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199,N1(C(C(=O)OCC)=O)CCCC(C2OCCCC2NC(=O)CC(C)(C)OC)C1 200,c1(C(N(Cc2cn(CC3(C)CC(F)(F)C3)nn2)O)=O)nc(Br)cnc1N 201,c1(C(=O)NC2CN(C(Cc3cc(C)sc3)=O)CC23CC3)ccc2nnc(C)n2c1 202,N1(C(CCC(N)=O)=O)CCCC2CN(C(c3ccc(CCF)cc3)=O)CC12 203,Cn1cc(S(N)(=O)=O)c(C(N2CCC(C)(CNC(=O)CN3CCCCC3)C2)=O)n1 204,CC1=C(C(=O)NCC2CC2NC(c2cccc(NS(=O)(=O)C(C)C)c2)=O)CCC1 205,c1(OC)cc(C(=O)NC2CCCC(C(=O)Nc3sc(C)cc3C#N)C2)cc(C)c1 206,c1(C(=O)NC(C(C)C)(C)CNC(C2CCOC2)=O)cc2c(F)cc(F)cc2o1 207,c1(C(N(CC(N2CCCCC(O)C2)=O)C2CC2)=O)cccn2ccnc12 208,CCCC(CC(=O)NC1CCN(C)C1)NC(=O)CC1CC(OC)C1 209,C(=O)(CN=C(NC(C)CF)NC1CN(C(=O)OC(C)(C)C)CC1C#N)NC 210,c1(C(=O)NC2CCCCN(C(c3c(CC)non3)=O)C2)nc2cc(F)ccc2s1 211,C1(NCCNCc2cc(C)cc(C)n2)CCCCC1C1CCCCC1 212,CC1CC(C(=O)NC(c2ccc(Br)cc2)CO)N(C(=O)CCc2ccco2)C1 213,N1(C(C2CCN(C(CC)=O)C2)=O)CCC2CCC(NC(c3ccns3)=O)C12 214,C1(SC(CC)C(=O)NC(c2nnc(CC(=O)OCC)s2)=O)CCOC(CC)C1 215,c1(C(N(CCCNC(=O)C2CC2)CC)=O)nc(C(C)C)ncc1Cl 216,C(C(C(=O)N1CC(Cn2cc(C(C)NC(c3nonc3N)=O)nn2)C1)OC)OC 217,C(=O)(CC1(N(C)C)CC1)NCCN(C(C1CC1NC(=O)OC)=O)CC 218,Cc1cc(CC(=O)NCCC2CN(C(=O)C(C)OCC(C)C)CC2C)ccc1F 219,CC1(C)CC(C)(NC(=O)C(CNC(=O)CCCC2CCCO2)CC2CC2)C1 220,N1(C(CC(C)O)=O)CC2(CNC(c3csc(-c4ncc[nH]4)n3)=O)CC1CO2 221,C1(CNC(=O)CCC2CC2(F)F)CCCCN1C(c1coc(C(F)F)n1)=O 222,C(=O)(C(CC(C)(C)C)NC(=O)CC(C)(F)F)N(CC(CN(C)C)O)C 223,N1(CC(=O)NCC(CN(C(CCN(CC)CC)=O)C)C)CCCC1=O 224,C(CC(C(=O)N1CCC(OCC)CC1)NC(C1CCOC1(C)C)=O)=CC 225,c1(COC)nc(NCc2c[nH]c(=N)s2)cc(N(C)Cc2nnc(O)o2)n1 226,C(=O)(C(C)(C)CCCN=[N+]=[N-])N1CCC(CCNC(C(C)C2CC2)=O)C1 227,C=CCCCC(C(=O)NCC1CC12CCOCC2)NC(c1ncc(C)s1)=O 228,c1(C(=O)NC2CC(NC(=O)CCSc3ccccc3)C2)csc2ccccc12 229,CCC(C)(F)C(=O)N1CC(NC(c2cc(-c3ccc(F)cc3)no2)=O)C(C)C1 230,C1(NC(C2C(C=C)OCC2)=O)CC12CCN(C(c1ncoc1C1CCC1)=O)CC2 231,C=CC(C)(C)C(=O)NC(CN(C)C(c1ccncc1CC)=O)CC 232,C(CCCCC(=O)N1CCC1CNC(c1cc2c(s1)CCC2)=O)OCC 233,CC(C)C(CC(=O)NC1(C)CCN(C(C2CC3CC3C2)=O)CC1)C(C)C 234,c1(NC(=O)NCCC2CCN(C(C)=O)CC2)ccc(I)nc1Cl 235,Cc1ccc2sc(C(=O)NCCC3CC(NC(=O)C(O)C(C)(C)C)C3)c(C)c2c1 236,c1(OC)cc(CN(CC(F)(F)F)Cc2ccccc2)c(O)cc1F 237,C(C(C(=O)NC1CCC1)N(C)CC1(S(C)=O)CC1)(C1CCOC1)OCC 238,c1(CNC(=O)OC(C)(C)C)cccc(CC(=O)NCCCCCO)c1 239,c1(C(CC(=O)OCC)NC(=O)C(C)(C)CNC(C)=O)ccc(O)nc1 240,N#CC1CN(C(c2ccnc(Br)c2)=O)CC1NC(=O)Nc1cccc(Cl)c1 241,c1(C(=O)NCC(CN(C)C(c2c[nH]nc2C2CCC2)=O)O)cnccc1N(C)C 242,C(C(N=c1[nH]c(SC)nc(Cl)c1C)c1ccccc1)NC(CCC=CC)=O 243,Cc1nn(CC(F)(F)F)c(Cl)c1C(=O)NC1CCN(C(c2cnc[nH]2)=O)C(C)C1 244,C1(N(C(CN2CCC(C)C2)=O)C)CCN(C(c2cc(C(N)=O)co2)=O)CC1 245,CC(C)CCC(C)NC(C1(CNC(C2CCCOCC2)=O)CC12CCC2)=O 246,N1(C(c2cn(C(C)C)nn2)=O)CCC(C)(NC(=O)CCC2OCCO2)C1 247,Cc1cc(NC(C2OCCN(C)C2=O)=O)ccc1NC(=O)CCC(C)(C)F 248,c1(CNC(=O)COc2cncc(C(=O)NC3CC3)c2)nc2cc(Br)ccc2o1 249,c1(C(=O)NC2CCCN(C(Cc3cn(CC)nc3C)=O)C2)cn2ccnc2cn1 250,c1(OC)cc(C(N2CCCCC2c2nc[nH]n2)=O)nc2ccccc12 251,CC1(O)CC(NC(C2CSCN2C(=O)CCC2CCCC2)=O)C1 252,N1(C(c2c(CC)nco2)=O)CC2CCC1CN2C(=O)Cc1cnc(C2CC2)[nH]1.C 253,N1(C(C23C(NC(CC(C)(C)O)=O)C4CC2C3C4)=O)CCC(CO)C(C)(C)C1 254,Cc1cc(F)ccc1CCC(=O)N(CCCNC(C12CCCC1(C(N)=O)C2)=O)C 255,c1(CCNC(C(=O)NCC2(C)ON=C(C)C2)=O)c[nH]c(=N)nc1O 256,c1(C(c2nnnn2CC)NCC(CC)CO)cccc(OC)c1Cl 257,C1(CNC(CC=C=C)=O)CC2(CC2)CN1C(=O)C(C)C=Cc1ccccc1 258,CC(CC1CCCC1)CN=c1[nH]c(=N)[nH]c(=NC2CCCCC2)[nH]1 259,C(=O)(C(C)(F)C(=O)N1CCN(C(=O)CCc2ncc[nH]2)C(c2ccncc2)C1)OC 260,Cc1ccc(Cl)c(C(=O)Nc2ccc(C(=O)Nc3ncnc(Cl)c3Br)nc2)c1 261,CC(CC(F)(F)F)C(=O)NC1CC(C)(C(=O)N(C2CCCC(C)C2C)C)C1 262,C1(NC(c2c(OCCOC)nccc2)=O)CCN(C(c2cnc[nH]2)=O)C1(C)C 263,CCC(C)CC(=O)C(=O)N(C1CCCC1)CCCNC(=O)C=CC=C(Cl)Cl 264,c1(NC(CCOCCN(C)C(c2ccc(OCCF)cc2)=O)=O)ccc(Cl)cc1 265,C1(NC(c2cccc(OC)c2O)=O)C2CC3CN(C(=O)CCOC(C)C)C1C3C2 266,N1(C(CCC(C)SC)=O)CCC(C2(NC(=O)CC(C)n3ccnc3)CC2)C1 267,c1(OC)ccc(C(=O)NCCN(CC(C)O)C(=O)CSc2ccc(C)cc2)c(Cl)c1 268,N1(C(CCNC(=O)OC)=O)CC=CC1(C)C(=O)NCCc1ccc(O)cn1 269,C(CC(=O)N1CCN(C(C2CC23CC3)=O)CC1)(C(F)F)NC(=O)OC(C)(C)C 270,N1(CCCC)CCC(C(=O)NCC(C)N(C(=O)CC2CCCO2)C)CC1 271,C(=O)(CCCCCF)N(CC(C)O)C.C1C(=O)N1CC.N(CCS)(CC)CC 272,C1(CC)C(=O)N(C)CCN1C(C1COCCN(Cc2scnc2C)C1)=O 273,CN1CCC(CCNC(C2(NC(=O)CNC(=O)CC(C)(C)C)CCCC2)=O)C1=O 274,C1(C)(C(=O)NC(CC=C)CC=C)CCCN(C(C2CCN(C(C)=O)C2)=O)C1 275,c1(C(=O)NCC2C=CC(NC(C(C3CCCC3)OC)=O)C2)ccc(C(C)C)cc1 276,c1(C(=O)NCC=CCNC(C(CCC)C)=O)cc([N+](=O)[O-])ccc1NC 277,c1(OC(C)C(N2CCCC(CCNC(=O)C3CC3)C2)=O)ccc(F)c(F)c1 278,C=CC(CC)C(=O)NC(c1ccccc1)C(=O)NCC1CC(N(C)C)C1 279,N1(C(c2cc(C(C)(C)C)on2)=O)CCCC2CCN(C(=O)C3=CCCS3)CC12 280,c1(C(CNC(Cc2nc(CC)[nH]n2)=O)O)cc(Br)ccc1OC 281,S(=O)(=O)(c1ccc(Cl)c2ncccc12)NC1C(=O)N(c2ccccc2Cl)CCC1 282,C(CN=C(NCc1cc(Br)ccc1C(F)(F)F)NC1CCC1)OCC(=C)C 283,CCC(C(=O)NCC(C(=O)NC(C)Cc1ncn(C)n1)C(C)(C)C)C(C)(C)CC 284,N1(C(C2N(C(C)(C)C)CC2)=O)CC2CC(NC(=O)C(F)=C3CCCC3)CC(C2)C1 285,C(=O)(C1=CC2CCCCCC12)NC1(C)CCN(C(=O)C(C2CCCO2)C2CC2)C1 286,C(c1cccnc1)=C(C)C(N1CC(NC(c2cnn(CCF)c2)=O)C(CO)C1)=O 287,c1(CC(N2CCC(NC(c3c(C)onc3CO)=O)C2)=O)ccc([N+](=O)[O-])cc1F 288,CCCC(CCCNC(=O)CCCOC(C)C)N=c1[nH]c(Cl)nc(C)c1F 289,c1(C(=O)NCC(C)NC(C2OCCN(CC)C2)=O)ccc2c(c1)OCCN2 290,CCCC(C)(CCC)C(=O)NC1CCCC1NC(c1cnn2cccnc12)=O 291,CCC(CC(=O)N1CC(CNC(C2OCCC2C)=O)C1)C(C)C 292,Cc1cc(CC(=O)NC2CC3CC2N(C(=O)C=CCN2CCCC2)C3)cc(F)c1 293,c1(C(N2CCC(CC=C)(NC(C3CC=CCC3)=O)C2)=O)ccc(C#N)n1C 294,C12(C(=O)NCCN(C(=O)CC3CN4CCC3CC4)C)CCCCC1NC(=O)CC2 295,C1(CNC(C(C2CCCC2)OCC)=O)CC2(CCC2)CN1C(=O)C(C)=C1CC1 296,C1(C(N(CC(O)CN(C)C(C2CC2F)=O)C)=O)CCCN(c2ccn(C)n2)C1=O 297,C(N=c1[nH]c2c(c(=NCC3CC4(CCC4)CO3)[nH]1)CCC2)c1c(C)cc(Br)cc1 298,Cc1ncsc1COCC(=O)N(C)CCc1cn(CCCN2CCOCC2)nn1 299,N1(C(c2cc(OC)no2)=O)CCC2(CC1)CC2NC(C1CCC(C)(C)OC1)=O 300,C#CC1(NC(C2CN(C(c3cc(C)n(CC)n3)=O)CC2(F)F)=O)CC2CCCC12 301,Cc1ccc(C(=O)NC2CN(C(=O)CCc3cn[nH]c3)CC2C)c(Cl)c1C 302,C#CCCC(O)C(=O)NCC1CCN1C(c1ccnc(C(C)(F)F)c1)=O 303,c1(C(c2n(CCC)nnn2)NCC2CCSC2)nc(Br)c2ccccn12 304,N1(C(c2ccc(Cl)cc2CSc2cc[nH]c2)=O)CCCC12CCOC2 305,c1(NC(=O)NCc2c(C)occ2)ccc(C2CCCO2)cc1 306,Cc1ccc(F)c(C(N2CC3CC2C3CNC(=O)CNc2ccccn2)=O)c1F 307,CCCC(O)(CCC)CC(=O)NC(CNC(=O)C(C1CC1)OC)CCOC 308,c1(C(=O)NCC(C2CCCC2)O)ccc(CNC(=O)C(C2CCCCC2)O)nc1 309,CC1(C(=O)NCCC2CCCN2C(=O)CCCN2CCOC2=O)CC2CCC1C2 310,N(S(=O)(=O)N(C)C)CC(=O)NCC(C1CC1)NC(C(C)N(c1cnccn1)C)=O 311,c1(CC(=O)NC(C2CCCCN2C(c2cccnc2CO)=O)C)ccc(O)nc1 312,N1(CC)CCN(C(=O)C(c2n(CC)cnn2)NC(=O)C(CC)N(C)C)CC1 313,S1(=O)(=O)c2ccc(cc2)OCCCN1.N1(CCC)CC(CNC)CC1=O 314,C=CCCCC(C1CC1)NC(=O)NCCc1nccn1-c1ccccc1 315,c1(C(N2CCN(C(=O)CC3CC34CC4)C(C3CCC3)C2)=O)cncc2c[nH]nc12 316,C1(C)(NC(c2c(CCC)occ2)=O)CCCN(C(=O)CSc2ccccc2)C1 317,CC1(CNC(=O)C(O)C2CC2)CC(F)(F)CN1C(c1ccc(SC(F)F)cc1)=O 318,c1(C(N2CCCCC(NC(C(CC=C)(F)F)=O)C2)=O)cccc2c1NCC2 319,C(=O)(C(=O)C(C)(C)C)NC1CC(C)(NC(CN2CC(C)(C)C2)=O)C1 320,N1(C(CCC2OCC(C)(C)C2)=O)CCc2[nH]nc(CNC(=O)C=CCO)c2C1 321,c1(OC)ccc(F)c(C(N2CCN(C(c3cc(OC)cc(F)c3)=O)C3CC23)=O)n1 322,O=C(C#CC1CCCCC1)NC(CC(=O)NC(CCO)CF)C1CC1 323,c1(C(N(CC(C)N(C)C(c2ccn(C3CCC3)n2)=O)C)=O)cc2cccnc2s1 324,N1(CC)CCN(C(C2(CNC(=O)CC3OCCO3)CCCC2)=O)C(C)C1 325,Cc1ncccc1C(=O)NC1CC(CC(=O)Nc2cnccc2C(C)C)C1 326,C1(CNC)CC(C(=O)Nc2csnc2C)CCO1 327,C1(N(C)C)CCCCN(c2cc(C(=O)O)cnc2C#N)C1 328,N1(C(C2(N(C(C(CSC)O)=O)C3CC3)CCC2)=O)CCCC(C)(C#N)C1 329,N1(C(c2cc(OC)n[nH]2)=O)CC2CC1(C(=O)NOC(C)(C)CO)C2 330,c1(C(=O)NCC(C(C)C)NC(C(C(C)C)SC)=O)c(C)nn(C(C)(C)C)c1C 331,c1(C(=O)NCCCNC(C(CNC(C)=O)(C)C)=O)nn(C)c(Cl)c1Br 332,FCCN=c1[nH]c(N2CCCC2c2ccccc2)nc2c1CCC2 333,c1(C(=O)NCC=CCNC(CCn2ccc(C)n2)=O)cc2c(s1)CCCNC2=O 334,N1(C(C=CCCC=C(C)C)=O)CC2CCC1CN2C(=O)Cc1ccccc1C 335,c1(C(=O)NC2(C)CN(C(C3(C(F)(F)F)CC3)=O)C2)ccc(=O)n(CCF)n1 336,CC(C(=O)N1CCC(C(=O)N(C)C)C1(C)C)C(C)(C)C.C1(=O)CC2(CC2)N1 337,c1(NC(c2cc(Cl)no2)C)[nH]c(=NCC2CCN(C)C(=O)C2)nc2c1cnn2C 338,C=CCCCC(C(=O)NCC1CC12CCC2)NC(=O)CC(C)COC 339,CC1(C)CC(C(N2CC(NC(c3c[nH]nc3F)=O)C(O)C2)=O)CC(C)(C)S1 340,c1(CNC(C2C3CCC23)=O)cnn2c1CN(C(C1CCCC13OCCO3)=O)CC2 341,c1(C(=O)NC(CCC)C(=O)OCC(F)(F)F)ccc([N+](=O)[O-])c(NCCN)c1 342,c1(C(=O)NCC2C(C(=O)NC(CCCCC)C)C2)cc2cccnc2[nH]1 343,c1(C(=O)NC2C(NC(C(CC=C)c3ccccc3)=O)C2)csc([N+](=O)[O-])c1 344,c1(-c2nc(-c3n(CC4C(C)C4)ncc3)on2)cn(C)nc1-c1ccc(Cl)s1 345,N1(C(c2cc(CC)on2)=O)CCN(C(=O)COCC(=O)OC)C(CF)C1 346,N1(C(c2nnc(CC)s2)=O)CCCC(C2CC2NC(C2CCCO2)=O)C1 347,C1(CC(=O)NC2C(C)C2C)C=CC(NC(=O)COC2CC=CC2)C1 348,c1(C(N2C3CC(NC(C(C=C)O)=O)CC2CC3)=O)csc2ccc(Br)cc12 349,Cc1ccc(C(=O)NC(CNC(c2ccc(C#N)s2)=O)CO)c(=O)n1C 350,C#Cc1ccccc1CNC(=O)C(C)(C)NC(c1coc(CO)c1)=O 351,c1(OC(C)C)cccc(C(=O)NC2(CO)CN(C(=O)CCC3(C)CC3(F)F)C2)n1 352,C12(NC(CN(C)CCO)=O)CCCC1CN(C(=O)Cc1cncs1)C2 353,C1(CNC(CSCC(C)C)=O)CCCN1C(=O)Cc1cc(C2CC2)n[nH]1 354,N1(C(CC(CCC)O)=O)CCc2nc(CNC(C34CCCC3CCC4)=O)sc2C1 355,C1(C(N2CC(C)(CCC(=O)NC(C3CCOCC3)(C)C)C2)=O)CCS(=O)(=O)C1 356,C(=O)(CCCC1CC1)NC(c1ccccc1)C(=O)N(CC(C)(C)OC)C 357,CCCC(C(=O)N1CC(NC(c2ccc(C(C)C)cc2)=O)C1)S(N)(=O)=O 358,CCCC(C(=O)OC)C(=O)NC12CC(CNC(=O)Cc3coc(C)n3)(C1)C2 359,CC1(CCC(N2CC(C#N)C2)=O)CN(C(=O)CNC(=O)C(C)(C)C)C1 360,CC1(CN)CN(C(c2ccc(F)cc2Br)=O)CCO1 361,c1(OC)ccc(F)cc1CC(=O)N(CCCN(C(=O)C1=CCCC1)C)C 362,c1(OC)cncc(C(N2CCC(C)C(NC(=O)C=Cc3ncc[nH]3)C2)=O)c1C 363,C(=O)(C1=C(Cl)CCOC1)NCc1cn(CC(=O)NC(c2ccccc2)C)nn1 364,C(=O)(CC(C)CC(=O)OC)N1CC2C(CNC(CC3(OC)CCC3)=O)C2C1 365,C1(C(=O)OC)CCN(C(C2CC(O)(CNC(=O)C=CC(C)(C)C)C2)=O)C1C 366,c1(CC(N2CCC(NC(CCC3C(C)C3)=O)C2C)=O)c[nH]c2cnccc12 367,C1(O)(CCc2cn(CCCCCC)nn2)CCN(C(C2CCC(C)(C)O2)=O)CC1 368,C1(C(=O)NC2CC=CC2)C2CC(O)C(C2)N1C(C1CN2CCN1CC2)=O 369,CCCCCCCCCC(C)CC(=O)NCCN(C)C(c1ccnc(Cl)c1O)=O 370,C(=O)(C(CN(C)C)C(C)C)N1C(CNC(CC2(OC)CCC2)=O)CC1 371,N1(CC(N2CCCN(C(C3CC(=O)N(O)C3)=O)CC2)=O)CCCC(C(F)(F)F)C1=O 372,N1(C(C(C2CCOC2)OC)=O)CCC(C)C(CNC(=O)C=CC2CC2)C1 373,O=C1NCC2CCCN(C(c3cncnc3)C(=O)NC3CCOC3)C12 374,N1(C(C(CC(C)C)ONC(=O)C(C)N(C)C)=O)CCN2C(=O)OCC2C1 375,c1(NCC)cccc(C(=O)NCC2CC2NC(C2CCNC2=O)=O)c1 376,C(=O)(C1=NOC(C)C1)N(c1scc(CC(N2CCCC2)=O)n1)CC.N(C)C 377,Cc1onc(Br)c1C(c1nnnn1C(C)C)Nc1cn(C)nc1SC(C)(C)C 378,c1(OC)cccc2c(C(N3CCN(C(=O)C(Cl)=CCl)CC3C(C)C)=O)cccc12 379,C(=O)(CCCCCF)NCc1c(C(N(C(C)C(C)(C)O)C)=O)nco1 380,C1(C(=O)NCc2nc(C)oc2)CCN(C(=O)CC(C)C)CCO1 381,N1(Cc2ccc(OC)s2)CCOCC(C(=O)Nc2cc(CO)cc(Br)c2)C1 382,C(=O)(C1Cc2cccc(Br)c21)NC1CCC(NC(C(C)=C(C)C)=O)C1 383,c1(C(N2CCN(C(C3CCCS3)=O)C3C2CCC3)=O)cc(=O)c2ccccc2o1 384,N1(C(c2c(C)nc(C3CC3)s2)=O)CCN(C(=O)CC2(O)CCC2)CC1C(C)C 385,C1(NC(Cc2cc(C)[nH]n2)=O)CCC2(CCCN(C(=O)C(C)C)C2)C1 386,N1(C(c2c(OC)nccc2)=O)CC(CC(=O)NC2CCCCC2C#N)C2(CC2)C1 387,c1(C(C)C)c(C(N2CCCC2C(C)NC(C2CCC(=O)N2)=O)=O)cccc1F 388,c1(OCC(=O)NC2CCC(N(C(Cn3ccc(C)n3)=O)C)C2)ccc(F)cc1Cl 389,n1(C(C)C)cnc2c(NCC=CCl)nc(N3CCC(C(F)(F)F)C(C)C3)nc12 390,C1(CC)CN(C(=NCc2cn(C(C)(C)C)nn2)NC2CC2)CC(C)S1(=O)=O 391,CC(CN(C)C(C1(N(C)C)CCC1)=O)C(=O)NCCc1cscn1 392,N1(C(C(C(CC)C)O)=O)CCC2(CCC(CNC(c3cn[nH]c3)=O)CC2)CC1 393,C1(C)(CCNC(CCC2C(C)C2)=O)CC(C(C(C)(C)C2(C)N=N2)=O)C1 394,CCC(CC(=O)NCC1CC(NC(=O)CCNC(C)=O)CCO1)SC1CCCC1 395,n1(C(CNC(c2scc(C(=O)OCC)n2)=O)(C)C)c(S)nc2ccccc2c1=O 396,CC(CNC(=O)OC(C)(C)C)CC(=O)N1CCC1NC(=O)CC1CC1 397,C1(F)(CNC(c2noc(CC)c2C)=O)CCCN(C(C2CC2c2nc[nH]n2)=O)CC1 398,Cn1ncc2ncnc(N3CCC(CNC(=O)CC4CC=CCC4)C3)c12 399,c1(C(C(N2CC(F)(CNC(C3(C=C)CCC3)=O)C2)=O)O)cc(F)c(F)c(F)c1 400,C1(CC(=O)NC(C(=O)OC)C)CC(C)(C)CN1C(C1CCC(OC)CC1)=O 401,CC(CCNCC(N1CCNCC1)(C)C)CC(C)(C)C 402,N1(C(C(=O)NCC(C)C)C)CCSC(C(=O)NC(C23CCC(CC2)C3)CO)C1 403,c1(CNC(NC(C)C2CC2)=NCCC2CC2)cn(C(C)(C)C)c(=O)nc1O 404,C(=O)(C1CCCc2ncnn21)NC1C(OC)CN(C(c2cncc(C#C)c2)=O)C1 405,n1(-c2ccn(CC)n2)nc(Cc2ccccn2)nc1CSC 406,N1(C(c2c(N)ccc(F)c2)=O)CCN(C(c2cc(O)ncn2)=O)C2CCCCC12 407,C(=O)(C(C)(F)C(=O)OC)N1CCC(OCCC(=O)NCC#C)C1 408,CCCCC(O)C(C)C(=O)NC1(CNC(C2CCCC(F)C2)=O)CCCCCC1 409,CN1N=C(CC(=O)N2CCC(F)(F)C(CNC(C3(O)CCSCC3)=O)C2)CC1=O 410,c1(C(=O)NCC2(O)CC(NC(CCCCC=C)=O)C2)cccc2c1OC(C)(C)C2 411,C1(C(COC)=O)CC(n2cc(C3C4CC5C(C4)C35)nn2)C(CCC(=O)O)C1 412,CCCCC(C(=O)NCC1CCCCS1)NC(c1cccc(C#N)c1)=O 413,N1(C(C2(CC)CN(C(=O)OC(C)(C)C)CCO2)=O)CCC(F)(F)CC(C)C1 414,c1(CN2CCC(CC(=O)NC(CCSC)CO)C2)c(C(C)C)nn(C)c1Cl 415,CCCC(C(=O)NCC1CCCCN1CCOc1cccc(Cl)c1)OC 416,CC(C(=O)OC(C)(C)C)C(=O)N1CCC(CCNC(c2ccnn2C2CC2)=O)C1 417,Cn1cnc(C(O)CNC(C2C=CCN2C(=O)Cc2nncs2)=O)c1 418,C1(C(C(=O)NCCOCC)NCC)CC=CCC1C.c1(COCC)cc(C=O)oc1C 419,N(C1c2ccccc2CC1NC(C12CCC(C1)C2)=O)C(C1(OC)CCCCC1)=O 420,C12(CC(=O)NCC(CC(C)C)NC(C3CCC4(CC4)C3)=O)CCC(CC1)OC2 421,C(=O)(C1CCc2cccc(O)c21)N1CCC(CC)(NC(C2CC(C)C2)=O)CC1 422,C1(C(=O)NCCOC2CN(C(c3ccc(=N)[nH]c3)=O)C2)CC2(CCOCC2)CO1 423,C1(NC(c2c(C)cc(SC)s2)=O)CCCC12CN(C(=O)CCC#N)C2 424,c1(NCC2(CNC(=O)Cc3cnns3)CCCC2)cc(C(N)=O)ccc1[N+](=O)[O-] 425,S(=O)(=O)(c1cccnc1)NC(c1csc(C)c1C)=O.C12CC(F)CN(C1)C2=O 426,c1(NC(c2n(CCSC)nnn2)c2cncs2)cc(F)cc(F)c1OC 427,N1(C(C2CN(S(CC)(=O)=O)C2)=O)CC2CCCC2(NC(c2cocn2)=O)C1 428,C1(NC(c2c(C)cno2)=O)C=CCN(C(=O)Cn2cccc2)C1 429,O=C1NC(C(=O)NCC2CCN2C(=O)Cn2cnccc2=O)CCO1 430,C(Cn1cccn1)(C(=O)NOC1CC1)NC(C1CCCC(=O)C1)=O 431,c1(C(CNC(C=CS(C)=O)=O)NC(=O)CCCN2CCCC2)ccc(Cl)c(Cl)c1 432,c1(C(=O)NCC2CC(C)N(C(c3cccnc3F)=O)C2)cn(C)c(=O)n(C)c1=O 433,C1(NC(C(Cc2ccco2)NC(C2N(C)CC(F)C2)=O)=O)CC(C)(C)OC1=O 434,C(N=C(NCC(F)F)N1CC(O)C2(CC2)C1)C1(O)C(C)(C)C2OCCCC21 435,N1(C(CCOCCC)=O)CCCC2CCN(C(c3cccn4cncc34)=O)CC12 436,N1(C(CCCSC)=O)CCC2(CC1)CC2C(=O)NC1(C)CCCC1(C)C 437,c1(C(=O)NCC(CNC(C(C)Cc2cnn(C)c2)=O)(C)O)cc2n(c1)CCOC2 438,C1(OCc2n(CC)nnc2C)CN(C(=O)NCCCOC(C)(C)C)CC(F)(F)C1 439,C1(NC(C(CC2CCC2)OC)=O)CCCCC1CNC=O.c1(C2CC2)cc[nH]n1 440,N1(C(C2(CC)CCC2)=O)CC(NC(c2cc(C(=O)OC)oc2C)=O)C(C)(C)C1 441,c1(NC(CCC(C)(C)C)CO)ccc2c(c1)C(=O)NCCC2 442,c1(C(=O)NC(C=CC(=O)NC(CCC=C)CO)(C)C)cccc2c[nH]nc12 443,c1(NC2C3CC32)cc([N+](=O)[O-])ccc1C.c1(CC)nnnn1C(C)(C)C 444,CCCC(C(=O)N1CCCCC12CC(NC(=O)C(C)(CC)CC)C2)S(N)(=O)=O 445,C1(NC(=O)NCc2c(OC)nc(C)cc2)CCOC2(CCSC2)C1 446,c1(COC)cccc2sc(Nc3sc(C(=O)OC)cc3S(N)(=O)=O)nc12 447,c1(C(N2CC3CCC(C2)N3C(C2CCCC(C(N)=O)C2)=O)=O)ccc2c(c1)OCO2 448,c1(C(=O)NC2C(CNC(c3cc(Cl)no3)=O)COC2)coc2ccc(Cl)cc12 449,CC(C)C(CO)C(=O)NC1CCCCC1CNC(c1cnc(-c2ccco2)s1)=O 450,C(=O)(C(CO)C(C)(C)C)N1C(CNC(Cc2nc(C(C)OC)sc2)=O)CCC1 451,CCC(CO)C(=O)N1CC(C(C)NC(c2c(OC)noc2C)=O)C1 452,C12(C(N(CC(N3CCCC(CO)C3)=O)CC)=O)CCC(CC1=O)C2 453,CCCC(C)(O)CC(=O)N(C)CCOCCN(c1nnccc1C#N)C 454,c1(C(=O)NC2(CCNC(CCC(=C)C)=O)CCCC2)ccc2c(=O)cc[nH]c2c1 455,C1(CC(=O)N(C)CC2CCN(C(=O)CCC3CCC3)C2)CCCC(=O)N1 456,C(N1CCOC2(C1)CN(C(C)=O)C2)n1c(C2CC2)nn(CCC=C)c1=S 457,N1(C(C(C2CCOCC2)C)=O)CC(NC)C(C)(C)C1.c1(C=O)c[nH]nc1Br 458,CC(C)C(C)C(CNC(C1CC1C(C)(F)F)=O)NC(=O)CCS(C)(=O)=O 459,Cc1ccc([N+](=O)[O-])c(NNC(=O)NC23CCCCC(Br)(C2)C3)n1 460,C1(CNc2nc(COC)nc(N3CCC(CF)C3)c2)CC2(CCC2)CCO1 461,c1(C(=O)OC)cnc(NC2CC(CNC(C3CCCO3)=O)C2)c([N+](=O)[O-])c1 462,N1(C(Cn2ccc(C)n2)=O)CC(C2CN(C(c3ccnc4ccnn34)=O)C2)C1 463,c1(OCC(=O)NC2(Nc3ccc(-n4cnnc4)cc3)CC2)cccc(F)c1 464,c1(C(=O)NCCC(C)CCNC(=O)C(F)CC2CC2)cccc2ccnn12 465,C(N=c1[nH]c(=NC2CC=CCC2C(F)(F)F)[nH]c2c1COC2)C1(N(C)C)CCC1 466,Cc1c(C(N2CCOC(C(=O)O)C2)=O)cnn1C(C)C(C)C 467,N1(C(C(CC)=CCCC)=O)CC(C)CN(C(c2ccc(C(F)F)cc2)=O)CC1C 468,C1(C(=O)NC(c2ccccc2F)C)CC(F)CN1C(=O)C(c1ccccc1)O 469,N1(C(C(C2CCOC2)NC(CCn2ncc(C)c2)=O)=O)CCC(CCO)CC1 470,N1(C(C(c2cccc(OC)c2)(F)F)=O)CC(NC(c2cnn(C)c2)=O)CC(O)C1 471,C=C(Cl)CCC(=O)NCC(C)(CNC(c1csc(C(C)=O)n1)=O)OC 472,c1(C(N2C(CNC(C(C)OC)=O)CC2)=O)ccc(N)c(F)c1 473,C1(CC=C)(NC(CCN(C(=O)C(O)CN(C)C)CC#C)=O)CCCC1 474,c1(CN(C(C)CN2CCSCC2)CC(=O)O)c2c(nn1C)CCCC2 475,C=CC1CN(C(c2ccc(F)c(C)c2)=O)CC1NC(C1CCCS1)=O 476,N1(C(C)=O)CCC(N(C)C(C2(NC(c3cc(CF)on3)=O)CCCC2)=O)C1 477,c1(C(=O)NCC(C2CC2)NC(c2cnc(CC)s2)=O)c(F)cncc1Cl 478,c1(C(N2CC(OC)(CNC(=O)CCCC(F)(F)F)C2)=O)cc(F)c(C#N)c(F)c1 479,C1(NC(c2c(C)oc(-c3cnn(C)c3)n2)=O)CCCCN(C(=O)C2=CCCC2)C1 480,c1(OC)ccc(C2(CNc3cnc(I)cn3)CCC2)cn1 481,C1(C(=O)NCCCC(CC)C)CCN(C(C2CC3(CC(=O)C3)C2)=O)C1(C)C 482,C1(CNC(c2c(SCC)cncc2)=O)COCCN(C(C2(C)CCCN2C)=O)C1 483,C1(CNC(C(C)N(C)C)=O)CC2CCC1N(C(=O)CC(C)c1cccnc1)C2 484,c1(OC)ccc(Cl)cc1C(N1CCN(Cc2cn(C3C=CCCC3)nn2)CC1)=O 485,Cc1c(NCc2cnc(O)nc2O)ncnc1NC(c1ccc(F)cc1)CF 486,C(C)(CCCC(C)C)NC(C(CC=CC)NC(c1c[nH]c(C)c1)=O)=O 487,Cn1ccc2cccc(C(N3CC(F)CC3C(=O)Nc3cc(O)ccn3)=O)c12 488,C(=O)(CCCCC(=O)NC1CC(OC)CN(C(c2coc(N(C)C)n2)=O)C1)NC 489,C(=O)(C(O)C(C)CC)N1C(Nc2ccc(CCC)cc2)COCC1 490,c1(N2CCCC(CNC(=O)CSCc3ccncc3)C2)nc2ncc(Cl)cc2s1 491,C1(C(N(CCCCN(C)C(c2nnsc2C(F)F)=O)C)=O)CCS(=O)CC1 492,C(=O)(C1CCc2ccc(Br)cc21)N1C(CNC(CCCCOC)=O)CCC1 493,C1(NC(c2c(C)nc[nH]2)=O)CC2CC1N(C(c1sccc1Br)=O)C2 494,C#Cc1cc(NC(=O)CN(C(=O)C(C(C)CC)N(C)C)CC(C)(C)C)cc(F)c1 495,N1(C(C(CCC)O)=O)CCOC2(CCN(C(C3(C4CCCO4)CCCC3)=O)C2)C1 496,N#CC1CCCC(C(=O)NC2CCN(C(C3CN4CCC3C4)=O)CC2CO)C1 497,C(c1cnn(C)c1C)=CC(=O)NCC(CC(C)C)NC(c1nccc(CC)c1)=O 498,C1(C(=O)NCC(CN(C(C(CC)O)=O)C)(C)C)CCN(c2ccc(Cl)nn2)CC1 499,c1(OC)cn(CC(N2CC3C(CNC(=O)CCNC(N)=O)C3C2)=O)c(C)cc1=O 500,N1(C(C(=O)NC)=O)CCC(C(F)CNC(=O)CC2CCCC(C)O2)CC1 501,c1(C(=O)NCC(CO)NC(C2COCCOC2)=O)cn2c(Br)cnc2s1 502,C(=O)(CCCC(N)=O)NCCC1C(C)CN(C(c2c[nH]nc2Br)=O)C1 503,CC(O)(CC(=O)N1CC=CC(NC(=O)CCCCN2CCCC2)C1)C(F)(F)F 504,N1(C(C(N2CCOCC2)C)=O)CCC2(CCC(NC(c3cnc(O)o3)=O)C2)C1 505,CC(CNC(=O)C(N1CCNC1=O)C)CC(=O)N(C1CCCCC1)CCO 506,n1(CC)cc(Br)c(C(C(=O)N(CCNC(CC)=O)C)CC)n1 507,C1(c2ccc(Cl)cc2)(C(=O)NCCN(C(COC)=O)CC(C)O)CCN(C)C1 508,N1(C(CSCCC)=O)CCCCC(C2CN(C(=O)Cc3ccccc3C)C2)C1 509,c1(C(C)=O)ccc(C(=O)N(CC(C)NC(C2CCC3CC23)=O)C)c(F)c1 510,Cn1ncc2c1CCC(C(N1C3CCCC1CN(C(=O)CC(C)(C)O)C3)=O)C2 511,c1(C(N(CCC2C(C)C2)C2CC2)=O)cc2cc(Cl)ccc2o1 512,C1(C(CNC(C(C(C)C)c2cc(O)n[nH]2)=O)=O)CCC(F)(F)CC1 513,CC1CCCC1(C(=O)NC(C(O)CO)C1CC1)NC(c1cnn(C2CC2)c1)=O 514,CC(C)(C(=O)N1CCC1CNC(=O)CCN1CCCC1=O)c1ccccn1 515,CCN=c1[nH]cc(C(=O)NC(C)(CC)CCNC(=O)CN(c2ccccc2)C)s1 516,C(=O)(C(CC)C(=O)NC(c1cccnc1)C(=O)NCCOC1CCCC1)OCC 517,c1(OCC(=O)NCC(C)CNC(c2ccnc(C(F)(F)F)c2)=O)ccc(O)cc1 518,c1(OC)ccc(CNC2C3CC2N(C(c2n[nH]c(C)c2C)=O)C3)cc1[N+](=O)[O-] 519,N1(C(C(C(C)O)NC(=O)C2CC2)=O)CCCN(C(=O)CCc2cnc[nH]2)CC1 520,CC1CCC(O)(C(=O)NCCOCCNC(=O)CCc2cccc(F)c2Cl)CC1 521,c1(C(=O)NCC2(CCNC(c3n(C)ncc3)=O)CC2)cc(N2CCCC2)ccn1 522,N1(C(=O)OC(C)(C)C)CC2CC1C2NCCc1ncc(SC)s1 523,C1(CO)CCN(c2ccnc(N3CCCC(CC4CCC4)CC3)n2)C12CCC2 524,N1(C(c2c(=N)cc[nH]c2)=O)CCC2(CCCN(C(C34CCC(CC3)O4)=O)C2)CC1 525,c1(C(=O)NCCC2CCC(NC(C=CC(=O)OCC)=O)C2)n[nH]c2c1COCC2 526,c1(C(N2CC(C)C(NC(c3cc(F)c(F)cc3F)=O)C2)=O)c(F)cc(F)cc1F 527,n1(CCOC(=O)CC2(O)CN(CC)C2)ncc2c(NCC3CCCC3)ncnc12 528,CC1CC2(CCC(C(=O)NC3CN(c4ccnn4C)C3)O2)CO1 529,CC(C)C(C(C)NC(C1(N(C)C)CC1)=O)NC(c1ccsc1Cl)=O 530,CCC(C(C)(C)O)NC(c1c[nH]nc1C1CCCCN1C(c1cc(C)co1)=O)=O 531,C1(OC)CC(C)CN(C(C2C(O)CCN2C(=O)C(=O)N(C)C)=O)C1 532,c1(C(N2CCc3nnc(O)cc3C2)=O)c2c(nc3ccc(Cl)cc13)CCC2 533,C=CC1(C(=O)NCCC2CCCN(C(C3(C)CCCNC3=O)=O)C2)CCCCC1 534,c1(C(N2CC(NC(=O)Cc3cccs3)C(F)(F)C2)=O)[nH]nc2c(Cl)cccc12 535,c1(C(=O)OC)ccc(C=CC(=O)NC2CCN(C(=O)C(O)CC(C)C)C2)cc1 536,C#CCCCCCCCNC(=O)C(CC1CCOCC1)NC(c1cnsc1C)=O 537,CC1c2c[nH]nc2CCC1C(=O)NC1C=CCN(C(c2csc(Cl)n2)=O)C1 538,c1(C(=O)NC(CN(C(C(C=CC)O)=O)CC)CC)ccc2nc3n(c2c1)CCC3 539,C1(CNC(C2(C(=O)NC)CC2)=O)CC2(CO1)CN(C(=O)C(C)CC1CCC1)C2 540,C1(OCCC(=O)N(CCN(C(C(C)NC(=O)OC)=O)C)C)CCC(F)(F)CC1 541,C1(NC(=O)NCC(C)Oc2cccnc2)CCCCCC1C(N)=O 542,C1(CNC(CC2CCC(NC(c3c(C)nc(C)s3)=O)CC2)=O)OCCCC1(C)C 543,Cc1cc(C#N)ccc1C(=O)NCC(O)CNC(N)=O.C1(C)(C2CCC2)C(=O)N1 544,C(=O)(C(CNC(c1cccc(O)c1F)=O)CC(C)C)NCC1C(OC)CCC1 545,c1(C(N(CCN(C(C2(C)CCC(C)C2)=O)CC)CC)=O)cc(F)ccc1O 546,C(=O)(C1=CCN(C)C1)NCC(CN(C(C(C1CCC1)OCC)=O)C)(C)C 547,c1(NCCO)ccc(OC)nc1.C1(C(CC)N2C(=O)C(=O)N2)CCCOC1 548,CCC(C)C(O)CC(=O)N1CCC(F)CC1C(=O)NOCCCF 549,C(=O)(CCC(C)C)N(CC(OCC)OCC(C)COC)C 550,c1(NC(C2COCCN2C(c2cc[nH]c2)=O)=O)c(C(F)(F)F)cccc1C#N 551,C1(O)(CC#N)CC2CCC(C1)N2C(=O)CCc1nc(-c2ccsc2)no1 552,N1(C(c2c(N)nccn2)=O)C2CCC1C(CNC(=O)CCCc1cnccn1)C2 553,N1(C(C(C)(C)OC(C)=O)=O)CCC2CN(C(=O)Cc3nnc(C)s3)CCC2C1 554,C12(CC(N3C(CNC(C4CCC(C)C4)=O)C=CC3)=O)CC3CC(C1)CC(O)(C3)C2 555,C1(NC(CCc2cc(OC)no2)=O)CCN(C(c2ccc(Cl)nc2O)=O)C(C)C1 556,c1(C(N2CCC(NC(CCN(CCC)C)=O)C2)=O)ccc2[nH]c(=O)c(=O)[nH]c2c1 557,S(=O)(=O)(c1ccc2oc(O)nc2c1)N1CCN(Cc2cc(OC)c(Cl)cc2)CC1 558,c1(C(N2CC(CNC(C3C(C)(CC)C3)=O)C2)=O)ncoc1C1CCCO1 559,Cc1cc(F)c(C(N2CC(C(=O)NCCNC(C3COC(=O)C3)=O)C2)=O)cc1F 560,C(=O)(CC1=CCN(C)CC1)N1CC(C)C(N(C)C(c2ccnc(F)c2O)=O)CC1 561,Cc1cc(C(=O)NCCC2COCCN2C(c2ccc(C#N)o2)=O)c(C)s1 562,Cc1cnc(NC(C2CCN(C(c3ncc(F)cc3F)=O)C2)=O)c(Br)n1 563,c1(OC)ccc(S(=O)(=O)N2CCC(O)C(C)C2)c(C(=O)O)c1 564,c1(CC(=O)Nc2nc(C(=O)NCc3cncc(F)c3)cs2)cccc(Br)c1Cl 565,N1(C(C=CCC)=O)CCC2(NC(C3CCC(=O)NC3)=O)CCCC12 566,c1(C(=O)NC2CCC(C)(CNC(CCCC)=O)C2)ncc(N)cc1C 567,Cc1nn(C)c(Cl)c1CC(=O)NCCCCCCNC(C1CCC(C)(C)CO1)=O 568,C#CCC(O)C(=O)NCC1CC1NC(c1cccnc1OCCCC)=O 569,c1(C(=O)Nc2csc(CO)c2)ccc2c(c1)OCCN2.N12CC3C(C3C1)CC2=O 570,C(=O)(C1=CCC(C)(C)CC1)NCC(CC)NC(=O)CCc1ccc(=N)[nH]c1 571,Cc1ccc(C)c(C2CCCN2C(=O)NCCCc2nccs2)c1N 572,C(=O)(C1=NN2CCCN=C2N1)NC(C)(CO)c1nn[nH]n1 573,CC1(C)OCCC1CC(=O)NCCc1ocnc1CNC(=O)CN1CC2CC2C1 574,C1(C(=O)NC2C(CNC(c3ccc(CCC)cc3)=O)C2)CC2CC(=O)C1O2 575,C1(CNC(C2CC(CC)(CC)C2)=O)CC2(CO1)CN(C(=O)C=CSC)C2 576,N1(C(CCC=C)=O)CCC(CNC(C2CCC(F)CC2)=O)(COC)CC1 577,N1(C(c2ccc(C#C)cc2C)=O)CCC(NC(=O)C(O)C=C)C2(CCC2)C1 578,c1(OC)ccncc1CC(N1CC2CC1C2NC(=O)C(CO)NC(=O)C(C)C)=O 579,C1(NC(C(C)(C)c2cnsc2)=O)CCC(F)(CNC(c2ccc(O)nc2)=O)C1 580,c1(NCC2(NC(=O)C=CC3CCCO3)C(C)CCCC2)ncnn2cccc12 581,N1(C(CC2CCC(C)C2)=O)CC2(CCN2C(=O)CC(C)(F)F)C1 582,CCCCCS(=O)(=O)CC(=O)N1C2CCCC1CN(C(=O)CCSC1CCCC1)C2 583,C1(C(=O)NCC2CCN(C)C2)(CNC(=O)CC2COCCO2)CCCCC1 584,Cn1c(O)nc2cccc(C(N3CCCCC(NC(=O)CCS(C)(=O)=O)C3)=O)c12 585,c1(CC(=O)NC(C=CC(N2C(C)(CCC)CC2)=O)C)ccc(F)nc1 586,CC(C)(C(=O)NCC1CC(F)CN1C(C1CC(=C2CCC2)C1)=O)C1=CCSCC1 587,C1(CNC(c2n(C)cc(F)c2)=O)COCCN(C(C2(C)CCOCC2)=O)C1 588,N1(C(c2nc(CC)sc2N)=O)CC2(C)CN(C(c3csc(C)c3C)=O)CC2(C)C1 589,CCCCC#CC(C)(C)NC(=O)CC(CC)N(C(=O)CCc1nccn1C)C 590,Cc1cc(C(=O)NC2C=CC(CNC(c3ccncc3Br)=O)C2)[nH]c1C 591,N1(Cc2c(C)ccnc2)CCC(NC(=O)Cc2cccc(F)c2)C(F)C1 592,CC(=O)C(C)CC(C)C(=O)NCC=CCC(=O)Nc1ccccc1C(C)C 593,C1(CCOC)CN(C(C2CC(C)(C)C2)=O)CCN1C(c1ccc(F)cc1F)=O 594,C(=O)(C(C)CC1CC1)NCC(C1CCCC1)NC(CSCC=C)=O 595,Cc1ccn(C)c(=O)c1NC(=O)CC1CCCC(NC(=O)CCCF)C1 596,Cc1cncc(C(N2CCC(CNC(c3cc(N)cc(O)n3)=O)CC2)=O)c1C 597,c1(C(N2CC(C)(NC(C3C(C)C3C)=O)C2)=O)c(Br)nnn1C 598,c1(NC(C(C)Cc2ccc(-c3ccccc3)cc2)=O)ccc(O)c(Br)c1 599,N1(C(c2c[nH]c(C)cc2=O)=O)CCC(NCc2ccc(C(=O)OC)cc2)C(C)C1 600,N1(C(C(COC)O)=O)CC(CNC(c2cncn2-c2cccn2C)=O)C(C)(C)C1 601,C12(CNC(C(CC(C)C)SC)=O)CC(C(N)=O)(C1)C1(CN(C(=O)C=C(Cl)Cl)C1)O2 602,c1(CC(=O)NCC2(COCC(=C)C)COC2)cc(F)ccc1F.C1C(=O)N1 603,N1(C(c2cscc2F)=O)CCN(C(c2cccc(F)c2Cl)=O)C2COCC12 604,CC1(CNC(=O)Cc2ccc(C3CC3)cc2)CN(C(=O)C2=CSCCO2)CCO1 605,C1(C(N)=O)CCCC(C(=O)NCCNC(=O)C(=O)Nc2ccc(OCCO)cc2)C1 606,c1(SCC(N2CCC(C(=O)NC(=O)OC)C2)=O)nc2ccccc2[nH]1 607,c1(C(N(CCC)CCNC(=O)C(F)CC2CC2)=O)ccc2c(C)nn(C)c2n1 608,C=C(C)CC(C)C(=O)NCC(=O)NOC(C)C 609,C1(NC(CSC(C)(C)C)=O)CC2(NC(=O)CC3CC4CCC3CC4)COC1C2 610,C#CC1CCCN(C(=O)COC(C)(C)CNC(=O)CC(C)C(F)F)CC1 611,Cc1cc(C(=O)N(C)CCc2cn(CC3CNC(=O)O3)nn2)ccc1S(N)(=O)=O 612,C(c1ccc([N+](=O)[O-])cc1)=CC(=O)NC1CN(C(c2cc(Cl)cnn2)=O)C1 613,C(=O)(C(C(C)(C)O)NC(C1(c2ccno2)CC1)=O)NCCC(CC)(F)F 614,C1(F)(C(N(CCC(C)NC(C2CCCC23CC3)=O)C)=O)CCC(F)(F)CC1 615,C1(NC(C(c2ccc(C)s2)C)=O)CCCC2CN(c3cc(Cl)nc(C)n3)CC12 616,C1(CNC(CCOCCCNC(C(C)=C2CCC2)=O)=O)CC(O)C12CCC2 617,C(=O)(C1=CCS(=O)(=O)C1)N1CC(N(C(=O)Cc2ccc(F)cc2Cl)C)C2(C1)CC2 618,C1(C2CC2)(NC(=O)C(F)n2cccn2)CCN(C(c2ccc(Cl)o2)=O)C1 619,C1(C)(CC(=O)NC2CN(C(CCOCCOC)=O)C(C)C2)CCS(=O)(=O)N1 620,C=C(C(=O)N(CCC(=O)OC)CC=Cc1ccc(OC)c(OC)c1)C1CCCC1 621,c1(OC)ccc(C(N2CCCC2(C)C(N2CCC2c2ccccc2)=O)=O)cn1 622,N1(C(CS(CC)=O)=O)CCN(C(=O)CCC(=O)NC)C(CO)C1 623,C1(CSC)CCCN(C(=O)CN(C(C2CC(F)(F)C2)=O)C(C)C)C1 624,C1(CNC(=O)CC2CCCCO2)CCCN(C(c2ccnc(SC3CC3)c2)=O)C1 625,c1(C(=O)NC(C)CNC(=O)C(C)n2cnnn2)c(O)cc(Cl)cc1F 626,c1(CC)cccc(C(=O)NC2(C(=O)NCC(C)CC3CC3)CC2(C)C)n1 627,C1(C(=O)OCc2cccc(CCCCC)n2)Cc2cccnc2C1 628,c1(OC)oc(C)nc1C(=O)NCC1CCN(C(=O)Cc2ccn(C)n2)C1 629,C(=O)(C(C)(C)C(=O)N(CC(C)N(C(=O)C(C)SC(C)C)C)C)OC 630,c1(-c2cn(C3CC(C(=O)NCC(CC)(C)OC)C3)nn2)ccc(C)cc1.C1CC1 631,c1(CC)ccccc1Br.n12cc(nn1)CC(=O)NCC2.C1C(=O)N1CC 632,CS(=O)(=O)C1(C(=O)NC2CCCC2NC(=O)CC2CCCO2)CCC1 633,c1(CC)[nH]c(=N)sc1C(=O)NCC1CCCC1NC(=O)C=CSC 634,C1(COC)CN(C(c2ccc(Cl)cn2)=O)CCN1C(c1ccc(F)c(CO)c1)=O 635,CCC(CC)C(=O)N1CC=CC1(C(=O)NC1C(C)C1(C)C)COC 636,c1(OCC)ccc(OC)c(C2CC2C(=O)NCC(C)CN(C)C)c1 637,N1(C(C2(CC#C)CCN(C(=O)CC(C3CC3)C3CC3)C2)=O)CC2(COC(=O)C2)C1 638,C1(C)(CNC(C(CC)N(CC)CC)=O)CCN(C(C2CCCOCC2)=O)CC1 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657,c1(C(N2CCCCC(NC(C(C(CC)C)C)=O)C2)=O)cc(OC)cc(OC)c1N 658,CC(C(=O)N1CCC(CN(C)C(c2ccc(Cl)o2)=O)CC1)C(C)(C)C 659,c1(CCC)onc(C)c1C(=O)NCC(F)CNC(=O)C(F)(F)c1ccccn1 660,N#Cc1ccc2cc(C(=O)NCCCCNC(c3ccc(Br)o3)=O)ccc2c1 661,Cc1c(CN2CCCC(C(=O)N(CCC(C)(C)O)C)C2)cnn1C 662,C(C(C(=O)NCC1CC1C(=O)OC)C(C)C)NC(C=C(CCC)C)=O 663,C(N=c1ncnc(N2CCCCC2)[nH]1)c1c(COC)snn1 664,Cc1c(F)ccc(N)c1C(N1CC(CNC(=O)CNC(=O)C2CC2)C(C)C1)=O 665,N1(C(c2cc(CC)no2)=O)CC(NC(=O)C(C)NC(=O)NC)CC2(CC2)C1 666,n1(CC)nc(C(=O)NCCC2CN(C(=O)CC(F)F)C2)c(Cl)c1Br 667,[N-]=[N+]=NC1(C(N2CCC(OCCO)CC2)=O)CCN(C(=O)Cc2ccco2)C1 668,N1(C(C2(OC)CCN(C(C=CCC)=O)C2)=O)CCCC(C)(C#N)C1 669,Cc1nc(C2OCCC2C(=O)NCCCC(C)O)n[nH]1 670,N1(C(=O)Cc2cc[nH]n2)CCN(C(C2CS(=O)(=O)CCO2)=O)C(CC2CC2)C1 671,C12(NC(CC(C(C)C)O)=O)CCCCC1CN(C(c1ccc(Cl)c(F)c1F)=O)C2 672,c1(NC(C2(F)CCN(Cc3n(CC)ncc3)C2)=O)ccc(C)nc1F 673,c1(OC)nc(C)ncc1C(=O)NC1CCN(C(c2cc(CN(C)C)on2)=O)C1C 674,c1(NC(C2C(C(C)C)OCC2)=O)cccc(CC2CCNCC2)c1 675,c1(C(N2C(CNC(C3CCC(C)(C)CC3)=O)CC2)=O)ccc(F)cc1[N+](=O)[O-] 676,CCC1=NOC(C(N2CC3CC3(CNC(=O)C(F)=C3CCC3)C2)=O)C1 677,CCCC(C(=O)NC(c1ncccc1F)C)NC(c1csc(Cl)n1)=O 678,N1(C(=O)Nc2scc(COC)n2)CC2CC(C(=O)OC)C1C2 679,Cc1cc(=NC2COCCOC2)[nH]c(=NCc2c(F)c(F)c(F)c(F)c2F)[nH]1 680,c1(C(N(CC(C)NC(c2cnc(O)s2)=O)CC)=O)cc(C(F)(F)F)cnc1C 681,C(c1ccccc1OC)=CC(=O)NCC(CNC(c1cc(CCC)nn1C)=O)F 682,N1(C(CCSCCC)=O)CCCC2C1CCN2C(=O)C(C)CC1CCCC1 683,c1(C(=O)NCC(C(C)C)NC(C2CCCN(CC)C2)=O)cn(C)c(C)cc1=O 684,C1(NCc2cn(C3CC(C(=O)OC)C3)nn2)(CC2CCCO2)CCC1(C)C 685,CC(CS(C)(=O)=O)C(=O)NC1CN(C(c2cc(O)c(O)c(O)c2)=O)CC1F 686,CN1C(=O)CCCC1C(=O)NC1CN(C(C2(C#N)CCCCC2)=O)CC1C(F)F 687,CCCC(C(=O)N1CCC(CC(C)NC(C2CC2C#N)=O)CC1)OCC 688,n1(CC(=O)NC(c2csc(CC(F)F)n2)C)cc(CC(C2CCOCC2)=O)nn1.N 