)OCC)F)=O)CCN(C(c2cc(Cl)n[nH]2)=O)CCC1(F)F C(=O)(CCN(OC)C(=O)C(C)C1CCN(C(=O)CCNC(C)=O)C1)OC c1(C(C)C)cnc(O)c(C(=O)NCCCN(C(=O)C(C)(C)COCC(F)F)C)c1 N1(C(C(CC)NC(C)=O)=O)CC2=C(C1)CN(C(C1CCCCN1N=O)=O)C2 N1(C(C=CC=CCOC)=O)CC(NC(=O)COc2cccc(OC)c2)CCC1C N1(C(C(C)Oc2cccc(F)c2)=O)CC(n2cc(C3CCCOC3)nn2)C(C)C1 C1(C(=O)NCc2cnc(Cl)s2)COCCC12CN(C(c1cccnn1)=O)C2 N1(C(C2(OC(C)=O)CC2)=O)CCCC(C)C1CNC(c1ccn(C2CC2)c1C)=O Cc1ccc(C(=O)NC(CNC(c2cc[n+]([O-])cc2)=O)C(C)C(C)C)c(=O)n1C Cc1ccc(Cl)c(OCC(=O)NC2CC3C2CCN3C(c2ccnc(C)c2)=O)c1 C1(CCOC)CN(C(C2CNC(=O)O2)=O)CCN1C(=O)COCCSC C1(NC(C(c2c(F)cccc2F)C)=O)CC(F)CN(C(=O)Nc2cnn(C)c2)C1 Cc1cc(OC(C)C)ncc1-c1cnn(NC(c2c(Br)cnn2C(C)C)=O)c1 N1(C(C(F)OC)=O)CCN(C(c2cn(-c3cccnc3)nn2)C)CC1 Cc1nc(N2CCCC(NC(C3CN(CC(F)(F)F)C3)=O)CC2)[nH]c(=N)n1 C(=O)(CCC(N)=O)N(C1CCN(C(=O)C(=Cc2ccncc2)C)CC1)CC c1(CNS(=O)(=O)CCC2CCCN2)c[nH]c(=O)cn1 N1(C(CCSC)=O)CCN(C(=O)CC2CCC(C(N)=O)O2)CC1c1nccn1C c1(C(=O)NCC(CN(C(c2ccc(C(C)=O)o2)=O)C)O)cc(=O)cc[nH]1 C(=O)(CC(C)C(F)(F)C(F)(F)F)N1CCC(NC(CC(CCCC)O)=O)CC1 N1(C(C)C)CC(C(=O)N(CCC(C)NC(=O)Cc2cccn2C)C)CC1=O C1(C(=O)NCCCCCNC(C2CCC(F)CC2)=O)CC2CC1CC2O C1(C(N2C(CNC(c3cc(Cl)ccn3)=O)CCCC2)=O)CCCC2CCCCC12 c1(CC)cc(C(N2CC3CC3(CNC(c3ncccc3C(F)F)=O)C2)=O)ccn1 CC1OCCC1(C)C(=O)NCC1(C(=O)NCC(c2ccccc2)C)CCC1 CC1CC(NC(C2(C)CC2)=O)CCN1C(c1csc(C(C)(F)F)n1)=O N1(C(c2nnn(COCC)c2N)=O)CCCN(C(C2CC2(C)CC)=O)CCC1 N1(C(c2ccc(C)n2C)=O)CCC(CNC(C2CCCC3CCCC23)=O)C1(C)C c1(C(=O)NC(C2CCN(C(C=CC)=O)C2)C)cc(Cl)cc(Cl)c1OC C1(C(N(CCNC(CCc2ccc(C)cc2)=O)C)=O)CC(c2ccncc2)=NO1 CCC(CC(=O)NCC(CC)N(C)C(C1CC(N(C)C)C1)=O)C1CCC1 Cc1cc(=NC(=O)COCCNC(=O)Cn2cc(C#N)cn2)[nH]n1C C(C(=O)NC1CCC(NC(c2occc2-c2cnn(C)c2)=O)C1)(C(C)C)OC C(C)(N=c1[nH]c(=NC2CC=CC2)[nH]c2c1CSC2)c1c(C)cc(Br)cn1 N1(C(C=CC)=O)CCN(C(=O)CC(F)(F)F)CC1CS(C)(=O)=O c1(C(=O)OCc2cccc(O)c2)cc2c(O)cccc2s1 N1(C(C(F)=C(C)C)=O)CC(C)OC2(CCN(C(c3cc(O)cc(Cl)c3)=O)CC2)C1 C(CCCC(=O)NCCc1ocnc1CNC(=O)C(C1CC1)C1CC1)OC N1(C(N)=O)CCCC(C2CCCCN2C(c2cn(-c3ccccc3)nn2)=O)C1 c1(C(=O)NCCCCNC(c2nc(COCC)sc2)=O)cnn2cccc(C)c12 c1(CC)[nH]nc(C(=O)NC(C2CC=CCC2)C(=O)NCC2(C)CCN(C)C2)c1C CCC(COC)(C(=O)OC(C)(C)C)NC(C1CCC(NC(=O)NC)CC1)=O C1(NC(c2cc(C)no2)=O)CCCN(C(=O)C(C)n2cccc2)C1C S(=O)(=O)(c1cc(F)c(F)cc1F)N1C2CN(C(c3cc(C)cc(C)c3)=O)CC21 c1(C(N(C2CC(NC(C3(C)SCCCS3)=O)C2)C)=O)ncc2[nH]ncc2n1 C=C(C)CC(C(=O)N1CC2CC2(NC(=O)C(N2CCCCC2=O)C)C1)OC C(=O)(C(O)CCCCC)NC(C(=O)N(CCCCCCC)C)C(C)COC C1(NC(COCCNC(c2cc(CC)ncn2)=O)=O)CC12CCCCCC2 CCCCCCC(=O)N1CCC(CF)(NC(c2cnc(COC)cn2)=O)C1 C1(C(=O)NCC(C2CCC2)NC(CC=C(C)C)=O)COC2(CCC2)CO1 Cc1cnn(C(C)C(N2CC(c3ccccc3)(NC(=O)CCC3CCC3)C2)=O)c1 O=C(CC1OCCc2sccc21)NC(CNC(c1c[nH]ccc1=N)=O)CO C1(CC(=O)NCC2CC(NC(C(c3ccccc3Cl)C)=O)C2)CCC(C)(C)O1 c1(C(C(=O)NC(CNC(C=CC)=O)(C)CC2CCC2)C)ccc(S(N)(=O)=O)cc1 C1(NC(C2CC3CC3C2)=O)CCCC12CN(C(c1csc(Cl)c1Cl)=O)C2 C1(NC(CCNC(C)=O)=O)CCCC(NC(c2cn(C(C)C)nc2Br)=O)CC1 C(=O)(C1CCCc2c[nH]nc21)N1C2C(NC(C(C)(C)N3CCCCC3)=O)C(C2)C1 C1(c2onc(C)n2)CCCN(C(=O)Nc2ccccc2C(C)C)C1 N1(C(c2ccccc2Br)=O)CCN2C(=O)[N+]([O-])(CC(F)(F)F)C2C1 CCC(CCCC(=O)NC(CO)CCC(C)C)NC(C1(CCOC)CCC1)=O C1(CC(NCP(C)(C)=O)=O)CCCCN(C(C)=O)CC1 c1(OC)cccc2c(C(=O)NC(C)(CNC(=O)C3=COCCC3)CO)c(C)[nH]c12 c1(C(=O)NCC2OCC(CNC(C3(OC)CCC3)=O)C2)n[nH]cc1[N+](=O)[O-] CCC(C)(C)C(=O)C(=O)N1CC2CC1CN(C(=O)COC1CCOC1)C2 C(=O)(C1=CC(F)C(N(c2cccc(F)c2)C(=O)OC(C)(C)C)C1)N(C)CCN(C)C c1(C(=O)NCCS)cc2cccnc2[nH]1.C1(C(=O)NCC)CCN(C(=O)C)CC1 C1(C(N2CC(C(C=C)CCC)(NC(=O)CCOC(C)C)C2)=O)CCC(NC)CC1 C1(CNC(Cc2c(C)noc2)=O)CC(C)N(C(c2cn(C(C)C)nc2C)=O)C1 N1(C(=O)Cc2noc(-c3cccs3)n2)CC2CCC1CN2CC1CCCCN1 c1(C(N2CCC(NC(C34CC(CC(F)F)(C3)C4)=O)C2)=O)ccc(C2CC2)nc1 C1(C(=O)NC(CC=C)CNC(=O)C(C)Cc2ccc(C)cc2)CCCCCC1 N1(C(CSCC(C)C)=O)CC2(C1)C(NC(C1CC(C(F)(F)F)C1)=O)CCS2(=O)=O c1(SCC)ccc(C(N2CCC(CCNC(C3CC3COC)=O)CC2)=O)cc1 C1(C(=O)NC2(CNC(C3CCO3)=O)CCOCC2)CC12CCSCC2 C1(C(N(CCOCCN(C(=O)C(F)(F)C2CC2)C)C)=O)CCCC(N(C)C)C1 CC1CCC(CC(=O)N(CCCN(C)C(c2cnn(C)n2)=O)C)O1 N1(C2CCN(C(c3cc[nH]n3)=O)C2)CCN(C(=O)C(F)CC2CCC2)CC1 C1(O)(C(N2CCC(C(C)O)C2)=O)CCN(CC=Cc2ccco2)CC1 N1(C(C(N2CCN(C)CC2)C)=O)CCC(C(F)(F)F)C(NC(C2(CF)CC2)=O)C1 c1(CC)ccc(C(=O)NCC2CC(C)N(C(c3onc(CC)c3C)=O)C2)cc1 C=CC(C)CC(=O)N1CCOC(CCCNC(c2ccc(CC)[nH]2)=O)C1 c1(NC2CC3CN(C(Cc4cc(COC)on4)=O)CC32)ccc2nnnn2n1 C=C(C)CC(C)C(=O)NCCCC(CCC)NC(c1csc(C(C)(C)C)n1)=O c1(NC(=O)NCC2N(C(CNC(CCC)=O)=O)CC2)ccsc1-n1cnnn1 c1(C(=O)NCC(C)N(C(=O)CC2CSCCS2)CC)cnc(C)nc1C1CC1 C(N=c1cc(C2(OC)CCC2)nc[nH]1)c1c(CSC(C(CC)C(C)O)=O)cccc1 n1(CC)ncc(C(=O)NCC2C(C)CCN2C(c2ccc(C(C)=O)cn2)=O)c1C c1(C(=O)NC(CN(C(C2(OC)CCOC2)=O)CC)C)cc(C)c(O)nn1 N1(C(C(Br)=C(C)C)=O)CCC2(CCC2CNC(=O)CC2CC2C2CC2)CC1 c1(OCC=C)ccccc1NC(c1nnnn1CCCSC)CC1(C)CCCO1 CC1CN(C(=O)CC2CCC(C)(C)CO2)CCC1NC(=O)COc1cnc(Cl)cn1 c1(N2CCC(NC(CCCC)=O)CC2)nn(C)cc1[N+](=O)[O-] c1(CC(=O)NCC(CNC(C(C2CC2)SC)=O)C)ccc(C(N)=O)nc1 c1(NC(=O)C(=O)NCc2ccco2)cncc(C(F)(F)CF)c1 N1(C(c2cnc(C)[nH]2)=O)CCC(F)(F)C(CNC(=O)CN2CCCNC2=O)C1 C1(NC(C(C)=CC)=O)CCC(C)(CNC(=O)C(C)NC(=O)COC)CC1 n1(CC)ncc(Cl)c1C(=O)NC(CNC(c1cnc(C(N)=O)cn1)=O)C1CC1 CCCC(C)CCCC(=O)N1CC(O)(CCNC(=O)C(C)SC)C1 Cc1nc(C(=O)NCC2(F)CCN(C(C3(CO)CCCO3)=O)C2)cc(O)n1 N=c1[nH]c(=NCC2CCSC2)[nH]c(=NC2CCN(c3cccs3)C(=O)C2)[nH]1 N1(C(C2(OCC)CCCOC2)=O)C2CCC1CC(NC(c1nc(C)c(C)[nH]1)=O)C2 c1(OC)ccc2c(c1)cc(C(=O)OCC1CC3(CCC3)C1)n2C1CC1 N(C(=NCCN1CCC(C)(C)CC1)NCC1CCCO1)CC1(OC)CCCSC1 C1(NC(C(C)(C)OC)=O)CCCN(C(=O)C=C2CCCC2)C1 C(=O)(C1NCCc2ccccc21)NC1CC(=O)CN1c1ccc([N+](=O)[O-])cc1 C1(C(=O)NCCN(CCC)C(C)C)C2CCC1(c1ccn(C)n1)C2 Cc1cc2c[nH]nc2cc1C(=O)NC1(C)CCN(C(c2ccc(C#N)cn2)=O)C1 N1(C(c2n(CC)nnc2)C(=O)NCCC2CC2)C(CO)CC2CCCCC12 CC1CN(C(=O)C(F)=C2CCCC2)CC1NC(c1csc(-c2ccoc2)n1)=O N1(C(CCC(=O)NCC)=O)CC(NC(=O)C(O)C(C)(C)CC)CC12CCCC2 C1(C(=O)NC2CC(CNC(=O)Cc3cccc(Cl)c3)CC2O)OC2CCC1CC2 N1(C(C(C)O)=O)CC(C)(NC(c2ccoc2I)=O)C1 C(C)(N=c1[nH]c(N2CCCNC(=O)C2)nc2ccsc12)c1cncc(OC)c1 Cc1ncccc1NC(c1nnnn1CC(F)F)C1CC=CCC1 N1(C(c2n(C=C)nnc2)=O)CCC2(CC1)CC2CNC(=O)CCCCOC c1(C(N(C(CC)CNC(c2cn(CCOC)nn2)=O)C)=O)cnc2ccccn12 C1(CNC(CC(c2ccccc2Cl)C)=O)CCN(C(=O)C=CCN(C)C)CC1C C1(C(=O)NCC(C)(C)c2ccsc2)CC12CCC(F)(F)CC2 N1(C(C(CCC)OC)=O)CCCN(C(=O)COc2cccnc2)CC1CO C(N=c1[nH]c(C)cc(OC)c1[N+](=O)[O-])C1OCC(NC(C(CCOC)C)=O)C1 C(CCF)(C(=O)NCC1CC(C)(C)CO1)NC(C(C)OCCOCC)=O C1(CC)CCCC1(C)C(N1CCN(CCCNC(=O)C2CC2)CC1)=O N1(C(C2CC(C)C2)=O)CCC(C)C(NC(C2(C)CCN(C)CC2)=O)C1 CP(C)(=O)CC(=O)NCCS(=O)(=O)Cc1cn(-c2ccc(Cl)cc2)nn1 C1(CNC(CC(C)C)=O)(CNC(c2cncc(Cl)c2)=O)CC12CCC2 C(=O)(CCCC(=O)c1cnn[nH]1)NC1CC(NC(C(C)O)=O)C(O)C1 O=C(CCC1CC1(F)F)NCCOCCNC(=O)COCC(=O)NCCF C(C(C)(O)CC(=O)N1CCCCC1CNC(=O)CCCc1cc[nH]c(=N)c1)OC C#Cc1cccc(C(=O)NCCCOCCNC(C2(CC)CCOC2)=O)c1F c1(OC)c(Br)ccc(F)c1S(=O)(=O)NC(c1ccc([N+](=O)[O-])cc1)C C1(NC(c2nc(CC)sc2)=O)CN(C(=O)COCC2CCCC2)C2CC12 Cc1nc2c(C(N3CCC(NC(=O)COCCN(C)C)C3)=O)cccc2o1 C12(C(=O)NCCC(C#C)C)C(NC(C3CC4(CC4)C3)=O)C3CC1C2C3 C(CCCCCC(=O)NCCC1CC(C)(C)CO1)NC(c1c(OC)ccs1)=O C(Cc1ccco1)(C(=O)N1CCC1CF)NC(c1coc(Cl)c1)=O c1(C(C2C(NC)CN(C(C(CC)C(C)C)=O)C2)=O)cc(S(C)(=O)=O)ccc1OC N1(C(c2c(CC)cno2)=O)CCCC(F)(C(=O)N(C2CC2)CC2CC2)C1 c1(C(N2C(CNC(C(C)C(F)F)=O)CCC2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 c1(C(=O)NCC(CC=C)NC(c2cncc(SCC)c2)=O)cnc(Cl)cc1N CC1=C(C(=O)N2CCC(NC(C3CCn4ncnc4C3)=O)CC2)SCCO1 N1(C(=O)SCC(N2CC(NC(C3CCCCC3)=O)C(F)CC2)=O)CCCCS1(=O)=O C1(CNC(C(C)OC2CCCC2)=O)CCCC2(CN(C(c3csc(Cl)n3)=O)C2)O1 c1(C(=O)NC2(CC(=O)N(CCOC)C)CCC2)ccc(C)cc1O C=CC(CC)CC(=O)N1CCCC(NC(=O)C(=O)Nc2ccc(C)cc2)C1CC C1(CCC(=O)NC(C(c2ccccc2)NC(C2CC(OC)C2)=O)C)CCOCC1 CCCN=C(NCc1ccc(CC(=O)OC)cc1)NCc1ncn(C)n1 C1(N(C(=O)CCc2ccc(O)cc2)C)CN(C(C2CCCC(=O)N2)=O)CC12CC2 N#Cc1cc(S(=O)(=O)N2CCCC(C(=O)Nc3ccsc3)C2)ccc1Br CC(C)(C)C(CC(=O)N1CC(O)C(F)C1)NC(C1CCCC(CF)C1)=O Cc1ccc(C(=O)NC2CC3CCC2N3C(=O)CC(O)C2CCCC2)nc1C Cc1cccc(C)c1C(N1CC(NC(=O)CCc2ncco2)CC(F)C1)=O c1(C(=O)NC2CN(C(C(N)=O)=O)CC2c2ccccc2)ccnc2ccncc12 C12CC3CN(CC3C1)C(=O)C(CCC#C)NC(=O)N2.C(C)(C)(C)NC(=O)C#CC c1(C(=O)NCC2CCC(NC(c3c(CC)nn[nH]3)=O)C2)cnc(C2CC2)nc1O c1(C(N2CCN(C(c3c(CC)c[nH]n3)=O)CC(O)C2)=O)ccn2c(C)ncc2c1 Cc1cc(C)c(NC(C2(NC(=O)CCCn3ccnc3)CCC2)=O)cn1 O=C(CC1OCc2ncccc21)NCCSCC(O)CO c1(C(=O)NCC2CN(C(c3c(C)nc(CO)s3)=O)CC2C)csc([N+](=O)[O-])c1 CCC(C#N)C(=O)N1CCC1C(=O)NCCC(=O)N1CCCC1 C1(C(N2CC(CC(C)(C)C)C2)=O)CCN(C(c2ccc(F)s2)=O)CC1O c1(C(=O)NCCN(C(C2(C3CCOCC3)CC2)=O)CC)cccc2ncccc12 C(C(O)CC(=O)NCc1nocc1C(=O)N(C1CC=CC1)C)N(C)C Cc1cnc(N2CCCCC2CNC(=O)CCc2nncs2)nc1C N1(C(CC(C(=C)C)NC(=O)OC(C)(C)C)=O)CC(C)(C)OCC1CC#N.OCC c1(C(N2CCCC(C(N(C(C(=O)OC)C)C)=O)CC2)=O)ccc2cncn2c1 c1(C(N2C3CC(NC(C4N(C(C)=O)CSC4)=O)(C3)C2)=O)c(F)ccc(F)c1F N1(C(C(C=CC)O)=O)CCC(F)(C(N2CCN(C(=O)NC)CC2)=O)C1 c1(C(=O)OC)[nH]c(=NC2CC23CC(NC(=O)C(C2CCCO2)C2CC2)C3)sc1C c1(OCC)ccc(C(=O)N(CCCNC(C2COC(C)C2)=O)CC)cn1 C1(C2CCN(C(c3cnc(S)n3C)=O)C2)(NC(CC=CCC)=O)CC1 C1(=O)CC(C(F)(F)F)N1C.CC(C)C#CC(=O)NC1CCN(C(=O)C=CCF)C1 N1(c2nc(OC)c(Cl)cn2)CCC2(CC1)CC(NC(=O)CS(C)(=O)=O)CO2 C(=O)(C1CCCc2n[nH]cc21)N(CCNC(c1c(C)cc(CO)o1)=O)C1CC1 C1(C(N2CC(NC(c3c(C)con3)=O)CC3(C2)CC3)=O)Cc2cc(Cl)ccc2O1 C1(NC(c2ccccc2O)=O)CCC(C(=O)NC2CCN(C3CC3)C2=O)CC1 Cc1csc2c(C(=O)NCC3CCN3C(=O)CC3(O)CCCCCC3)cccc12 C1(NC(COCCCC(C)C)=O)CN(C(C2CC(S(C)(=O)=O)C2)=O)CCC1C C1(C(C(=O)NCC(CC)NC(=O)C=CC2CCC2)NC(N)=O)CCCCC1 C1(NC(c2ccccc2)=O)CCC(S)CC1.C1(CCC)CCCN1C(=O)C=CCO CC(C)(C(=O)NCC1(F)CC(NC(c2ccnn2C(F)F)=O)C1)c1cccs1 N1(C(C(=O)NCc2ccn(C)n2)=O)CCC(N)CC1 N#Cc1c[nH]cnc1=NC1CCC(NC(=O)CN2CCCCCCC2=O)CC1 C1(C)(CC)CCC(NC(C23CCC(OC)C2C3)=O)CC1.C12CC(C1)NC(=O)C2 c1(C(=O)NCCCCC(C)NC(C2C(CC(C)C)C2)=O)cc2c[nH]cnc-2n1 C1(C(=O)NCC2CN(C(=O)C3=CCOC3)CC2O)CC2CCC(C1)S2(=O)=O c1(-c2nc(CC(CC)C)nn2C(C)CC2CC2)cc(C)ccc1Br C(C(C)(C)CN=[N+]=[N-])NC(C(C(C)OCC1CC1)NC(C1CC(OCC)C1)=O)=O c1(C(C(=O)OCCc2cccc(OC(F)F)c2)=O)cc2ccccc2s1 O=C(C1CCc2ccccc21)N1CCCCC1CC1CSc2ccccc2O1 c1(C(C(=O)OC)OC(C2CCCNC2C)=O)cccc(Br)c1C C=C(Cl)C(C)(C)C(=O)NCC1CCN(C(=O)C(C)Oc2cccc(C)c2)C(C)C1 C1(NC(C2C(C(C)(C)O)C2)=O)CCC(NC(c2cncc(C(F)(F)F)c2)=O)CC1 C(C(COC)C(=O)NCCCCCN(C)C(C1CCCOC1C)=O)OC c1(SCC(CC)OCC)ccc(Cc2cccc(Br)c2)c(OC)c1 C1(CN(C(C)=O)CC)CCCCN1C(=O)Cc1cnn(C)c1C N1(C(C2CN(C(COC(CC)(C)C)=O)CC2F)=O)CC(C)=CC(C)C1.C(C)(=O)O c1(OCCCC(=O)OC2CN(C3CCOCC3)C2=O)cccc2ccccc12 CCC(CN(C)C)CC(=O)NC1CCCCCC1C(=O)NOCC(F)(F)F C12CCC(CC1)NC(=O)CCC(=O)N2C.c1(OCC)nc(C(=O)OC)ns1 CCC(CC)CC(F)C(=O)OC1CC(N2CCNC2=O)C1 c1(C(=O)NC(C(CO)NC(C)=O)C)c[nH]cc(F)c1=O.c1(N)ccc(OC(F)F)nc1 C1(C(=O)NCC2(OC)CCC2)CC=CCC1NC(=O)COc1ccn(C)n1 C(C)(C(=O)N(CC(N1CCC(N2CCC2)C1)=O)CCO)(C(C)C)OC c1(C(=O)NC(c2ccsc2)C)ccc2c(c1)CCN(Cc1cccc(F)c1)C2 C(=O)(C(C)CC)ONC(c1sccc1)=O.CCC(C1CC1)N(C)CC1CC1 CCCC(CNC(C1CCN(C(=O)C=Cc2cc[nH]c2)C1)=O)OC C(=O)(C(O)(C(F)(F)F)c1ccccc1)NCC(C)NC(c1c(C(=O)OC)c[nH]n1)=O c1(OCC)cc(Cl)ccc1C(N1C2CCC1(CNC(C1CCC1C)=O)CC2)=O c1(OC)nsc(C(=O)NCCn2ccccc2=O)c1Br N1(C(CCCOC)=O)CC(CO)C2(CCN(C(c3csc(CO)n3)=O)CC2)C1 N1(C(C(C)(c2cccs2)N(C)C)=O)CCC(F)(CNC(=O)C#CC(C)(C)O)CC1 C1(C(NOCCCCC)=O)(NC(c2nnn(CC)c2C)=O)CCCC1C c1(C(c2nnnn2CCCF)NCCCC=CC)cnn(Cc2ccccc2)c1 C(=O)(C(C)(F)C(=O)OC)N(CC(=O)NCC1CNC(=O)O1)CCC Cc1csc(=O)n1CC(N1CCC(C)C1)=O C(=O)(C1=NOC2COCC12)N(CCC(=O)NC1C(COC)CCC1)C N1(C(C(C=C)O)=O)CCc2[nH]nc(CNC(c3nocc3Br)=O)c2C1 C1(C)(CSc2cc(C(=O)COC(CC=C)C)sc2)CCCNC1=O CCS(=O)(=O)CC(C)(C)CNC(c1ccc2c(n1)CCC2)=O CCC(CC(=O)N(Cc1ccccc1)CC1COC2(CCCCC2)C1)C(C)(C)C N1(C(C(C)NC(COC)=O)=O)CCC(CCNC(c2ncc(C(F)F)s2)=O)CC1 c1(CCNC(COC)=O)n[nH]cc1N(C(CO)C(C)C)C(=O)CC1CC(C#N)C1 N1(C(C(CCOCCO)NC(C(CC(C)C)C)=O)=O)CCc2ncsc2C1 c1(C(N2CCCC(NC(=O)Cc3ccns3)C(F)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 c1(NC(C2(F)CCC2)=O)ccc(C2CCN(Cc3ccnnc3)CC2)cc1 N1(C(C2C(C=C)CC2)=O)CC(CNC(c2coc(C)c2)=O)C(C)C1 CC1CC(NC(=O)C#CCNC(=O)COCCN(C)C)CS1 c1(C(C)C)cc(=NC(=O)C(F)(F)C2CCCN(Cc3ccccc3)C2)[nH]n1C c1(N2C(CC(N)=O)CC(C)C2)ccc(S(=O)(=O)N(c2ccccc2)C)cn1 CC1(C(=O)NCc2cn(Cc3cc(-c4cccnc4)no3)nn2)CCNC1=O CCCC(C)(C)CC(=O)NCC1CN(C)CCN1C(C1CCC2(CCC2)OC1)=O c1(C(=O)OCC)cccc(N(C(=O)Nc2ccc(C)cn2)CCN(C)C)c1 N1(C(C2CCCN2C(=O)CCn2cccc2)=O)CCCC(N(C)C)C1 c1(C(=O)NCC2CCCC(NC(=O)CSC(F)F)C2)ccc2nc[nH]c2c1 C1(C(N(C)CCC2CC2)=O)CSCCN1C(C1CC1C(C)(F)F)=O C1(C2CN(C(C(CC#C)C3CCCCC3)=O)C2)CC(C)(C)CN1C S(=O)(=O)(c1ccc(-c2cccc(C)c2F)s1)N(CC=C)C c1(C(=O)NCC(=O)CNC(C2(F)CN(C(C3CC3F)=O)C2)=O)cccnc1 c1(CNC(=O)CC2CCCCCN2)ccc(S(=O)(=O)N2CCOCC2)cc1 C(=O)(C1CCc2cccc(O)c21)N1CC(CNC(C=CCOC)=O)C(F)(F)CC1 CCCC(C)C(c1nnnn1CC)NCCCc1noc(C(C)(C)C)n1 C(=O)(C(F)(F)C(F)F)NCCC1CCC(NC(CCc2scc(C)n2)=O)C1 N1(C(C(C(C)NC(C(C)OC2CCCC2)=O)(C)C)=O)Cc2ccnn2CC1C CCC1=C(C(=O)N2CCN(C(=O)C(=Cc3ccncc3)C)C3CC23)CCCO1 C(CN=c1[nH]nc(C(F)(F)F)s1)=CCNC(C1=C(C)CCC1)=O c1(CC)ccc(C(=O)NC(C)(CNC(=O)C(C(C)C)NC(N)=O)C(C)C)c(C)n1 CCC(C)(C)CCCC(=O)NCC1CCN(C(c2cc(Cl)n[nH]c2=N)=O)CC1C CC(C)CC(C(=O)NC1CN(C(=O)C(C)(C)c2ccccc2)CC1C)C(N)=O c1(C(=O)NCCCCN(C(=O)C=CC(F)(F)F)C)ccc(C(C)(C)C)cc1N Cc1cccc(Br)c1C(=O)NC(CNC(c1ccc(Cl)s1)=O)C(C)C C1(CNC(c2ccn(C(C)(C)C)c2)=O)CC2(CC2)CN1C(=O)CCC(=O)C1CC1 C1(NC(C2CC(C(F)(F)F)(OC)C2)=O)CN(C(=O)CCC(F)(F)F)C(C)(CO)C1 Cc1c(C(=O)NCC23CCC2CN(C(c2ncn(C)n2)=O)C3)ccc(F)c1F c1(COCC(=O)NCCC2(NC(=O)CSC3CCCC3)CCC2)ccc(Cl)cc1 C1(CC)CN(C(=O)CC=CCNC(=O)C(C2CCOCC2)F)CCS1 C12(NC(C3CCN(C(C(C(CC)C)=O)=O)C3(C)C)=O)CC3CC(CC1C3)C2 C1(C(=O)NC2CCCC2NC(=O)C2=CCSC2)CCC(O)CC1 C(CCN=C(NCc1ccc(F)c(F)c1)N1CCC(C)(F)C1)SC c1(OC(C(=O)OC)C(=O)Nc2ccnc(OC)c2)ccc(Cl)cc1C C1(C(=O)NCC2(C3CC3)CC2)CC2(CC2)C1.C12(CC1)C(=O)N2 C1(NCCC(C)(C)Nc2ncnc(Cl)c2F)C2Cc3ccccc3C12 c1(C(N(C)CC2CCCN(C(C3C(C)C3C)=O)C2)=O)cn(CCO)c(=O)nc1O C(C(C)(CO)CO)N(C(=O)C(=O)Nc1nnc(C(C)(C)C)s1)C C(CC(C(=O)N1CC(CO)CC1CO)NC(=O)CC1(O)CCC1)N(C)C CC(C)CC(C)(CNc1ncccn1)NC(c1ccc(C(F)(F)F)[nH]1)=O Cc1cc(N)c(C(=O)NC2CC2NC(C2CC2(Cl)Cl)=O)c(F)c1 C1(NC(Cc2c(C)ccnc2)=O)CC2CCCC(C1)N2C(=O)C(C)C(O)C(C)C C(=O)(C1=NN(CCO)C(=O)CC1)NC(C1(O)CCN(C(=O)CCCN=[N+]=[N-])C1)C C1(NC(C(C2CCCOC2)OC)=O)CC2CC(C1)N(C(C1CCCN1C=O)=O)C2 N1(C(C2(CC=C)CCCN2C(=O)C(CC)=CC)=O)CCOCC(C)(O)C1 c1(C(=O)NCC2(CC(=O)N(CC(CC)O)C)CC2)cncc(NC)c1 C1(C)(CNC(CC(C)=C(C)C)=O)CCN(C(C2(C)CCCCO2)=O)CC1 Cc1cccc(C(C)NC(=O)C(O)CNC(C2(Cl)CC2)=O)n1 C1(C(=O)Nc2ccc(CN(CC)CC)cc2)(OC)CCC(F)(F)CC1 CON1CC(C(N2CC(C)(C(=O)NC3(CCO)CCCC3)C2)=O)CC1=O N(C(=NCCCCC(F)(F)F)NCC1C=CCC1)Cc1c(O)cccn1 c12ccc(cc1)CC(=O)NC2.c1(CC)cccnc1CNC(=O)C(C)(C)CO c1(OC)ccc(C)cc1C=CC(=O)NCC1(NC(=O)CC2SC(=N)NC2=O)CC1 C(C)(C(CO)NC(c1ccsc1SC)=O)NC(C1C(CCOC)C1)=O c1(C(N(C(C)CNC(c2cccnc2)=O)CC)=O)cnc(N(C)C)o1 c1(OCC(N2CCC(=CCNC(C3C(C)C3)=O)CC2)=O)cccc(F)c1 N1(C(C2(C3N(C(C4OCCC(C)C4)=O)CCC3)CC2)=O)CCC2(CCC2)CC1 C1(C(=O)NC2C(NC(c3c(C)nc(CO)o3)=O)CCC2)CCc2c(n[nH]c2C)C1 c1(SC)ccc(C(=O)NCC(C)NC(c2c(SC)ccs2)=O)o1 C1(C(N2CCCC(CNC(=O)COC(F)(F)F)C2)=O)(OCC)CCOCC1 C(=O)(C1(C)CCc2ccccc21)N1C(CNC(CN(C(C)=O)C)=O)C(C)(C)CCC1 N1(C(C2CC(CC)OCC2)=O)CCCC(O)(CNC(c2nc(C)oc2C)=O)CC1 N1(C(C(CC(=O)OC)C)=O)CCCc2cc(OC(C)(C)C)cc(Br)c21 c1(-c2cccc(NC(Cc3c(OC)cncc3)=O)n2)c[nH]c2ccc(CNC)cc12 C1(NC(c2nc(C(C)(F)F)sc2)=O)CC(F)CN(C(=O)COCc2ccccc2)C1 c1(CN2CC3C(C(=O)Nc4ccc(F)cc4O)(C3)C2)ccncc1[N+](=O)[O-] Cn1cc2c(n1)CC(C(=O)NC1COCC1CNC(=O)C(=O)NC1CC1)CC2 CCC(CCC(=O)N(CC(F)(F)COC)C)NC(c1cc(C)oc1C)=O c1(OC)ccc(CN2CC(F)(F)CC2C(=O)Nc2cncnc2Cl)c(Br)c1O C(=O)(C(O)(C(F)(F)F)C1CC1)NC(C(C)NC(c1c(C)n(C)cn1)=O)C N1(C(C(C)C)=O)CC2(NC(c3ccc(=O)n(CC(F)(F)F)n3)=O)CCC1C2 C(=O)(C1CCCn2ncnc21)N1CC(C(C)NC(C2CC3(C2)CC(O)C3)=O)C1 C1(CNC(=O)Cc2cncnc2)CC2(CCN(C(c3cnccc3Cl)=O)C2)CO1 c1(C(=O)NCCCN(C(c2ncoc2C2CC2)=O)CC)cnn2c1OCC(O)C2 c1(C(=O)NCC(C(C)(C)C)NC(C2OCC2(C)C)=O)n[nH]c2c1CS(=O)(=O)CC2 C1(C(=O)NC2C=C(C)CCC2)COCCN(C(=O)CCN(C)C(=O)C2CC2)C1 N1(C(C2(CC#C)CCCCO2)=O)CCN(C(=O)C(C)(O)C2CC2)CC1CO N(C1CCOc2c(Br)cccc21)C(=O)Nc1cc(SC)cc(NC(=O)OCC)c1 N1(C(C2C(NC(C3CC(=O)N3)=O)CC2)=O)CCc2ccccc21 O(P(=O)(COCc1cn(CC2CCCN2C(=O)C(N)=O)nn1)OC(C)C)C(C)C c1(CC)oc(C(=O)NCC2C3CC=CCC23)cc1C C1(NC(c2ccc(-c3nc[nH]n3)nc2)=O)(CO)CCN(C(c2ccc[nH]2)=O)C1 c1(C(=O)NCCC(C)N(C(=O)C(C)(C)O)C)ccc2c(c1)S(=O)(=O)NC=N2 CC(C)(C)C(O)C(=O)NCC1COCC1C(N)=O.C12(CCCCC1)C(=O)NC2 N1(C(C(c2ccn(C)n2)C)=O)CCCC(C(=O)N(CC(C)(O)C2CC2)C)C1 C(=O)(C#CC1(C)CC1)N(C1CC(NC(c2c(OCC)nccc2)=O)C1)C c1(C(=O)NCC(CCCC)NC(=O)C(O)CCSC)cc(N)ccc1SC CS(=O)(=O)C1(c2cn(C3CCC(C(=O)Nc4ccsc4)C3)nn2)CC1 c1(CCC(=O)NC2CNOCC2F)ccc(Cl)nc1 C1(CNC(C(CC)OC)=O)Cc2ccccc2CN1C(=O)COC1CCCOC1 c1(C(C)=O)cc(C(=O)NC2(CNC(C3(c4ccsc4)CC3)=O)CCOC2)oc1C N1(C(Cc2c(C)con2)=O)CCC(CNC(=O)C(C)C(C)C)C12CCC2 C=CC(COC)N=c1[nH]c(=NCCCCCCCCSC)[nH]c2ccc(Cl)cc12 c1(C(C)C)conc1C(=O)NC(CC1CCCC1)C(=O)NC(CC1CC1)CO C=CCCC(C)(C)CNC(=O)C=CC1CCCN1C(=O)C(O)C1CCCC1 c1(C(=O)NCCC(C)NC(C2ON=C(C)C2)=O)ccc2c(c1)nc(C)n2CCO C1(N2CCN(c3c(C)nccc3)CC2)CCCCN(C(C2CCC(C)C2)=O)C1 C12(C)CCN1C2=O.c1(CC)conc1CNC(=O)C(C)(C)OC(C)=O C1(NC(C(CCC#C)O)=O)CN(C(=O)C=Cc2ccc(F)cc2)CCC1(C)C c1(OCC(=O)NCC2CC(NC(=O)Cn3cnc(Br)c3)C2)ccc(F)cc1 C(=O)(C(C)(C)Cc1cnn[nH]1)NC1(CC=C)CN(C(=O)CSCC2CCCO2)C1 C1(CNC(c2c(C)csc2)=O)CC12CCN(C(c1scnc1C)=O)CC2 Cc1ccoc1C(=O)N(CC(=O)NCC(C)(C)C1CCCO1)C C1(NC(c2cccc(Cl)c2)C)CCC(C)(CN)CC1 c1(C(=O)NC(C2CCCCN2C(=O)C(C2CC2)C2CC2)C)ccc(C(F)F)cn1 C(=O)(C(O)C(F)(F)F)N(CC(CNC(c1n[nH]c(C)c1Br)=O)C)C C(CNC(c1cc(O)cc(O)n1)=O)(C(C)C(C)C)NC(c1ccc(C)nn1)=O N1(C(=O)Cc2ccc(Cl)nc2)CCN(C(C23CCCC2CC3)=O)CC12CC2 CC(CC(=O)N1CC(C(C)O)C1)C(C)(C)NC(C1CCCCCCC1)=O N1(C(CC(=C)C)=O)CCCCCC(NC(=O)Cc2nnc3n2CCOC3)C1 c1(C(=O)NC2CCCC(NC(C3(SCC)CC3)=O)C2)ccnc(Cl)c1OC C(=O)(C#CC1CCOC1)N1C(C(=O)NCc2cocn2)CC2(CC1)CC2 C(CCCCCNC(=O)CC)NC(c1c(C)nco1)=O.C(C)(C)(C)OC(C)=O C1(CC)CN(C(=O)C2CC2)CCC1NC(c1ccc(=O)n(-c2ccccc2)c1)=O c1(C(N2CC(C)(NC(c3c(OC)cccc3)=O)C2)=O)cc2cccnc2s1 N1(C(C(C)=O)=O)CCN(C2CCN(C(=O)CC(C)C3CCCO3)C2)CC1 c1(C(N2CC(NC(C=C)=O)C(C)C2)=O)nc(Cl)ccc1F CC1(C)CC(NC(=O)Cc2cnn(C(F)F)c2)CN1C(=O)CC12COCC(C1)C2 N1(C(c2cn(CCOC)nc2)=O)CCN(CC2C=CCC2)C(C)C1 N1(C(C(COC)N(C)C)=O)CCOCC(CNC(=O)CCc2cc(C)on2)C1 C1(NC(c2ccc(CC)s2)=O)CCN(C(c2ccc(N)cc2C)=O)C(C)C1 N1(C(CC=C)=O)CCC(CN(C(c2cc(C3CCC3)[nH]n2)=O)CC)C1 C1(CC)CCC(NC(=O)C(CCNC(=O)CCCN(C)C(C)=O)OC)CC1 C12(C(=O)NCCOCCCNC(c3c(C)[nH]cc3)=O)CC1COC2(C)C C(C)(C)(C(=O)N1CC(CCO)(NC(=O)C(C)CN(C)C)C1)OC N1(C(c2cn(CCC)nc2C)=O)CCN(C(=O)C(O)COC)C(C)C1 c1(C(=O)NCC2(Cn3cc(CC(=O)OC)nn3)CC2)c(Cl)cnn1C CN(Cc1ccc(C#N)cc1)N1CCOC(C2(N(C)C)CCC2)C1 c1(C(C)(C)O)ccc(C(=O)NCC(C)(O)CNC(=O)CNC=O)cc1 N1(C(CNC(C2CCCC2)=O)=O)CCC(CCNC(c2csc(C3CC3)n2)=O)C1 C1(C(=O)NNC(=O)c2ccccc2C2CCC2)CC(O)C12CCOCC2 N1(C(C(C)OCC)=O)CCOCCC1C(=O)Nc1ccc(C)cc1OC C1(NC(C(N(C(C(C)OCCCC)=O)C)C2CC2)=O)CNC(=O)C1(C)C C1(C(=O)NCCNC(C(C)C)=O)(CNC(c2cc(Cl)cs2)=O)CC2(CC2)C1 C(=O)(CC1=CCN(C(c2cnc(C3CC3)o2)=O)CC1)N(C)Cc1nc(C)[nH]n1 c1(OC)cc(CCNCC(Cc2ccccc2[N+](=O)[O-])CO)ccc1S(C)(=O)=O CC(C)(C(=O)NCC(C)(C)C#CC(=O)NC1CCC(CO)C1)C(F)(F)F c1(C(N2CC(C(C)(C)O)(CNC(CCc3nc(C)sc3)=O)C2)=O)nc(=O)n(C)[nH]1 C1(OC)CNCCC1C(=O)Nc1cnc(NCC(=O)N(C)C)n1C C(=O)(C1=CC2CCC1C2)N1CC(NC(c2ccc(C3CC3)[nH]2)=O)C1 c1(C(=O)NCC2N(CC(=O)NC3CCC4CC34)CCCC2)cccn2cncc12 CN1CCN(c2ncc(OCF)cn2)C(NC(C2CCCCC2)=O)C1 c1(C(=O)NCCN(C(CN2C(C)CCC2C)=O)C)cc(Cl)c(F)cc1F C1(C(N2C(C)(CC)CC2)=O)CN(C(C2COCC(C)O2)=O)CCC1O c1(C(=O)NC2CC(C)CN(Cc3ccoc3)C2)n[nH]c2ccc(C(F)(F)F)cc12 C(=O)(C1CCc2ccc(Cl)nc21)N1CCC(CNC(c2ncc(F)cc2F)=O)C1 c1(CCC(=O)N(CCNC(C2(Cl)CC2)=O)CC)ccc(C(=O)OC)cc1 C(=O)(CCCCCC#N)NC(CNC(COc1c(C)ccc(Cl)c1)=O)C C1(C)(CNC(CSCC)=O)CCCN1C(c1nc(-c2nc[nH]n2)sc1C)=O N1(C(CCCCC)=O)CCOC(C)(CNC(C23CC(CC)(CO2)C3)=O)C1 Cc1cc(C(=O)NCC2CC(CNC(=O)CNc3ccccc3)C2)c(Cl)cc1N c1(C(=O)NC(C)CC(C)NC(C23CC(F)(C2)C3)=O)cc(=O)c(Br)c[nH]1 C=C(C)CC(C)C(=O)NC(C1CCCCN1C(=O)CCCn1nc(C)nc1C)C C1(C(=O)NC2CC(C)(CC)C2)CC2CCC(C1)N2C(C1C2CCCC(=O)C12)=O c1(C(=O)NCC2(F)CC(NC(C#CC3(C)CC3)=O)C2)ccc2c(c1)OCCC2 c1(OC)ccc(C=CC(=O)N(CC(C)(C)NC(=O)C(C)CS(C)=O)C)nc1 c1(C(N2C(C)(C(=O)Nc3cn(COC)nc3)CCC2)=O)cc2cc(F)ccc2s1 C1(c2ccc(OC)cc2)COCCN(C(=O)Cc2ncc(F)cc2Cl)C1 C(=O)(CC(C)C(F)(F)F)NC(C(=O)NCC1CCCN(CC)C1)C(C)O C(CCC(C(=O)NOCCc1ccccc1)NC(=O)CCC1CCCN1C)OC C1(NC(c2cn(C)nc2O)=O)CC2(CCN(C(c3cc(Cl)cnc3O)=O)CC2)C1 CC1OCCN(C(=O)CC2(C#N)CC2)C1C(N1CCCN(C(N)=O)CC1)=O N1(c2cc(CC)nc(Cl)n2)CCCC12CCN(C(=O)COCCN1CCCC1)C2 C1(C(=O)NCC(C2CCN(C(COC)=O)CC2)(C)C)CCn2c(O)nnc2C1 N1(c2sc(C)c(Br)n2)CCOC(C)C1.C(=O)(C(O)Cc1ccccc1)N c1(C(N(C2CCCN(C(=O)CCS(=O)(=O)NC)C2)CC)=O)csc2nccn12 C=CC1(CC(=O)NCc2coc(C)n2)CN(C(c2cccnc2OC)=O)C1 c1(C(N2CCN(CCCNC(C3CNC(=O)C3)=O)CC2)=O)cc2c[nH]nc2s1 C(C(F)(F)C(F)(F)F)n1c(C)nc(-c2cccs2)n1 c1(COC)nn(C)cc1-c1cn(C2CC(NC(c3cnsn3)=O)C2)nn1 N1(C(c2c(CC)nccn2)=O)CCC(C(=O)NC(C)CN2CCOCC2)=C(F)C1 c1(SCCC(=O)OC)ccccc1N1CCCS1(=O)=O N1(C(C2(OC)CC2)=O)CCN(C(c2ccc(CC3CC3)s2)=O)C(CF)C1 c1(NC(C2(C)CCN(CCCCCC)C2)=O)ccc(OC)cc1C c1(C(=O)NC(C2CCN(C(C3CCS3(=O)=O)=O)C2)(C)C)ccc2oc(=N)[nH]c2c1 C1(NC(c2c(CC)noc2)=O)CC(CO)N(C(=O)C=Cc2ccc(Br)o2)C1 CC(C)CC(C(=O)NCCC(N1CCCC1C1CCC1)=O)C(C)C c1(OC)c(C(N2CCC(CNC(=O)CC3CCCCC3)C2)=O)oc2ccccc12 Nc1ccc(Cl)c(C(=O)NC2CC3(C2)CN(C(=O)Cc2cccs2)C3)c1 c1(C(N2CCC(C(=O)NCCCC)C2)C(=O)NC2(C)CC2)cc(Cl)c(F)c(Cl)c1 C(CC(C)(C)C)(C(=O)N1CCCC(C)(NC(c2ccc(N(C)C)c(F)c2)=O)C1)OC N1(C(c2cc(OCC)no2)=O)CCCC2(NC(=O)C(C)(C)CC)CCCC12 c1(C(=O)NCC2N(C(CC=C)=O)CC3(CC3)C2)cc2c(nc3ccccn23)s1 C(C)(CCC(=O)N(C1COCC1OC)C)NC(c1ccc(CC)s1)=O c1(C(=O)NCC2N(C(C3CC(C)C(C)CC3)=O)CCC2)ccc2c(c1)CCN2C c1(OCC(=O)OC)cccc(C(=O)NC2CCCCC2NC(C2CC(O)C2)=O)c1 C(C)(C)(CC(=O)NC(CNC(c1ccn(-c2ccncc2)n1)=O)C(C)C)SC N1(C(CC=C)=O)CC(C)(C)CC1CNC(=O)CC1C=CCC1 C1(OC)CCN(C(=O)C(=O)NCCC2(O)CCOCC2)C1CN Cn1cc(C(N2CCN(c3ncc[nH]3)CC2)=O)c(=O)c2cnn(C)c12 Cc1ccc(C(N2CCN(C(C3CC3C)=O)CC2c2cccnc2)=O)c(=O)n1C C1(CC=C)(NC(c2ccco2)=O)CC2CCC(C1)N2C(c1nn(C)c(N)c1C)=O CC(C)CS(=O)(=O)CC(=O)NC1CCN(C(=O)CC2CCCS2(=O)=O)C1 N1(C(=O)CC2CCCCC2)CC2CC(C1)N(C(c1cnc3[nH]ncc3c1)=O)C2 C1(C(=O)NCC2(O)CN(C(C3C(C(N)=O)CC3)=O)C2)CCN(CCO)C(=O)C1 c1(OCCCC)ccc(C(=O)NCC(F)CNC(C2(C)CCNC2=O)=O)cc1 c1(CC(=O)NCC2OCCC(NC(CC3C(C)(C)C3)=O)C2)ccc2occc2c1 N1(C(C2(CC#C)CCCO2)=O)CCCC(O)(CCNC(C2CC(F)(F)CS2)=O)C1 c1(C(=O)NCC2N(CC=C(C)C)CCCC2)cccc2nncn12 CCC(C(=O)NCCCCC(=O)N1CCCC(CCF)C1)C(C)C c1(NCCN2CCC(OCCN)C2)ccccc1[N+](=O)[O-] N12CS(=O)(=O)CC1C2=O.C1(OC(C)=O)CC12CC(NC(=O)CSC(C)C)C2 c1(NC(CNS(CCC)(=O)=O)=O)noc(C)c1C(=O)OCC CC1=C(C(=O)NC2CCC(CC(=O)NCC3C=CCC3)CC2)CCCO1 C(=O)(C(F)CC(CC)CC)N(CCN(C(C(C1CCCC1)OCC)=O)C)C C=CCCCCC(=O)NC1COCC1C(=O)NC1CCCSCC1 c1(C(=O)NC(CC)(C)CNC(c2cnco2)=O)cnc2cc(Br)ccc2c1 c1(C(=O)NCC(CC)NC(=O)C(C2CCCCC2)C)cc(CO)nn1C C1(C)(CNC(c2ccc(OCC)c(OC)c2)=O)CN(C(=O)C(C)(C)O)C(C)(C)C1 C1(CC)CC(CC(=O)NC2CCCC2NC(=O)C=CCO)CCO1 C1(NC(C#CCNC(C(C)NC(=O)OC)=O)=O)CC(CN(C)C)C1(C)C C(=O)(C1CCc2cc(Cl)ccc21)NCCC1N(C(C(CCCCC)O)=O)CCC1 C(C1CCc2cccnc21)O.N(C(=NCCCF)NC)CC1N(C(=O)OC)CCC1 