689,C1(CNC(CNC(=O)C2CC2)=O)CCN(C(c2cc(=O)c(O)c[nH]2)=O)C12CCC2 690,O=C(CC1COCCN1C(=O)CCCOc1ccc(Cl)cc1)N=c1cc(Br)[nH][nH]1 691,c1(CC)cc(C)c(C(=O)NCc2ncccc2C(=O)NOCC2CCOCC2)o1 692,Cc1nc(N2CCCC(C)(CNC(C34CCC(C)(C3)OC4)=O)C2)cc(C#N)n1 693,c1(N2CCCC(C(N(C)CC3(OC)CCOC3)=O)C2)nc(=N)nc(C(C)(C)C)[nH]1 694,C=CCC(C(=O)N1CC=CC1)NC(=O)CCCNC(C)=O 695,N1(C(c2c(NC)scn2)=O)CCOC(CC(=O)NC(C)CCCCO)C1 696,c1(NC(C2N(C(C(C)n3cccn3)=O)C3C(C2)C3)=O)ccc(F)c(Cl)c1 697,C(CCN=c1[nH]c(C)ncc1F)OCCSC 698,CCCC(CC(=O)NCC1(O)CCCC1(C)C)NC(=O)C(C)(C)C(N)=O 699,c12nn(C)cc1NC2c1nnnn1C1COC1.c1(CSC)cc(C(C)C)no1 700,c1(CC(N2C(Cn3cc(CCC(C)(C)O)nn3)C=CC2)=O)cc(F)ccc1F 701,CCC1=C(C(=O)NC2CCC2NC(=O)C(N2CCN(C)CC2)C)CCCO1 702,C1(CC(=O)NC(C(=O)N(C23CC(C2)C3)CCOC)C)CCCCN1C 703,C1(CCCN(C(=O)CONC(=O)C2CCOC2)CCO)(CO)CCOC1 704,Cc1nc(NC2CN(C(C3CC(C)CO3)=O)CCC2C(F)(F)F)c(C)c(O)n1 705,C1(CNC(CC(C)C)=O)CN(C(C2(c3cccs3)CC2)=O)CC1C 706,c1(CC(C)NC(=O)NC(C2(O)COC2)C)ccccc1F 707,c1(CC)cc(C(=O)NC2C3CN(C(c4cc(C)c(Cl)cn4)=O)CC23)ccc1F 708,CC1CC(NC(c2ccc(CCF)cc2)=O)CN1C(=O)C=C1CC1 709,c1(C(N2CCC(CCCNC(C3CCCC3)=O)CC2)=O)c(O)cc(F)cc1F 710,N1(C(CC(C)NC(c2c(C)noc2N)=O)=O)CCC2(CCC2)C1 711,c1(C(=O)OC)ccc(C(=O)NC2CN(Cc3cc(Br)ccc3Cl)C2)cc1Br 712,c1(NC(C(C)NC(c2ccc(CO)nc2)=O)=O)cccc2ccoc12 713,C(=O)(C(O)C1=CCCCC1)NCCCCCCC(=O)NCC1CCC(C)CC1 714,N1(C(C(CCC)C)=O)CCC2(CNC(C3(C(N)=O)CC3)=O)CCCCC12 715,c1(C(=O)NC(C(C)NC(C2COCCO2)=O)(C)C)ccc2cn(C)nc2c1 716,c1(NC(c2c(C)nc(-c3cccc(CO)c3C)s2)=O)ncc(Cl)cc1C(=O)N(C)C 717,N1(C(C(CCCC)O)=O)CC2CCCC(C1)N2C(c1[nH]cnc1CC)=O 718,C1(C(CC)NC(=O)CCCn2cc(C(C)(C)C(=O)O)nn2)COCCO1 719,C1(C(N2CCC(CCOC)(NC(=O)CCOCC(F)F)C2)=O)CCCC(C)(C)O1 720,C1(C(=O)OCC)CC(NC)CCN1CC1COCCO1 721,N1(C(c2cc(C)c(C)o2)=O)CCC(C(=O)NCCC2CCCC2(C)C)C(C)(C)C1 722,N1(C(C2(C)CC(C)OCC2)=O)CC(C)OC2(CCN(C(C3CCCSC3)=O)C2)C1 723,O=C(C(O)CC(F)F)NCc1cc(Cl)cnc1Cl 724,N1(C(C(C)C(F)F)=O)CCC2CC2(C(N2CCC3C(O)CC23)=O)CC1 725,O=C(CC(C(F)F)n1cccn1)N1CC(NC(C2CC(O)C2)=O)C(C(F)(F)F)C1 726,c1(C(=O)OCC)ncc(S(=O)(=O)N2CCC(F)CC2COC(C2(CC)CC2)=O)s1 727,c1(C(=O)NCC(Cn2cc(C(C)OC)nn2)(C)C)c(Cl)n[nH]c1C1CC1.C 728,C1(CNC(c2cccs2)=O)CN(C(c2c[nH]nc2Br)=O)CCO1 729,c1(C(N(C2CCCN(C(c3ccc(NC)nc3)=O)C2)CC)=O)cccc(N)c1F 730,C1(CC(=O)NC2C(C)C2(C)C)C2CCCC2N1C(C1(C2CC2)CC1)=O 731,C1(C(=O)NCC(C)NC(=O)CN2CC(C)(C)C2)COc2ccc(O)cc2O1 732,C(=O)(CS(=O)(=O)c1ccc(Cl)cc1)N1C2C(NC(CCCCCC#C)=O)C(C2)C1 733,C1(C(=O)OCC23CC(C(=O)OC)(C2)C3)CCCC(NC(=O)CC2CC2)C1 734,N1(C(C(=O)Nc2ccc(OCCOC)cc2)=O)CCn2cc(C)nc2C1 735,C1(c2nnnn2Cc2ccco2)(CCC2C(=O)NCCC2)CC2CC(OC)C2C1 736,CC(C)CC(C(=O)NC)NC1CC1.c1(CCCOC(C2CC2C=O)=O)cccnn1 737,C1(C(=O)NC(C2C(C(=O)OC)C2)C)CC=CCN1C(c1csc(Cl)n1)=O 738,N1(C(c2sc(CCC)c(CC)c2)=O)CCN(C(=O)CNc2ccccn2)C(C)C1 739,C1(N(C(C=CC)=O)C(c2cnc(N3CCCCC3)nc2)=O)CCS(=O)(=O)C1 740,C(=O)(C#CC1CCCO1)N1CC(NC(c2c(O)ccc(C)c2)=O)C2(C1)CC2 741,S(=O)(=O)(c1cc(C(=O)O)ccc1Cl)N1C(C)CC(NC(=O)OC(C)(C)C)CC1 742,CCC(C(=O)NCCCC(C)NC(c1ccc(C)nc1N)=O)C(C)C 743,C1(CC(N2CC(SCC)(OC)C2)=O)CC(NC(c2ccoc2)=O)C1(C)C 744,N1(C(C2CC(C)CN2C(c2c(Cl)cnn2C)=O)=O)CCC(=O)N(C)CC1 745,C1(C(N(CC(C)NC(=O)C=CC(=O)N(C)C)CC)=O)CN(c2nncs2)C1.C 746,Cc1ccc(=N)[nH]c1C(N1CCN(C(=O)C(C)C2CCCC2)CC1C)=O 747,C1(C(C(C)C)NC(C(F)OC)=O)CCN(C(c2ccccc2OC(F)F)=O)CC1 748,C1(C)(NC(CC2CCCN(C(C(C)NC(CC)=O)=O)CC2)=O)CCC2(CC1)CC2 749,N1(C(c2cc(CC)oc2C)=O)C2CCC(C2)C1C(=O)NC1CCNC(=O)C1 750,c1(NC(C(=O)Nc2nnc(CCC)s2)=O)ccc(OCC(=O)OC)c(Cl)c1 751,c1(OCC)nc(N(CCCN(C(=O)C(CO)c2ccccc2)C)C)ncc1Cl 752,C1(C(=O)N(C2CCC(NC(=O)C(C)NC=O)CC2)C)(OC)CCCCC1 753,N1(C(c2c(C)nncc2)=O)CCC(n2cccn2)(CNC(C2CCSCC2)=O)CC1 754,N1(C(C(OC)OC)=O)CC(CO)C2(C1)CN(C(=O)C(CC(C)C)NC(C)=O)C2 755,Cc1cccc(CCC(=O)NCC23CC2CN(C(=O)Cn2cnnc2)C3)c1Br 756,c1(NC(CNC(C2(C)CCC(C)C2)=O)C2CC2)cc(=O)n2cc(Cl)ccc2n1 757,n1(CC(=O)NCC(CC)N(C(=O)C(F)CC2CCC2)CC2CC2)ccnc1C 758,C1(C(N(C(C)CNC(c2cnccc2Cl)=O)CC)=O)CCCCN1C 759,C1(C(=O)NCC2(NC(C3OCCN(C)C3=O)=O)CC2)CCc2nnc(O)cc2C1 760,C#CCC(CC(=O)NCc1ccncn1)NC(c1ccc(C)cc1F)=O 761,c1(N2C(C(=O)NCc3cn(C(C)C)nc3)CC(F)C2)ncnc2c(Br)csc12 762,C1(C(=O)NCC2N(C(C34OCCC(C)(C3)C4)=O)CCOC2)CCc2ccnn2C1 763,C1(CC(=O)NCC2N(C(c3ccc(C)o3)=O)CCC2)COCC(C)O1 764,C(=O)(CCCCCC(C)(C)C)NC1(CO)CCN(C(C=C(CC)CC)=O)C1 765,N1(C(C=C(C)C)=O)CCCC2(CCN(C(c3c(Cl)ccc(Cl)c3O)=O)CC2)C1 766,C1(NC(CCC(C)N(C)C)=O)CC2(C1)CC(NC(C1CCC1C)=O)C2 767,Cc1cc(C(=O)NC2CCC2CNC(c2cn(CC(N)=O)nn2)=O)n[nH]1 768,c1(CC(=O)NCC(CN(C(C(C2CCCC2)OC)=O)C)O)cccc2occc12 769,C(=O)(C1=CCCCCC1)NC1C(N(C)C(C2CC23CCOCC3)=O)CCCC1 770,C1(C)(C(=O)NCC2CCCC(NC(COCC#C)=O)C2)CCOC(C)C1 771,c1(NC)c(C(=O)NC(C)(C)CNC(=O)CC2CC3CC3C2)cccc1[N+](=O)[O-] 772,Cc1cnn(C(C)C(=O)NCCCCNC(=O)C(C)OCCN(C)C)c1 773,C(=O)(CCS(=O)(=O)CC(C)C)NC(C1CN(C(C2CCOC2C(F)(F)F)=O)C1)C 774,N1(C(c2c(CC)nccn2)=O)CCC2(CC1)CCN2C(=O)CCC1CCOC1 775,C1(CC)CCN(C(c2coc(CO)c2)=O)C(C(=O)NC(COC)C(C)C)C1 776,c1(C(N2CCCC(CN(C(C3CC(C(=O)OC)C3)=O)C)C2)=O)cnc(O)c(C)c1 777,C1(C)(C(N(CCNC(=O)C(C)(CC)CO)CC)=O)CC2(C1)CC(F)(F)C2 778,N1(C(C2C(CC)C2)=O)CC2(CCN(C(c3sc(Cl)c(Cl)c3OC)=O)CC2)CC1C 779,C1(NC(CN(C)C(=O)C2CC2)=O)CCC(CC(N2CCCC2CO)=O)CC1 780,CCC(F)(F)C(C)(C)C(=O)NC1CCCCCC1NC(=O)CC1CCN(C)CC1 781,Cc1cnc(CCCC(=O)NCCN(C(=O)C(C)Oc2cccnc2)C(C)C)o1 782,C1(CC(=O)NC2CC2(F)F)CCN(C(C2CC2(Cl)Cl)=O)C1 783,C#CCCN=C(NCC(c1cc(C)oc1C)C)NC1CC1F 784,Cc1cccc(CC(=O)NC2CC(CNC(C3CC4CCN4C3)=O)CC2O)c1 785,C1(NC(CCCc2cc(C)no2)=O)CC2CN(C(C3CCC3)=O)CC2C1 786,C=CCCCCC(=O)N1C2CCC1C(C(=O)N(C)CC1CCCOC1)C2 787,Cc1cc(Br)oc1C(N1CCC(Cn2cc(CC(CO)C3CC3)nn2)CC1)=O 788,S(=O)(=O)(c1ccc(=NC(CCO)C2CC2)[nH]c1)N(CCCc1c(C)cccn1)C 789,C1(c2cn(CCN(C(CC(C)(C)SC)=O)CC)nn2)COc2ccccc2C1 790,c1(C(C)NC(CCN(C(=O)CC2CCCCO2)CC)=O)ncccc1F 791,C1(NC(=O)COCCN(C)C)CCC(F)(C(N2CCC(COC)(OC)C2)=O)CC1 792,N1(C(CCCOCCC)=O)CC(O)CC1C(=O)Nc1cnccc1C1CC1 793,N1(C(C=C(C)C)=O)CCN(C(c2ccc(C(C)(C)C)cc2C)=O)C(C(F)(F)F)C1 794,CCCCC(C)CCC(=O)NCCCOCCNC(c1cc2nnn(C)c2s1)=O 795,C1(C(=O)NCC(C2(O)CN(C(c3cc(C)[nH]n3)=O)C2)(C)C)CCC(=C(F)F)CC1 796,N1(C(C(CC)(C)CC)=O)CCCC2(C1)C(NC(=O)C(C)SC)CCN2C 797,C(c1ccc([N+](=O)[O-])s1)=CC(=O)NC1CCN(C(CSCC(=O)OC)=O)C(C)C1 798,c1(C(N2C(CCOC)CN(C(C3CC3(C)C)=O)CC2)=O)nc(C)n2ccccc12 799,c1(C(=O)NC23CCN(C(c4ccc(Br)o4)=O)CC2C3)ccc2occc2c1 800,CCN=C(NCCNCCOCCOC)NC(C)(C)C.C12CCC(C1)NC2=O 801,c1(OC(C(=O)NC2C(CNC(CCC=CCC=C)=O)C2)CC)cccc(C)c1 802,c1(CN(C(=O)COCCF)CC)ccccc1C(N1CCCC(COC)C1)=O 803,c1(C(N(C2CN(C(CSCC=C)=O)CC2F)C)=O)cc(Cl)c(F)cc1C 804,c1(C(=O)NCC(CN(C(c2c(C)nn(C)n2)=O)C)(C)C)nc2ncccn2n1 805,C1(F)(CNC(C2(OCC)CCOC2)=O)CCCN(C(=O)C=Cc2ccsc2)CC1 806,C(CC(C(C)(C)C)NC(=O)C1=CSCS1)N(C(=O)C(=O)NC1CC1)C 807,C1(NC(=O)NCc2ccc(Cl)c(C(F)(F)F)c2)CNCCS(=O)(=O)C1 808,Cc1ncc(-c2cn(Cc3ncoc3CNC(=O)C(C)(C)Br)nn2)[nH]1 809,Cc1cccc(C(N2CCC(C(=O)N(CC(O)C(C)(C)C)C)C23CC3)=O)c1C#N 810,CCC(CC(C)C)C(=O)N(C)CC1COCCN1C(c1nn[nH]c1Cl)=O 811,S(=O)(=O)(c1ccc(Br)cc1NCCc1ncc(C)cn1)N(C(CC)CO)C 812,N1(C(C2C(CC)CCN2C(c2ccc(N)cn2)=O)=O)CCC2(CCCO2)CC1 813,N1(C(CC2CC(C)N(C(c3cc(N)cc(F)c3)=O)C2)=O)CC2(CCC(=O)NC2)C1 814,N1(C(C(CC)CC2CCCC2)=O)CC2CC(NC(c3cc(Cl)cc(Cl)c3)=O)C1C2 815,N1(C(CSCCOC)=O)CCCC2C1CCN2C(c1ccc2ccn(C)c2c1)=O 816,c1(CNC(COCCOCCOC)=O)cccnc1C.n1(CC(=O)N)ncccc1=O 817,c1(C(C)C)ccc(C(O)C(=O)N(C(C)CNC(C2(C)CNC(=O)C2)=O)C)cc1 818,C(=O)(C(F)(F)C(F)(F)F)NCC1(C)CN(C(c2cscc2C#N)=O)CCO1 819,C1(NC(C2CCCc3ccccc32)=O)CC2CCC(C1)N2C(c1ccc(Br)s1)=O 820,C1(C(NOCCCC#C)=O)COCCN1C(C1CCCN(C)C1)=O 821,c1(C(c2n(CC)nnn2)NCC(c2nnnn2C)OC)ccncc1Br 822,CCC(C)(CO)C(N=c1[nH]c(N(CC(Cl)Cl)C)nc2ccsc12)c1nncn1C 823,C1(N(C(CN(CC)CC)=O)C)CCCC2CN(C(=O)CCc3cn(C)nn3)CC12 824,c1(C(N2CCC(N3C(CSC)CCC3)C2=O)=O)cccc2c1OCO2 825,C(C(C)(C)C(=O)NC(C1CN(C(=O)CC(C)C2CCCO2)C1)C)OC(C)C 826,c1(C(=O)NCC(C)(C)NC(c2c[nH]ccc2=N)=O)cccc2c1CCOC2 827,C1CS(=O)(=O)N1.C1(CNS(CC)(=O)=O)CCC(O)C1 828,C(=O)(C(CCC(C)C)NC(c1ccncc1O)=O)N1C(COC)CCC1 829,c1(C(=O)NC2CC(CNC(C(CC)F)=O)C2)cc(C)c2c(c1)CCC2 830,Cc1nccc(C(=O)NCc2cc(C(=O)NC3CCCC3C)n(C)n2)n1 831,c1(C(=O)NC2C3CN(C(COCC)=O)C2CC3)cc2ccc(NC(C)C)cc2[nH]1 832,N1(C(CC2C(NC(C(CSC)(C)C)=O)CC2O)=O)CCCC(O)(C(N)=O)C1 833,c1(C(N(C2CC(=O)CCC(=O)N2)CC(=O)OC(C)(C)C)=O)cc2ccccc2[nH]1 834,c1(C(=O)OC)cc(C(=O)NCC23CC2CN(C(C2CC(N(C)C)C2)=O)C3)n(C)n1 835,C(=O)(C(F)(F)CC(C)C)N1CCCC(CC=C)(NC(c2ncccc2O)=O)C1 836,c1(C(=O)O)ccnc(C2CCN(CCCN3CCOC3=O)CC2)c1 837,N1(C(CCC(=O)NC)=O)CCC(NC(C2CCN2C2CCCC2)=O)C(C)C1 838,c1(CN2C(CC(=O)Nc3ncc(C)nc3Br)COCC2)ccc2nc(C)oc2c1 839,C1(NC(Cn2ncc(C)c2)=O)CCC(C)N(C(=O)Cc2cncn2C)C1 840,C12(CNC(C(C3CC3)OC)=O)CCCC1N(C(C1CCC(=O)N(C)C1)=O)CCC2 841,c1(CNC2(c3n(CCCC)nnn3)COC(C)(C)C2)ccc2[nH]nc(F)c2c1 842,CC1CCC(C)(C(N2CCN(c3nccc(C#N)n3)C(CCO)C2)=O)CC1 843,N1(C(C(C)N(C(C)=O)C)=O)CC2C(CNC(c3cc[nH]c3C3CCCC3)=O)C2C1 844,N1(C(C2CC(C#N)C2)=O)CCCC2(NC(=O)Cc3cc(O)nnc3O)CCCC12 845,c1(C(N2CC(NC(C(C)(C)F)=O)C2)=O)cc(Cl)ncc1Br 846,Cc1[nH]cc([N+](=O)[O-])c(=O)c1C(=O)NC1CCCC1NC(=O)C1=CCOC1 847,c1(C(N2CCC(O)(CN(C(C(CC)O)=O)C)C2)=O)cnc2ccccn2c1=O 848,C#CC1CCCC1NC(=O)CC(CC1CC1)NC(=O)C=CC1CCCC1 849,Cc1cc(F)c(C(=O)N(C2CN(C(=O)C(C)(C)c3cccs3)C2)C)cc1F 850,c1(C(=O)NC2CCC(N(C(c3nc(C)n(C)c3)=O)C)C2)ccnc2ccccc12 851,C(=O)(C(C)C(O)CC(C)C)N(CCCNC(CC=C)=O)C(C)C 852,c1(C(=O)NCC(C)NC(c2c(SC)cccc2)=O)cnn2c(C)ccnc12 853,C(=O)(C1CCCc2n[nH]cc21)N1CC(CNC(C=CC)=O)C(F)(F)CC1 854,c1(C(=O)OC)ccc(NC(c2cccc(C3CC3(F)F)c2)=O)c(OC)c1Cl 855,c1(COC)nn(C)c(Cl)c1C(N1CCC(F)C(NC(=O)Cc2cc(C)no2)C1)=O 856,c1(C(F)(F)F)cccc(-c2nc(O)n[nH]2)c1.CC1CCNC(=O)C(=O)N1 857,c1(C(N(CC(CC)NC(=O)CCCN=[N+]=[N-])C)=O)cc2cncn2c(O)n1 858,c1(C(=O)NCC(CCC)C(=O)NCc2scnc2C)n[nH]c2ccccc12 859,CC1CCCC(C)N1C(=O)C(N1CCN(Cn2cc(C(F)(F)CO)nn2)CC1)=O 860,c1(C(=O)NCC(CC)NC(C2CC(C)(C)C2)=O)cc(OC)cc2c1NC(=O)CO2 861,c1(N(CC#C)C)ccc(CNCC(=O)OCCc2ccccc2CS)cc1.SCC 862,c1(NC(=O)NC2C(NC(=O)CCN3CCOC3=O)CC2)ccc(C2CC2)cn1 863,O=C(C1SCCc2sccc21)N1CC(c2cn(CC3CCOCC3)nn2)C1 864,N1(C(C2CCC(=O)O2)=O)CC=C(C(=O)NCC2C3COCC23)C1 865,c1(C(=O)NC(CCN(C)C)C(=O)NC2CCN(CCF)C2)ccnc(O)c1F 866,c1(C(C)(C)C(=O)NC2CCC2NC(C2CCCN2S(C)(=O)=O)=O)cccnc1F 867,C1(CNC(C2C(C)(C)C2)=O)CCC2(CCN(C(c3n[nH]cc3[N+](=O)[O-])=O)CC2)O1 868,c1(OC)cc(C(C)NC(=O)Nc2c(OC)ccc(F)c2OC)c(F)cc1F 869,C1(CC(C)C)(C(=O)NCC2(NC(=O)CC(C)(C)C)CCOC2)CCNC1=O 870,c1(N(C)C)ccc(-c2cccc(NC(C3(C(C)(C)O)CCC3)=O)n2)cc1 871,C1(NC(CC(C=C)(C)C)=O)CC2CC(C1)N(C(=O)CC(=O)N(C)C)C2 872,N1(C(c2on(C)c(=O)c2)=O)CCC(NC(c2ccsn2)=O)CC(C)(C)C1 873,N1(C(c2ccc(CNC(CCSC)=O)cn2)=O)CC(=O)NC2(CC2)C1 874,N1(C(c2cc(C)sc2)=O)CC(CNC(C2CCCC(C)O2)=O)CC1C 875,C(=O)(C1CCc2snnc21)NCC(c1ccccc1)NC(=O)C=CC1CC1 876,c1(NC2C(C)CN(C(C=C(C)C(F)F)=O)CC2C)cc(C)ccc1[N+](=O)[O-] 877,C1(CNC(c2ccc(CC)o2)=O)CCCCN(C(=O)C=C(C)C2CC2)C1 878,N1(CC(N2CCOCC(C(CC)CC)C2)C)CCc2ccccc21 879,C1(CNC(=O)CC2(C)CCCO2)CN(CC2CCCC2)CCC1(F)F 880,C(C1=CCCN(C(=O)C=CC2(C)COC2)C1)NC(c1c(C)occ1)=O 881,N1(C(c2n(C(C)C)nnc2)=O)CCC(O)(C(C)CNC(=O)CCn2cccn2)C1 882,N1(CC(=O)NC2C(NC(C3CCC(CC)CC3)=O)COC2)C(=O)NC(C)(C)C1=O 883,CC1(C)CCCCCC1NC(=O)C(CNC(C1OC2CCC1C2)=O)C(C)(C)C 884,C1(C(=O)NC2CCC(O)CC2)C2CC(CC2F)N1C(C1(Br)CC1)=O 885,N#Cc1c(CN2CC3CC2CN3S(=O)(=O)Cc2ccc(Cl)cc2)cccc1Cl 886,N1(C(=O)OC)CCC(C(=O)NCC2CCN2C(c2ncsc2C(C)C)=O)CC1 887,N1(C(C2(CC)CCN(C(C3CC4C=CC3CC4)=O)C2)=O)CCC2(CCCCC2)C1 888,C1(CCC)(NC(=O)CC2CC(O)CN2C(c2cccnn2)=O)CCNC1=O 889,N1(C(CCCOCC)=O)CC(NC(=O)CC2CCCC3(CC3)C2)CC2(CCC2)C1 890,C1(CNC(C(=O)NC(C)C)=O)CC2(CCC2)CN1C(C1CCCC1C(C)C)=O 891,c1(C(=O)OC)ccc(C(=O)NCC2N(C(=O)CC3CC(CF)C3)CCC2)cc1C 892,c1(OCC)cc(-c2cnccc2C(=O)NCCc2ccc(F)cc2)ccc1F 893,C1(C(C)=O)C(C(=O)N(CC(=O)NC2CCCS2)CC2CC2)C1(C)C 894,c1(C(N2CCC(OCCNC(C3(CC)CCOC3)=O)C2)=O)c([N+](=O)[O-])cnn1C 895,N1(C(C(F)OC)=O)CCN(C(=O)CC2CCN(S(C)(=O)=O)CC2)C2COCC12 896,S(=O)(=O)(C1CC12CCC2)NC(c1ncccc1C(F)(F)F)C 897,c1(CN(C(c2ccc(O)nn2)C(=O)NC2C(C)CCC2)C)ccc2c(c1)N(C)CC2 898,N1(C(c2c(C)c(C3CC3)on2)=O)CC2CCCC1C2CNC(=O)Cn1cnnc1 899,Cc1cc(C(=O)NC2CC3CC2N(C(=O)COCc2cc(C)on2)C3)nc(C)c1 900,c1(C(N2CCN(C(C)=O)CC2)=O)cc2c(s1)CCN(C(C1CCC=CO1)=O)C2 901,CC1=C(C(=O)NCC2CN(C)CCN2C(=O)C(CO)NC(=O)C(C)C)CCO1 902,N1(C(C(C(CC)C)O)=O)CC2CCN(C(C3C4(CC4)C34CC4)=O)CC2C1 903,c1(C(N2CCC3CN(C(CCCSC)=O)CC32)=O)cc2cc(C)ccc2[nH]1 904,CCC(C)(F)C(=O)NC(C)CNC(C1(Sc2ccccc2)CC1)=O 905,O=C(CC1=CCCC1)NCc1ncccc1C(=O)NC1CCCCC12CC2 906,c1(N(CCCCN(C(=O)CC2COC(=O)C2)C)C)nnc(C2CC2)o1 907,CC1(C)CC2CCCC12NC(=O)C(C1(C)CC1)NC(=O)COCC1CCOC1 908,C1(OCCC(=O)NC(CCNC(Cn2c(C)ncc2)=O)(C)C)CCN(C)CC1 909,c1(OC)cc(O)ncc1C(N1CC2C(CNC(c3n[nH]cc3[N+](=O)[O-])=O)C2C1)=O 910,CCC(CC)C(=O)N1CC(O)CC1CNC(C1CCCN(c2nccs2)C1)=O 911,C(=O)(C(CO)C(F)(F)F)N1CCC(C)(CC(=O)NCCCOCC(F)F)C1 912,c1(C(N2C3C(NC(C(CC)(C)CO)=O)CC(C3)C2)=O)cc2ccnc(Cl)c2[nH]1 913,c1(C(=O)NCCCN(C)C(C2CCC(OC(F)F)C2)=O)cncc2ncccc12 914,C#CC1(C(=O)NCC(C)(C)C(C)O)CCN(C(=O)COCCCN=[N+]=[N-])C1 915,c1(C(=O)OC)ccnc(C)c1NC(C1CCN(Cc2ncccc2F)CC1O)=O 916,CCC(CCCC(=O)O)NC(=O)Nc1cccc(N(C)Cc2cccc(C)c2)c1 917,N1(C(=O)CC23CC(C2)C3)CCC2C1CCCN2C(=O)CCc1cccnc1 918,N1(C(=O)NCCCC2CC2(F)F)CC2CCCCC12c1ccccc1 919,C(CCC(O)C(=O)N(C1CCCC(O)C1)C)NC(C(C)NC(=O)C1CC1)=O 920,C1(CNC(C=C(C)CNC(=O)Cc2cn(C)nc2C)=O)CC(F)(F)CO1 921,N1(C(c2c(C(C)C)cco2)=O)CCC(NC(c2cc(Cl)cs2)=O)C(C)(C)C1 922,CC(C)C(C)(C)C(=O)NC1CN(C(C2CCCN(CC(F)F)C2)=O)CC1O 923,CC#CCCCC(=O)NC(CCc1ccccc1)C(C)NC(=O)C(=O)NC1CC1 924,Cc1nc(NC(=O)NC2CCC(O)(c3ccccc3)C2)sc1C 925,N1(C(c2c(N)c(Br)cc(Cl)c2)=O)CCC2CN(C(=O)CC3CC3)CCC12 926,c1(C(N2C(CCNC(c3c(CC)scn3)=O)CSCC2)=O)cc(F)c(O)c(F)c1 927,c1(COCC)cc(Cl)c(OC)c(OC)c1O.N12CSCC1C2=O 928,N1(C(c2c(O)cc(C)c(Br)c2)=O)CC(NC(C2COC2)=O)CC12CCOCC2 929,Cc1nc(C(N2CCC(C)(NC(c3cc(C(C)(C)C)c[nH]3)=O)C2)=O)c(C)o1 930,CC(C)CC(CNC(C1CCCCC(=O)C1)=O)C(=O)NC(c1nn(C)cc1O)C 931,c1(C(N2CC(Cn3cc(C(C)(C)C(N)=O)nn3)C2)=O)c[nH]c2ccncc12 932,c1(C2C(C(=O)NCCN(C(=O)Cc3ccnn3C)CCC)CC2)nnc(S)n1C 933,c1(C(N2CC(F)(CNC(c3cncc(C#C)c3)=O)C2)=O)cc2cc(Cl)cnc2[nH]1 934,C(=O)(C1CCCc2n[nH]cc21)N1CC(CN(C(C(CC)(F)F)=O)C)C1 935,CC1(C)CC(C(=O)NNC(=O)C2CC(=O)NC2)C(C)(C)S1 936,C(CCCCC(=O)N(C)CC1CN(C(=O)C=Cc2ccc(F)cc2)C1)N(C)C 937,c1(N2C3CC(CN(C(c4ccc5ncnn5c4)=O)C3)C2)cccc(F)c1[N+](=O)[O-] 938,N1(C(c2ccc(C)c(O)c2)=O)C2CCC(C(=O)NCCOC(C)C)C1CC2 939,c1(C(N(C(C)CCNC(C2CC(O)C2)=O)C)=O)cc(F)c(F)c(C#N)c1 940,CC(C)C(C)CC(=O)NCCCOCCCNC(=O)C(c1cccc(F)c1)(C)C 941,N1(C(CNC(C)=O)=O)CC=CC(NC(=O)CC(c2ccccc2)NC(N)=O)C1 942,c1(NCC2CCCN(C(c3ccc(OC)nn3)=O)C2)cc(F)ccc1C 943,c1(CC)cc(F)ccc1C(=O)NC1CCN(C(C2CC(F)C(=O)N2)=O)C1(C)C 944,C(=O)(C(C)CC(C)(C)C)N1CCC(NC(C(CCCC)O)=O)C1C 945,C1(NC(c2ccc(F)o2)=O)CN(C(C2CC2c2cccs2)=O)CCC12CCC2 946,c1(C(N(CC(CNC(CCNS(CC)(=O)=O)=O)(C)C)C)=O)nnn(C)c1C(F)F 947,c1(C(N2CC(C)N(C(c3cccc(C(F)F)c3)=O)CC2)=O)ncc(C#N)cc1Cl 948,c1(CC(N2CCN(C(C(CSC)C)=O)C(C)C2)=O)ccc(Cl)c2cccnc12 949,N1(C(COCCC)=O)CCC(N(C)C(c2ccc(C(C)(C)C)s2)=O)C(C)C1 950,c1(NC(C(=O)NC)=O)cc(Cl)nc(S(C)(=O)=O)n1.N12CCCN(CC1)C1CC2C1 951,C1(NC(CC(CCC)C)=O)CN(C(c2ccc3scnc3c2)=O)CCC12CCC2 952,Cc1oc(C(F)(F)F)nc1C(=O)NC(C)CCNC(C1CN(C)CCO1)=O 953,N1(C(C(C)Sc2ncccn2)=O)CCN(C(=O)CC2COCC(C)(C)O2)CC1C 954,CC(CC(=O)NC(Cc1ccoc1)C(=O)N(CCC(C)(C)C)C)c1ccco1 955,Cc1cc(N)c(C(N2CC(NC(c3ccc(CC4CC4)s3)=O)CC2C)=O)cc1C 956,C1(NC(C(C)NC(=O)NC)=O)CC12CCN(C(C1CCCN(C)C1)=O)CC2 957,CC1(C)COC(C(N2CCN(C(c3cscn3)=O)CC2CC2CC2)=O)CO1 958,CCS(=O)(=O)CC(=O)NC1C=CC(C(=O)NC(c2cccc(C)c2)CO)C1 959,C1(CN(C(COCCOC)=O)C2CC2)CCCCN1C(=O)C(F)CC1CCC1 960,C1(C(=O)NC(C2CCN(C(CC(COC)C)=O)C2)C)OCCN(C)C1=O 961,C1(NC(C(C)(C)OCC)=O)CC2CC(NC(=O)C(C)CCCOC)C1C2 962,c1(CNC(=NC)NC2CCCC(F)(F)C2)cc(OC(C)C)ccc1Cl 963,Cc1cc(Cl)c(C(N2CCCCC(NC(c3coc(Br)c3)=O)C2)=O)cn1 964,C1(N(C(c2c(C)noc2C)=O)C)CN(C(=O)C2=CC(C)CC2)CC1(C)C 965,N1(C(CN(C(=O)C=C(C)C(C)C)CC)=O)CC2(COCC(=O)N2)C1 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1147,C1(C(=O)NC2(C)CCN(C(c3cc(C(C)(C)C)ncc3)=O)C2)CCOCC1(C)C 1148,C12(CNC(COCC(=O)OC)=O)CC1CN(C(=O)CNC(=O)CC(C)(C)C)C2 1149,Cc1cc(=NC(C)c2ccnn2C)[nH]c(=NCCOCCOCCO)[nH]1 1150,Cc1cnc(F)c(CNC(=O)CC2(NC(=O)CC(C)N(C)C)CCC2)c1 1151,Cc1cc(C(=O)N(C)CC2CN(C(c3cccc(C(F)F)c3)=O)C2)nn1C(F)F 1152,c1(C(=O)NC(C2CCN(C(=O)C(O)CN3CCCC3)C2)C)ccc(F)cc1F 1153,CC1CCC(NC(C2CC3CCC3C2)=O)CN1C(C1CCCO1)=O 1154,c1(C(N2CC(NC(Cc3c(C)cccc3)=O)C(C)C2)=O)ccc(C)n(C)c1=O 1155,C(=O)C(CCCO)c1ccccc1.CC1(C)CC(OC=O)CO1 1156,CCCC(C(=O)N(CC(CC)NC(c1[nH]nnc1C)=O)CC)NC(C)=O 1157,Cc1nn(C)c(C)c1C(=O)NCC1(NCc2ccc(-c3nn[nH]n3)cc2)CC1 1158,C1(C(=O)NCc2cccc(NC(C(C)(C)F)=O)c2)CCn2cncc2C1 1159,O=C1NCCCC12CCCN(c1cc(NCCCCN3CCCCC3)ncn1)C2 1160,c1(CNC2CC(NC(c3nccnc3Cl)=O)C2)ccccc1N1CCOCC1 1161,N1(CC)CCC1C(=O)NC1CC(C(C)NC(=O)Cc2ccco2)C1 1162,c1(C(=O)NCC(CC)(C)OC)c(CNC(c2ccc(C(N)=O)o2)=O)cnn1C 1163,c1(C(N2CCCN(C(c3n(C(C)C)ccn3)=O)CC2)=O)ccc2cnoc2c1 1164,O=C(C1=COCCC1)NCC12CC1CN(C(c1ccccc1C1CC1)=O)C2 1165,C1(NC(C(C)C2CCOC2)=O)CCN(C(=O)COc2ccc(Cl)cc2)C12CCC2 1166,N1(C(CSCCC(C)C)=O)CCCN(C(C2CCOC2=O)=O)C(C)C1 1167,c12cn(nn1)CC(=O)N2c1ccncc1.c1(CN(CCC#N)C)ccccn1 1168,CC1CCOCC1C(N1CC(F)(CNC(=O)Cn2ccc(O)nc2=O)C1)=O 1169,C1(NC(C(C)NC(CC)=O)=O)CC2CC1CN2C(c1cncc(Cl)c1)=O 1170,n1(CC)nc(C(N2CC(C(F)Cn3cc(Cc4ccccc4)nn3)C2)=O)c(C)n1 1171,C(CC(C(C)C)NC(c1nn(C)cc1CC)=O)N(C(c1c(CCC)n[nH]c1)=O)C 1172,c1(C(=O)OCC)ccc2nc(O)n(C3CCCC3)c2c1.c12ccc(o1)CN(C)C2 1173,c1(NC(c2c(C)sc(-c3ccc(F)c(O)c3)n2)=O)cc(Cl)cc(Cl)c1O 1174,C(=O)(C(Cn1ccnn1)NC(c1cc(Cl)no1)=O)N(CCOCC)CC 1175,C1(C)(CNC(CC(C)(C)N(C(=O)CCC23CCC(CC2)C3)C)=O)CCC(=O)N1C 1176,C1(CC(=O)NCC2CN(C(c3c(C)nnn3C)=O)CC2O)CCC(C)(C)CC1 1177,c1(C(=O)NC2C3(CC(NC(=O)Cn4ncnn4)C3)C2)cccc2[nH]cc(Cl)c12 1178,N1(C(C(c2scc(C)n2)C)=O)CCC(NC(=O)CC(C)(F)F)C12CC2 1179,C(N=c1nc2c(F)cccn2[nH]1)c1ccc(OCC)cc1 1180,c1(C(N2C(COC)CN(C(=O)CCC3CC3(Cl)Cl)CC2)=O)cccc2cncn12 1181,c1(N(C)C)nc(C(=O)NC2CC(O)CN(C(=O)Cc3cnc[nH]3)C2)cc(O)n1 1182,CCCC(C)(C)CC(=O)N1CCC(OCCCNC(c2cnc(C)[nH]2)=O)CC1 1183,N1(C(C(C)SC)=O)CCN(C(C2CCS(=O)(=O)CC2)=O)C(CC(C)(C)C)C1 1184,c1(C(=O)NC2CC(NC(C(C3CC3)OC)=O)C2)cncc2nc(C)[nH]c12 1185,c1(OC)cccc2c(C(=O)NC3CN(C(c4cncc5sccc45)=O)C3)n[nH]c12 1186,c1(C(=O)NCC(CC=C)NC(=O)CSSC)ccc(=O)n(C)c1 1187,CC1=C(C(=O)N2CCC(C(C)CNC(=O)C(O)(C3CC3)C3CC3)CC2)SCCO1 1188,c1(C(N2C(CNC(CC)=O)C(C)CC2)=O)cc(Br)c([N+](=O)[O-])[nH]1 1189,C(CNC(c1cn(C)nc1C)=O)(N=c1cc(C)nc(Cl)[nH]1)c1scc(C)n1 1190,Cc1nnccc1C(=O)NCC1CCC(N(C(=O)C(CO)N(C)C)C)CC1 1191,c1(CC)ccccc1C1CC1C(=O)NCC(C)CNC(C1CCC2(CC2)C1)=O 1192,C1(C(=O)NC(C2(O)CCN(C(C(C)OC(C)=O)=O)C2)C)CC(C(C)C)=NO1 1193,C#Cc1ccccc1CC(=O)NCCCN(C(=O)CC(C)OC)C 1194,CN1C(CNC(=O)N(CC(c2cccs2)O)C2CC2)CCS1(=O)=O 1195,S(=O)(=O)(c1cccc(Br)c1F)N1CC2CCN(C(C(C)OC)=O)C2CC1 1196,C12(N(C(C(CC=C)C)=O)CCCOC)CC(c3ccccc3)(C1)C2(F)Cl 1197,Cc1ncc(Br)c(NC2CN(C(=O)C(C)Cc3ccccn3)CCC2(F)F)n1 1198,c1(CC)cc(NC(=O)C(CC)NC(C2CC(C)(CC)C2)=O)cc(O)c1 1199,C(=O)(CCCC(C)(C)NC(C1CCC1(F)F)=O)NC(c1cnn(C)c1)C 1200,N1(c2ccnc(NCC3CC(n4cncn4)C3)n2)CCSC2(CCC2)C1 1201,c1(C(=O)NCC2(C)OCCO2)c[nH]c2cnccc12 1202,CC(CC(F)(F)F)C(=O)N1CCN(C(=O)COc2cccc(Cl)c2)CC1CF 1203,C1(NC(c2cc(CC)ncn2)=O)CN(C(=O)Cc2csc(Cl)c2)C2(CCOC2)C1 1204,C(C(C)(O)CC(=O)NC(CCF)C(=O)N(C)Cc1ncnn1C)OC 1205,C1(C(=O)NCCN(CCC)C(C2CC(O)C(F)C2)=O)CC(C)CC(=O)N1 1206,N1(C(NNC(c2c(C)n(C)nc2)=O)=O)CC2CC3CC1C2O3 1207,C(=O)(CCCCC(=O)NC)NC(C)COC(CC(CC)OC)=O 1208,c1(CN=[N+]=[N-])ccc(C(=O)NC(CNC(c2ccncc2O)=O)C(C)(C)C)cc1 1209,C12(C(=O)OC)CCCC1N(C(C1CN(C)NC1=O)=O)CCC2 1210,CCC(CC)CC(F)C(=O)NC1(C)CCCCC1C(=O)N(CC1CC1)CC1CC1 1211,c1(NC(c2cncc(-c3cc(=N)[nH]cc3)n2)=O)ccc(Br)cc1OC(F)(F)F 1212,N1(C(c2cc(C#C)cc(N)c2)=O)CCC(C2CCCN(C(c3cnsn3)=O)C2)C1 1213,C1(F)(C(C)=O)CC(OC(=O)CCN(C(=O)CC2CCCCC2)C)C1 1214,C1(NC(C(C)SCCCC)=O)CN(C(c2cnc3sccn23)=O)CC12CCC2 1215,c1(NC(c2sccc2NC(C2CCCO2)=O)=O)ccc(OC(F)F)cn1 1216,c1(C(=O)NC2(CC)CCN(C(=O)CCC3CCCOC3)C2)cc2cccnc2[nH]1 1217,C(=O)(CC(C(F)(F)F)OC)NCCCCC1CN(C(C(=O)OCC)=O)C1 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1236,c1(C(=O)NCCC2N(C(C(CCC)C#N)=O)CCC2)[nH]c2ccccc2c1OC 1237,C(=O)(CCC(F)(F)C(=O)NC(C)CN(C)C(C12CC(CO1)C2)=O)OCC 1238,C(=O)(CC(CC)C(C)C)NCC1CN(C(C2(CC=C)CCCCC2)=O)CC(C)C1 1239,c1(C(N2C(CNC(c3cc4occc4s3)=O)CC2)=O)ccc2nncn2c1 1240,c1(OCC)ccc2c(c1)CN(c1cc(C)c(C#N)cc1[N+](=O)[O-])C(C)C2 1241,C1(C(N(C(CCN(C(CCC#C)=O)CC)C)C)=O)(N(C)CO)CCCOC1 1242,N1(CC(=O)NCC2N(C(CC3C(=O)NC(=N)S3)=O)CC=C2)CCC(=O)NC1=O 1243,c1(CC)ccnc(C(=O)NCC(CC(=O)N2CCC(O)C2)C2CCC2)c1 1244,c1(CNC(CC2(C)N(C(c3c(CC)cco3)=O)CC2)=O)cnc(O)nc1O 1245,C12(NC(COCC)=O)CCC(CC1)N(C(=O)CCc1nc(C)cs1)C2 1246,CC(C(=O)NNC(=O)Cc1ccc2c(c1)OCO2)NC(=O)OC(C)(C)C 1247,CN(C(=NCC1CCCO1)NCc1cnc(-n2cccn2)o1)Cc1nnn(C)n1 1248,c1(CCC(c2nnnn2C)NCC2(OC)CC2)ccccc1F 1249,c1(C(N2CC(NC(=O)COC3CCCC3)C(O)CC2)=O)ncc(Br)cc1[N+](=O)[O-] 1250,C1(C(c2n(C)nnn2)Nc2ccc(Cl)cc2)CCC2(CC1)OCCCO2 1251,C1(CNC(C(C(=C)C)(C)C)=O)CC2(CO1)CN(C(c1ncc(C)cc1F)=O)C2 1252,Cc1cc(Br)cc(C)c1C(=O)OCC(N1CCCC(C(C)(C)O)C1)=O 1253,CCC(CC(=O)N1CCN(C(C2CCCN2C(=O)OC)=O)C(CO)C1)C(F)F 1254,N1(C(CC(CC)CN(C)C)=O)CC2CCC1C(CN=c1ncc(OC)c[nH]1)C2 1255,c1(N2C(CCNC(C(C(COC)C)C)=O)CSCC2)ccc([N+](=O)[O-])cc1 1256,c1(N(C)CC2CCN(C)CC2)nc(N2CCOC(C)(C)C2)nc2c1COCC2 1257,Cc1cc(=O)oc(C)c1C(N1CCN(C(C23CCC(CC2)C3)=O)C(CF)C1)=O 1258,C1(C(C)NC(C=CCOCCOC)=O)CCCN(C(c2[nH]cnc2C#N)=O)C1 1259,C(=O)(C1=C(C)N(C)c2ncnn2C1)N1CC(N(C(C=CC=CC)=O)C)C2(C1)CC2 1260,c1(C(=O)NC(C2CCN(C(C3CC=CC3)=O)C2)C)cc(F)c(F)cc1N 1261,c1(N(C2CN(C(C(C=C)c3ccccc3)=O)C2)C)nc(C)ncc1F 1262,c1(SCc2cn(C)nc2)ccc(C(N2CC(O)CC2CNC(=O)CO)=O)cc1 1263,N1(C(c2nn(CC)nc2C)=O)CCC(C)C(CC(=O)NC2(COC)CC2)C1 1264,S(=O)(=O)(c1ccc(NC(=O)CCC2CC2)o1)NNC(=O)C1CC1.C12CC(C1)C2.C1(C)CC1 1265,c1(CCC)cc(C(=O)N(C2CCCC(NC(c3cnc(O)n3C)=O)C2)C)sc1C 1266,c1(CC(C)C)cc(C(N2CC(F)(CNC(=O)CC3CC(O)C3)C2)=O)n[nH]1 1267,Cn1nccc1C=CC(N1CC(NC(=O)C(F)C2CCC2)C1)=O 1268,c1(C(=O)NCC2N(C(C(n3c(C)ccn3)C)=O)CCC2)cnc(Cl)c(F)c1N 1269,Cc1cc(NC(c2cc(NC(c3ccc(CO)cc3)=O)cn2C)=O)cc(F)c1Br 1270,N1(C(c2sc(C(=O)OC)c(C)c2)=O)CCC2CCN(C(=O)C(N)=O)C2C1 1271,C=C(C)CC(C(=O)NCCc1cnc(C)[nH]1)NC(C1CCC(=O)NC1)=O 1272,N1(C(c2cc(C(=O)OC)oc2C)=O)CC2CN(C(=O)CN3CCOCC3)CC2C1 1273,N1(C(c2c(SCC)cccn2)=O)CC2CC(NC(=O)Cn3ccnn3)CC2C1 1274,C1(N(C(c2c(C)snn2)=O)C)CCN(C(=O)Cc2sccc2Cl)CC1C 1275,Cc1ccc(C)c(C(=O)N(CCCC(=O)NCC2CCC(CN(C)C)O2)C)c1 1276,C1(F)(C(=O)NC(c2c(C)ncs2)C)CCN(C(c2ccc(C#N)[nH]2)=O)C1 1277,c1(CNC(NC(c2nc(CC)no2)CC)=NCC2CC2)cn2c(C)cc(C)cc2n1 1278,c1(C(c2n(C(C)C)nnn2)NCc2cncn2C)cccc(C(F)F)c1F 1279,C1(CNC(C2N(CC(C)C)CCC2)=O)CC(F)(F)CN1C(C1CN(C)CCO1)=O 1280,N1(CCO)CCCNC(=O)C12CC2.c12cncc(c1)NCCNC2=O 1281,N1(C(CCC)C)CC(C(N2CCCC2CNC(C2(CO)CCCC2)=O)=O)CC1=O 1282,CC#CCC(C(=O)NCCC(O)C1CCC1)NC(c1ccccc1OC)=O 1283,c1(CCNC(C2CCC(C#N)CC2)=O)cc2ncc(C(F)F)cc2[nH]1 1284,C1(CC)(NC(c2sc(-n3cccc3)nc2C)=O)CCCN(C(=O)C(C)COC)C1 1285,N1(C(c2n(CC(C)C)ncc2)=O)CCN(C)C(CNC(=O)CC2CC2C)C1 1286,c1(C(=O)Nc2cccc(CO)c2F)ncn2cc(-c3cnoc3)sc12 1287,c1(OC)ncc(C)cc1C(=O)NC1CC1CNC(=O)CC1COC(=O)C1 1288,Cc1c(F)ccc(C(=O)NC2CC3CC(NC(=O)C#CC(C)C)CC23)c1C#N 1289,C(=O)(C(CC(C)C)NC(=O)CCCCC#N)OCC#C 1290,N1(C(C2CC(=O)N(CC3CC3)C2)=O)CCOCC1CC(N1CCCCCCC1)=O 1291,c1(OC)cc(C(N2CC(NC(=O)C(F)(F)CN(C)C)C(O)C2)=O)cc(Cl)c1O 1292,c1(C(=O)OCC)cnc(N2CC(NC(=O)CN=S(C)(C)=O)CC2C)nc1C 1293,C(=O)(CCC(F)(F)C(F)F)N(C)CC1(C)C(NC(C(C)n2ccnn2)=O)CCC1 1294,C1(C)(C(N(CCCNC(=O)CC(=O)Nc2nccs2)C)=O)CS(=O)(=O)C1 1295,Cc1nc2ncnn2c(C)c1C(=O)NCCCNC(c1sc(N(C)C)nc1C)=O 1296,C1(NC(CC(=C)C)=O)CN(C(=O)COC(C)(C)C(F)(F)F)C2(CCOC2)C1 1297,N1(Cc2n(C)c(Br)nn2)C2CCC1CN(C(c1cccc(-n3cnnc3)c1)=O)C2 1298,Cc1c(C(=O)NC2CCCC2CNC(c2nnc(S)n2C)=O)ccn1CCO 1299,C(CCSC)(C(=O)NCC(C12CCC(CC1)C2)NC(C1(C)CC1(Cl)Cl)=O)OC 1300,N1(C(C2C(CC3N(C(c4ccccc4)=O)CC(F)C3)C2)=O)CCC(CO)C(O)C1 1301,c1(C(=O)NCC23OCC(CNC(c4cnc(SC)s4)=O)(C2)C3)cnc(O)c(C)c1 1302,C1(C(N2C(C#C)CC2)=O)CN(C(c2occc2COC)=O)CC12CCC2 1303,c1(C(=O)NC23CCC(CNC(=O)C4=CCCC4)(OC2)C3)cccc2ccsc12 1304,N1(C(C2C3(CC(=O)NC2)CCC3)=O)CCN(C(C2CC3CC3C2)=O)C2COCC12 1305,C1(CC)CN(C(=O)CCn2cc(C)cn2)CCC1NC(=O)C(C(F)(F)F)OC 1306,N1(c2nc(=NCCOCCC)s[nH]2)CC2(C)CN(C)CC2(C)C1 1307,N1(CCC(N2C(CNC(c3[nH]cc(C(=O)OC)c3)=O)CC2)=O)CCOCC1C 1308,CC(C)C(C)C(=O)N1CCN(C2CN(C(=O)C(C)N(CC(F)(F)F)C)C2)CC1 1309,C(=O)(CC(F)(F)C(F)(F)F)N1CCC(C)(CNC(C(C(C)C)n2cccc2)=O)C1 1310,N1(C(c2cc(C(C)C)on2)=O)CC(NC(C2CC2(Cl)Cl)=O)C2(CCOCC2)C1 1311,N1(C(Cc2cc(C)sc2C)=O)CC2CC(NC(C3(C#N)CCCC3)=O)C(C2)C1 1312,CCC(CC(=O)NC1CC2(C1)CC2NC(c1ncsc1C)=O)C(C)C 1313,c1(-c2ccc(CNC(c3cnn(C4(CO)CCNC4)c3)=O)s2)ccnc(F)c1 1314,C1(NC(C(CN(C)C)(C)C)=O)CC12CCN(C(c1sccc1I)=O)CC2 1315,N12CCCCC1C(C)(C)CNC(=S)NC(C(C)C)CC2.CS.OC 1316,C1(CNC(c2ccncn2)=O)CN(C(C2CC3(C2)CC(F)(F)C3)=O)CCC1(F)F 1317,N1(C(CN(C)C(N)=O)=O)CCC(C)(N(C(C2CCCN(CC(F)F)C2)=O)CCO)C1 1318,C=CCCC(C(=O)OC)NC(=O)CC1CN(C(=O)Cc2ccoc2)CC1C=CC 1319,C1(CNC(CC2C(CNC(C(CC)OC)=O)C2)=O)CCC2(CC1)CC2 1320,c1(N(C=O)C(C)C2CC2)ccc(OC(F)F)cc1F.C1(n2ccnc2)CCCCC1 1321,C(CCCCCNC(=O)CCn1cccn1)NC(C(C)C1CCCO1)=O 1322,N1(C(c2nccc(C)c2N)=O)CCC2(CCCC(CNC(=O)C=CCO)O2)CC1 1323,C1(NC(c2cccc(C#C)c2)=O)CC2CCC(C1F)N2C(C1(CF)CC1)=O 1324,Cc1ccc2c(c1)CC(NC(=O)N(C)C(c1cccs1)C)CO2 1325,C1(NC(CCC(C)(C)F)=O)CN(C(c2ncccc2O)=O)CC2(CCC2)C1 1326,C(=O)(C1=CCCC1(C)C)NC1CCCN(C(c2csc(C)c2C2CC2)=O)C1 1327,C1(c2nnnn2CCOC)(CNCCCOC)CCCC1CCF 1328,N1(C(C=CSC)=O)CCCC(CNC(=O)C(F)(F)C2CCOCC2)CC1 1329,C1(C2CCCO2)CCOCC1.c1(CC)ccc(C(=O)NCC(C)N(C=O)CC)[nH]1 1330,N1(C(c2ccc(C)s2)=O)CCC2C(C(=O)NC3(C)CCCC3C)C2C1 1331,C1(C(=O)NC2C3CN(C(C(C=C)(C)C)=O)C2C3)Cc2cc(C)ccc2O1 1332,Cc1nc2c(o1)CCN(C(=O)C(CCOCCO)NC(c1ccoc1Cl)=O)C2 1333,c1(C(=O)NCC2C(NC(c3c(C#C)ccc(F)c3)=O)C2)csc2c(F)cccc12 1334,N1(C(CCC2CC(OC)C2)=O)CCN(C(c2ccc(O)cc2Cl)=O)C(C(C)C)C1 1335,c1(CCC)ncoc1C(=O)NC1(CCNC(=O)CCn2ccc(C)n2)CCC1 1336,C1(NC(c2c(C)ncs2)=O)COC2(CCN(C(C3(C#N)CCCOC3)=O)CC2)C1 1337,c1(NC(C2C3CC2N(C(=O)C(Cl)(Cl)Cl)C3)=O)cnc(Br)nc1 1338,c1(SCC)ccccc1C(N1CCC(NC(c2oc(CN(C)C)nc2C)=O)C1)=O 1339,C(CC)(C(=O)N(C)CC1CCN(C(C2(C3CCCO3)CCC2)=O)C1)=CC 1340,C1(C(=O)NC2(C(=O)Nc3c(OC)ncnc3)CCC2)CCCCC(=O)N1 1341,C(=O)(C#CC1CCOCC1)NC(C1CCN(C(c2cc(Cl)cc(C)c2O)=O)C1)C 1342,C1(C(=O)N)CCN(C(N2CCCC2)=O)C1.CC(CCCl)N(C1CC1)C 1343,c1(C(=O)NC2(CC=C)CCN(C(=O)C(O)CSC)CC2)cc2cc(C)ccc2[nH]1 1344,c1(C(=O)NC2(C)CC(NC(c3cn(C)c(=O)cc3)=O)C2)coc2ccc(F)cc12 1345,c1(C(=O)NC(CC)(C)CNC(=O)COCc2nc(CC)no2)cc(Cl)ccc1N 1346,C(=O)(C(CS(C)(=O)=O)NC(=O)OC(C)(C)C)NCC(C(C)C)(C)C 1347,c1(C(N2CCN(C(=O)Cc3ccc(O)nc3)CC2)=O)ccc(O)c(Cl)n1 1348,C1(C(=O)NCC(C)CN(C)C(C2CC3CC3C2)=O)CCc2ccnn2C1 1349,C1(OC)CC(NC(c2ccsc2)=O)CN(C(c2cncc(OC(C)C)c2)=O)C1 1350,C1(C(N2CCC(OC(C)C)CC2)=O)CN(C(C2CC(=O)C2)=O)CCC1O 1351,O=C(CCC(=O)N1CCC(NC(C23CCCCC2C3)=O)CC1)C1CC1 1352,CCCC(C(=O)NCC1CC2CN(C(c3ccc(Cl)cc3OC)=O)CC12)C(C)C 1353,CC#CCCCC(=O)NCc1ccc(C(=O)NC(C)CN(C)C)cc1 1354,C1(NC(c2ccc(C)c(O)c2)c2nnnn2C2CC2)CC(F)(F)CCC1(C)C 1355,c1(C(c2cnc[nH]2)NC(S(C)(=O)=O)=O)ccccc1.CC1C(=O)NC(CO)CN1 1356,C1(O)(CN(C(=O)C(=O)NC2CC2)C)CCCN(C(=O)CC(F)(F)Cl)C1 1357,c1(C(N2C(CNC(COCCCC(C)C)=O)C=CC2)=O)cc2nnn(C)c2s1 1358,c1(NC(C2CCN(Cc3ccc(C)s3)C2)=O)cncc(F)c1I 1359,C1(NC(C2C(CNC(CNS(N)(=O)=O)=O)OCC2)=O)C2C=CC(C2)C1CO 1360,C1(N(C(C(C=C=C)C)=O)C)CN(C(=O)C(F)(F)Cc2ccccc2)CC12CC2 1361,C1(NC(c2cc(CSCC)on2)=O)CCC(O)CN(C(c2ccn(C)c2C)=O)C1 1362,c1(CNC(C(=O)Nc2c(C(=O)OC)scc2)=O)cccc(NC(C)=O)c1 1363,C1(C(N(C2(CO)CC2)C)=O)CN(C(=O)CC2CCSC2)CCC1(C)C 1364,N1(C(C(CC)(F)F)=O)CC2C3CCC(C2C1)N(C(=O)C(c1cscn1)C1CC1)C3 1365,CCC(C(=O)NC(C)(C)CN(C(=O)CCc1ncccc1C)C)C(C)O 1366,C1(CC)CCC(C(=O)NC(C2CCCN(C(C3(SC)CC3)=O)C2)C)CC1 1367,N1(CC(N2CC(CN(C)C(C3COCCO3)=O)C2)=O)CCCCC1=O 1368,c1(C(N2C(CNC(CCC#C)=O)CC(O)C2)=O)cc(OC)cc(F)c1 1369,CO[Si](C)(CCCOC(C1(CC(C)C)CC1)=O)OC 1370,C12(NC(C(CC)OC)=O)CCC(CNC(c3cn(C)c(C)n3)=O)(CC1)OC2 1371,CCCCC(C(=O)N1CCC(C)C1CNC(=O)C(C(C)C)SC)C(C)C 1372,N1(C(CCCOC)=O)CCCC2(NC(=O)CN(c3ccccc3)C)CC12 1373,N1(C(CCCC=C)=O)CCN(C(C23CC=CC(C2)OC3)=O)C(CC)C1 1374,c1(C(N2CC(NC(CSC(C)C)=O)C(C)(C)C2)=O)c(F)cccc1[N+](=O)[O-] 1375,c1(C(=O)NC2CC3(C2)CC(NC(C2CC2(F)Cl)=O)C3)cc2cccnn2n1 1376,CCC#CCCNC(C1CC1NC(=O)COC1(C)CCC1)=O 1377,c1(C(=O)NCC(CO)NC(CCNC(N)=O)=O)coc2c1C(=O)NCC2 1378,c1(C(=O)NCc2nc(N(C(C(C)C)=O)C(=O)CN(C)C)sc2)ccccc1[N+](=O)[O-] 1379,CCC(CC(=O)NC(CC(F)F)C(=O)N1CCCC(C(C)C)CC1)CC(C)C 1380,CN1CC=C(CC(=O)NC2CCN(C(C3CC3C(=O)NCCO)=O)C23CCC3)CC1 1381,Cc1cc(Cl)cc(C(N2CC(NC(C3(F)CCC3)=O)CC(C)C2)=O)c1N 1382,C1(C(=O)NC(C)(CNC(c2cc(C(F)(F)F)n[nH]2)=O)CO)COC2(CCC2)CO1 1383,c1(C(N(CC(CO)(CO)NC(CC(=O)OCC)=O)C)=O)c[nH]c2c(F)cccc12 1384,C(C(O)CCNC(C1CCC12CC2)=O)NC(CSCCC(C)C)=O 1385,C(=O)(C(CNC(c1ccc(C)c(F)c1)=O)C(C)(C)C)NCC1N(CC)CC1 1386,c1(CC(=O)NCCCN(C)C(C2(CF)CCC2)=O)cnoc1 1387,C(=O)(C1=CCCCO1)NC1(C(=O)NCCC2CCCC(C)C2)CCCCC1 1388,N1(C(C23CC(OC)C2C3)=O)CCC2(CCC(N(C(=O)C=CC(C)C)C3CC3)CC2)C1 1389,N1(CCNC(=O)NC2(C(F)F)CCCC2)CCCC(c2ccccc2)C1 1390,C(=O)(N=c1ccn(CCN(C)C)[nH]1)N(CC(c1ccccn1)(C)C)C 1391,c1(OC)ccccc1C(O)Cn1cc(C(C)N(C)C(c2cc(O)cs2)=O)nn1 1392,C(=O)(CS(=O)(=O)C(C)C)N1CC(CNC(CC2(C(=O)OC)CC2)=O)N(C)CC1 1393,Cc1ccc(N)cc1C(N1CC2(C1)CN(C(=O)C(c1ccccc1Cl)O)C2)=O 1394,C1(C(N2C(CCNC(C(C)C3CCCC3)=O)CCCC2)=O)CCC([N+](=O)[O-])CC1 1395,C1(NC(CCSC)=O)CCN(C(c2ccc(C(O)C(F)(F)F)cc2)=O)C1C1CC1 1396,c1(C(=O)NC(CC)CN(C(=O)C(C)Oc2ccccc2F)CC)cccc(F)c1N 1397,N1(C(C2CCC(C)CC2)=O)CCOC2(CCN(C(=O)C=C3CCC3)C2)C1 1398,N1(C(c2n[nH]cc2Br)=O)CCC(C2CC2)C1CNC(C1(CF)CCC1)=O 1399,c1(C(N(C2CCN(C(CCC(=C)C)=O)CC2)C)=O)c(Cl)cccc1[N+](=O)[O-] 1400,C(=O)(C(C)(CO)OC)NCC(c1cccnc1)Nc1cn(CC(=O)OC)nn1 1401,C12(C(=O)NCC(CNC(CC3(C)CC3)=O)O)COCC1CN(S(C)(=O)=O)C2 1402,C1(C(=O)NC(C=CC(=O)N(CCSC)CC)(C)C)CCCN1CC 1403,C(CC(C)(C)C)(C(=O)N1CCCC1)NC(C(CCC#C)O)=O 1404,c1(SC)ccc(C(N2CC3CC3(CNC(=O)CC(C)C)C2)=O)cc1Br 1405,c1(C(=O)NC2(CC(=O)NC3CC(CC)(CC)C3)CC2)cccc(F)c1O 1406,N1(C(CC2ON=C(C)C2)=O)CCCC(CN(C(=O)C(c2ccc(Cl)cc2)O)C)C1 1407,c1(C(=O)NC2C=CC(CNC(c3n(CC)ncc3)=O)C2)c(F)cccc1F 1408,C(c1cc(F)c(F)c(F)c1)=CC(N1CCC(N(C(C(C)OC)=O)C)C1)=O 1409,N1(C(c2c(C)csn2)=O)CC(C(=O)N(C2CCCC2C#N)C)CC(C)C1 1410,C1(NC(c2c(C)cn(C)n2)=O)CC2(C1)CC(NC(c1csc(C)c1N)=O)C2 1411,N1(C(CC2CN(C)C2)=O)CCC(NC(=O)CC(O)C2CC2)C2(CCC2)C1 1412,c1(CNC(C2(C)CCCN(C(C=C(C)C(=O)O)=O)C2)=O)ccc(C#N)cc1F 1413,C(=O)(C1CCCc2nncn21)N1CCC2(C(NC(C3C(=O)NCCCC3)=O)C2)CC1 1414,c1(C(=O)NCC(CNC(c2c(CC)nns2)=O)(C)O)ccc2ncncc2c1 1415,CON(CCC(=O)NCC1CCCC(O)C1)C(=O)Cc1cc(C)on1 1416,n1(CC)nc2c(c1NC(=O)Nc1cc(Cl)ccc1Oc1ccccc1)CCCC2 1417,Cn1c(=O)[nH]c(NCC2CCN(c3ccccc3Cl)C2)c(C#N)c1=O 1418,C1(CC#C)(C(=O)O)CCN(C(C2CCC(N)CC2)=O)CC1 1419,c1(C(N2CC(C)OC(C(=O)NCC3CC34CC4)C2)=O)ccn2cncc2c1 1420,Cc1nc(C(=O)NC2CCC2CNC(c2cccnc2)=O)cn1C(F)F 1421,c1(OC)ccc(Br)cc1NC1COCCC1NC(=O)NC1CCC(CF)CC1 1422,C1(C(N(C(CCNC(CNC(=O)NC)=O)C)C)=O)CC(C)CO1 1423,CC(C)(C)CC(=O)NC1CC2C(NC(C3(NC(N)=O)CC3)=O)C2C1 1424,Cc1ccc(CC2(NC(=O)C(C)CC(=O)O)CN(C(C3C(C)CC3C)=O)C2)cc1 1425,c1(C(N(CC(N2CC(OC(N)=O)C2)=O)C2CCC2)=O)coc(CO)c1 1426,c1(C(N(C(C)CNC(c2ccc(C)nc2C)=O)CC)=O)nsc2c(Cl)cccc12 1427,n1(CCCC)nnnc1C(CCC1CC=CCC1)NCC(F)=C(C)C 1428,CC1CCN(C(c2cc(Cc3ccc(F)cc3)[nH]n2)=O)CC1NC(=O)C(C)(Cl)Cl 1429,C(C)(CCC(=O)NC1(CC(=O)NC2CCCC2(C)C)CCC1)OC 1430,C1(C(=O)Nc2cn(CC#C)nc2)CC2C=CC1N(C(=O)Cc1cnn(CC)c1)C2 1431,c1(CC)cccc(C(=O)NCC2(O)CCN(C(=O)Cc3cnn(C(F)F)c3)C2)c1 1432,C(N=c1cc(C)nc(Cl)[nH]1)C1CN(C(C2(COC)CCCCO2)=O)C(C)C1 1433,C=CC(C)(O)C(=O)NCC(C)(C(C)C)NC(c1cc(Cl)sc1Cl)=O 1434,C1(C(N2CC(CC(CNC(Cc3n(C)ccc3)=O)(C)C)C2)=O)CCCCC(C)(C)C1 1435,CC1CCC(CC(N2CC(CC(F)C(=O)N3CCC3(C)C)C2)=O)C1 1436,N1(C(c2c(C)nsc2)=O)CC(N(C)C(c2cncs2)=O)C(F)C1 1437,CCC(CCOCC)NCc1cc(C(N)=O)co1 1438,C=CCC(CC(C)C)C(=O)NCCCC1(NC(=O)CCCCC(C)C)CC1 1439,CCC(c1cccc(Cl)c1)=CC(=O)NCC1CCC1NC(=O)CC1CC1 1440,CC1CCCC1(C)C(=O)NCC1CCC(C(=O)N(C)CCO)C1 1441,CC1CCCC(C(N2CCN(CCCCNC(=O)C(=O)N(C)C)CC2)=O)CC1 1442,c1(CNC(CC2CCC(C)O2)=O)ccc(Cl)cn1.C1(=O)CCCC2(CCC2)N1 1443,c1(N2CCOCC(c3nnc(CC)o3)C2)ncc(Br)c2ccc(C)cc12 1444,N1(C(C#CC2(C)COC2)=O)CCCC2CN(C(c3ccn4ccsc34)=O)CCC12 1445,C(=O)(NNc1c(Cl)cccc1Br)NC1CC(=O)C2C1CNC2 1446,c1(C(=O)OC)c(Cl)nc[nH]c1=NCCN(C)C(c1ccc(OC)cc1)=O 1447,c1(C(N2C(C(N3C(COC)C(O)CC3)=O)CC2)=O)ccc(C)c(C#N)c1 1448,C1(C#CC(=O)N2CCC(O)C2CNC(C2(CC(=O)OC)CC2)=O)(CC)COC1 1449,N1(C(CCC(C)(C)F)=O)CCC2(CCCN(C(=O)CCCCCC3CC3)C2)C1 1450,n1(CC)cc(NC(C2CC(C)CN2Cc2cnc(N(C)C)cn2)=O)c(C)n1 1451,N1(C(N(C(C)(CO)C(F)F)C)=O)CCC2(C1)CN(Cc1ccccc1)CCO2 1452,C#CCC(C)(C(=O)NCC1NC(=O)CC1(C)C)NC(=O)CCc1nc(=N)[nH][nH]1 1453,c1(C(N2C(CNC(c3cnn(C)n3)=O)CC(OC)C2)=O)cc(Br)cnc1N 1454,c1(C(N2CC(CNC(c3cc(C)n(C)n3)=O)C(C)C2)=O)ccn2cnnc2c1 1455,c1(OCC)ccc(C(=O)NCC2CC(C3CC3)CCN2C(C23CC2C3)=O)c(F)c1 1456,c1(C(=O)NCC2(F)CCC(NC(c3c(C)noc3)=O)C2)cnc2ccccn12 1457,n1(CC(N2CCCC(N(C(C(CCC)C)=O)C)C2)=O)ncc(C#N)c1Br 1458,C1(C(=O)NC2CCC(C(N3CC(N(C)C)C(F)C3)=O)CC2)CCCC(C#N)C1 1459,c1(C(N(C)CCNC(=O)CCc2cn[nH]c2)=O)ccc(CSC(F)F)o1 1460,C1(C(=O)Nc2cccc(CNC(C(CC)O)=O)c2)Cc2cc(C)c(C)cc2O1 1461,CCCCCC(O)CC(=O)NC(CNC(=O)COc1cccnc1)CCC 1462,C(=O)CC1=NNC(=O)C1.C(CC(C)CCNC(=O)CSCCC(F)(F)F)OC 1463,N1(C(c2c(C(C)C)c[nH]n2)=O)CCC2CN(C(c3csc(C(N)=O)n3)=O)CC2C1 1464,C(=O)(C1=C(C#N)CCC1)N1CCC(OC)(CNC(C2CN(C)C2)=O)CC1 1465,C(C(=O)NCC1C2CN(C(=O)CC(C)CN(C)C)CC12)(C(C)C)n1cc(C)nc1 1466,c1(CC)cc(CC(=O)NC2C=CC(CNC(c3scnc3C(C)(C)C)=O)C2)on1 1467,C12(CNC(CC3CCN(C(C)=O)C3)=O)CC(NC(C3CCCSC3)=O)(CCO1)C2 1468,C1(CC=C)(C(=O)NCCc2cnc[nH]2)CCN(C(c2ccn(C)n2)=O)C1 1469,C1(C(N(CCCC)CCO)=O)CCC(NC(=O)Cn2cc(CO)nn2)CC1 1470,C(=O)(C1=CS(=O)CCC1)N1CCC(C(C)NC(C(C)c2cccs2)=O)CC1 1471,Cc1ccnc2c(C(=O)NCC3CC(NC(c4[nH]cnc4C)=O)C3(C)C)cnn12 1472,O=C(C=CC(C1CCC1)NC(=O)CN1CCCCC1)NOCCOC1CC1 1473,n1(CC)c(C)cc2c1CCCC2NC(=O)C(=O)NCC1OC(=O)NC1(C)C 1474,c1(OC)cc2[nH]ncc2cc1C(N1CC(NC(=O)C=CC(C)C)CC(F)(F)C1)=O 1475,N1(C(C(C(Cn2cc(-c3nc(C4CC4)cs3)nn2)CO)C)=O)CCCCCC1C 1476,N1(C(C2C(COC)CC2)=O)CCc2ccccc2C1CO 1477,c1(C(=O)NC2C(CNC(CN(C(C)C)C)=O)C2)coc(Cl)n1 1478,C1(CNC(=O)C(O)C(F)F)COCCN(C(c2c[nH]nc2-c2ccns2)=O)C1 1479,C1(NC(N(c2ccc(-n3cccn3)cc2)C)=O)CC2(C1)CC(N)C2 1480,C1(NC(Cc2ccc(C)cc2)=O)CCN(C(c2ccc(C)n2C)=O)CC1C(N)=O 1481,c1(C(=O)NC2(C(=O)NCC)CC2)sc2nccnc2c1CSC 1482,O(NC(=O)C(c1cn(C)nn1)NC(c1cc(C)[nH]n1)=O)C(C=C)C 1483,CC1CCN(C(=O)C(O)CC2CCCC2)CC1CNC(c1ccc(C2CC2)nc1)=O 1484,c1(OC)cc(CN2CCC(NC(c3ccc(O)c(O)c3)=O)C(F)C2)ccc1C 1485,CN1C(=O)CN(CC(=O)NC2CN(C(c3cnccn3)=O)CCC2C)C1=O 1486,C1(C2CCN(C(=O)C(C)P(C)(C)=O)CC2)(NC(CCCC(C)C)=O)CC1 1487,N1(C(c2c(CC)non2)=O)CC2(CCCC2NC(=O)CS(=O)C(F)(F)F)C1 1488,c1(C(=O)NC(C(C)NC(c2cncc(NCC)c2)=O)(C)C)nccc(Cl)c1O 1489,c1(C(=O)NCC2N(C(CC3CC(C)C3)=O)CCOC2)cnn2c1S(=O)(=O)NCC2 1490,c1(NC(C2(C)CCN(C(=O)Cn3cc([N+](=O)[O-])cn3)C2)=O)ccc2oncc2c1 1491,Cc1csc(C(=O)NC2(C(=O)N(C)CC3(O)CCOC3)CC(O)C2)c1 1492,N1(C(C2CCN(C(=O)OCC)CC2)=O)CCCC(NC(C2CC(C)(O)C2)=O)C1C 1493,C1(CNC(C2CCC(=C)CC2)=O)CC2CN(C(c3coc(C)c3)=O)CC12 1494,c1(OCCC)cccc(C(N2CC(O)CC2CNC(C2(C)CCNC2=O)=O)=O)c1 1495,C(C(C)C(F)C(=O)NCC1CCC(=O)NC1C)NC(CC=CC=C)=O 1496,C12CCN(C13CCC3)C2=O.O=C(CCCOc1ccccc1)NC1CC1 1497,Cc1cc(C)n(CC(N2CC(O)(C(F)C(=O)NC3(CO)CC(F)(F)C3)C2)=O)n1 1498,C1(CNC(C=CC(=O)OC)=O)(NC(C2CC2C(=O)OC)=O)CCOC1 1499,C1(CC)CCCC1(C)C(=O)NCC1CCCC1NC(c1cc(C)[nH]n1)=O 1500,N1(c2nnc(C(=O)OCC)s2)CC2CC(NC(C3COC(C)C3)=O)CC1C2 1501,N1(C(C)C)CCC(CNC(=O)C(O)CNC(=O)C(F)=CC2CC2)C1 1502,C1(NC(Cc2cn(C)nc2)=O)CCC2(CC1)CN(C(C1COC(=O)C1)=O)C2 1503,CC(C(=O)NC1CCCN(C(=O)C(=O)NCC(F)F)CC1)C(F)(F)C(F)F 1504,Cc1ccc(C=CC(=O)N(C2CCN(C(=O)C=C3CCC(C)C3)CC2)C)cn1 1505,c1(C(CCOC)C(c2n(CC(=C)C)nnn2)C2(N)CC2)ccc(OC)cc1 1506,C1(NC(C(C2CCCCC2)OC)=O)C2CCCN(C(=O)COC(F)F)C2C1(C)C 1507,c1(C(N(C2CCCN(C(C3CCCCN3C)=O)C2)CC)=O)[nH]c(O)nc1C 1508,c1(SC(c2ccccc2)C(=O)NC2C(NC(C)=O)CC2)ccc(O)c(Br)c1 1509,N1(C(C(C)(C)c2ccccn2)=O)CCC2CC(NC(C3CSC3)=O)CCC2C1 1510,N1(C(CC(=O)NCC#C)=O)CC2CC(NC(=O)CC3COCC3(C)C)C(C2)C1 1511,c1(C(N2CCN(C(C3(CF)CC3(F)F)=O)CC2)=O)cc(F)cc(Cl)c1O 1512,C(=O)(C(C)CC(=C)C)NCCN(C(CC=C=C)=O)C(C)C 1513,C1(NC(c2nc(COC)[nH]n2)=O)CCN(C(c2cc(SC)oc2C)=O)CC1F 1514,c1(C(=O)NC(CC)CNC(=O)C(=O)NC(C)C)sc(C(C)C)nc1C 1515,CCCC(C)CCN=c1[nH]c(N(CCCOC)C)nc2c(F)cc(F)cc12 1516,CC(C(=O)NC1CCCCC1CNC(=O)CSCCC(F)(F)F)C(C)(F)F 1517,c1(C(N2CCN(C(c3cc(C)ncn3)=O)CC2)C(=O)NCC)ccc2nsnc2c1 1518,Cc1[nH]c(C)c(C(=O)NCc2ccoc2C(=O)N(C)CC2CCN(C)CC2)c1C 1519,S(=O)(=O)(c1cccc(=NC2CCCc3sccc32)[nH]1)NC(c1cc(Br)n(C)n1)C 1520,C1(C(=O)NCC(C(N)=O)(F)F)CC(N=[N+]=[N-])CN1C(=O)CN1C(=O)CNC1=O 1521,C(=O)(C(C)(O)CCC)NCC(C)(CO)NC(c1c(CC)nn(C2CC2)c1)=O 1522,N1(C(CC2CC(C)(C)C2)=O)CCN(C(C2CCO2)=O)CC1c1cccc(Cl)c1 1523,CN1C(=O)NCC1C(=O)NCCN(C1CCCC1)C(c1ccc(F)cc1)=O 1524,C1(C)(C(=O)NC2C=CC(CC(=O)NCc3c(C)ocn3)C2)CCC(=O)C1 1525,C(C)(CCCN=c1c(Br)c[nH]cc1[N+](=O)[O-])NC(C=CCC)=O 1526,C(=O)(C#CC1CCOCC1)NC1C(CNC(CC2(CC(=O)OC)CC2)=O)CCC1 1527,N1(C(C2C(=C)C2)=O)CCc2ccccc2C1CNC(c1cnn(C2CC2)c1Cl)=O 1528,C1(CN(C)C(C2CC23CC(NC(C24CCC(C2)C4)=O)C3)=O)CCCCC1(C)C 1529,C#CCC(C)(CC)C(=O)N1CCC1CNC(C1(O)CCSCC1)=O 1530,Cc1ccc2c(N(CCCF)C)nc(N(C)CC3CCCS3(=O)=O)nc2c1 1531,C(C)(C(CC(=O)NCCc1ccc(F)nc1)NC(=O)CCN1CCCCC1)OC 1532,C1(NC(CCc2cncc(C)c2)=O)CCN(C(=O)C(C)C2CCOC2)C(C)C1 1533,CC(C(C(=O)NCCSC)N1CCCCC1CNC(=O)OC(C)(C)C)C(C)(C)C 1534,C1(CNC(c2cn(CC(C)C)nc2C(F)F)=O)CCCCN(C(=O)C=CCF)C1 1535,c1(CCC(=O)NC(CCNC(C2C(C(=O)OC)CCC2)=O)C)ccccc1OC 1536,CCCCCC(=O)NCC(C)N(C(=O)Cc1cccnc1)C 1537,Cc1cc(F)ccc1CC(=O)NC1(CN(C(=O)C(C)(C)c2ccccn2)C)CC1 1538,c1(C(=O)Nc2cccc(NC(C3(NC(C)C)CC3)=O)c2)ncnc2cc[nH]c12 1539,N1(C(COC(C)(C)C)=O)CCCC(O)(CNC(=O)C(O)Cc2ccccc2)C1 1540,C1(O)(CNC(C2CCCS2)=O)CCCN(C(=O)CN2CCCC2)CC1 1541,C(=O)(C(CO)c1ccccc1)NC(C1CCN(C(=O)CCc2cc[nH]n2)C1)(C)C 1542,n1(CC)ccc(CNC(=O)C(C)C2CCOC2)n1.C(=O)(COCCSC)N(C)CC 1543,c1(C(=O)NC(CNC(CC2(OC)CCCC2)=O)C2CC2)ccc(F)cc1C1CC1 1544,N1(C(CC(C=C)CC)=O)CCC(C(=O)NCc2ccc(C)nc2)C(C)(C)C1 1545,C1(NC(C2C=CCN(C(c3ccccc3)=O)C2)=O)CC2(CCC2)C1O 1546,C1(C(N2CCN(C(CC(n3ccc(C)n3)C)=O)CC2C)=O)CC2CCCCN2C1 1547,C1(CC(=O)NC(CNC(C(C(C)C)OC)=O)(C)C)CCC(=O)NC1=O 1548,Cc1nc2ccc(C(=O)OC3CCC(=O)NC3=O)cc2s1 1549,C1(N(C)C(C23CCC(C2)C3)=O)CCCC(NC(C2(C)CC2)=O)C1 1550,C1(CNC(c2c(C)noc2)=O)CCN(C(=O)C2=NOC(C3(O)COC3)C2)C1(C)C 1551,C#Cc1ccc(C(=O)NCC(O)CCNC(c2c[nH]cc2C)=O)cc1 1552,C(C(N=c1cc[nH]c(-c2ccc(N(C)C)cn2)n1)C1CC1)NC(CCC=C)=O 1553,C1(NC(C(CCF)NC(COCCC)=O)=O)C2CCC(C2)C1C 1554,C(=O)(C#CC1CCCOC1)NCCCN(c1nccc(OC)n1)C(C)C 1555,N1(C(c2ccn(-c3ccccc3)n2)C(=O)NCCC)CC(=O)N(C)CCC1 1556,c1(NC(=O)NCc2ccc(OC)c(C#N)c2)cccc2c(OC)ccnc12 1557,CC(CCC(=O)N1CCN(C(=O)CNC(N)=O)CC1)NC(=O)C(C)n1cccn1 1558,C1(N(C(=O)CCSc2ccccc2)C)CCCN(C(C2CCC2(C)C)=O)C1 1559,c1(CC)nn(C)c(C(C(=O)NC(C)C)N(C)CC2OCCC2(C)C)c1Br 1560,N1(C(CS(=O)(=O)NC)=O)CC(NC(=O)C=CC2CCCCCC2)CC(C)(C)C1 1561,c1(N(C2CCNC2)C(c2cc(OC)cc(C)c2)=O)ncnc2ncn(C)c12 1562,c1(OC)nc(C)sc1C(=O)NCC1CCC(NC(c2ccc(C(F)F)nc2)=O)C1 1563,C1(CNC(CN2CC(C)C2)=O)CC2CN(C(=O)CCCC#N)CC12 1564,C(=O)(CCCS(C)(=O)=O)N1CC(NC(C(C=C)(C)C)=O)C2C(C1)C2 1565,C1(C(=O)OCC)CC2CCC1N(C(=O)C(=O)NCc1cccc3c[nH]nc13)C2 1566,C1(CCNC(c2ncc(C)cn2)=O)CCCN(C(C2CC2C)=O)CC1 1567,N(C(=NCCC(C)(C)C(F)(F)F)N1CCN2C(CCS2(=O)=O)C1)C(C)C 1568,S(=O)(=O)(c1cc(C(N)=O)oc1C)N1CC(C(=O)O)(COC)C1 1569,C1(CCOCC2CC(CSC)C2)(OC)CCN(C(=O)OC(C)(C)C)C1 1570,CCCC(CCCNC(c1coc(C(C)C)n1)=O)NC(c1cc(Br)n[nH]1)=O 1571,c1(C(=O)NC(C2CCN(C(=O)C(c3cnn(C)c3)O)C2)C)ncc(F)cn1 1572,CC1(C)CC(NC(C2CC2F)=O)CCN(C(=O)CCc2cc(Cl)cs2)C1 1573,C12(CCOCC1)C(=O)N2.c1(C(=O)NC2CCN(CC)C2)cn(CCOC)nc1C 1574,N1(C(CC(C)C)=O)CCCC(C2CCN(C(C3(C#N)CC4CCC3CC4)=O)C2)C1 1575,CN=c1[nH]c(C(N2CCN(CC(C)(C)NC(C3CC34CC(O)C4)=O)CC2)=O)cs1 1576,C1(CNC(c2n(C(CC)C)ncc2)=O)CN(C(C2CC2(F)F)=O)CCC1(C)C 1577,c1(SC)nccc(=NC2CCC3(C2)CN(C(c2ccc(C(C)C)nc2)=O)C3)[nH]1 1578,N1(C(C=CC=CCC)=O)CC(CNC(c2c(C)csc2Cl)=O)N2CCC1C2 1579,c1(C(N(CCCCNC(=O)CC2CC=CCC2)C)=O)ccnc2cc[nH]c12 1580,Cn1c(O)ncc(-c2nccn2-c2ccc(C3CC3(F)F)cc2)c1=O 1581,c1(N2CCC(NC(c3ccc(C)cc3)=O)C(C)C2)cc2nncn2c(C)n1 1582,C1(C(N(C(CC(F)F)C(=O)NCC(C)(C)C#N)C)=O)CN2CCC1CC2 1583,C(=O)(C(C)CCCC(C)=O)N1CCC(CCOC)(C(N2CC(C)C(F)(F)C2)=O)CC1 1584,c1(N2CCCC(C)(OC)CC2)nc(N2CCn3ncc(Cl)c3C2)c2c(n1)CCC2 1585,N1(S(CC)(=O)=O)CC2CCN(S(=O)(=O)Cc3nc4ccccc4[nH]3)C2C1 1586,CCC(CC(=O)N1CC(CC(F)C(=O)N2CC(N3CCC3)C2)C1)C(C)C 1587,C(CC(C(=O)NCC12CC(F)(C1)C2)NC(c1cnc(Cl)n1C)=O)N(C)C 1588,C1(CC)CCN(C(C2COCCO2)=O)C1CNC(c1cccnn1)=O 1589,Cc1ccccc1CNC(C1(CNC(=O)CO)CCCC1)=O.N1(C2CC2)CCC1C 1590,N1(C(C23OC(C)C(C2)C3)=O)CCCN(C(C2CCCN2C)=O)C(CO)C1 1591,C=CCCCC(C)(C)C(=O)NC(C)CNC(=O)Cc1ccc(O)c(Cl)c1 1592,Cn1nc(C(N2CCOC(CNC(C3C4CC(=O)CC34)=O)C2)=O)cc1F 1593,c1(OC)cc(CC(N2CCN(C(c3cc(C)on3)=O)C3CCC23)=O)c(F)cc1O 1594,c1(CC(N2CC(C)N(C(c3cccn(C)c3=O)=O)CC2)=O)cc(F)c(F)cc1F 1595,S(=O)(=O)(c1cccc(OCC(c2ccccc2)C)c1)N.CCCC1CCCN1 1596,Cc1cccc2[nH]cc(C(=O)N(CCCCNC(C34CCC(CC3)OC4)=O)C)c12 1597,Cc1ccc2oc(N3CC(CO)(NC(c4cnc(F)c(Cl)c4)=O)C3)nc2c1 1598,N1(S(CCC)(=O)=O)CCCCC1C(=O)NCCCN(C(=O)CCC(C)O)C 1599,C1(C)(NC(C(CC)C)=O)CCCN(C(c2ccnn2CCOC)=O)C1 1600,c1(C(=O)NC2CCN(C(C3(C=C)CCC3)=O)C2)cc(C)nc2ccc(C)cc12 1601,Cc1cccc(CNCc2ccc(-c3ccc(C4(C#N)CC4)cc3)cn2)n1 1602,N1(C(C(C(C)C)O)=O)C(C(=O)NC2(C)CCC(C)(C)C2)C2CC(O)C1C2 1603,N1(C(C2(CC=C)CC2)=O)CC(CNC(=O)C(COC)N(C)C)CC(C)(C)C1 1604,N1(C(CCC(=O)NCC)=O)CC2(CNC(=O)C(C)(C)C3(C)CC3(F)F)CC1CO2 1605,CC1(NC(c2cccc(Cl)c2O)=O)CCC(NC(=O)C(F)(F)c2cscn2)CC1 1606,N(C1CCc2c(C(F)(F)F)cccc21)C(c1ccc(Br)c(Cl)c1)C(F)(F)F 1607,c1(C(=O)NCC2CCCN(C(C3CCCC3)=O)C2)cc2cc(Cl)ccc2o1 1608,N1(C(C2N(C(C3CCC(C)(C)OC3)=O)CCOCC2)=O)CCC2(CC1)CSC2 1609,CCC(CC)(CO)C(=O)N1CCC1CNC(c1ccccc1-n1ccc(C)n1)=O 1610,C1(O)(CNc2ncc(C(=O)OCC)nc2)CCCN(C(=O)Cn2cccn2)C1 1611,c1(C(=O)NC2(F)CN(C(CC(c3ccccn3)C)=O)C2)ccc(Cl)nc1 1612,C1(NC(C2C(NC(C3CCC(C#N)CC3)=O)CCCC2)=O)CCC2(CCCC2)C1 1613,O=C(C1c2c[nH]nc2CN1C(c1nocc1Cl)=O)NCCC(O)C(F)(F)F 1614,c1(C(=O)NCCCC(C)NC(CC(CC)(C)C)=O)cc2ncccc2o1 1615,CCC(C)CCCCC(=O)N(CC)CC1CCCN1c1ncnc2[nH]cnc12 1616,C(=O)(CCS(N)(=O)=O)NC1CN(C(C(CC=C)N(C)C)=O)CC1C 1617,C1(CNC(C(n2cc(-c3nccs3)nn2)C)=O)CC(C2CC2)=NO1 1618,C12(C(=O)NCc3c(CCNC(C(CC)C)=O)ocn3)CC3CC1C2C3 1619,Nc1ccc(C(N2CC(NC(C3CC3C3CCC3)=O)C(F)C2)=O)cc1[N+](=O)[O-] 1620,c1(C(=O)NCCC2N(C(c3c(C)ccs3)=O)CCOC2)ccc(=O)n(CCF)n1 1621,c1(C(=O)NC(COC)CC(=O)NCC(O)CN(C)C)cc(C)cc(O)n1 1622,c1(CC(COC2CC(=O)C2)O)cn(C2CCc3c(F)cc(Cl)cc32)nn1 1623,C(=O)(C(C)CS(C)(=O)=O)N1C(NC(N(C2CCCCCC2)CC)=O)C2CCC1C2 1624,C1(CC)CN(C(=O)CCc2ccco2)CCC1CNC(c1cnc(C)cc1Cl)=O 1625,C(=O)(CCC(F)(F)F)NC(C(C)C)CNC(c1cccnc1N(C)C)=O 1626,C#CC1(NC(C2CC2C(C)NC(=O)C(CC)n2ccnc2)=O)CCCCC1 1627,c1(OC)cc(F)c(C(=O)NCC2CCC(C)CN2C(=O)CCNC(N)=O)cc1N 1628,c1(C(n2cc(C(C)(O)CCO)nn2)C(=O)NC)ccc2c(c1)CC(C)(C)O2 1629,C1(C(N2CC(C(C)NC(=O)C(C)C3=CCCC3)C2)=O)CCc2[nH]nc(O)c2C1 1630,c1(C(=O)NCCCCC(C)NC(C(C)NC(C)=O)=O)cc(C)c(F)cc1N 1631,CC1c2ccccc2CN1C(=O)CCN(CC(N1CCCCC1)=O)C 1632,Cc1nc2sccn2c1C(=O)NCC1(O)CC(NC(=O)Cc2ccsn2)C1 1633,Cc1c[nH]cc(C(=O)NCCCC2(NC(=O)COC3CC=CC3)CC2)c1=O 1634,c1(C(=O)NC2CN(C(c3c(C)[nH]c(=NCC)s3)=O)C2)cc2ccccc2n1C 1635,c1(C(N2C(C(N3CCN4CCC3CC4)=O)CC(=C)C2)=O)cc2nc(C)ccc2o1 1636,C1(CNC(Cn2c(C)cnc2)=O)CCCN(C(=O)Cc2cscn2)CC1 1637,N1(C(C(C(CC)C)C)=O)CCOC2(C1)CN(C(=O)CCCOC(=O)C(C)C)C2 1638,C1(C(=O)NC2(C3CN(C(COCCC#C)=O)C3)CC2)CCCCC12CC2(F)F 1639,c1(C(N(C(C(=O)N(C)CCOCCO)C2CC2)C)=O)ccc2n[nH]cc2c1 1640,Cc1cc(F)ccc1CC1(C(=O)NCC(CNC(C2CC2F)=O)CO)CC1 1641,C1(NC(C(C2CN(C(c3ccncc3Cl)=O)C2)OC)=O)CC=CCC1C 1642,Cc1cc(-n2nc(-c3nccs3)nc2C(C)CF)cc(C)n1 1643,c1(C(N(CC(C)(C)NC(=O)CNS(C)(=O)=O)C)=O)ccncc1F 1644,c1(C(=O)NC2CCC(N(C(=O)CNc3cccnc3)C)C2)cnn2ccccc12 1645,C1(F)(C(N(CCC(=O)OCC)C)=O)CCCN(C(C2CCC3(CCC3)C2)=O)C1 1646,CC1CCCn2ncc(C(N3CCN(C(=O)C(C)C(F)(F)F)CC3)=O)c21 1647,C1(OCC)CN(C(=O)C(C)(C)F)CC1CNC(c1cc(C)no1)=O 1648,C#CC1(O)CCN(C(=NCCC(=O)NC)NC)C1.S(=O)(=O)(CC)N 1649,c1(C(N(C)CCNC(=O)CC(F)(F)c2ccccc2)=O)cccc2oncc12 1650,c1(CCC(=O)NC(CNC(C(C)SC)=O)(C)C2CCC2)ccc(C)nc1 1651,c1(OC)cc(Nc2ccccc2)ccc1Br.N1CCN(C(=O)C(C)(COC)OC)CC1C 1652,C1(NC(=O)Cc2ccc(Cl)cn2)CC(F)CN(C(C2CC23CC3)=O)C1 1653,C12(C(=O)NC3C(CNC(c4ncc(C)cc4F)=O)C3)C3CCC(CC13)C2(F)F 1654,c1(C(N(C2CCCN(C(C(COC)C)=O)C2)CCF)=O)cccc(C)c1Cl 1655,C12(CNC(C(C3CCC3)OC)=O)CC(CO1)N(C(=O)C(C)(CO)NC(C)=O)C2 1656,c1(C(=O)O)nc(C(=O)NC2COC(C3CC3)C2)cs1 1657,O(N=C1CCCCCC1)CC(N1CCC2(NC(COC)=O)C(C1)C2)=O 1658,C1(NC(c2c(C)nns2)=O)CCCN(C(C2CCCN(c3ccccn3)C2)=O)C1 1659,Cn1cnc2ccc(C(=O)NCC3CCC(NC(C4CS(=O)(=O)C4)=O)C3)nc12 1660,N1(C(c2c(CCC)n[nH]c2)=O)CC2CC2C1C(N1CCC1C1CCOCC1)=O 1661,C(=O)(C(=O)N=S(C)(C)=O)N1C(CNC(c2ccc(CC)cc2Cl)=O)CC2CC21 1662,C12(CC(=O)NC3C(C(=O)Nc4c(Cl)cc(C)c(O)c4)C3)CC3CC(CC(C3)C1)C2 1663,C1(C(N2CCC(=CCC)C2)=O)CCN(C(c2cscc2C)=O)C12CC2 1664,c1(C(N2CCN(C(CCC=C)=O)CC2)=O)cc(S(=O)(=O)NC(C)C)c[nH]1 1665,C1(O)(C(C)NC(c2c(C)c[nH]c2CC(N)=O)=O)CCN(C(c2ccns2)=O)CC1 1666,C1(CC(=O)NC(c2c(C(N(CC#CC)C)=O)con2)C)CCN(C)C1=O 1667,c1(CC)cc(=NC(=O)c2conc2C(C)NC(C2CNC(=O)CC2C)=O)[nH]n1C 1668,C(=O)(C1COc2ccccc21)N1C2CCC(NC(CCC(CC)C)=O)(CC2)C1 1669,C1(C(=O)OC)(CNC(CCN(C(=O)CC(C)n2cccn2)CC)=O)CCCO1 1670,N1(C(c2cn(CC=C)nn2)=O)CCOC(C)(CNC(=O)CC=CCC)C1 1671,N1(C(=O)NC(CCF)C(=O)O)CCN(CCc2nc(C3CC3)no2)CC1 1672,CC1(C)C2CN(C(C3COC4(C3)CN(C(c3cnsn3)=O)C4)=O)CC12 1673,C(=O)(CC(CN(C)C)C(F)(F)F)NC(C(CO)NC(C1(CC)CCCC1)=O)C 1674,C1(C(=O)NC(C2CCN(C(c3ccc(N)c(N)c3)=O)C2)C)CCc2nnnn2CC1 1675,C#CCCCCCC(=O)N1CC2(CC(CNC(=O)C(C)C3=CCCC3)C2)C1 1676,c1(C(=O)NCc2ccc(C(N3CCC(CN(C)CC)C3)=O)s2)n[nH]c(C)c1Cl 1677,c1(C(=O)NCC2CC(NC(CCC=C(C)C)=O)C2)cc(F)cc(Br)c1F 1678,N1(C(C(C(C)C)(F)CNC(=O)C(C)CO)=O)CC2(CCC(O)CC2)C1 1679,C(=O)(C(C)S(=O)(=O)C(C)C)NCCN(C(c1c(N)sc(C)c1C)=O)C1CC1 1680,c1(C(C)SCC(c2ccc(OC)cc2)NC(C)=O)c(F)cc(Cl)cc1F 1681,c1(C(N2C(CNC(c3ccc(Cl)s3)=O)CCC2)=O)cc(O)nc(C2CC2)n1 1682,N1(C(C(CCC=C)NC(c2ccc(N)c(F)n2)=O)=O)CC2CCC(O)C2C1 1683,C(C(=O)N1CCN(C(=O)CC(C)(O)C2CC2)CC1CCO)(C(C)(C)C)NC(C)=O 1684,N1(C(c2cc(COC)no2)=O)CCC(O)(C(C)NC(=O)C(Cl)=CCl)C1 1685,C(C(CO)(CO)NC(c1ccn(C)n1)=O)N(C(C=CC=CCC)=O)C 1686,C1(C(=O)NC(c2cncnc2)C)(CC)CCN(C(=O)CC2CSCCO2)CC1 1687,C1(NC(c2ccc(C(N)=O)[nH]2)=O)COCCN(C(c2cc3occc3[nH]2)=O)C1 1688,CP(C)(=O)C(O)C(=O)N1CCC(O)(CNC(c2ccc(=O)oc2)=O)CC1 1689,c1(NC(=O)CC2CCN(CC(C)(C)C(N)=O)C2)cc(N)c(=O)n2c1CCCC2 1690,c1(NCCCCCC)ccc(S(=O)(=O)N2CCCC(C)C2CO)cc1C#N 1691,c1(C(=O)NCC2(CCNC(C3(CC)CCC3)=O)CC2)ccc(F)cc1C(F)F 1692,C1(C(=O)NCC2N(C(C(C(C)C)N(CC)CC)=O)CCOC2)CCCCCCC1 1693,S(=O)(=O)(c1cn(C)cn1)NCC(=O)N(CCN(C(c1c(C)cc(C)o1)=O)C)C 1694,CC1(C(=O)NC2C=CC(CC(=O)NCCc3noc(=O)n3C)C2)CC=CCC1 1695,N1(C(c2c(C)nn(C3CCO3)c2)C(=O)NC2CCCC2)CCNC(=O)CC1(C)C 1696,N1(c2nc(C(C)C)nc(Cl)c2)CCS(=O)(=O)C(CCNC(=O)CC=C(C)C)C1 1697,N1(C(C2C(COC)CC2)=O)CC2(CC2)CC1CO 1698,N1(C(c2cc(C)ns2)=O)CCC(NC(=O)Cc2ccsn2)C1C 1699,Cc1nc(O)ccc1C(N1CSCC1C(=O)NCC(C)(C)C#N)=O 1700,c1(N)ccc(Br)nc1.C(=O)(CC(=O)N1CC(CO)(NC(=O)CCCc2nccs2)C1)OC 1701,c1(OC)ccc2[nH]c(C(N3CC(C4CCCO4)C3)=O)cc2c1OC(F)F 1702,CCC(C)C(C(=O)N1CCOCC(CNC(c2ccsc2OC)=O)C1)OC 1703,CN1CC=C(CC(=O)NCC2C=CCN2C(=O)Cc2c(O)ncnc2O)CC1 1704,C1(C)(C(=O)NC(C)CNC(=O)C(Cc2ccccc2)n2cnnn2)COCCO1 1705,c1(C(=O)NC2(CNC(=O)COC3CCOC3)CCC2)ccn2nncc2c1 1706,C1(CC=C)(NC(=O)CC(C)(C)CC)CCCN(C(=O)CC2(C)CCCO2)C1 1707,CC1(C)CCC(O)(C(N2CC(CNC(c3csc(C(F)F)n3)=O)C(O)C2)=O)CC1 1708,CC1CN(C(=O)Cc2cccnc2Cl)CC1NC(=O)C(O)C1CCCC1 1709,C1(N(C(=O)CC2CC2(Cl)Cl)CC)CCN(C(=O)Cc2cncnc2O)CC1 1710,CC(C)(C)C(O)C(=O)NC1CCCN(C(c2cc(F)ccc2Cl)=O)CC1 1711,c1(C(n2ccnc2)CNC2(c3n(CC)nnn3)CCOC2)ncc(C)cc1C 1712,N1(C(c2c(C(C)C)n[nH]c2)=O)CC2CN(C(=O)C(c3cnccn3)C)CC2(C)C1 1713,c1(NC(c2n(C)ccn2)=O)sc2c(c1C(N1CCNCC13CCC3)=O)CCOC2 1714,c1(C(=O)NC2CCN(C(c3cc(C)c(C)o3)=O)C23CC3)cncc2ccsc12 1715,n1(C(C(=O)NCC2(C)CCN(C(COC)=O)C2)C)cc2ccccc2n1 1716,S(=O)(=O)(c1ccc2oc(=O)ccc2c1)N1CC2CCN(Cc3c(C)c[nH]c3)C2C1 1717,Cc1cc(C(N2CCC2C(N2CCC(O)C(C)C2)=O)=O)ccc1F 1718,N1(C(c2ccc(C=C)cc2)=O)CCN(C(=O)C(C)(C)C(=C)C)CC2CCCCC12 1719,N1(C(c2cc(C)[nH]n2)C(=O)NC(CC)(C)C)CCCC(S(C)(=O)=O)CC1 1720,c1(C(=O)NCC(CN(C(C(c2cccc(C)c2)=O)=O)C)(C)C)cc2n(n1)CCC2 1721,c1(CSC)cc(C(=O)NCC(C)CN(C(=O)CCNC(C2CCC2)=O)C)sc1C 1722,CCC(O)C(C)C(=O)NCC1CN(C)CCN1C(C1C=CCS1)=O 1723,N1(C(c2ccc(Cl)s2)=O)CC(CNC(C2CC(N3CCCC3)C2)=O)CC12CCC2 1724,CC(C(=O)NC1C=CCN(C(c2ccc(-c3cn[nH]c3)cn2)=O)C1)C(F)(F)F 1725,n1(CC(=O)N(CC(CO)(CO)NC(C2CC(C)(C)CO2)=O)C)cnc([N+](=O)[O-])c1 1726,C(C)(CO)(C(=O)NC(C)C(=O)NC(c1ncc(C)[nH]1)(C)C)OC 1727,c1(C(N(C2CN(C(c3c(F)ccc(F)c3N)=O)C2)C)=O)cccn2c(O)nnc12 1728,c1(NC(c2cnc3c(F)cccc3c2)C)nc(C2CC2)nc2[nH]ccc12 1729,CCCC(CNC(=O)CCNC(=O)CO)C(=O)NCC1COC(=O)N1 1730,N1(C(C2(NC(CC(CC)C(F)F)=O)CCCC2)=O)CCC2C(CCN2C)C1 1731,c1(CC(=O)NC2C3(CC(NC(C4N(CCC)CCC4)=O)C3)C2)cccc(F)c1F 1732,N1(CCC(=O)NC2(C)CN(C(CC3CC(OC)C3)=O)C2)C(=O)NC(C)(C)C1=O 1733,C1(NC(CCC#C)=O)(CNC(=O)CC(C)(C)C)CCCCCC1 1734,C1(COC)CC(N=c2[nH]c(=NCc3ccoc3C)[nH]c3c2CC(C)CC3)C1 1735,C(=O)(C1Cc2ccc(C)cc21)NCC(CNC(C(CC=C)CC)=O)(C)C 1736,C1(CCNC(C(CC#C)O)=O)CCN(C(c2cc(C(N)=O)no2)=O)CC1(F)F 1737,c1(C(N2CCC(CNC(C(C=C=C)C)=O)C2)=O)cc(C)nc2ccnn12 1738,CC(C)CC(C(=O)N(C)CC1C2CN(C(=O)C(C)(C)CN(C)C)CC12)NC(N)=O 1739,c1(C(=O)NCC(CC(C)C)NC(C)=O)cc(C(N)=O)cc(C)c1 1740,CN1CC(C(=O)NCCC2CCN(C(c3c[nH]c(=O)cn3)=O)C2)CCC1=O 1741,c1(C(C(=O)N(C(CN(C(C(C)OCC=C)=O)C)C)C)=O)ccc(Cl)cc1O 1742,C1(NC(C(C)C(F)F)=O)CCN(Cc2ccccc2)CC1NC(=O)OC(C)(C)C 1743,c1(CC(N2C(CNC(C3(C=C)CCCCC3)=O)CCC2)=O)ccc2c(c1)COC2 1744,C1(CC(=O)NCC=CCNC(c2c(N)cc(O)cc2)=O)Cc2ccccc2O1 1745,n1(Cc2ccc(C)o2)ccc2ccccc12.n12cc(nn1)C1CCN1C(=O)CC2 1746,c1(C(=O)NCC2N(C)CCN(C(=O)CCn3ccnc3)C2)cccn2cncc12 1747,c1(OCCCC(=O)OCC2C3CCC23)ccc2ccccc2c1 1748,C1(C)(NC(c2c(C)csc2)=O)CCN(C(=O)CC(c2ccccc2)N(C)C)C1 1749,CCC(C)(C)C(=O)C(=O)N1CCC(C2CCCN2C(c2ccc(Cl)o2)=O)C1 1750,c1(C(N(C2CN(C(CN(C)C)=O)C2)C)=O)cc(=O)cc[nH]1 1751,C(=O)(C1=CC2(CCOC2)C1)N1CCC(C(N(CC(CC)CC)CC)=O)CC1 1752,c1(CN(CCNC(c2cc(F)c(OCC)c(Br)c2)=O)C)ccc2occ(C)c2c1 1753,C1(C2CCCN(C(C3C(C)(C)C3(F)F)=O)C2)(NC(C=C(CCC)C)=O)CC1 1754,c1(OC)ccc([N+](=O)[O-])cc1C(N1CCN(C(=O)COc2nnc(C)s2)CC1)=O 1755,c1(C(=O)NC(C(=O)NC(CC#C)CCOC)CCC)cccc(C#N)c1C 1756,c1(CN2C(CC(=O)NC(C3CCCC3)C)CCC2)c(F)cccc1F 1757,c1(CNC2C(C(=O)NC(c3cncs3)C)CCC2)c2c(nn1C)CCC2 1758,c1(OC)cc(C)cnc1C(=O)NC(CCO)C(F)(F)F 1759,Cc1nc2cc(C(=O)NCC(O)CNC(=O)CC3=CCN(C)CC3)cc(O)c2o1 1760,CC(C(=O)N1CCC1CNC(=O)Cc1cscn1)n1ccnc1 1761,C1(C(N2CC3(CN(C(C(=C(C)C4CC4)F)=O)C3)C2)=O)CCC2(CC1)CNC(=O)C2 1762,C(=O)(C(C)CCCOC)NCCCC(C)(C)NC(c1cc(CC)[nH]n1)=O 1763,C#CCCCC(C)C(=O)NCC(CO)NC(c1cc(C(N)=O)[nH]n1)=O 1764,C(C(CC(=O)N1CCC(C)(N(C)C)C1)NC(C1CCCN1C1CC1)=O)OC 1765,C(=O)(C1CCOc2ccc(F)cc21)N1CC(CNC(C(Br)=C(C)C)=O)C1 1766,N1(S(C)(=O)=O)CCCCC(N=c2ccnc(NCC3CCCCCC3)[nH]2)C1 1767,Cc1[nH]c(C#N)cc1C(=O)NC1(CO)CCN(C(C2CC(C)(C)CN2C)=O)C1 1768,CP(C)(=O)CCC(=O)NC1CCN(C(=O)CCCc2csc(=N)[nH]2)C1 1769,Cn1ccc2c(C(=O)NCCC3CN(C(=O)Cn4ccnn4)CCO3)ccnc12 1770,c1(C2C(C(=O)NCC3(COC)CN(C(C4CCC4(C)C)=O)C3)C2)ccccc1Br 1771,c1(CC(=O)NCC=CCNC(c2n(CC)ccc2)=O)cnc(Cl)cc1C 1772,S(=O)(=O)(c1cccc(C(=O)NCCc2nc(=O)o[nH]2)c1)N(CC(=O)NC(C)C)C 1773,Cc1cnn(C)c1C(=O)NCC(c1ccccc1)N(C(=O)CCS(C)=O)C 1774,C(CCC(=O)NC(C)CN(C(=O)CCc1nc(C)no1)C)=CC 1775,C12(NC(CC3CCC(C)CO3)=O)CC(CNC(c3cncn3C)=O)(C1)OC2C 1776,C1(C(=O)Nc2nnc(C(C)C)s2)CC12CCN(C(c1ccc(CO)cc1)=O)C2 1777,CS(=O)CCC(O)C(=O)NC1(C)CN(C(=O)Cc2csc(-c3ncccn3)n2)C1 1778,C1(CC(=O)NC2CCOC2=O)CCCC2CN(C(=O)C3Cc4ccccc43)CC12 1779,N1(C(=O)NC(C(C)NC(=O)OC(C)(C)C)C)CC2CS(=O)(=O)CC2(C#N)C1 1780,N1(C(CCCCCC)=O)CCCC(CCn2cc(C(=O)N(C)OC)nn2)C1 1781,c1(N(CCNC(C2CC23CCOC3)=O)CC)c(Cl)cncc1[N+](=O)[O-] 1782,Cc1noc(C)c1C=CC(=O)NC1CC2CC1N(C(c1coc(C(N)=O)c1)=O)C2 1783,c1(CC(=O)NC2CCN(C(c3c(C)c[nH]c3)=O)CC2CO)cn2ccccc2n1 1784,c1(OC)ccc(Cl)cc1C(=O)NC(C)CNC(c1cccc(F)c1O)=O 1785,CC(CC(F)(F)F)C(=O)NC(CC1CC1)C(=O)N1CC(N2CCC2)C1 1786,c1(OC)c(C(=O)NCC2CSCN2)ccc(Cl)c1Cl 1787,C1(COC)(CNC(=O)CSCCN(C)C)CCCN1C(=O)C(C)(F)F 1788,c1(CCC)cccc(C(=O)N(C)CC2COCCN2C(=O)COC(=O)N(C)C)c1 1789,C1(CC(=O)NCCC(CNC(=O)CC(=O)Nc2nccs2)O)CC2C=CC1CC2 1790,c1(C(N2CC(OC(=O)NC(=O)C3CC3)C2)=O)ccc(I)nc1 1791,N1(C(CC(C(CC)C)O)=O)CC2N(C(=O)Cc3nnc(C)o3)CCC2(C)C1 1792,CCCCC(C(=O)N1CCN(C(C2CC3C(C2)C3(F)F)=O)CC1)NC(N)=O 1793,c1(C(N2CC(C)OCCC2)C(=O)NCCCF)ccc2c(Cl)n[nH]c2c1 1794,C(=O)(C(=O)N=S(C)(C)=O)N(CC(C)NC(C1CC(O)CN1C)=O)C 1795,C(=O)(C1SCCc2sccc21)N1C(CCNC(c2cc(C)ncc2)=O)CCC1 1796,c1(C(=O)NCC23CC(NC(C(C(C)C)OC)=O)(C2)C3)cc(NCC2CC2)nc(C)c1 1797,N1(C(=O)CC2(O)CCC2)CCCCC1CCNc1nccc(C(F)(F)F)n1 1798,N1(C(COCC(C)C)=O)CC(CNC(c2csc(Cl)n2)=O)OC(C(F)(F)F)C1 1799,C(C1CN(C(c2cc(C(N)=O)co2)=O)CC1C(N1CCC(C(N)=O)C1)=O)=CC 1800,c1(CC(=O)NC2CN(C(=O)C(O)CC(F)F)CC2O)cnc2ccccc2c1 1801,CC(O)C(C)(C)C(=O)NC1CCOC1C(=O)NC(c1nncs1)C 1802,C=CCCC(c1nnnn1C)(C1CCOCC1)NC(C)CCC(=C)C 1803,c1(C(=O)NC2C(NC(c3c(C)ccc(OC)c3)=O)C2)cccc2oc(C)cc12 1804,c1(C(=O)NCC(CN(C(=O)CC2(O)CC2)C)O)n[nH]cc1-c1ccccc1 1805,c1(C(=O)NC2COCCN(Cc3cccc(OC)c3)C2)n[nH]c2cc(Br)ccc12 1806,N1(C(COCCCCC)=O)CCC(NC(=O)C=COCC)C(C)C1 1807,C1(NC(C2(C)ON=C(C)C2)=O)CC2CC(NC(C3SCCS3)=O)C1C2 1808,C1(C(=O)NC2C=CC(CC(=O)NC(C)C(C)(C)C#N)C2)CC2CC(=O)C1O2 1809,c1(NCC2C(C)CN(C(C3CC(C)(C)C3)=O)C2)ncnc2c1nnn2CC1CC1 1810,C1(NC(COCCCC#C)=O)CC2(C1)CC2NC(=O)CCCOC1CCCCC1 1811,c1(CC)ccc(C=CC(N2CCCC2CN(C(=O)Cc2ncc(C)o2)C)=O)cc1 1812,N1(C(c2cc(OC)n[nH]2)=O)CCC(C)(CNC(C2CCC(=O)CC2C)=O)CC1 