C1(F)(C(=O)Nc2c[nH]nc2Cl)CC(C(=O)NCCNC(=O)Cc2cccs2)C1 c1(OCOC)ccc(CN2CCNC(C(=O)Nc3ccc(C(N)=O)nc3)C2)cc1 c1(C(N2CCN(C(c3cccc(C)c3C)=O)C(CF)C2)=O)cnn2cccc2c1 CC1=C(C(=O)N2CCC(NC(=O)CC(F)(F)Cl)C(CO)CC2)C(C)(C)CCC1 CC(N=c1nc2scnc2c(NCCCN2CCOC(C)C2)[nH]1)C1CCCC1 N1(C(c2ccn(C)c2C2CCC2)=O)CC2(C1)CN(C(c1ccc(Br)cc1)=O)C2 C1(NC(N2CCC(C(=O)NC)C2)=O)CCCN(C(=O)CC(C)SC)C1 c1(C(N(CCC(NOCCCC=C)=O)CCO)=O)ccc2cc[nH]c2c1 c1(OC)ccc(C(C)(C)C)cc1Br.C12CC3(CC1C3)NC2=O C(C(C)C(C)C(=O)NC1CCC(CNC(C2(CF)COC2)=O)CC1)OC N1(C(CSC(C)=O)=O)CCC2C1CCCN2C(=O)C(O)CC c1(C(=O)NCC(CNC(C2(C#N)CCOCC2)=O)O)ccc(O)c([N+](=O)[O-])c1 c1(C(CC)C)nc(C)cc(=NC2C3CN(C(=O)C(C)CC)CC23)[nH]1 Cc1cnc(O)c(NC(c2n[nH]cc2CNC(C2CCC3(CC3)C2)=O)=O)c1 Cc1cc(F)cnc1C(N1CCC(C)C(NC(C2CCS(=O)(=O)C2)=O)C1)=O C=CC(C)(C)C(=O)N(C)CC1CCN(C(=O)C(C)c2ncco2)C1 N1(C(C(CCCC)O)=O)C2CCC1C(F)C(NC(=O)CN1CCOCC1=O)C2 N1(C(CN(C2CC2)CC)=O)CCCC(NC(=O)C(C)OCC(C)C)C1.C1CN1 C1(Cl)(C(=O)NCC(C)(C)CNC(=O)CCCOC2CCCC2)CC12CCOCC2 N1(C(c2c(C)oc(C(C)(C)C)c2)=O)C2CCC1CC(NC(c1n[nH]cc1Cl)=O)C2 C#CCC(C)C(=O)OCCc1ccc(NC(c2cscc2C)=O)cc1 Cc1ccc(-n2nc(C3CCOC3)nc2-c2ccc(NS(N)(=O)=O)cc2)cc1 N1(C(COCC=C)=O)CCN(C(=O)Cn2cnc(C(F)(F)F)n2)CC1C(C)C c1(C(N2C(CN(C(=O)C(F)n3cccn3)CC)CCC2)=O)cc(F)cc(N)c1F C1(NC(c2n(C=C)nnc2)=O)CN(C(c2cnoc2CC)=O)C2CCCC12 C1(NC(C(c2ccccn2)C)=O)CN(C(=O)C(F)=CC2CC2)CC1(C)C C1(c2cn(CC3CCC(NC(C4CCC(C)C4)=O)C3)nn2)CCN(C)C1=O C1(NC(=O)C=Cc2cccnc2)CC(O)CN(C(c2c[nH]nc2F)=O)C1 c1(C(=O)NC2C(NC(C(C)OC)=O)CCCC2)cc(F)c(Cl)cc1Cl c1(C(N2CC(O)CC(NC(C3CCSC3)=O)C2)=O)cccc([N+](=O)[O-])c1Br c1(OC)cc(C(=O)N(CC(C)NC(C2(C)CNC(=O)C2)=O)C)cc(Cl)c1 C(C(C)(CO)N)NC(=O)C(C)CC1CCC1.C(CCOCCO)N(C(C)=O)C C(=O)(C(O)C(F)(F)C(F)(F)F)NCC1OCCN(C(c2c(C#C)cnn2C)=O)C1 Cc1ccnc2c(NC(=O)CN3CCN(C(C)C)C4CC34)cnn12 C12(C(N(CCCCCC)C)=O)C(NC(c3ccccc3OC)=O)C3CC1C2C3 C1(C(=O)NC2(C(=O)O)CCCC2)CCC2(CN(CCCCc3nccs3)C2)O1 c1(C(N2CC3C(CNC(C(CC)OC)=O)(C3)C2)=O)cc(Cl)c(OC)cc1OC c1(COC)cc(=NCc2cccc(Br)c2Br)[nH]c(Cl)n1 c1(C(N2CCC(NC(c3c(CC)n(C)nn3)=O)CC2)=O)c(F)ccc(Br)c1C c1(NC(C(CCC=C)NC(C2CC(=O)NC2(C)C)=O)=O)cc(C#N)ccc1C C1(CC)CN(C(C2(COC)COC2)=O)CCN1C(=O)CCS(N)(=O)=O c1(C(=O)NC2CCCC2NC(C2CC(n3ccnn3)C2)=O)coc2c1COC2 C1(F)(CNC(C2(C#C)CC2)=O)CCCN(C(=O)CCC(=O)Nc2nccs2)C1 CC1CCn2c(C(=O)NC3CN(C(c4ccccc4CO)=O)CC3O)cnc2C1 Cc1cn2cccc(C(=O)NC3CCC3NC(=O)CCc3cccc(Cl)c3)c2n1 C1(C(=O)NCC2C(C)C2C)CC2CC1CN(C(=O)C#CC1CCC1)C2 C1(C(=O)NCc2c(C)noc2)CCC(C2CC2)N1C(=O)CC1CSCCO1 N1(C(c2c(CC)oc(C)c2)=O)CCCC(C)C1CNC(c1cccc(=O)o1)=O Cc1noc(C2C(C(=O)NC3CCC3CNC(c3ccsc3)=O)C2(C)C)n1 C(=O)(C1COc2ccc(F)cc21)NCC1CN(C(CC2CC(C)(C)OCC2)=O)C1 c1(C(=O)OC)n[nH]c(=NCCCC(C)NC(C2CC(=O)NC2(C)C)=O)s1 c1(CC(=O)NC(C(=O)NCCC=CC)CC2CCCC2)ccc(F)nc1 N1(C(COCCOCC#C)=O)CC(C)(C(=O)N(C)CC2CCOCC2)CC1(C)C C12(NC(c3c(C)con3)=O)CCCC1N(C(c1cc(Cl)sc1Cl)C)CC2 CC(C)CC(C(=O)NCCC1(O)CCOC1)ONC(C1(C)CCCC1C)=O N1(C(Cn2c(C)nc(C)n2)=O)CC(CNC(=O)C(C)C2CC2)OC(C)(C)C1 C(=O)(C(C(=O)N1CCC(C(=O)N(C)CC2CCCC2(C)C)(CO)C1)OC)OCC N1(C(c2cn(CCC(F)(F)Cl)nn2)C)CCOC(C)(CO)C1 c1(C(=O)NC2CC(CCNC(c3c(CCC)n[nH]c3)=O)C2)ccc(CC#N)cc1 C1(OC)CN(C(=O)Cc2cn[nH]c2)CC1NC(c1c(C2CC2)n[nH]c1C)=O Cc1cccc(C(=O)NCCC(=O)NCCC(O)C2CC2)c1 N1(C(CCc2ncn(C)c2)=O)CC=C(C(=O)NC2CC(O)C2(C)C)C1 C(=O)(CCS(N)(=O)=O)N(CC(CC)NC(=O)C=CSC)CC N1(C(C(COC)COC)=O)CC(CO)C2(C1)CN(C(c1nn(C)c(C)c1Cl)=O)C2 C#Cc1cn(C)nc1C(=O)NC1CC12CC(NC(=O)Cc1cnc(C)[nH]1)C2 C1(CCNC(C(C)NC(COC)=O)=O)CCCCN1C(c1cc(C)c[nH]1)=O C(=O)(C(F)(F)C(C)(C)O)N1CC(C(=O)NC(C)C(C)(C)CO)CC(C)C1 Cc1ccc(C(=O)NC2CC3CC(NC(=O)C=CCN4CCCC4)C2C3)c(C)n1 C1(CNC(C2(c3c(C)ccc(C)c3)CC2)=O)CC2COCC2N1C(=O)C(C)C#N c1(N2CCC(OCCCC)CC2)nc(Cl)cc(=NC2CCC3(C2)CC3(F)F)[nH]1 C1(CNC(CC2C3CN(C(C(CC#C)C4CC4)=O)CC32)=O)CC2(CCCO2)C1 N1(C(c2cccc(CC#N)c2)=O)CC2CCC(C1)N2C(=O)CC1COCCOC1 Cc1cc(C#N)ccc1-c1cn(CC(=O)O)nn1.C(=O)(CCCCN1C(=O)CCC1=O)N CC(C)(F)C(C)(F)C(=O)N1CC(CO)C2(C1)CN(C(c1cncc3cnccc13)=O)C2 c1(OC)ccccc1CCC(=O)NC1CN(C(=O)CCc2cnoc2)CC1C N1(C(C2C(CC)CCCC2)=O)C(C(=O)N(CCCO)C2CCC2)C2CCCC12 c1(N(CCCCCCC=C)CC2CC2)cc(OC)c(OC)cc1[N+](=O)[O-].CO c1(C(=O)NCC(COC)NC(c2nnn(C)c2N)=O)cc2c(s1)CCCC2 N1(C(C(=O)NC(c2ccc(OC)cc2)CC)=O)CC2(CCC2N(C)C)C1 C[Si](C)(C)c1ccc(C(=O)NC2CCN(C(c3cc(Br)cnc3O)=O)C2)cc1 c1(C(=O)NC(C)CCNC(=O)CNS(N)(=O)=O)cncc(Cl)c1Cl c1(C(N2CCCN(C(C3C(C)CCS3)=O)CCC2)=O)sc2ncccc2c1Cl N1(C(c2ccc(OCCN(C)C)c(F)c2)C(=O)NC)CCC(P(C)(C)=O)C1 C1(NC(COC2CN(C(C)=O)C2)=O)CCCN(C(=O)CCCOCCNC(N)=O)C1 c1(CCC(=O)NC2CN(CCn3cc(CO)nn3)CC2F)ccc2c(c1)CCO2 C(=O)(CC(C)(C)CC(F)F)N1CCC(O)(CCNC(C2C(C)(CC)C2)=O)CC1 c1(C(=O)NCC#CCNC(C(C)c2ccco2)=O)sccc1Cl C(=O)(C(CCOCC)NC(=O)CCn1ccnc1)N1CC(C#C)C1 C1(N(C(=O)CCC2CCC2)CC)CCN(C(=O)C=CCOC(C)(C)C)C1 C1(C(N2CCC(CNC(C(C)(C)N(C)C)=O)C23CC3)=O)CCCC(C)(F)CC1 Cc1ccc(CCCNC(=O)NCC2CCC2)s1 N1(C(C(F)=C(C)C)=O)CCC2(CC1)CC(NC(=O)C(F)(F)C(C)O)CCO2 C1(O)(C(=O)NCC(CC)NC(c2c[nH]c(C(F)(F)F)c2)=O)CCCC(C)CC1 c1(C(N2C(C(C)NC(C(CC#C)O)=O)CCC2)=O)ccc(Br)c(C)n1 C(CC(C(=O)NCc1cccc(Cl)n1)OC)NC(Cc1cc(OC)no1)=O C(=O)(C(F)CC(C)(C)NC(c1cn(C)cn1)=O)N(C1CC(N(C)C)C1)C N1(c2c(C)cccc2)C(=S)NC(c2csc(C#N)c2)C2=C1CCNC2=O C1(C(N2CC(O)CC(NC(c3ncc(Cl)cc3Cl)=O)C2)=O)CCc2nc[nH]c2C1 CN1CCC(OCC2(F)CC2(Cl)Cl)C1c1ccccc1 c1(-c2n(CC(=C)C)nc(-c3cnn(C)c3)n2)cc2c(COC)nn(C)c2s1 Cc1cc(NC(c2cnn(C(C)C)c2Cl)=O)c(C)n1C1CCCCC1 c1(C(N2C(CC(=O)N(C)CC3N(CC)CCC3)CCC2)=O)ccnc2cc[nH]c12 NS(=O)(=O)c1cc(C(=O)NCC2C=CCN2C(=O)Cc2cc[nH]c(=N)c2)co1 N1(C(C(C)C2CCOC2)=O)CCCC(CNC(c2cnn(C(F)F)c2)=O)CC1 c1(C(C(=O)NCCCN(C(C=C(CC)CC)=O)C(C)C)(F)F)cccc(C)n1 c1(NC(C=CC(=O)NC2(C)CCN(C(=O)CN3CCCC3)C2)=O)cc(O)ccc1Cl C1(NC(CSCC=C)=O)CCN(C(=O)CC2CCC(F)(F)CC2)CC1CO Cc1nc(C(N2CCC(NC(c3cc(O)nn3C)=O)C(CO)C2)=O)c(C)n1C C(=O)(C1CCCn2nccc21)N1CCN(C(COc2ccc(C)cc2F)=O)CC1 N1(C(C(C)(C)O)=O)CC2CC1CN2C(C1CCCS(=O)(=O)C1)=O C1(NC(CN(c2ncccn2)C)=O)CCCCN(C(c2cccc(F)c2Cl)=O)C1 CC1CCCCC1(CNC(=O)CC1CC2(CC2)CO1)NC(C12CC(F)(C1)C2)=O N1(C(c2cccc(CNC(c3cc(C)nc(C)n3)=O)n2)=O)CCC(O)C(F)(F)C1 C[Si](C)(C)C1(CNC(C2(CCNC(=O)CC3CCCO3)CC2)=O)CC1 C1(CNC(C2N(C(C)=O)CCC2)=O)CCN(C(C2CC2(C)C)=O)C12CCC2 c1(C(=O)NC23CC(CNC(c4nc(CCC)sc4)=O)(C2)C3)ccc2sncc2c1 c1(C(=O)NCC2C(NC(C=COCC)=O)CCCC2)cc2ccccc2o1 c1(SCC(N2CC(O)C2)=O)ncc(C)[nH]1.C1(O)C(C(=O)NCCCC)C1C c1(N2CC3C(C(N4Cc5c(nn(C)c5N)C4)=O)C3C2)ncnc2c(F)cccc12 c1(C(N2C(CNC(=O)C3CC3)CCC2)=O)cccc(C2(O)COC2)c1 c1(C(=O)NC2C(CC)CN(C(=O)C(F)=CC3CC3)CC2)cn(C)c2ccccc12 Cc1noc(C)c1C(C)CC(=O)N(C)CCN(C(=O)CCNc1ccccn1)C C1(C(=O)NCC2N(C(c3cc(C)sc3)=O)CCC2)CCCCCS1(=O)=O N1(C(C(C)(C)c2cccs2)=O)CCC2(C(=O)NCC(c3ccco3)O)CCCC12 N1(C(c2cc(=N)[nH]cc2)=O)CCC(CNC(c2scnc2Cl)=O)C12CC2 N1(C(=O)Nc2c(C)c(C)cc(C)c2C)CCCC2(CC1)CNC(=O)O2 N1(C(c2c(C)cc(=N)[nH]c2)=O)CC(C)CN(C(=O)CC23CC(C2)C3)C(C)C1 C1(CC(=O)NC(C)CCCNC(=O)CCC(F)F)CC2CCC1CC2 C(CCS(C)(=O)=O)NC(c1cc(CNC(Cc2cc(C)no2)=O)no1)=O Cc1oc(CO)cc1C(=O)NCC(C)=CC(=O)N(C(=O)C1CC1)CC1CC1 C1(C(=O)NCCOCCC=C)C(CC)CCN1C(C1CSC1)=O C(CCC)(C(=O)N1CCC(N(C(=O)CN2CC3CC3C2)C)C1)=CCC CN1CCC2(CC1)CN(C(C1CCC3(CCOCC3)CO1)=O)CCN2C C(CO)(C(F)(F)F)NC(c1cc(CNC(c2cc(=N)[nH][nH]2)=O)on1)=O C1(N(C(c2c(CC)ocn2)=O)C)CCCN(C(=O)Cc2ccccc2O)CC1 C(=O)(CC(F)(F)C(F)F)NC(CC(C)NC(C=CCC)=O)C CCCC(C(=O)NCc1ccnc(C(=O)Nc2cccc(CC)c2)c1)C(C)C N(C1CCCn2ncnc21)C(C(C)N(C(=O)CCc1cnn(C)c1)CC)=O c1(C(N2CC(N(c3ncccn3)C)C2)=O)ccc2[nH]nc(O)c2c1 CC(CC(F)(F)F)N(C(=O)CCC1CC(NC(=O)CCc2ccc[nH]2)C1)C Cc1[nH]c(=N)nc(O)c1CC(N1CCC(NC(c2cc(Br)c[nH]2)=O)C12CC2)=O Cc1ncncc1C(=O)NC1CCN(C(=O)C(O)CNC(=O)OC(C)(C)C)CC1 c1(C(=O)NC2CN(C(CN3CC(C)C3)=O)C(C)C2)cc(S(=O)(=O)N(C)C)c[nH]1 C1(=CC(=O)NCC(C2(C)CC2)O)CCCCC1(C)C c1(C(=O)NCCN2CCN(C)CC2)ccc(NC(C2CC3CCC2N3)=O)cc1Cl c1(CC(=O)NCC(CNC(Cc2cn(CC)nn2)=O)(C)O)ccc(Cl)nc1F C(=O)(C(O)C1=CCCCC1)NCC1N(C)CCN(C(=O)COC2CCC2)C1 c1(COC)nc(NC(=O)C(c2cn(C)nn2)NC(c2cnn(C(C)C)c2)=O)n[nH]1 N1(C(C(C)(C)C(F)F)=O)CC2(C1)CN(C(C1CCCN3CCCC13)=O)C2 N1(C(c2cn(CCC)nn2)=O)CC(CNC(c2cncn2C)=O)CCC1C N1(C(CC2ON=C(CC)C2)=O)CCc2ccc(C(=O)NCCCSC)nc2C1 C(=O)(C1=CCCOCC1)N1C(CNC(c2ccn(C(C)C)n2)=O)CCC1 C(C)(C(C)C(=O)N1CCN(C(C)C)CC1)NC(c1cnc(CC)s1)=O S(=O)(=O)(CCCN=c1[nH]c2c(c(=NCCS(=O)C(C)(C)C)[nH]1)COC2)N(C)C C1(C(=O)NCC2(CNC(c3[nH]cc(C)c3)=O)CC2)CC(S(N)(=O)=O)C1 c1(C(N(CC(C)NC(=O)CCCn2cnnn2)C)=O)cc(F)cc2ccncc12 N1(C(c2c(C)nc(C)s2)=O)CCC2CN(C(=O)C(C)O)CC2C1 c1(CNc2cc(Cl)cc(OC)c2N)cccc2cccc(C)c12 c1(CN(C(CCN(C(c2nc(C)oc2)=O)C)=O)C)cccc(O)n1 C1(C(N(C)CC2CCN(C(=O)COc3ccon3)C2)=O)CN(C)C(=O)N1 N1(C(=O)Cn2cccc(C(F)(F)F)c2=O)C2CC3C4CC(C3C2O)C1C4O.C1COC1 N1(c2snc(SC)n2)C2CCC1CC(NC(=O)COC1CCCC(C)C1)C2 C12=CC(=NCCC(=O)N1)NC=N2.C(CN(C)C)(C1CC1)OC C(=O)(C1=CCCN(C(=O)OC(C)(C)C)CC1)NC(C)CNC(C1(Cl)CC1)=O C1(C)(C(N(CC=C)C)=O)C=CCN1C(c1cnc(C2CC2)o1)=O c1(OCC)ccc(C)cc1NC(C1CC1NCc1nccn1C)=O CC1CCCN(C(=O)C(=O)NC2(C)CCN(C(c3cc[nH]n3)=O)C2)C1 N1(C(C2CC(=O)OC2)=O)CCOCC(CNC(=O)CN2CCC(F)CC2)C1 C(=O)(C(COC)CC(C)C)N1C(CC(=O)NC2C(CC=C)COC2)C2CCCC21 c1(OC)cccc(C(=O)N(CC(O)CNC(c2ccnc(S)c2)=O)C)c1 C1(CNC(CCCc2c(C)ccs2)=O)(NC(=O)CC2CC2C2CC2)CCOCC1 C1(C(=O)NC2(CC)CC2(F)F)(CNC(CC)=O)CCC(=O)N1 N1(C(C(CC)O)=O)CCc2sccc2C1CNC(c1ccc[n+]([O-])c1)=O c1(C(N2C(CNC(C(C(CC)O)C)=O)C3CCC2C3)=O)ccnc2[nH]cnc12 CCCC(O)(CCC)CC(=O)NCCC(C)NC(C1COCCC1C1CC1)=O c1(SC)cccc(C(=O)NC(CNC(=O)C2=CCC2C)CO)c1[N+](=O)[O-] CN1CCC(F)(C(=O)NCCOCCCN(C)C(c2cnc(O)n2C)=O)CC1 N1(C(C)=O)CC(O)CC1C(=O)NCCNC(c1nc(O)c(C)s1)=O c1(C(=O)NCC2(O)CN(C(=O)C=C(Cl)Cl)C2)coc2c1CS(=O)(=O)C2 c1(OCCCN(C)Cc2cccc(OC3CC3)c2)ccccc1C c1(C(N2C(CNC(c3csnc3C3CC3)=O)CC(OC)C2)=O)ccc(C)cc1C C1(C(=O)NCCCCNC(C2CC(C)OC2C)=O)CCCNS1(=O)=O N1(C(Cn2c(C)ncc2)=O)CCN2CCN(C(c3cc(C(F)F)no3)=O)CC2C1 N1(C(c2c(OC)ccs2)=O)CCN(C(=O)CC(C)(C)C2CC2)CCC1C C12(C(N3CCOCC(CNC(C4C(=C)C4)=O)C3)=O)CC3CC(C1)CC(C)(C3)C2 Cc1ccc(CC(=O)NCCC2CC(Nc3nc(C#N)c(Cl)s3)C2)cc1[N+](=O)[O-] c1(C(=O)NCC(CN(C(=O)CN2CCSCC2)C)O)cnc2nc(O)ccc2c1 c1(C(=O)NC2C(NC(c3ccc[nH]3)=O)CC2)cnc(O)c2cccnc12 CCCC(CC(C)C)C(=O)N(C1CCC(NC(=O)C(C)OC(C)C)CC1)C CN1CCC(CC(=O)NCC2(C(N3CC4C=CC4C3)=O)CC2)CC1 N1(C(C(CCC=C)CCC)=O)CCC2(CCOC2)CC1 C12CC(N=C3NC(=NC(=N)N3)N(C)C1)C2.C(C(=O)NC)N(C1CC1)CC C1(O)(CCNC(CCNS(CC)(=O)=O)=O)CCN(C(=O)C(C)(F)CC)C1 C1(C(=O)NC2CCC(F)C2)CC2(C1)CN(C(C1CC1c1ccccc1)=O)C2 C(CS(=O)(=O)CC(=O)NCC1(C(=O)NCCc2cccn2C)CC1)OC C(=O)(CCCCCCC(=O)O)OC(C1CC(OC)C12CCCC2)=O C(=O)(C(C)(C=C)CCOC)NC(CC=C)CNC(=O)CC=CC Cn1cc(CN2CC3(CCCN3C(c3ccc(F)c(Cl)c3)=O)C2)c2cccnc12 c1(C(N(CCNC(c2ccc(C)s2)=O)CC)=O)cccc(C=C(F)F)c1 C(=O)(CC(C(C)(C)C)NC(C1CC1(Cl)Cl)=O)NC(C(=O)OC)C N1(C(CCC(CC)C)=O)Cc2ccc(CNC(=O)C(C)NC(N)=O)cc2C1 c1(C(C)=O)cc(C(=O)NCC(O)CN(C)C(c2n[nH]cc2Br)=O)c(C)o1 C1(C(C)C)CCc2nc(O)c(C(=O)NCCn3cc(CC(C)O)nn3)cc2C1 CC1(C(=O)O)CCCC1N(S(C)(=O)=O)C(c1ccc(C(=O)NC2CC2)cc1)=O C1(NC(C2(SC)CC2)=O)CCCCC12CCCN(c1cc(C)nc(C(C)C)n1)C2 N1(C(c2cccc(C(C)C)n2)=O)CC2CCC(NC(c3ccnnc3Cl)=O)C2C1 c1(COC(N2CCC(C(=O)OCC)C2SC(F)(F)C(F)(F)F)=O)cccc(C)c1 N1(C(c2c(-c3c(C)ccnc3)ncs2)=O)CC2(CC2)n2nccc21 C(=O)(CC1=C(C)NS(=O)(=O)N=C1C)N1CC(C)CC(CNC(C(CSC)C)=O)C1 CCC(O)C(C)(C)C(=O)N1CCC(CO)(NC(c2ccc(O)c(C(N)=O)c2)=O)C1 c1(CC)cccc(C(=O)NC2CC(NC(=O)C(F)CC3CC3)C2)n1 c1(C(=O)NCC(C2CCCCN2C(=O)CC2CC(CF)C2)(C)C)ccc(F)cc1 CCC(C)(F)C(=O)NCC1(CNC(=O)Cc2cc(C)sc2C)CCCC1 N1(C(CN(CCC)C)=O)CC(NC(=O)CCCc2cc(C)no2)CCC1C c1(OC(C)C)n[nH]c(=NC(=O)N2CCC2c2cccc(Cl)c2F)s1 CN1CC2CCC(C1)N2C(=O)C(C)(C)CNC(=O)CC1CCCO1 C1(CC(=O)NC(C(=O)NC(C(=O)N(C)C)CO)CO)CCCC1(C)C