1813,C(=O)(C(C(C)CCC(=O)OC)N1CC2(C(=O)OC)CCCC12CO)NCC=C 1814,C1(OC)CC(C(=O)NC(CNC(c2cc(C(C)=O)on2)=O)C2CC2)CC1OC 1815,Cc1cc(N2CCC(NC(C3C(F)(F)C34CCC4)=O)C2C)n2nc(C)nc2n1 1816,C(=O)(CN=c1[nH]c(=NC2CC3C=CC2C3)c2ccccc2[nH]1)NC 1817,C(=O)(C1=CC2CCC=CCCC12)N1CC(NC(C2CC(O)(CC#C)C2)=O)C1 1818,C1(CC(=O)NC(C=CC=CCCCCCOC(C)(C)C)=O)COCC2(CCC2)O1 1819,c1(C(=O)NCC(C)(C)NC(Cc2c(C)noc2)=O)cnc2c(c1)nnn2C 1820,C1(CNC(C(CC)C)=O)COC(C)(C)CN1C(c1cnc(SC)nc1O)=O 1821,C12(OC)CCC(C(=O)NCCCNC(=O)Cc3cc(F)ccc3Cl)(CC1)C2 1822,c1(CC(=O)NC2C(CNC(c3cc(OC)n[nH]3)=O)C2)c(CC)cccc1CC 1823,CC1CCCCN1C(c1cccnc1CNC(C1CCN(C2CC2)C1)=O)=O 1824,c1(C(N(CCNC(=O)C=CSC)CC)=O)ccc(O)c(CO)c1 1825,C1C(C)CC(=O)N1.C(CC(=O)OC)N(C(=O)COCC(C)(C)C)CC#C 1826,C1(NC(CCc2nc(C)c(C)o2)=O)CC2CC(NC(C3OCCC3(C)C)=O)CC12 1827,C=CC(CCC)CC(=O)NC(CN=[N+]=[N-])C(=O)N(CC(C)C(=O)NC)C 1828,C(CC(O)CNC(=O)Cc1cnc[nH]1)NC(c1sccc1Cl)=O 1829,Cc1ccc(C(=O)NC2CCC(NC(C3CCCN3N=O)=O)CC2)c(F)c1 1830,CC(CC(=O)N(C1CCCN(C(=O)CCN2CCC2)C1)C)C(F)F 1831,c1(NC(C2CN(C(c3cnc(Cl)nc3)=O)CCC2O)=O)cc2c[nH]nc2cc1Br 1832,c1(C(C)=O)cn(CC(N2CC(C)(OCC(=O)NC3CCCCS3)C2)=O)nn1 1833,c1(OCC(=O)NC(CNC(C2(CC#C)CCCC2)=O)(C)CO)ccc(F)cn1 1834,c1(C(N(C(CNC(CCCC=C)=O)C)C)=O)cccc([N+](=O)[O-])c1O 1835,N1(C(CCc2n(C)cnn2)=O)CC2CC2(NC(=O)CCC2CCCOC2)C1 1836,c1(CC(N2C(C(C3CC3)NC(CCC)=O)CCC2)=O)cc(O)ccc1Br 1837,C1(NC(c2n(CC=C)ccc2)=O)CN(C(=O)C(C)(C)SC)CCC1CO 1838,c1(C2C(C(N(CC(C)(C)C)Cc3csnn3)=O)C2)ccccc1 1839,Cc1nc(C(N2CC3(NC(c4cnoc4C)=O)CC2C3)=O)ccc1C#N 1840,CC1CCCCCN1S(=O)(=O)CNc1ccccc1-c1ccc(Cl)c(F)c1 1841,C1(C(N2C3(CN(C(C(CCC)CC)=O)C3)CC2)=O)Cc2ccccc2C(C)(C)C1 1842,Cc1cc(C(N2CCC(C(=O)NCC3CCCC3O)(CF)C2)=O)ncc1N 1843,C1(C(=O)N(C(C(=O)N(C(C)C)C2CC2)C2CCCC2)C2CC2)CCC2CC1CO2 1844,Cc1cc(C)c(CN2CCC2(C)C(=O)Nc2ccc(C#N)cc2F)cc1C 1845,c1(C(=O)N(C(CO)CCc2ccncc2)CCO)cc(C(c2ccco2)=O)cs1 1846,Cc1cc(S(=O)(=O)NC(C)CCCCCO)c(C)cc1-c1sccc1C 1847,CC1(CNC(c2ccoc2)=O)CCN(C(=O)Cc2nnc(-c3ccccc3)o2)C1 1848,C(=O)(CC1C(=O)Nc2ccccc21)NC(C)C(CO)NC(=O)Cc1csc(Cl)n1 1849,C(=O)(CC(F)(F)CS(C)(=O)=O)NCC(CNC(C(CC#C)C1CC1)=O)O 1850,N1(C(C)=O)CCC(C2OCCC2NC(=O)C=C(C)C(C)C)CC1 1851,C12(C(=O)NCCCNC(C3(c4ccc(Cl)cc4)CCC3)=O)C=CC(CC1)C2 1852,C(C)(CC(=O)N1CCCCC1CNC(=O)CCCCCF)(C(F)(F)F)N(C)C 1853,n1(C2C(C)C2)nc(-c2ccccn2)nc1C1CC(c2ccc(Cl)s2)C1 1854,c1(CC)cc(C(N2CCCC2C(N2CC(CC(=O)OC)C2)=O)=O)ccn1 1855,c1(C(N2CC(C)C(N(C)CC34CCC(CO)(CC3)C4)CC2)=O)ccnc2cc[nH]c12 1856,Cn1cc(CNC(C2CC=CCN2C(=O)C(O)CC2CCCC2)=O)ccc1=O 1857,Cc1cnsc1C(=O)N(CC(C)C(=O)NC1CC(CF)C1)C 1858,CCCCC(CNC(C1(C(=O)N(C)C)CC1)=O)NC(=O)C(N1CCN(C)CC1)C 1859,c1(CC)nnc(CNC(=O)C=CC(C)NC(=O)Cc2ccc[nH]2)o1 1860,CCCC(C)CC(=O)NC1CC12CC(NC(c1c(C)nc(C)n1O)=O)C2 1861,CC1=NOC(C(=O)N(CCNC(=O)Cn2ccc(C)n2)CCOCCO)C1 1862,c1(C(N2CC(NC(C(C)(C(C)C)OC)=O)C2)=O)c(C)nc(C(C)(C)C)nc1O 1863,c1(C(N2CCC(C)(NC(COC)=O)CC2)=O)nccc2cnn(C)c12 1864,c1(C(=O)NC23C(CN(C(C4CC(=O)N(O)C4)=O)C2)CC3)sc2sccc2c1Cl 1865,C1(NC(c2ccc(CN(CCC)C)o2)=O)CCCN(C(=O)CCNC(C)=O)C1 1866,c1(CC)ccc(C(=O)NC(COC)C(=O)NCC(=O)NCC(F)F)o1 1867,c1(C(N2CCCC(N3CC(O)C3)C2)=O)ccc2ncsc2c1 1868,Cc1ccc(=O)n(CC(=O)NCC2CC2NC(=O)COC2(C)CCCC2)n1 1869,C1(NC(c2c(OC)cccn2)=O)CCCC12CN(C(=O)CC(C)(C)F)C2 1870,O=C(C1=CCCN(C(C2CCC2(F)F)=O)C1)NC(C(F)(F)F)C1CC1 1871,C12(C(=O)NC(C(=O)OC)C3CC3)CC1CN(C(=O)C(C)(C)CCl)C2 1872,C1(C(N2CCCC(C)(NC(c3cccc(F)c3F)=O)C2)=O)Cc2cccnc2C1 1873,c1(OC)ccc(O)cc1C(N1CC=C(CNC(C2(OC)CC2)=O)CC1)=O 1874,CC1CCN(C(c2cc(C(C)(C)C)no2)=O)CCN1C(C1CC1C(F)F)=O 1875,CN1CC(C(=O)NC(C)(C)CCNC(=O)COCC2CCCO2)NC1=O 1876,c1(C(=O)OC(C(=O)OCC)Cc2ccccc2)noc2c1CCCCC2 1877,N1(C(c2cnc(=N)[nH]c2)=O)CC2(CCC(CNC(C34CC5CC3C4C5O)=O)O2)C1 1878,C1(N(C(C2CC(C)(O)C2)=O)C)CCN(C(=O)C(F)(F)CO)CC12CC2 1879,N1(C(c2c(CC)nc[nH]2)=O)CCCC(O)(CCNC(c2cnc(C3CC3)[nH]2)=O)C1 1880,c1(C(C(C)C)NC(=O)NCC2CS(=O)(=O)C2)ccc(Cl)cc1 1881,N1(C(=O)CN2CCOCC2)CCC(CNC(C2CCCCO2)=O)C(O)C1 1882,C(=O)(C(C)(C)C(C)C)NCC(C)N(C(C1N(C(CCC)=O)CCCC1)=O)C 1883,C1(C(=O)NCCOC2CCN(C(C3(C(N)=O)CCC3)=O)C2)CCOC(=O)CC1 1884,CC1CCN(C(c2cnn(C(F)F)c2)=O)C1CNC(=O)CCOC1CCOCC1 1885,CCCC(CNC(=O)CCC(C)(F)F)C(=O)N1CCC(CC(F)F)C1 1886,c1(C(=O)NCC2COC(CNC(c3cc(Cl)no3)=O)C2)cccc(CO)n1 1887,CC(C)(C)C(=O)NCC1CCC1NC(C1CCCN1C(=O)Cc1ncc(Cl)s1)=O 1888,Cc1sc(N2CCCCC2)nc1CC(=O)NC1COCC1n1ccnc1 1889,C1(C(N2CCC(CNC(c3c(CC)noc3)=O)CC2)=O)CC1C1CCCC1 1890,CC1CCC(NC(=O)OC(C)(C)C)CN1C(c1ccoc1I)=O 1891,c1(C(N2CCN(C(c3ccc(C)cc3)=O)C3C2C3)=O)ccnc2ccnn12 1892,c1(C(C)NC(C2CC=CC2)=O)ccc(CNC(C2(c3cccs3)CC2)=O)cc1 1893,c1(OC)ccc(C(N2CC(CCO)(NC(=O)CSCCOC)C2)=O)c(N)c1Br 1894,C1(CC)CCN(c2nnc(O)s2)C1(C)C.c12cccc(c1)CC(C)CC(=O)N2 1895,CCCC(O)CC(=O)N1CCC(C(C)(C)C)(CNC(=O)CCS(C)(=O)=O)C1 1896,CC(C)S(=O)(=O)CC(=O)NCC1(F)CC(NC(C2CCC3(CCC3)O2)=O)C1 1897,CCC(C)(COC)CNC(C1CCN(C(=O)CCCCN(C)C)C1C)=O 1898,N1(C(CC2(COC)CC2)=O)CCCC(N(c2ncc(F)cn2)C)C1 1899,N1(C(COCC(=C)C)=O)CCC(N(C)Cc2cncs2)CC1 1900,N1(C(c2cc(Cl)cc(Cl)c2O)=O)CCC2CCN(C(C34CCC(C3)C4)=O)CC12 1901,C1(C)(C(N(CC(CNC(c2c(C)n(C3CC3)nc2)=O)(C)C)C)=O)COC(C)CO1 1902,CC1(C)CC(NC(=O)C(N)CCc2ccncc2)c2ccccc2O1 1903,C(C)(CN=c1[nH]c(C2(COC)CC2)nc(C)c1I)(C(C)C)c1c(OC)cccn1 1904,C(=O)(CC(C)(C)CCC)NCC1CC(C(=O)NC(CCCC)(C)C)C1 1905,n1(CC)cnc2c(NC(C)(COC)CCO)[nH]c(=NCCCCCN(C)C)nc12 1906,Cc1noc2ncc(OCC(C)N=c3nc[nH]s3)cc12 1907,N1(Cc2nc(CCCC)sc2)CCC(C)C(NC(C2CCS(=O)(=O)C2)=O)C1 1908,Cc1ccc(C)c(C(=O)NCC(CC(C)C)NC(c2cccnc2)=O)c1O 1909,C1(NC(C(C)SCC)=O)CCC2(CCN(C(c3ccsc3C(F)(F)F)=O)CC2)C1 1910,c1(C(N2CCC(O)(CC(N3CCC(C#N)CC3)=O)CC2)=O)c(Cl)cc(Br)cc1Cl 1911,C(CN=c1nc(Cl)[nH]c(C)c1C#N)CC.C12CCCCN1CC(=O)NC21COC1 1912,C1(CNC(C(C)Cc2cnc[nH]2)=O)(NC(=O)COCCCF)CCCCC1 1913,C1(C(=O)OC)CCC(CC(=O)N(Cc2cccc(C)c2)CC2CCCC2)CC1 1914,c1(C(=O)NCCCN(C)C(C2CCCS2)=O)cc(S(=O)(=O)N2CCOCC2)c[nH]1 1915,C1(NC(c2c(C(N)=O)csc2)=O)CS(=O)(=O)C2CN(C(c3cnns3)=O)CC12 1916,c1(C(=O)NCCNC(CC2(OCC)CCC2)=O)cncnc1C 1917,c1(CC)cnoc1C(=O)NC1CC(C)(NC(=O)C(C)C2CCCO2)C1 1918,N(C(=NCc1ccc(C)cc1)NCc1ccccc1NC(C)=O)C(CC)C 1919,CC(C)S(=O)(=O)c1cnc(NC(=O)Nc2ccc(CS(C)(=N)=O)cc2)nc1 1920,N1(C(C(=O)NC(C)COC2CCCOC2)=O)CC(N(C)CCO)C2(CC2)C1 1921,C(CCC(C)(C)NC(C1CC1C(C)(F)F)=O)NC(COCCOCC)=O 1922,CC1OCCCC1C(=O)NCC1CCCCC1NC(=O)CSc1nncn1C 1923,CCC(CC)(CO)C(=O)NCC1(CN(C)C(C2CCC3CCC23)=O)CC1 1924,Cc1cnc2c(C(=O)N(CC(O)CNC(=O)C=C3CCC(C)C3)C)cccn12 1925,C1(C)(CNC(=O)NC2CCC(SCC)C2)CC2(C1)OCCO2 1926,N1(C(CN2CC3(CN(C(=O)CCc4cscn4)C3)C2)=O)CCC(O)C(F)(F)C1 1927,C1(C)(CC(=O)N(C)CCNC(c2ccnc(OC(C)(C)C)c2)=O)CCS(=O)(=O)N1 1928,c1(C(=O)NC(CNC(CC(C=C)C)=O)C(C)(C)C)ccc(N)c(Cl)c1 1929,c1(C(=O)NCC2CCN(C(c3c(CCC)n(C)nc3)=O)C2)cc(Cl)ccc1OC 1930,c1(OC)ccccc1CC(=O)N(C1CN(C(c2c(Cl)nsc2Cl)=O)C1)C 1931,c1(C(=O)NCCOC2CN(C(c3c(C)oc(Cl)n3)=O)C2)ccc2c(c1)CC(=O)N2 1932,c1(CN(C(CC)C)CC2CCCC23CC3)ccc(F)cc1 1933,c1(OC)ccc(O)c(CNC2CCC(C(=O)Nc3nnc(Br)s3)CC2)c1 1934,c1(OC)nc(C)cc2ccc(C(=O)NC(C)CN(C)C(C3C=CCCC3)=O)cc12 1935,c1(C(=O)NC2CC(NC(C=CC3(C)COC3)=O)CC2O)cc2cnccc2o1 1936,C1(CN(C)C(c2ccnc(C(C)(C)C)n2)=O)CCN(C(=O)C(F)(F)CO)CC1 1937,C1(CNC(C(CSC)O)=O)CN(C(c2ccc3nccn3c2)=O)CCC12CCC2 1938,Cc1scc(C(=O)NC(c2ccc(F)cc2)CNC(c2cnc[nH]2)=O)c1C 1939,CC1CCC(NC(c2cn(C)ccc2=O)=O)CN1C(=O)CCc1ccon1 1940,Cc1cc(F)c(C(=O)NC2CCCCC2CNC(c2nc(O)sc2C)=O)c(Br)c1 1941,c1(C(=O)NC2C(C(F)(F)F)CCN(C(CC(=C)C)=O)C2)c(F)ccc2occc12 1942,Cc1cc(C(=O)NC2CN(C(C34CCCC3C4(F)F)=O)CC2C)cc(C)n1 1943,C1(C(=O)NC2CC(c3ccccn3)C2)C2Cc3cc(Br)ccc3C12 1944,c1(OC)ccnc(O)c1C(=O)NCC(C)N(C)C(c1cc(CO)[nH]n1)=O 1945,CC(C)(CCCCNC(=O)C(O)C1CC1)NC(c1cc(Cl)n[nH]1)=O 1946,C(=O)(C1CCCn2ccnc21)OC.C1(=O)C(C)(C)NCCCN1C(C)C 1947,c1(NCC(C(C)C)OC)ccc(S(=O)(=O)Nc2ccnc(CN(C)C)c2)c(Cl)c1 1948,C1(CC=C)N(c2ccnc(NCC3COCCC3(F)F)n2)CCCC1(C)C 1949,c1(C(N2C(C)(CNC(=O)C(F)CC3CC3)CCC2)=O)cccc2c1NCCC2 1950,N#Cc1sc(=NC2(C3CN(C(=O)CSC(F)(F)F)CC3)CCC2)[nH]c1Cl 1951,c1(C(N(CCCNC(C=C(C)C)=O)C(C)C)=O)nncn1C1CC1 1952,C1(NC(C(C)Cc2cnn(C)c2)=O)CCN(C(C23CCN(CC2)C3)=O)C12CCC2 1953,C1(CCNC(=O)C(O)C2CC2)CCCCN1C(C1CCC(O)CC1)=O 1954,c1(NC(N2CCC(CN(CCC)C)CC2)=O)c(Br)ccc(C)c1F 1955,S(=O)(=O)(c1ccc(NCc2ccn(C3CC3)n2)cc1Cl)NC(c1cnoc1)C 1956,C1(OC)CCN(C(=O)C(CC2CCC2)OC(=O)C=CCn2cncn2)CC1(C)C 1957,c1(C(=O)NCC2CN(C(C3COCC3C(F)F)=O)C2)ccc(-n2cccn2)cc1 1958,N1(C(CCCN(C)C)=O)CCC(C2(NC(=O)COc3nc(O)nc(O)n3)CC2)C1 1959,C1(CC(=O)NCC2CCN(Cc3ccc(O)cc3)CC2)CCc2ccccc2C1 1960,C1(C(N2CC3CN(C(CCCC(C)C)=O)CC3C2)=O)CCc2nn(C)cc2C1 1961,C(=O)(C(C)(CC)CO)NCC(N1CCN(C(C=CC=CCC)=O)CC1)C 1962,C(CCN=c1nc2c(c[nH]1)CCCC2)NC(=O)NCCCN1CCCCC1 1963,N1(C(C2(OC)CCCCCC2)=O)CC2CCCC1C2CNC(=O)C(C)(C)OC 1964,CC1(C)CN(C(c2cccnc2)=O)CC(CNC(=O)Cc2ccc(F)cc2Cl)O1 1965,Cc1cnc(CC(N2CCC(n3cc(C4CCCNC4=O)nn3)CC2)=O)cn1 1966,C1(NC(C(COC)(C)C)=O)CCN(C(=O)C(C)OCC(C)C)C12CC2 1967,N1(C(C(C)OCCOC)=O)CCN(C(c2sccc2CNN(C)C)=O)CC1.C(CO)C 1968,c1(C(=O)NCC2CCN(C(C3CN(CCC)C(=O)C3)=O)CC2)cc(C#N)[nH]c1C 1969,C(CC(=O)N1CC2(CCCC2)C1)(C(F)(F)F)NC(=O)C=CC1CCOCC1 1970,c1(NC(N2C(C)CN(CCc3ccc(Cl)cc3)CC2)=O)cn2cccnc2n1 1971,C=C(C)CCCC(=O)NC(C)Cn1cc(CN(CC)CC)nn1 1972,N1(C(C=C2CCN(C)CC2)=O)CC2CN(C(=O)CC3CCCO3)CC2C1 1973,C1(NC(=O)NC2CCCC2c2nc[nH]n2)CC2CCN(C1)C2 1974,CN1CCN2N1CCCC(OC(F)F)C(=O)N(C)C(CC)CCOCC2 1975,C12(C(=O)NC3CCN(CCNC(C4CC4F)=O)CC3)CCCC(CCC1)C2 1976,CCCCC(O)CC(=O)NC1CCCN(C(=O)C(C)(C)C(C)C)CC1 1977,C12(NC(c3cccc(OC)c3N)=O)CCC(CC1)N(C(C1CC(O)C(F)C1)=O)C2 1978,N1(C(CC2(C=C)CC2)=O)CC2CCC1CN2C(C1CC1CC(C)(C)C)=O 1979,c1(OC)ccccc1C(CNC(c1csc(Cl)c1)=O)NC(C1CCC12CCC2)=O 1980,C1(C(N2CCC(OCCNC(c3sc(CC)c(C)c3)=O)C2)=O)C(C2CC2)C1(F)F 1981,N1(C(CC=C=C)=O)CC(C(=O)NCc2nccc(=N)[nH]2)C(F)(F)C1 1982,C=CCCCCCCC(=O)NC1(C)CCCC1NC(=O)CC1C=CS(=O)(=O)C1 1983,N1(CC)CCCCC(N(c2cc(C(F)(F)F)ncn2)C2(C)CC2)C1 1984,C1(C(N2CCC(NC(C=CC(=O)N(C)C)=O)C(CO)C2)=O)C2(CCC2)C12CCC2 1985,n1(C(C)C)cc(CC(=O)NC2CCCC2NC(=O)CCOC2CCCCC2)nn1 1986,c1(C(=O)NCC2C(NC(=O)Cn3ccnn3)CC2)ccc(O)c(Br)c1 1987,C1(NC(C(C#C)(C)C)=O)CC2CCC1CN(C(C1CCC(F)CC1)=O)C2 1988,c1(C(N(C)CC2(O)CCN(C(C34OC(C)C(C3)C4)=O)C2)=O)cccc2occc12 1989,c1(OC)ccc(C(=O)Nc2ccc(-c3c[nH]nc3C3CC3)cn2)c(OC)c1OC 1990,n1(CCC)ncc(C(C(=O)Nc2ccccc2OC)N(C)CC)c1C 1991,c1(C(N(CCCCCNC(c2csc(Cl)n2)=O)C)=O)ccc([N+](=O)[O-])cn1 1992,C12(NC(C3CC3[N+](=O)[O-])=O)CCC(C1)N(C(=O)CNc1ccc(C(N)=O)cn1)C2 1993,C12(CNC(CSC)=O)CN(C(C3CCc4n[nH]cc4C3)=O)CC1CCO2 1994,N1(C(CC2(N(C(CC(C)C(F)F)=O)C)CC2)=O)CCC2(CCC(O)C2)C1 1995,C1(CNC(C2CCC(CC)O2)=O)(OC)CCN(C(=O)C(F)(F)c2ccccc2)C1 1996,Cc1ncnc(C)c1CC(=O)NCCCNC(C1CC2(F)CC1C2)=O 1997,c1(C(=O)NC(CC=C)CNC(=O)C(F)n2ccnc2)ccc(Cl)nc1O 1998,Nc1cc(C(N2CCCC2C2(NC(=O)C3=COCCC3)CC2)=O)cc(Br)n1 1999,C1(CNC(CSCCCC)=O)CCN(C(=O)CC2(CSC)CC2)C1 2000,C1(CC(=O)NCCOCCn2cc(-c3ccncc3)nn2)CC2COCC12 2001,N1(C(C2C3(CCN(C(CC4(N(C)C)CCC4)=O)C3)C2)=O)CCC(C2(C)CC2)CC1 2002,c1(C(N(C2CCN(C(=O)Cc3ccco3)C2)CCC)=O)ccc(C(C)=O)[nH]1 2003,N1(C(CCC2CC(NC(C3C(CC)OCC3)=O)C2)=O)CCc2oc(C)nc2C1 2004,C1(NC(C=CCOC)=O)CCCCC12CCN(C(=O)C(O)C(C)CC)C2 2005,c1(OCC)ccccc1C(=O)N(CCCNC(=O)CC1CC1C)C 2006,CCC(C)(CCCNC(=O)NCCCc1ccc(F)cc1)c1nccn1C 2007,C1(NC(c2ccc(-n3cncn3)cc2)=O)CCOCC1NC(c1ccns1)=O 2008,N1(C(c2ccc(CN3CCCC3=O)cc2)=O)CCC2(CC1)CC(O)CCO2 2009,C(=O)(C(O)C1=CCCCC1)N(C1CCN(C(=O)CSC2CC2)CC1)CC 2010,N1(C(c2cccc(C)c2)=O)CC(NC(=O)CSc2nc[nH]n2)C(C#N)C1 2011,c1(-c2c(C)n[nH]c2)cccc2c1CN(C(=O)Nc1ccc(Cl)cc1)CC2 2012,c1(NC2CCC(NC(c3cccc4nc(O)[nH]c34)=O)C2)ncc(Cl)cc1[N+](=O)[O-] 2013,CCCC(O)CC(=O)NC(C)(C)C(C)NC(=O)Nc1cc(N2CCCC2)ncn1 2014,Cc1cccn2cc(C(=O)NC3CC(CNC(=O)C(O)P(C)(C)=O)C(O)C3)cc12 2015,C(=O)(C(C)C(CC)CC)N1CC(CC(=O)N(CC(NOCC)=O)CC)C2(C1)CC2 2016,c1(C(=O)NC(C2CN(C)C2)C)ccc(CNC(c2cccn2C)=O)o1 2017,c1(NC(C2(NC(C3CC(Cl)(Cl)C3)=O)CCSC2)=O)cccc(F)c1 2018,C=C=C(C)CC(=O)NCC1(F)CCC(NC(=O)Cn2ncc(Br)c2C)C1 2019,CC(N=c1ccnc(Cl)[nH]1)C1CCN(C(=O)C(C)Cc2ccccc2)C1 2020,C1(C(N2CCC(N(C)C(C3CC4CC4C3)=O)CC2)=O)CCc2ccc(F)cc2C1 2021,c1(C(N2CCC(N(C(c3cc(C)cc(O)n3)=O)C)C2)=O)ccc2c(c1)N(C)CC2 2022,Cn1cc(C(N)=O)c(=NC(=O)C2CC(NS(=O)(=O)c3ccc(Cl)cc3)C2)[nH]1 2023,C1(OC)(CNC(=O)Cn2cc(Br)cn2)CCN(C(C2C3COCC23)=O)C1 2024,C1(C(=O)NC(c2nccc(O)n2)C)C=CCN(C(=O)Cn2ccnc2)C1 2025,C=CCCC(F)(F)C(=O)NC1CN(C(c2cc3ccccc3s2)=O)C1 2026,Cc1nc2cc(C(=O)NC(C)CCNC(C3CC(C)CC(=O)N3)=O)[nH]c2s1 2027,C(C(C)C(=O)NC1COCC1NC(C12CCC(C1)C2)=O)SC 2028,C1(C(=O)NC(C)CNC(=O)Cn2cnnc2)CCCCC12CCC2 2029,N1(C(c2c(C)noc2N)=O)CCCC(C)(C(=O)NC2CC(CC(C)(C)C)C2)C1 2030,C1(CNC(c2nocc2Cl)=O)CCN(C(=O)CCn2cc([N+](=O)[O-])cn2)C12CC2 2031,c1(C(C(=O)NCCOC)N(CC(C)S(C)(=O)=O)C)cnn(C)c1Cl 2032,C1(NC(C(C(COC)C)C)=O)CCCC12CCN(C(=O)Cn1nnc(=N)[nH]1)CC2 2033,C1(C(N(C)CC2COCCN2C(c2n[nH]cc2Br)=O)=O)CCC2(CCC2)O1 2034,c1(C(C)C)ccc(C(=O)NCC2CC2CNC(C2CCCO2)=O)cc1Br 2035,C1(NC(C2C(C(=O)OC)C=C2)=O)CCN(C(=O)C(C)OC)CC1NC(C)=O 2036,C1(C(=O)NCC2CCCC(CNC(=O)CCF)C2)CN2CCCC1C2 2037,c1(N2C(C)C(N(C)C)CC2)ccc(S(=O)(=O)NCCCc2cnoc2)cn1 2038,C1(C(N(CCC(=O)Nc2cncs2)C2CC2)=O)C=CCCC1 2039,c1(OC)ccc(C(=O)NCCNC(C2CCCN(C(C3CC3[N+](=O)[O-])=O)C2)=O)cc1 2040,c1(OCC)c(Cl)cc(NC(c2ccc([N+](=O)[O-])o2)=O)cc1Cl 2041,O=S(=O)(c1cccc(=NCCn2cnnn2)[nH]1)NC1(CO)CCCC1 2042,N1(C(C2CCN(C)CC2)=O)CCC(NC(=O)CO)C(F)(F)CC1 2043,N1(C(C(C)(C)c2cscn2)=O)CCC2(CCC2NC(=O)C=Cc2ccsc2)CC1 2044,c1(CC(=O)N(CCCNC(C(C)C2CCC2)=O)C)ccc(Cl)c2cccnc12 2045,N1(C(CC(C)(C)O)=O)CCN(C(=O)C=Cc2ccccn2)CC1CS(C)(=O)=O 2046,C1(CNC(=O)COc2ccccc2)CCC(NC(C2CC2C2CC2)=O)CC1 2047,CCCC(C)CC(=O)NC1CCC(NC(C2CCCO2)=O)C1 2048,C1(CNC(c2cc(C)sn2)=O)CCCCN(C(c2cc3[nH]ccc3s2)=O)C1 2049,c1(CC(=O)NCCNC(c2c(Cl)csc2Cl)=O)ccc2cccnc2c1 2050,c1(C(=O)NCCSCCC(F)(F)F)cnc2c(Br)cc(Br)cc2c1 2051,C1(C(=O)NC(c2cccc(C)n2)CC)CCCN(C(=O)C(=O)N(C)C)C1 2052,C(CC1CCN(C(=O)Nc2ccc(SC)c(C#N)c2)c2ccccc21)OC 2053,N1(C(CCCOCCC)=O)CCCC2CN(C(C3(F)CC34CCCCC4)=O)CC12 2054,c1(C(=O)NCCCCCNC(c2c[nH]c(=O)cn2)=O)cccc2cnccc12 2055,C=CCC(CNC(c1ccn(CCOC)c1)c1nnnn1C1COC1)CC(C)C 2056,C(=O)(CS(=O)(=O)C1CC1)NC1CC(CNC(c2c(C(F)(F)F)cccc2F)=O)C1 2057,C1(CC)CCCN(C(c2ccc(OC)s2)=O)C1C(=O)NC(C12CCC(CO1)C2)C 2058,c1(CC)c(C(=O)NCC2CN(C(c3csc(COC)n3)=O)CCO2)cccc1F 2059,c1(CC)nnsc1C(=O)NC1CN(C(=O)CCc2ncccn2)C1 2060,c12cc(ccc1OC(C)C)CCNc1ccc-2cc1.N1(CC)CCOCC1 2061,C12(NC(c3ccns3)=O)CCN(C(c3cncc(CO)c3)=O)CC1C2 2062,N1(C(c2nn(CC)c(C)c2)=O)CCN(C(=O)C=CCO)CC1CC(C)(C)C 2063,c12c(Cl)ccc-1c2F.N1(C(c2cc(Br)c[nH]2)=O)CCN(c2ccnc(O)c2)CC1 2064,c1(C(=O)NC2CN(C(c3ccc(OC)o3)=O)C2)cnc(OC)cc1C(F)F 2065,N1(C(C(CC)N2CCCC2=O)=O)CCN(C(C2(CO)CCC2)=O)CC1C1CC1 2066,C=CCC(CC)C(=O)NCCC1CN(C(=O)C(=O)NC2CC2)CCS1(=O)=O 2067,c1(C(N2CCC(CNC(C3CN4CCC3C4)=O)C2)=O)cn2ccccc2n1 2068,C1(C(=O)NC(CNC(C2(C)ON=C(C)C2)=O)(C)C2CCC2)CC2CC1CC2O 2069,CS(=O)(=O)c1ccccc1C1=CCN(C(=O)OC(C)(C)C)C1 2070,C(C(=O)NCc1ccco1)(c1ccns1)N(CCOC)CC1CC1 2071,C1(NC(c2cc(COC)sc2)=O)C=CCN(C(=O)CCN2CCC(F)C2)C1 2072,c1(CC)ccc(N)c(C(=O)NC2CN(C(=O)C(O)CC)CCC2C(F)(F)F)c1 2073,Cn1ncnc1C(=O)NCCNC(=O)CC1OCCO1 2074,O(C=CC(=O)N(C1CN(C(=O)CCc2ccc(Br)s2)C1)C)CC 2075,c1(C(=O)NCC(CO)NC(c2c(C)nn(C(C)(C)C)c2)=O)ccc(N=[N+]=[N-])cc1 2076,C=Cc1cncc(C(=O)NCCN(CCC)C(C2SCCS2)=O)c1 2077,C12(CC3(CCC3)C1)SC2.c1(NC(=O)NCCS(N)(=O)=O)nccc(C(F)(F)F)n1 2078,N1(C(C2(OC)CCOC2)=O)CC2=C(C1)CN(C(=O)C(c1cncnc1)C)C2 2079,N1(C(C2N(C(CCc3cc(C)[nH]n3)=O)CCC2)=O)CCC(O)C(C)C1 2080,C1(C(N2CCC(Nc3ccccc3F)CC2)=O)CCCCC12CCC2 2081,N(C1CCCOc2c(Br)cccc21)C(C)(C)C1CC1.C1(CC)(NC(=O)N)CCCOC1 2082,C12(CC(=O)NCC3(F)CN(C(C4C(C)C4)=O)C3)CCCN1CCC2 2083,C(C(C)(C)C)SCCCC1CCC1.C1(=O)CNC(=O)CC2(CC2)N1C 2084,c1(C(CC(N2CCC(N(C(C3CN(C4COC4)C3)=O)CC)C2)=O)C)c(C)noc1C 2085,n1(CC(=O)NC2CCn3nncc3C2)nc2ccccn2c1=O 2086,c1(C(=O)NCC(CNC(COCC(=O)OC)=O)O)cc(C)n(C2CCOC2)c1C 2087,c1(C(C)(C)C)nccc(C(N2CCC(C)(NC(C3CCCS3)=O)C2)=O)n1 2088,c1(COC)cccc(S(=O)(=O)NC(CCc2ccccc2)C(F)F)c1 2089,c1(C(N2C(CNC(CC(CC)C)=O)CCCC2)=O)cnc2sc(C)nc2c1 2090,CCCC(CC(=O)N1CCC(C(N)=O)(OC)C1)NC(C1(n2cnnn2)CC1)=O 2091,Cc1cc(C(N2CC3CC(C(N4CCOC(C(C)(C)C)C4)=O)(C3)C2)=O)cc(O)c1 2092,Cc1nccnc1C(=O)NC1CN(C(c2ccc(OCC3CC3)nc2)=O)CC1C 2093,c1(C(N2CCC(C#N)(NC(C3CCNC(=O)C3)=O)C2)=O)cc(O)c(O)c(O)c1 2094,CC1CC2N(C1)C2=O.c1(C(C(=O)NCCC(=O)OC(C)(C)C)=O)ccc(F)cc1 2095,C1(NC(c2c(C)cn(C)c2)=O)CN(C(=O)CC(O)CC2CC2)C2(CCOCC2)C1 2096,C1(NC(C2N(C(CNC(CCC)=O)=O)C3C(C2)C3)=O)CCN(C)C(=O)C1 2097,CCCCC(O)C(C)C(=O)NC(C)CCNC(=O)C1=CCCCCC1 2098,c1(-c2cnc(N3CCC(O)C(C)C3)nc2)cnc2ccccn12.C[SH](=O)=O 2099,N1(C(c2c(=N)[nH]cnc2)=O)CCOCC(CNC(c2sccc2CO)=O)C1 2100,CCCCC(C)C(=O)NC(c1nc(C(=O)NCCc2cccc(O)c2)co1)C 2101,c1(C(=O)NCC2C(NC(CC(C)F)=O)CC2)ccc(N2CCCC2)cn1 2102,Cc1c(C(=O)NC2CC(NC(c3cc(Cl)cc(Cl)c3)=O)C2)c[nH]c2nccc1-2 2103,Cc1c(F)ccc(O)c1C(=O)NC1CCN(C(=O)CC=C(Cl)Cl)CC1C(C)C 2104,c1(C(N(CC(CNC(c2[nH]cc(C)c2)=O)C)C)=O)cn(C2CCC2)nc1C 2105,c1(CC)ccc(C(=O)NC2(C)CCCN(C(c3ccnc(C)c3Cl)=O)C2)c(F)c1 2106,C(=O)(CC(C)CC(F)(F)F)NC(CC1CN(C(CC2(COC)CC2)=O)C1)C 2107,c1(C(N2CCC(Nc3cccnc3)CC2)=O)ccc(Br)cc1OC1CCCCC1 2108,C(=O)(C(F)C1=CCCCC1)N1CC2(C(NC(c3nc(OCC)oc3)=O)CCC2)C1 2109,C12(COC)CCC(C(N3CCC(CNC(=O)CC(C)(F)F)C3)=O)(CO1)C2 2110,N1(C(CCc2n(C)c(S)nn2)=O)CCCC(S(=O)(=O)N(C)C)C1 2111,C1(C(N2CC(CF)C2)=O)CCC2C(C1)C2(F)F.c12ccccc1Cn1cc-2nn1 2112,c1(C(=O)NC2CCCN(Cc3nc(C)[nH]n3)CC2)ccc(S(N)(=O)=O)cc1Cl 2113,C#Cc1ccc(NC(=O)C(C)(C)C2CCN(C(=O)CCOCC)C2)cn1 2114,N1(C(c2cncc(OC)c2)=O)CCN(C(c2cc(N)c(Cl)cn2)=O)CC(C)(F)C1 2115,N1(C(c2c(COC)ncs2)=O)CC(NC(c2cnn(C)c2C)=O)CC1C 2116,C12(CNC(c3c(C)scc3)=O)CCCC1CN(C(c1cnc3scc(C)n13)=O)C2 2117,c1(C(=O)NC(CC2CN(C(C3(CCOC)CC3)=O)C2)C)ccc(O)nc1 2118,Cc1cc(NC(C2CC2NC(c2cc(Cl)ccc2O)=O)=O)ncc1F 2119,C(=O)(C1=CCSC1)NC(C)CN(C)C(C1CN(C(=O)OC(C)(C)C)C1)=O.C(=O)N(C)C 2120,Cc1ccccc1OCCC(=O)NCC1CC(F)CN1C(=O)CC(C)(F)F 2121,N1(C(C2CN(C(CCC)C)C(=O)C2)=O)CCN(C(=O)C=C(C)C)C2COCC12 2122,C(CC(F)F)(C(=O)NCC1(O)CCN(C)C1)N(C(c1n(CC)ccc1)=O)C 2123,C1(CNC(C2(OC)CCOC2)=O)CN(C(=O)CC2(C)OCCO2)CCC1(C)C 2124,C(CCCCC(=O)NC1CCCC(CC)C1)=CCCC 2125,C1(NC(C2C(NC(C34CCC(CC3)CC4)=O)CCCC2)=O)CCC=CCCC1 2126,c1(CC(=O)NCCCC(C)NC(=O)COC2CCC2)c[nH]c2ncccc12 2127,c1(C(=O)NCC23C(CN(C(C4C(C)(C)OC(=O)C4)=O)C2)C3)cccn2nnnc12 2128,c1(Cc2cccc(NC(CN3CCC(=CCC)C3)=O)c2)ccn(C)c(=O)c1 2129,N1(C(CNS(NC)(=O)=O)=O)CCC2CCN(C(c3n[nH]c4c3CCC4)=O)CC12 2130,C12(C(=O)NC3(COCC)CC3)CC(NC(C3CCSC3)=O)(C1)C2 2131,c1(C(=O)NC2CC3(C(C(=O)NC4(C)CC(=C)C4)C3)C2)ccc(C#N)cn1 2132,N1(C(C(C=CCCC)O)=O)CCCCC(NC(c2ccc(CSC)cc2)=O)C1 2133,CCC(CCC(=O)N1CC2C(C(=O)NCN)C2C1)NC(C1CC(OC)(OC)C1)=O 2134,C(=O)(C1=CSCS1)NC(CNC(=O)C=Cc1ccccn1)C1CCC1 2135,C1(NC(=O)CSC(F)(F)F)(CO)CCN(C(c2ccc(CF)cc2)=O)C1 2136,c1(C(=O)NC2C3CN(C(C#CC4(CC)CC4)=O)C2C3)cccc2cc(F)ccc12 2137,N1(C(c2cn(CC(N)=O)nn2)=O)CCCC(N(CCO)C(c2cnccn2)=O)C1 2138,Cc1nn(CC(=O)NC(C)CNC(=O)Cc2ncc(Cl)s2)c2ncccc12 2139,CC(F)CC(=O)N(C1(CC(N2CC=CC2CF)=O)CC1)C 2140,c1(OC(C)C(N2CCCCC2CNC(c2ccc(Cl)cn2)=O)=O)ccccc1F 2141,n1(CC(=O)OC(C)(C)C)nnnc1C(=O)Nc1nccn1-c1ccccn1 2142,c1(C(=O)NC2CCN(C(C3CCC(CC)CC3)=O)C2)nn(C)c2ccc(Br)cc12 2143,N1(C(C2C(C)(C)C2(C)C)=O)CCC2C(NC(c3cc(=O)cc[nH]3)=O)C2CC1 2144,c1(OC)ncc(C(=O)NCC2CCN(C(C3CC(F)C3)=O)C2)cn1 2145,c1(C(=O)NCC(c2ccccc2)NC(C2(CC=C)CCC2)=O)ccc(N)c(N)n1 2146,c1(OC)c(NCC2CCN(C(=O)CC3(OC)CCCC3)C2)ncnc1C 2147,Cc1cc(CC(=O)NC2CN(C(c3cn[nH]c3C(C)C)=O)CC2(C)C)cc(F)c1 2148,CC(O)CCC(=O)NCC(C)N(C(=O)CCc1ccco1)C 2149,Cc1ncc(Cl)cc1NC(C1CCC(NC(=O)CCOCC(C)C)CC1)=O 2150,CS(=O)(=O)c1cnn(CC(O)CNCC2OCCC2CC2CCCC2)c1 2151,C(=O)(CN1C(=O)C(N(C)CC2CCCN2C)CCc2ccccc21)NC(C#C)C 2152,N1(C(c2c(C)cc[nH]2)=O)CCOCC12COCCN(C(c1ccn(C)n1)=O)C2 2153,c1(C(N2CC(C(C)NC(=O)CC(C)F)C2)=O)ccc(S(N)(=O)=O)o1 2154,C1(CCNC(C2C(OC)CCC2)=O)CCN(C(=O)C=CCCC=C(C)C)CC1 2155,c1(C(N2CC3C(N(C(c4c(OC)ccs4)=O)C)C3C2)=O)cccc(C)c1O 2156,C(=O)(CC(C(F)(F)F)NC(C1(C2(C)CC2)CC1)=O)NCc1ccc(C)cc1 2157,N1(C(=O)CC2(C)CCCO2)CCC(CCN(CC(N2CCCC2CC)=O)C)CC1 2158,C1(C(=O)O)(N(C(=O)CCc2nc(-c3ccncc3)no2)CCO)CCC12CCC2 2159,N1(C(c2cc(CCC)on2)=O)CCC(NC(C2CC(CCC)C2)=O)CC(C)(C)C1 2160,c1(N2CCCC(N(C(COCc3cc(C)on3)=O)C)C2)ncc(Br)cc1C#N 2161,N1(C(CCNC(COC)=O)=O)CCCC(C)(C)C1C(N1CC(c2nncs2)C1)=O 2162,c1(C(N(C(CC)C(=O)N(C2(C)CC2)C)C)=O)ccc2n[nH]cc2c1 2163,N1(C(Cc2cc(C)no2)=O)CC2C(C(N3CCC3Cc3ccccc3)=O)C2C1 2164,c1(NC2CN(C(C)=O)C2)ncccc1S(=O)(=O)N1CCC(=C(F)F)CC1 2165,C1(C(=O)NCCN(C(CCCCN(C)C)=O)CC2CC2)CC1C1CCCCC1 2166,C1(C(=O)NCCC(CNC(c2c(C)ccs2)=O)O)Cc2c(F)cccc2O1 2167,N1(C(=O)CC2(CBr)CCCC2)CCS(=O)(=O)CC1c1ccccc1 2168,N1(C(Cn2c(CCC)ncc2)=O)CCOCC1CCNC(C1C=CCS1)=O 2169,c1(OC)ccc(C(N2CCC(NC(=O)Cc3ccoc3C)CC2)=O)cc1[N+](=O)[O-] 2170,c1(C(=O)OC)c(C)[nH]c(C(=O)NC2CC2NC(c2c[nH]cc2C(C)C)=O)c1C 2171,N1(C(=O)Nc2ccc(C(=O)NC)c(Cl)c2)Cc2cccc(Cl)c2C1 2172,c1(C(=O)OC)cc(Br)ccc1CN1CC(C(=O)N(C)CCF)CC(C)C1 2173,C1(NC(C2(NC(c3cccc(=O)n3C)=O)CCN(C)C2)=O)CN2CCC1(F)CC2 2174,C1(O)(C(c2cn(CC3CCCN3C(=O)Cn3cccn3)nn2)C)CCN(C)CC1 2175,c1(SCC#C)cccc(C(=O)NCCOCCN(C(=O)C(C)=C2CCC2)C)c1 2176,C1(NC(C2CCCC(NC(c3c(C)nsc3)=O)C2)=O)CC(=O)NC(=O)C1 2177,C1(NC(c2c(CN(C(CCn3ncc(C)c3)=O)C3CC3)n[nH]c2)=O)C=CC(C)(C)CC1 2178,c1(-n2c(CCCCCOC)nc(CCOC)n2)cc(C)ccc1C 2179,C1(NC(COCC)=O)(CO)CCCN(C(c2cnc(N)c(Br)c2)=O)C1 2180,C(=O)(C(CC(F)F)NC(=O)CC1CCCCN1C)NCC1CCCN(C)C1 2181,C1(C(=O)NCC(CNC(C2(Br)CC2)=O)O)CC12CCOCC2 2182,N1(C(C(C2CCOC2)NC(CCCCCC#N)=O)=O)CC2(CCC(=O)NC2)C1 2183,CCC(Cc1ccccc1C)C(=O)NCC(C)(O)CNC(C1(C(C)(F)F)CC1)=O 2184,C12(NC(C(CSC)OC)=O)CCCC1(F)CN(C(=O)CCCC(F)(F)F)C2 2185,N1(C(c2c(F)ccc(OC)c2F)=O)CC(C)CN(C(c2cc[nH]c2C)=O)C(C)C1 2186,N1(C(c2ccc(OC)cc2)=O)CCC(F)CC1C(=O)Nc1cc(C)cc(O)c1 2187,c1(OCC)nccc(C)c1NC(c1ccc(-c2c[nH]c(=N)c(C)c2)c(C)n1)=O 2188,C(=O)(CC(C)C(C)(C)C)N1CC(C=CC)C(C(=O)NC2CN(CCC)C2)C1 2189,c1(C(=O)NC2CC(C(F)C(N3CCC(CCO)C3)=O)C2)cncc(Cl)c1 2190,c1(OC)ccc(C)c(C(N2CC3(CC3)CC2CNC(C2CCC3CCC23)=O)=O)c1 2191,C1(C(=O)NC2CC(O)C2)C2CC(O)C(C2)N1C(c1ccn2ccnc2c1)=O 2192,Cc1cc(C(N2CCOCC(NC(c3ccc(C(N)=O)o3)=O)C2)=O)nc(C)c1 2193,CCCCCC(C)CC(=O)NC1CN(C(C2CC(F)(F)C2)=O)CC1SC 2194,C1(CCC)CN(C(=O)C=Cc2csc(C(F)(F)F)c2)CCN1C(=O)C(O)CC 2195,CCC(C(=O)NCc1cn(CC(C)NC(=O)C(O)C2CC2)nn1)SC 2196,c1(C(c2cn(CCOCC(N3C(C(N(C)C)=O)CCC3)=O)nn2)O)ccccc1Cl 2197,c1(C(=O)NCC2(NC(C3CCCCC3F)=O)CC2)c(F)ccc(F)c1Cl 2198,C1(NC(C2CCCC2C(F)F)=O)CC2CC1N(C(c1ccncc1)=O)C2 2199,c1(CC)onc(C)c1CNC(=O)C(C1CCN(C(=O)CC2(C)CC2)CC1)C 2200,Cc1c(OC(F)F)cccc1Cl.n1(C2CNC2)cc(Br)ccc1=O 2201,Cc1nc(C(=O)N(C2CN(C(c3conc3C)=O)C2)C)ccc1F 2202,C1(NC(C2C(C(C)=O)C2(C)C)=O)CC(NC(c2nn(C)cc2Cl)=O)C12CCC2 2203,N1(C(C(C)n2ccnc2)=O)CC(S)CC12CCOCC2 2204,c1(C(=O)NC2C(CNC(C(CC#C)O)=O)C2)ccc(COC)c(F)c1 2205,C1(C(=O)O)(NC(C2C(CCC)C2)=O)CCOc2ccccc21 2206,c1(CC)cnc(O)c(C(=O)NC2CN(C(=O)Cn3cc(CO)nn3)CC2C)c1 2207,c1(C(=O)NCC(C)N(C(c2c(C)ncs2)=O)C)cccc(Br)c1Cl 2208,C(=O)(CC(C)CC(C)(C)C)N1C(COC)(CNC(C2CCCC(C)C2)=O)CCC1 2209,c1(CCNC(C2(NC(C3CCCC3)=O)CC2)=O)cccc(F)c1F 2210,c1(N(CCCS(C)(=O)=O)C)ccc(S(=O)(=O)N2CCSC3CCC23)cn1 2211,CC1CN(C(c2cccc(=S)n2O)=O)CCCN1C(C1CCCCS1)=O 2212,N1(c2cc(C)nc(C(F)(F)F)n2)CC2CCN(Cc3ccccc3)CC(C2)C1 2213,N1(C(C(C2CCC2)OC)=O)CC2(CC2)CC1CNC(=O)CCOCCN(C)C 2214,C1(CNC(c2c(OCC)scc2)=O)CCC(C)(C)CN1C(=O)C(C)CF 2215,c1(C(=O)NCC(C2CC2)NC(c2c[nH]cc2Br)=O)ccc(C(F)F)c(F)c1 2216,N1(C(Cn2cc(-c3cn(C(C)C)nc3)nn2)=O)CC(F)(F)CCC1C 2217,C(C)(CCC(=O)NCC1CC(C(=O)NCc2cccc(F)n2)C1)SC 2218,N1(C(C2C(=C)C2)=O)CCOCC12COCCN(C(c1ccc3ccnn3c1)=O)C2 2219,N1(C(C(CCCC)F)=O)CC2CCN(C(=O)CS(=O)(=O)C(C)(C)C)CC2C1 2220,N1(C(C=C(CCC)C)=O)CCN(C(=O)CC2COCC2O)CC1COC 2221,c1(C(=O)NCC(CC(=O)NC(CN(CCOC)C)C)OC)ccc2[nH]ccc2n1 2222,C(C(C)(CC)C(=O)NCC(C)(COC)CC)NC(C1CN(CC)C(=O)C1)=O 2223,N1(C(C(C(C)C)O)=O)CCC(C)(C)C1C(=O)NC1(CC(C)(C)C)CC1 2224,C1(CNC(CC2CC(OC)C2)=O)OCCC1C(=O)NC1(c2nc(C)no2)CC1 2225,c1(C(=O)NCCCCCN(C(=O)CCCN=[N+]=[N-])C)cc2n(n1)CCCC2O 2226,c1(C(=O)NC2C(NC(c3ncn(CC)n3)=O)CCC2)cc2ccc(Cl)cc2[nH]1 2227,C(=O)(CC1=CCOCC1)NCC(CC(F)(F)F)NC(C(CC#C)(C)C)=O 2228,C(CCN=C(NCCF)NC1CC1(C)C)OC(Cn1cccn1)OC 2229,C=Cc1ccc(C(N2CC3CCC2C3NC(=O)Cc2ccn(C)n2)=O)cc1 2230,C(=O)(C(O)CC(F)F)NCC1C(NC(c2c(C)nsc2N)=O)CCC1 2231,C1(CNC(c2c(CC)con2)=O)CN(c2cc(C)nc(COC)n2)CC(C)(C)O1 2232,c1(-c2nc(CCOC)nn2CC(C)(C)CO)cc(C)nc2c1nc(C)n2C 2233,CC(C)(CC#N)C(=O)N1CCC(NC(=O)C(c2ccccc2F)(F)F)C(O)C1 2234,Cc1cc(NC(C)CCCCNC(=O)C(O)C2CCC2)c(Br)cc1[N+](=O)[O-] 2235,c1(C(N(CC(=O)C(C)=O)C)=O)cnn(CCNC(=O)C(C)C#N)c1.NC(C)C 2236,c1(C(=O)NC2CN(C(C3(CC=C)CC3)=O)CC23CC3)ccc2c(Br)cnn2c1 2237,c1(OCCCC(=O)NCC(CNC(C(C=C)O)=O)OC)ccc(C)cc1 2238,C(=O)(C(C)(C)C(C)(F)F)NC(CN(C(C1N(CC)CC1)=O)C)Cc1ccccc1 2239,c1(C(=O)NC(C(C(C)C)NC(c2ccccc2O)=O)C)cncn(C)c1=O 2240,N1(C(CC2CCCN(C)C2)=O)CCC(F)(CNC(c2sccc2C(F)F)=O)CC1 2241,CC1CCN(C(c2cccc(C3CC3)c2)=O)CCN1C(=O)Cc1ncc(Cl)s1 2242,C(=O)(CCCCCCS(N)(=O)=O)NCCC(C)NC(Cn1ncc(CC)c1)=O 2243,c1(CC(N2CCOCC(NC(c3cn(C)c(O)n3)=O)C2)=O)cnc2ncccn12 2244,c1(C(N2C(C)CC(NC(C=C(C)C)=O)C2)=O)[nH]c2c(c1C)CCCC2 2245,C1(CC)CCCCCCN1C(=O)CC(C)C(C)(C)NC(c1cccc(O)c1F)=O 2246,C(=O)(CC1=CCN(C(C2(SC)CC(=O)C2)=O)CC1)N1CC(CC)OCC1C 2247,CCS(=O)(=O)c1ccc(C(=O)NCC2CCN2C(C2CC3(CCC3O)C2)=O)cc1 2248,C=C=C(C)CC(=O)NCC(CNC(c1ccc(OC(C)C)nn1)=O)CO 2249,N1(C(c2nnc(CC)o2)C)CCC(NC(c2nccn2C)=O)C(C)C1 2250,C(CO)(C(=O)NCCOCCN=[N+]=[N-])NC(C(C)OCCC(C)C)=O 2251,c1(NC(C2N(C(c3cc(C)no3)=O)CC(F)C2)=O)cc2nccn2cn1 2252,Cc1nn(CC(C)C)c(C)c1CNC(C12CCC(CN1C(=O)OC(C)(C)C)C2)C 2253,CCC(C)C(C(=O)NCC1N(C(C2CC3CC2CC3O)=O)CCC1)N(C)C 2254,CCC(CC)CCC(=O)NCC1(NC(=O)CCC2CC2(Cl)Cl)CCOC1 2255,c1(C(N2CCCC(N(C(CC(C=C)C)=O)CC)C2)=O)ccc2c(c1)OCCN2 2256,N1(C(CS(CC)=O)=O)CCN(C(c2cn(C3CC3)nc2C)=O)C2(CC2)C1 2257,N1(N(c2ncccn2)CC)CCOC2(CCN(C(=O)CC(C)(O)COC)C2)C1.C(C)=O 2258,c1(OC)cc(C)c(C(N2CC(C)(NC(c3cnn4cccnc34)=O)C2)=O)c(C)c1 2259,C(CCC(N)=O)(C(=O)NCC1CCN(C(c2cc(C3CC3)ns2)=O)CC1)N(C)C 2260,C(=O)(C(C)(C)CC#N)NC(CCOCC)C(=O)NC(CC(N)=O)C1CC1 2261,c1(N(C)C)ccnc(C(=O)NC2CCC2CNC(=O)CNc2cccnc2)c1 2262,N1(C(C(C)NC(CC)=O)=O)CCc2ccccc2C(NC(=O)Cc2csnn2)C1 2263,N1(C(c2c(C)nc(C)s2)=O)CCN(C(c2cccc(Cl)c2O)=O)C(C2CC2)C1 2264,Cc1ccc(C(N2CCN(C(=O)C(N3CCCC3)C3CC3)CC2C)=O)c(C)n1 2265,C12(C(=O)NCC#CCNC(c3c(N)c(F)ccc3)=O)CC1COC21CCC1 2266,O(C1CCCc2ccccc21)Cc1c(C(=O)O)nn(C)c1Cl 2267,Cc1cc[nH]c(=N)c1C(=O)NCC(C)NC(c1cnn(-c2cccc(F)c2)c1)=O 2268,C(CC(C(=O)N1CCC(CCCO)CC1)NC(c1ccccc1)=O)OC 2269,c1(C(=O)NCC(CC)NC(c2cn(C)c(C(F)F)n2)=O)cc(C)cc2c1CCC2 2270,N1(C(CCc2ccn(C)n2)=O)CC(CNC(C2(C#N)CC3CC3C2)=O)C(C)(C)C1 2271,C(=O)(C(CC(C)C)C(C)C)N(CC(C)NC(c1c(C)cc(C)nc1S)=O)C 2272,c1(C(=O)NCCN(C(=O)CC2CC2(C)C)C)cccnn1 2273,N1(C(C(C)C2(O)CCC2)=O)CCN(c2ncnn3cccc23)C(C#N)C1 2274,C(=O)(CC(CC)C(C)C)N1CCC(CC)C1C(=O)NCCCn1cncn1 2275,C1(C(N2C(CCCNC(c3cn(CC)nn3)=O)CCC2)=O)CN(C)CC(C)O1 2276,c1(C(=O)NC2CC(CNC(Cc3c(C)cco3)=O)C2)cc(F)ccc1N 2277,c1(C(=O)NCC2N(C(C3CCN(CC)C3)=O)CCOC2)[nH]cc2c1CCCC2 