Cc1n[nH]c(=NCCCN(C)C(c2cn(CC3CC3)nn2)=O)s1 CC(C(C)(C)C(=O)NCCN1CCNC1=O)NC(=O)Cc1ccccn1 N1(C(C=CCCC)=O)CCC(CC(=O)NC(C2CC2)C2CC2)CC1 CC#CCCCC(=O)NCC(C)NC(=O)C(C)OCc1ccncc1 CP(C)(=O)C1(C(=O)NCCC2(CNC(c3ccc(Cl)cc3)=O)CC2)CC1 c1(C(=O)NCC(CC)(C)NC(=O)CCC2CCCN2C)cnn2c1CCC2 c1(CC(=O)N(CC(C)O)CCNC(C(CC2CC2)OC)=O)cc(C)sc1C CC1=C(C(=O)NC2CCC2NC(C2CC(C(C)C)=NO2)=O)CCCO1 C1(NC(C(CCSC)O)=O)CCCC2CN(c3cc(C#N)nc(C)n3)CC12 C(c1cccc(O)c1)=CC(N1CCCC(CNC(C=Cc2occ(C)n2)=O)C1)=O N1(C(CCC)C)Cc2ccc(NC(=O)N(C)CCC3CCC(=O)N3)cc2C1 c1(CC(=O)NCC(CC)NC(c2ccc(C)cc2O)=O)c(F)c(F)cc(F)c1F C1(CN2C(CS(=O)(=O)Cc3nnc(SCC)s3)CCC2)CCC(F)(F)CC1 N1(C(c2cn(CC(CC)O)nn2)=O)CCC2C(CCN2C(C2CCCC2C)=O)C1 c1(C(C)NC(C2CC2c2sccc2C)=O)ccc(OCC(F)F)cc1[N+](=O)[O-] C1(NC(CC(CC=C)NC(=O)C=Cc2ccc(C)o2)=O)C2CCC(C2)C1(C)C c1(NC(=O)NCC2CCCC(CC)C2)c(N=[N+]=[N-])cnnc1O c1(CNC2CC(C(=O)NC(c3c(C)n[nH]c3C)C)C2)ccc2ncsc2c1 CC(C)(C#N)CCCC(=O)NCCC1CC(NC(C2CCCCN2C(N)=O)=O)C1 Cn1cnc2cc(C(=O)NC3(C)CC(NC(=O)OC(C)(C)C)C3)ccc12 Cc1cc(C)c([N+](=O)[O-])cc1C(=O)NC1CC1NC(=O)Cc1ccsc1 c1(C(C(F)(F)F)OC(C(C)=CC2CC2)=O)ccccc1C#N c1(C(=O)NCCC2(NC(C3=C(C)OCC3)=O)CCC2)ccc(S(N)(=O)=O)cc1 C1(NC(c2c(C)nncc2)=O)(CO)CCCN(C(C2(C#N)CCCO2)=O)C1 C=CCC(CC(=O)NCC(C)CC(=O)OC)NC(C1CCC1C#N)=O c1(CCC(=O)NCC(C)N(C(C(C(C)C)CO)=O)C)cc2ccccc2o1 c1(NCCNC(CC)=O)nc(=NCC(C(C)C)OC)[nH]c2ncn(CC)c12 c1(OCC(=O)NC2C(NC(C(C)c3cccs3)=O)C2)ccccc1C(F)F C12(C(N(CCCSC)C)=O)COCC1CN(C(=O)CC1(NC(C)=O)CC1)C2 c1(C(=O)NCC(CC(=O)NCCn2c(C)cc(C)n2)O)cc2n(n1)CCC2 c1(C(N2CCC(O)(CO)C(O)C2)C(=O)NCC(F)F)n[nH]c2c(F)cccc12 S(=O)(=O)(c1ccccc1OC(F)(F)F)N1CC(NS(CC)(=O)=O)C1 c1(C(CC)NC(=O)NCC2CN(C)C(=O)O2)ccc2cc(Br)ccc2c1 CC(C)C(C)(O)C(=O)NC(CNC(c1cc(-c2cccs2)on1)=O)CO c1(C(=O)NCC(CC(C)C)NC(C=CSC)=O)coc2cc(C3CC3)ccc12 C1(C(N2CC(C)C(NC(=O)CCn3cccc3)C2)=O)CC2CCC1CC2 N1(CC)CCOCC1C(=O)NCCC(C)N(C)C(c1cnns1)=O CC1CC2CN(C(=O)C3=NN(C)C(=O)CC3)CC2N1C(c1ccncc1)=O Cc1ncc(C(=O)N(CC(C)NC(=O)Cc2ncccc2C)C)c(O)n1 c1(C(N2CCC(CC(=O)N(CC)CC3CCC3)C2)=O)ccc(F)cc1Cl CC1CC2CN(C(C3CCC(C)(C)OC3)=O)CC2N1C(=O)C(F)CC1CCOC1 c1(OC(c2csc(-c3cnccn3)n2)=O)ccc(N2CCOC2=O)cc1 N1(C(CCC#CC)=O)CC(OC)CC1(C)NC(=O)C(=O)Nc1ccccc1C#N C1(OC)CC(CF)N(C(C2CCCCN2C(=O)C(C2CCCCC2)C)=O)C1 C(CCC(=O)NCC(C)NC(C1CC1(C)C(C)C)=O)OCC(C)C CC1CN(C(=O)Cn2cccn2)CCCN1C(C1OC2CCC1CC2)=O c1(N(CC(C)CO)C)ncccc1S(=O)(=O)NCCN=c1cc[nH]cc1 C1CC2CC1CC2=O.CC1(C(=O)N(CCCF)CCO)CN(C=O)C1 N=c1[nH]c(=NCCC2CC(=O)NC2=O)[nH]c(=NCCN2CCCCC2)[nH]1 C1(COC(=O)Cc2nc(=N)[nH][nH]2)CCCCC1c1ccccc1.CCC1C(=O)O1 c1(NCc2cc(C)c(C)[nH]2)c(C)cccc1F c1(C(N2C(CNC(C3(COC)CCCO3)=O)CCC2)=O)cc(Cl)c(N)cc1F C1(NC(c2ncnc(C)c2C)=O)CC2CC(NC(=O)CC(C)(C)C)CC2C1 N1(C(C(CCCC)O)=O)CCCN(C(=O)Cn2cc(C(F)(F)F)nn2)C(CO)C1 Nc1c(C(N2CCCCC2CCCNC(C2CC(O)C2)=O)=O)cccc1[N+](=O)[O-] N1(C(C2CN(C(C3C(C)OCCO3)=O)C3(C2)CCC3)=O)CC2CCC(C1)C(=O)N2 N#Cc1cnc(NC(=O)Cc2csc(NC(c3ccc(O)nc3)=O)n2)cn1 c1(C(C)SCC(N2CCC(C(OCC)OCC)C2)=O)nc2ccccc2o1 C(=O)(C(O)CC(C)C)NC(C(=O)NC(CC)C(N)=O)C(C)OC Cc1ncc(C(N2CC=CC2(C)C(N2CCC(OCC(C)C)C2)=O)=O)n1C Cc1csc(C=CC(=O)NCCC(O)CNC(=O)C(C)c2cccs2)n1 c1(C(=O)NC(CC)C(=O)N(C)Cc2cccc(O)n2)ccn2nccc2c1 N1(C(COc2cccc(CC)c2)=O)CC(C)(C)OCC1CNC(=O)C(C)CF CCC(O)C(C)C(=O)N1CC(F)CC1CNC(c1cnn(C2CC2)c1Cl)=O c1(C(=O)NCC2(F)CC(CNC(c3c(CC)scn3)=O)C2)cccc(O)c1 CC1=NOC2(C1)CC(C(=O)NCCC1(O)CN(C(=O)CSCc3cscn3)C1)C2 c12nc(cn(N)c1=O)N2.C1(CN(C)C)CCN(C(=O)OC(C)(C)C)C1 c1(C(=O)NC2C(CNC(C=C(CC)CC)=O)CC2)cc(S(N)(=O)=O)c(C)cc1C C1(CCC=C)(C(=O)N(CC(C)(C)NC(=O)CN(C)CCOC)C)CCCC1 c1(C(=O)NCC2C(NC(c3c(OC)cccn3)=O)C2)ccc2scc(C)c2c1 c1(C(N2CC(CCC)N(C(=O)C(OC)OC)CC2)=O)ccc(C)c(F)c1N N1(C(COCC)=O)CC(CNC(C2CCCN2C(C)=O)=O)C(O)C1.C(=O)(CC)N N1(C(c2ncc(C)cn2)=O)CC2(CNC(=O)COC(=O)CO)CC1CCO2 C(=O)(C(CO)C(F)(F)F)NCC1CN(C(C2C(C)(C)C2Cc2ccccc2)=O)C1 N1(C(C2C(NC(C=C(COC)C)=O)C=CCC2)=O)CCC(C2CCCC2)C1 c1(C(N2C(CNC(=O)CC3CC3(Cl)Cl)C=CC2)=O)ccc(CN2CCC2)cc1F C(=O)(CC1=CCN(C(C2(Cl)CC2C(C)=O)=O)CC1)NCC(CC(=O)OC)O Cc1nccc(C(=O)NC2CN(C(c3n[nH]c4c3CCC4)=O)C2)c1C C1(C(=O)NCC=CC=CCNC(=O)CC2CSCCS2)CCCOCC1 N12CCc3ccccc3C1CN1C(=CC=C([N+](=O)[O-])C=NC(CCCl)C1=O)C2=O c1(C(=O)NCC2N(C(C3CC(=O)NC3)=O)CCC2)cc2c(cn1)COCC2 C1(C(=O)NCC2CCCN(C(CNS(C)(=O)=O)=O)C2)CC2(C1)CC1(CC1)C2 Cc1c(C(=O)NCC2CCCN(C(=O)CCOCC3CCCO3)C2)ncn1C c1(C(=O)NC2CCN(C(=O)Cc3sc(O)nc3O)C2)cc(F)c(C(F)F)c(F)c1 C1(CC(=O)NC(CCOC)COC)COCCN1C(=O)CC1C(=O)NN=C1C C1(C(C(N2C(CC(=O)N(CC(C)(C)C)C)CCC2)=O)=O)CCCCCC1 C12(NC(c3c(C)ncnc3)=O)CC(CNC(=O)C(c3ccccc3)C)(C1)OC2C C1(C(=O)NC(CC#C)C(=O)NCC)C2CCC(C2)C1NC(=O)C=Cc1ccsc1 C1(CC=C)(NC(=O)C(C)=C(C)C)CCN(C(=O)CC2(OC)CC2)C1 c1(C(N2CC(CNC(c3cnc[nH]3)=O)C3C2C3)=O)cc(Cl)c2c(c1)OCO2 C1(C2(C(N(CC(CNC(COCC(C)C)=O)O)C)=O)CC2)CCCCO1 CCC(CC(C)C)C(=O)NC1CN(C(=O)CN(c2ccc(Cl)cn2)C)CC1F C(=O)(CC(C)C(=O)c1ccccc1)N1C(CN(C(c2ccc(C)s2)=O)CC)CC1 C1(C(N2CC=CC(NC(c3c(C)nc(C)o3)=O)C2)=O)CCC12CCCO2 C(=O)(C1=CSCS1)NC(C(C)NC(C1CC(F)C1)=O)(C)C CCC(C(=O)NCC1C2CCC(C2)N1C(c1cc(C)cc(N)c1)=O)C(F)(F)F c1(NC(C2CN(C(c3ccc(C(C)=O)o3)=O)C2)=O)cn(C)c(=O)nc1O C1(C(C)(C)C)(CNC(c2ccc(O)nc2)=O)CCN(C(=O)C=CC2CCOC2)C1 N1(C(C(N2CCNC2=O)C)=O)CCC(C)(C2CC2)C1.C12CC1C(=O)NC2 C1(C(N2CCC(NC(Cc3c(C)non3)=O)CC2C)=O)CN2CCN1CC2C c1(-c2scc(C(=O)Nc3cccc(Cl)c3Br)n2)ccc([N+](=O)[O-])cc1 C#Cc1cnc(C(=O)NCC2N(C(=O)OCC)CC2(C)C)c(C)c1.C(C)(C)(C)O Cc1cnc(-c2nc(CCCO)nn2C2CCC(C)(C)C2)c(C)c1 CC1CN(C(=O)C(Cc2cc[nH]n2)NC(C2CCC(=O)O2)=O)CCC1CO CCN=C(NCC1(N2CCCCC2)CCCC1)NC1CCN(Cc2cccs2)C1 CC1(CCNC(=O)C2=CCSC2)CCN(C(C2CCC(C3CC3)O2)=O)C1 S(=O)(=O)(c1ccccc1)N1C(c2ccccc2)CCC(C)C1 N1(C(CNC(CSCCC)=O)=O)CCCC(C)(OCCOCC2CCOC2)C1 CCC(CCCO)N(C(=O)C(N1CCCC1(C)C)=O)C(N1CCCC1)=O N1(C(CCC(=O)NCCC)=O)C2CCC1CN(C(C1CC(=O)N(C3CC3)C1)=O)C2 Cc1nc2ncccc2cc1C(=O)NNC(=O)CC12CC3CC1C2C3 c1(C(N(C2CC(OC)C2)C)=O)ccc(CNC(C2(C#N)CCCO2)=O)cc1 C12(CC(=O)NC(C(C(C)C)NC(=O)CNC(=O)C(F)(F)F)C)CCC(CC1)CC2 CN1CCCC(NC(CCCCc2onc(CN(C)Cc3ccccc3)n2)=O)C1 c1(C(N(C(CNC(C(=O)Nc2ccc(C)cc2)=O)C)C)=O)c(C)cncc1C N1(C(C(CC2CN(C(C3(CC#C)CC3)=O)C2)F)=O)CCCCCCC1C c1(C(=O)Nc2c(C)c(Cl)ccc2)n[nH]c2c1CN(C(=O)C(C1(O)CCCC1)F)C2 c1(CC(=O)OC(c2cccc3ccccc23)C)c[nH]c2cc(OC)c(OC)cc12 CC(CCCc1ccccc1)C(=O)N1CCCC(NC(c2ncn(C)n2)=O)C1C C(c1ccc(Cl)c(Cl)c1)=CC(N1CC(CC)N(Cc2cncs2)CC1)=O c1(NC(CC2(O)CCN(C(c3nc(C)oc3)=O)CC2)=O)ccc([N+](=O)[O-])cc1 c1(C(=O)NC2CC3CN(C(c4c(COC)cco4)=O)C2C3)cnn2cc[nH]c(=O)c12 N1(C(CC2C(NC(C3CNC(=O)N3)=O)CC2O)=O)CC2C=CC1CC2 C1(NC(C)=O)CCN(C(c2ccn(C(C)C)c2)C(=O)NCC2CCOC2)CC1 Cc1ccn2ncc(C(=O)NCC3CCCCC3NC(=O)CCC3(C)N=N3)c2c1 CC(C)(O)C(F)CNC(=O)CC1(C)CCN1C(C1CC=CCC1)=O N1(C(c2cccc(NC(c3ccc(=N)[nH]c3)=O)c2)=O)CCC2CCC(C1)S2 C1(CNC(c2c(C)ccs2)=O)CN(C(=O)CNC(C2CCC2)=O)C2CC12 c1(C(N2CC(NC(=O)Cc3c[nH]nc3O)C(CO)CC2)=O)cc(F)c(F)cc1F N1(C(C(C(C)C)c2ccncc2)=O)CC(C)(C)CC1CNC(C1CC1C(C)O)=O N1(C(c2cnc(Cl)cn2)=O)CC2(CCC(NC(C3CC(O)C3)=O)C2)C1 C=C(F)C1(CC(=O)N(CCCNC(=O)CC2C=CCC2)C2CC2)CCOCC1 c1(C(=O)NCc2cc(-c3ccc(O)cc3)on2)ccc(N2CCC2)nc1 C1(C(=O)NCC(C(C)C)NC(c2c[nH]c(=NCC)s2)=O)CCc2cncn2C1 CC1=CC(C)CN(C(C2CN(C(=O)CC(C)N(C)C)CC2C)=O)C1 c1(C(=O)NCC23C(CN(C(c4cnc(C)[nH]4)=O)C2)C3)nc2cccnc2s1 C1(OC)CN(C(=O)CCC(N)=O)CCC1NC(=O)Cc1cn(C)cn1 N1(C(C=C(C)c2ccco2)=O)CC2(CCC2)CC1C(=O)NC1CNC(=O)C12CC2 C1(C(N(C(C)COC)CC)=O)(NC(=O)CC2C=NN(C)C2=O)CC(F)(F)C1 N1(C(CNC(N)=O)=O)CCC(C2CCCN(C(c3sccc3C(F)F)=O)C2)C1 Cn1ncc(C(N2CCC(OCCCNC(c3cc(O)no3)=O)CC2)=O)c1N C12(C(N3CC(C)C(NC(C4COC5(CCC5)C4)=O)C3)=O)CCC(CO)(CC1)CC2 C1(C(=O)NCC2(F)CC(CNC(=O)CCF)C2)CN2CCN1CC2 N1(C(COC2CN(S(C)(=O)=O)C2)=O)CCC(N(CC(F)F)CC(N)=O)CC1 C1(NC(=O)CC2CC=CC2)CC2CN(C(=O)Cc3ccnc(F)c3F)CC12 C=CC(CC)CC(=O)N1CCC(C)C(CNC(C23CC4CC2C3C4)=O)C1 Cc1nc(C(N2C(C(=O)N(C3CCC3(C)C)C)CC3CC23)=O)c(C)s1 c1(OCC)cccc(C(=O)NCCC(C)N(C(=O)C2=CCSC2)C)c1O CCC(C(=O)N1CCC(NC(c2cnc(S)n2C2CC2)=O)C(F)C1)C(C)C c1(C(CC)C)nc(N2CC3(CN(C(c4cc5sccc5[nH]4)=O)C3)C2)cc(C)n1 N1(C(c2ncc(C)o2)C(=O)NCC(C)C)CCCC(C)C1CO CC(CS(C)=O)C(=O)N1CC2CC1(CNC(=O)CCSCc1ccccc1)C2 c1(C(N2CC(C)(C(=O)Nc3cnn(C4CC4)c3)C2)=O)cc([N+](=O)[O-])c(Cl)cc1Cl Cc1c(C)c(C)c(C(=O)NC2CCCC(NC(C3CC3C)=O)C2)c(C)c1C N1(C(C2(CC=C)CC2)=O)CCC(NC(=O)C=CCSn2cncn2)CC1 C1(CNC(C=CSC)=O)CCCC(CNC(=O)C(C)n2ccnn2)C1 c1(CC)ncc(CNC(=O)NCC2CN(C(=O)OC(C)(C)C)C2)[nH]1 C(CC(F)(F)F)N(C(=O)CN(C(c1n[nH]c(O)n1)=O)CC1CC1)CC CC1CN(C(C2OCCCO2)=O)CCCN1C(C1CN(C)CCN(C)C1)=O C(C#CC1CCCCC1)N(CCC(=C)Br)C CC(CC(=O)NCc1cncn1C)N(C(=O)CCOC1CCC1)C N1(C(C2(CC=C)CC2)=O)CCC2(CC1)CC(NC(c1cn(C3CC3)nc1C)=O)C2 C1(NC(C2CCCCC2)=O)CCCN(C(=O)C(O)C(F)(F)F)CCC1 C1(NC(c2ccc(Cl)c(-n3nnnc3C3CC3)c2)=O)CCCNC12CCC2 C1(C2CCN(C(C=NOC)=O)C2)CCCN(C(=O)C=Cc2cn[nH]c2)C1 C1(C)(NC(c2cc(SC)oc2)=O)CCCN(C(C2CC3C=CC2O3)=O)C1 CC(C)C(C)C(=O)NCCC1(CNC(=O)C(C)Oc2cccc(F)c2)CC1 c1(CNC(=O)NC2CCCC(N(C)C)C2)nnc2ccccn12 N1(C(N(c2cc(C(=O)OC(C)(C)C)ncc2)C)=O)CCCC2CC12C(=O)O Cc1ccc(C(F)F)c(C(=O)NCC(C)N(C)C(C2CCN(C3CC3)C2=O)=O)c1 c1(C(NCP(OCC)(C)=O)=O)cnc(CNC(=O)CC2CC3(CC3)CO2)nc1O C1(NC(C(n2cc(-c3c(F)ncc(C)c3)nn2)C)=O)CC2(CCCCC2)C1 CC1CCCCC1C(=O)NCCCCNC(=O)CS(=O)(=O)N1CCCC1 Cc1nc(C(=O)NCC(C(C)C)NC(C2(O)CC2(C)C)=O)nn1C C(CC(=O)OC)N(C(=O)C(O)C1CC1)CC=C.C1(C2(C)CC2)C(=O)N1C C=CCCCC(=O)N1CCC(N(CCC)C(c2cnccc2Br)=O)C1 c1(OC)ccc2c(C(=O)NCC3CN(C(c4cc(CO)[nH]n4)=O)C3)ccnc2c1 C(=O)(CC(C(F)(F)F)c1ccon1)NCC(CC)NC(c1nc(C)ccc1F)=O C1(C(N2CC(O)(CN(C(c3cc(CC)on3)=O)C)C2)=O)CC(OC)C(OC)C1 c1(C(=O)NC2CC(NC(C3CC(CC)C3)=O)C2)cc(-c2ccccc2)[nH]n1 N1(C(C(C(CC)C)C)=O)CC2(C1)CN(C(c1cccn3ccnc13)=O)CC2CO C(CC(C)(C)C(=O)NC1(CC(=O)NCC2(C)CCCOC2)CC1)OC N1(C(CCC=CC(C)C)=O)CCC(C(=O)NCC(C)(O)C(C)C)CC1(C)C C(=O)(CCC(CC)CC)NCC(CCC)NC(=O)C(F)CC1CCOCC1 C1(C(=O)NC2CCN(C(Cc3cccc(CC)c3)=O)C2C)OCCN(C)C1=O CCC(O)C(C)(C)C(=O)NCC1(F)CC(NC(c2cccc(SC)c2)=O)C1 c1(CN(CCNC(Cn2ncn(C)c2=O)=O)C2CC2)cnc2nccn2c1 N1(C(C=Cc2cnc(C)s2)=O)CCC(NC(C2CCCC(=O)N2C)=O)C(C)C1 N1(C(CCCC)=O)CCC(C(C)CNC(C2(CC)CC(C)(C)C2)=O)CC1 c1(C(=O)NCC=CCNC(c2c(C)noc2)=O)cncc2n[nH]c(C(C)C)c12 C(=O)(CN1C(=O)Cc2ccccc21)NCC(CC=C)NC(=O)CC1CCCCC1 CN1CC2(CC2)CC1C(=O)NC1(C)CC(C(N2CCC(O)(C(N)=O)C2)=O)C1 c1(N(C)C(=O)O)ccc(F)c(CNC2CCC23CCCC3)c1F c1(NC(C2CCN(Cc3ccc(CO)o3)CC2O)=O)cccc2c(I)n[nH]c12 N1(C(C(=O)N(CC(C)(C2CC2)OC)CC)=O)CC(C)C1 CC1OCCC1CC(N1CC(C)(NC(C2CCC2)=O)C1)=O.C1C(=O)N1 c1(C(=O)NC(CN(C(c2csc(N3CCCCC3)n2)=O)CC)C)cnc(C)[nH]1 C#CC1(NC(=O)NC2CCCCC2CC(F)(F)F)CCC(C)(C)CC1 c1(C(N2C(CN(C(C3C(CC)C3)=O)C)CCCC2)=O)cc2c(=O)[nH]ccn2n1 C1(NC(c2c(C)cnc(F)c2)=O)CN(C(=O)C(CC)CC=C(C)C)C2CCCCC12 Cc1nccnc1C(=O)N(CC(=O)NCC(O)C(F)(F)F)C1CC1 Cc1c(C(N2CCN(CCNC(C3CCCC34CC4)=O)CC2)=O)nnn1C C(CCCCC(=O)N(C(C)CNC(c1scc(Br)c1C)=O)C)SC CC(C)(CF)C(=O)NCCC1CCN(C(c2ncc(C(F)(F)F)s2)=O)C1 C1(C(C(=O)NC2CC2)N(C)Cc2ccncc2F)CC2C(C1)C2(F)F.C1(CN)CC1 c1(C(c2n(CCCSC)nnn2)NCCc2ncccc2C)ccc(Cl)cc1F c1(CNC(C2OCC(C)(C)OC2)=O)ccc2c(c1)CN(C(=O)C(O)C(F)(F)F)C2 C1(NC(c2c(C)[nH]cc2)=O)CCC2(CCNC2=O)CC1 c1(C(=O)NC(CC)CNC(=O)C(C)(O)C2CCC2)noc2cc(Cl)ccc12 C(=O)(CCC(=O)C1CC1)NC1C(NC(C23CC(C(=O)OC)(C2)C3)=O)CCC1 C=C(C)C(CC(=O)NC1CN(C(c2cnc(C)s2)=O)CCC1C)OCC Cc1cc(=NC(=O)CN2CC3C(CNC(=O)CN4CCCNC4=O)C3C2)[nH]o1 N1(C(C2N(C(C(CC#C)C3CC3)=O)CSC2)=O)CCC2CCCC2C1 C1(NC(=O)CN2CC(F)C2)(CF)CCN(C(=O)Cc2cccc(C(F)(F)F)n2)C1 N1(C(C(CCC)OC)=O)CCC2(CC1)CN(C(C1CC(F)C(=O)N1)=O)C2 C1(c2nnnn2CCCOC)(NCC2(CC)COC2)CC2CCC(C2)C1 n1(CCCC(=O)NCC(C)(NC(c2cnc(C3CC3)s2)=O)C2CC2)c(O)nnc1O N1(C(c2c(C#C)cc(Cl)cc2C)=O)CCc2cc(OC)c(S(N)(=O)=O)cc2C1 CCC(C)(C(=O)N1CC(O)(C(C)NC(=O)Cn2ncnn2)C1)OC C(c1ccc(F)c(F)c1)=CC(=O)NCCCC(CCC)NC(c1cc(C)no1)=O C1(C(=O)NC(C2CC2NC(=O)CN(C)C)C)CC12CC(NC1(C)CC1)C2 CC1CC(C(=O)N2CCC23CN(C(C2COCCN2C)=O)C3)=NO1 CCC(C(=O)N1CCC(C2CCCCN2C(=O)CSCC(N)=O)CC1)C(C)C C(=O)(C(CCF)NC(=O)C(C)C(C)C)NCC(=O)OC(=O)OCCCC C1(CC(=O)NC2C(OC)COC2)N(C(=O)CN(c2ccncc2)C)CCC1(C)C CS(=O)(=O)c1ccnc(N2CCC(NS(=O)(=O)CCCCl)C2)n1 C(=O)(C(C)CC(C)CC)N1CCC(CNC(CC=CCC)=O)C12CC2 c1(C(=O)NC(C(C)NC(CCCC=C)=O)CO)cc2occc2n1C N1(C(c2c(C)noc2)=O)CCN(C(=O)CCc2cccnc2Cl)CC1CF C#Cc1ccc(C(N2CCN(C(=O)C(C)N3CCC3)C(CO)C2)=O)cc1 c1(CCC)c(C(=O)N(C)CCNC(c2c(C)coc2CC(=O)OC)=O)cnn1C C(=O)(NNc1c(F)cccc1Br)NC1(C(=O)O)C(C(C)(C)C)CC1 c1(C(=O)NC(CC2CCN(C(c3c(SC)ccs3)=O)CC2)C)cccc(Cl)c1Cl c1(OCC(N2CCC(N(C(c3ncc(C)cn3)=O)C)C2)=O)ccc(C)cc1F N1(C(c2ccc(OC)s2)=O)CCC2CCC(NC(C3CCC4CC4C3)=O)C1C2 N1(C(C(CCC)NC(N)=O)=O)CCOC2(CCC(NC(=O)C(F)(F)CO)CC2)C1 C(=O)(C(O)C(C)(C)C)NC1CCN(C(CC(C)SC)=O)C1 C(=O)(CC(C)C(F)F)NCC(CNC(CNC(c1nccc(OC)n1)=O)=O)(C)O CC1C(=O)CC1C(=O)NCC1CC(NC(=O)CCC2CCCO2)C1 C1(NC(C(C2CC2)NC(CCCCOC)=O)=O)C(O)C2CCCC12 C(N=c1nc2c(ncn2C)c(N(C)Cc2ncc[nH]2)[nH]1)c1cc(C)nc(C)c1 N#Cc1cnn2ccc(N(C(=O)CCCC(F)(F)F)C3CC34CCNCC4)nc12 Cc1cc(C(N2CC(CNC(=O)C=CC(=O)N(C)C)C3(CC3)C2)=O)ccc1F N1(C(c2c(C)nns2)C(=O)NCc2ccc(F)cc2)CCCC2CC1C2(C)C N12CCOC(C1)CCC2.C1(CCC)CC(c2nnnn2CC)(NC2CCCC2)C1 c1(C(C(=O)N(CCC(=O)NCCOCC=C)C)C)ccnn1C C1(O)(C(=O)NCCC2(NC(c3ccn(C)n3)=O)CC2)CCCC(C)(C)C1 C1(CNC(c2cc(C(=O)OC)sn2)=O)CC2COCC2N1C(=O)C=COCC CC1CC(NC(=O)CCCF)CCN1C(C1CC1C(C)(C)O)=O N1(C(c2n(CC)ncn2)=O)CCCC(n2cc(CNC(=O)C(C)CSC)nn2)C1 c1(OC(C)C)cccc(C(=O)NCC(O)CNC(=O)C2=CCCOC2)c1F C(=O)(C1=Cc2cc(Cl)ccc2OC1)N(CC(C)O)CCNC(C12CCC1C2)=O Fc1ccc2c(-c3cnccc3C(=O)Nc3c[nH]c4ncccc34)c[nH]c2c1 CC(C)(C)CC(O)C(=O)N1CC(C)(C)C1C1CCN(C(c2cc[nH]n2)=O)CC1 N1(C(CC2CCC(C)CC2)=O)CC2CN(C(=O)CN(C3CCCC3)C)CC2C1 C1(C(N2CCC(CSC)C2)=O)(NC(=O)C=Cc2ccc[nH]2)CCOCC1 CC(C(=O)NCCC1CC(F)(F)CN1C(c1cn(C)nc1Cl)=O)C(C)(C)C c1(C(C)(C)C(=O)NCC2CC(NC(c3cncn3C3CC3)=O)C2)ccc(Cl)nc1 c1(CC)nc(C)c(C(=O)NCC2(O)CN(C(c3ccc(CC4CC4)o3)=O)C2)s1 C(=O)(C1CCCn2nccc21)NC1CC(C(=O)Nc2ccc(O)c(=O)cc2)OCC1 C(CC(C(=O)N(CC(CO)(CO)NC(C12CCCCC1C2)=O)C)N(C)C)SC N1(C(CC=CCCCCC)=O)CCN(C(c2ccc(F)cc2)=O)C(CC)C1 C1(NC(CCNC(C2CCN(CC)C2)=O)=O)C2CC3C(C2)C13 N1(C(C=CCCC)=O)CC(CNC(=O)CC2CC2)C(O)C1 CC1CC1(F)C(=O)NC1CC(NC(=O)CNC(N)=O)C1 c1(OCC)cc(Br)c(CN2CC3CC2CN3C(=O)CC2NC(=O)NC2=O)cc1OC N1(C(CC2CCC(N)C2)=O)CCCC(N2CC3CC3C2)C1 C#Cc1c[nH]nc1C(N1CCC(OCC(=O)NCCSC2CC2)C1)=O c1(C(C)(C)C)n[nH]c(=NC2CC(CCNC(=O)CCc3c(F)cccc3F)C2)s1 c1(C(N2CCC(CC(=O)NCCc3scc(CC)n3)C2)=O)cn(C)nc1C1CC1 C1(C)(C(=O)NC(CN(C)C)C)CCCC1NC(=O)C(C#N)N(C)C(=O)OC(C)(C)C N1(C(c2cc(C)ns2)=O)CC(C)CN(C(C2(N(C)C)CCCC2)=O)CC1C N1(C(C(C)Oc2ccccn2)=O)CCC(NC(=O)C=CC2CCCC2)CC1 C1(NC2CCN(CC(=O)OC)C2=O)CCN(C(=O)C=Cc2cncn2C)C(C)C1 C1(NC(=O)C=C2CCC2)CN(C(=O)COc2ccc(F)nc2)CC1n1ccnn1 N1(C(c2nccc(OC)c2)=O)CCN(C(=O)Cc2ccc(F)cc2)CC1C(C)C C1(C(=O)NN2CCCC2)C2CC3C(C2N)C13.c1(C(C(=O)C2CC2)=O)ccc(S)o1 N1(C(C2N(C)CC(O)C2)=O)CCC(C2CCN(C(=O)C=CBr)C2)C1 N1(C(c2c(OCC=C)cccn2)=O)CCN(C(=O)COC2CCCC2)C(CO)C1 c1(CCC(=O)OC)ccc(CNC2CN(C(=O)COC3COC3)CC2C)cc1 O=S(=O)(c1ccn(CC(F)F)n1)N1C2CCC1CC(CN1CCC1)C2 c1(C(=O)NC(C)C(C)NC(c2cccn2C2CC2)=O)ncn(-c2nc[nH]n2)n1 CC(C(=O)NCCCN(C)C(c1cn(C)nc1-c1ccccc1)=O)P(C)(C)=O N1(C(C(C)Oc2ccc(F)cc2)=O)CCN(C(=O)CCCF)C(C)C1 N1(C(c2ccc(CO)o2)=O)CCC2C(CCCN2C(=O)CC(F)F)C1 C1(O)(CN(C(c2cc(C)nn2C)=O)C)CCN(C(C2CCCCC2F)=O)CC1 N1(C(C(CCC)C)=O)CCC2C(CCCN2C(c2ccc(C#N)cc2)=O)C1 C1(C(N2C(C#C)CCC2)=O)CC2CC1CC2NC(c1cnc(C)o1)=O C(=O)(CC(C)C(F)F)NCC1(CCCNC(C2C(OC)C2)=O)CCCC1 O=C(CS(=O)(=O)C1CCCC1)NCCCCCNC(C12CCCN(CC1)C2)=O c1(C(=O)NCC(C)N(C(=O)C(C)NC(C2CCC2)=O)C)nnn2c1COCC2 C1(NC(C(C)C)=O)CCCCC1NC(=O)CN(C1CCSCC1)C N1(C(C=CCOC)=O)CC2(CCN(C(=O)C(c3ccc(O)cc3)=O)C2)C1 c1(C(=O)NCC2CN(C(CC3CC(=C)C3)=O)C3C2C3)ccc(C(C)C)c(F)c1 Cc1cccc(C(=O)NC2(CO)CCCN(C(C3CCCN3C3CC3)=O)C2)c1O N1(C(Cn2ccc(C)cc2=O)=O)CCN(C(c2cnc(O)cc2C)=O)CCC1C C1(C(N(C(C)C)CCNC(=O)C=C2CCC(C)C2)=O)CCc2ccccc2C1 CC1(C)COC(C(=O)NCC(=O)NC2C=CCCC2)C1 C1(C(=O)NCC)CCCN1C(c1nc(C(C)(C)C)co1)C(=O)NCC(C)C c1(C(N)=O)ccc(NC(=O)C(=O)Nc2ccnc(Br)c2)cn1 N1(C(=O)NCC(C)C(=O)OCOC)CC2CCOC2C1.c1(SC)ccccc1 c1(CC(=O)NC2CN(C(c3n(CCC)ncc3)=O)C(C)C2)c(OC)cccc1C c1(CNC(C2C(NC(c3cc(C)cc(CO)c3)=O)C2)=O)c(Br)cc(F)c(Cl)c1F Cn1nc(C(=O)NCC(C2CCCCC2)NC(C2CC2C(F)F)=O)c(Cl)c1Cl C=CCCC(CC(C)C)C(=O)N(C)CCN(C)C(c1cn(C)nc1O)=O C#Cc1cccc(C(=O)NCC2CC2CNC(=O)C=Cc2ccc(Cl)cc2)c1C N1(C(c2ccc(S)cc2)=O)CC2CC1CN2Cc1c(Cl)cccc1Cl C1(C(N2CCC(N(C(=O)CCc3ccc(Cl)s3)C)C2)=O)CCCC12CCC2 CC1(C)OCC(CC(=O)NCC2CN(C(c3cscn3)=O)CCO2)O1 C(=O)(C1=CCCCC1)N1CCC(CC)C1C(=O)NCC1CCN1C(=O)OC(C)(C)C C1(NC(C[SH](c2ccccc2)C)=O)CN(C(=O)C(c2cncn2C)N(C)C)CC1O c1(C(=O)NC(CC2CN(C(C3(C#C)CC3)=O)C2)C)ccnc(O)c1 C1(C(=O)NCCCC2(NC(C(C)C3CCCC3)=O)CC2)CCC(C)CC1 c1(C(=O)NCC2(O)CCN(C(C(C)(C3CC3)NC(C)=O)=O)C2)cccc(F)c1C N#Cc1ccc(CNc2cccc(Cl)c2-n2nccn2)nc1 c1(NC(c2cccc(OC)c2OC)CC)nc(=NCC2CC2)[nH]c2cccnc12 C1(CCNC(c2c(Br)n[nH]c2C)c2n(CC)nnn2)CC2C=CC1C2 C1(NC(CC(CC)CC)=O)(CN(C(=O)C(C)N(C)C)C)CCC(C)(C)CC1 N1(C(CC=C(C)C)=O)CCCC2(NC(=O)CN(C)S(N)(=O)=O)CCCC12 C12(C(N(CCC(C)(C)C)C)=O)CCN(C(c3cc(Cl)n(C)n3)=O)CCC1C2 C=CCC(Cc1ccccc1)C(=O)NC(C)(CNC(=O)CCCC(C)=O)CC N1(C(C2CCN(CCC)CC2)=O)CCN(C(=O)C2=CCCC2)C(CO)C1 C1(NC(c2c(CC)ccc(F)c2)=O)CCC2(CCCN2C(c2coc(Cl)n2)=O)CC1 N1(C(CC(C)CF)=O)CCN(C(=O)C=Cc2c(F)ccc(Cl)c2F)CC2(CC2)C1 Cc1cc(C(F)(F)F)c(C#N)c(NCC2CCCN2C(=O)C2=NNC(=O)C2)n1 CC1(C)CCC(C(N2CCC(C)(CNC(C3(CC(F)F)CCC3)=O)C2)=O)OC1 N1(C(CCN(CCCO)C(C2C(CC)CC2)=O)=O)CCC(F)(F)C(C)C1 N1(C(c2cc(C)sc2Cl)=O)CCCC(NC(=O)C(C)CC2CCC2)C1C C1(C(=O)NCCOCCNC(C2CC(F)C2)=O)CCCC2CCCN12 c1(C(=O)NC2C3(CO)C4CC2CC34)cccc2ccnn12.C12(CC(CC)C1)C(=O)N2 C1(NC(COCCC)=O)CCC(N(C)C(c2cc(C3CCCC3)no2)=O)C1 Cn1c(C(=O)NCCCCCCNC(C2C(C(F)F)C2(C)C)=O)cnc1Cl N1(CC(=O)NC(=O)NC2CC2)C2CCC1CC(NC(c1cccc(F)c1Cl)=O)C2 [N-]=[N+]=Nc1ccc(Cl)cc1NC(c1ccc(OCCF)cc1)=O Cc1nn2cc(CC(N3CCCC(CNC(c4oncc4C)=O)CC3)=O)nc2s1 Cc1ccc(F)c(C(N2CCC(N(c3cc(F)ncn3)C)CC2)=O)c1Cl C1(C(C)NC(CSCC(C)=O)=O)CCN(C(=O)Cc2nc(O)n[nH]2)C1 N1(C(C(=O)NCC(F)F)=O)CCCC2(CCN(C(c3cscc3F)=O)C2)C1 CCC(CC)CC(=O)NC1CC2(C1)CN(C(=O)CC(C)SC)C2 CCCC(CCC)CC(=O)N1CC=C(C(=O)N2CC(O)(C(F)(F)F)C2)C1 C1(OC)CN(C(C2CCCC2)=O)CC1NC(c1cnoc1C1CCC1)=O c1(NC(CCNc2cnc3sc(C)c(C)n32)C)ncnc2cc(F)c(F)cc12 c1(C(N2CCC(Cc3cn(C4CC4)nn3)C2)=O)cnc2ccccc2c1 N1(C(C(N2C(c3cnc(C)[nH]3)CCC2)=O)=O)CCN(C(=O)C(C)OCC2CC2)CC1 c1(C(=O)NCCCC(=O)NC2CC2NC(=O)C(F)F)cccc(Br)n1 C1(CCC(C)C)CCN(C(C2CCCN2C(=O)CCOC2CC2)=O)CC1 CCC(CCC(=O)N1C2CCC1(CNC(=O)C(CC1CC1)OC)CC2)OC CC1(NC(C2CN(S(N)(=O)=O)C2)=O)CCN(C(C2CCCC2C(F)(F)F)=O)CC1 c1(C(N2CCC(F)(CNC(c3coc(Cl)c3)=O)C2)=O)coc2ccc(Cl)cc12 C1(C)(OC)CC(NC(C2(O)CCN(C(c3ccnn3C)=O)CC2)=O)C1(C)C C(COC(C)(C)C)(C(=O)NNC=O)N(CC(C)C)CC.Cc1ccccc1 c1(COCC(N2C(C3CCN(C(=O)C=C(Cl)Cl)C3)CCC2)=O)ccc(F)cc1 c1(OC)ccc(C(N2CCOC(CN(C)C(C3(CO)CC3)=O)C2)=O)nc1N N1(Cc2c(C)[nH]c(C(=O)OCC)c2C)CCC2(CCC(C)(O)CC2)C1 C(=O)(CCC(F)(F)F)N1CC(C)CC(C(=O)NCc2c(C)nc[nH]2)C1 N1(C(C(COC)C)=O)CCC(C2CCC2)(CNC(c2nnc(S)n2C)=O)CC1 N1(C(C(CCC)O)=O)CCN(C(C2(F)CCOCC2)=O)CC1CC C(c1nc(CNC(CC(C)C)c2nnnn2C2CC(F)(F)C2)co1)=C(C)C N1(C(c2[nH]cc(C(N)=O)c2)=O)CCOCCC1C(=O)NCCC1COCCO1 Cc1cc(S(=O)(=O)N2CCCC(C)(C(N3CCOC(C)C3)=O)C2)ccc1Br CP(C)(=O)CCC(=O)NCCn1cc(CNC(C2CC3CCC2O3)=O)nn1 C1(CC(=O)NC2(C(=O)NCCS(=O)(=O)NC)CCC2)CC(O)C1(C)C N1(C(C2(C=C)CC2)=O)CCC(CN(C(=O)C=C(C)CN2CCCCCC2)C)CC1 N1(C(c2c(N)n(CCO)nc2)=O)CCN(C(=O)CC=C(Cl)Cl)C2CCCCC2C1 C1(CN(C(=O)CC2CC3C=CC2C3)CC)CCCCN1C(=O)C(C)C1CC1 C1(OCC)CC2CN(C(=O)C(CC(C)C)NC(=O)CC3(C#N)CC3)CC12 C1(N(C(C2(CCOC)CC2)=O)C)CCN(C(=O)C=C2CCC(C)C2)CC1 C(C(=O)NC1CC1C(=O)N(CC1=CCCOC1)C)(C(C)C)NC(CC(C)C)=O c1(C(=O)NC(CCOCC)CNC(C2(CC)CCCCO2)=O)cc(C)ccc1O N1(C(c2c(NC)ccc(F)c2)=O)CCC2CC1CN(C(=O)CCC=C(C)C)C2 C1(NC(C2C=CCCC2)=O)CCC2(CC1)CN(C(=O)COCCF)C2 c1(C(=O)NCC2CCN(C(C(C)NC(C)=O)=O)C2)sc2nc(C)nc(C)c2c1C C1(NC(C2N(C(Cn3ncc(C)c3)=O)CC=CC2)=O)CN(C)CCC1O N1(C(C2CC2(F)Cl)=O)CCCOC(c2cn(-c3ccccc3Cl)nn2)C1 S(=O)(=O)(CC(=O)C1CC1CN)N1C(C2CCC(C)C2)CCC1 C1(C(N2C3C(NC(=O)CC4CCS(=O)(=O)C4)C(C3)C2)=O)CC12CCOCC2 C=CC1CCCCN1C(=O)COC1CC(NC(c2ccccc2CSC)=O)C1 C=CC(C)C(C)C(=O)N1CC2(NC(c3cnc(OC)cn3)=O)CC1C2 c1(C(N2CC(COC)N(C(c3nccn3C)=O)CC2)=O)ccc2c(c1)COCO2 C(=O)(CC(C)P(C)(C)=O)NC(CCCNC(CN(C)CC)=O)C c1(C(=O)NCC(C)(C)CNC(=O)C(CC(F)F)C2CCC2)ccc(N)cc1F CC(F)(F)CCCC(=O)NCC1CC(NC(=O)C(F)(F)c2ccccn2)CC1O C1(CNC(C2(C)C(C(=O)OC)CC2)=O)CN(C(c2nccn2C(C)C)=O)CCO1 O=C(N=c1ccn(C2CC2)[nH]1)c1ccnc(NCc2ccc(I)c(F)c2)c1 c1(CC(=O)N(C)CC2(NC(c3ccnnc3)=O)CC2)nc(F)c(F)cc1F C1(C(=O)NCC2(F)CN(C(C3(OC)CCOCC3)=O)C2)C2Cc3ccccc3C12 C1(NC(c2cc(CC)on2)=O)CCN(c2ncc3c(n2)COC3)C12CCC2 N1(CCCC)CC2CCC1C(NC(=O)C(C)Oc1ccc(OC)cc1)C2 CS(=O)(=O)c1cccc(-n2nc(CN3CCCC3=O)nc2CCCn2ccnn2)c1 N1(C(c2nc(C(C)C)oc2)=O)CC(C2CN(C(C3SC4C=CC3C4)=O)C2)C1 CC(C(=O)N1CCC(O)(CNC(C2CCC3(CCC3)C2)=O)CC1)C1=CCCC1 Cc1nn(C(C)C(=O)N(C(C)CS(C)(=O)=O)C)c(C)c1[N+](=O)[O-] C1(CCC)COCCN1C(c1cccnc1OC(F)F)=O C1(C(=O)NC2C(NC(c3ccc(F)c(Cl)c3F)=O)C2)CCc2cc(F)ccc2O1 C1(CCC)CCc2nc(NC(=O)Nc3cc(F)cc(Cl)c3)sc2C1 c1(NC(CN(C(=O)C(C)CF)CC(C)C)=O)cccc(CNC(N)=O)c1 CCC(C)(CNC(=O)CCC1CCCC1NC(=O)CCOC1CCC1)C(N)=O C12N(CC13CCCC3)C(=O)C1C(C(C)C)CN(C1)C2=O.C(C=C(Cl)Cl)N(C)C c1(CC(=O)NC(C)CCN(C)C(C2(Cl)CC2)=O)csc2ccccc12 C1(N(C(=O)CNC(=O)CNC(N)=O)C)CN(C(c2ccoc2)=O)CC1(F)F Cn1ncc(C(N2CC(O)(CNC(=O)CCNS(=O)(=O)CCCl)C2)=O)c1F N1(C(c2c(C)scc2)=O)CCC2CN(C(c3cnc4n3CCS4)=O)C2C1 c1(CC(=O)N(CCNC(=O)CC2COCCN2CC)CC)nc2c([nH]1)CCCC2 c1(C(N(C(CNC(c2cnc(C)nc2C)=O)C)C)=O)scc2c1OCCO2 c1(C(=O)NC(C2CCCN(C(c3cn(C)cn3)=O)C2)C)cccc2ncnc(O)c12 CC1(C)CC(NC(C2CC3CC2C2CC32)=O)CN(C(c2ccnc(Cl)c2)=O)C1 c1(C(=O)NC(CNC(c2ccc(COC)s2)=O)CO)ccc2ccccc2c1O O=C(C1=CCCS1)NC1CCN(C(=O)C(O)CC2CCOCC2)CC1 C(=O)(C1Cc2ccc(C)cc21)NCC1N(C(CCNC(=O)OCC)=O)CCOC1 c1(C(=O)NC2CC(CNC(CN(C)CC)=O)C2(C)C)cc(S(N)(=O)=O)oc1C c1(C(N2C(C)C(C(=O)NC3(C4CCCC4)CC3)CCC2)=O)cn(C)c(=O)n1C c1(C2(Cc3cccc(-c4n(CCCC(C)C)ccn4)c3)CC2)cccc(Cl)c1Cl C1(CC(=O)NC(CCSC)C)C2CCC(C2)N1C(c1ncccc1CO)=O c1(C(=O)NCC2C(NC(c3c(SC)csc3)=O)C2)cc2c(nc1O)CCCCC2 c1(OCC(N2C(CNC(CSCCC)=O)C=CC2)=O)ccc(F)cc1O C1(CNC(=O)C=C(Cl)Cl)CCCC(CNC(c2snc(O)c2Cl)=O)C1 CC1CC(C(=O)N2CCC(NC(c3cc(C4CC4)ns3)=O)C2(C)C)=NO1 c1(C(=O)NC2CCN(C(c3ccon3)=O)C2)cnn2cc[nH]c12 c1(C(=O)NCCC(C)NC(C2(C(F)(F)F)CC=CCO2)=O)cc(F)c(F)cc1N C1(NC(C(C)NC(CC)=O)=O)C2CCN(C(=O)CN3CCCCC3=O)C12 CC1CCN(C(c2c[nH]ccc2=N)=O)CCN1C(C1(C2CCCCO2)CC1)=O N1(C(CCC=CCC=C)=O)CC(C)CCC1CNC(c1cc(C)sc1C)=O c1(NC(C2CC(NC(c3c(C)nn(C)c3)=O)C2)=O)cccc(Cl)c1C c1(C(=O)NC(c2ccco2)CO)ccc(-c2ccccc2F)cc1 C1(C(=O)NC2CCCCO2)(C(N2CCN(CCO)CC2)=O)CC2(CC2)C1 Cc1cc(C(F)F)nn1CC(=O)NC(CNC(c1ccc(C(N)=O)[nH]1)=O)CC(C)C C1(NC(C2CC2)OC)CCCN(C2CC2)CC1 CCC(C(=O)N(C)CC=CC(=O)NCC1(CC(C)C)CC1)C(C)C n1(C(CC(=O)NC2C(c3onc(C)n3)C2(C)C)C)cnc2ccccc12 c1(NC)cnn(C(=O)OC2(C)CN(C(C(N3CC(CO)C3)=O)=O)C2)c1.C1CO1 O=C(N=c1[nH]oc2ncccc12)C1CC(C(=O)NCc2cc(Br)cnc2F)C1 c1(N2CCN(C)CC2)ccc2c(c1)CCN(C(c1ccnn1C(C)(C)C)=O)C2 C1(CNC(CCn2c(C)cc(C)n2)=O)CCCCCN1C(=O)Cc1ncc(C)o1 N1(C(C2(OC)CCCC2)=O)CC2C(NC(C3CCCC3C)=O)C2C1 c1(C(=O)NC(C2CN(C(C=C(C)C)=O)C2)C)nn(C)c(C(F)(F)F)c1Cl c1(NC=O)nc(CC(=O)N(C2CCN(C(C3(CCF)CC3)=O)C2)CCO)cs1 