2278,N1(C(Cn2ncc(C)c2)=O)CCC2CCC(C1)N2C(=O)CC1CN2CCCC1C2 2279,C(C(C)CN(C)N1CCC(C(c2nccs2)O)CC1)c1ccc(C)cc1 2280,c1(C(=O)NC2CC(C(=O)NC(CCC)CCO)CC2O)cccc(O)c1C 2281,C=C=CC(C)C(=O)NCc1ccc(C(=O)NCCC2CCCCC2)cc1 2282,N1(C(=O)Cn2cnnc2)CCC2(CCN(C(c3c(F)ccc(F)c3F)=O)C2)C1 2283,c1(CCC(=O)NC2CCCC(N(C(=O)Cn3ccnn3)C)C2)cccc(F)c1Cl 2284,C(=O)(CCC(=O)N1CCCC1(CC(C)C)C(=O)O)OCC 2285,n1(CC)ncc(CNC(C2C=CCCN2C(C2CC3CCC3C2)=O)=O)c1C 2286,FC1(F)C2(CCC2)C12CC(NCC1(c3ccccc3Cl)CCC1)C2 2287,C1(NC(c2cc(OCC)ncc2)=O)C2CC1CN(C(c1cscn1)=O)C2 2288,CC(CC(=O)N1CC(NC(c2ccc(CO)o2)=O)C2(CC2)C1)C(F)(F)C(F)(F)F 2289,C1(CNC(C2(C(=O)NC)CCC2)=O)CCC(C(=O)NCc2ncc(C)o2)C1 2290,c12ccccc1OC2.c1(C(=O)OCCNC(CCN(CC)CC)=O)ccc(Cl)s1 2291,N1(C(C(CCC)OC)=O)CC2(CCCCN(C(=O)C(c3cncc(F)c3)C)C2)C1 2292,c1(CNC2C(C(=O)NCC3(C)CCC3)CCCC2)ccc(O)c(O)c1 2293,C1(C(=O)NCCC=CCCC)CN(C(=O)CCC=C(C)C)CCC1(C)C 2294,c1(C(=O)NCCN(C(=O)C(n2ccc(Br)n2)C)CC)c(C)ncn1O 2295,c1(OC)cc(C)ccc1C(=O)NC1C=CCN(C(C2(C#N)CC3CC3C2)=O)C1 2296,c1(C(=O)NCC2(CNC(c3cc(COC)no3)=O)CC2(F)F)cnc[nH]c1=N 2297,c1(C(=O)NCCCC2N(C(C(C)SC(C)C)=O)CCC2)cc(Br)n(C)c1 2298,c1(C(C(N2CCN(C(c3cc(C)nnc3)=O)CC2)=O)=O)c(C)nn(C)c1C 2299,C1(NC(=O)Cn2cnnn2)CN(C(c2cc(F)c[nH]2)=O)CC2(CCC2)C1 2300,c1(CCC)[nH]ccc1C(=O)NCC(C)N(C)C(c1cnc(-c2cccnc2)s1)=O 2301,c1(C(N2CC(N(C)C(C3CC4C=CC3O4)=O)C3(C2)CC3)=O)ccc(S(C)(=O)=O)[nH]1 2302,C(=O)(C(C)(C)CC(=O)N(C)CC1(O)CCN(C(=O)C2=NNC(=O)CC2)CC1)OC 2303,C(Cc1ccccc1)(CCNC(=O)CN(C1CCC1)C)NC(C(C)O)=O 2304,N1(C(c2csc(Cl)c2)=O)CCCN(C(=O)C(O)C2CCCC2)C(CO)C1 2305,O=C(C1NCCc2ccccc21)NCC(C1CCCCC1)=O 2306,c1(C(=O)NCC2N(C)CCN(C(C(C(C)C)C)=O)C2)cncc([N+](=O)[O-])c1 2307,CCC(F)(CNC(=O)NC(c1ccc(Cl)nc1)C1CC1)CC 2308,c1(CNC(C=C(C)C(F)F)=O)nc(CNC(=O)CCc2nccn2C)cs1 2309,c1(C(=O)NCC2CCCC(NC(C(C#C)(C)C)=O)C2)nccc(F)c1Cl 2310,c1(C(=O)NCC(CNC(C2(OC)CCOC2)=O)OC)cc(C2CC2)n(C)n1 2311,C1(CN(C)C(C2(NC(=O)CC34CCCC3C4)CC2(C)C)=O)COC(=O)N1 2312,C1(NC(c2c(C)nn[nH]2)=O)CCN(C(=O)Cc2cc(F)cc(Cl)c2)C(C2CC2)C1 2313,c1(C(=O)NC2CCC(CCNC(CCCC=C)=O)C2)c(C)cnc2ccccc12 2314,c1(C(=O)NCC(C)CNC(c2cc[nH]c2)=O)cc(OC(F)(F)F)ccc1F 2315,n1(C(C)C)ccc2cc(C(N3CCCC(NC(=O)C(O)CC(C)C)C3)=O)ccc12 2316,C1(CCCC(=O)NC(C(C)C)CNc2ccccc2)CCCC(=O)N1 2317,CC1CN(C)CC1C(=O)NCC1CC(NC(c2ccc(OCC(N)=O)cc2)=O)C1 2318,C1(C(N(C(C2CCCCC2)C)C)=O)COC2(CNC2)C1 2319,c1(C(=O)NCC2(C(C)NC(=O)CN3CC4CC4C3)CC2)ccc2[nH]c(=N)[nH]c2c1 2320,Cc1cc(C(=O)NCC2CC(NC(=O)C(C#N)C(C)C)C2)c2c(C)nn(C)c2n1 2321,C(C(O)CC(=O)NC(C)(C)CN(C)C)NC(COCCC(C)C)=O 2322,c1(N2C3CC(CN(C(C4C(C)OCC4)=O)C3)C2)ncc([N+](=O)[O-])cc1CO 2323,CC1=CCC(C(=O)NCC(C)(C)OCCNC(c2cnn(CCF)c2)=O)CC1 2324,C1(CC(=O)NCC2(F)CN(C(c3ccc(C(F)(F)F)cc3)=O)C2)CCCC1(F)F 2325,N1(C(Cc2c(C)nc[nH]2)=O)CCC(NC(=O)CCc2cncn2C)C12CCC2 2326,CCC(CCC(=O)NCCOCC1CCCC1)NC(=O)CS(=O)CC 2327,c1(NC(=O)NNC(=O)c2ccccc2F)ccc2cc[nH]c2n1 2328,c1(OC)ccc(C(=O)NCC(C2CCC2)NC(=O)C(C)CF)cc1 2329,C1(c2nnc(CC)o2)CCN(c2nncs2)CC1 2330,C1(C(=O)NC(CC#C)C(=O)NC(CO)C(O)CCC)CC2C(C1)C2(F)F 2331,CC1(C)C(C(=O)NCC(CO)NC(=O)C2=NOCC2)CC1(F)F 2332,N1(C(c2ccc(OCC)cc2)=O)CCC2(CC2)CC1C(N1CC2CC2C2CC12)=O 2333,Cc1noc(Cl)c1CC(N1CCCC(C2CCCCN2C(C2SCCS2)=O)C1)=O 2334,N1(C(C23CCCC2C3)=O)CC2(C1)CN(C(=O)CN1CCCC1)CC2CO 2335,c1(CC(CC)C)nc(-c2nn(C)cc2Br)n(-c2cnnn2C)n1 2336,Cc1ccc(C(N2CCCC2CN(C(=O)C(F)CC2CC2)C)=O)[nH]1 2337,Cc1ccn(CC(=O)NCc2ccsc2C(=O)NCCCO)n1 2338,C=CCC(C)C(=O)NC1CC(NC(=O)CCSc2nccn2C)C1 2339,c1(OC)cc(C(N2CC(CCCCNC(c3csc(Cl)n3)=O)C2)=O)cc(F)c1 2340,c1(C(=O)NCC(CC)NC(C2CCCC23CC3)=O)cnn(C(C)(C)C)c1Cl 2341,Cc1nn(C2CC2)cc1C(=O)NCCC1CCCN(C(C2CC2(Cl)Cl)=O)C1 2342,CC(C)(C)CCC(=O)N1CCCC(CC(=O)NCC2CN(C3CC3)C2)CC1 2343,C1(C(N2CCN(C)CC2COC2(C)CCC2)=O)CCCC2CCCCC12 2344,C(=O)(CCC1=CCCCC1)N(CCC(C)NC(=O)CC(C)O)C 2345,N1(C(C)C)CC(N2CCC(C)C(CO)C2)CCC1=O 2346,S(=O)(=O)(c1cccc2scnc12)NC1(C#N)CCN(Cc2n(C)ncc2Br)C1 2347,CON(CCC(=O)N(C(C)C(F)F)C)C(=O)C1(CSC)CC1 2348,c1(-c2ccc(NC(CCC(=O)N(CCC(O)CCO)C)=O)s2)cc2ncccn2n1 2349,N1CCN(C(=O)CC2CC2)C2CCCCC12.Cc1cc(-c2nn[nH]n2)cc(C)c1 2350,CC1CC(NC(=O)Cc2cc(F)ccc2O)CN(C(c2cc(Cl)c(Cl)[nH]2)=O)C1 2351,C12(C(=O)NCCCCNC(C(CC)OC)=O)CC(c3ccccc3)(C1)C2(F)F 2352,C1(CC(=O)NC(C)CNC(c2cccnc2)=O)CC(F)(F)C1(F)F 2353,C1(C(C)(C)NC(=O)C(n2ncnn2)=O)CCCCN1C(=O)CC1(O)CCC1 2354,C=CC(C)(CCOC)C(=O)NCc1cc(C(=O)N(CC(C)N(C)C)CC)co1 2355,C1(OC)CN(C)C(C)(C(N2CCCC(CNC(c3cnn[nH]3)=O)C2)=O)C1 2356,c1(SCC(=O)NCC(C)CNC(c2ccnnc2S)=O)ccc(Cl)c(C(F)F)c1 2357,Cc1cc(P(C)(C)=O)oc1C(N1CCC1CNC(=O)Cn1cc([N+](=O)[O-])cn1)=O 2358,N1(C(=O)NC23N(C(c4cnn(C(F)F)c4)=O)CC(C)(C2)C3)Cc2cncnc2C1 2359,C(=O)(C(C)(c1cccs1)N(C)C)N(CCN(C(=O)C(F)C1CCC1)C)C 2360,c1(N2CC3CN(C(c4ccc(C)nc4O)=O)C3C2)ncc2cn[nH]c2n1 2361,c1(C(=O)NC2C(C)N(C(c3csc(C(F)F)n3)=O)CC2)cccc2nn(C)cc12 2362,c1(NC(C(C=C)F)=O)ccccc1NC(=O)CCc1ccc(C)cc1 2363,C(C)(CO)(C(=O)N(C)CC1(CNC(=O)CCn2ccnc2C)CC1)NC(C)=O 2364,N1(C(C(C)n2cccn2)=O)CC2CN(C(=O)CN3CCCOC3=O)CC2(C)C1 2365,CC1CCN(C(c2cccc3c2CCC3)=O)CCN1C(c1ccn2c1CCC2)=O 2366,CC1=NOC(C)(C(=O)NC2CCN(C(=O)Cc3sc(S)nc3C)C2C)C1 2367,C1(C(=O)NC(C(=O)OCC)CO)CCC=CC1NC(=O)CC12CCC(CC1)C2 2368,Cc1ccccc1CN1CCC1CN(C(=O)C(C)(C)c1sccc1Cl)C(C)C 2369,C=C(C)C1CN(C(c2cc(C)c(=O)n(C)c2)=O)CCO1.C12CCN1C2 2370,c1(C(N2C3(CNC(c4nn(C)c(Cl)c4)=O)CCC3CC2)=O)cc(S(C)(=O)=O)cs1 2371,N1(C(C(C)=CC)=O)CCC(NC(c2nccc(OC)c2OC)=O)C(CC)C1 2372,Cc1cccc(N)c1C(N1CC(CCNC(c2ccnn2C(C)C)=O)C(C)C1)=O 2373,CC1(N=[N+]=[N-])CC(C(CN=[N+]=[N-])C2CNCC(O)CCC2)C1 2374,CCC(C)C(C)C(=O)NCCCCn1cc(-c2cn(C)nc2C(=O)OC)nn1 2375,c1(CSC)ccc(NC(c2sc(C(C)C)nc2C)=O)cc1 2376,CC1CN(C(=O)Cc2ccn(C)n2)CC1(C)CNC(=O)Cn1ccccc1=O 2377,c1(C(=O)OCC)cn(C)nc1NCCC1CCCN1C(=O)C(C)NS(=O)(=O)CC 2378,Cc1cc(C)c(C(=O)NCC2C=CCN2C(=O)CN2CCCCCC2)s1 2379,Cc1cc(C(=O)NCc2csc(C(=O)NCCCS(C)(=O)=O)c2)nc(O)c1 2380,c1(N2CCC(C(C)C)C2)nc(N2CCC(C)(c3ccccc3)C2)c2ncsc2n1 2381,C=CCCCC(C(=O)NCCNC(c1ccoc1)=O)NC(=O)Cc1csc(C)n1 2382,CS(=O)(=O)c1cc(C(=O)NCCc2ccn(CC(F)(F)F)n2)c(Cl)cn1 2383,CS(=O)(=O)C1(C(N2CC(CNC(c3cnns3)=O)C2)=O)CCNCC1 2384,N1(C(C=CCOC)=O)CCC(C2CC2)(CNc2ncnc3c2CCO3)C1 2385,C1(C(N2CCSCC(C)C2)=O)COC2(C1)CN(C(c1c[nH]c(C#N)c1)=O)C2 2386,N1(C(c2cc(C)c(Cl)s2)=O)CCN(C(=O)Cc2conc2C)C2CC12 2387,N1(C(C2C(C)OCC2)=O)CCC2OCCN(C(c3ns[nH]c3=O)=O)C2C1 2388,c1(C(N2CC(C3(NC(CCCCCC)=O)CC3)C2)=O)cc(Cl)c(F)cc1OC 2389,c1(OCCCCNC(C(=O)N(C2CCCC2(F)F)C)=O)c[nH]ccc1=N 2390,C1(OCC)CC2CN(C(=O)C(CCF)NC(c3cc(C(N)=O)co3)=O)CC12 2391,c1(N2CC(C=C)OCC2)cc(S(=O)(=O)NC2CC3(CCC3)C2)ccc1C#N 2392,c1(C(N2CC(c3cn(C4CC(O)C4)nn3)C(O)C2)=O)ccc2c(O)ncnc2c1 2393,c1(C(=O)NC(C(C)C)CNC(c2cc(Br)ccn2)=O)ccc([N+](=O)[O-])cn1 2394,C1(CC(=O)NCC(CC)NC(c2n[nH]c(C)c2C)=O)OCCCC1(C)C 2395,Cc1cc(Cl)cc(C)c1C(=O)O.C(=O)(CCOC1COC1)NCC=CC 2396,C12(CNC(c3n(CC=C)ccc3)=O)CN(C(=O)CN3CC4CC4C3)C(COC)(C1)C2 2397,C1(O)(C(C)NC(=O)CC2NC(=O)NC2=O)CCN(C(C2(C)CC2(F)Cl)=O)CC1 2398,C1(C(N(CCCN(CC)CC)C)=O)CN(C(=O)Cn2cccnc2=O)C(C)(C)C1 2399,N1(C(CNC(CN(S(C)(=O)=O)C)=O)C(F)F)CCN(C(C2(C)CC(C)C2)=O)CC1 2400,C(C(C)C(=O)NCCC(C)N(C(=O)CCCNC(=O)O)C)OC.OC 2401,C1(C(N(C2CN(C(C(F)=CC)=O)C2)CC)=O)CCC(C)N(C(=O)OC(C)(C)C)C1 2402,C1(CCC(=O)NC2CC(C(F)F)(NC(=O)COCCC=C(Cl)Cl)C2)CCCCO1 2403,C1(CC)C(NC(C2CCOC2)=O)CCCN1C(c1cnc(C2CC2)o1)=O 2404,c1(C(N2C(CNC(C3N(N=O)CCCC3)=O)CC3CC32)=O)ncnc2ccsc12 2405,N1(C(c2nc(CCC)sc2)=O)CCCCC1CCCNC(C1(C)COC1)=O 2406,CC(C)(C)CC(C)(C)C(=O)NCC1COCCN1C(=O)CCF 2407,Cn1ncc2ncnc(N3CCN(CC4CCCC4)CC3)c12 2408,N1(C(CCNS(CC)(=O)=O)=O)CCCC1CCCNC(=O)C(F)=CCCF 2409,Cn1c(O)nc2c(C(=O)NC3CCN(C(c4cnc(O)s4)=O)CC3F)cccc12 2410,c1(SC)cc(C(=O)NCC=CCNC(=O)CCC2(C)CC2(F)F)cc(Cl)c1 2411,c1(C(N(CC(C)CNC(=O)Cc2cccnc2Cl)C)=O)ccnc2c1CC(=O)N2 2412,n1(CC)nncc1C(=O)NCC(CNC(C1CC=CCC1)=O)CO 2413,N1(C(C(C(=C)C)(C)C)=O)CC(NC(=O)C(C)(C2CC2)OC)CC2(CCC2)C1 2414,c1(OC)ccc(Br)c(C)c1C(N1CC2(CCC(NC(=O)C=CC3CC3)C2)C1)=O 2415,C(=O)(C#CC1(C)CCCO1)NC(CC(C)NC(c1nnc(C(C)C)s1)=O)C 2416,C1(N(C(=O)CSC2CCOCC2)CCC2CC2)CCCCC1 2417,C1(C(N2CC(CNC(CCn3c(C)cc(C)n3)=O)OCC2)=O)CCC2CC2CC1 2418,O=S(=O)(c1ccc(NCCC2CCCO2)c(F)c1)N1CC2CC3CCCN3C2C1 2419,C1(CC(=O)NCCn2cc(CNC(c3scc(C)c3)=O)nn2)CCCC(C)C1 2420,N1(C(CS(N)(=O)=O)=O)CCC2CCN(C(=O)COCc3nc(C4CC4)no3)CC12 2421,C1(CN(C)C(c2cscc2C2CC2)=O)CCCN1C(c1ccnnc1)=O 2422,CCC(C(=O)N(CC(Cc1ccccc1)NC(C12CC(CO1)C2)=O)C)N(C)C 2423,C(=O)(C(F)C1=CCCCC1)NC(CCNC(c1ncc(CC)s1)=O)C 2424,Cn1cnc(C(=O)NC2C3CC2N(C(c2ccc(C#N)cc2)=O)C3)cc1=O 2425,Cn1ncc(C(=O)Nc2ccc(C(C)(C)C#N)cc2)c1F 2426,C1(C)(C(=O)OC)CCN(C(C2CCN(C(C3CC4CC4C3)=O)CC2)=O)C1 2427,C(=O)(CC1=NNC(=O)C1)N1CCC(NC(C(C(C)C)N2CCCCC2)=O)C(C)C1 2428,C1(NC(CN(C(C)C)C(C2CCC3CC2CO3)=O)=O)CN2CCC1CC2 2429,n1(CC(=O)NCC2N(C(C(=Cc3ccccn3)C)=O)CC=C2)nc(Cl)ccc1=O 2430,CCC(C(=O)N1CCCC(C(C)C(N2CCCC2C(=O)OC)=O)C1)C(C)(C)CC 2431,C(=O)(C1CNC(=O)c2ccnn21)N(C(CNC(c1c(C)nc(C)[nH]1)=O)C)C 2432,C1(C(C)NC(c2cccnn2)=O)CCCN(C(C2CCC(C(F)(F)F)CC2)=O)C1 2433,CC(CCCCO)NC(=O)C=CCN(C)C(c1cscc1Cl)=O 2434,C1(CNC(C23CC(CC(F)F)(C2)C3)=O)CCCCN1C(=O)Cn1cc(Cl)cn1 2435,C1(CC(N2CC(CNC(C3CC(SC)C3)=O)C2)=O)COC2CC1C2 2436,c1(C(N2CCC(CN(C(=O)CC(O)C3CCCC3)C)C2)=O)ccccc1CC#N 2437,c1(C(N2C(C(=O)NC3(CC#C)CC3)CC2C)=O)ccc(C)c(F)c1 2438,C1(C(F)(F)F)(C(=O)NC2(C)CN(C(CC3C(C)CCC3)=O)C2)CCCCO1 2439,c1(NC(N2C(C(=O)Nc3ncn(CC(C)C)n3)CC2)=O)cc(OC)c(F)cc1F 2440,c1(C(=O)NCC2(O)CC(NC(CCCC3C(C)C3)=O)C2)cccc2occc12 2441,C1(C2CC2)(C(=O)NCCC(C)NC(=O)CC2(N3CCCC3)COC2)CC1 2442,N1(C(c2nc(C)[nH]n2)=O)CC2CCN(C(c3cc(C4CC4)no3)=O)C2C1 2443,Cc1oc(CO)cc1C(=O)NCCC(O)CNC(=O)C(C)Sc1ccccc1 2444,C(CCC(=O)NC(C1CCOC1)CNC(c1cc(C(C)C)[nH]n1)=O)=C(C)C 2445,C12(C(N3C(C(C)NC(c4cc(OC)ncc4)=O)CCC3)=O)CC1COC2(C)C 2446,C(=O)(CC(O)CC(C)(C)C)N1CC(NC(CCCOC)=O)C2(C1)CC2 2447,c1(NC)c(C(N2CCCC(NC(C3(C)CCC(F)(F)C3)=O)C2C)=O)cccc1N 2448,C12(C(N3CCC(NC(C4CC5CCCC45)=O)C(F)C3)=O)CCC(F)(CC1)CC2 2449,Cc1nscc1C(=O)NCCCC1CCCN1C(=O)COCC1CCCCO1 2450,N1(C(C2(CC)CCN(C(=O)CC#N)C2)=O)CCOC(CO)CC1 2451,C1(CCSCC(=O)N(C2CCCCC2)CCC)CCN(C)C1 2452,N1(C(C2N(CC)CCCC2)=O)CCCC(C2CCN(C(=O)C(C)CCO)C2)C1 2453,c1(C(N2CCC(NC(CC=C(C)C)=O)C2C)=O)ccc2c(c1)CCC(C)(C)O2 2454,C1(NC(c2cc(C3CCC3)no2)=O)C2CN(C(c3cc(C(N)=O)co3)=O)CC12 2455,N1(C(CCCN(C)C)=O)CCC(CC(=O)NCCCOCCCO)CC1 2456,c1(COC)ccccc1C(=O)N(CC(C)N(C(=O)CC1OCCC1(C)C)C)C 2457,S(=O)(=O)(c1ccc(F)cc1)NC(C1(F)CCN(C(C(c2ccccc2)C)=O)C1)=O 2458,c1(C(=O)NCC(CNC(c2coc(Cl)c2)=O)OC)ccc2ccn(C)c2c1 2459,C(CCC(=O)NCCC(=C)CNC(=O)C(C)NC(=O)CC1C=CCC1)=CC 2460,C=C(Cl)CC(C(=O)N(C1CCCC1C)C)NC(C1CNC(=O)O1)=O 2461,c1(C(N2CCSCC(C)C2)C(=O)NCCCCCC)ncc(F)cc1F 2462,C1(N(C(=O)Cn2cccc2)C)CN(C(=O)Cc2cnns2)CC1(C)C 2463,C(CN=C(NCCc1ccccn1)NCC(C)(C)CO)c1ncc(C)nc1 2464,C12(C(=O)NCC=CCNC(c3cccc(O)c3F)=O)CCC(CC1)CC2 2465,C1(C(N2C(CCNC(c3cc(C)sn3)=O)CCCC2)=O)CN2CCN1CC2C 2466,CCC(CC(=O)NCC(C)(C)C#CC(=O)NC(C)Cn1cncn1)CC(C)C 2467,C1(CNC(C(CC)OCC)=O)CCCCCN1C(C1CC(N(C)C)C1)=O 2468,C1(NC(C(N2CCC(n3ccc4ccccc34)C2)C)=O)CC2(CCC2)C12CCC2 2469,c1(N(CC(=O)N(C)C)C)ccc(S(=O)(=O)N(C(CO)C2CCC2)CCO)c(Br)c1 2470,N1(C(CNC(C2(C#N)CC2)=O)=O)CCN(C(=O)CC2CC3(CC3)CO2)CC1 2471,c1(C(=O)NC(C(C)NC(=O)CN(S(C)(=O)=O)C)CO)cccc(C#N)c1Br 2472,C1(NC(c2c(C3C(C)C3)noc2)=O)CC(F)CN(C(=O)Cc2cn(C)nn2)C1 2473,c1(C(=O)NCCCCN(C(=O)Cn2cnnn2)C)sccc1Cl 2474,CC1CN(c2ccc(-c3cnccc3C(F)(F)F)cc2)CC(=O)N1 2475,N1(C(CCC)=O)CCCCC1CNC(C1(C)CC(C#N)C1)=O 2476,c1(CCC)c(C(N2CC(CNC(c3occc3C)=O)CC2C)=O)nnn1CC 2477,N1(C(CC(C)=C(C)C)=O)CCC(C)(CCNC(c2ccc(C3CC3)o2)=O)C1 2478,c1(C(N2CCOC(CCCN(C)C3CC3)C2)C(=O)NCC)ccc(C2CC2)cc1 2479,c1(CNC(c2ccc(NC(C3CCC(F)C3)=O)nc2)=O)cc(Cl)ccc1[N+](=O)[O-] 2480,c1(CC)c(C(=O)NCCC(C)(C)NC(=O)CCc2ncc(F)cn2)csc1C 2481,N1(C(c2nc(CC)oc2C)=O)CCN(C(C2CC(O)C2)=O)CC2CCCCC12 2482,C(=O)(C1=CCC2CCC1N2C(=O)C(C(C)C1CC1)OC)NC(C(=O)OC)C 2483,C1(O)(CCNC(c2cc(C)oc2)=O)CCN(C(C2CC(N(C)C)C2)=O)C1 2484,N1(C(c2c(CNC(C(C)(C3CC3)SC)=O)cco2)=O)CC=C(C(C)C)CC1 2485,N(C(=NCCn1cncn1)N1CCC(COC2CCCCC2)C1)CC(=C)C 2486,C(=O)(C1=NOC2(CCC2)C1)NC1C(NC(c2c(Cl)ccc(OC)c2F)=O)CC1 2487,c1(CC(=O)N(C)CCOCCCNC(c2cnc[nH]2)=O)ccccc1Br 2488,C1(NC(c2ccc(F)c(CO)c2)=O)COCCN(C(C2(CF)CC2(F)F)=O)C1 2489,c1(OCC(=O)N)cnn(C)c1CC1CC1.C1(C(=O)OC)(C(=O)N)CC(CF)C1 2490,Cc1cnc(C(N2CCC2CNC(=O)C(C)Cc2cccc(F)c2)=O)cn1 2491,c1(OCC(=O)OC(C2CS(=O)(=O)C2)C)cccc(Cl)c1Cl 2492,C1(C(=O)OC)CC(n2cc(C3(C(C)=O)CC3)nn2)CN1C(c1cccc(C)c1)=O 2493,c1(OCC)nn(C)c(Cc2nc(-c3ccn(C)n3)nn2C2CCC(C)C2)c1Cl 2494,c1(C(=O)NCc2cn(C(C)C)nc2)cccc2c1cnn2C 2495,c1(C(=O)NCC(CCCC)NC(=O)C(CC)CCC)cc2cccnc2cn1 2496,c1(C(=O)NC(CC)(C)CNC(=O)CC2CCN(C)C2=O)nccc2c1CNC2=O 2497,C1(C(=O)NCc2cc(Cl)no2)(NC(C(C(C)C)F)=O)CCc2cc(Br)ccc2C1 2498,O=C1CC(NC(=O)CC2CCN(C(C3(O)CCC3)=O)CC2)CCN1 2499,C(=O)(C(F)(F)CC1CN(C(=O)NCC2(n3cccn3)CC2)C1)OC 2500,CCCCC(CCCC)NC(=O)CC(C)(C)N(C(=O)Cc1cccc(C#N)c1)C 2501,N1(C(CC2(COC)CC2)=O)Cc2ccccc2OC2(C1)CN(C(C1CC1(Cl)Cl)=O)C2 2502,C(=O)(C1=NNC(=O)CC1)NCCCC(C)NC(C1N(C(C)=O)CSC1)=O 2503,c1(C(=O)NC(CC)CNC(=O)C(C)=CC2CC2)ccc2nnnn2c1 2504,c1(OC)ncc(C(=O)NCC2(C)CN(C(=O)C(C)N(C)C)CCO2)nc1C 2505,N1(C(CCC=C(C)C)=O)CC2CC1(C(=O)NC1(C)CS(=O)(=O)C1)C2 2506,CC1CN2CCN1C(C(N1CCCCC1CNC(C1(C)COC(=O)C1)=O)=O)C2 2507,C1(C(=O)NCCCCCCNC(CCCC)=O)C2CCC(C2)S1(=O)=O 2508,C(CC(=O)NCC1(NC(=O)C=CCC2CC2)CC1)OCC#C 2509,Cc1coc(C(N2CCC(N3CCC(NC(=O)C(=O)NC(C)C)CC3)C2)=O)c1C 2510,Cc1c(Cl)ccnc1NC(C1CC(F)CN(C(=O)C=CC(=O)N(C)C)C1)=O 2511,CCC(CC(=O)NCCC1CN(CCc2cnn(C)c2)CCS1(=O)=O)C(C)C 2512,N1(C2CN(C(=O)C(COC)OC)C2)CC(NC(c2c[nH]nc2CC)=O)CC1=O.CC 2513,C#CC1CN(C(=O)CN(CC(C)C)C(C2CN(C3CCC3)C2)=O)CCO1 2514,C#CCC(CC(=O)NC(C)CCNC(=O)CN1CCC(C)CC1)c1ccccc1 2515,N1(C(C2CCC(C)O2)=O)CC2C(N(C)C(c3cncn3C)=O)C2C1 2516,CC(CC(C)(C)C)C(=O)N(C1CCN(C(C2CCN(C)C(C)C2)=O)C1)CC1CC1 2517,CCC(CCOC)C(=O)NCC1(F)CN(C(C2Cc3nccn3C2)=O)C1 2518,c1(C2C(CN(C)C(C3(CC(F)(F)F)CC3)=O)C2)ccc(Br)nc1 2519,C(c1cc(C)no1)=CC(=O)NC(CNC(CNS(CC)(=O)=O)=O)(C)C 2520,N1(C(C2C(C)(C)N(C(=O)CC3(O)CCCOC3)CC2)=O)CC2(CCOC2=O)C1 2521,C1(C(=O)NCC(C)CNC(C2(C)CC(C#N)C2)=O)CC(c2cccc(F)c2)=NO1 2522,c1(C(N2CC(N(C(C(C=C)O)=O)C)C(O)C2)=O)nn(C)cc1S(N)(=O)=O 2523,C(=O)(C(C(=O)NC1(CNC(C2CC2C)=O)CCCCC1)C1CC1)OCC 2524,C1(OC)(CNC(c2cc(C(F)F)ccn2)=O)CCN(C(=O)C(C)(F)F)C1 2525,C1(CNC(C2(CC#C)CCC2)=O)CN(C(c2cnc(COC)[nH]2)=O)CC1(F)F 2526,CCCC(C)C(=O)N1CCC(CCC2CCCN2C(C(=O)C(F)F)=O)CC1 2527,C12(NC(C=COCC)=O)CCCC1N(C(c1cncs1)=O)CC2 2528,c1(CC)cnc(O)c(C(N2CC(NC(C3(CN(C)C)CC3)=O)C(C)C2)=O)c1 2529,N1(C(c2cnn(C)c2N)=O)CCCC(CCNC(=O)C(O)CC(F)F)CC1 2530,N1(C(C)C)CCCC1CC(=O)N(C(C)CCNC(=O)CCCN(C)C)C 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2549,CN1CCC(C(=O)N(C)CC2CCCN2C(=O)CNC(C2CCC2)=O)CC1=O 2550,c1(CN2CCC(NC(c3ccc(CN(C)C)cc3)=O)CC2)ccc(F)c(CO)c1 2551,C1(CSCC(=O)NCCCNC(Cc2nc(C)oc2)=O)CCc2ccccc2O1 2552,C(=O)(CC1OCc2ncccc21)NCCCN(C(C(CCSC)O)=O)C(C)C 2553,c1(C(C)(C)C)csc(C#N)c1.c1(C)ccc(C(=O)NCCCOCCCNC=O)s1 2554,N1(C(C2(F)CCN(C(c3ccnc(F)c3Cl)=O)C2)=O)CCN2CCCC2C1 2555,C(C(C)C(=O)NCCC(Cc1ccccc1)NC(c1nscc1N)=O)SC 2556,CC(C)C(C)C(CNC(C1CN(C)C1)=O)NC(c1cn(C)nc1C(F)F)=O 2557,N1(C(c2scc(C)c2)=O)CCCCC2(CCN(N3CCCCC3)C2)C1.CC=O 2558,CCC(C)CCCC(=O)N1CC2(CC2)CC1C(N1CCC2(CC1)CC2)=O 2559,C(CCCC(C)NC(C1(c2ccccc2)CC1(C)C)=O)NC(CCSC)=O 2560,C1(C(=O)NC(CSC)C)CC2CC1CN(C(c1ccc(O)cc1F)=O)C2 2561,C=Cn1nccc1C(=O)NC1CN(C(=O)CC2CC3(COC3)C2)C1 2562,C(=O)(CC(O)C(Cl)(Cl)Cl)NCCCCNC(c1c(C)cc(N)cc1)=O 2563,C1(CC#C)(C(N2CC(CC=C)(NC(=O)C(O)Cc3cnc[nH]3)C2)=O)CCCCO1 2564,N1(C(C2(C(=O)NCCOCCOCCOC)CC2)=O)CCOC(C)(C)CC1 2565,C1(C(N2CCC(C)(F)C2)=O)N(C(=O)Cc2csnn2)CC12CCCC2 2566,c1(CC)n[nH]c(CC)c1CC(=O)NC12CC(CNC(=O)C(C)(C)C)(C1)C2 2567,C(=O)(C(C)(C)CCCCC)N(CC(CN(C(Cc1cccc(C#C)c1)=O)C)O)C 2568,C#Cc1cn(C)nc1C(=O)NCC(C1CCOC1)NC(=O)C(C)(C)C#N 2569,c1(NCC2N(C(c3c(C)ccc(F)c3)=O)CCC2)ncnc2occc12 2570,C1(CNC(C2(C(CC)(F)F)CC2)=O)(NC(=O)Cc2ncccc2C)CCOCC1 2571,N1(C(C(CC)CO)=O)CCC(O)(C2(NC(=O)CSc3cnn(C)c3)CC2)CC1 2572,C1(CNC(C2(CC)CC2)=O)CN(C(=O)Cc2cn3ccccc3n2)CCC1(C)C 2573,c1(N(C(CCC2CCN(C(CCCOCCOC)=O)C2)=O)CC)c(C)n[nH]c1C 2574,C(=O)(CC(C)C(C)C)NCC(CC(C)C)NC(c1scnc1C1CCCC1)=O 2575,C1(CC(=O)NC2CCC(N(C)C(c3cc(CO)[nH]n3)=O)C2)CC2CCC1CC2 2576,CN1CCN(C(=O)C=Cc2ccc[nH]2)C(C(=O)N(C2(C)CC2)C)C1 2577,CC1(C)OCC2CC12CNC(=O)CC1CCC(NC(=O)Cc2ncccc2F)C1 2578,C1(NC(c2ccccc2F)C)CCS(=O)(=O)C2(C1)CC(CN)C2 2579,C(CC=C)(CC(=O)N(CC(C1CCCC1)O)C)NC(C(C=C=C)C)=O 2580,C(C(=O)O)(C(C)OCC(C)C)NC(C1CCN(CCOC)C1)=O 2581,Cc1c(C(=O)NC2CCC23CN(C(C2COC(=O)C2)=O)C3)oc2ccc(F)cc12 2582,Cc1c(NC(=O)CN2CCN(C(c3ccccc3O)=O)CC2)cnn1C 2583,C1(NC(C2(C)CC3(CC3)C2)=O)CCCC(C(N2CCC(F)CC2)=O)CC1 2584,C1(C(=O)NC2(CC=C)CC2)CN(C(c2c(C)cccc2C)=O)CCC1(C)C 2585,c1(NCC(N(C)C(c2ncn3ccccc23)=O)C2CC2)ncnc(Cl)c1C#N 2586,C=C(C)CCCC(=O)N1CC(NC(c2c[nH]cc(Cl)c2=O)=O)C(C)C1 2587,CCC1=C(C(=O)N(C(CNC(=O)Cn2ncc(O)nc2=O)C2CC2)C)CCCO1 2588,c1(C(N(CCN(C(C)C)C(C2(C)CCCCO2)=O)C)=O)ccnc(CO)c1 2589,c1(-c2ccc(OCCO)cc2)ccc2cc(C(N3C(C)COCC3)=O)cn2c1 2590,S(=O)(=O)(C1CN(C(=O)Nc2nnc(C(C)(C)C(F)F)o2)C1)Cc1ccccc1 2591,N1(C(Cn2c(C)ccn2)=O)CCC2CN(C(c3sccc3F)=O)CC12 2592,c1(OC)ccc(F)cc1CC(=O)NC1(CNC(c2ncsc2C2CC2)=O)CCC1 2593,c1(N(CCNC(COCCC=C)=O)C2CC2)nc(C)nc(Cl)c1C 2594,C1(c2nc(-c3c(OCC)nccc3)nn2-c2cccc(Cl)c2)CC2CCCCC12 2595,c1(C(N2C3CC(NC(C4CC4F)=O)C2CC3)=O)cc(Br)cc(Cl)c1O 2596,C=CCC(C(=O)N1CC(C(=O)N(C2CC3CC3C2)C)C1)OC 2597,N1(C(CC(COC)C)=O)CCC(F)(CNC(C2(C)CCC(C)C2)=O)CC1 2598,C1(=CCC)CN(C(=O)C(C)NC(=O)C(C)SC)C1 2599,C1(NC(CCC(=O)OC)=O)CCN(C(C2CCCC2OC)=O)CC1C 2600,C1(CN(C(=O)CCn2ccccc2=O)C)CN(C(c2ccsc2)=O)CC12CC2 2601,Cn1ccc2c(C(=O)NC3CCCCN(C(C4CC4C#N)=O)C3)[nH]cc2c1=O 2602,C1(CC)(NC(c2ccc(N(C)C)nn2)=O)CCCN(C(C2CCC(=O)N2)=O)C1 2603,C1(OC)C(F)CCC(C(N2C3CCC2COC3)=O)N1C(=O)OC(C)(C)C 2604,N1(C(c2cc(CNC(C(CC)(C)CC)=O)on2)=O)CC(C)CC(C)(C)C1 2605,C1(C(=O)NCCCN(C(=O)CN(C)C(C)C)C(C)C)(COC)CC1 2606,N1CCC(O)(c2cccc(C(F)(F)F)c2)CC1.O=C1CC(c2ccccc2)CN1CCCCl 2607,c1(COCC(=O)NC(c2ccccc2)C2(c3cccs3)C(C)C2)sccc1C#N 2608,C1(C)(CC)C=C(C(=O)N2CC(CNC(=O)CSc3nncn3C)CC2(C)C)C1 2609,N1(C(CCC)=O)CCC(C(=O)NCC2CCOCC2)=C(F)C1 2610,C1(CC(C)NC(CC(C)SC)=O)CCN(C(=O)C(C)C(C)C)CC1 2611,CC(=O)CCCCC(=O)NCC(C)(C)OCC(=O)NC(C1CC=CCC1)CO 2612,N1(C(c2ncn(C)n2)=O)CC(O)CC1CNC(c1cc(C2CC2)n(C)n1)=O 2613,C1(CNC(C2CC(C)=C(C)CC2)=O)COC(C)(C)CN1C(c1cn(CCO)nn1)=O 2614,C1(C)(C(=O)NCC2CN(C(C(C)(C)CF)=O)CC23CC3)CCc2ccccc2C1 2615,c1(C(=O)NC2(C(N(CCC#C)CCOC)=O)CC2C)ncc(F)cc1F 2616,C1(OC(c2ccc(-n3cncn3)cc2Cl)=O)CCOC2(CCCC2)C1 2617,C12(NC(c3nc(C(C)=O)sc3)=O)CC1CN(C(C1CCC(C)(C)C1)=O)C2 2618,c1(C(N2CC(C(C(=O)NCc3c(CC)con3)OC)C2)=O)ncncc1C 2619,C(C)(CO)(C(=O)N1CC(CCNC(c2cnn(C)c2Cl)=O)(OC)C1)OC 2620,c1(C(=O)NCC(CC)NC(=O)C(C)C(C)CC)cc(C(=O)OC)ccc1C 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2655,C(=O)(C1=NNC(=O)C1)N1CCC(CNC(=O)C=Cc2ccccn2)(CO)C1 2656,c1(NC)cnc(C(N2CCC(C)(CNC(c3ncccc3C3CC3)=O)C2)=O)nc1 2657,C1(C(=O)NC(C(=O)NCc2n(C)cnn2)C2CCCO2)CC(=O)CCO1 2658,CC1(C)CCN(C(=O)CCC2CCOC2)C1C(N1CCOCC1C1CC1)=O 2659,C1(F)(C(=O)NCC2C=CC(NC(C3CCN(c4nncs4)C3)=O)C2)CCCCC1 2660,N1(C(c2cccc(C(=O)NC)c2)=O)CCC(NC(=O)Cc2cnn(C)c2)C(O)C1 2661,c1(C(=O)NC2CCCN(C(C=C(C)C(C)(C)C)=O)CC2)c[nH]c2c(F)cccc12 2662,C1(C(=O)NC2CC3CN(C(c4ccc(C#N)cn4)=O)C2C3)CCCCC1C1CC1 2663,N1(c2cc(NCC3CSC3)nc(C)n2)CCC(C)C(C)(C)C1 2664,C1(NC(NCC(C)COC(F)F)=NCCN2CCC2)CCc2ccccc2C1 2665,c1(OCCNC(=O)NC2C(=C)COC2)ccccc1F 2666,c1(C(=O)NC2CCN(C(CCCCCC)=O)C2C)cc(OC)cc(Cl)c1F 2667,C1(C(N(c2cnn(C)c2)C)=O)CCCCCCN1C(c1cnn(C)c1Cl)=O 2668,c1(C(=O)NC2CC(F)(CNC(C(C)OC)=O)C2)n[nH]c2c1C(=O)CCC2 2669,c1(N(CCOC(COC)=O)C(C)C)ccc(CC(=O)OC)cc1 2670,C1(NC(c2n(C(C)C)ncc2)=O)CCCC(NC(=O)C(C)(C)c2cnc[nH]2)C1 2671,C(C)(CO)(C(F)F)NC(C(C1CN(C(=O)Cc2ncoc2C)C1)OC)=O 2672,C(=O)(CCC(=O)NC(c1ccccc1)CNC(=O)CSCC1CCCCO1)NC 2673,CCC(C)(O)C(=O)NCC1(C)CC(NC(=O)Cn2nccn2)C1 2674,C1(OC(C)=O)C(C(C)C)CN1C(=O)C(c1ccoc1)NC(=O)CC1OCCC1C 2675,c1(COC)ccsc1C(=O)N(C(C)CCNC(c1ncn(C(C)(C)C)n1)=O)C 2676,C1(NC(C2CCC(C)CN2C(c2ncsc2NC)=O)=O)CCn2nnnc2C1 2677,CCCC(O)CC(=O)N(C1CCCC1)CCCNC(=O)CN(CC(C)(C)C)C 2678,N1(C(C2(CNC(C(C)C3CCC3)=O)CC23CCC3)=O)CCC2(CCCCC2)C1 2679,Cc1cc2[nH]c(C(=O)NCC3CC3NC(c3ccc(Br)c(N)n3)=O)cc2o1 2680,C1(NC(COCCC=C)=O)CCCCC12CCCN(C(=O)Cc1ccc(C)o1)C2 2681,C(CC(C(C)(C)C)NC(=O)Cc1c[nH]nc1O)N(C(=O)C=C(Cl)Cl)C 2682,C=C(C)CCC(C)NC(=O)C=CC(C)(C)NC(c1ccn(C)n1)=O 2683,c1(N(CC(=O)OCC)CC2CCCCC2)ncc(C(F)(F)F)n1C 2684,C(CN=c1nc2ncn(C)c2c(NCCC(C(C)CC)OC)[nH]1)OCCOCC 2685,C1(CC)CN(C(=O)C(C)(C)F)CCN1Cc1cc(C(F)(F)F)cc(Cl)c1 2686,c1(C(=O)NCC2(NC(C(C=C=C)C)=O)CC(F)(F)C2)ccc2nonc2c1 2687,C1(CNC(=O)C=C2CCC2)CCCCC1NC(=O)C(=O)NC1CC1 2688,C12(C(=O)NCC3OCC(CNC(c4cnc(SC)[nH]4)=O)C3)CCC(CC1O)C2 2689,C(C(O)CNC(=O)CC1CCSC1)NC(C=C)=O 2690,c1(C(N2CC(NC(C=C(C)C(F)F)=O)C(F)CC2)=O)cc(S(N)(=O)=O)co1 2691,C1(CNC(c2cn(C)nn2)=O)CN(C(C2C3CCCC23)=O)C2CC12 2692,N1(C(c2cc(C)sn2)=O)CCOCC(NC(c2cnc(C)c(C(F)(F)F)c2)=O)C1 2693,N1(C(C(C)CC2CCC2)=O)CCN(C(N2CCN(C(=O)C3=CCC3)CC2)=O)CC1 2694,C(C)(C(C(=O)N1CC(O)CC1CC(=O)N(C)CC1CCCCC1)N(C)C)OC 2695,C1(F)(CNC(c2ccc(CC#N)nc2)=O)CCC(CNC(c2ccsc2)=O)CC1 2696,C1(N(C)C(c2ccccc2C(N2C(C)C(C)(C)C2)=O)=O)(CO)CC2CCCC12 2697,c1(C(=O)NC2CN(C(COCCC)=O)C(C)(C)C2)nn(C)c2c1CCCC2 2698,C(C(C)(CC)C(=O)NCCCS(C)=O)NC(C(c1ccc(C)o1)C)=O 2699,Nc1cc(Cl)c(Cl)cc1C(N1CCN(C(c2ccoc2Br)=O)C2CC12)=O 2700,O=C(C1=CCCOCC1)NCC1CC2CCCC2N1C(c1cc(C2CC2)on1)=O 2701,C12(CNC(c3c(CC)nc[nH]3)=O)CCCC(CN1C(=O)C1=NOC(C)C1)C2 2702,C1(C(=O)NCCCN(C)C(C2(c3cccs3)CCCC2)=O)CCN(S(C)(=O)=O)C1 2703,C1(OC)CN(C(=O)Cc2c[nH]ccc2=O)CC1NC(=O)CC1(OC)CCCCC1 2704,Cc1cc(CNC(C2CC3CCC2C3)=O)oc1C(=O)NCC1(n2nccn2)CC1 2705,c1(OCC)cccc(C(N2CC(O)(CNC(C3CCC3C(F)(F)F)=O)C2)=O)c1N 2706,C(CC)(C(=O)N(CCCNC(c1nsnc1O)=O)CC1CCCC1)=CC 2707,C1(O)(CNC(c2nc(C)oc2)=O)CCCN(C(=O)CN2CCOCC2=O)C1 2708,C1(NC(C2C(OCC)C2)=O)CN(C(=O)CCc2cccnc2C)CCC1CO 2709,c1(C(N(CCCNC(c2conc2C(C)C)=O)CC)=O)cc(O)cnc1Cl 2710,C1(NC(=O)C=Cc2ccoc2)CC2(NC(=O)C(=C3CCCCC3)F)COC1C2 2711,C1(NC(C(CC)OCC)=O)CCN(C(=O)C2=COCCO2)CC12CCC2 2712,CCCC(C)C(=O)NCC1(C(N)=O)CN(C(=O)CC2(C#N)CCC2)C1 2713,c1(C(=O)NC(C2OCCN(C(CC=CC=C)=O)C2)C)cc2cncn2c(O)n1 2714,N1(C(C(c2cccc(C)c2)C)=O)CC2CC(NC(c3c(C)n[nH]c3C)=O)C2C1 2715,C(=O)(CC(F)(F)C(F)(F)F)NCCC(C)NC(C1CC1(Cl)Cl)=O 2716,C1(C(N(C)CCF)=O)CCN(C(C2CC3CCC2CC3)=O)C(C)(C)C1 2717,c1(NC(CSCc2nnc(C(C)=O)s2)=O)cccc(N(C2CC3C=CC2C3)C)c1 2718,CCCC(C(O)C(=O)N(C)CC1CC1(C)C)NC(c1ncc(C)cc1C)=O 2719,C1(CC(=O)NC2CC(N(C(=O)CC3COCCO3)C)C2)COCC1(C)C 2720,CC(C(=O)NCC1(C)CCCN1C(c1n[nH]cc1Br)=O)P(C)(C)=O 2721,C1(C)(CNC(=O)NCC2(NC)CCCC2)COCC(C)(C)O1 2722,C1(C(N2CCC(O)(CN(C(C3(CC)CC(C)(C)C3)=O)C)C2)=O)CC2C=CC1CC2 2723,C1(CNC(CSC(C)C)=O)CC(O)CN1C(=O)C(Cc1ccc(F)cc1)N(C)C 2724,CCCC(C)(O)C(=O)N1CCC(NC(c2cccc(CSC)c2)=O)C1 2725,C1(C(N2C(CN(C(CCOCCOC)=O)C)CCC2)=O)CC2(CC(=O)N2)C1 2726,Cc1nc(C)c(C(=O)NCC(O)CNC(c2ccsc2)=O)o1 2727,N1(C(C=CC)=O)CCCC(C)(NC(=O)C(C)Oc2ccccc2C#N)C1.C1CO1 2728,C1(NC(CCS(N)(=O)=O)=O)CC12CCN(C(c1cc3occc3[nH]1)=O)CC2 2729,C1(CN(C)C(c2cn(C3CC3)cn2)=O)CCCN(C(c2cnc(Cl)n2C)=O)C1 2730,c1(C(=O)NCC(CNC(c2n(CC)ncc2)=O)O)cc(C(F)F)cc(C)c1 2731,Cc1c(C(=O)N(CCNC(C2CC23CCC3)=O)C2CC2)cncc1Br 2732,C(=O)(N1OC2C=CC1CC2)c1nc(CNC(CC2N(C)CCC2)=O)oc1 2733,Cc1ncnc(C)c1OCC(=O)NCCC(C)CCNC(c1ccc(O)nn1)=O 2734,c1(CN(C(c2cnc(C(=O)OC)s2)C(=O)NCCC2(C)CC2)C)ccc(C)cn1 2735,C1(C(=O)NCCc2ccsc2)CCCCCN1C(C1CC(O)C1)=O 2736,C(N=c1[nH]c(=NC2CCC2OC)[nH]c2c(F)cc(F)cc12)C1C(CC)C1 2737,N1(C(CC(C)OC)=O)CCC(C2CCCN(CCc3ccnn3C)C2)CC1 2738,C1(NC(CSCC(C)C)=O)CN(C(C2(C#N)CCCC2)=O)CC(C)(C)C1 2739,S(=O)(=O)(c1ccc(F)cc1C)N(c1cc(SC)nc(C)n1)C1CCNCC1O 2740,C(=O)(N(OC)C1CCC1)C1N(C(c2ccc(CC)cc2)=O)C2C(C1)C2 2741,N1(C(c2c(C)n(C)cn2)=O)CCCOC(CCNC(C2Cc3nccn3C2)=O)C1 2742,N1(C(C(C)OCCC=C)=O)CCCCC1CNC(=O)CC(O)C1CCCC1 2743,CC(C)CC(F)(F)C(=O)NCC(C1CCCC1)NC(c1ccoc1Cl)=O 2744,C(=O)(CC(C)(C)C)NC(C)C=CC(=O)NC1CC1c1ccn(C)n1 2745,C1(OC)CC(CNC(=O)Cc2ncoc2C)N(C(=O)Cc2ccc(Br)cn2)C1 2746,N1(C(c2c(CC)cns2)=O)CCCCC1CCC(=O)N(CCO)C(C)C 2747,c1(C(=O)NC2CC2CNC(C2(F)CCC2)=O)c(Br)ccc2ccccc12 2748,CC1CCc2sc(C(=O)NCC(C)(O)CNC(=O)Cn3ncn(C)c3=O)cc2C1 2749,C(=O)(C1=CCSC1)NC(C1CCN(C(=O)C(O)C2CCC2)C1)(C)C 2750,S(=O)(=O)(c1cnc(-c2cccc(-c3c(C)ccc(Cl)c3)c2)s1)NC(=O)C(C)S 2751,C1(CC(=O)NCC2CC(OC)CN2C(C2CC2C)=O)CC2(CCCC2)CO1 2752,c1(C(C)NC(C2CSCCN2C(c2nccn2C)=O)=O)cc(Cl)ccc1O 2753,c1(C(N2CC(OCCNC(CN3CCC(C)CC3)=O)C2)=O)ccc(F)nc1F 2754,c1(OCOC)cc(-c2ncsc2C(=O)NCCc2cccs2)c(F)cn1 2755,Cc1nc(C(=O)NCC(F)CNC(c2ncoc2C2CCC2)=O)c2ccccn12 2756,C(=O)(C(C)C(C)NC(=O)CC1(C#N)CC1)N(CCc1nc(C)on1)C 2757,C#CCCCCCCC(=O)N1CCC(C(C)C(N2CC=CC2CF)=O)CC1 2758,C1(N(C)C)(CNCCC(=O)NC(CNC(c2ccsc2)=O)C2CC2)CCCC1 2759,c1(N2CC(O)(C(C)NC(CC(C(C)C)O)=O)C2)ccc(S(=O)(=O)NC2CC2)cn1 2760,N1(C(c2c(C)cc(CO)o2)=O)CCN(C(c2ccon2)=O)C2CCCCC12 2761,Cc1cc(Cl)ccc1C(=O)NC1COCCN(C(=O)CC2(O)CCCOC2)C1 2762,Cc1ccc2c(N(CC(C)C)C)nc(=NCCCOCCNCC(C)C)[nH]c2c1 2763,Cc1c(C(=O)NC(C)(C)CNC(=O)C(F)CC2CCCC2)cccc1N 2764,c1(C(N(CC(c2ccccc2)O)C)=O)ccc(=O)n(-c2ccccc2F)c1 2765,c1(C(=O)NCC(CC)NC(c2cnnn2C2CC2)=O)ccncc1Cl 2766,Cc1coc(C)c1C(=O)Nc1ccccc1.N12CC3C(C3C1)c1cn(nn1)CC2=O 2767,N#Cc1ncc(CC(N2CCC(Cn3cc(-c4ccncc4)nn3)C2)=O)s1 2768,Cc1nn(C(C)(C)C)cc1C(=O)NC1CCN(c2cccnc2)C1 2769,CCC(CC)C(=O)NCC(=O)NCCC(C)(C)CNC(C)=O.C12CCN(C1)C2=O 2770,Cc1c(O)ccc(C(N2CCCCC2CNC(C2CC23CCC3)=O)=O)c1C 2771,C(=O)(C(F)C1CC(CCN2CCCC2)C1)N(CC(=O)NC(=O)COC(C)(C)C)C 2772,c1(C(N2CC(CC(C)NC(C3CC4CC4C3)=O)C2)=O)scc(Cl)c1Cl 2773,Cc1ccc(C=CC(=O)NCC2CCC(C)N(C(=O)C=CCCC(C)C)C2)nc1 2774,C(CC)(CCCC(=O)N1CCCC(C#N)C1)NC(CCCCCC)=O 2775,C12(C(=O)NCCCN(C(=O)CC(=O)Nc3n[nH]c(O)n3)CC)CC(CC(F)F)(C1)C2 2776,N1(C(c2c(NCC)scn2)=O)CCCC2(CCCN2C(=O)CN2CC=CC2)C1 2777,c1(C(c2nnnn2-c2ccccc2Br)NC2CC(=C)C2)sc(C)cc1Br 2778,c1(C(N2CC3CCN(C(C4N(C)CCC4)=O)C3C2)=O)ccc(Br)c2cn[nH]c12 2779,C(=O)(C1=CN=C2N=CNN2C1)NC1(C)CCCN(C(C2(F)CC3(CCC3)C2)=O)C1 2780,c1(OC)ccc(Br)cc1CNC1C2CN(C(c3ccncc3O)=O)CC12 2781,NC(=O)CCC(=O)NCc1nc(C2CCCN(C(c3cnsn3)=O)C2)n[nH]1 2782,c1(C(=O)NC(C2(O)CN(C(=O)C(O)C(F)F)C2)C)ccc(C(=O)OC(C)(C)C)cc1 2783,c1(C(=O)NCC(CNC(C(CC=CC)C)=O)(C)C)c(C)ncnc1O 2784,C1(CC(=O)NC(C2N(CC(=O)N)CCC2)C2CC2)CCCC12CC2.C1(C)CC1 2785,N1(C(C2CCN(C(=O)NC)CC2)=O)CC2CCC2(NC(c2cn(CC)cn2)=O)C1 2786,C1(CCCNC(CCCC)=O)CCN(C(=O)C(C)(C)Oc2ccc(Cl)cc2)CC1 2787,c1(C(=O)OC)cc(NC(=O)C(C)n2ccnc2)cc(Cl)c1 2788,c1(C(=O)NC2C(CNC(CCCCOC)=O)CC2)nc(OC)cc(OC)n1 2789,c1(C(N(CC(C)NC(=O)CN2CC=CC2)C)=O)cn2c(n1)CCC2 2790,c1(C(C(=O)NC(C(C)NC(=O)CCc2cccn2C)C)O)cc(F)cc(F)c1 2791,C1(C(=O)NCCc2c(CNC(C3(CC)CCOC3)=O)nco2)CN=C2N=CNN2C1 2792,C1(NC(C(CC)OC)=O)CCN(Cc2nnnn2CCC2CCCCC2)CC1O 2793,C#CC1(C(=O)NCC2CC(C)(C)CO2)CCN(C(c2ccnc(CO)c2)=O)CC1 2794,C12(NC(C3N(CC)CCOC3)=O)CCOC(CNC(=O)C(C3CC3)SC)(C1)C2 2795,CC(CN(C(=O)C=CC1CC1)C1CC1)(CO)NC(=O)COCC1CCOC1 2796,C1(NC(CNC(CC)=O)=O)CCC2(CC1)CN(C(=O)C=CC)CCO2.