C#CC1(C(=O)NCCCCC(=O)OC)CCN(C(=O)CC23CCCC2C3)C1.C=O C1(NC(=O)CCOC2CCCOC2)CCCC(CNC(=O)CCC2CCCC2)C1 C(C(C)(C(=O)N1CC(C)(NC(=O)Cc2ccn(C3CCCC3)n2)C1)OC)OC N1(C(C(C)(C)C#N)=O)Cc2ccc(CNC(=O)C(CO)c3ccccc3)cc2C1 CCCCC(C(=O)N1CCCC(CO)CC1)NC(c1cc(=N)[nH][nH]1)=O CN=c1nc(C(N2CCC(O)C(NC(c3cc(C4CC4)on3)=O)C2)=O)cc(C)[nH]1 C(=O)(CCCCC(=O)N(C1CCCCC1)CCNC(C1CCCOC1)=O)N(C)C c1(C(=O)NCC2C(C)CCN2C(c2cc3sccc3[nH]2)=O)cn2cnnc2cn1 c1(C(=O)NCC2C(CNC(=O)C=Cc3cn[nH]c3)C2)ncc2n1CCCC2 C(=O)(CCCCCC#N)NC(C(C)NC(c1cc(C)nc(C)n1)=O)CO Cc1nc(N(C)C)sc1C(=O)NC1CCCN(C(=O)COC(F)F)C1 C1(NC(Cn2c(C)cc(C)n2)C2CC2)CC12CCN(C(=O)CC13CCCC1C3)C2 N1(C(C)=O)CCCC(C(N2CCN(C(=O)C(C)(C)Oc3ccccc3)CC2)=O)C1 N1(C(C2C=CCN(C(c3n(CCC)ncc3)=O)C2)=O)CCOC2CN(C)CC12 S(=O)(=O)(c1ccc(C2CC2)o1)N(C)C.C12CN(C(=O)C=C(Cl)Cl)CCC1N2 C12(C(N(CC(CC)NC(=O)COc3cccc(Cl)c3)C)=O)CCN(CC1)CC2 O=C(C(F)C(F)(F)C(F)(F)F)NCCC1(O)CCN(C(=O)COc2ccsn2)C1 N1(C(C(C)OC)=O)CCC2(CNC(=O)C(O)C(C)(C)C)CCCCC12 C=C(Cl)CCC(=O)NC1(C(=O)N(CCN2CC=CC2)CC)CC(CO)C1 c1(OC)ccc(C)c(C(=O)NC(C)(CNC(=O)C(C2CC2)C2CC2)C2CCC2)c1 c1(C(N2CC(CNC(C3(F)CCOC3)=O)OCC2)=O)cccc2occc12 CCCCC(CC)CC(=O)NC1CCCN(C(=O)COCc2ccccn2)CC1 C1(CCCNC(=O)CC2CSC2)CN(C(=O)C(F)(F)Cc2ccccc2)CCO1 c1(C(=O)NCC2C(NC(c3nc(CCCCC)sc3)=O)C2)cc(CCC)oc1C C12(C(=O)Nc3ccc(CC)s3)C(NC(=O)CC3CCCC4CC34)C3CC1C2C3 C(N=c1nc(N2CC3CCC3C2)c2c([nH]1)CCC2)C1(C)CCCC1 c1(CCC=C)ccccc1C(N1CC2CC1CO2)C(=O)NCSc1ccc(Br)cc1 CCCC(C)(O)C(=O)NCCOCCOCCNC(=O)C(c1cnn(C)c1)SC C(CCCC(=O)N1CC(O)CC1CNC(C1C2CCN1CC2)=O)NC(N)=O C1(N(C(Cn2ncc(CC)c2)=O)C)CCCC2CN(C(c3scnc3C)=O)CC12 Cc1c(Br)cc(C(=O)NCC2C3CN(C(c4cn[nH]c4)=O)CC23)c(=O)n1C CCCCCCN1CCOCC1.N12CCCC1N(CCCCCOC(C)(C)C)C2=O C(=O)(CC(C)C(C)(C)NC(N1CC(=O)NC(=O)C1C)=O)OC N1(C(CCC(C)=O)=O)CCC2(CC1)CN(C(c1cnn(C)n1)=O)CCO2 C(=O)(CS(=O)CC)N1CC(C(=O)NCc2ncco2)(CC)C1 c1(CNC(CC2C(C)C2)=O)ccc(CNC(C2CCCOCC2)=O)cc1 N1(C(c2n(CC)ncc2Cl)=O)CCCC(O)(CN(C(=O)C(O)CN(C)C)C)C1 O=C(C#CC1CCC1)N1CC(NC(C23CCCCC2C3)=O)C1 N1(C(C2(CC)CN(C(=O)CN(C)C(C)C)C2)=O)CC2(CCOC(=O)N2)C1 C(CCC(=O)NC1(C(=O)NOCCF)CCSC1)OCCOC C1(C(N(CCCCNC(Cc2cc(C)no2)=O)C)=O)CCCC(CF)C1 N1(C(CC2(OC)CC2)=O)CCC(O)(C(C)NC(=O)Cc2cc(C3CC3)no2)CC1 c1(C(N2CCC23CN(C(c2ccncn2)=O)C3)=O)cnc(Cl)cc1Cl c1(C(N2CC(NC(c3cc(C)n(C)n3)=O)C(F)C2)=O)ccc2c(n1)NC(=O)CC2 Cc1ccc2ncc(C(N3CCC4CN(C(c5cnn(C)n5)=O)CCC34)=O)n2c1 N1(C(=O)C(F)OC(F)(F)F)CC2(C(=O)NCC3CCCSC3)CC1CO2 c1(C(=O)NC2CCC(NC(=O)CSc3ccccc3Cl)C2)cccc2nncn12 CCC(CC)CCC(=O)NC1CCC1NC(C1(Br)CC1)=O Cc1ccc(C(=O)NCC2CCCCC2NC(C2OCCCO2)=O)c(Br)c1 c1(CC(=O)NC2CC(NC(C3CCC=CCCC3)=O)C2)ccc2cnccc2c1 C(=O)(CCC(=O)NC)NCC(CC)NC(c1c[nH]nc1C(C)(C)C)=O c1(C(N(C)CCNC(=O)C=CBr)=O)cc(C(C)(C)C)n(C)n1 N1(C(c2ccc(OCC#C)cc2)=O)CCC(N(C)C(c2ccsc2)=O)C(C)C1 N1(C(C2(CC(=O)OC(C)(C)C)CCC2)=O)CCCC(NC(=O)C=CI)C1 C(=O)(CC(C(F)F)NC(=O)C#CC(C)(C)O)N(CC(C)(C)CCO)C1CC1 C1(C(N2CC(OC)(CNC(=O)C(C)CC(F)F)C2)=O)CC2CCC(C1)C2O c1(C(N2CCC(CCNC(c3c(CC)n(CC)nc3)=O)C2)=O)cc2n(n1)CCO2 C1(NC(c2ncc(C)c(Br)c2)=O)CCC2(C1)CN(C(C1CNC(=O)C1)=O)C2 C=CCCCCCCCCC(=O)NC(CNC(C1CCCN1N=O)=O)CCCC c12cc(ncc1Br)CNC2=O.c1(CC(=O)OC)cc(CN)on1 N1(C(C(=O)OC)=O)CCN(CC(O)CC(F)(F)F)CC1C(F)F c1(C(=O)NC(C)CCCc2ccc(O)cc2)cnc2cccnn12 N1(C(c2cnc(Cl)c(Br)c2)=O)CCN(Cc2ccc(OC(F)(F)F)cc2)C2CC12 c1(C(=O)OC)cc(C(=O)NC(CC(=O)CC2CC2(Cl)Cl)(C)C)co1 N1(C(C2CCC(C(C)C)CC2)=O)C2CCC1CN(C(C1(C)CC3CC3C1)=O)CC2 C1(CNC(=O)CSCC2CCCCO2)COCCN1C(=O)C1=CSCS1 C(=O)(C(CCC(C)C)NC(c1ncccc1F)=O)NCc1nc(C)sc1C c1(C(=O)NC(C2CCN(C(C3(S(C)(=O)=O)CC3)=O)CC2)C)cccc(C#N)c1 C1(CC)CCCC1(C)C(=O)NCCC1(O)CN(C(=O)CC2COCC(C)O2)C1 N1(C(C(=O)Nc2cccc(C)c2)=O)CCC12CN(C(=O)C(C)CC#N)C2 c1(C(=O)NCC2C(CNC(c3ncncc3F)=O)C2)c(F)cccc1Br c1(C(=O)NC2CCN(C(c3nc(CC)sc3N)=O)CC2)cccc2nnn(C)c12 c1(CC2CN(Cc3cc(C(=O)OCC)n[nH]3)C2)cccc(F)c1.C1(C(C)N)CCCC1 C1(O)(CN(C)C(C2(c3cccs3)CC2)=O)CN(C(C2CC(C)(C)C2)=O)C1 N1(CC)CCOC(C(=O)NCC(CC2CC2)C(=O)NC(c2nnnn2C)C)C1 C1(NC(c2c(C)oc(CNC(=O)C(C)CC3CCC3)n2)=O)CCCCC1(C)C C1(C(N2CCC(C3N(C(c4cnc(C(C)(C)C)o4)=O)CCC3)C2)=O)CCCC12CC2 N1(C(C2(NC(CCCOC(C)C)=O)CCOCC2)=O)CCOC2CCOCC12 FCCN=C(NCc1c(C2CC2)cccc1F)NC1CC2CCC1O2 c1(OC)cccc(C2CCCC2NC(c2cccc(I)c2)C)c1 Cc1cc(C(=O)NC2(C)CC(NC(=O)CC34CCC(CC3)CC4)C2)nc(C)c1 c1(CN(c2ccc(-c3ccc(CC)cc3)nc2)CC)ccc2ncccc2c1.CCl c1(NC)cnc(Cl)cc1C(=O)NCC1COCCN1C(=O)CCCn1ccnc1 C12(C(N3CCC(COC)(CNC(c4ccnnc4)=O)C3)=O)CCC(C)(CC1)OC2 C1(C(N2C(CC#N)CN(C(=O)C(O)CCl)CC2)=O)CCC2CNCCC2C1 CCCC(C(=O)NCC1CC(NC(=O)C(C)(C)CF)C1)NC(=O)OC(C)(C)C c1(C(N2CC(CNC(CCC)=O)C(C(F)(F)F)C2)=O)c(S(C)(=O)=O)cnn1C C1(CNC(C2CC2Sc2ccccc2)=O)CN(C(=O)CC2(C)CC2)CCO1 CCC(F)(F)CC(=O)NCC1CCN(Cc2ccnn2C)CC1O c1(CCC)cc(C(=O)NCC2(CNC(=O)CCC(C)N(C)C)CC2)cc(O)n1 N1(C(CN(C(CSCC=C)=O)C)=O)CC(F)(F)C(F)(F)C1 c1(C(N2CCCC(NC(C(CCC)(C)C)=O)C(F)C2)=O)cc2c(nc1N)CCC2 C(CCCCCNC(c1cc(C(F)F)[nH]n1)=O)N(C(CC1CCC(C)O1)=O)C C#Cc1ccc(C(=O)NCCC2(C(N3CCC(N(C)CC)C3)=O)CC2)c(C)c1 N12CCC(C)(C)C1C2=O.c1(CNC(c2onc(COC)n2)=O)ccc(OC)nc1 N1(CC(=O)NC(C)CC2CC(NC(=O)C(c3ccc(Cl)nc3)(C)C)C2)CC(=O)NC1=O N1(C(c2cc(C)oc2C)=O)CCC2(CC(NC(c3sc(C)c(C)c3C)=O)C2)C1 CCCCC(C)CCC(=O)N1CC2CC1CN(C(c1cnn(CCC)c1)=O)C2 C1(NC(C(C)N(C)C)=O)C(C)CCN(C(c2cc3ncccc3[nH]2)=O)C1C c1(OC)cc(OC)cc(C(N2CC(NC(c3nocc3Br)=O)C(C)C2)=O)c1 c1(C(N2C(CNC(CC)=O)C(CC)CC2)=O)cc(Cl)cnc1O N1(C(c2c(C)cc(F)s2)=O)CCC(CO)(NC(c2ccc(O)nc2)=O)CC1 N1(C(C2C(CC)N(C)CC2)=O)CC2CCCC(CNC(c3cc(Cl)no3)=O)C2C1 c1(N2CC(C(=O)NC(C#C)C)OCC2)nc(C)nc2ccsc12 C#Cc1ccc(C(=O)NCC(C(C)(C)C)NC(C2(CC)CC2)=O)o1 C1(C(N2CC(C(C(=O)O)OC)C2)=O)CC(=O)N(c2cccc(C(F)(F)F)c2)C1 C(=O)(CCCCCCCC(=O)N(CCCNC(=O)CC1(C)CCCCC1)C)OC C(=O)(C#CC1(C)CCCO1)NCC1(C)CCCN(C(c2nnc(O)nc2O)=O)C1 C(=O)(C(=O)C=Cc1cccs1)NCC(C)N(C)C(c1ccnn1C)=O C1(C(N(CC=C)CC=C)=O)CCC(n2cc(C3CCN(C)C3)nn2)C1 c1(CC(=O)NCC(=O)OC)ccccc1Br.c1(C(=O)NC2CC2N)cn[nH]c1 C1(CC)CN(C(C2CCC2)=O)CCN1C(C1CC(C(F)(F)F)(OC)C1)=O CC1CC(C(N2CCOCC(CNC(C34CCC(CC3)C4)=O)C2)=O)CC(C)C1 C#Cc1cncc(C(=O)NC2CC3CC(NC(=O)CSC(F)F)C3C2)c1.C(C)(=O)O c1(CC(N2CCC(N(C(=O)C(F)n3cccn3)C)CC2)=O)cnn2c1CCCC2 N#Cc1cc(NC(C2CC23CCN(C(c2ccnc(O)c2)=O)CC3)=O)ccc1O c1(C(=O)NCC(CO)NC(CC(CCC)CCC)=O)c(C)ccc2ncccc12 C1(C(=O)NCCN(C(COC(C)=O)=O)C2CC2)Cc2cc(C)ccc2O1 c1(C(N2CC(CC(=O)NCCC(C)CO)OCC2)=O)ccc(C#N)cn1 CCC(CC(=O)NCC(C)(C)CN(C)C(C1(CO)CCCO1)=O)c1ccccc1 O=C(CCSC)N1CCCc2c(Br)cnn21.C1CCCC1 C1(CC)C2Cc3ccc(Cl)cc3C12.c1(OCC)cncc(C(=O)NCCOCC)c1 c1(C(=O)NC2(CO)CCSCC2)ccc(S(=O)(=O)NC2CC(C(N)=O)C2)c(Cl)c1 C(=O)(CC(C)(C)C(=O)NCc1ccoc1C(N1CC2COC(=O)C2C1)=O)OCC c1(C(N(CCCNC(C2CC2Cl)=O)C)=O)cccnc1-c1ccccc1 N=c1[nH]c2ncc(C(=O)NC(c3cccc(Cl)c3)CNC(C3COC3)=O)cc2s1 Cc1ccc(OCC(=O)NCC2(O)CCN(C(C3(C)CC=CC3)=O)C2)c(F)c1 N1(C(Cc2cc(C)[nH]n2)=O)CCC(NC(=O)C(C)(C)CCF)C(O)C1 C1(CNC(C2C(C(=O)OC)C2)=O)CC2(CC2)CN1C(c1cc(C2CC2)no1)=O CC1(C)CC2(CN(C(C3CN(C(C4CCC4(F)F)=O)C(C)(C)C3)=O)C2)C1 S(=O)(=O)(c1ccc(NC2CCC(C)C2)cc1Br)N1CCC(C(C)C)CC1 Cc1c(CC(=O)NCCNC(C2CC3CCC2CC3)=O)nc(Br)n1C Cc1nc2c(C(=O)NCCCCNC(C34CC3C4)=O)cccc2o1 c1(CNCCC(C)N(C)C)cc(Br)ccc1Br C1(NC(C=CC)=O)CCC12CCN(C(c1c(F)ccc(Br)c1F)=O)CC2 c1(CNC(c2cccc(NC3CN(C(=O)OC)C3)c2)=O)cc(Cl)ccc1I N#CCC(C(F)(F)F)NC(=O)NC1(C(=O)N(C)C)CCCC1 c1(NC(CN(CCC)C)=O)c[nH]c2cc(C)ccc12.c12ccc(cc1)OC2 N1(C(CCC=CC(C)C)=O)CCC2(CC1)C(N(C(=O)CC(C)(F)F)C)CS2(=O)=O CC1CN(C(C2(C(F)(F)F)CCCC2)=O)CCN1C(=O)C(C)C1CCC1 Cc1cnc(CNC2CCCCC2C(=O)Nc2ncc(Br)cc2C(F)F)cc1Br N1(C(C(CC)(F)F)=O)CCC(CNC(=O)Cc2ccc(C)o2)C(C)C1 N(C(=NCCCCl)NC(c1cc(F)cc(Br)c1)COC)CC(C)(CO)OC c1(C(C(=O)NC(CC)C)N(CCCO)C2CC2)cn(C2CCC2)nc1C Nc1cccn(CC(=O)N(c2cccc(F)c2)C2CCC2)c1=O Cc1[nH]cc(C(=O)NC2CCCCC2NC(=O)CCC(N)=O)c(=O)c1Cl c1ccc(Br)cc1.C1CCON(C)N1C.C(C)(C)(C)OC=O N1(C(C2(COC)CC2)=O)CC(C2CCCCN(C(=O)CC3CCCO3)C2)C1 c1(CC)cc(C)ccc1C(=O)N(CCCNC(=O)Cc1nonc1C)CC c1(C(N(CC(C)NC(=O)CC2CSC2)CC)=O)snnc1C(C)C c1(C(C2CCN(C(=O)C(=O)NOCC(C)O)CC2)C)cc(C)nc(C)c1 c1(C(c2n(CC(=C)C)nnn2)NCCc2ccc(Cl)s2)ccc(OCCC)nc1 C#CCCN=C(NCC(CC)C1CC1)N1CC(OCCSC(C)(C)C)C(OCCS)C1.CC CCC(C)C(CNC(=O)C(C)(C)C1CCN(C(=O)Cn2ncn(C)c2=O)C1)CO c1(OCC)cc(C(N2CSCC2C(=O)Nc2ccsc2C)=O)on1 c1(C(N2C(CN(C(=O)C(F)C(C)C)CC)CCC2)=O)cnc(COC)nc1C N1(C(C(=O)NCCc2ccc(OCC)cc2)=O)CCN(C(=O)COC)C(C)C1C c1(-c2cn(C3CCC(C(=O)NCCCCN(C)C)C3)nn2)cn(C)nc1CC1CC1 C1(O)(C(C)NC(C(c2ccc(Cl)cc2)CC)=O)CCN(C(C2(OC)CCC2)=O)C1 c1(CCC(=O)NC(C)CC2CN(C(=O)CCC3CC3(Cl)Cl)C2)cn(C)cn1 C=C(C)CC(C)C(=O)NC1(CC=C)CCN(C(c2cccc(CO)c2)=O)C1 N1(C(c2cncc(CC)c2)=O)CCN(C(C2CC(=C3CC3)C2)=O)C(COC)C1 C=CCC(C(=O)N1CCC1CNC(c1cnc(CC)[nH]1)=O)NC(C)=O C1(C)COCCN1CC(F)F.n1(C2C(C(=O)NCCO)C2)cc(CS)nn1 Cc1cc(C(=O)NCCc2n[nH]cc2C(=O)NC(C)CCC2CC2)ncc1N CC(C)CC(C)CC(=O)NC1C2CC1N(C(=O)CCn1ncn(C)c1=O)C2 c1(C(N2CCC(NC(C=NOC)=O)C2)=O)ccc(C)c(F)c1 C1(NC(CSCC(N)=O)=O)COCC1CNC(=O)COCC1CCCOC1 N1(CC)CCOCC1C(=O)NCC(CNC(c1c[nH]nc1)=O)OC.C(C)(=O)OC Cc1cccc(O)c1C(N1CC2(CCC2NC(c2cnn(C)c2)=O)C1)=O CC(CCC(=O)N1CCC(c2cc[nH]n2)C1)NC(=O)CC1CC(F)(F)C1 c1(CNC(C(C)Oc2ccccc2Cl)=O)cncc2n[nH]cc12 c1(NC(C)C)ccc(C(=O)NCCCCCNC(=O)CC2(O)CCC2)cn1 n1(CC(=O)NC(CCNC(C(C(CC)O)(C)C)=O)C)ccc(=O)c([N+](=O)[O-])c1 c1(OC)ccc(NC(=O)Cc2ccccc2NC(C)=O)cc1S(N)(=O)=O N1(C(C(CC2CCC2)OC)=O)CC(N(C)C(c2cc[nH]c2)=O)C(C)(C)C1 c1(C(C(=O)NCC)N(C(C#C)C2CCC2)C)cc(Cl)c(Cl)s1 c1(CNC(C2CCOC(c3ccccc3)O2)=O)sccc1SC1CC1 CN1CCN(C(=O)CCC2CC2(F)F)CC1CNC(=O)C(O)CF C(=O)(CC(CNC=O)CC(C)C)N(C1CCCN(C(=O)CNC=O)C1)CC C1(F)(CNC(=O)CS(=O)(=O)Cc2cccs2)COCCN(C(=O)CC(F)(F)F)C1 N1(CCN(CC(CNC)O)CC(O)CC)CCOCC1.C1C(=O)N1 N1(C(CC2(NC(C)=O)CC2)=O)CC2CC1CN(C(C1CN=C3N=CNN3C1)=O)C2 N1(C(CC2C(C)C2)=O)CC(C2CCN(C(C3(O)CCCCC3)=O)CC2)C1 C1(CC)CN(c2nnc(CC(C)C)n2C2CC2CS(C)(=O)=O)CCS1 N1(C(c2n(C(C)C)ncc2)=O)C(CNC(=O)CNC(N)=O)CC2COCC12 Cc1nn(C)cc1C(O)C(=O)NCCCNC(=O)CC1CCCCN1C C1(NC(=O)Cc2cccc(Cl)c2)CN(C(=O)CCn2cncn2)CC12CC2 C1(CC)(NC(c2ncn(C)c2C)=O)CCCN(C(=O)CC2(O)CCCOC2)C1 C(CCS(=O)(=O)NC(=O)CC1CCCN1c1nccc(C(F)F)n1)OC c1(OCC)ccc(Cl)c(C(=O)NC2CCCN(C(=O)CC(C)F)C2)c1F Cc1cnn2cc(C(N3CCCC4(NC(=O)CC5CC=CC5)CC4C3)=O)cnc12 C(=O)(N1CCC(C(N)=O)O1)n1ccc(CC)n1.C1=C(C)CNC1=O C(CCS(C)(=O)=O)(C(=O)OC(C)(C)C)NC(=O)OCC(CCO)C(F)(F)F c1(C(CNS(CC(C2CCCC2)OC)(=O)=O)=O)ccc2c(c1)CCC(=O)N2 C(=O)(CCCC(=O)N(C)C)N1CCC(C(C)CN(C(=O)C(C)CC2CC2)C)CC1 c1(CC(=O)NC2CCN(C(=O)C=Cc3cc[nH]c3)C2)nccc2ccccc12 C1(OC)CC(CNC(=O)CNC(=O)CCC(C)C)N(C(c2nc(C)nn2C)=O)C1 N1(C(c2scc(C)c2)=O)CCC2(CC1)CCN(C(=O)C(=O)C(C)C)CC2 C1(NC(C2(C=C)CC2)=O)CC2CCC1C(NC(=O)C(C)Cc1cccc(Cl)c1)C2 c1(C(=O)NCCOCC(=O)NCC(N2CCOCC2)C)cc(CCO)on1 C1(C(=O)NC2(CC(=O)NCCC3CCOCC3)CC2)CCC2CC12 N1(C(c2c(C)cn(C)c2)=O)CCC(C)C(NC(c2ccncc2Cl)=O)C1C c1(OC)nc(C(F)(F)F)c(C(=O)N(C2CCN(C(=O)OC(C)(C)C)C2)C)s1 C(CCCCC(=O)N(C1CCCN(C(C2(C)CC=CC2)=O)CC1)CC)OC N1(C(CNC=O)=O)CCC(C2CCN(C(c3coc(O)n3)=O)C2)C1 Cc1cc2occ(CN(N3CC(O)(CN)C3)C)c2cc1C.C1(C=O)CC1F Cc1cc2ccccc2nc1C(=O)NC1CN(C(=O)C(C)c2cc[nH]n2)CC1C C(C)(CNC(=O)C(=Cc1ccccc1)C)(C(C)C)NC(CCCNC(C)=O)=O N1(C(CCC(=O)NCCC)=O)CCOCC(C)(CNC(=O)C(C)c2ccsc2)C1 N1(C(C(CNC(C(CC)C(=O)OC)=O)C)=O)CCc2cncnc2C1 Cc1cc(C(=O)NC2C=CCCC3CC23)sc1-c1ccc(F)cc1 N1(C(c2cc(C)ns2)=O)CC(NC(=O)C=C2CCCCC2)C(F)C1 c1(C(c2nnnn2CSc2ccccc2)NC(C)CCCO)nnc2n1CCC2 C1(C(=O)NCCOC2CN(C(CN(CCC)C)=O)C2)CC2(C1)CC(F)C2 C1(CC(=O)N(CCC)C2CC2)CN(C(c2[nH]ccc2COC)=O)CCC1C C(C)(CCC(=O)NC(C)(CNC(=O)COCC(=O)OC(C)(C)C)CO)SC C1(CN(C)C(c2ccc(Br)nc2)=O)CN(C(C2CC2C2CC2)=O)CCO1 C1(NC(C2CCCC(C(N)=O)C2)=O)(CO)CCN(C(c2ccc(Cl)s2)=O)CC1 C1(C(N2CCC(C(C)C(=O)NCC(C)(C)C3CCCC3)C2)=O)CCC(F)CC1 