[nH]1cncn1 2797,N1(C(=O)CSc2nnc(S)s2)CC(C2CN(C(c3ncc(Cl)cc3F)=O)C2)C1 2798,Cn1cnc(C(C(=O)NC2(C)CC2)N(C)CC2CCOC2)n1 2799,C(C)(C(O)C(=O)N(CC(C)(C)CNC(C1CCC=CCC1)=O)C)OC 2800,C1(CC(N2CC(NC(C(C)(C)OC)=O)CC2(C)C)=O)CCc2ccccc2C1=O 2801,c1(OC(C)C(=O)NCC2(F)CCC(NC(C3(C(N)=O)CC3)=O)C2)cccc(F)c1 2802,N1(C(CC(COC)(C)O)=O)CCC2CN(C(c3cn4nc(C)sc4n3)=O)CC12 2803,c1(NC(C2(C(N)=O)CCC2)=O)cnccc1N1CCCCC1 2804,N1(C(=O)NCc2cc(C(F)(F)F)no2)CCC(c2nn[nH]n2)C12CC2 2805,c1(OC(CC)C)ccc(C(N2CCCC(CCNC(=O)CC(F)(F)F)C2)=O)cc1 2806,N1(C(c2ncc3ccccn23)=O)CCOC2CN(C(C3(CCF)CC3)=O)CC12 2807,CCCCC(C)C(=O)N(C1(C(=O)NC2(COC)CC=CC2)CC1)C 2808,C12(CNC(c3c(C)nn(C)c3)=O)CC(CCO1)N(C(=O)COC(C)(C)C)C2 2809,C1(F)(C(=O)NCC2N(C(CC(=O)NC)=O)CCC2C)C(C)(C)C1(C)C 2810,C(CCC(C)(C)NC(C1CCCN1CC(F)(F)F)=O)NC(C1(SC)CC1)=O 2811,CC1(NC(C23CC(CN2C(c2cn(C4CC4)nn2)=O)C3)=O)CC2CCC1C2 2812,c1(C(N2CC3CCN(C(c4[nH]cc(C)c4)=O)CC32)=O)ccc2c(c1)COCCN2 2813,C(=O)(C(F)CCC(C)(C)C)NC(C1CCN1C(c1cncc2c1CCC2)=O)C 2814,CC(C)(CCNC(=O)Cn1ccnc1)C(=O)NCC1CSCCO1 2815,CCC(C(=O)N(C)C)NC(C1CC(O)(CNC(c2c[nH]nc2C(=O)NC)=O)C1)=O 2816,C(=O)(C(C)(C)CS(N)(=O)=O)NC1CCN(C(C2(Oc3cn(C)nc3)CC2)=O)C1 2817,CC1NC(=O)OC12CN(C(C1(CNC(C3COC(=O)N3)=O)CCC1)=O)C2 2818,C1(C(N2C(CNC(c3cn(CCN(C)C)nn3)=O)C=CC2)=O)CC(=O)C12CCC2 2819,CC#CCCCC(=O)N1CCC(O)C(NC(C2CCCC(C)(C)C2)=O)C1 2820,CC(C)C(CO)C(=O)N(C(CNC(c1cnn(C2CC2)c1)=O)C1CC1)C 2821,C1(C(=O)NCC2(SC)CCC2)CN(C(=O)CCc2ccoc2)CCO1 2822,c1(CN2CC(CC(=O)NCc3nc(C)[nH]n3)OCC2)cccc([N+](=O)[O-])c1 2823,C1(O)(CCNC(c2ccccc2Cn2cnnn2)=O)CCCN(C(=O)C2CC2)C1 2824,c1(CN2CC(NC(c3c(Cl)ncc(C)c3)=O)(CO)C2)ccc2nc(O)[nH]c2c1 2825,C1(CN(C)C(C2CC2(C)C)=O)CCCN(C(c2snnc2C2CCC2)=O)C1 2826,N1(C(c2c(CC)c(F)ccc2)=O)CCC2(CC1)CC2NC(=O)CC1CC1 2827,Cc1cccc(CC(c2ncc[nH]2)NC(=O)N(C)Cc2ccccc2C)c1 2828,C1(OC(C(COC)N(C(C)(C)C)C)=O)CN(C(=O)OC(C)(C)C)CC12CC2 2829,Cc1nn(CC(N2CC(NC(C34CC(CN3C3CC3)C4)=O)CC2CO)=O)c(=O)o1 2830,c1(CC(=O)NCC(C)=CC(=O)NC2CCOC(C)C2)ccc(C)nc1O 2831,CC(C(=O)N1OC2C=CC1CC2)C1CCN(C(C2CC(C)(C)CO2)=O)C1 2832,c1(-c2c(C)nc[nH]2)nc(C2CCCO2)nn1C1CCSC1 2833,c1(C(=O)OCC)c(NC(=O)N(C2CCCC(=O)N2)C)c(C#N)cn1C 2834,c1(C(C(C2CCN(OC)CC2)C)NC(N2CCOCC2CF)=O)ccccc1F 2835,C1(CNC(c2ccc(C#C)cc2)=O)CN(C(c2cnn(C)c2F)=O)CC(C)(C)O1 2836,CCCCC(C(=O)N1CCN(C(=O)CCOC)C(C2CC2)C1)COC 2837,N1(C(C(CC)C(C)C)=O)CCOC2CN(C(c3ccc(OC)cc3C)=O)CC12 2838,N1(C(C2OCCC(NC(=O)CC3CCCCCC3)C2)=O)Cc2ncsc2C1 2839,c1(C(=O)NCC2C(C)CCN2C(=O)COc2ccc(Cl)cc2)ncc(F)cc1F 2840,N1(C(COC(C)=O)=O)CCCC2C1CCN2C(c1snc(O)c1Cl)=O 2841,C1(C(=O)NC(CCNC(C(N2CC(C)C2)C)=O)(C)C)CCC(F)(F)C1 2842,CCCC(CCC)=CC(N1CCN(CCNC(=O)CCc2cnc(O)[nH]2)CC1)=O 2843,FC1(F)CCC2C(CCN2CC(C2CCCCC2)F)C1 2844,N1(C(c2ccc(OCC)cc2)=O)CCCC(C)(C(=O)OC(C)(C)C)C1 2845,CCC(CC(=O)NC(C)C(C)C(=O)NCCOCCN=[N+]=[N-])CC(C)C 2846,c1(SC)ncc(Br)c(N2CC(NC(=O)C(C)(CO)CO)C(F)C2)n1 2847,N1(C(C2CN(CCC)C(=O)C2)C(=O)NCC2CCOCC2)CC(CO)C2(CC2)C1 2848,N1(C(c2n(C)ncn2)=O)CCC(O)(CNC(c2cnccc2Cl)=O)C1 2849,C(c1cccnc1)=CC(=O)N(C1CCN(C(C2COC(=O)O2)=O)C1)CC 2850,Cc1ccc(CCC(=O)N(CC(C)NC(c2c(C)ccn2C)=O)C)c(Br)c1 2851,C1(CNC(c2n(CCOC)ccc2)=O)CCCCN1C(=O)Cc1cnccc1C 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2870,C(C(CNC(c1cnn(-c2ccc(Cl)cc2)c1)=O)C(F)(F)F)NC(=O)C=CCF 2871,C12(C(N3CCC(NC(CC4CCN(C(C)C)CC4)=O)CC3)=O)CCCC1C2(F)F 2872,C1(C(=O)NC2CCCC(F)(F)C2)Cc2cc(O)ccc2CN1C(=O)CCBr 2873,c1(C(=O)NC(C)CCN(C)C(C2CC2C2CCC2)=O)ccc2c(c1)C=CS2(=O)=O 2874,Cc1cc(=NCC(C)(C)C2CCN(C(=O)CN3CCCC3=O)CC2)[nH]cc1C#N 2875,C(N=c1cc(C(C)=O)c([N+](=O)[O-])c[nH]1)C1CCN(C(C(CC)(F)F)=O)CC1C 2876,C1(C)(C(N(C)CC2CCN(C(C(C=C=C)C)=O)CC2)=O)CC(OC)CN1C 2877,C(=O)(C1c2c[nH]nc2CN1C(c1cc2ccccn2c1)=O)NCCOCCC#C 2878,CCCCC(CC)C(=O)NCCC(C)(C)NC(=O)CC1C=CCCC1 2879,C1(C(=O)NCC2N(C(C3(C)CC(C)(C)C3)=O)CCC2)CC2C(C1)C2(F)F 2880,C1(C#N)(C(=O)NCCCCCN(C(=O)CC2CCC23CCC3)C)CC1(C)C 2881,C#CC1CN(C(=O)CC(CCC)NC(=O)CNC(=O)CC)CC1O 2882,c1(C(=O)NC2C3CN(C(C=C(C)C(F)F)=O)C2C3)ccc(F)cc1C(F)(F)F 2883,c1(C(=O)NC2(COC)CN(C(C3CC(O)C3)=O)C2)cc(C2CC2)nc(O)c1 2884,C(=O)(CC1=NNC(=O)C1)NCCC1OCCCN(C(CC2CC(C)OC2C)=O)C1 2885,C1(C)(C(N(CCN(C(C)C)C(C2CCC(F)(F)C2)=O)C)=O)CCCN1C 2886,CC(C)CC(O)C(C)C(=O)NCc1nnn(C)c1C(=O)NC1COCC1C 2887,CC(CCCCCO)NC(=O)C=CC(C)(C)NC(C1CC(=O)OC1(C)C)=O 2888,N1(C(c2nc(C(=O)OC)sc2)=O)CCC2C(C1)CN2C(=O)CCCCC1CC1 2889,C12(NC(C3(OC)CC3)=O)CC1CN(C(C1(C(=O)CCNC(C)=O)CC1)=O)C2 2890,c1(CC(=O)NC2C(C)CN(C(C3CC3C)=O)CC2)ccc2c(c1)CCN2C 2891,C1(CN2C(C(=O)OC)CC(OC)CC2)CN(C(=O)OC(C)(C)C)CCN1C 2892,C(=O)(CC(CC)CC)NC(C(=O)NC(CCCCC)C)COC 2893,Cn1c(=O)c2ccc(NC(=O)NCC3(CCCO)CC3)cc2n(C)c1=O 2894,N1(C(Cc2c(CC)con2)=O)CCC(NC(C2(C)CC(C)=NO2)=O)C(O)C1 2895,N1(C(c2cc(C)oc2)=O)CC2COCCC2(NC(c2cccc3[nH]ncc23)=O)C1 2896,C12COCCN(C1)C(=O)C1(CCC1)C(=O)N2.c1(C(=O)OCC)c[nH]n(CC)c1=N 2897,CC1CC(CNC(C2CN(C3COC3)C2)=O)CN1C(=O)CCCCN(C)C 2898,C1(CC#C)(C(=O)NCCC#CCO)CCN(C(=O)C(CC)n2cncn2)C1 2899,C(=O)(CC(C)(C)CNC(C1CCCN1C=O)=O)NC(C)(C)CC1CCC1 2900,CC1=C(C(=O)NC2CN(C(C3(C(F)F)CCCC3)=O)CC3CC23)CCO1 2901,c1(C(=O)NCC2C(C(=O)Nc3ccc(CC)s3)C2(C)C)cnn(CC2CC2)c1C 2902,c1(C(=O)OC)[nH]c(C)c(C(=O)NCC2CCN2C(C2CC(Cl)(Cl)C2)=O)c1C 2903,C1(NC(C(=O)NCCC(C=C)C)=O)CC12CCOCC2 2904,CCC(C)CCCC(=O)NCC1(NC(C2(C(=O)N(C)C(C)C)CC2)=O)CC1 2905,C1(C(=O)NCC=CCNC(Cn2c(C)ncc2)=O)CCc2cnnn2C1 2906,N1(C(c2cn(CC)nc2)=O)CC(NC(c2coc(C(C)OC)n2)=O)C2(CCC2)C1 2907,c1(C(N(CCCCNC(C(C2CCCOC2)OC)=O)C)=O)c(C)nnn1C 2908,c1(CC)ccc(C(=O)NC(C(=O)NCCC2(C)OCCO2)c2cccs2)cc1 2909,C1(C(N2CCC(COC)(NC(=O)C=CCOC)CC2)=O)Cc2cccnc2C1 2910,c1(C(=O)NCCN(C(=O)C(C)NC(=O)NC)CC)ccc(NC)c(F)c1 2911,N1(C(CCN(C2CCCC(C)C2)CC=C)=O)CC2CCCC(C1)N2C 2912,c1(SC)nc(C(F)(F)F)c(C(N2CCC(C)(O)C2)=O)s1 2913,c1(C(=O)NCC(=C)CCNC(=O)C(F)=C2CCC2)cncc(P(C)(C)=O)c1 2914,C(C)(C)(CCC(=O)N1CC(NC(C2CCCCC(=O)N2)=O)CC1CO)OC 2915,n1(CC)ccnc1C=CC(=O)NN(C(=O)C(CCSC)OC)CCSC 2916,N1(C(C2(C#N)CC=CC2)=O)CC(C2CCCN(C(=O)CCCN=[N+]=[N-])C2)C1 2917,N1(C(Cn2ncc(C)c2)=O)CCC(NC(C2(c3cncs3)CC2)=O)C(O)C1 2918,C12CCCN(C1)C2=O.C1(CCNC(C2C(C(=O)OC)CC2)=O)CCSCC1 2919,Cc1ncsc1C=CC(=O)NC(C1(O)CCN(C(=O)Cc2cnn(C)c2)C1)C 2920,C(=O)(C1CCCCn2nnnc21)N1CC(CC)C(N2CCOCC2)C1 2921,C1(NC(=O)Nc2cc(CC)ncn2)CCN2CCC1C2 2922,c1(CC(=O)NC2C(NC(CCCNS(C)(=O)=O)=O)C2)c[nH]c2cc(F)ccc12 2923,c1(NC(c2cc(OC)c(-c3cccnc3O)cn2)=O)nccc2occc12 2924,C1(CNC(c2c(C)non2)=O)CC(F)CN1C(=O)C(C)Cc1cnn(C)c1 2925,C1(COC)(NC(=O)CC(C)COC)CCN(C(C2(OC)CCC2)=O)CC1 2926,c1(CC)nc(C)c(C(=O)NCC2(C(N)=O)CN(C(=O)C(Cl)=CCl)C2)s1 2927,C1(C(=O)NCCNC(c2cc3sccc3[nH]2)=O)Cc2ccccc2C(=O)O1 2928,c1(OC)nc(C(=O)NCCCCCN(C(C2CCCC(C)C2)=O)C(C)C)cc(O)n1 2929,c1(C(N2CCC(N(C(c3nncc(CCC)c3)=O)C)C2)=O)cc(OC)ccc1N 2930,C1(NC(CC2N(CC)C(=O)CC2)=O)CC12CCN(C(=O)CCc1ncco1)CC2 2931,n1(CC(=O)NCC=CCNC(c2oc(CC)c(C)c2)=O)nc(O)ccc1=O 2932,C1(NC(CCC=C(C)C)=O)CCOC(C(=O)NCCc2c[nH]nc2O)C1 2933,CCC(CCC(=O)N(CC(N1CCN(C(=O)Cc2cccnc2)CC1)=O)C)OC 2934,N1(C(CCC#CC)=O)CCC(C(=O)NCc2ncccc2Cl)C(C)C1 2935,N1(C(C2(NC(c3cn(CC=C)nc3)=O)CCN(C)C2)=O)CCC2C(=O)NCC2C1 2936,c1(-c2cn(CC(CCNC(C3(C)CC(=C)C3)=O)F)nn2)cccc2c1CCCC2 2937,C(C(C)(O)CC(=O)NC1CCCCN(C(=O)CC2CCSCC2)C1)OC 2938,c1(C(N2CCC(N(C(c3c(CC)c[nH]c3)=O)C)C(C)C2)=O)cc2ccccn2c1 2939,C(=O)(C#CC(=O)NC(CNC(=O)C(=O)N(C)C)C(C)(C)C)NC(C)C 2940,c1(C(N(CC(CC)NC(=O)Cn2ccnc2C)C)=O)ccc(CO)o1 2941,C(C(=O)O)(C1CC1C(F)(F)F)C(=O)NC(CC1(C)CC1)=O 2942,C1(C(C)NC(c2cn(CCN(C)C)nn2)=O)CCCN1C(=O)CC1CC(C)(F)C1 2943,C(=O)(CN1C(=O)COc2ccccc21)N(C)Cc1cn(Cc2ncon2)nn1 2944,c1(NC(C(C2C3COCC23)N(C)CCN2CCCC2=O)=O)cccc(Cl)c1 2945,C1(C(=O)NC2(CCNC(CC3C(CC)C3(F)F)=O)CC2)CCCCCCC1 2946,C1(C(N(CC(CC)NC(c2cccc(C)c2O)=O)C)=O)CC12CCCCC2 2947,Cc1cc(OCC(=O)N(CCN(C)C(c2nc(O)c(C)s2)=O)C(C)C)ccc1F 2948,C#Cc1cc(C(=O)NCC(C2CC2)N(C(=O)CCc2nccs2)C)ccc1C 2949,C1(NC(c2cn[nH]c2)=O)CC2(C1)CC(C(=O)NC1(CO)CC(F)C1)C2 2950,CC(C)C(O)C(F)(F)C(=O)N(C)CC1COCCN1C(c1ccc2c(c1)CC2)=O 2951,N1(c2nc(C)nc(O)c2)CC2(CN(C(=O)C=Cc3ccco3)CC2CO)C1 2952,CCC(CC(=O)N1CCC(N(CCO)C(C23CSCC2C3)=O)C1)SC 2953,c1(CC)noc(CN(C(CNC(C)CC#N)=O)C)n1 2954,C1(OC)CCN(C(=O)CN(C(=O)CCCN2CCCC2)C2CCC2)CC1 2955,C1(NC(C=CCC)=O)CC2CC(C1)CN(C(C1CCCN1C(C)C)=O)C2 2956,c1(C(=O)NC(CC(C)NC(=O)Cc2ccon2)C)sc2sccc2c1Cl 2957,c1(C(=O)NCCC2CN(C(C3(C(C)C)CCC3)=O)C2)csc2c1CCCCCC2 2958,c1(CC(=O)NCC2CCN(CC(=O)Nc3cccc(Cl)c3)C2)ccc([N+](=O)[O-])cc1 2959,C12CN(CCN1C(=O)OC(C)(C)C)C2=O.c1(CCC(=O)NC)cnc(C2CC2)o1 2960,c1(C(=O)NCCC2(C)CCN(C(=O)CSc3nc[nH]n3)C2)cc(O)nc(O)n1 2961,CC1(NC(=O)CN2CCCC2)CCN(C(c2sccc2C(F)F)=O)CC1 2962,c1(C(C)NCc2ncnn2CC(F)F)ccc(NC2CC2)cc1 2963,C(=O)(C(C)(C)CC(F)(F)F)N(CC(CNC(C(C(C)C)SC)=O)C)C 2964,C(c1ccc([N+](=O)[O-])cc1)=CC(=O)NC1CC(CN=c2[nH]nco2)C12CCC2 2965,C(=O)(CCC(=O)N1CC2C(NC(C3CCCOC3)=O)C2C1)N(C)C 2966,c1(C(=O)OC)c(C)[nH]c(C(N2CC(C)(NC(=O)CNS(N)(=O)=O)C2)=O)c1C 2967,C(=O)(C(C)(C)CN(C(=O)CC=C(Cl)Cl)C)NCC1CCC(C(=O)OC)O1 2968,C(CCCCC(=O)N1CC(CC)C1)n1cc(C(NOOCC)=O)nn1 2969,C(CCC(=O)NC(C)CC(C)NC(c1occc1-c1cnn(C)c1)=O)OC(C)C 2970,c1(C(=O)NCC2(c3ccccc3)C(C)C2)ccc2nc(O)oc2c1 2971,C12(C(N3CCC(N(C(C4CCC5CC5C4)=O)CC)C3)=O)CCOC(C)(C1)C2 2972,N1(C(c2n(CC)nc(C)c2)=O)CC(NC(=O)CC2CCOC2)CC(F)C1 2973,C1(CC)(OC)CN(C(=O)CCCC2(NC(c3sccc3CO)=O)CCC2)C1 2974,c1(C(N2CCC(CCOC)CC2)=O)cc(C(F)(F)F)cnc1O 2975,N1(C(=O)C=CCF)CC2CCCC(C1)N(C(=O)Cc1ccsn1)C2 2976,c1(OC)nc(C)cc(=NC2CC23CC(NC(=O)C(C)CC(N)=O)C3)[nH]1 2977,C1(C(=O)OCCCC2CCCC2)CC2(CCCC2)CO1 2978,c1(OC)cc(C(N2CCCC(NC(=O)CC3SC(=N)NC3=O)CC2)=O)cc(C)n1 2979,C#Cc1cncc(C(=O)NC23CCN(C(=O)Cn4nc(C)ccc4=O)CC2C3)c1 2980,CN1CC(C)(C(N2CC3(CCN3C(C3COCOC3)=O)C2)=O)CCC1=O 2981,N1(C(c2ccc(C)s2)=O)CCN(C(=O)CCC2(C)CC2)C(C(F)F)C1 2982,N1(C(CP(C)(C)=O)=O)CC2C3CCC(C2C1)N(C(=O)C=C1CN2CCC1CC2)C3 2983,C(=O)(C1CCCc2nn[nH]c21)NC1CC(C)(NC(c2ccc(Br)c(O)n2)=O)C1 2984,Cc1ccc(CC(=O)NCC2CN(C(C3CC3C)=O)CC23CC3)cc1Cl 2985,N1(C(CCCC#CC)=O)CCC2(CCC2NC(=O)CC2OCCC2(C)C)CC1 2986,c1(C(N)=O)cc2oc(C(N3CCC4C(C3)CN4C(=O)C#CC3CC3)=O)cc2[nH]1 2987,N1(C(C(CCSC)O)=O)CCCC(NC(C2CCN(C(C)=O)CC2)=O)CC1 2988,N1(C(C2(C)CCCN(C(c3cc(C)n(C)c3)=O)C2)=O)CCC2(CCC2)CC1 2989,N1(C(C(CC=C)C)=O)CCC(C2CN(C(=O)Cc3cccc(Br)c3)C2)C1 2990,C1(C(=O)NC2CN(C(=O)COC3CCCC3O)C2)C2C3CC4C1C1C2CC3C41 2991,Fc1ccc2c(c1)C(c1nc(Cc3ccccc3Cl)nn1-c1ccno1)CO2 2992,Cc1nc(C(=O)NCCNC(C2CC2C(=O)NCCO)=O)cs1 2993,CC1CCC(C)C1NC(c1c(CNC(=O)CN=[N+]=[N-])nnn1C)=O 2994,c1(CC(=O)OCCC2C(C)(C)CCO2)cccc2nsnc12 2995,Cc1cc(C(=O)NCCCNC(=O)C=CC2CCOC2)nn1-c1ccc(F)cc1 2996,Cc1nn(C)c(NNC(=O)N(c2nnc(CO)n2C)C)c1C#N 2997,c1(CNC(C2C(O)CCN(c3c(C)cncn3)C2)=O)ccc(F)c2ccccc12 2998,Cc1ccc(C(=O)NCCCN(CCCNC(=O)C(C)n2ccnn2)C)cc1 2999,c1(C(c2n(CC=C)nnn2)NCc2cncn2C(C)C)ccc(C(F)(F)F)cn1 3000,C(CCC[Si](C)(C)C)Nc1cc(C)c(-c2cccc(CCN)c2)s1.CCO 3001,n1(CC)ccc(C(=O)NCC2CCN(C(c3ccc(CO)c(C)c3)=O)C2)cc1=O 3002,C#CCCCCC(=O)NC1CC(C(C)NC(C23CCCN2CCC3)=O)C1 3003,c1(-c2ccnc(N3C(C(=O)Nc4cnncc4Br)CC3)n2)cccc([N+](=O)[O-])c1 3004,c1(C(=O)NCC(N(C(C=CC)=O)C)C2CC2)cc2cccc(O)c2[nH]1 3005,c1(CC)cc(F)ccc1C(=O)NCC1CN(C(C2CC3C(C2)C3(F)F)=O)CC1O 3006,N1(C(C2(C)CCC2)=O)CCC2(CCOC2)C(CNC(=O)CCCCNC(N)=O)C1 3007,C12CC3CC1CN(C3)C(=O)CN2C1CC1.CC(C(=O)NC1CCCC1)C1CCC1 3008,Cc1ncccc1C(N1CCC(C)(CCNC(C2(NC(C)C)CC2)=O)C1)=O 3009,C(C1CCCN1C(c1csc(Cl)c1)=O)=CC(=O)NCCSC 3010,C1(NC(c2c(CC)ccs2)=O)CC2CN(C(c3c(C)noc3CC)=O)CC2C1 3011,C1(C(=O)NC(C(C)O)(C)C)CCCCCC1NC(=O)CC1OCCO1 3012,c1(SCC(=O)N(CC(C)NC(C2CCCCN2C)=O)C)ccc(N)cc1 3013,n1(CCSC)nnnc1C(c1ncco1)NCC1CC12CC2 3014,Cn1cc(C2OCCC2C(=O)NC2CC(NC(c3cc(O)cs3)=O)C2)cn1 3015,N1(C(=O)NCC(c2ccc(CC)cc2)O)CC=C(c2cccc(Cl)c2C)C1 3016,C(=O)(CCCC(=O)N1CC2CC2(NC(C2CCC3CCC2O3)=O)C1)NC(C)C 3017,CN=c1ncc(-c2ccc(F)c(CN3CCC(N(C)CC4CC4)CC3)c2)c[nH]1 3018,C1(C(C)NC(C2(C(=O)NC)CCC2)=O)CCCN(C(c2sc(C)cc2Cl)=O)C1 3019,Cc1c[nH]cc1C(=O)NCCC(O)CNC(c1cnn(Cc2ccccc2)c1)=O 3020,c1(CC)[nH]nc(C=O)c1Cl.N12CC(C(=O)NCCC(=O)N(CC)CC)C1C2.CC 3021,Cc1nc2c(cc1C(=O)NCCC1COCCN1C(=O)C=C1CC1)c(C)nn2C 3022,C1(C(=O)NCC(CN(C(c2c(CC)cco2)=O)C)(C)C)CC12CCC(=O)CC2 3023,Cc1ccc(NC(C2C(NC(=O)CCN=[N+]=[N-])C2(C)C)=O)c(C)n1 3024,C(C(=O)NCCC1CCN(C(c2nccnc2N)=O)C1)(C(C)C)SCC 3025,C(=O)(C(O)CC(C)(C)C)N(CC(CNC(CC(C)(C)OC)=O)C)C 3026,CCCCC(O)C(=O)N(CCCCCCNC(=O)Cc1cccc(C(N)=O)c1)C 3027,c1(OC)c(F)cc(C(=O)NC(C2CN(C(c3cc[nH]n3)=O)C2)C)cc1Cl 3028,N1(OC(=O)NCCC(C(F)F)NC(=O)OC(C)(C)C)CC(C)(C)C1(C)C 3029,C#CCCC(O)C(=O)NC(C)CCNC(c1snnc1CC)=O 3030,C1(C(N2CCCC(NC(CCc3ncc(C)[nH]3)=O)C2C)=O)CS(=O)(=O)CC(=O)N1 3031,C(=O)(CCCCC#N)NC1CN(C(c2c(CC)non2)=O)CC1C 3032,N1(C(CC)C(C)C)CC2COCC2(C(=O)NCC(=O)NC2CC2)C1 3033,C1(NC(Cc2nc(C)sc2)=O)CCC2(CCN(C(c3ccn(C)c(=O)c3)=O)C2)C1 3034,N1(C(C(C(CC)C)N(C(=O)CN2CCCCC2)C)=O)CCN2CC(O)CC2C1 3035,N1(C(c2c(C)nc(=N)[nH]c2)=O)CC2CN(C(=O)C(C)(C)F)CCC2(CO)C1 3036,C1(C(=O)NCC(C)N(C(=O)Cc2ccn(C)n2)C)OC2CCC1CC2 3037,CC1C(C)C(C)CN1C(=O)NCc1ccc(N(C)C(N)=O)cc1 3038,CCC(CCC(=O)NCc1ccon1)NC(=O)Cc1cn(C)nc1C 3039,Cc1cc(=NC(=O)C(C)C(C)NC(c2cc(C3CC3)no2)=O)[nH]n1C 3040,c1(C(N(CCNC(C2CCCC2n2cccc2)=O)CC)=O)ncc(C)cn1 3041,CC(C)CC(F)C(=O)NCC(CNC(=O)Cc1ccc(Br)cn1)CO 3042,C(CC(C)C)(C(=O)NC1C(C)C1C)ON(C(COC(CC)CC)=O)C 3043,c1(CNC(C)=O)ccc(C(=O)NCC2C(NC(=O)CCCF)C2(C)C)cc1 3044,c1(C(=O)NCCN(C(CCn2c(C)ncc2)=O)CC(C)O)c[nH]c(=S)cn1 3045,CCCC(C)CC(=O)NC1(CCCC(=O)NCCOC)CC1 3046,c1(OC)ccc(NC(C2CCN(Cc3ccnc(Cl)c3Br)CC2O)=O)cc1Br 3047,C(=O)(CC1OCc2ccccc21)N(CCOCC)CCNC(=O)C(=O)N(C)C 3048,Cc1nnc2n1CCN(C(C1CCCN(CCS(C)(=O)=O)C1)=O)C2 3049,c1(CCNC(c2n(C(CC)C)nnn2)c2cnn[nH]2)cccc2ccncc12 3050,CC1CN(C(=O)Cc2cc(Cl)ccc2O)CCC1NC(=O)Cn1ccnn1 3051,N1(C(c2cnn(C)c2C)C(=O)NCCCSCC)CC(C)CCCC1C 3052,C1(C(=O)NCC(CC)N(C)C)(CNC(c2cc(Cl)cs2)=O)CCCC1 3053,C(C(CC(C)C)C(=O)NC(C)Cc1nc[nH]n1)NC(c1c(C)noc1)=O 3054,c1(C(N2CC(CC=C)(NC(C3CC3CF)=O)C2)=O)cn2cccc(C)c2n1 3055,C12(NC(c3cncc(-n4ccnn4)c3)=O)CC1CN(C(C1CCC13CCC3)=O)C2 3056,N12CC3(CC(F)(C1)C3)C2.C12CC(C1)C2c1cc[nH]n1.CS(=O)(=S)NCc1ccco1 3057,CN1C(=O)CC(C(N2CC(F)(CNC(=O)CSC3CC3)C2)=O)C1c1ccnn1C 3058,S(=O)(=O)(c1ccc(N2CCOC(C#N)C2)c(F)c1)N1Cc2c(ccc(OC)c2)C1 3059,C(=O)(CC(C(F)(F)F)c1ccon1)N1CC(O)(CNC(C(C)(C2CC2)OC)=O)C1 3060,N1(C(C=C(COC)C)=O)CCC(N(C(=O)COC2CC2(F)F)CCO)C1 3061,c1(OC)ccccc1C=CC(=O)N(C)CCNC(=O)CC(c1c(C)noc1C)C 3062,C1(NC(C=CCC(C)(C)NC(=O)CC2(O)CCOCC2)=O)CC2(CNC(=O)O2)C1 3063,CC1CCN(C(c2cc(Cl)cn2C)=O)C(C(=O)NCC2(CO)CC2C)C1.C(N)=O 3064,Cc1cc(CC(=O)NCC2(O)CCN(C(=O)CC3CCCN(C)C3)C2)cc(O)n1 3065,C1(CN(C(C(C=CCCC)O)=O)C)CN(C(=O)C(C)(C)CF)CCO1 3066,C(C(O)CN=c1[nH]c(C2CCCC2)nc(=N)[nH]1)NC(C=C(CCC)CCC)=O 3067,C(N=c1[nH]nc(-c2cccnc2)s1)C1CCC(NC(c2cc(C)ncc2)=O)C1 3068,c1(N2CC(CNC(Cc3cccc(C)c3C)=O)OCCC2)nc2cccc(C)c2o1 3069,Cc1nn(CC(=O)NC(C)CCNC(C2CCCCCC2)=O)cc1[N+](=O)[O-] 3070,N1(C(Cn2c(C(=O)OC)cc(C)n2)=O)CCC(F)C(NC(c2sc(=N)[nH]c2C)=O)C1 3071,CC1CCN(C(=O)C(C2CCCCCC2)O)CC1N(C(=O)Cc1cncnc1)C 3072,N1(C(CCCCCOCC)=O)CCC2CCN(C(=O)C(C(C)C)C(C)C)CC12 3073,C(=O)(C(C)(C)CN(C)C(C1COCC(C)O1)=O)N(CC(CC)OC)C 3074,c1(N2C(CCO)CN(Cc3ccncc3Br)CC2)ncnc2ccc(F)cc12 3075,c1(C(=O)NCC(CNC(=O)C=CCO)O)cc(Cl)cc2c1CCC2 3076,Cc1cccc(C(N2CCC(CNC(=O)CCCF)C2(C)C)=O)c1C 3077,c1(N2CCN(C(=O)Cc3ccc(C(CC)C)cc3)CC2)ncnc2oc(C)nc12 3078,C1(CNC(c2cc(O)ncn2)=O)CN(C(C2C(F)(F)C23CC3)=O)CCCO1 3079,c1(C(=O)NC(CNC(CCCCC)=O)CC(C)C)cc(C2CC2)ccc1F 3080,C(C(CC(C)C)C(=O)NCC1(C)CNC(=O)O1)NC(C1(CC=C)CC1)=O 3081,C1(CN(C)C(C2CCCOC2)=O)CCN(C(=O)Cn2ccc(C(F)(F)F)n2)CC1 3082,c1(C(=O)NC2CC(N(C(C=CSC)=O)C)C2)ccc(NC(=O)N(C)C)cc1 3083,C1(C(N(C2(CC(=O)NCC3(O)CN(C)C3)CC2)C)=O)CCCC12CCC2 3084,N1(CC(=O)NCCNC(C2C(C)OC(=O)N2)=O)CCC(=O)NC1=O 3085,c1(OC)ccc(Cl)cc1CNCC(CC(F)F)NC(=O)OC(C)(C)C 3086,CC1CC(C)(C(N2CCCC(C)(CNC(=O)CC3CC3(Cl)Cl)C2)=O)CC(C)O1 3087,c1(CN(C2(C#N)CCC2)CCOCc2ccc(OC)cc2)c(C)cc(C)cc1C 3088,c1(C(C)NC(C2CCN(C(C3CCCC4CC34)=O)C2)=O)ccc(Cl)c(Cl)c1 3089,c1(C(=O)NCCOCC)nc(C)cnc1NC(c1cccc(OCC)c1)=O 3090,c1(C(=O)NCC(c2c(CC)cccc2)NC(=O)C(C)(Cl)Cl)cc(N)c(F)cn1 3091,C(=O)(CCCNC(=O)C1CC1)NC(CN(C(=O)CC1CC1(C)C)C)(C)C 3092,c1(OCC)cccnc1C(=O)NC1CCOCC1NC(=O)C(C1CCCCC1)O 3093,N1(c2ncc(CCC)cn2)CCOCC(NC(c2ccon2)=O)C1 3094,c1(C(=O)Nc2c(C)ccc(NC(=O)C(C)N(C)C)c2)ccnc2c1c(C)nn2C 3095,C(=O)(C(C(C)CC)N(C)C(c1cscc1Cl)=O)NC(CCC)(C)CC 3096,c1(C(N2CCC(CNC(=O)Cc3csnc3C)CC2)=O)cnc(N(C)CC)nc1 3097,c1(C(=O)NC(C(=O)OC(C)C)C)ccc(CNC(c2nonc2N)=O)cc1 3098,C1(C(CN2CC(C(N(c3ncn(C)n3)C)=O)C2)=O)CCCC2CC12 3099,N1(C(c2c(C(=O)OC)cccn2)=O)CCC2CC2(NC(=O)CCS(N)(=O)=O)CC1 3100,C1(N(C(CCCC)=O)C(=O)Cc2cc(C)[nH]n2)CCNC1=O 3101,c1(N2C(CNC(C3N(C(C)C)CCC3)=O)C(C)CC2)nc(Cl)ncc1C(F)(F)F 3102,N1(C(C(C)(O)C2CCC2)=O)CC2CC(C1)C2NC(c1sc(Cl)cc1Cl)=O 3103,C1(CNC(C=C)=O)C(C)CCCN1C(c1ccc(CC(C)C)nc1)=O 3104,c1(C(=O)NC2CCCC(CNC(c3cnsn3)=O)C2)ccc2c(c1)CCCS2 3105,N1(C(c2c(SC)cccc2)=O)CCCC2C1CCCN2C(=O)CSc1ccco1 3106,C1(C(N(C)CC2CCCN2C(c2ccccc2CO)=O)=O)CCC(C)(C)OC1 3107,c1(C(N2C(CC)C(NC(c3ccccc3Cl)=O)CC2)=O)ccc2c(c1)N(C)CC2 3108,n1(CC=C)c(SC(=O)CCCS(C)(=O)=O)nc2ccccc2c1=O 3109,C1(NC(Cn2cc(C(=O)OC)nc2)=O)CCN(C(=O)C(C)CC(C)C)C(C)C1 3110,N#Cc1cc(C(N2CC(NC(C3CC3(F)F)=O)C3(CCC3)C2)=O)cc(F)c1F 3111,N1(C(C=C(C)CNC(=O)Cc2scnc2C)=O)CCCC1C(C)O 3112,CN1CC(NC(C2CN(C(=O)CN3CCNC3=O)CC23CC3)=O)CCC1=O 3113,C1(NC(C2CC2C2CCC2)=O)COC2(CCN(C(=O)C=C(Cl)Cl)CC2)C1 3114,CCC(C)(C)C(C)CC(=O)N1CCC(C)N(C(C2CCCCCCC2)=O)CC1 3115,CCCC(C)C(=O)N1CCCC1CN(C(=O)Cn1cccc1)CC 3116,c1(OC)cc(C(=O)NCC2COCCN2C(c2ccccc2C#N)=O)ccc1Cl 3117,C1(NC2CC(C(=O)OCC)N(C3CC3)C2)CC2CCC(C1)N2C(=O)OC(C)(C)C 3118,c1(C(=O)NC(CC(C)NC(c2cc[nH]c2)=O)C)ccc(-c2cnc[nH]2)cc1 3119,N1(C(c2c(CC)n(C)cc2)=O)CC2COCC2(C(=O)NCC2CCCN2C)C1 3120,C1(NC(C(C)C2(O)CCC2)=O)COCCC1C(=O)NOCC1CCOCC1 3121,C1(C(N(CC(CCC)O)C)=O)CC(OC)CN1C(=O)CC1CC2(CCC2)C1 3122,C1(NC(C2C(=C)C2C(=O)OC)=O)CCCN(C(=O)C(C)(C)C(C)C)CC1 3123,C1(C(=O)NC2(C)CC(=C)C2)CCN(C(C2CCCCCN2C)=O)C(C)(C)C1 3124,C(=O)(C(=O)CC(C)C)NCCCC(N1CCCC(CC=CC)C1)=O 3125,C(=O)(C(C)CC(C)CC(C)C)NCC1(F)CC(NC(c2nnn(CC)c2C)=O)C1 3126,c1(CNc2cc(N3CC4C(CO)(C4)C3)ncn2)ccc2c(c1)NCCO2 3127,C1(C(N2CCCC2)=O)CCCC(SCC)C1.C1(C(=O)OCC)(C(=O)NC)CC1 3128,C1(SC)CN(C(=O)OC(C)(C)C)CC1N(CC(c1ccccc1)c1ccccc1)CCl 3129,C1(C(=O)NCC2(O)CCN(C(CCCN(C)C)=O)CC2)CC12CCC(F)(F)CC2 3130,O=S(=O)(c1cnccc1N1CC=CC(O)C1)NCC(c1cccnc1)CO 3131,Cc1ncc(NC(=O)C(C)NC(=O)C(C)C2(O)CCC2)c(C)c1C 3132,c1(CN(C(=O)C(=O)Nc2ccc3nn[nH]c3c2)CCOC)ccc(S(C)(=O)=O)cc1 3133,c1(CC)cc(C(=O)NC(C)C(C)NC(=O)C(F)C2CCCC2)ccc1O 3134,C(=O)(C(F)C(C)CNC(=O)CC1(CO)CC1)N(C)Cc1c(OC)cccc1 3135,C12(C(=O)NCc3cnc(C)o3)CC1CN(C(C1CCO1)=O)C2 3136,N12CCC3CC(CCC3C1)C2=O.N=c1ccc(Cl)c(CSc2nn[nH]n2)[nH]1 3137,c1(C(=O)OC)cn(C)nc1C(=O)NC(C)CNC(=O)Cc1cnns1 3138,Cc1nc2cc(NC(=O)C(C(C)(C)C)NC(N)=O)cnc2[nH]1 3139,C(CNC(=O)C(F)(F)C(F)F)(CC(F)(F)F)NC(C1CN(S(CC)(=O)=O)C1)=O 3140,C1(NC(C)=O)CCN(C(=S)Nc2ccc(Cl)c(F)c2)C1 3141,N1(C(CC2(CSC)CC2)=O)CC(O)(CCCNC(C2CCC3CC23)=O)C1 3142,C1(C(=O)NCCn2ccc(C(N3CC(C)=C(C)C3)=O)c2)CC2(CC(=O)C2)C1 3143,C12CCCN(C1)C(=O)c1cccc(c1)OC(=O)C2C.Cc1csc(CNC)n1 3144,C1(c2nc(CCCCCC)nn2C(C)C(C)(C)C)CCn2c(C)cnc2C1 3145,C(=O)(CCCCCn1cc(CO)nn1)NC1CCCC1CN.Cc1cc(OC)n(C)n1 3146,Cc1ccc(CCC(N2CCC(C)N(C(=O)C=CC(N)=O)CC2)=O)cc1[N+](=O)[O-] 3147,N1(C(C=CC)=O)CC(NC(=O)CCC(=O)NCC2CC2)C(C(F)F)C1 3148,C1(C#N)(C(N2CCCN(CCC(C)(C)O)CC2)=O)CCC(F)(F)CC1 3149,C1(NC(CCOC)=O)CC2CCC1C(NC(=O)C=Cc1ccc(OC)cc1C)C2 3150,CCCC(C(=O)NC1(C)CCN(C(c2nccn3ccnc23)=O)C1)C(C)C 3151,CC1(NC(c2cnc(Br)s2)=O)CCN(C(C2(O)CCC2)=O)C1 3152,CC(C)(C#N)CCCC(=O)NC1CCCC(NC(C2CC23CCSCC3)=O)C1 3153,c1(CCC)cc(C(N2CC(F)CC2CNC(=O)C(C)O)=O)sc1C 3154,c1(OC)ccc(Br)cc1CNC(c1ccnn1C(F)(F)F)c1nnnn1C(C)C 3155,c1ccccc1[N+](=O)[O-].CC(CCNC(=O)C=CC(N)=O)NC 3156,C1(CC(N2C(C(=O)NCC=C3CCSCC3)CC2)=O)CC2(CCC2)C1 3157,c1(C(=O)NCC#CCNC(C(C)C2CCC2)=O)cc(C(F)(F)F)cc(O)n1 3158,c1(C(N2CCCCC2c2n[nH]c(C(C)C)n2)C(=O)NCC(C)C)nc(Br)nn1C 3159,C1(CCC)CN(C(=O)Cn2nc(C)nc2C)CCN1C(=O)C1=C(Cl)CCC1 3160,N1(C(C2N(C(C3CC3c3ccc(Br)cc3)=O)CCC2)=O)CCN2CC(O)CC2C1 3161,C1(NC(C2(NC(C)=O)CC2)=O)CCC(N(C(=O)CCN(C)C)C)CC1 3162,C(=O)(C(C)(C)C(C)C)N(CCCCN(C(C1C(C)=CCS1)=O)C)C 3163,C1(NC(CC(C)N(C)C)=O)CC(C(=O)NC(C)(C)CC2CCC2)C1(C)C 3164,c1(OC)ccc(Br)c(C(=O)NCC(C)NC(C2CC3(C2)CC(O)C3)=O)c1 3165,C(=O)(C1=NN(C)C(=O)CC1)NC1(c2c(F)ccc(-c3ccc(OC)cn3)c2)CC1 3166,C(=O)(CCCCCF)NCCN(CCOC)C(C1CC1C1CCCC1)=O 3167,CCCC(C)(O)CC(=O)NC1(C)CCCCC1C(N1CC=CC1CF)=O 3168,CC(CNC(c1csc(O)n1)=O)C(F)C(=O)NCCF 3169,N1(C(c2cnc(OC)s2)=O)CC2(CCC2NC(=O)C(O)Cc2cn(C)cn2)C1 3170,CCC(CC)(CCNC(C1CC1(Cl)Cl)=O)NC(=O)C(N)=O 3171,c1(OC)cccc(CC(=O)NC2CN(C(=O)CN3CC=CC3)CC2C)c1Cl 3172,C1(CNC(c2ccc(Cl)s2)=O)CCCN1C(=O)CC(C1CC1)NC1CC1.C1CC1 3173,N1(C(CCCOC(C)C)=O)CC2CC(NC(=O)C(CC(F)F)C3CCC3)C(C2)C1 3174,N1(C(C(C)OCC2CC2)=O)CC(C(=O)N(C)CC2CCCOC2)C(F)(F)C1 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3193,N1(C(c2c(COC)noc2)=O)CCC2CCCC(C1)N2C(c1ccnnc1S)=O 3194,C1(C(N2CCC(N(C(c3c(Cl)n[nH]c3C)=O)CC)C2)=O)CCOC(=O)CC1 3195,C#Cc1cncc(C(=O)NC(CN(C)C(C2CCS(=O)(=O)N2)=O)CC)c1 3196,n1(CC)nncc1C(=O)NC1CC(NC(=O)C(F)(F)c2nc(C)cs2)C1 3197,c1(CN2CC3C(C(N4CCCC(C(C)(C)O)C4)=O)C3C2)ccnc(F)c1Cl 3198,c1(NC2C(C)C2)cc(S(=O)(=O)NCc2ccc(F)cc2)ccc1C#N 3199,C1(C(N(CC(F)F)CCC)=O)CSCN1C(c1cc(OCC)no1)=O 3200,CCC(CCC(=O)NC1CCN(CC2CC2)C1)NC(c1ccnnc1C)=O 3201,c1(C(=O)NC2CC(CNC(C3CC(C#C)(O)C3)=O)C2)ccc2ncc(=O)[nH]c2c1 3202,c1(OC)cccc2c1CC(C(=O)N(C)CCN(C)C(C1CC(C#N)C1)=O)CO2 3203,C1(C(N2CCC(NC(=O)C3=CCCCO3)C(F)C2)=O)CC2CCC(C1)S2(=O)=O 3204,N1(C(c2ccc(C)o2)=O)CC2CCC(C1)N2Cc1ccc(C(N)=O)cc1 3205,CCCCCCCCC(=O)NCC(F)CNC(=O)CC(C)(C)C1CCCCC1 3206,C(=O)(C(C)(C)C(=O)NC(N)=O)N(C)CCN1CCN(C(=O)CCOC(C)(C)C)CC1 3207,N1(C(c2cscn2)=O)CCC2(CCCCN(C(C34CC(C3)C4)=O)C2)C1 3208,N1(C(C(C=C)(F)F)=O)CCCC(CCNC(C2CC3CCC3C2)=O)CC1 3209,C1(OC)CN(C(=O)Cn2nnc(C)n2)C(C)(CNC(c2ccc(CO)cn2)=O)C1 3210,Cc1cc(CC(N2CCC(NC(=O)Cc3ccc(Br)s3)C2)=O)c(C)s1 3211,Cc1nc2ccc(COC(=O)CNC(=O)Cc3cccc4c3SCCC4)cc2s1 3212,C1(C(=O)NCCCCCN(C(COCC(C)C)=O)C)CC(S(C)(=O)=O)C1 3213,c1(C(=O)NC(C2CCCN2C(C2CCC2C(F)F)=O)(C)C)cncc(F)c1 3214,C1(C(N2CCC(NC(c3cccc(Cl)c3F)=O)CC2)=O)CCCCCCC1 3215,Cc1cc(C(=O)NCC2CCN(C(c3ncc(Cl)cc3Cl)=O)CC2)ccc1F 3216,c1(C(N2C(CN(C)C(C3CCNC(=O)C3)=O)CC(F)C2)=O)cn2cnnc2cn1 3217,C(=O)(C(C)C(C)n1cccn1)N.C(CCC(=O)NC1CN(C(C)=O)C1)NC(=O)OC 3218,C1(C)(C(N(C2CCN(C)C2)CCC)=O)CCN(C(c2ccccc2Cl)=O)C1 3219,C1(NC(CN2CC(C)C2)=O)CCC2CN(C(c3ccc(N)c(N)c3)=O)CC2C1 3220,C1(C(=O)NCC2(C3(O)CN(C(C(=O)NCC)=O)C3)CC2)CC2(C1)NC(=O)NC2=O 3221,c1(NC(C2(C#C)CN(C(c3cncc(F)c3)=O)C2)=O)c(C)[nH]c(C)cc1=O 3222,c1(OC)ncc(C=CC(N2CCC(NC(=O)Cc3ccns3)CC2)=O)cn1 3223,C(=O)(N=c1[nH]nc(C(F)(F)F)s1)OC(C)(C)C.C12(CCOC)CCN(C1)C2=O 3224,c1(C(C)C)cc(C(N2CCC(CN3CCC(N)C3)CC2)=O)nn1-c1ccccn1 3225,C1(N(C(=O)Cc2ccsn2)C)C2CN(C(C3(C)CCCS3)=O)CC12 3226,c1(C(=O)NC(CC)CNC(=O)C(O)c2ccco2)ccnc(SC(C)(C)C)c1 3227,CCCCCCN(C(=O)CNC(=O)CCNC(=O)C(C)SCC)C 3228,N1(C(CC=C)=O)CCCC(C)(NC(=O)C(C)OCCOC)C1 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3264,C1(C2CN(C(=O)C(c3ccccc3Cl)N(C)C)C2)(CNC(C(C)CN(C)C)=O)CC1 3265,C=C=CCCC(=O)N(CC)CC1CCCCN1C(=O)CC1(OCC)CCC1 3266,N#CC1(C(N2CCCN(C(=O)C(c3cccc(F)c3)O)CC2)=O)CC2CC2C1 3267,c12cc(ncn1)C(=O)O2.c1(N(C(=O)C(F)(F)F)CC2CCCNC2)cccc(F)n1 3268,C1(C(N(CC(C)NC(=O)CCSC)CC)=O)(OC)CC(CF)C1 3269,C(=O)(C(CCCC)N(C)C)N1CCC(O)(CN(C(CCC=CCC=C)=O)C)C1 3270,c1(C)ncc(NC(C2CC(NC(CSC(C)(C)C)C3CC3)C2)=O)cn1.C1CC1 3271,N1(C(C2(CCC=C)CC2)=O)CCN(C(=O)CCn2nc(C)cc2C)CC(C)C1 3272,C1(C)(C(=O)NCC2(NC(C(N3CCC(O)CC3)C)=O)CCCC2)COCCO1 3273,c1(C(N(c2ncnc(OC)c2C)C2CNCC2F)=O)ccc(F)c(Br)c1F 3274,CC1(C)CCc2cc(C(N3CCOCC3CNC(=O)C#CC3CC3)=O)ccc21 3275,c1(OC)ccc(C2(CNC3CC(CN)C(O)C3)CC2)cc1O 3276,c1(-c2cn(C3CCC(C(=O)NC4CCCC4C(=O)O)C3)nn2)c(F)cccc1Cl 3277,C1(C(N(CCC(=O)NC2C=CCCC2)CC#C)=O)CCCC(=O)CC1 3278,C(=O)(C1=NOC2(CCN(Cc3csc(Br)n3)C2)C1)NCC1(C)CC1 3279,c1(C(N2CC(N(C(c3c(C)onc3)=O)C)C2)=O)cn2c(n1)CCC2 3280,CC1Cc2cc(C(N3CCN(C(=O)CC(C)(C)C(F)(F)F)CC3C)=O)ccc2O1 3281,N1(C(C(CC)C(=O)OC)=O)CCC2CN(C(C3CC(F)(F)C3(C)C)=O)C(C)C12 3282,CC1COC(CNC(=O)NC(CC2CC2)Cc2cccc(F)c2)CO1 3283,c1(C(N)=O)c[nH]c(C(=O)NCCOCCNC(c2nncs2)=O)c1 3284,C1(OC)COCCC1NC(=O)COC(C)(C)CNC(C1(SC)CC(=O)C1)=O 3285,c1(CCNC(Cc2nc(NC(=O)OC(C)(C)C)sc2)=O)c(C#N)ccc(Cl)c1F 3286,C1(N2CC(c3ccc(OC)c(OC(F)F)c3)C2)Cc2ccccc2C1C 3287,Cc1[nH]c2ccc(C(=O)NCC(C(C)C)NC(=O)C(=O)C3CCCC3)cc2c1C 3288,N1(C(C2=CC(C)(C)C2)=O)CCC2CN(C(c3ccc4c(c3)CCOC4)=O)CC2C1 3289,C1(NC(c2c(C)cccc2)=O)CC2CC1CN2C(c1ccc(F)cc1)=O 3290,N1(C(C2(C)CCCCCC2)=O)CC2(CC(NC(C3CCCS(=O)(=O)N3)=O)CO2)C1 3291,C1(CC=C)(C(=O)NCC[Si](C)(C)C)CN(C(=O)C(C)c2cccs2)C1 3292,Cc1cc(C(=O)NC(c2nccs2)C)c(C)n1N 3293,C1(CC(=O)NCC2C(C(=O)NCCc3onc(C)n3)C2)C(C)(C)C1(C)C 3294,c1(C(=O)NCC2CC(NC(C(c3n(C)ncc3)O)=O)C2)cc2cc(F)ccc2o1 3295,CN=c1[nH]cc(C(N2CCCC2C2CCN(C(c3scnc3C)=O)C2)=O)o1 3296,c1(OC)ccc(Cn2nc(C(C3CC3)OC)nc2-c2cnns2)cc1 3297,c1(CCNC(=O)NC(c2cnn(C)c2)CC)cn(C)cn1 3298,C(=O)(N=S(C)(=O)c1cccc(F)c1)c1cn(C)nc1C(N1CCOCC1)=O 3299,Cc1cncc(CC(=O)NCC(C)(C)CN(C)C(C2NC(=O)OC2C)=O)c1 3300,C=CC(C)(CCOC)C(=O)NCCCCC(C)NC(C1CCC(C)CC1)=O 3301,C(=O)(CC(C)CCC=C(C)C)N(C1CCN(C(C2CCCC(C)O2)=O)CC1)CC 3302,CN1CCOCC(NC(C2(NC(=O)C(O)CC(N)=O)CSC2)=O)C1 3303,c1(CC)nc(N(CCOC)CCNC(c2ccco2)=O)cc(Cl)n1.C1C(=O)N1 3304,CC#CCC(C(=O)N1CCC(C(C)C#N)CC1)NC(=O)C(n1cc(C)cn1)C 3305,N1(C(C2(SCC)CC2)=O)CCC(C)(CCNC(=O)COc2ccsn2)CC1 3306,c1(C(=O)NCCN(C2CCCCC2)C(c2ncccn2)=O)cnc2ccsc2c1 3307,c1(C(N2C(CNC(c3c(CC)ncs3)=O)CC(O)C2)=O)cncc(F)c1C 3308,C(=O)(CCCC(F)(F)F)NC1CC(C)(C)N(C(=O)C=CCN2CCOCC2)C1 3309,C12(C(=O)NCC(CNC(c3ccccc3-n3cccc3)=O)F)CC1CCC2(F)F 3310,C#Cc1ccnc(C(=O)NC(c2cccnc2)C(=O)NCc2cccs2)c1 3311,c1(C(C)C)cc(C(=O)NC2CCC(N(C(=O)CC3CN(C)C3)C)CC2)cc(F)c1 3312,C1(CC)CC(CC(=O)NC2CC(CNC(=O)CC(C)(F)F)C2)CCO1 3313,c1(SC)cccc(CC(=O)NCCC2(CNC(=O)CC(C)n3cccc3)CC2)c1 3314,c1(NCC(C)(C2CC2)NC(C(CCCC)C)=O)cc(=O)n2cc(Cl)ccc2n1 3315,C1(c2cccnc2)CC2C(C1)C2(F)F.C1(OC(N(C)C)=O)CC1 3316,Cc1ccc(NC(=O)C(c2ccoc2)NC(=O)Cn2ccnn2)cc1CO 3317,N1(C(CN(S(CC)(=O)=O)C)=O)CC(CNC(=O)CC2CCCCC2)CC1C 3318,c1(OC)csc(C(=O)NCCN(C(=O)C(n2ccnc2C)C)CC2CC2)c1 3319,n1(C(CC)C)ncc(C(=O)NC2(CCF)CC2)c1C 3320,N1(C(c2c(OC)c(Cl)ccc2)=O)CCC2(CCN(C(=O)CN(S(C)(=O)=O)C)C2)C1 3321,C(=O)(C(C)P(C)(C)=O)NCc1c(CNC(CCNC(CC(C)C)=O)=O)ocn1 3322,N1(C(c2c(C)nsc2)=O)CC(NC(=O)CC2CC23CC3)C(c2cncn2C)C1 3323,N1(C(CCNC(c2ccoc2)=O)=O)CC2CC1CN2C(C1(O)CCC1)=O 3324,N1(CCOCCCC)CCC2(CC1)CC(C(=O)OC)C2 3325,C1(C(=O)OC)C(C(N2CCC(NC(=O)Cc3cscn3)C2)=O)C1(F)F 3326,C(CCN=C(NCC1CC(=O)N(c2ccccc2)C1)NC1CSC(C)C1)OC 3327,C12(NC(C3C(CN(C)C)C3)=O)CC1CN(C(=O)C(C)(C)c1ccccn1)C2 