c1(NC(C(C2CC(NC(c3c(C)cncc3)=O)C2)F)=O)ccc(F)c(F)c1 S(=O)(=O)(c1cc(F)cc(F)c1)N(C1CC2CCC1N2C(=O)OCCSC)C.C(C)(C)(C)O C(=O)(CC(O)CCC)NC1(CC=C)CCN(C(=O)Nc2ccccc2F)C1 N1(C(C2CCN(CCC#C)CC2)=O)CCC(C)N(C(=O)Cc2cccnc2)CC1 O(NC(=O)C(C(C)O)N(C)C)C(C(=O)NC(C1CCCCC1)CC)CC(C)C C(N=c1nc(O)c2cnn(C)c2[nH]1)C1(F)CC(NC(c2c(C)onc2C2CC2)=O)C1 c1(NC(c2nc(NC(C3(COC)CC3)=O)sc2)=O)cc(Br)ccc1F C(=O)(CC(CNC(C1CSC(C)=N1)=O)C1CCC1)NC(C)C C1(CC=C)(NC(C2CCCC2O)=O)CCCN(C(C2CCC3(C2)N=N3)=O)C1 C(=O)(CCCCCN(C(C1CCC1)=O)C1CC1)N(C)CCc1ncon1 c1(C(=O)NC(CCCCNC(CCC=C=C)=O)C)ccn(CC)c(=O)c1 C1(C(=O)Nc2c(C)cc(F)cc2Br)CCc2ccccc2N1 c1(C(=O)NCC2CCCN(C(C(C(C=C)C)C)=O)C2)cc(N(C)C)cc(C#N)c1 C1(CNC(c2c(CC)[nH]nc2Cl)=O)CN(C(c2cccnc2)=O)C2CCCC2O1 c1(C(=O)NC2CCC(N(C(=O)COC3CC=CC3)C)C2)cnc2c(F)cccn12 c1(CSC(C)C)ccc(C(=O)NC(C)C(C)NC(C2(C)CS(=O)(=O)C2)=O)cc1 c1(CC(=O)C(=O)N2CC(c3cnc(-c4ccncc4F)cn3)C2)ccccc1F CCCC(C#N)C(=O)NC1CC(C(=O)NC2CCCCCC2F)C1 C(CC(=O)NC(C1CCC1)CO)N(C(=O)CCC1CCCC1)CC#C C1(C(=O)NCCCC=CC)C2CC2CN1C(=O)CC1CCCCCC1 c1(CC)oc2ccccc2c1CC(=O)NCC(C)(C)NC(=O)CC(C)CC c1(CC(=O)NC2C(NC(C(C3CC3)SC)=O)COCC2)cc(C)cc(F)c1 N1(C(C2CC(=C)C2)=O)CC(NC(=O)COCCCC)CC1C c1(C(=O)OC)cnc(N2CCN(C(=O)C(c3cnn(C)c3)O)CC2C)nc1C c1(CC(=O)NC2C3(CCCN(C(C(CSC)OC)=O)C3)C2)n[nH]c2ccccc12 c1(C(C(=O)NC(C)C)NCCS(=O)(=O)NC)ccc2c(c1)OCO2 C1(C(N2CCC(CNC(=O)C(c3cccn3C)=O)C2)=O)(NC(C)=O)CC(F)(F)C1 N1(C(C(C)Sc2ccccn2)=O)C2CCC1C(NC(=O)CCc1ccc(Cl)s1)C2 c1(C(C)=O)c(C)[nH]c(C(N2CCN(C(C3(C(N)=O)CCC3)=O)CC2CO)=O)c1C Cc1cnc(C)c(C(=O)N(C)CC2CN(C(c3cc(C(C)C)on3)=O)CCO2)c1 C1(C(N2C(CNC(C(C)=C3CCCC3)=O)CC(O)C2)=O)CC12CCSCC2 Cc1n[nH]c(C)c1CC(=O)NC1(CNC(C2CC23CC3)=O)CCOC1 C1(CN(C(c2c(C)n[nH]c2)=O)C)CCCN(C(C2(Cl)CC2(C)C)=O)C1 c1(CNC(C2OCCN(C(c3ccc(C)o3)=O)C2)=O)ccc(Cl)c(Cl)c1 Cc1ccc(F)cc1CCNC(=O)COc1cccc(F)c1 C(CC(=O)NCCC1CCC(C)(C)CO1)(C(N)=O)NC(C)=O c1(C(=O)NC2CCN(C(CCN3CC(=O)NCC3)=O)CC2)occ2c1CCCC2 CN1C(=O)NCC12CN(C(C1CN(C(C3(C)COCCO3)=O)CC13CCC3)=O)C2 C(=O)(CCCC(=O)NCC(C)(C)CN(C(=O)Cc1cc(Cl)ccc1OC)C)NC C1(NC(C(C)O)=O)CCOC12CCN(C(=O)Cc1cncn1C1CC1)CC2 C1(CNC(C(CC)OC)=O)Cc2ccccc2CN1C(c1cn(CC)cn1)=O c1(C(=O)NCC(=O)NC(C2CCOCC2)C2CC2)ccc(C2CCCN2)o1 C1(CC)CN(C(=O)C=CCN(C)CC)CCC1CNC(C1CCCC1O)=O C1(NC(c2c(Cl)cn(C)n2)=O)CN(C(=O)CC2CCCC2(F)F)CCC1CO C(=O)(C(C(C)(C)C)NC(=O)C=CC1CCN(C(c2cccc(=O)o2)=O)CC1)NC C#Cc1cnc(C(=O)NC(C)(CNC(=O)Cc2nncn2C)CC)c(C)c1 N1(C(CCN(C(CC(C)SC)=O)C2CC2)=O)CCCC2(C1)N=N2 Cc1noc(C)c1C(C)(C)C(=O)OCCn1ccnc1C CC1(C)CCNC(C(=O)NCc2cccc(C#N)c2)C1 c1(-c2c(C(N)=O)cccn2)ccc2c(c1)CN(C(C1CC(O)CN1)=O)CC2 c1(OC)nc(C)ncc1C(=O)NCC1C2CC1N(C(C1CCCC(C)(C)C1)=O)C2 N1(C(CCCCNC(C)=O)=O)CCCC(NC(=O)CC2CCC(=O)N2)C1C N1(C(c2c(C)nc(C)[nH]2)=O)CCC2(CC1)CCN(C(C1CC3(C1)CC3(F)F)=O)C2 n1(CC)ccc(C(=O)NC2CCC(C)(NC(=O)CN3CCC(O)CC3)C2)c1C c1(CNCC2(O)CN(C(C(C)C(C)n3cccn3)=O)C2)cc(S(N)(=O)=O)cs1 c1(N2CCC(C)(CC(C)C)CC2)nc2ccc(Cl)cc2c(=NCCCOC2CC2)[nH]1 Cc1ccn(CC(N2CC(NC(C3CN(S(C)(=O)=O)C3)=O)CC2CO)=O)c(=O)c1 C1(C(=O)NCC(c2ccccc2)O)CC(F)CN1C(c1cccc(O)c1)=O N1(c2nc(SC)nc(C)c2)CC2CC(NC(c3ncc(Cl)s3)=O)CC2C1 C12(NC(CC(=C)C)=O)CCOCC1CN(C(C1(CCOC)CCCC1)=O)C2 O(NC(=O)C(CNC(=O)C(C)C=C)CCC)CC(=O)OCC Cc1nc2ncnn2cc1C(=O)NCCOC1CN(C(c2cc(O)ccc2F)=O)C1 c1(C(N(C2CCN(c3nnc(C(F)F)s3)C2)CC)=O)ccc(C)nc1Cl c1(SCC(=O)OCC(NOCC(c2ccc(C)cc2)C)=O)ccc2ncnn2c1 N(C(=NCCCc1nccs1)NCCC1CCOC1)C1CCCN(CC)C1 C(C)(C(=O)NC1CCCN(C(c2oc(C3CC3)nc2C)=O)C1)(C(C)C)OC CCCS(=O)(=O)CC(=O)NC(C1CCN(Cc2occc2C(=O)O)C12CCC2)=O c1(C(C(=O)NC(CC(C)NC(C2N(CC)CCC2)=O)C)F)ccc(F)cc1 n1(CC=C)nnnc1C(c1cc(C(=O)N(C)C)no1)NCC(C)COC C(=O)(C(O)CC(F)(F)F)NC1C(SC)CN(C(c2ccnnc2)=O)C1 C1(N(C(C(CC)F)=O)CCO)CCN(C(c2cc(C3CCOCC3)on2)=O)CC1 C1(COC)(CNC(=O)CC2CCN2C(=O)CC2(C#N)CC2)CCCCO1 c1(CC)ccnc(NC(c2noc(=O)n2C)c2nnnn2CC2CCCO2)c1 C=CCC(C)(O)C(=O)NC1CCC(CC(=O)NC2CCC3CC23)C1 c1(C2(C(N(CCNC(c3nc(OCC)oc3)=O)C)=O)CCC2)ccccc1F N1(C(Cc2nc(C)oc2)=O)CC(NC(C2CC3(CCO2)CC3)=O)C2(CC2)C1 C1(CCC)CCC(CN(c2cc(O)ncn2)CCNC(C)=O)CC1 C(=O)(C1COc2ccc(Cl)cc21)NCCC(C)NC(CS(CCC)(=O)=O)=O N1(C(=O)OCC)CCC(C(=O)NC2CCCC(NC(C3(CNC)CC3)=O)C2)CC1.SC c1(NCCC(CC)OC)[nH]c(=NC2CC2c2cnn(C)c2)nc2c1ncn2CC C(=O)(C1=COCC1)NCC(CCOC)NC(=O)C(C)SCc1ccccc1F C1(CCNC(CSc2cn(C)nc2)=O)CCN(C(=O)CC#N)CCC1(F)F c1(C(C2CC2)NC(CN2CC(C)C=C(C)C2)=O)ccc([N+](=O)[O-])cc1 O=C(C(O)C1=CCCCC1)NCCC(F)Cn1cc(C2CCCC2)nn1 CCC(C)(C)C(O)C(=O)NCCC(O)CNC(C1CC2(CCC2)C1)=O N1(C(C2(CC)CCOCC2)=O)CC(NC(=O)C(CO)OC)C2(CC2)C1 C(C(O)CC(C)(C)CO)N(C=O)CC1CCC(C#C)CC1 c1(C(=O)NCC2(O)CC(NC(CC(CC)C3CC3)=O)C2)cnc2cnccc2c1 c1(C(=O)NC2CCCN(C(c3c(Cl)ncc(N)c3)=O)C2)ccc(O)c([N+](=O)[O-])c1 Cc1nn(C)c(C)c1C(=O)NCC1(CC(N2CCCC(C#N)C2)=O)CC1 O(NC(=O)C(C(C)CC)NC(=O)C(CC(C)C)OC)CCCC=C N12CCC(C(F)C1)NC(=O)CSc1c(cccc1)CC2=O.CCCCSCC CC1C(NC(C2(CF)CCC2)=O)CCN1C(C1CCN1Cc1ccccc1)=O C(=O)(C1=CC(C)(CC)C1)NC1(CNC(C2C(CCCC)CCC2)=O)CC1 CCCCC(CO)NC(=O)CCN(C(=O)CC1CCC(=O)C1)C1CC1 c1(C(=O)NCC(CNC(C(C(=O)OC)C)=O)(C)O)ccc2c(c1)NC(=O)C2 N1(C(C(C)OC)=O)C2CCC1CC(NC(=O)C(F)(F)CCn1ccnn1)C2 c1(C(=O)NC(C)C(C)NC(=O)CNS(N)(=O)=O)coc(-c2cccnc2)n1 C1(C(N2CCC(CC)C2)=O)(CNC(c2ccn(C)c2)=O)CC2(CC2)C1 N1(C(C#C)Cc2ccc(F)cc2)CCC(O)(C(=O)NC(C)C(=O)O)CC1 c1(C2(C(=O)Nc3ccc(CC)cn3)CC2)ccccc1C#N N1(C(CCCC#CC)=O)CCC2C(CCCN2C(c2cc(Cl)cc(F)c2F)=O)C1 Cc1cc2c(CC(=O)NCC(F)CNC(=O)Cn3cc(C(F)F)cn3)csc2s1 C1(OCC(C)OC(C)(C)C)CCN(Cc2cc(C)[nH]n2)C1(C)C C(=O)(C1=NNC(=O)CC1)NC1CC(NC(C(C)NC(C)=O)=O)C1 C(c1cccc(O)c1)=CC(N1CCC(CCCNC(CCC#C)=O)CC1)=O C1(C(N2CC(CC(C)NC(C3(CC)CCC3)=O)C2)=O)CCOCC12CCC2 C(CCCCNC(c1ccoc1)=O)NC(C(C)NS(CC)(=O)=O)=O c1(OC)cccc(C(C)CC(=O)NCC(C(C)(C)C)NC(=O)C2=CCCS2)c1 C(=O)(C(C#N)C)NC(C)(C)CNC(C1C(C(=O)NC(C)(C)C)C1)=O.C1(C(=O)O)CC1 c1(NC2CCC(CCC)CC2)ncccc1S(=O)(=O)N1CC(OC)C2(CC2)C1 C1(C(N(CC(COC)C)C)=O)CN(C(C2CN(C)CCN2C)=O)CC12CCC2 c1(CCC(N2CC3C(NC(C(N)=O)=O)C3C2)=O)ccc(OC(F)(F)F)cc1Br c1(C(=O)NCCCN(C(c2csc(CSC)n2)=O)CC)nccc2nn[nH]c12 C1(NC(=O)CCc2ncc[nH]2)CC2CCCC(C1)N2C(c1ncncc1Cl)=O C(=O)(CC(F)(F)Br)NCCOCCN(C(=O)C=CC=C(Cl)Cl)C C1(C)(NC(CC2CCC(NC(Cn3nnc(C)n3)=O)C2)=O)CCSCC1 C1(NC(CC=CCC)=O)CCC2(CC1)CCN(C(c1cc(OC)n[nH]1)=O)CC2 N1(C(C=NOC)=O)CC=C(CNC(=O)CCc2csc(C)n2)CC1 c1(C(N(CC(C)N(C)C(c2cnc(O)o2)=O)C)=O)n[nH]c2c1CS(=O)(=O)CC2 C1(C)(NC(C=CCOC)=O)CCCN(C(C2CC(C)CCCO2)=O)C1 c1(C(=O)NC(C(C)C)C(C2CCCCC2)NC(C2CCC2)=O)ncc(F)cc1F C1(C(=O)NC2CCN(C(C(c3ccc(F)cc3)=O)=O)C2)CCC12CCOCC2 c1(C(=O)NC2CC(F)(CNC(CCOCCN(C)C)=O)C2)c(F)cccc1F N1(C(CSC)=O)CC(F)CC1CNC(=O)C=C(Cl)Cl c1(NC(C2C3(CC(NC(c4c(C)[nH]c(C)c4C)=O)C3)C2)=O)ccc2c(c1)CCC2 c1(C(N(CC(=O)N(CCCC#C)C)CC2CC2)=O)cc(C)nc(O)n1 c1(C(N2CC(C)CN(C(C3CC3F)=O)CC2)=O)ccn2cc(Br)cc2c1 C1(C(N(C)CCNC(c2cnsn2)=O)=O)CCC(c2nc[nH]n2)CC1 O=C(C1=NOCC1)NC1CN(C(c2ncsc2-c2ccccn2)=O)CC1O CC1CN(c2ccnc(N3CCOC(C4CCCC4)C3)n2)Cc2cccc(Br)c21 C(C(C)CN=c1[nH]c(=NC2COC3(CCC3)C2)[nH]c2cc(C)ccc12)NC(=O)OC C12(CC(=O)NC3(CNC(CC4C(C)(C)C4)=O)CCOCC3)CCCCC1C2(F)F c1(NC(C(=O)Nc2cccc(CS(C(C)C)(=O)=O)c2)=O)cc(F)c(F)cc1I C1(CNC(C(=O)NCC)=O)CCC(C(=O)N(C)CCC)CC1 C1(C(=O)NC(CC)C(F)(F)F)CC(N=[N+]=[N-])CN1C(c1coc(CO)c1)=O C#Cc1ccc(C(N2CCC=CC2C(=O)Nc2cnn(C(C)C)c2)=O)cc1 C1(C(=O)NCC2C(CNC(COc3cn(C)nc3)=O)C2)C(F)(F)C12CCC2 C=CC1(C(=O)NCCn2cncn2)CCN(C(c2cn(CCO)nn2)=O)C1 C1(NCc2ccc(CC(C)C)cc2)CCS(=O)(=O)CC1 Cc1cc(C)c(C(=O)NC2CC2CNC(=O)C(C)Cc2ccco2)s1 C(CO)(CCCCNC(=O)C(C)(C)F)NC(c1cccc(SCC)c1)=O N1(C(c2c(CC)nn(C)c2)=O)CCC(C)(C)C1CC(=O)NCC(C)C(C)(C)C C12(C(=O)NCC(CNC(CCn3c(C)ncc3)=O)O)CCOC(C)(C1)C2 c1(C(=O)NCC(CC)NC(c2cnn(C(C)C)c2F)=O)oc(C(F)F)cc1C C(CC(C)C(=O)NCC1C(O)C(O)CN1C(c1ccnc(C2CC2)n1)=O)=CC c1(COC)ccc(C(=O)N(CC(O)CN(C)CC#N)C)s1 c1(C(=O)NC2C(NC(C(CC)CC)=O)CCOC2)ccc2c(c1)NC(=O)CN2C N1(C(CC(CC2CC2)NC(CCN(CCC)C)=O)=O)CCCC(C)CC1 N1(C(C(F)=CC)=O)CC(NC(=O)Cc2cccc(C)c2)CC(C)C1 Cc1cc(C(N2CCC(C(C)NC(c3cscn3)=O)CC2)=O)cc(Br)c1C C1(CC)CC(C)(C)CN1c1ccccc1.C12CC(CN1C(=O)COC)OC2=O C1(NC(C2CC(C)(NC(Cc3cc(C)[nH]n3)=O)C2)=O)CC(CO)C12CCC2 CC(=O)CC(C)(C)CC(=O)N1CCC2(CCC(NC(=O)CCC(=O)N(C)C)C2)C1 C#CC1(C)CCCN(C(C2CCCN(C(=O)CCCCC3CC3)C2)=O)C1 c1(C(=O)NC2C(NC(COCP(C)(C)=O)=O)COCC2)cnc(O)c2ccccc12 Cc1cnn(C)c1S(=O)(=O)NC1(CF)CCN(C(=O)OC(C)(C)C)C1 c1(NC(c2c(CNC(c3scc(C)c3Cl)=O)ccs2)=O)cc(Br)c(O)cc1Br c1(C(N2CC(OC)C(NC(C34COCC3C4)=O)CC2)=O)cccc2nn[nH]c12 CC(C)C(CC(=O)NCC12CCC(CC1)N(C(c1cnc(S)[nH]1)=O)C2)C(C)C CCCC(CC)CCC(=O)N1CCCN(C(=O)C(c2ccc(O)cc2)=O)C(C)C1 C1(N(C(C(C)NC(=O)NC)=O)C2CC2)COC2(C1)CN(C(C1CC1C(C)O)=O)C2 c1(CNC2CC(C(=O)NC3CCCC(C)C3)C2)ccc(F)c(Br)c1F c1(NC2CCN(C(c3cccs3)=O)CC2)nc(Cl)nc2sccc12 C1(NC(CCCCC)=O)CC2(C1)CC(CNC(C1(C(=O)N(C)C(C)C)CC1)=O)C2 CN1CC=C(CC(=O)NCCn2cc(-c3ccc(Br)cc3)nn2)CC1 C(=O)(C(CC)C(C)C)N(CCCC(=O)N(CC=C)CC1CC1)C(C)C Cc1cc(C(=O)NC(CNC(c2cc(CF)on2)=O)C(C)(C)C)[nH]c1C n1(C(=O)N(CCO)C2CC2)ncn2nccc2c1=O CC1CCN(CC(N2CC(SCC(=O)N(CCNS(=O)(=O)C3CC3)C)C2)=O)CC1 N1(C(CC(=C)C)=O)CCCC(CNC(=O)Cc2cn(CCC)nc2C)C1 c1(OC)ccc2c(c1)CC(=O)N(CCC(C)=O)CCC(=O)N2NC(C)C c1(OC)cc(C(=O)N(CCCNC(C2(c3ccccc3C)CC2)=O)C)c(F)cn1 C(C(C(=O)NCc1cn(C2CC2)cn1)NC(=O)CC1CC1)OC Cc1ccc(N(C)CCCC(N)CC2CCCO2)cc1 C(=O)(CS(=O)(=O)C(C)C)NC1CCN(C(Cc2ncc(C)s2)=O)C1(C)C C=CCC(C(=O)N1CC(C)C1C(=O)NC(C)C(C)C)OC C(=O)(C(C(C)(C)C)N(C)C)NCC(CNC(c1nn(C)c(F)c1)=O)(C)F CC1=C(C(=O)NCC#CCNC(c2ccc(C)c(N(C)C)c2)=O)CCCO1 C(=O)(C(CO)C(C)(C)C)NC(CCC)CCCNC(c1cc(C)c(Cl)s1)=O Cc1nc(NC2CC2)sc1C(=O)NCC1(NC(=O)C(F)n2cccn2)CCC1 c1(NC2(C3CN(C(C4(CC)CCC4)=O)C3)CC2)nc(C)nc(O)c1C c1(C(N(CCNC(=O)C(F)(F)C2CCCCC2)CC)=O)ccc2c(c1)C=CCC2 C(=O)(CCC#Cc1ccccc1)N1CC(C)C(NC(C2(C3CCC3)CCC2)=O)C1 CC(C)C(CCN(C)C(C1CC1(F)F)=O)NC(c1c(Cl)cnn1C1CCCC1)=O C1(C(=O)NCCN2C(C)CC2)CC(C)N1C(=O)C=Cc1cc[nH]n1 N1(C(c2c(Cl)cc(C)s2)=O)CCOC(C(=O)NCCOCC(F)F)CC1 NS(=O)(=O)CCC(=O)NC1CN(C(=O)Cn2nnc(-c3ccco3)n2)CC1O C1(C(=O)NC(C2CCOC2)CC)CN(C(=O)Cc2csnc2C)CC12CC2 c1(C(C)=O)ccsc1C(=O)NCCC(C)NC(=O)C(c1ccccn1)C c1(CC(=O)NC(C2CCCN(C(C=CSC)=O)C2)C)cc2ccccc2c(=O)o1 C1(NC(COCC(C)C)=O)CCSC12CN(C(=O)C=Cc1ccccc1C#N)C2 c1(C(=O)Nc2ncc(-c3cncc(CO)c3)s2)nc(Cl)ccc1[N+](=O)[O-] N1(C(CNC(CC(C)C)=O)=O)CC(F)CC1CN(C(=O)CC1CC2CC2C1)C CC1(NC(c2ccnc(C3CC3)c2)=O)CCC(NC(C2CC(=C3CCC3)C2)=O)CC1 C1(NC(c2ccc(C#C)cc2C)=O)CCC2(CC1)CC(NC(C1CC1OC)=O)C2 c1(C(C)OC)nc(C(=O)NCC(O)CCNC(=O)C=CC2CC2)cs1 n1(CC(=O)NC(CCOCC)C)cc(CNC(=O)COCC2CC2)nn1 C1(NC(CCC(CC)NC(C2CC=C(C)CC2)=O)=O)CCCCC1N=[N+]=[N-] C1(C(N(CC(C)NC(CSCCC)=O)C)=O)CC2(C1)CC(C)(C)C2 C(=O)(CC(C)CC(=O)NCc1cc(C(N2CCCC(C(N)=O)C2)=O)no1)OC C(N=c1[nH]c(SC)ncc1Br)C1CCCCN(C(C(COCC)N=[N+]=[N-])=O)C1 C(CCCCCCn1cc(-c2cn(C)cn2)nn1)NC(C(C)c1ccco1)=O c1(C(N(C)CC2(CNC(C(CN(C)C)O)=O)CC2)=O)ccccc1F C12(C(=O)NCC3C(C)CN(C(=O)CCC=CBr)C3)CCCCN1CCC2 c1(C(N(C(C)C(=O)NCc2ccc(O)nn2)C)=O)ccnc2cc[nH]c12 N1(C(C(C)OCCC(C)C)=O)CCN(C(=O)C=CC2CCCO2)CC(C)(C)C1 C1(C(=O)NCC2(F)CC(NC(c3c(OC)n[nH]c3)=O)C2)CN=C2N=CNN2C1 N#Cc1ccc(CNc2cn(-c3cc(C(=O)O)ccn3)nn2)cn1 C(=O)(CS(=O)(=O)C1CC1)N1C(CCCNC(c2c(C(N)=O)nccn2)=O)CCC1 c1(C(N(CCC(=O)N(C(C(=O)OCC)C)C)C2CC2)=O)cnc(N)cn1 c1(C(N(CC(=O)NCC(C2CCC2)NC(c2ccoc2)=O)C)=O)cc(F)cc(F)c1 c1(C(=O)NCC2CC(NC(C3(C(F)F)CC(=C)C3)=O)C2)cccc(C=C(F)F)c1 N1(CC(C)NC2C3CC4C(C3=O)C24)CCN(C(C)C)CCC1C C1(CC=C)(C(=O)N(C2CN(C(C3(SCC)CC3)=O)C2)CCC)CCOC1 C(CCC(C)(C)C(=O)NC(CN1CCCC1)CC)NC(c1ccc(CC)[nH]1)=O N1(C(CCC(CC)OC)=O)CCCC12CCN(C(c1cnn(C)n1)=O)C2 C1(C(=O)OC)CS(=O)(=NC(=O)CC(C)Cc2ccc(Br)cc2)C(C)CO1 N1(c2cc(C)nc(NCC(C)(F)F)n2)C(C)C2CCCCC2C1C