3328,c1(OC)cncc(C(=O)NC2CCOCC2C(=O)Nc2ccsc2C)n1 3329,C(=O)(C(C)(C)C(C)(C)C)N1CC(NC(c2c(C(C)C)con2)=O)C(F)C1 3330,C(=O)(C(C)(F)C(C)(C)F)NC(CC)CNC(=O)CCSc1ccc(C)c(C)c1 3331,C12(C(=O)NC3C(C)CN(C(c4coc(Br)n4)=O)C3)CC(C)(C1)OC21CCC1 3332,c1(NC(N2CC(N(C(CC=C)=O)CCCCl)C(C)C2)=O)cccc(C)c1F 3333,c1(C(N2CCCC(CNC(CCCCSC)=O)C2)=O)cc(F)c(F)cc1C 3334,CC1CCN(C(=O)CCc2ccccn2)C1C(=O)N(C)Cc1nc(=O)o[nH]1 3335,C1(O)(C(C)NC(=O)CCC2CCC(O)CC2)CCN(C(c2ccon2)=O)CC1 3336,C1(C)(C(N(CC(CC)(C)OC)C)=O)CCN(C(=O)Cc2cnccc2C)CC1 3337,n1(CC#N)ccc(C(N2CC(n3cc(CNC(c4n[nH]cc4Br)=O)nn3)C2)=O)n1 3338,c1(C(=O)NCc2nc(CNC(C)=O)sc2)c(-c2ccccc2)noc1C 3339,c1(SC)cc(F)c(CCNC(c2ccn(C(F)F)c2)=O)cc1F 3340,N1(C(CC2N(C)C(=O)CC2)=O)CCC2(CC1)CC2NC(C1(c2cc[nH]n2)CC1)=O 3341,C1(C(=O)NCCC2(O)CCCC2)CCCN(C(c2ccn(CCOCCO)n2)=O)C1 3342,c1(C(C(=O)N2CCCC2)NC(CC(=O)OCC)=O)c(C)cccc1Br 3343,N(C(=NCCCCC(F)(F)F)NCCSc1nc(C)cc(C)n1)CC(C=C)C 3344,C1(c2ccccc2)(CC(=O)NCCC2(O)CN(C(C34CCC3C4)=O)C2)CCCO1 3345,c1(CC(=O)NCC2CCCCN2C(=O)OC(C)(C)C)cc(F)cc(F)c1Br 3346,Cc1cccc(C(N2CCC(C)C2CNC(c2cc(=O)cc[nH]2)=O)=O)c1 3347,C1(NC(c2c(C)cns2)=O)CN(C(C2CC2c2cncn2C)=O)C2(CCC2)C1 3348,C1(NCc2nnn(C)n2)CCN(C(c2cccc(Cl)c2)=O)CC1(C)C 3349,C1(CC)CCC(NC(=O)CCCn2cncn2)CC1 3350,c1(C(N2CCN(C(CC=CC)=O)CC2c2ccncc2)=O)ccc2c(c1)CCC2 3351,c1(C(=O)NCC2(F)CCC(NC(C3(C(F)F)CC(=C)C3)=O)C2)ccc(N)c(Cl)n1 3352,C1(COC)CN(C(c2cccc(C(C)(C)C)c2)=O)CCN1Cc1ccc(Cl)nc1 3353,c1(OC)cc(CC(=O)NCC2CCN2C(=O)C(F)OC(F)(F)F)on1 3354,Cc1oc2ccccc2c1C(=O)NCC1CCCC1NC(c1cc(O)nn1C)=O 3355,N1(C(C2CCN(C(c3ccc4cncn4c3)=O)C2)=O)C2COCC1CC(F)C2 3356,c1(C(N2CCC(C)(CNC(C3C(C)C3(F)F)=O)C2)=O)n[nH]c2cccnc12 3357,N1(C(C2(CC)COC2)=O)CCC(NC(=O)CCOc2cccc(C)c2C)C(O)C1 3358,C(=O)(C(CNC(=O)Cc1nccn1C)C(C)(C)C)N(C)Cc1ccccn1 3359,CC(N=c1[nH]c(N(C)Cc2ccn(C3CC3)n2)nc2c1CCC2)c1csc(Br)c1 3360,c1(C(N(CCCCNC(=O)CN2CC3CC3C2)C)=O)ccc(F)c(N)c1 3361,c1(OC)cc(O)c(C(=O)Nc2ccc(C3CCNCC3)cc2)cc1OC 3362,c1(OC(c2oc(CC)c(C)c2)=O)cc(C2CC2)cc(F)c1 3363,N1(C(C(C)SC(C)C)=O)CC2(NC(C3CCCC3)=O)CC1C2 3364,c1(CCC)cccc(C(N2CCN(C(=O)C(C3CCCO3)OC)CC2)=O)c1 3365,C1(NC(C(CC2CCOCC2C)N(CC(=O)NCC)CC)=O)CCC(F)(F)CC1 3366,c1(C(=O)NCC23C(CN(C(c4ncnc(C)c4C)=O)C2)C3)cc2scc(C)c2[nH]1 3367,N1(C(c2c(C)coc2)=O)CCCC(C)(C)C1C(N1CCOCC1CO)=O 3368,c1(C(=O)NC2(CNC(C3C(C(N)=O)COC3)=O)CC2)ccnc(N2CCCC2)c1 3369,C=C1CC2(C1)CC(C(=O)NCC1CCCCN(C(=O)COC3(C)CCC3)C1)C2 3370,C1(CNC(C(c2ccc(OC)cc2)(C)C)=O)CC2COCC2N1C(=O)CC1CC1 3371,CC1(C(=O)NCCC2CCN(C(=O)C(C3CCCCC3)O)C2)CCS(=O)(=O)CC1 3372,C1(O)(CC(=O)NCCC(C)N(C(=O)CCN(C)CCO)C)CCOC1 3373,CC1CC(CCNC(c2csc(C(C)(C)C)n2)=O)CCN1C(=O)Cc1cncs1 3374,C1(C(=O)NC2CC(NC(c3noc(CC)c3C)=O)C2)CCc2n[nH]cc2C1 3375,N#Cc1c[nH]c(C(N2CC3C(CNC(=O)CCCc4ccncc4)C3C2)=O)c1 3376,CC(C(=O)NC1(CC(=O)NCCc2ncon2)CC1)C1CCCO1 3377,C12(CNC(COCC#C)=O)CCC(NC(=O)CCC3CCCCC3)(CC1)CO2 3378,c1(C(=O)NC2C(NC(C=CCN(CC)CC)=O)COC2)cccc(C#N)c1 3379,N1(C(C(CC(C)C)=O)=O)CC2C=CC1C(C(=O)NCc1nn[nH]n1)C2 3380,C=CC(C)(CCOC)C(=O)N(C1CCCC1)CCNC(=O)CC(F)(F)C(F)F 3381,C12(CNC(c3cn(CC)nc3)=O)CC1CN(C(c1sccc1SC)=O)C2 3382,N1(C(C(c2nc(C)sc2)=O)=O)CC(NC(c2ccc(C(F)F)nc2)=O)C(C)(C)C1 3383,N1(C(C2CC2C(N2CCCC2)COC)=O)CCC(Cn2cc(COC)nn2)CC1 3384,CN1CC=C(C(=O)NC2COCCN(C(=O)Cc3ccoc3)C2)C1 3385,c1(CN2CC(C(CF)(F)F)(C(=O)O)C2)cnn2c1OCC2 3386,C(c1cccc(Cl)c1)=C(C(N1CC(NC(C(C)(C)SC)=O)C1)=O)C 3387,CCCCC(CC)(c1nnnn1CCSC)NCCS(=O)CCSC 3388,C1(NC(c2n(CCC)ncc2)=O)CCN(C(=O)Cn2ccnc2C)CCC1(F)F 3389,N1(C(CN(C(C#C)C)C)=O)CCC(N2CC(C)(O)C2)CC1 3390,N1(C(CCc2ccnc(C)n2)=O)CCN(C)C(CNC(C2CC2(F)F)=O)C1 3391,c1(N2CC(C)C(NC(=O)Cc3ccc4c(c3)CC4)CC2)ccc([N+](=O)[O-])cn1 3392,c1(C(N2C(CN(C)Cc3c(C)ccs3)CCCC2)=O)cnc2c(c1)CCCC2 3393,CC1CC2(C(N3CC(F)(CNC(C4(Oc5ccccc5)CC4)=O)C3)=O)CC12 3394,CC1CCCN(C(C2CCS2(=O)=O)=O)C1CNC(=O)CCN1CCOC1=O 3395,c1(C(=O)NCC2(C)C(C)CN(C(C(CCSC)O)=O)C2)cc(Cl)c(Cl)cc1N 3396,C1(CNC(CCSCCC)=O)C(C)CCCN1C(c1cc(C2(C)CC2)on1)=O 3397,C(=O)(C1c2c[nH]nc2CN1C(c1cncn1C)=O)NC(C1(O)CCC1)C 3398,c1(C(N2CC(OCC)(CNC(=O)Cc3nocc3CC)C2)=O)cn(C)nc1CC 3399,N1(C(C2(C)CC(=C)C2)=O)CCC(CNC(c2cnn(C3CC3)c2)=O)C(O)C1 3400,C=CCCC(C)(C)C(=O)NCCC(C)(C)NC(C1CCCC(C(F)(F)F)C1)=O 3401,N1(C(C(C)N(C(=O)CCN2CCCCC2)CC)=O)CCc2ccncc2C1 3402,CC1CCC(NC(c2cnn(C)n2)=O)CN1C(c1cccc(Cl)c1N)=O 3403,C=C(C)C(CC(=O)NCC(N1CCCC1C(=O)N=Cc1ccccn1)=O)OCC 3404,C1(NC(C2(COC)CC=CC2)=O)COCCC1NC(=O)Cc1cn(C)nn1 3405,c1(-c2c(C(c3c(O)ccc(C)c3)=O)scn2)c(C)cc(C)c(N(C)C)c1C 3406,c1(N2CCC(=C)C2)nc(N2CCOC(C(=C)C)C2)nc2c1CSC2 3407,C(=O)(C1=CC2CCCC12)N(C1CCN(C(c2ccc3nncn3c2)=O)C1)CC 3408,C(=O)(CCCCC(=O)OC(C)(C)C)N1CCN(C(C(CC=C)C)=O)CC1CCO 3409,CCC(F)(F)C(=O)NCC1CCCC1NC(=O)Cc1cn(C2CC2)cn1 3410,CC1(CNC(=O)Cc2ccc(Cl)s2)CCCN1C(=O)CCc1cocn1 3411,C1(N(C(=O)Cc2csc(Cl)n2)C)CN(C(=O)C#CC2CC2)CC12CC2 3412,C1(CNC(c2n(C=C)nnc2)=O)CN(C(=O)C(C2CC2)N(C)C)CC12CC2 3413,c1(NC(=O)NCC(C#C)OC)cc(F)ccc1N1CCCCC1 3414,N1(C(C(C)C(F)F)=O)CC(CC(=O)NC2CCN(C(N)=O)CC2)C2(CC2)C1 3415,N1(CC(=O)NC2C3CN(C(c4n(C)ncc4Cl)=O)CC2C3)C(=O)NC(C)(C)C1=O 3416,C1(C(N2C(C(=O)NC3(CC=C)CC=CC3)CCCC2)=O)C2CCCC(=O)C12 3417,Cc1ncc(C(=O)NC2CCC(N(C)C(C3CCN(C)C3C)=O)CC2)n1C 3418,CCCC(CNC(c1cccn1C)=O)C(=O)N(CC)CC1CCCO1 3419,c1(C(C)Cc2cnn(C)c2)nnc(-c2cnsn2)n1C 3420,C1(CCNC(=O)C=CCO)CCN(C(c2cnc(N3CCOCC3)cn2)=O)CC1 3421,N1(C(C=CC)=O)CC(C)(C)OC2(C1)CN(C(c1ccc(S(N)(=O)=O)c(N)c1)=O)C2 3422,Cc1cc(=O)ccn1CC(=O)NCC1CCN1C(c1coc(C2CCC2)n1)=O 3423,C12(C(=O)NCC(C)NC(C)=O)CC(CN(C(=O)CC3CC(C4CC4)C3)C1)C2 3424,c1(C(N2CCCN(C(C3CC(OC)C3)=O)CC2)=O)nc(C)ccc1C(=O)OC.CN 3425,Cc1cc(S(=O)(=O)NCCN2CC(C)(C#N)C2)c(C)cc1-c1ccno1 3426,C=CCC(CC)C(=O)N1CCOC(CCNC(C2(CC3CC3)CC2)=O)C1 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3445,c1(C(=O)NC2CN(C(C(C)(C)N3CCOCC3)=O)C2)ccc2cc[nH]c2c1 3446,c1(C(N2CCC(NC(CC3=NNC(=O)C3)=O)C(F)C2)=O)cc(=O)n2nccc2[nH]1 3447,c1(C(=O)NC(C(C)(C)NC(C=CC)=O)C)cc2[nH]nc(C)c2cn1 3448,N1(C(CC=CC)=O)CCN(C(C2CCCN(C)C2)=O)C(c2cn[nH]c2)C1 3449,CCCC(C(=O)NCCC1CN(C(c2cccnc2-n2ccnc2)=O)C1)OC 3450,C1(NC(C(C(C)NC(=O)CC(C)=C(C)C)C)=O)CCC2(CCC2)CC1 3451,c1(C(=O)NCC(=O)N(C(C)C)CC)ccc(Nc2nc(C)cs2)c(SC2CC2)c1 3452,C(=O)(C(CCOCC)NC(=O)COC(C)CC)NCC(=C)CC 3453,CC1(CNC(C2C3(CC3)C23CC3)=O)CCN(C(=O)C=Cc2cnc[nH]2)CC1 3454,C=CCCCC(C(=O)N1CCC1(C)CCC)NC(=O)C(=O)C(C)CC 3455,Cc1nn(C)c2c(N3CCC4(CCC4)C3)nc(=NC(C)CC3CCCN3C)[nH]c12 3456,C(CNC(C1CCN(CC(C)C)CC1)=O)(C(C)C(C)C)NC(c1cc(C)ns1)=O 3457,C1(NC(C(CC#C)O)=O)CN(C(=O)C=C2CCC2)CCC1(C)C 3458,C1(CC)CN(C(C2C(C)(C)C2(C)C)=O)CCN1C(c1cc(OC)ccn1)=O 3459,c1(OCC(=O)NC2(CCNC(Cc3n(C)ccn3)=O)CCC2)cccc(F)c1F 3460,N1(C(c2cc(C)sc2)=O)CC(C)OC2(CCN(C(c3ncccc3F)=O)CC2)C1 3461,N1(C(C(C(=O)NC)(C)C)=O)CCC2(CCN(C(=O)COC3(C)CCC3)C2)C1 3462,C1(C(=O)NCCCCCN(C(C(C)CC(F)F)=O)C)CCCC(F)(F)CC1 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3552,c1(C(N2C(CCC(=O)NC(CC=C)C3CC3)CCC2)=O)ccc([N+](=O)[O-])[nH]1 3553,C(=O)(C1=NN2CCCN=C2N1)NC(CNC(=O)C=CC=C(Cl)Cl)C1CCC1 3554,C1(CNC(C2CC(O)CN2)=O)C2CN(Cc3cn(C(C)C)nc3)CC12 3555,c1(OC)ccc2c(C)c(C(=O)NC3CCC4(CC3)CC4)[nH]c2c1 3556,c1(C(N(CC(CN(C(=O)Cc2cnoc2)C)O)C)=O)ccn(CCF)n1 3557,C1(F)(CNC(c2nc(CC)oc2C)=O)CCCN(C(c2ccon2)=O)C1 3558,N1(C(=O)Cn2ccc(C(F)(F)F)n2)CCCC2CCN(C(=O)C3=COCC3)CC12 3559,CN1CCN(c2ccc(N(C(c3ccc(=N)[nH]n3)=O)C3CC3)cc2)CC1 3560,c1(CCCSCC)cn(CC(=O)N(C2CC2(C)C)C)nn1 3561,S(=O)(=O)(c1c[nH]ccc1=NC(CF)CF)NC(c1cc(C)no1)C 3562,Cc1nc(O)ccc1C(N1CCC2CCC12CNC(=O)Cc1ccsc1)=O 3563,c1(C(=O)NC(CC)CNC(c2cc(C)no2)=O)c(Cl)ccc(Cl)c1OC 3564,C1(CNC(CCCCC=C)=O)CN(C(=O)C(F)(F)C(O)CC)CCC1(C)C 3565,C(=O)(C(C)(CC)CCC)N1CCC(CC=C)(C(=O)NCc2snnc2C)C1 3566,CCS(=O)(=O)CC(=O)NC(C)C(C)NC(c1ccoc1CC(N)=O)=O 3567,C(=O)(C(CN(C)C)c1ccccc1)NCCN(CC)CC1CCCCC1 3568,C1(C(=O)NCC(=O)OCCCC)(CO)CCN(C(c2cnn(C)c2N)=O)C1 3569,C1(C(=O)NC(C(=O)N2CC(OCCCCC)C2)CO)COCCN1CC 3570,c1(C(=O)NC2C(CNC(C3(C#C)CC3)=O)C2)ccc2c(c1)CCN2S(C)(=O)=O 3571,N1(C(c2c(CC)ncnc2)=O)CC2(CCC(NC(C3CCC3C(N)=O)=O)CC2)C1 3572,C1(C)(C(=O)NCCC2(O)CN(C(c3cc(COC)[nH]n3)=O)C2)CCCC(F)(F)C1 3573,C1(C(=O)NCCCNC(C(C(C)(C)C)O)=O)CC(O)c2ccccc2O1 3574,C(=O)(C1CCc2nccn21)NCC(=O)NCc1c(C)nsc1 3575,CC1=C(C(=O)N(C2CCCC(N(C)C(C)C)C2)C)CCS1(=O)=O 3576,N1(C(C2CCC(NC(C3(OC)CC3)=O)CC2)=O)CCN2C(=O)OCC2C1 3577,c1(C(N2CCN(C(C(c3scc(C)n3)C)=O)CC2C)=O)nn(C)c2c1CCC2 3578,c1(CC)nc(O)c(C(=O)NCC(C)NC(c2oc(Br)cc2C)=O)cc1C 3579,C(CC(C)N=c1[nH]c(=NCc2ccc(Cl)cc2Cl)c2ccccc2[nH]1)SC 3580,C1(C(=O)NC(C2(CCOC)CCCC2)=O)CCN(C(c2cn(C)nn2)=O)C1 3581,CCC(CN(C)C)CC(=O)N(C1CN(C(=O)C(C)NC(C2CCCC2)=O)C1)C 3582,C(=O)(CC(C)(C)NC(C1C=CCS1)=O)N(C)C 3583,C1(O)(CN(C(COCC)=O)C)CCN(C(c2c(C)ncnc2C)=O)CC1 3584,Cc1cnc(NC(CNC(C2CC23CCOC3)=O)C2CCC2)nc1O 3585,C#CCCCCC(=O)N(C)Cc1ccc(CNC(C2(C)CC2)=O)cc1 3586,C1(NC(c2ccc(CNC(CC(C)O)=O)cn2)=O)CCCN(C)C1C 3587,c1(C(N2CC(NC(c3n(C)nc(C4CCC4)c3)=O)C2)=O)cnn2c(=O)cc[nH]c12 3588,C(=O)(CC(C)CC(C)(C)C)NCC1N(C(C(C)C)=O)CC1 3589,C(CCC)(C(O)C(=O)N1CC=CC1CF)NC(C(C)OCC#C)=O 3590,N1(C(c2c(OC)csc2)=O)CCCN(C(c2cn(CC(F)F)cn2)=O)C(CO)C1 3591,c1(C(=O)NCCC(CNC(=O)C=Cc2ccccc2)O)cccc2ccnn12 3592,C(CC(=O)NC1CC1C(N1CCC1C)=O)OC 3593,c1(CNC(c2sc(C(=O)NC3(C)CN(CC)C3)c(C)c2)=O)ccc(C)c(C)c1 3594,N1(C(C(C(CC)(C)C)O)=O)C2CCCC1CN(C(=O)C(CO)OC)C2 3595,N1(C(CN(C(C)C)C(C2CCOC2C)=O)=O)CCC2(CC1)CC2C#N 3596,C1(CNC(C2C(C(=O)OC)CC2)=O)CC2CN(C(c3cc(C)nc(C)c3)=O)CC12 3597,C(=O)(C1=C2CCN=C2NC=C1)N1CCC(N(C(=O)CS(C)(=O)=O)C)CC1 3598,C(N=c1nc(N2CCC3(CCCN(C)C3)C2)c2[nH]ccc2[nH]1)C1CCC(C)CC1 3599,c1(CC)ccc(Cl)nc1C(=O)NCCC1CCN(C(=O)N(CCN(C)C)CC)C1 3600,CC1CC(c2nn[nH]n2)CC(C)N1CC(C)(C)CO 3601,Cc1ccc(C(N2CC(NC(=O)COC3CCC(C)CC3)C2)=O)cc1CO 3602,c1(C(=O)OC)cccc(NC(=O)C(=O)NCCOc2ccc(C)cc2)c1C 3603,N1(C(CC2C(OC)COCC2)=O)CCC2(CCNC2)C1 3604,C1(CC(=O)NCC(=C)F)CN(C(c2ccnnc2)=O)C(C)(C)C1 3605,N1(C(COCCC)=O)CCC(C(=O)NCc2cn(C3CC3)nn2)C1C 3606,c1(C(=O)NC(C)C(C)NC(c2cc(C(C)(C)C)no2)=O)cnc(O)n1C 3607,c1(C(N2C(CNC(c3cc(C(F)(F)F)ns3)=O)CCC2)=O)cccc[n+]1[O-] 3608,c1(C(=O)NC2CC(c3ccccc3)(NC(C3C(C)C3)=O)C2)ccc(C2CC2)cn1 3609,CN1CCC(C(=O)N(CCNC(c2ccsc2)=O)CC2CC2)CC1 3610,c1(SC)ccc(C)c(C(N2CCOCC2CNC(c2ccc(C)c(C)c2)=O)=O)c1 3611,C(C(C)(O)CC(=O)N(C1CN(C(c2c[nH]nc2C)=O)CC1(C)C)C)OC 3612,c1(CC(=O)OC)ccc(C2CNC2)cc1.C1C(C)C(=O)NC(=O)C(=O)N1 3613,C1(C)(C(N(C(CNC(=O)CCC2CCCOC2)C2CC2)C)=O)CCCO1 3614,C(=O)(C(C)(C)C(C)(C)O)N1C(CNC(c2cccc(COC)c2)=O)CCC1 3615,c1(OC)nc(NC(c2ncn3ccccc23)=O)nc2ccccc12 3616,c1(C(N(C2CCCCC2)CCNC(C(c2ccccc2)C)=O)=O)nsnc1O 3617,Cc1nc(N2CC3CC(NC(c4cc(=O)cc(Cl)[nH]4)=O)CC3C2)cc(C#N)n1 3618,C(CC(CC)C(=O)NC1C=CCC(C(=O)N(CCN2CCOCC2)CC)C1)=CC 3619,C1(CNC(c2n(C(C)C)ccc2)=O)CCC2CN(C(C3CN(C)C(=O)N3)=O)CC12 3620,C(=O)(C(CNC(c1cc(C2CC2)no1)=O)C(C)(C)C)NC(c1nn[nH]n1)CC 3621,N1(C(CCCC(C)NC(=O)OCC(C)(C)C)=O)CC2(CCCCC2)CC1C 3622,C(=O)(C1CNC(=O)c2ccccc21)NCC1C2CN(C(C(N)=O)=O)C1CCC2 3623,C=CC(O)(C(=O)NC1CCCCC1N(C(=O)CSc1ccccc1)C)C(F)(F)F 3624,c1(OC)cc(C)c(CC(=O)NCCN(C(=O)C(N2CCCCC2=O)C)C2CC2)o1 3625,C1(CNC(CC(C)C)=O)CC(NC(C2CC(C)(C)CO2)=O)C(O)C1 3626,C1(CN(C(C2(CCOCC)CCCC2)=O)C)CN(C(=O)C(=O)NOC)CCO1 3627,n1(CC(=O)N(CCCCCNC(C2CC2Cl)=O)C)ccc([N+](=O)[O-])n1 3628,CCC(CNC(C1CN(C(=O)C(C)CC#N)CC(C)O1)=O)CC(C)C 3629,C1(C(F)(F)F)CC(=O)N2CC(C2)O1.C1(c2ccc(F)cc2)(COC)CCOCC1 3630,N1(C(=O)CC(F)(F)c2ccccn2)CCC2(CC1)CC(F)CO2 3631,C1(NC(C2CN(C)C2)=O)CCN(C(=O)CCNC(N)=O)CCC1c1ccccc1 3632,C=CCC(CC(C)C)C(=O)N(C(C)CCNC(=O)Cc1nsc2ccccc12)C 3633,N1(C(C(C)CSC(F)(F)F)=O)CC2CCN(C(c3nnn4c3CSCC4)=O)CC12 3634,c1(C(=O)NC2C(CNC(Cc3nc(C)sc3C)=O)CCCC2)cccc(Cl)c1N 3635,C1(NC(c2ccc(CC)nc2)=O)CC(O)CN(C(=O)Cn2cc(F)ccc2=O)C1 3636,C(CC(O)C(F)(F)F)NC(C(CC=CC)NC(=O)CC1CCOC1=O)=O 3637,C(=O)(C1=COCCC1)NCC(C)(F)CNC(C1CN(CCF)CCO1)=O 3638,N1(C(C2CCCC(OC)C2)=O)CCC2(CC1)CCN(C(C1CC1C)=O)CC2 3639,CCC(C)C(CC(=O)NCC(C)(O)C1CCCC1)NC(c1c[nH]c(=NC)o1)=O 3640,N1(C(CCC2C(C=C)C2)=O)CC2CC(NC(c3cnc(C4CC4)o3)=O)CC1C2 3641,c1(C(=O)NC(CNC(C(C(C)C)n2cccc2)=O)CO)cn2cnnc2cn1 3642,c1(CC(C)C(=O)NC(C)(C)C)ccc(F)cc1.c12ccc(o1)COCCNC2=O 3643,N1(C(C2(CC#C)CCCOC2)=O)CCC2(CC1)CC2CNC(=O)CCOC 3644,C(=O)(CCN(OC)C(=O)c1ccc(C#N)[nH]1)N1C(C)=CCC1 3645,N1(C(CC(c2ccc(C)cc2)C)=O)CCCC(C)C1CNC(C1CCCCC1)=O 3646,C1(F)(CNC(c2c(CC)non2)=O)CCN(C(=O)C(C2CCCCCC2)O)C1 3647,C1(C(=O)NCC)CCC(C)(C)N(C(=O)Cn2cc(COC3CC3(F)F)nn2)C1 3648,CC1CC2(CCO1)CC2C(N1CC2CC(NC(c3c(N)cnn3C)=O)CC1C2)=O 3649,c1(C(N2CCC(OCCNC(c3c(OC)nccc3)=O)C2)=O)c(C)cnnc1O 3650,N1(C(CCCC(N)=O)=O)CCC2CN(C(=O)C=CC(N3CCOCC3)=O)CC12 3651,N1(C(C2(N(C)C)CC2)=O)CC(NC(C2(c3cccc(Cl)c3)CC2)=O)CC(C)(C)C1 3652,N1(C(C(=O)N(CC(=C)C)CC)C(CC)CC)CC2CN(C)CC(C1)O2 3653,Cc1c[nH]c(C(N2CCOCC2CCNC(C2(C(F)(F)F)CCC2)=O)=O)cc1=O 3654,C(c1cscn1)=CC(=O)N(C1CCN(C(c2sccc2CO)=O)C1)CCC 3655,c1(C(N(CCNC(C=C(CNC(C)=O)C)=O)CCC2CC2)=O)ccnc(C)n1.C 3656,c1(NCC(C)NC(C2(OC)CCCC2)=O)ncnc2ccccc12 3657,c1(C(=O)NCC#CCNC(=O)C2=CCCS2)coc2c(Cl)cccc12 3658,Cc1nc2cccc(C(=O)NC3CC(NC(c4cc5sc(C)nc5[nH]4)=O)C3)n2n1 3659,CCC(C)C(O)C(C)C(=O)N(CCC(N1CCCC(O)(CC)C1)=O)CC 3660,N1(C(c2cc(CC)c(CC)o2)=O)CCCC(CO)(NC(=O)CN(C2CCC2)C)C1 3661,c1(C(N2CCCC(C(=O)NC3CC34CCC4)C2)=O)cn2c(n1)CCC2 3662,N1(C(CONC(C2CN(OC)C(=O)C2)=O)=O)CCN(C)CC(O)C1 3663,C1(C(=O)NC(CN(C(c2cnc(CC)s2)=O)C)C)(OC)CCC(F)(F)CC1 3664,Cc1cc(C)c(C(N2CC(NC(c3cncc4ccsc34)=O)CC2C)=O)cc1C 3665,C1(NC(c2n(CC)ccc2)=O)CN(C(=O)C=CC2CCCO2)CC2(CCC2)C1 3666,N1(C(C)C)CCCC1CC(=O)NC(C)CCCNC(=O)CCc1cc[nH]n1 3667,c1(NC(C(=O)NCCC(=O)NC2CCC2O)=O)ccc(Br)cc1 3668,N1(C(C(CC)C(C)C)=O)CC2CCCC(NC(C3CCCS(=O)(=O)C3)=O)C2C1 3669,c1(C(=O)NCC(COC)NC(c2c[nH]nc2C)=O)ccc2n[nH]cc2c1Cl 3670,n1(CC(=O)NCCc2ccc(F)cc2F)ncc2cccc(Br)c2c1=O 3671,c1(OC)c(Cl)ccc(C(=O)NC(C)CNC(C2CCS(=O)(=O)CC2)=O)c1N 3672,N12CCC(CC1)CC(=O)OC2.c1(C(CC(C)(C)C)O)ccc(O)cc1 3673,C(=O)(C(O)CCS(C)=O)NC(C1CCCCC1)CNC(CCCCOC)=O 3674,N1(C(CC(C)c2ccco2)=O)CCN(C(=O)CNC(C2CCCS2(=O)=O)=O)CC1 3675,c1(C(N(C2CCCC(NC(c3cc(C)oc3C)=O)C2)C)=O)cnc2n1CCCC2 3676,N1(C(C(C2CC(F)(F)C2)OC)=O)CCC2CC(C1)CN(C(=O)Cc1cnc(C)s1)C2 3677,C1(C(=O)NCC(CCC)OCC)CC2CCC1N2C(=O)CCS(N)(=O)=O 3678,C(=O)(C(CNC(=O)C=Cc1ccncn1)CC1CCCC1)NC1C(C(N)=O)CCC1 3679,N1(C(C2(CC)CCCCC2)=O)CCC(O)(CCNC(=O)Cc2cn[nH]c2)CC1 3680,Cc1ncccc1N(C(N1CCC(Sc2ccc(Br)cc2)C1)=O)CC1COC1 3681,C(=O)(C#CC1(C)CCCO1)NC(C1CC1C(=O)NC1(C)CCCC1(F)F)C 3682,CC1(C)OC(=O)NC1C(N1CCCC(C(=O)Nc2ccc(F)cc2)C1)=O 3683,N1(C(C(CC)=O)=O)CCC(C)(C(=O)Nc2cnc(C(C)(C)C)nc2)C1 3684,C1(NC(C(CC)(C)O)=O)CN(C(=O)CCn2ccnc2C)CC(C)(C)C1 3685,N1(C(c2nc(C)nc(O)c2)=O)CC2(C1)SCCC2NC(=O)C1=CS(=O)CCC1 3686,c1(C(N2C(C(CNC(c3c(CCC)occ3)=O)(C)C)CCC2)=O)[nH]cnc1C#N 3687,C(=O)(C(C(=O)N(C1CCN(C(=O)C(c2cccc(C)c2)(C)C)C1)C)OC)OCC 3688,N1(C(CCc2cnc(C)o2)=O)CCN(C(C2CCCC2C(F)(F)F)=O)CC1CO 3689,C(=O)(CC1CCc2ccccc21)NCCCNC(=O)CCOCC1CCCO1 3690,c1(C(c2n(C3(C)CC3)nnn2)NCCC2CCCOC2)cc2cc(Cl)cnc2o1 3691,CC1CCCN(C(C2(n3nccn3)CC2)=O)C1CNC(=O)CC(C1CC1)C1CC1 3692,N(C1CN(C(C2(c3ccno3)CC2)=O)Cc2ccccc21)C(c1c(C)ocn1)=O 3693,Cc1cc(F)cnc1C(c1nnnn1C1CCCCCC1)NC1C(C)C1(C)C 3694,C1(NC(CCCc2n(C)cnn2)=O)CC2C(NC(=O)Cc3ccccc3O)C2C1 3695,c1(N2CCC(NC(c3c(C)ccs3)=O)C(C)C2)nc2ccc(Br)cc2o1 3696,c1(COCC(=O)NC(CNC(c2c(OC)n[nH]c2)=O)(C)C2CC2)nnc(S)n1C 3697,C1(C(N(CC(CNC(c2c(CC)cns2)=O)C)C)=O)(CO)CC(C)(C)C1 3698,Cn1ncc(C(=O)NCCCOCCC(=O)NCC2C(C)(C)C2(F)F)c1Cl 3699,n1(CC(=O)NCC2CCC2NC(=O)C(=O)N2CCC2)ccc(Br)cc1=O 3700,CC(C)(C(=O)NCC1CC1CNC(=O)COCP(C)(C)=O)n1cccn1 3701,N1(C(C2(C#C)CC(=O)C2)=O)CCCC(C(=O)NCC(C)CC2CCC2)CC1 3702,c1(OC)cc(OC)cc(OCC(=O)NCC(O)CSc2cc(F)ccc2Cl)c1 3703,N1(C(c2c(C)oc(-c3ccc(OC(F)(F)F)cc3)n2)=O)CCC(O)C(F)(F)C1 3704,C1(CNC(C2(C(=O)OCC)CCC2)=O)CCN(C(=O)C(F)(F)c2ccncc2)C1 3705,C(=O)(CCS(=O)(=O)N(C)C)N(CC(O)CN(C(=O)CC(F)(F)F)C)C 3706,O(NC(=O)C(C(C)NC(c1cn2c(n1)CCC2)=O)C(C)C)C(C(=O)OC)(C)C 3707,CC(C)(C)C(C(=O)NC1CCN(C(C2CCCCNC2=O)=O)CC1)NC(N)=O 3708,N1(C(C2C(CNC(C=Cc3cc(C)no3)=O)C2)=O)CC(CO)CC(C)(C)C1 3709,C(CCC(C)C)(C(=O)N1CCC(O)(C(=O)NC23CC2CNC3=O)CC1)OC 3710,N1(C(C(C(C)(C)C)F)=O)CC2(CCC(CNC(C3(Cl)CC3(F)F)=O)O2)C1 3711,c1(-c2cn(CCCNC(c3cc(C4(C)CC4)n[nH]3)=O)nn2)ccc(O)nn1 3712,c1(NC(=O)Nc2cc(C)c(I)cn2)cc(O)c2c(C(C)(C)C)n[nH]c2c1 3713,c1(C(N2CC(COC)(CNC(=O)CNS(C)(=O)=O)C2)=O)cc(F)cc(F)c1O 3714,N#Cc1cc(C(N2CCN(CC(N3CCC(CO)C(O)C3)=O)CC2)=O)ccc1Cl 3715,N1(C(C23CCC(OC)C2C3)=O)CC2CCCC(C1)N2C(=O)CCc1cnoc1 3716,c1(OC)ccc(C)cc1NC(C1CCN(C(=O)C2=COCC2)C1(C)C)=O 3717,C=CC1(C(N2CCN(C(c3cc(C)ns3)=O)C(CCC)C2)=O)CCOCC1 3718,CC(CC(=O)N1CCCCC1C(N)=O)C(C)(C)NC(=O)Cn1cnnc1O 3719,C(=O)(CC(C)(CN(C)C)C(F)(F)F)N1CCC2(CCN(C(C3C(C)C3C)=O)C2)C1 3720,N1(CC(N2C(CNC(Cc3ncc(C)s3)=O)CCC2)=O)CCN(S(C)(=O)=O)CC1 3721,c1(CCC(=O)NC2(CNC(c3cc(C)nc(C)n3)=O)CC2)cc2ccccc2[nH]1 3722,c1(C(=O)NC(c2ccc(I)cc2)C(=O)NCC(=C)C)ccc(OC)c(F)c1F 3723,c1(C(N(CCCOCCNC(=O)CCn2ccnn2)C)=O)cc(C(C)(C)C)c[nH]1 3724,C=CCCN=C(NCc1cc(Cl)cn1C)NC1CCOC(c2ccccc2)C1 3725,C1(C(NC[Si](C)(C)C)=O)CCOC2(CCC2)C1 3726,C=CC1CCN(C(C2(NC(C3CC4CC4C3)=O)CC(O)C2)=O)C1 3727,c1(OC)ccc(CNC(=O)NCC2CCCC(F)C2)nc1 3728,N1(C(Cc2cc(C)sc2)=O)CCCC(CN(C)C(C2CC(F)C(=O)N2)=O)C1 3729,C1(SC)CCCC(N=c2cc(NCCc3c[nH]nc3C)nc(C(C)C)[nH]2)C1 3730,N1(C(=O)COCCF)CCC(F)(C(N2CCC(F)(CO)C2)=O)CC1 3731,C1(CCC(=O)NCC(C)(C)NC(CN(C)C2CC2)=O)CCN(C)C1 3732,CC1CN(C)CC(C(=O)NC(C)C(N2CC(O)(CC(N)=O)C2)=O)O1 3733,CCC(CC)C(=O)NC1CCC(NC(=O)CNC(=O)CCC2CC2C)C1 3734,C12(NC(CC=C)=O)COC(CNC(=O)Cc3ccc(C(=O)C(C)(C)C)s3)(C1)C2 3735,c1(CC)ccc(C)c(C(N2CC3(C2)CN(C(=O)C(c2ccc(Cl)s2)C)C3)=O)c1 3736,N1(C(c2c(OC)n(C)nc2C)=O)C2CCC1CN(C(C1CN(CC(C)C)C1)=O)C2 3737,c1(C(N2CCN(C(C3(C)C=CCCC3)=O)CC2)=O)ccc2ocnc2n1 3738,C12(C(=O)NCCC(C(C)C)OC)CC1CN(C(=O)C(C)C(F)F)C2 3739,c1(C(=O)NC(C)CC2CN(C(C3(CO)COC3)=O)C2)cc(Br)cnc1O 3740,c1(CC(N2CC(O)(CN(C)C(c3ccoc3Cl)=O)C2)=O)cnccc1C(=O)O 3741,c1(OCC)ccc(CNC(=O)CC23CC(NC(=O)C=C(C)C)(C2)C3)cc1OC 3742,c1(OC)cccc(OC)c1C(=O)NCCC1CCCN(C(=O)C(C(C)C)OC)C1 3743,c1(OC)ccc2nc(N3CCC4(CCC(CNC(=O)COC5CC5)O4)CC3)sc2c1 3744,CN1C2CCC1CC(=CC(=O)NCC1CCN(C(C3(O)CC(C)(C)C3)=O)CC1)C2 3745,c1(C(=O)NCC2CCC(C(N(CC=C)Cc3ccco3)=O)O2)c(C)noc1C 3746,c1(-n2cc(CCN(CC)CC)nn2)ccc(C(F)(F)F)cc1.C(=O)(C(C)O)N 3747,c1(C(C(=O)NCc2ccccc2Br)N(C2CCNC2=O)C)cc2n(n1)CCCC2 3748,CCC(C)(C)CC(=O)NC1(CO)CCN(C(c2csc3cncn23)=O)C1 3749,C1(CC(=O)N(C)CCC2CCCO2)COCCN1C(c1nocc1Cl)=O 3750,c1(C(N(C2CCN(C(=O)CCC3CC(C)C3)C2)CC)=O)ccc2nc(O)[nH]c2c1 3751,C1(C(N(CC(F)(F)F)CC)=O)C2C(CN1Cc1cccc(C(=O)OC)c1Cl)C2(C)C 3752,c1(C(=O)NCC2(CNC(CCC(=O)OCC)=O)CC2)ccc(C)cc1OC 3753,C(=O)(C1CCc2c[nH]nc21)NCC1(C)CCN(C(C(CCCC)O)=O)CC1 3754,C1(NC(C2(C)CN(C(C(C=CC)O)=O)C2)=O)CNC(=O)OC1 3755,c1(NC(=O)NC(CCCC#C)c2ccccn2)ccc(F)c(C)c1F 3756,N1(C(C2CC(C)N(C)C2)=O)C2CCC(C(=O)NCCC(C)c3cn[nH]c3)C1CC2 3757,C1(F)(C(=O)NCC2CCCC(CNC(C(C)NC(C)=O)=O)C2)CCC2(CC1)CC2 3758,c1(C(CC)C)ccc(NC(=O)Nc2cccc(C(=O)NC3CC3)c2)cc1 3759,c1(C(N(CCNC(=O)C(C)S(N)(=O)=O)CC)=O)c(OC)ccc(F)c1N 3760,C(C(CC(C)C)C(=O)NCC1CN(C(c2coc3ccccc23)=O)CC1O)OC 3761,c1(OC)cc(OCCNC(c2ccncc2)=O)cc(S(N)(=O)=O)c1 3762,C#CCC1CC(=O)N1.C(=O)(CC(=O)OC(C)C(=C)C)OC(C)(C)C 3763,Cc1nn(C)c2nc(N3CC4CC(C)C4C3)c(C#N)cc12 3764,C1(C(=O)NCCC(CC)(F)F)CC2(CCN(C(=O)C(O)CC(C)(C)C)C2)C1 3765,CCCC(CC1CCCCC1)C(=O)NC1CCCC1NC(c1coc(C)c1)=O 3766,C1(NC(c2cn(CCNC(C(C(C)(F)F)F)=O)nn2)=O)CCn2nnnc2C1 3767,c1(-c2ccc(C)o2)ccc2ccnc(NC(c3ccn(C(F)F)n3)=O)c2c1 3768,Cc1cc(C(=O)NC2CCC2NC(=O)C(C)N(C)C)ccc1O 3769,CC1(C)COC(CC(=O)NCC2CC(NC(C3(CO)CCCC3)=O)C2)CO1 3770,C1(NC(CC(N(C)C)C2CC2)=O)(CF)CCN(C(=O)Cc2cnc[nH]2)C1 3771,c1(CC)cc(C(=O)NCC(CO)NC(c2ccnnc2O)=O)c2c(c1)CCO2 3772,c1(OCC)cc(NC2CC3CCCC(C2)N3C(=O)CSSC)ccc1[N+](=O)[O-] 3773,C1(C(N(CCOC)C2CC2)=O)CN(C(=O)C(C)C(F)F)CCO1 3774,Cc1ccc(C(C)NCCC(C2(O)CCOCC2)C)cc1C#N 3775,C(c1cccc(F)c1)=C(C(=O)NC(C)CNC(=O)CC1(CN(C)C)CCCC1)F 3776,c1(NC(=O)OCC)ccc(C(=O)NCC(C)(CO)NC(=O)CCC(C)C)cc1 3777,C(C)(CC(C)(C)O)NC(C=C(C)CNC(C1CN(C(C)C)C1)=O)=O 3778,CC1CC2(CCN(c3nc(N4CCC5(CC4)CC(O)C5)nc4c3SCC4)C2)CO1 3779,C1(C(N(C)CCc2ccccn2)=O)C2CC1N(C(=O)Cc1ccn(C)c1)C2 3780,C(CCCC(C)C)(c1n(C(CC)C)nnn1)NCc1nnn(C(C)(C)C)n1 3781,N1(C(c2ccc3nonc3c2)=O)CC2CCCC(C1)N(C(C1CC(O)C1)=O)C2 3782,c1(C(=O)NCCN(C)C(C2(C)CCOCC2)=O)sc2cccnc2c1Cl 3783,N1(C(=O)CCC2CCCCC2)C2CCC1CC(C(N1CC3(COCCO3)C1)=O)C2 3784,c1(C(N2CC3(N(C(C(C(C)C)F)=O)CC3)C2)=O)ccc2ncn(C)c(=O)c2c1 3785,CCC(CC(=O)NCC1CCN1C(=O)CNC(=O)Nc1ccncc1)C(C)C 3786,N1(C(C)(C)C)CCC2C(C(N3CSCC3C(=O)O)=O)C2C1.N12CC(C1)CC2=O 3787,C1(NC(CCCOC(C)=O)=O)C2CC3C1C3C2C(=O)NC1(C)CCCC1C 3788,C1(N(C)C)CCN(C)C(COC(c2cc(Br)ccc2OC(F)(F)F)=O)C1 3789,C1(C(=O)NCCCN=[N+]=[N-])CN(C(=O)CCOCC2CCC2)CC12CC2 3790,C=CCC(C(=O)NC(C1CC1C(=O)OCC)C)Nc1cccc(OCF)c1 3791,CC(C)C(O)C(F)(F)C(=O)N1CC(O)(CN(C)C(c2cc(N(C)C)ccn2)=O)C1 3792,n1(CC)c(CC(N2CC(N(C)C(C3CC4C=CN4C3)=O)C2)=O)nc2ccccc12 3793,C(N=c1[nH]c(N(C)Cc2ccc(Br)nc2)nc2c1CSC2)C1(OC)CCOCC1 3794,N1(C(C2N(C(C)=O)CCC2)=O)CCCCC1CCC(C)(C)NC(=O)C=NOC 3795,CC1CN(c2ccnc(NCC3CCCCN(C)C3)n2)CC(C)O1 3796,C1(CCN(C)C(c2cscn2)=O)CCCCN1C(C1CCCC1(C)C)=O 3797,C(=O)(C(C)CC(=O)N1CCN(Cc2ccc(Cl)cc2OC)CC1)OC 3798,c1(C(=O)NCCCN2CCN(C(C3C(OC)CC3)=O)CC2)cccc(=S)n1O 3799,C1(C(=O)N(CCCNC(c2csc(C(C)(F)F)n2)=O)C)(COC)CC1(F)F 3800,N1(C(C(C(C)C)NC(CC(C)C)=O)=O)CCC2(CCN(C(=O)C(=O)N(C)C)C2)C1 3801,c1(C(=O)NC2C(OC)CN(C(=O)CCc3csc(=N)[nH]3)C2)cc(C)nc(C)n1 3802,CC(C)(C)C(C)(C)C(=O)N1CCOC(C2CN(C(=O)CCP(C)(C)=O)C2)C1 3803,Cc1ccc(CCCNC(CC2CCC2)C2CC2)c(C)c1 3804,C(C)(C1=CCN(C)CC1)NC(C(c1cn(C)nn1)NC(c1[nH]cc(C)c1)=O)=O 3805,c1(C(=O)NCC(C)CNC(c2n[nH]c3c2CCC3)=O)cc(O)nc(Br)c1 3806,C1(C(N(CCCN(C(=O)C=CCO)C)C)=O)CC(=O)N(c2ccccc2F)C1 3807,CCC1=C(C(=O)NC(C)CCCCNC(c2ccc(C)nc2N)=O)CCCO1 3808,c1(C(=O)NC2CCC(CCC(=O)NC(C#C)(C)CC)C2)cnc(C)n1C 3809,c1(C(=O)NC2CC3(C(NC(C(C)NC(C)(C)C)=O)C3)C2)cc(Cl)ccc1[N+](=O)[O-] 3810,c1(C(=O)NC(CNC(C2N(C)CCC2)=O)(C)C)ccc2c(=N)[nH]cnc2c1 3811,CC(=O)CCCC(=O)NCC12CC1CN(C(=O)COc1ccc(F)nc1)C2 3812,n1(CCC)cc(C(N2CCOC(C(C)NC(=O)C=C(C)C(C)(C)C)C2)=O)c(C)n1 3813,c1(NC(=O)Nc2c(SCC)cc(Br)cc2)ccc([N+](=O)[O-])cc1Cl 3814,c1(C(=O)NCC2C(NC(C3(CC)CC3)=O)CC2)ccccn1.C1C(=O)N1 3815,c1(C(=O)Nc2ccc3ncc(C(=O)OC)n3c2)cc(COC)c2c(c1)CCO2 3816,CCC(C)(C)CCCC(=O)NC(CN(C)C(c1cc[nH]c(=NC)c1)=O)(CO)CO 3817,c1(CC(=O)N(CC(=O)N(C(C)C=C)CC)CC#C)cncnc1 3818,c1(C(=O)NCC2C(N(C)C(C3(C)CCC3)=O)C2)ccc(C(F)(F)F)c([N+](=O)[O-])c1 3819,C1(C(=O)NC(CC(=O)NCC(CCC)C)COC)CC2CC1CC2=O 3820,C(=O)(C1=CCCN(C(=O)Cc2ccccc2O)C1)NCc1cc(C#N)ncc1 3821,CC1CN(C(=O)CSCC(N)=O)CCC1CNC(c1ccnn1CC(F)F)=O 3822,c1(OC)cccc(C(=O)NCCC2CC(NC(=O)C(C)CS(C)=O)C2)c1C 3823,C#Cc1ccc(F)c(C(N2CCCC(CCNC(C3CCC(=O)C3)=O)C2)=O)c1 3824,N1(C(CCOC(C)=O)=O)CCC(O)(C2CCN(C(=O)C(C)=C(C)C)CC2)C1 3825,CN1CC=CCC1C(N1CCC(CC(=O)NCC2CCC(=O)N2)C1)=O 3826,N1(C(CCC=C)=O)CCCC(C2CCCN(C(=O)CCc3cncc(F)c3)C2)C1 3827,N1(C(C(C)N(C(C)=O)C)=O)CC(O)(C(C)NC(=O)Cc2cnsc2)C1 3828,CC1CN(C(=O)CC2C=CCC2)C1C(=O)NCC(C)(C)CC1CC1 3829,C#Cc1ccc(C(=O)NC2CCN(C(C3NC(=O)CC3C)=O)CC2)cn1 3830,c1(NC(CNC(CNC(=O)CN2CCSCC2C2CC2)=O)=O)ccc2ccoc2c1 3831,c1(C(N(CC2N(C(CCC=CCC=C)=O)CCC2)CC)=O)cn(C)cc1C 3832,N1(C(C(=O)NCCSCC)c2cccs2)CCOC(C2CC2)CC1 3833,c1(C(C)(C)C)cc(C(N2CCC(C)(NC(=O)Cc3ccoc3)C2)=O)ccc1O 3834,c1(OC)c(C(=O)NCCCNC(=O)COC(F)F)ncnc1C 3835,C(=O)(C(C)COC)NC(C(=O)N(CCC)CCO)c1cccs1 3836,c1(OC)ccc(F)cc1CC1CCCCC1C(N1CCCC(Cn2cccn2)C1)=O 3837,C1(N(C(=O)C(O)CC)CCC)CCN(C(c2csc(C)c2Br)=O)CC1 3838,C12(CNC(C34CC(C)C3C4)=O)CC1CN(C(C1(CO)CC(C)(C)C1)=O)C2 3839,c1(C(N2CCC(F)(CNC(CCOCC#C)=O)C2)=O)cc2ccncc2s1 3840,N1(C(C2(NC(C34CCCC3C4)=O)CCC2)=O)CCCC(C(=O)O)C1.N1(CC)CCOCC1 3841,N1(C(C(=O)NCC)=O)CCC2(CCCN2C(=O)C(O)CC(C)(C)C)C1 3842,n1(CCC(N2CCC(O)(CNC(C3C(C)C3C)=O)CC2)=O)ccc2cccnc12 3843,CC(C)CC(F)C(=O)NC1(C2CN(C(=O)Cc3cc(-c4ccco4)on3)C2)CC1 3844,C1(NC(c2ccc(-c3ccco3)[nH]2)=O)CC2CC(NC(c3cccnc3)=O)C2C1 3845,C=CCCC(C)NC(C1CCCC1CNC(C1CN(C)C1)=O)=O 3846,C(=O)(C(N=[N+]=[N-])C(C)C)OC.C12(C)CC(O)CN1C2=O 3847,CC1(C)OCC2CC12C(N1CCN(CCCNC(=O)CC2=CCCC2)CC1)=O 3848,Cc1nc(CNC(C2CCOC2C(C)NC(=O)CNC(C)C)=O)sc1CC1CC1 3849,c1(CN2CCC(OCCOCC)C2)ccc(Br)c(C)c1O 3850,C(=O)(CS(=O)C(F)(F)F)NC(CNC(c1c(CC)ocn1)=O)C1CCC1 3851,CC#CCC(C(=O)Nc1ccc(CC)nc1)NC(=O)CCn1cncn1 3852,CCCCCC(O)C(=O)N1CCC2CC12C(=O)NCC1C=CCCC1 3853,N1(C(C(C=CCCC)O)=O)CC(CNC(C2(C3CC3)CC2)=O)CC1(C)C 3854,C(=O)(C(C(C1CCC1)OCC)N(C1CC1)C1CC1)NCC 3855,c1(C(=O)NCC2(C)CCC(NC(COCCOC)=O)C2)cc([N+](=O)[O-])ccc1N 3856,C1(COCC(=O)NC2CCCOC2)CCCNC12CC2 3857,C1(CC=C)(NC(C2CCS(=O)(=O)C2)=O)CCN(C(C2CCCNS2(=O)=O)=O)CC1 3858,Cc1cc(C)c(C(=O)NC2CCN(C(=O)NCc3ccccc3C)C2)c(Cl)n1 3859,CC1(C)OC(=O)NC1C(=O)NCC1CCCN1C(C1CCCCC1C(F)(F)F)=O 3860,c1(C(=O)OC)cccc(Br)c1NC1CCN(C(=O)C(C)CC(F)F)C1 3861,Cc1onc(CO)c1C(=O)NCCCN(C(=O)C=C(Cl)Cl)CCO 3862,C(=O)(C#CC1CCOCC1)NCC1C(C)CCN(C(=O)C=CC(C)(C)C)C1 3863,CC(C)C(C(=O)NCC1(NC(C2(C)COC2)=O)CCOC1)c1ccn(C)n1 3864,C1(C(C)C(=O)NCC(CO)NC(c2ccon2)=O)CCC(=O)N1 3865,CC(C)C(CCNC(c1nnnn1C1CCOCC1)c1nccs1)N(C)C 3866,c1(OCC(=O)NC(CCNC(CC(=C=C)C)=O)C)ccc(C)cc1C(F)(F)F 3867,C1(C(N2C(C)CC2NC(c2cc(O)n(C)n2)=O)=O)CCc2ccccc2C1 3868,C12(C(=O)NCCCC(C)(C)OC)CC(CN(C(c3nn(C)cc3Cl)=O)C1)C2 3869,C1(CNC(COCCC)=O)CC2(CC2)CN1C(c1cn(C2CCOC2)cn1)=O 3870,Cc1ccccc1NC(C1CCOC1NC(C1CCC1C#N)=O)=O 3871,c1(C(N(CC#CCNC(=O)CNC(c2ccsc2)=O)C)=O)cc(O)nc(O)n1 3872,C=CC(C)(CC)C(=O)N(CCCNC(c1ccc(C(=O)OC)nc1)=O)CCO 3873,c1(C(=O)NC(C2CC(F)CN2C(=O)CC2COCCO2)C)ccnc(C(C)(C)C)c1 3874,C12(CNC(=O)OC(C)(C)C)CCC1CCN2C(C1CCC(C)CC1)=O 3875,C(=O)(CCCCN=[N+]=[N-])NC1CN(C(C(CC=C)(F)F)=O)CC1CC1CC1 3876,C1(CCC)(C(=O)NCC(c2cccc(Cl)c2)NC(c2ccco2)=O)CCNC1=O 3877,Nc1cccnc1C(=O)NCC1CCCCC1C(=O)NCc1ncc(CO)[nH]1 3878,C(=O)(CC(C)C(F)F)NC(C(=O)N(CC(CC)(O)CC)C)COC(C)C 3879,C=CCC(CNC(C1(CC=C)CCCC1)=O)NC(C1(c2cc[nH]n2)CCC1)=O 3880,C1(NC(Cc2nn(C)nc2Br)=O)CN(C(C2CCCN2C=O)=O)CCC1CO 3881,C(CCCCCN=c1[nH]ccnc1C(=O)OC)NC(C(C)SCC)=O 3882,c1(C(=O)OCC)c(NC(=O)NC2CC2c2ccc(Cl)c(Cl)c2)sc2c1CCSC2 3883,C=CCC(C)(CNC(C1(C)CCN(C(=O)C(C(C)C)OCC)CC1)=O)CO 3884,c1(CC)cccc(C(=O)N(CCNC(=O)CCc2ccn(C)n2)C2CC2)c1 3885,C#CC1CCCN1C(C1(CC=C)CN(C(c2c[nH]c(=N)o2)=O)C1)=O 3886,N1(C(C(COCC)C)=O)CCSCC1C(=O)Nc1ccc(Cl)nc1 3887,C1(NC(C2(OC)CC2)=O)CC(O)CN(C(c2cnc(C3CCC3)s2)=O)C1 3888,C1(CSCC(=O)N(CCCNC(C2N(CC)CC2)=O)C)CCCCO1 3889,Cc1nsc(NC(C2CCN(C(=O)CCC3(O)CCC3)CC2)C)c1C#N 3890,N1(C(C2CN(C)CC2C(F)(F)F)=O)CCCC(NC(C2(CF)CCC2)=O)CC1 3891,N1(CC(C)NC(=O)CS(=O)(=O)N(C)C)CCN(C(=O)CC2COC(=O)C2)CC1 3892,C1(N(C(C=C(CC)C)=O)C)CCCCN(C(c2cn(C)c(O)n2)=O)C1 3893,Cc1c(F)cc(C(N2CCC(C(N3CC(C#N)C3)=O)C(O)C2)=O)cc1F 3894,N1(C(COC(C)C)=O)CCC2CCCN(C(c3c[nH]c4ccc(Cl)cc34)=O)C2C1 3895,C1(CN(C)C(c2sccc2C2CC2)=O)COCCN1C(C1CCCNC1=O)=O 3896,c1(OC)cc(CN(C(=O)NCC23CC(CN2)C3)C2CC2)ccc1O 3897,c1(C(N(CCN(C(C(C)OCC)=O)C)C)=O)cc(Cl)cnn1 3898,CC1=CCC(C(=O)NCCCCN(C(=O)CCSc2nccn2C)C)CC1 