N1(C(=O)CN2CCCS2(=O)=O)CC2C3CCC(C2C1)N(CCn1cccn1)C3 C(C(=O)N1CC2C(NC(=O)CCOC3COC3)C2C1)(C(C)(C)C)N(C)C C1(C)(C(N2CC(C#C)C(OC)C2)=O)CN(O)C(C)(C)C1.C1(C(=O)CC)C2CC3C(C2)C13 c1(C(N2CCC(C)(NC(=O)CCCC3CCCCC3)C2)=O)ncc(Cl)nc1Cl N1(C(C=CC)=O)CCn2c(CNC(C3(C)CNC(=O)C3)=O)nnc2C1 C(=O)(CCS(=O)(=O)C(F)(F)F)N1CCCC(C2CN(C(CC(C)C(F)F)=O)C2)C1 C1(CS(C)(=O)=O)(N(C)C(=O)Nc2ccnc(OC(F)(F)F)c2)CC(F)(F)C1 C1(C(N2C(CNC(CCC)=O)CC(C)(C)C2)=O)Cc2ccccc2N1S(C)(=O)=O C1(c2nnnn2C2CCC2)(NC(N2CCOCC2)c2cnc[nH]2)CC2CC2C1 C(C)(C)(CCCC(=O)NC1CC(CO)C1)NC(CC1N(C)CCC1)=O CN(CCCC(=O)NCC1(O)CCN(C(C2(C3CCC3)CC2(F)F)=O)C1)N=O N1(C(C(CC)C)=O)CC2(CCN(C(C3(c4cccc(C)c4)CCC3)=O)CC2)C1 C1(CC=C)(C(=O)NCC(O)CC)CCCN1C(c1cn[nH]c1)=O c1(C(N2CC(NC(COCC(=C)C)=O)C2)=O)cc(N)ccc1C(F)(F)F C1(CC(=O)NC2C(NC(C3(C#N)CCOC3)=O)C2)CCCCCCC1 C(=O)(C#CC1CCOC1)N1C2CCC(NC(=O)CCOC3CC3)(C2)C1 c1(C(N2CCCCCC(NC(CC=C(C)C)=O)C2)=O)[nH]nc2c1CCCC2(C)C c1(C(N2CC(NC(c3ccc(N(C)C)cc3)=O)C(F)C2)=O)cccc(Cl)c1Br c1(C(=O)NC(C2CCN(C(C(COCC)(C)C)=O)C2)C)cc(C)cc(Cl)c1N N1(C(=O)Cc2csnn2)CC2(C1)CN(C(c1ccoc1C(F)(F)F)=O)C2 Cc1cc(F)ccc1C(O)C(=O)NC1CC(C)N(C(C2CCC=CO2)=O)C1 CC1(CNC(C23CSCC2C3)=O)CCCN(C(c2ccc(O)nc2)=O)C1 N1(CCNC(C2CCC3CCC23)=O)CCCN(C(c2cccnc2)=O)CC1 N1(C(Cc2nc(-c3ccc(OC)cc3)sc2)=O)CC2(CCC2NC(=O)CCF)C1 Cc1ccc(C=CC(N2CCCC(C)(C)C2CNC(C2(F)CC2)=O)=O)cc1Cl C(=O)(C1=C(C)OCCC1)NC(C(N1C(C#C)COCC1)=O)Cc1ccoc1 c1(C(=O)NC(CC(C)C)(C)CNC(C2CCNC2=O)=O)ccc2occc2n1 CCCC(C)(O)CC(=O)N1CCN(C(c2nccnc2C)=O)CC1c1cn[nH]c1 C(=O)(C(F)C(C)(C)O)NCC1(CCNC(C(C)(C)c2ccccc2)=O)CC1 C1(C)(NC(C2(NC(c3c(CC)ocn3)=O)CC(O)C2)=O)CCCC1(C)C c1(C(N(C2CCCN(C(c3ccoc3CC(N)=O)=O)C2)C)=O)cnc(Cl)n1C N1(C(COCCC)=O)CCN(C2(NC(=O)CCOCC)CC2)CC1.COC C1(CC(=O)NCC(CC=C)NC(C2C3CCCCC23)=O)OCCC1(C)C C1(CNC(C2CC(C)C2)=O)CN(C)CCN1C(c1ccon1)=O c1(CC)nc(C(=O)NCC2CCC(C(=O)NCC3CCC3)O2)cs1.C1(C)CC1 C1(CC)CCC(C)CN1C(=O)CCCN(C(=O)Cc1cccn1C)C c1(C(=O)NC(CNC(Cc2cc(CC)nn2C)=O)C(C)C)cccc([N+](=O)[O-])c1 c1(CC)nnc2n1CCCC2C(=O)NC1CN(S(=O)(=O)CCCSC)CC1(C)C c1(C(=O)NC2CCN(C(=O)COCC3CCCO3)C2)c(Cl)cc(F)cc1Br C(=O)(CCC(C)(C)C(=O)N=c1ccc(OC)n[nH]1)NC(CC)C C1(C)(C(=O)NCCCc2n(C)ccn2)CCCN(C(=O)C(F)n2ccnc2)C1 CCCC(CC)C(=O)NCCN(C(C1CCCN1C1CCCC1)=O)C(C)C N1(C(C=C(C)CNC(c2cnc(S)nc2)=O)=O)CCC(C)OC(C)C1 N1(C(c2cnc(C)s2)=O)CC2(CCNC(=O)C(F)n3ccnc3)CCC1CC2 c1(N(C(=O)C(N2CCCC3NCCC3C2)=O)C2CCCC2)ccc2ccccc2c1 c1(C(SS(Cc2c(C#N)cccc2)(=O)=O)=O)ccc2c(c1)OCCO2 Cc1cc(C)c(C(=O)NC2CC3CC2CN(C(=O)Cc2cccnc2)C3)c(N)c1 C1(CC(=O)NCC(CC)(CC)OC)CC2(C1)CN(C(=O)Cc1ccn(C)c1)C2 n1(CCC=C)cc(C#CCNC(c2ccc(-c3cnnn3C)cc2)=O)nn1 Cc1ccc(C(=O)NCc2ccc(C(=O)NCC(c3ccsc3)C)cc2)c(O)n1 c1(CC)ccc2occ(C(=O)NC3CCC(NC(=O)CCn4ccnn4)C3)c2c1 N1(C(CCCOCCOC)=O)CC2CCC1C2NC(=O)Cn1cccnc1=O c1(N(C(CNCC(OC)C)=O)C(C)C)cc(Cl)ccc1C.C(C)(C)(C)O.CCC c1(CC(=O)N(CCCCN(C)C(c2cc(Cl)cs2)=O)C)nc(C2CC2)cs1 c1(NC(C2CC2c2cccc(-c3cnn(CCO)c3)c2)=O)cc(F)cc(Cl)c1 c1(C(=O)NC(c2cc(Br)cs2)C(=O)OC)cc2n[nH]cc2cc1C C1(NC(C(n2c(C)ccn2)C)=O)CN(C(=O)Cn2cnnc2O)CCC1F C1(N(C)C(c2cnc(C(C)(F)F)s2)=O)CCC(NC(C2CCC2(F)F)=O)CC1 C1(C(N2C(CC)CC(O)C2)=O)C2CC3C(C2NC(=O)C(C)(C)C2CCCC2)C13 N1(c2ccnc(NCc3c(OC)cc(C)cn3)n2)CC(C)(C)OC2(CCC2)C1 C(=O)(CC(C)(C)O)N(CC(=O)NCCOCCCC)CC1CC1 O=C1CN(C(=O)CC2CCCCC2NC(C2COCCO2)=O)CCCN1 CC(C(C)(C)C(=O)NC1C(O)CC1O)NC(C1COCCC1C)=O N1(C(CCCOCC)=O)C2CCC(C2)C1CC(=O)NCC(C)CC(=O)OCC C(c1ccc(OCC)cc1)=CCCC(=O)NC(CCCC)CNC(=O)C=C(C)C C1(NC(c2n(COC)ncc2)=O)(CNC(c2scc(C)c2C)=O)CC2CCC1C2 C1(C(=O)Nc2ccc(COC3CCN(C(C)=O)CC(N)C3)cc2)C2CS(=O)(=O)CC12 N1(CC)CC2(CN(C(=O)CN(C(=O)CC3CCCOC3)CC)C2)C1 N1(C(=O)CC2CC(NC(=O)CC3CSC3)C2)CCc2n[nH]cc2C1 CC(CC(F)F)C(=O)NCC(c1ccccc1F)NC(c1n[nH]cc1F)=O c1(OC)c(C(=O)NCCN(C)C(c2c(C)cc[nH]c2=N)=O)cc(Cl)cc1Cl CN1CCC(C)(C(=O)NCC2(C(C)(C)C)CCN(C(C34CC(CO3)C4)=O)C2)C1=O c1(OC)ccnc(C(N2CC(N3CC(C(C4CC4(C)C)=O)CC3=O)C2)=O)c1O C1(CNC(c2c(Cl)cn(C)n2)=O)CC2(C1)CN(C(=O)COC1CC(F)(F)C1)C2 c1(C(=O)NC(C)C(=O)NC(C23CC(CO2)C3)C)cnccn1 C(=O)(C1=NOC(C)C1)N1C(CNC(CCc2scc(C)n2)=O)CC(O)C1 C1(OC)CN(C(=O)CN(CC(C)(C)C)C)CCC1NC(=O)C(C)CC1CCCO1 C1(NC(c2cnc(OC)nc2C)=O)CN(C(=O)C(C)C2CC2)CC(C)(C)C1 c1(C(=O)NCC23C(CN(C(CSc4c(C)noc4C)=O)C2)C3)cc2[nH]ccc2s1 C(C(COC)CC(=O)N1CC2CC(NC(c3ccc(C4CC4)cn3)=O)C2C1)OC CCC1=NOC(C(=O)NCC2CCCC(CNC(=O)CCCNS(C)(=O)=O)C2)C1 C(=O)(CC(O)c1ccccc1)N(C)CC1COCC1NC(c1cnoc1)=O c1(C(=O)NC(COC)CNC(=O)C(C)CCCOC)ccc2nc(C)sc2c1 C1(C(=O)NC23CC(COC)(OC2)C3)COCCN(C(C2(N(C)C)CCC2)=O)C1 N1(C(c2cccc(OCC)c2)C(=O)NC2CC2)CCC2(C1)CC(F)(F)C2 c1(OC)cc(OC)c(C(=O)NC2CCCCN(C(C3CCC(C)(C)O3)=O)C2)cn1 C1(NC(c2cc(C)c(C)nn2)=O)COC2(C1)CN(C(c1ccc(Br)o1)=O)C2 C1(C(=O)OCC(=C)OCOC)CC(N=[N+]=[N-])C1 C1(NC(C(C)OCC)=O)CN(C(=O)CCC(C)(C)F)CCC12CCC2 Cn1ccc(CCC(=O)NCC2CCN2C(C2CSCCS2)=O)c1 N1(C(c2c(OC)c(C)ncn2)=O)CCCC2CN(C(=O)CC3CCN(C)C3)CC12 Cc1cnc(C(N2CCCOC(CCNC(C3CC3C)=O)C2)=O)c(C)c1 C(=O)(C1=CCC(C)CC1)N1CC(NC(c2c(C)nc(C(C)(C)C)s2)=O)(CO)C1 N1(C(c2cc(C)nc(Cl)c2N)=O)CC2CCCC(NC(C3C4COCC34)=O)C2C1 C1(C(=O)NCc2cc(C)cc(O)c2)N(C(=O)Cn2ccnc2C)CCCC1(C)C N(C1COc2ccccc21)C(C1CC2CC2N1C(c1c[nH]ccc1=O)=O)=O N1(C(CC2(CSC)CC2)=O)CCC2CCC(C1)N2C(=O)C(c1nc(C)cs1)C C1(CC)CCC(C(=O)NC(CN)CCc2ccc(F)cc2)CC1 CC(C(=O)NC1(CCNC(=O)COCC2CCCOC2)CCC1)C(F)F C1(NCc2cccc(OC(c3ccccc3)CC)c2)CCCC2(CCCC2)C1 N1(C(C=C(C)Cl)=O)CC2CS(=O)(=O)CC2(CNC(=O)C2=CC(C)(C)C2)C1 c1(C(=O)NCCNC(CCC)=O)sc2ccc(Br)cc2c1C N1(C(C=C(C)C)=O)CCC2(CCCN(C(=O)Cc3cc(F)cc(Br)c3)C2)C1 C1(NC(C2(CNC(C=CCOC)=O)CC2)=O)C=CCCCC1 C1(CCCC)CCCN(c2nnc(C3CCOC3)n2CCOCCOCC)C1 N1(C(=O)CN2CCNS2(=O)=O)CCCN(C(=O)C(O)Cc2ccccc2)CCC1 c1(OCC)cc(F)ccc1C(N1CCCC1C)C(=O)NC1CCCCC1 CCC(C(=O)NCCC(C)(C)C(=O)NCC1(O)CCCCC1)C(C)(C)CC c1(OCC)ccc(C(=O)NCCCC(CO)NC(=O)C(O)C2CCCC2)cc1 C1(N(C(=O)Cc2scnc2C)CC)CCCN(C(c2csc(S)n2)=O)C1 N1(C(CNC(=O)NC)=O)CCC(O)(CN(C)C(C2CCC3(CC3)C2)=O)C1 N(C(=NCCC1CCCCC1)NCC1C2COCC12)Cc1cn(C)nc1 N1(C(C2N(Cc3ccc(C(C)(C)C)cc3)CC=C2)=O)CCC2(CCC2)C1 c1(NC(C)=O)cccc(CC(=O)NC2CCC2NC(c2cc(C)c(C)[nH]2)=O)c1 n1(CC(C)NC(c2cc(Cl)no2)=O)cc(-c2ccncc2)nn1 N1(C(C2(CSC)CC2)=O)CCC(O)C(C(=O)NCc2ccc(=O)n(C)c2)C1 Cc1c(C(N2CC3CCC3(CNC(=O)CN(C3CCCC3)C)C2)=O)cccc1Cl c1(CCC(N2CCC(NC(C3(C)CC3F)=O)CC2)=O)cccc(Br)c1Cl CC1c2cccc(F)c2CCN1Cc1sc(Cl)cc1Br C1(CNC(COCC#C)=O)CN(C(c2cc(N)cc(F)c2)=O)CC12CC2 c1(CCC(=O)NC2CC(NC(c3c(C)c[nH]n3)=O)C(O)C2)ccc(F)cc1F C1(NC(CC2C(C)C2(F)F)=O)CC=C(C(=O)NCc2ccc(C#N)s2)C1 C(=O)(C(F)CC(C)(C)C)NCC1C(C)CCN(C(C2(CC=C)CCCC2)=O)C1 c1(C(=O)NC(CC)CO)cnn2cccc(-c3cc(OC)ccc3[N+](=O)[O-])c12 C(=O)(CC(O)C(C)C)NC(C1CCN(C(C(C)NS(CCCC)(=O)=O)=O)CC1)C Cc1nn(CC(=O)NCC2C3CN(C(c4nnc(O)cc4O)=O)CC23)c(C)c1C C(=O)(C(CC1CCCC1)N(C)C(CC(=O)OC(C)(C)C)=O)NCCCOC=C c1(OC)ccc(CC(=O)NCCC2(O)CN(C(=O)Cn3cc(Br)cn3)C2)cn1 C(=O)(C(C(=O)N(C)CCNC(=O)CCSc1n[nH]c(C)n1)C(C)C)OCC c1(CCNC(C(C)NC=O)=O)nc2ccc(Cl)cc2[nH]1 Cn1nc(C(C)(C)C)cc1C(=O)Nc1cnn(CC(N2CCCC2)=O)c1 N1(C(C(C)C)=O)CCC2CCN(C(c3cnn(C4CC4)c3)=O)CC2C1 c1(OC)c(CC(=O)NCc2ccsc2Br)ccc(F)c1F.c12c[nH]c(c1)C(=O)N2 C1(NC(C2C(C)(C)C2(C)C)=O)CCCC12CN(C(C1CC3(C1)CC3F)=O)C2 c1(C(N2CCC(C)C2)C(=O)NCC(=C)C)ccc(CN(C)C)o1 c1(C(=O)NC2C(NS(C)(=O)=O)COCC2)cc(F)ccc1SC(c1ccco1)=O N1(C(c2c(SC)ccs2)=O)CCC(F)(CNC(=O)C(F)C2CC2)CC1 c1(N2CCC(N3CCC(C)C3c3cn(C4CC4)nn3)C2=O)cc(F)cc(F)c1F c1(CNC(c2csc(CNC(C3CCOCO3)=O)c2)=O)c[nH]ccc1=O CC1CCC(NC(=O)CCCC(=O)NC2CC2)CN1C(c1ccnnc1O)=O c1(C(=O)NC2CC(CC(=O)NC(C(C)SC)C)C2)coc2c1COC2 c1(NC(N2CCC(CO)C2)=O)cccc(C)c1CNC(C1CCN(CC)CC1)=O C1(C(N2C(CNC(C3CN4CCN3CC4)=O)CC(O)C2)=O)CCC(F)(F)CC1 Cc1cc(C(=O)NCC2CC2NC(C23CCC(CO)(CC2)CC3)=O)ccc1C#N CCC(C)(CC(=O)N1C2CCCC1CN(C(=O)C=Cc1cscn1)C2)C(=O)OC c1(C(N2CCC(C)(NC(C=CSC)=O)C2)=O)c(Br)cncc1[N+](=O)[O-] N1(Cc2cccc(C(=O)OC)c2F)CCC2(CC1)OCc1ccccc12 c1(N(C)Cc2nccn2C(C)(C)C)nc(=NCCc2cc[nH]n2)[nH]c2c1COC2 c1(OC)cccc(CCC(C)NC(c2ncccc2Br)=O)c1 N1(C(C=Cc2ccc(C)cc2)=O)CCCC12CCN(C(c1ccc(O)cn1)=O)C2 C1(NC(CCCCCOC)=O)CC12CCN(C(c1cc([N+](=O)[O-])n(C)n1)=O)CC2 C1(c2n(C(C)C)ncc2)CC(O)CN1N(C)C1CCC1C c1(C(N2CCN(C(c3n[nH]cc3Br)=O)CC2)=O)cccn(CC(F)(F)F)c1=O C1(C(N2CC(N3CCN(C(c4ccc(CO)s4)=O)CC3)C2)=O)C(F)(F)C12CCC2 CCC(CC(C)C)C(=O)N1CCCC(C)(CNC(C2CCC(F)(F)C2)=O)C1 c1(C(=O)NC2C3CN(C(c4c(C)cc(OC)nc4)=O)C2C3)ccn2c1CCCC2 C=C1CCCN(C(=O)CN(C(C2CC=CCO2)=O)C(C)C)C1 C1(C(C)NC(C2N(C(c3nc(C)oc3)=O)C(C)C2)=O)CN(C)CCO1 c1(C(N2CCC(C(C)NC(c3nccc(C)n3)=O)CC2)=O)ccnc(F)c1Cl Cc1cnc(C(=O)NCC2C(C(C)C)CCN2C(C23COC(CF)(C2)C3)=O)nc1 c1(NC(=O)NCCN2CCCN(S(C)(=O)=O)CC2)nc2cccc(Cl)c2[nH]1 c1(C(=O)NCC(CC)N(C(C(C)NC(CC)=O)=O)C)c(C)nc(C)nc1C N1(C(C(C)Cc2ccncc2)=O)CCCOC(CNC(=O)CC2(C(F)F)CC2)C1 N1(C(C(C)(C)OC)=O)CCCC(CCNC(C2CC2c2ccccn2)=O)C1 N1(C(CCCCC(=O)OC)=O)CC(C2CCN(C(c3ccc(C)s3)=O)CC2)C1 C1(NC(C2C(CCC)CCC2)=O)CN(C(=O)CNC(=O)NC2CC2)C(C)(C)C1 C1(NC(c2coc(Cl)n2)=O)CC(NC(c2cnnn2C2CC2)=O)C12CCC2 C12(C(N(C)CC3CCN(C(C4C(C)C4)=O)C3)=O)CC(CO)(C1)OC21COC1 CC1CC=C(C(=O)NC2CC3CCC(C2)N3C(=O)CC2CCC(=O)C2C)CC1 c1(C(N2CC(F)CC(NC(c3[nH]cc(C)c3)=O)C2)=O)c2c(nn1C)CCSC2 c1(C(=O)NC2CCN(C(=O)Cc3ccnnc3O)CC2F)nc(O)nc(O)c1F N1(C(C(Cn2cccn2)NC(CCC(C)SC)=O)=O)CCOC(C#N)C1 C(=O)(C(F)CC(C)(C)C)NC1CCC(C(=O)NC(C(C)O)CO)C1 N1(C(c2cc(-c3cc[nH]n3)on2)=O)CCCN(C(=O)CCC2CCCN2)CC1 S(=O)(=O)(c1cccc(N2CCC(CCO)C2)n1)NCCCCN(C)C c1(CC)cc2c(c(=O)o1)C(c1c(Cl)sc(C(=O)OC)c1C#N)NC(=O)N2C1CC1C C(=O)(C(C(=O)OC(C)(C)C)C(C)C)N(CC(CN(C(c1c(C)ocn1)=O)C)O)C N1(C(CCc2cc(C)no2)=O)CCC(C(=O)NCC(C)S(N)(=O)=O)CC1 C(N=c1[nH]cc2ncnc-2[nH]1)C1N(C(c2c(C)cccc2)=O)CCCC1 C1(=CCOC)CN(C(=O)COC2CC(NC(C3CS(=O)C3)=O)C2)C1 C(CCCCCCO)C(=O)NC1(C(C)NC(=O)CCc2ccoc2)CC1 n1(CC)nc(C(=O)NCC2(C)CCC(NC(=O)CN3CCC(C)CC3)C2)cc1C C(=O)(C1=CCCCC1)N1C(C)(CNC(C2(OC)CCSCC2)=O)CCC1 N1(C(C(c2ccccc2)OC)=O)CCC(CN(C)C(c2cc(Cl)nn2C)=O)CC1 c1(C(N2CCC(CCNC(CNC(C(CC)C)=O)=O)C2)=O)ncc(C)cc1F C(=O)(C(CC(F)F)NC(=O)C=Cc1ccccc1)NCC1C(N(C)C)COC1 CC1CCC(O)(C(=O)NCC2CC(O)(CNC(C3CCCCO3)=O)C2)CC1 N1(C(c2nc(Cl)cs2)C(=O)NCCC)C2C=C(c3ccccc3)CC1CC2 C(C)(C)(CCCNC(=O)C(c1cccc(Br)c1)(C)O)OC N1(CC(C)C)C(=S)NC(c2scc(Br)c2C)C2=C1CCN(C(C)(C)C)C2=O C(=O)(C(C)CC(C)C)N(CCC(=O)NC(c1ccnn1C)CC)CC#C CCCC(C(=O)N1CCN(C(c2cc(N)c(C)cc2C)=O)C(C)C1C)C(C)C c1(NC(CCC(CC)NC(C2CN3CCN2CC3)=O)=O)ccc2c(c1)OCO2 CC(C)(CC#N)C(=O)NC1CC2(C1)CC(NC(=O)CCCNC(=O)C(C)(C)C)C2 C(CNC(c1sccc1C#N)=O)(CC(F)(F)F)NC(CN1CCC(C)CC1)=O c1(CC)onc(C(N2CCCC2C2(O)CN(C(C3CCCC3O)=O)C2)=O)c1C c1(CCOC(CC2N(C)CC=CC2)=O)c(F)cc(Br)cc1F c1(C(N2CC(O)CC(NC(CSCCCC)=O)C2)=O)nc(C)c(C)nc1C c1(C(=O)NCCC(CC)(C)NC(=O)CCC(C)C)cncc2ncccc12 Cc1cccc(-c2nc(C3CC(n4cnnc4)C3)n(CCCN(C)C)n2)c1 Cc1nc2cc(C(=O)NC3CC(CCNC(=O)COCC(C)(C)C)C3)ccc2s1 C(=O)(C1=CCCC1)NCC(C(C)C)NC(C(C)NC(=O)NC)=O C1(CCNC(C2(OC)CC2)=O)CCN(C(=O)Cc2cncnc2O)C(C)C1 CC(C)(C)C(CCc1ccsc1)C(=O)N1CC2COCC2(c2n[nH]c(=N)o2)C1 Cc1cc(C(=O)NC(C)C(c2ccccc2)NC(c2cccs2)=O)nc(O)n1 C1(N(C(c2cnccn2)=O)CC)CCCN(C(=O)C(C)n2cnnn2)C1 c1(COC(CCC)=O)cccnc1N1CCCC1.c12ccc(cc1)CCC(=O)N2 Cc1ccn(CC(=O)NC2CC2CNC(=O)CCS(=O)(=O)N(C)C)c(=O)c1 C1(NC(CC(=O)NCC#C)=O)CC2CC(C1)N(Cc1ccc(F)cc1)C2 N1(C(c2c(C)c[nH]n2)=O)CC(NC(c2cc3occc3[nH]2)=O)CC(F)C1 Cn1cccc(C(N2CCC(C(C)(C)C(=O)NC3CCS(=O)(=O)C3)C2)=O)c1=O C(=O)(CC(C)CC(C)C)N(C1CN(C(c2ccc(C)c(C)n2)=O)CC12CC2)C C(C(=O)N(C)Cc1ccncc1)(C(C)(C)O)NC(C(C)=C1CC1)=O c1(C(=O)NC2CC3CN(C2)C(=O)CO3)cnc2ncc(Cl)cn12.C(COC)OC C12CCC(CC1)CC(=O)N2.N1(C(N(CC(=O)OCC)C)=O)CCCC(N(C)C)C1 N1(C(C2CC(O)(CC#C)C2)=O)CCCCC1CNC(=O)C(=Cc1cccnc1)F