3899,C1(OCCC)CCCN(C(=O)CCOCc2nc(OC)cc(OC)n2)CC1 3900,c1(N2CC(CC#N)N(C(C3CC3N)=O)CC2)ncnc2ccc(F)cc12 3901,N1(C(CC=C)=O)CCCC(CC)C1C(N1CCC(CCSC)CC1)=O 3902,C(C(CC(=O)NOCc1nc[nH]n1)OC)NC(C=CCCC)=O 3903,S(=O)(=O)(c1cc(C(N2CCCCC(CNC(=O)CNC=O)C2)=O)n(C)c1)NC 3904,C(=O)(CCCCCCCCCO)NCC1N(C(=O)C=CCF)CCCC1 3905,C1(C(N(CC(C)CNC(=O)COCC2CCCO2)C)=O)CCS(=O)(=O)N1 3906,C#CC1CN(C(=O)C(CNC(=O)C(CC)n2ccnc2)C(C)C)CCO1 3907,N1(C(C2C(C(=O)OC)CC2)=O)CCC2(CC(NC(=O)C(C)(C)CF)C2)C1 3908,c1(OC)cc(F)c(NC(=O)NCC2COCCC2C)c(F)c1 3909,c1(CCC)ccccc1C(=O)NC1CC(NC(=O)Cc2ccc(C)s2)C(O)C1 3910,C1(C(N2C(C)CN(C(C3C4CCCCCCC34)=O)CC2)=O)CNc2ccnn2C1 3911,C#CCC(CC#C)C(=O)N(C)CC1CCCC(NC(c2cc(C3CC3)on2)=O)C1 3912,C1(C(=O)NCC(CNC(c2c(C)c(N)ccc2)=O)C)Cc2c[nH]cc2S1(=O)=O 3913,C1(C(=O)NC2(c3cc(C)no3)CC2)CCCN(C(=O)CP(C)(C)=O)CC1 3914,Cc1nnc2ccc(C(N3CCCC3CCNC(c3occc3F)=O)=O)cn12 3915,Cc1c(F)ccc(C(=O)NCC2CC2CNC(C2CCS2(=O)=O)=O)c1Cl 3916,c1(C(N(Cc2cn(CC(C)CS(C)(=O)=O)nn2)O)=O)cccc([N+](=O)[O-])c1 3917,CCC(O)C(C)C(=O)N1CC(CNC(C2CCS(=O)CC2)=O)C(C)(C)C1 3918,C1(CCC)C(=O)NCCN1C(=O)C(=O)NCCc1ccc(F)cc1Br 3919,C1(CNC(C#CC(C)C)=O)CC2(CCOCC2)CN1C(=O)CC1CC(=O)NC1=O 3920,N1(C(C(C)OCCOC)=O)CCN(C(c2ccc(=N)[nH]n2)=O)CCC1C 3921,c1(C(=O)NC2(CNC(=O)CSCC(N)=O)CC(OC)C2)cccnc1Cl 3922,O=C(CCC(=O)c1ccc[nH]1)NCC1C=CCN1C(=O)C1=COCC1 3923,C1(C(=O)OC)CCCN(C(c2ccccc2C)C)C1=O.C(C(Cl)Cl)O 3924,C(C)(CC(C)(C)C)NC(C(=O)Nc1c(C)csc1)=O 3925,CC(C)(CC#N)C(=O)N1CCCC(NC(c2ccc(F)c(CO)c2)=O)C1 3926,c1(C(N2CC(NC(C3(C#C)CCC3)=O)(CO)C2)=O)cc(C(=O)OCC)ccc1C 3927,CCC(CC(=O)NCCC12CC(CCO1)C2)N(C(=O)C(CSC)OC)C 3928,C1(NC(c2c(C)nc(CO)s2)=O)CN(C(=O)C2=CCCOC2)CCC1C(F)(F)F 3929,Cn1ncc2c1CCC(C(=O)NCC1(C)CCN(C(=O)C(F)F)CC1)C2 3930,N12CCC(O)(CC1)C2.c1(C(C)OC)n[nH]c(=NCc2occc2C)o1 3931,CC1N=C2NN=C(O2)N2CCC1C2.c1ccccc1F.C(F)F 3932,O=C(CN=c1cc[nH]cc1)NCCc1ocnc1CNC(C1C2CCC1CC2)=O 3933,C1(NC(C=C(C)C(C)(C)C)=O)CCCCCN(C(=O)COC2CCN(C)CC2)C1 3934,C=Cc1cc(C(=O)N(CC(N2CCC(C(=O)NC)C2)=O)CC)cc(F)c1 3935,c1(C(N2CC(CC)N(Cc3c(OC)cccc3F)CC2)=O)c(F)ccc(F)c1F 3936,c1(OC)ccc(F)c(CC(=O)N(C2CN(C(c3ncccn3)=O)CC2F)C)c1 3937,N1(C(c2cc(N)cc(F)c2)=O)CCCC(NC(c2ncc[nH]c2=O)=O)C(F)C1 3938,C1(CC)CCN(Cc2ccc(C)cc2-n2cccn2)CC1OC 3939,C=CCCC(O)CNC(=O)CC(O)CNC(c1csc(C)c1C)=O 3940,C1(NC(C(Cc2ccoc2)NC(COCCCCC)=O)=O)CCCC2(CCC2)C1 3941,Cc1sc(C(=O)NCCC2CCCN2C(C2CC23CCC3)=O)cc1CS(C)(=O)=O 3942,C1(NC(C=C(C)C)=O)COC2(CCCN(C(=O)CC3(C(F)(F)F)SCCS3)C2)C1 3943,N1(C(C(C)C2CCCO2)=O)CCC(CCCNC(c2ncc[nH]c2=O)=O)CC1 3944,C1(C(=O)NCCS(C)(=N)=O)CC2(CCN(C(=O)CC3CC(=O)NC3=O)C2)C1 3945,N1(C(c2ccc(C(C)=O)nn2)=O)CC=C(CNC(c2cnn(C3CC3)c2)=O)CC1 3946,CC1(C)CC(NC(c2ccc3c(c2)CC3)=O)CN1C(=O)Cc1ccc(Cl)cn1 3947,c1(NC(C(C)(N(C(CC(C=C)C)=O)C)C2(CO)CC2)=O)cc(O)c(C)cc1C 3948,CC1C(O)CCCN1C(c1ccc(CNC(=O)CSc2nc[nH]n2)s1)=O 3949,Cc1[nH]nc(C(=O)N(C2CC(NC(=O)CCn3ccccc3=O)C2)C)c1C 3950,C(=O)(CCCC(F)(F)CO)NC1C(C)CN(C(=O)Cn2cc(Cl)cn2)C1 3951,c1(OC)cc(C(N2CCC(O)(CNC(=O)Cc3cccc(Cl)c3)C2)=O)ccn1 3952,N1(CC(=O)NC(C(=O)OC)CC(F)(F)F)CCC2C(O)CCCC2C1 3953,CC(CN(C)C)CCC(=O)NC1(C(=O)NC2(CO)CC3CCC2C3)CCOCC1 3954,CCC(CCC(=O)Nc1cncc(F)c1)NC(=O)C(C)(O)CCN(C)C 3955,N1(Cc2scc(CC)n2)C(=O)CN(CCN2CCC2CC)C1=O 3956,C12(C(N3CC4C(NC(c5c(N(C)C)scn5)=O)(C4)C3)=O)C3C4C1C1C2C3C41C(N)=O 3957,c1(N2CC(CNC(c3c(OC)ccnc3)=O)(OC)C2)nc2cc(F)cc(F)c2o1 3958,N1(C(C2C(C(=O)OC)C2)=O)CCCC(C2CCN(C(=O)C(O)C3CCC3)C2)C1 3959,C(=O)(C(CC)(CC)C(=O)OC(C)(C)C)NCCN(C(CCC(=C)Br)=O)CC(C)O 3960,c1(C(N(CCOCCNC(C(CC)F)=O)C)=O)cc(OC(C)C)ccc1C 3961,c1(C(=O)O)cc(=NCC2C3(CC3)C23CC3)cc[nH]1 3962,C(N=c1[nH]cnc2cc(F)c(F)cc12)C1N(C(C2(C)CCOCC2)=O)CCCC1 3963,C#CCCN(C)N1CCCC(Cc2ccc(Cl)cc2)C1 3964,CCCCCCCCC(=O)NC(C)CCCNC(=O)C1=COCCO1 3965,Cc1ccc(CCC(=O)NC2CCC2CNC(c2cn3ccsc3n2)=O)cc1Cl 3966,N1(C(CC(CC)C2CC2)=O)CCOCC(F)(CNC(=O)Cn2ccnn2)C1 3967,C12(CC)CN(C(=O)Cc3nnc(C)o3)C(CNC(C3(C)CC3(Cl)Cl)=O)(C1)C2 3968,n1(CC(=O)OCC)nccc1C(=O)N(CCNC(=O)C(O)c1cnc[nH]1)CC 3969,c1(CC(N2C(COC)CN(C(=O)CCCC(C)=O)CC2)=O)ccccc1[N+](=O)[O-] 3970,Cc1cnc2n1CCCC2C(=O)Nc1cc(C(C)C)nn1C(C)(C)C 3971,N1(Cc2c(C)cc(Cl)cc2)CCCN(C(c2cccc(F)c2C)=O)C(C)C1 3972,C#Cc1ccc(C)c(CNC(=O)NCCNC(=O)OCC)c1.C(C)(C)(C)O 3973,C(C)(N=c1[nH]c(N2CCC(C(C)C)C2)nc2ccccc12)c1cc(C)cc(Br)c1 3974,C(CCCCCN=C(NCC1CN(C)CCO1)NCC1(CC)CCC(=O)N1)SC 3975,c1(SC)nccnc1C(=O)NCC1(C(N)=O)CN(C(C2CCC(F)C2)=O)C1 3976,N(C1CCCc2sccc21)C(N1CC(CO)C(Cc2ccccc2)C1)=O 3977,C(=O)(C(CC(F)F)NC(=O)COc1ccsn1)NC1CC(C(=O)OC)C1 3978,c1(CC(=O)NC2C(C)(CNC(C3C(C#C)C3)=O)CCC2)cc(Cl)ccc1Br 3979,N1(c2c(C)nc(OC(C)C)cc2)Cc2cc(CN3CCCS(=O)(=O)CC3)ccc2C1 3980,C1(CNC(C(C(CC)C)O)=O)CC2(CCN(C(=O)CCc3cnc(O)[nH]3)CC2)C1 3981,C(=O)C(CCSC)NC(=O)C(Cl)Cl.C1(=O)CN1C.CO 3982,N1(C(c2csnc2Cl)=O)CCC2CCCC12C(=O)NCC1CCC1(F)F 3983,CCCC(C(=O)N1CC(CN2CCC(C(=O)NCC(C)C)C2)C1)OCC 3984,C1(C)(C(=O)NCC2CC(NC(c3c(OC)nn(C)c3)=O)C2)CC(O)CN1C 3985,CCC(CC1CCCC1)C(=O)NC1CN(C(c2sc(CO)nc2C)=O)C1 3986,c1(C(c2n(CCOC)nnn2)NCC2CCOC2)cc(OC)nc(Cl)c1 3987,C1(NC(=O)CCc2cnccn2)CCCCN(C(C2CCC(F)(F)CO2)=O)C1 3988,C1(C(=O)OC)CN(C(C2CNCC3(CCC3)C2)=O)C2(CCC2)C1 3989,CCCC(C(=O)NCC1CCN(C(=O)Cc2ccc3nn[nH]c3c2)C1)S(N)(=O)=O 3990,CC(F)(F)C(C)(C)C(=O)N1CC(CCCCNC(c2ccc(C(F)F)o2)=O)C1 3991,c1(C(=O)NC2C(C)CN(C(c3csc(Cl)n3)=O)CC2)nnn2c1CCCC2 3992,C1(CN=c2[nH]nc(C(C)C)o2)CC12CCN(C(c1nc3ncccn3n1)=O)CC2 3993,O=C1CCC(C(=O)NCCC2CCCCN2C(c2ccsc2C(F)F)=O)CN1 3994,c1(C(=O)NC2(CNC(C3C(CC)CCO3)=O)CCC2)[nH]c2ccc(F)cc2c1C 3995,CCCC(C(=O)NC1CCCCC1NC(c1cc(F)c(CO)c(F)c1)=O)C(C)C 3996,c1(C(N2C(CNC(c3ccns3)=O)CC(OC)C2)=O)cc(Cl)c(F)cc1O 3997,Cc1ccc(OCCC(N2CC(NC(=O)CCC(C)C#N)C3(CC3)C2)=O)cc1C 3998,CCCC(C(=O)NC(C)(C(N)=O)c1ccncc1)c1ccc(Cl)cc1 3999,c1(NC(c2cnc(-c3cccc(O)c3)cn2)=O)nc(F)ccc1Br 4000,CC(C)(C)CC(O)CC(=O)NC1CCCC1C(=O)NC(CCO)C(F)(F)F 4001,CCCC(C(=O)NC(C12CCC(CC1)C2)CNC(=O)C(F)(F)C1CCOCC1)OC 4002,c1(C(C)OC)nc(C(=O)NC(CNC(c2cn(CCF)nn2)=O)CO)co1 4003,c1(C(N2CCCC(CN(C(=O)Cc3nc(=N)[nH][nH]3)C)C2)=O)cc(O)cc(N)c1Cl 4004,N1(C(CC2C(OC)CC2)=O)CCN(C(=O)COCCN=[N+]=[N-])CC1C 4005,c1(CC(=O)NC2C(NC(c3cc(C)on3)=O)CCC2)c(C)[nH]c2ccnn2c1=O 4006,CCCCC(CC)CC(=O)N1CC=CCC1C(N1CC(C2=NOCC2)C1)=O 4007,Cc1nnc(O)c(C(=O)NCCC2CSCCN2C(=O)CC2CC(F)(F)C2)c1C 4008,c1(C(=O)NCC2(N3CCOCC3)CCCOC2)nc2ccc(F)cc2s1 4009,c1(C(=O)NCC2(F)CN(C(C=Cc3ccn(C)c3)=O)C2)n[nH]c2c1CC(C)(C)C2 4010,c1(CNC(C2CCCN(C(=O)COC3CCCCC3)C2)=O)cc(Br)ncc1F 4011,c1(C=O)ccc(Cl)c(F)c1.N1(N2C(CC(=O)NCC)CCC2)CC2C(C=O)C2C1 4012,N1(C(c2ccc(F)c(Cl)c2)=O)CC2CCC1CN2C(C1SC2C=CC1CC2)=O 4013,N1(C(C(C)OC2CCCC2)=O)C(CNC(=O)C2=NOC(C)C2)CC2COCC12 4014,C1(C(=O)NCCCC(C)NC(C(C)NS(C)(=O)=O)=O)CC2(C1)CC2F 4015,Cc1ccc2ccccc2c1CNC(c1sccc1Br)c1nnnn1CC1CC1 4016,c1(N2CCC(N(CC#C)C(c3cscc3C)=O)CC2)ncnc2cc(Br)sc12 4017,C1(C(N(CC(C)O)C)=O)CC(NC(c2cncc(F)c2)=O)CCO1 4018,C1(CC(=O)NCC(C2CC2)NC(C2CC2C2CCCC2)=O)CCCCC1(F)F 4019,C1(C(N(C(CC)C2CC2)C)=O)CN(C(C2(C(=O)OC)CC2)=O)CC(C)O1 4020,C(=O)(C(O)CC(N)=O)NC(C)CCC(=O)N(C)Cc1cccc(O)c1 4021,CC1CCC2(CC2)N(C(=O)CC2C3CN(C(c4cnc5ccccn45)=O)CC23)C1 4022,c1(C(=O)Nc2nc(C(=O)OC)c(C)s2)n[nH]c2cccc(C3=CCCC3)c12 4023,C1(C(=O)NCC(C2CCC2)NC(C(CC)=CC)=O)CCc2cn(C)nc2C1 4024,C1(NC(c2cn(Cc3onc(C)n3)nc2)=O)CCN(C(c2cn[nH]c2)=O)CC1F 4025,C(=O)(CCC(=O)N(C)C)NCC1OCC(C(N(C(C)C)C2CC2)=O)C1 4026,C1(O)(CNC(C(C)n2cccc2)=O)CCCN(C(=O)Cc2cccc(OCF)c2)C1 4027,c1(C(N(CC(C)O)CCNC(c2ncn(C(C)C)n2)=O)=O)onc2ccccc12 4028,C(CCC(C(=O)Nc1ccccc1)N(C1CCN(C)CC1)C)=C(C)C 4029,CCC(C)CC(C(=O)NCc1cc(C#N)n(C)c1C)NC(C)=O 4030,C(=O)(CC(F)(F)C(F)F)N1CCCN(C(c2ccc(-c3ccco3)[nH]2)=O)CC1 4031,c1(C(C)CN(C)C)ccc(-n2cc(C(C)(C)CO)nn2)cc1 4032,c1(OC)noc(C)c1NC(c1coc(C(C)NC(C2(C)CCCCC2)=O)n1)=O 4033,N1(C(CC=C(C)C)C(=O)NC2CC(N3CCCC3)C2)CC2(C1)CC2(F)F 4034,C(=O)(C(=O)CCCC)NC(CC=C)CNC(c1cnc(OC)cn1)=O 4035,N1(C(CC(=O)NCC)=O)CCC(C2CC2)C1C(N1CC(C)(N(C)C)C1)=O 4036,c1(C(=O)NCCC(C)NC(C2CCOC(C)C2)=O)cc2c(cc1F)NCCC2 4037,c1(C(=O)NCC2C=CCN2C(C2CCCC2(F)F)=O)ccc2c(n1)OCCO2 4038,C1(O)(CN(C(c2n(CC)cnn2)=O)C)CCCN(C(=O)C(=CC2CCCC2)C)C1 4039,C1(NC(C(C)N(CCSc2ccccc2)C)=O)CN(C(=O)C(=O)N(C)C)CC1O 4040,c1(C(=O)NC(CCCNC(c2cc(C(C)=O)c(C)o2)=O)C)nc[nH]c2ncnc1-2 4041,c1(OC)ccc(Cl)c(C(=O)NCC23CC2CN(C(=O)CC24CCCC2C4)C3)c1 4042,N1(CC(=O)N(CCC(=O)NC(CO)C2CC2)CC=C)CCOC1=O 4043,c1(C(N2CCCC(N(CCO)C(C3C=CCCC3)=O)C2)=O)cnccc1Cl 4044,C1(CNC(c2n(CC)ncc2)=O)CCN(C(C2CSC(C)=N2)=O)C12CCC2 4045,N1(C(c2c(C)cc[nH]2)=O)CCN(C(=O)COC2CCOC2)C(CC(F)(F)F)C1 4046,C(C(CC(F)(F)F)NC(c1cc(F)cc(F)c1)=O)NC(CC1CC(OC)C1)=O 4047,C1(C(N(C)Cc2c(C)n[nH]c2)=O)CC(NC(c2cnccc2C)=O)CCO1 4048,C(CCC(C)C)(C(=O)NC(c1ccccn1)C)NC(c1c(CC)nccn1)=O 4049,C(=O)(C(C)(O)C(F)(F)F)NCCC(=C)CNC(c1ccc(C)c(Cl)c1)=O 4050,c1(N2C=CC(C(=O)NC3(CCOCC)CCCC3)C2)nc2ccc(F)cc2s1 4051,Cc1ccc(C)c(CN2CCC(C)(CNC(C3CCN(C)C3=O)=O)C2)c1 4052,C1(c2onc(C3(c4ccc(F)cc4)CCC3)n2)CCCC2(C1)OCCO2 4053,N1(CC(=O)NC2(C)CC2)CCCC(C(N)=O)(CO)C1.C1(CC(N)=O)OCCO1 4054,C(=O)(C(C1=CCCSC1)N1CCOC(C(C)(C)O)C1)NCC=C 4055,C(N=c1ncc([N+](=O)[O-])c[nH]1)C1CN(c2nc(C(=O)OCC)c(C)s2)C(C)C1 4056,N1(C(c2c(C)con2)=O)CC=C(CC(=O)NCC2(O)CCCC2)CC1 4057,C1(NC(C2N(C(C3CC(CC)(CC)C3)=O)CC(OC)C2)=O)CC2(CC(OC)C2)C1 4058,C(CCC(C)(C)CO)NC(CC1CC(C)N(C(=O)CNC(N)=O)C1)=O 4059,C1(NC(c2c(C)ncs2)=O)CS(=O)(=O)CC1NC(c1cnc(CO)[nH]c1=N)=O 4060,C(C(C)(CO)CC=C)NC(C(CC#C)NC(C1CCN(C)C1)=O)=O 4061,C1(C(N(C2CCC2)CC#C)=O)CN(C(=O)CCn2cnc(=N)[nH]2)CC1(F)F 4062,c1(NC2CC(C(=O)Nc3nc(C)c(C#N)nc3)C2)ncnc2sc(Br)cc12 4063,c1(CNC2CC(NC(CNC(CC(C)C)=O)=O)C2)cc(F)cc(Cl)c1 4064,N1(C(=O)C=Cc2cocn2)CC2CCC(NC(C3(F)CCOC3)=O)C2C1 4065,c1(CCNC(=O)NCC2CCN(C)C(=O)C2)cccc2ncccc12 4066,C1(C)(C(=O)NCC(N2CC(C)(OC(C(=O)OCC)CO)C2)=O)CC2CCC1C2 4067,c1(C(=O)NC(CC)CN(C(c2ccc(SC)o2)=O)CC)ccccc1C 4068,C1(F)(NC(C(C)C)=O)CCS(=O)(=O)C1.C12CCCC1CN2C(=O)Cc1cccs1 4069,C1(NC(CCOCCN(C(=O)C(C)(C)C)C)=O)CCCSC1 4070,N1(C(C=CC)=O)CC2CC(NC(=O)C(C3CCC3)OC)CC1C2 4071,N1(C(CCN(CCC)C)=O)CC(F)CC1CC(=O)NCC(C1CCCCC1)O 4072,c1(CC)cc(C(=O)NC2(COC)CN(C(c3cc(Cl)ccn3)=O)C2)ccc1F 4073,Clc1cc(Br)c2ncnc(N3CCCCCC3c3ccco3)c2c1 4074,N1(C(CN2C(C)CCC2C)=O)CC2(CCC(CNC(=O)C(C)N3CC(C)C3)O2)C1 4075,C1(C(N2CC(C)(NC(C(C)=CC)=O)C2)=O)CCCOC1c1cn(C)nn1 4076,C12(NC(=O)Cc3ccoc3)CCCC1N(c1cc(Cl)nc(C(F)(F)F)n1)CC2 4077,O(N1CCC(N=c2cccc(S(=O)(=O)N3CCCC3C3CCCO3)[nH]2)CC1)CC 4078,c1(-c2cnc(C(C)OC(c3c(C)occ3)=O)o2)ccc(Cl)cc1 4079,C1(NC(CCC=C)=O)CCC(O)CN(C(c2ccc(C(=O)OC)cc2F)=O)C1 4080,C12(CNC(C)=O)CC(NC(=O)C(c3ccccc3)F)(CO1)C2 4081,C1(C(N(CCCOCCNC(CC2CC(C)C2)=O)C)=O)OCCC1(C)C 4082,c1(CC(=O)NC(CC)CNC(C23CC(O)C2C3)=O)cnc2c(C)cccn12 4083,c1(C(=O)NC(CCCNC(CCCCCSC)=O)C)ccnc2c1CCCN2 4084,C1(CNC(C2N(C(C)=O)CSC2)=O)COCCN1C(=O)CNC(=O)C(F)(F)F 4085,N1(C(C2(C)CN(C(C3CCN(CC)C3)=O)C2)=O)C2CSCC1C2 4086,Cc1cc2c(Br)cccc2c(=NC(C)C(O)c2ccc(F)c(Br)c2)[nH]1 4087,c1(C(N2CC(n3cc(C(CC(C)C)(C)O)nn3)C2)=O)ncc2c(Br)cccc2n1 4088,Cc1cc(Br)cnc1C(=O)NC1(CC2CC2)CCN(C(=O)C#CC2CCC2)C1 4089,c1(C(=O)NC2CC(CNC(c3cc(CCOC)on3)=O)C2)nc(Cl)c(Cl)s1 4090,CC1=C(C)CC(C)(C(=O)N(CCNC(=O)CCC#N)C(C)C)CC1 4091,c1(C(=O)NCC(C)NC(CC(=O)N(CC)CNc2nccs2)=O)ncsc1C 4092,c1(NC(CCC)CO)ccc(S(=O)(=O)NC2COc3cc(Br)cnc32)cc1Br 4093,Cc1nc(N2CCC3(NC(=O)C4=NNC(=O)CC4)CCCC23)c2ccsc2n1 4094,C1(C)(C(N2CCN(C(COCCCC#C)=O)CC2CF)=O)CC(C(C)(C)C)=NO1 4095,C1(CNC(c2cc(C(CC)CC)no2)=O)C2CN(C(C3CSC3)=O)CC12 4096,N1(C(c2nc(C(C)NC(CSCC#C)=O)oc2)=O)CCC2(CCCN2C)C1 4097,c1(-c2cc(C(=O)NCCNC(C3CC(C(N)=O)C3)=O)no2)ccccc1O 4098,Cn1cnc(CNC(C2CC2CNC(=O)CC2CCCCO2)=O)n1 4099,c1(C(N(C)CC2CCCC(NC(C(CC)(C)CO)=O)C2)=O)ccc2cnoc2c1 4100,Cc1ncc(N)cc1C(=O)N(CC(C)NC(=O)C(C)NC(c1ccco1)=O)CCO 4101,Cc1cnc(CNC(=O)CCCC2CN(C(=O)OC(C)(C)C)C2)o1 4102,Cc1nc(N2CC(C)(CC(=O)Nc3ncc(F)c(Cl)n3)C2)c2ccccc2n1 4103,n1(CC)ncc(C)c1C(=O)NC1CN(C(c2csc(C)n2)=O)CC1OC 4104,c1(-c2ccc(C(N3CCC(c4ccc(F)nc4)CC3)=O)o2)cccc(F)c1 4105,c1(C(=O)NC2(C(=O)NC3CN(C(C)=O)C3)CC(O)C2)cn(C)cc1C 4106,C1(C(=O)OC)CCOC1C(=O)NCCCNC(=O)CC1(C)CCC1 4107,[N-]=[N+]=NC1CN(C(c2n[nH]c3c2COC3)=O)CC1NC(=O)Cc1csc(S)n1 4108,Cc1ccc(CC(N2C3CCC2C(NC(=O)CC2CC4CCC2C4)C3)=O)cc1C 4109,C1(CN(C)C(c2ccc[n+]([O-])c2)=O)CCCN(C(C2(CO)CCCCC2)=O)C1 4110,C(=O)(C1CC=Cc2ccccc21)N1C2CN(C(C#CC3(C)COC3)=O)C(C2)CC1 4111,Cc1nc(CNC(=O)CCc2cccn2C)oc1C(=O)NC(C)Cn1cnnc1 4112,N1(C(C2CC(C(C)C)OCC2)=O)CCC(F)(CNC(C2CN(C)C2)=O)CC1 4113,c1(OC)cc(OC)cc(NC(=O)CC(=O)OCC(C(=O)NC(C)C)N)c1 4114,C1(NC(C(C)n2cccc2)=O)CCN(C(C2CCC(C(F)(F)F)C2)=O)CC1 4115,Cc1ccc2c(C(=O)NCC3CC(NC(=O)C(=O)N(C)C)C3(C)C)csc2c1 4116,C(=O)(C#CC1(C(F)(F)F)CC1)N1CCC(OCCNC(C=C(CC)CC)=O)C1 4117,C=CCCC(C(=O)N1CCCC(O)(CC)C1)NC(=O)CN(C)CCOC 4118,C1(F)(C(N(CCN(C(C)C)C(C2CCOC2)=O)C)=O)C2CCCC12 4119,C1(C(C(=O)NC)CC)CCN(CC(=O)NCC(N)Cc2ccccc2)CC1 4120,c1(C(=O)OC)ccccc1-c1nc(C)c(NCC2(CC(C)C)CCC2)s1 4121,CCCS(=O)(=O)CC(=O)N1CCCC1CN(C)C(C1(c2ccc(Cl)nc2)CC1)=O 4122,Cc1nc(C(=O)NC2CC(C(N3CC(C)CC3C(N)=O)=O)C2)c(C)o1 4123,CC1CC(C(N2CC(NC(c3c(Cl)noc3C)=O)C2)=O)CC(C)C1 4124,N1(C(c2c(C)cnnc2)=O)CCC2(CC1)CC2NC(c1cc(C#N)ccc1F)=O 4125,N1(CC(=O)Nc2ccc(F)nc2)CC2(CCN(Cc3cccnc3)C2)C1 4126,c1(CC)c(C(N2CCCC(NC(=O)C(C)c3ccsn3)C2)=O)cnn1CCC#N 4127,C(=O)(C(CO)C(C)C)NCC1N(C(CCC(=O)N(C(C)C)C)=O)CC(F)C1 4128,N1(C(C2ON=C(CC)C2)=O)CC2CC1CC2NC(=O)Cn1cc(CC)cn1 4129,c1(C(N(C)CC2(NC(C3N(C(C)C)CCC3)=O)CC2)=O)nc2ccccc2s1 4130,C12(C(=O)NC3C(C(C)C)C3)CCCC1CCN2C(=O)CCCN(C)C 4131,c1(C(CC)NC(=O)NC2CONC2=O)ccc2c(CO)n[nH]c2c1 4132,C1(CNC(Cc2c(C)scc2)=O)CC2CCC1N2C(C1(N(C)C)CC1)=O 4133,c1(N2CCC3(C(CNC(c4cc(C)on4)=O)C3)CC2)ccnc2c1CCO2 4134,C1(CN(C2CCC(C)(C)C2)CC=C)CCN(C(=O)C(C)CC=CCC)CC1 4135,C=C=CCCC(=O)NCC1CN(C(=O)C=C(CCC)CCC)C1 4136,Cc1ncc(Br)c(C(N2CCC(NC(=O)C3=CCCCO3)C(O)C2)=O)n1 4137,C1(S(C)(=O)=O)(CNC(C(n2cc(-c3ccc(F)nc3)nn2)C)=O)CCCCC1 4138,C1(C(N2CC(CCCNC(C3CC(CCC)C3)=O)OCC2)=O)CC(=O)CC(=O)N1 4139,C1(NC(C(C)CC(N)=O)=O)CCC2(CC1)CC2NC(C1CC(=O)N(C)C(=O)N1)=O 4140,c1(C(=O)NCC(C2CCC(F)(F)CC2)OCC)ccc2n[nH]cc2c1 4141,N1(c2ncc(CC)cn2)CCCC2C1CCN2Cc1cc(C(=O)O)sc1Cl 4142,S(=O)(=O)(c1cccc(=NCCc2cnccn2)[nH]1)N(C(C)CC#N)C 4143,C(CCCCCN=[N+]=[N-])NC(C1C(c2c(OC)cccc2)C1)=O 4144,CC1(C)C(=O)CCCN1C(=O)CC(C(F)F)Nc1ccccc1 4145,N1(C(C2(C(N)=O)CCC2)=O)CCOC2(CCC2)CC1.C12CCCC1CC(=O)N2 4146,C1(NC(c2c(C)sc(-c3ccco3)n2)=O)CN(C(C2CCC2C)=O)CC12CCC2 4147,c1(C(=O)NC2C=CCN(C(c3nnn(C)c3C(F)F)=O)C2)ccc(C2CC2)nc1O 4148,Cc1cccc(C)c1CC(=O)NCC(c1ccc(F)cc1)NC(C1CCOC1)=O 4149,C1(C(N2CCC(C)(NC(C=CC=CCCCCC)=O)C2)=O)COC2COCC12 4150,C1(NC(CCCC=C)=O)CN(C(c2ccc(C3OCCO3)cc2)=O)CCC1CO 4151,N1(C(c2nn(C)c(O)c2)=O)CC2CN(C(c3cnc[nH]3)=O)CC12 4152,O=C(C1CCCn2ccnc21)N1CCCC1c1ccccc1 4153,Cc1c(C(N2CC(NC(C3CCC3C#N)=O)C(C)C2)=O)cccc1Cl 4154,c1(C(=O)NCC(CCOC)NC(C2CC(=O)N(C)C2)=O)[nH]c(C2CC2)nc1C 4155,C(=O)(C1=CC2(CCOCC2)C1)N1C(CCCNC(=O)CC2CCC2)CCC1 4156,c1(CC)ccc(O)c(NC(=O)C(F)C2CC(NC(C34CCC(OC)C3C4)=O)C2)c1 4157,C1(C(N2CCN(C(CC3CNC(=O)O3)=O)C(CCO)C2)=O)CC2C=CCC(C1)C2 4158,N1(C(c2ccc(C(C)O)cc2)=O)CCCCC(NC(C2(n3cnnn3)CC2)=O)C1 4159,C1(CC(=O)NCCC2(C(=O)NCC3(OC)CCOC3)CCCC2)C(=O)NN=C1C 4160,c1(CCC)nc(C(=O)N(C2CCN(C(C3(C)CCCO3)=O)C2)CC)cs1 4161,c1(OC)cccc(OCCC(=O)NCCC2COCCN2C(=O)C(F)C(C)C)c1 4162,C1(O)(CCNC(c2cn(C3CCOCC3)nn2)=O)CN(C(C2CCC2(F)F)=O)C1 4163,C(=O)(C1=CS(=O)CCC1)NCC(N)CC(F)(F)F 4164,c1(NC(C2(c3ccc(F)c(F)c3)CCN(C(C)=O)C2)=O)nc2ccc(Cl)cc2[nH]1 4165,n1(CC=C)cc(CNC(c2cn(CCNC(=O)C(F)C3CCOC3)nn2)=O)nn1 4166,c1(C(=O)NC2CC3N(C(C(CC)OC)=O)C(CC3)C2)cc2ccccc2cc1F 4167,c1(SC)ncc(Br)c(C(=O)NCC2CC(F)CN2C(=O)C(c2ccccc2)C)n1 4168,c1(CC)oc(C)cc1C(=O)NC1CCOC(NC(C23CC(COC)(CO2)C3)=O)C1 4169,C1(CCCNC(c2c(C)c[nH]n2)=O)CCN(C(c2cccnc2C2CC2)=O)CC1 4170,C1(CC)(CF)CCOCC1.c12cc(n[nH]1)C(=O)NCC1(CC1)CNC2=O 4171,C1C(=O)N(OC)CCC(=O)N1CC(=O)NC1CC1.C(C)(C)(C)OC 4172,N1(C(C(C(CC)C)O)=O)CCC2CCCC12C(=O)NCC(F)(F)C(F)F 4173,Cn1nc(C(=O)NC2CCC2NC(C2(O)CCOCC2)=O)cc1C(F)F 4174,c1(C(C(=O)NCCCF)N(C(C)C2CC2)C2CC2)ccc2ccccc2c1 4175,c1(OC)ccncc1NC(=O)C=C(C)CNC(=O)Cc1ccncc1Cl 4176,C1(C2(C)CC2)CCCN1C(=O)C(Cn1cncn1)NC(c1cn[nH]c1)=O 4177,N1(C(c2nncc(C)c2)=O)CCC(F)(F)C(CNC(C2CC=CCC2)=O)C1 4178,O=C(N=c1[nH]nc(Cl)cc1Br)C1CC2CC2N1C(c1cn2cc(F)ccc2n1)=O 4179,C(=O)(CC(C(F)F)NC(C1COC(=O)N1C)=O)N(C)Cc1nc(C)[nH]n1 4180,CCC(CC)CCCC(=O)N1CC(OC)C(OC)C1.C1(=O)C(C)=CCN1 4181,c1(C(C(=O)N(C(CNC(CCCN(C(C)=O)C)=O)C)C)C)ccc(C)cc1 4182,c1ccccc1Br.c1(CONC(C2CCCN2CC)=O)cc(CO)on1 4183,C1(C(=O)NCCCOCC)CCCN(C(c2nc(C)sc2C)=O)CC1 4184,C1(CC)CCN(C(c2cc(F)n(C)n2)=O)C1CNC(=O)CCc1ccnn1C 4185,Cc1ccc(OC(C)C(=O)N2CCC2CNC(=O)CCC=CC(C)C)c(C)c1 4186,C=CC(CC)CC(=O)N1CC(NC(=O)C=CCN2CCCC2)C(C=C)C1 4187,C(=O)(C(O)CCC(F)(F)F)N1CCC(N(CCC)C(c2cnn[nH]2)=O)CC1 4188,c1(CCC(N2CC3C(CNC(C(C)C)=O)C3C2)=O)c[nH]c2ccccc12 4189,CCCC(C)(CC)C(=O)NCC1(NC(c2cc(Br)cn2C)=O)CCCCC1 4190,C1(NC(c2c(CC)nc[nH]2)=O)COCCC1NC(C1(C2CCC2)CC1)=O 4191,c1(C2(C(=O)NC3CCC(CCNC(c4n(C)nnc4)=O)C3)CC2)ccc(Cl)cc1 4192,c1(C(=O)NC(C)C(C)NC(c2csc(O)n2)=O)ccc(-c2cnnn2C)cc1 4193,C(C(=O)N(C)C)(C(C)(C)C)NC1(c2cn(C)nc2)CC1.c1nnnn1CCCC1CC1 4194,C=CC1OCCC1C(N1CCCCC1CC(=O)NCC1CCC1COC)=O 4195,C1(NC(c2n[nH]cc2[N+](=O)[O-])=O)CCCCN(Cc2ccc(C3CC3)cc2)C1 4196,N1(C(CCC#C)=O)CCC2CCC(NC(=O)CCCC#C)C12.C12CCCN1C2=O 4197,C1(C(=O)NCC(c2ccccc2)NC(=O)CC2CCC2)CC2(COC(=O)N2)C1 4198,c1(C(=O)NC(CC)(CNC(C2(C)COCCO2)=O)CC)cccc2ncnn12 4199,C1(NC(COCCCC)=O)CCCC1(C)CNC(=O)CC1CC1C(F)(F)F 4200,C1(NC(C(c2ccn(C)n2)C)=O)C2CCN(C(=O)C(C)(O)C3CCC3)CC12 4201,C1(NC(c2cccc(C3(O)CC3)c2)=O)CCn2c(C(F)(F)F)nnc2C1 4202,c1(CN2C(NS(=O)(=O)C3CC3)CCC2)nc2ccccc2n1Cc1ccccc1 4203,Cc1cc(C(=O)NC2(c3cn(-c4ccc(Br)cc4F)nn3)CCC2)cc(O)c1 4204,CC1CCn2cc(C(=O)NC34CCCC3CN(C(=O)C(C)N3CCC3)C4)nc2C1 4205,c1(N(S(CC2C(C(=O)OC)CCO2)(=O)=O)Cc2cccc(F)c2)cccc(Br)c1 4206,Cc1ccc(C(N2CC3CC3(NC(=O)C(=O)NCCN(C)C)C2)=O)cc1F 4207,N1(C(C(C)OC)=O)CCC(F)(C(=O)NCCc2cnn(C)c2C)C1 4208,S(=O)(=O)(c1cncc(C(F)F)c1)NCCC1CC(OC)(OC)C1 4209,c1(NC(C(C)NC(=O)OC)=O)cncc(C2CC2c2ccncc2)c1 4210,c1(NC(c2cccc(O)n2)=O)cccc(NC(=O)CN2CCOCC2)c1 4211,c1(C(=O)NC2CN(C(C(CC)OC3CCCC3)=O)C2)c([N+](=O)[O-])cnn1CC 4212,C1(C(C(=O)N(CCC)CCNC(c2coc(C(C)C)n2)=O)C)CCC(F)(F)CC1 4213,CC1(C)CCN(C(=O)C(c2ccc(F)cc2)(C)F)C(C(=O)O)C1 4214,c1(C(=O)N(CC2(CCNC(=O)Cn3cncn3)CC2)CC)coc2c1C(O)CCC2 4215,c1(CCC)cc(C(=O)N(C2CCC(NC(C3CC4CC3C4)=O)C2)C)cc(O)n1 4216,N1(C(Cc2c(C)nccc2)=O)C(C(=O)NCC2(C)CSC(C)=N2)C2CC(O)C1C2 4217,N1(C(C(CC2CC2)OC)=O)CCC(C2CCN(C(=O)C(C)(C)CF)C2)CC1 4218,CCC(C(=O)NC(C)CCCNC(=O)C(=O)N(C)C)C(C)(C)CC 4219,c1(C(=O)NC2C(OC)CN(C(=O)CC=C(C)C)C2)cc2occc2[nH]1 4220,c1(-c2ccc(CN(C(C)(C)C)CC)cc2)ccc(F)c(C)c1 4221,S(=O)(=O)(c1ccc(Br)cc1NC)NC(C)(C)C.C(C(C(F)F)C1CC1)CCOCC(F)F 4222,Cc1ccc(C=C(C#N)C(=O)NCC2(CNC(=O)C(C)OCC(C)C)CC2)cc1 4223,C(CC(C(=O)N1OC(C)(C)C1)NC(=O)CCCCCNC(C)=O)=CC 4224,Cc1nc2cc(C(N3CC4CC3C4CNC(C3COCCN3C)=O)=O)cnc2[nH]1 4225,c1(-n2cc(NC(=O)NC(c3cn(C)nc3Cl)C)nn2)ccc(C(C)(C)C)cc1 4226,N1(C(CCn2c(C)ncc2)=O)CCN(C(c2cc(Cl)ccc2N)=O)C(C)C1 4227,C1(C(=O)NC(C(=O)OC)C)CCC(C)(C)N(C(=O)C=C2CCC2)C1 4228,CC(CC(F)F)C(=O)N1C(C(=O)NCC(=O)NCC2CC2)CCC1C 4229,N1(C(CC(=C=C)C)=O)CCN(C)CC1C(=O)N(CCC(O)CO)C 4230,c1(C(=O)NC(C2CCN(C(CC3(OC)CCC3)=O)C2)(C)C)cn2ccccc2n1 4231,c1(C(=O)NCC(CNC(COCCCOC)=O)C(F)(F)F)cc(C)c(F)c(C)c1 4232,C1(C(=O)NC(c2cn(CCCCN3CC(OC)C3)nn2)=O)C2CCC(C2)C1C 4233,c1(CCNC(C(=O)Nc2c(C(C)(C)C)cccc2)=O)nc2ccccc2s1 4234,C(C(CC(=O)N1CCC(NC(C2(C)CCCCCCC2)=O)C1C)C(F)F)N(C)C 4235,c1(C(C(=O)OC(C(C)=O)C(C)=O)=O)c[nH]c2ccc(F)cc12 4236,S(=O)(=O)(c1cc(F)ccc1Cl)OS(CC1(C)CCOC1)(=O)=O 4237,C1(NC(CC2COCC(C)O2)=O)CC=C(C(=O)NCCC(C)N(C)C)C1 4238,c1(OC)ccccc1CN1CCC1C(=O)Nc1nnccc1-n1ccnc1 4239,c1(-c2cn(C(C)C(N3CCC(OCCO)C3)=O)nn2)c(Cl)cncc1Cl 4240,c1(C(N2C(CNC(CC(C)SC)=O)CC(O)C2)=O)cc2c(s1)CCOC2 4241,C(C)(C)(CC(=O)NC1CCC2CC12)N(C)C(c1ccns1)=O 4242,c1(N(CCC)CCNC(=O)C(CC)C(C)O)ncnc2[nH]cc(C(=O)NC)c12 4243,S(=O)(=O)(c1ccc(NCC2(C)CSC(C)=N2)c2cnccc12)N1C(CC)CC1 4244,N1(C(C(C2(O)CCC2)NC(c2ccnn2C(F)(F)F)=O)=O)CCCC(CCO)C1 4245,Cc1ccc(C#N)c(NC(=O)CC2CN(Cc3ccc4c[nH]nc4c3)CCO2)c1 4246,CCC(CC(F)(F)F)C(=O)NC1(C)CC(NC(c2cc(Br)cn2C)=O)C1 4247,N(C(=NCCCCl)NC1CC2(CC2)C1)Cc1c(C)nns1 4248,C(C)(C(=O)NC1CCC(n2cc(-c3ccc(C)nc3)nn2)CC1)(C(C)C)OC 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4285,CCCC(O)C(=O)NC(Cc1cn[nH]c1)C(=O)NCC(F)F 4286,CC(C)CCN=C(NCC1CN(c2ncccn2)C1)NC1CCCOC1 4287,N1(C(C2(OC)CCSC2)=O)CCC2(C1)CN(C(=O)C(C)(C)CC(C)=O)CCO2 4288,C1(NC(C(C)(N(C(C=CCC)=O)C)C2CC2)=O)CCCCNC1=O 4289,C(=O)(CCP(C)(C)=O)N(C1CCOC1)C(C)CNC(C1(c2cccc(Cl)n2)CC1)=O 4290,N1(C(c2c(C)[nH]nc2Br)=O)CCN(C(=O)CCC2CCCOC2)C(CO)C1 4291,c1(CC(c2cnc(C)[nH]2)C)cc(F)cc(Cl)c1.c12nnnn1CC2c1ccccc1C.N 4292,CC1(CNC(=O)CC2(O)CCCC2)CCN(C(C2C(c3ccccc3)C2(F)F)=O)C1 4293,N1(CC(N2CC(OC)C(NC(c3ccoc3)=O)C2)=O)CCCCC(O)C1=O 4294,c1(C(N(c2cnc(F)cn2)Cc2onc(CC)n2)=O)c(C)nn(CO)c1Cl.C1(N)CC1 4295,N1(C(C2CC(=C)C2)=O)CC2CCC1C1CN(c3c([N+](=O)[O-])c(C)nn3CC)CC21 4296,c1(OC)cc(C)ccc1C(N1CC2CC1C2NC(c1ccnnc1)=O)=O 4297,c1(CNCC(c2ccc(O)c(O)c2)N(CC)CC)cc2cc(C)ccc2s1 4298,CC1COCC(C(=O)NCC#CCNC(c2cnn(C)c2Cl)=O)O1 4299,C1(C(=O)NC(CNC(CC)=O)C)CCC2(CC1)CC(OC)C2 4300,c1(OC(C)C)cc(C(N2CC(CNC(=O)CC(C)O)C(O)C2)=O)ccc1F 4301,c1(C(=O)NCC2CC(OC)CN2C(=O)CN(C)C(C)C)ccc2c(c1)N(C)CC2 4302,C(CCCCCS(=O)(=O)CCO)NC(=O)NC1CCC=CO1 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4446,C1(NC(c2cnc(Cl)[nH]2)=O)CCN(C(c2nccnc2C(F)F)=O)CC1F 4447,c1(NC(=O)NCc2ccc(N3CCS(=O)(=O)CC3)nc2)cc(I)c(O)c(I)c1 4448,C1(C(=O)NCCC2N(C(c3c(OC)ccs3)=O)CCOC2)CCOCC12CCC2 4449,N1(C(CN(C(c2nn(C)cc2Cl)=O)CC)=O)CCC(CO)C(O)C1 4450,n1(CC(N2CC(CC)C(NC(=O)CNS(N)(=O)=O)C2)=O)nc(Cl)ccc1=O 4451,N1(C(c2c(C#N)csc2)=O)CC2CCCC1CN(C(=O)CNC(C1CCC1)=O)C2 4452,C(CCN=c1[nH]cnc2c1SCCC2)OCCC(=O)NC(CCCC(C)C)C.C(N)=O 4453,N1(C(Cc2cccc(NC(=O)OC(C)(C)C)c2)=O)CCC2CCOCC2C1 4454,CCS(=O)(=O)CC(=O)N1CC(C)CCC1C(=O)NCCC1CC=CCC1 4455,C1(CNC(Cc2c(C)con2)=O)CCCCC1NC(=O)C(=C1CCCCC1)F 4456,c1(CC(N2CCC(N(C(c3[nH]cc(C)c3C)=O)CC)C2)=O)ccc(F)cc1F 4457,N1(C(C2(OC)CC2)=O)CCC(CNC(=O)CO)CC1C.C1(C)CCOC1 4458,C1(C(N2CCC(OC)(CNC(c3cncc(CO)c3)=O)C2)=O)CC(=O)NC(=O)N1 4459,CC1(C)CCC(CC(=O)NCC(=C2CN(C(=O)Cn3ncnn3)C2)F)OC1 4460,Cc1cc(N2CCN(CCF)CC2)nc(=NCCC(C)OCC(F)(F)F)[nH]1 4461,N(C)(S(=O)(=O)NOC(C1(OCC)CC=CCC1)=O)CC#C 4462,CCC(CNC(=O)C=Cc1ccccc1C)(CC)C(=O)N1CCC(C(N)=O)C1 4463,N1(C(c2cnc(COC)s2)=O)CCCC(NC(C2CCC(C(N)=O)CC2)=O)C1 4464,C(CCCC(C)(C)C(=O)NNC(=O)c1c[nH]c(C#N)c1)NC(C(C)OC)=O 4465,c1(NC(C)C)[nH]c(=NC(C)Cc2c(Cl)cccc2Cl)[nH]c2ncnc1-2 4466,C(=O)(C(C(C)C)C1CCC1)NCC1(OC)CN(C(c2cnc(O)o2)=O)C1 4467,Cn1ncc(N(C(C2(C)C=CCC2)=O)CC2CC2)n1 4468,c1(-n2cc(C(N3CCN(C(C(C)O)=O)CC3)(C)C)nn2)ccc(F)cc1F 4469,C1(OC)(CNC(C2(F)CCN(C(=O)Cn3cnnc3)C2)=O)CCCCC1 4470,C1(O)(CNC(C(N2CCNC2=O)C)=O)CCCN(C(=O)CCc2cnn[nH]2)CC1 4471,C1(CNC(c2c(C)nn[nH]2)=O)CC(C)N(C(c2nc(C(C)(C)C)no2)=O)C1 4472,c1(C(=O)NC2CCN(C(CCC=CC)=O)CC2CO)cc2ccccc2nc1O 4473,C(=O)(C(C(=O)NCCCCC(C)NC(=O)C(C)Sc1ccccc1)OC)OC 4474,c1(C(=O)NCC2CC(F)(CNC(C3(CCCC)CC3)=O)C2)cnn(CC)c1C 4475,C1(C2CCN(C(=O)CC3CC3)C2)(NC(c2ccccc2Cl)=O)CC1.O=C1CCN1 4476,c1(CC(=O)NCC(CN(C)C(C2CCC(=O)N2)=O)O)cncn1C 4477,CC(C)C(CCN(C(=O)CC1C(C)C1(F)F)C)NC(c1cnc(S)n1C)=O 4478,c1(NC(C23CC2CN(C(C2(C(=O)O)CC2)=O)C3)=O)cncc(-n2nccn2)n1 4479,C(N=c1nc(N2CCC(=NO)CC2)c2c([nH]1)COC2)c1ccc(N)cn1 4480,N1(C(c2ccc(C)cc2Cl)=O)CCC2(CC1)CN(C(=O)C(O)Cn1cncn1)C2 4481,c1(NC(C)C)ccc(C(=O)NCC2CC2CNC(c2cc(Cl)no2)=O)cn1 4482,O=C(C1CCCc2ccnn21)NCC1CCN1C(c1cnc(O)n(C2CC2)c1=O)=O 4483,N1(C(CN(CC(C)C)C(C2CC(=C)C2)=O)=O)CCOC(CCF)C1 4484,c1(C(=O)NCC(C2CCOC2)NC(C(C)(C)C(N)=O)=O)csc2c(F)cccc12 4485,CC1CCN(C(=O)CN2CC3CCC2C3)CC1CNC(c1cc(Cl)on1)=O 4486,c1(NC(CCC)c2ccco2)[nH]c(=NCCc2cccnc2C)nc2scnc12 4487,C1(C(=O)OC)CN(C(C2CN(Cc3ncccc3Br)CCN2)=O)CCC1O 4488,N1(C(c2cc(F)cs2)=O)CCCC(Cl)(O)CC1 4489,N#Cc1ccc(C(=O)NC2(C(N3CCC3CO)=O)CCSC2)s1 4490,CN1C2(CCN(c3nnc(C(C)(C)C)o3)CC2)C(NC(=O)CC2CC2)CS1(=O)=O 4491,C1(CNC(Cc2cc(C)sc2)=O)COCCN1C(c1cnc(C2CCC2)s1)=O 4492,c1(C(=O)NC2CCC(CCC(=O)N(C(C=C)C)C)C2)c[nH]c(=S)cn1 4493,N1(C(C(CC2CCC2)NC(=O)Cc2cnns2)=O)CCC12CCCC2 4494,n1(C(C(N2CC(NC(COCc3onc(C)n3)=O)C2)=O)C)nc(C)cc1C 4495,CC12CN(C(=O)CC3CCCN3C(C34CCC(C3)C4)=O)C(C(N)=O)(C1)C2 4496,c1(C(=O)Nc2c(F)cc(C3CCNCC3)cc2F)ncc2cc(Br)cc(F)c2n1 4497,N1(C(CCNC(=O)NC)=O)CCC=CC1C(=O)NCC12CC(CCO1)C2 4498,Cn1nc(C(N2CC3CC(O)C2C3NC(c2ccc(F)s2)=O)=O)c2c1CCC2 4499,c1(CC(=O)NCC23C(CN(C(C(CC#C)O)=O)C2)CC3)ccc(F)cc1[N+](=O)[O-] 4500,C1(C2CCN(C(=O)NCC(=O)OC)C2)(NC(=O)COC(CC(C)(C)C)=O)CC1 4501,C1(C(N(CC(=O)NCCCc2nncn2C(O)C2CC2)C2CC2)=O)CCC(O)CC1 4502,C1(CNC(C2C(=C)C2)=O)(COC)CCN(C(c2cc(C)ccc2N)=O)CC1 4503,N1(C(C(C(C)C)O)=O)CCC2(CCN(Cc3cc(-c4ccc(F)cc4)n[nH]3)C2)C1 4504,Cc1cnc(C(=O)N(C2CN(C(c3cnnc(O)c3)=O)CC2F)C)c(Br)c1 4505,N1(C(C2=NOC(C)C2)=O)CCC2(C1)CN(C(=O)CCC1CCCCO1)CCO2 4506,N1(C(c2c(CC)cn(C)n2)=O)CC(NC(C2(C(=O)OC)CC2)=O)CC(C)C1 4507,C(=O)(CCCC(=O)C(C)OC(=O)C(F)CC1CC(F)(F)C1)OC 4508,c1(C(N(C2CCN(C(C3CC(C#C)(O)C3)=O)C2)C)=O)cnc2c(Cl)cccn12 4509,N1(C(CCCCCOCC)=O)CCCC2CN(C(=O)CSC(C)(C)C)CCC12 4510,CCCC(CCCNC(=O)C1CC1)NC(c1ncccc1CC)=O 4511,C1(C2CCN(C(=O)C(F)CC3CCC3)CC2)(NC(C(CC)C)=O)CC1 4512,C1(C(N2CCC(C(F)F)(CNC(C3CN(C(C)C)C3)=O)C2)=O)CC2C(C1)C2(F)F 4513,C1(N=[N+]=[N-])(C(N(CC#C)CC=C)=O)CCN(C(=O)CN2CCSCC2)C1 4514,c1(NC)cc(N2CCOCC2)ccc1Cl.C1(=O)C(C)(C)n2cc(cn2)N1 4515,c1(-c2cc(C(=O)NC3CN(C(c4cnn(CC(F)F)n4)=O)C3)n[nH]2)ccccc1O 4516,C(=O)(CCCC(C)NC(=O)CN1CCCCC1)NCC(C)C#N 4517,N1(C(C(C)CCN(C)C)=O)CCN(C(=O)CC2(C)OCCO2)CC(C)(F)C1 4518,Cc1cc(CC(=O)NCc2nc(C(=O)N(CC(C)O)C)co2)no1 4519,C(=O)(C1=CCCC1(C)C)N1CCC(C(C)(C)NC(c2n(CC)cnn2)=O)C1 4520,C1(NC(CCCOCC)=O)CCCN(C(=O)CCC(C)(C)F)CC1F 4521,CC(N=c1[nH]ccc(C#N)c1[N+](=O)[O-])C1CN(C(c2ccnc3[nH]ncc23)=O)C1 4522,CC(C)C(C(=O)NCC(c1ccncc1)C)C(C)NC(C1CC(=O)C1)=O 4523,C(=O)(CCN(OC)C(=O)C(C)N(C(=O)C(C)C#N)C1CC1)OC 4524,N1(C(CC#N)=O)CCC2(NC(c3ccc(-c4ccon4)cc3)=O)CCCC12 4525,CC1(C)OC(=O)CC1C(N1CCN(C(=O)Cc2ccc(Cl)s2)C(CF)C1)=O 4526,Cc1ccsc1CC(=O)N(C(c1ccccc1)CNC(C1(CC2CC2)CC1)=O)C 4527,c1(-c2c(C)ccnc2F)ccc2ccnc(NC(=O)C3=CCCCO3)c2c1 4528,c1(CC(=O)NCC2C(CNC(c3c(C#N)nc[nH]3)=O)C2)cc2ccccc2o1 4529,n1(CC)c(C(=O)N(CCC(=O)NC2(C(O)COC)CCC2)C)cnc1O 4530,C(=O)(CCCCCNC(c1cn(C2CC2)nn1)=O)NCC(CCCC)O 4531,C1(NC(C(c2cncc(F)c2)C)=O)C2CC1CN(C(c1ccc([N+](=O)[O-])[nH]1)=O)C2 4532,N1(C(CC(C)C)=O)CCC(CNC(=O)C(O)CN2CCOCC2)C1(C)C 4533,c1(CC(C)OC)nc(-c2ccc(C3CC3(F)F)cc2)n(C2CCN(C)CC2)n1 4534,N1(C(C2CC(F)CN2C(c2cc(O)ccc2Cl)=O)=O)Cc2ccc(Cl)cc2C1 4535,C=CCC(C)C(=O)NCC1(C)CC(NC(C2CCCC(C(F)(F)F)C2)=O)C1 4536,C(N=C(NC(C)C)N(C)Cc1ccc(Br)cc1)C1(COC)CCCO1 4537,c1(CN2C(CNC(Cc3cccc(NC(C)=O)c3)=O)CCC2)cc(Cl)ncc1Cl 4538,C1(C)(NC(c2nc(C)sc2)=O)CCCCC1C(=O)NCCc1cscn1 4539,CCC(O)CC(=O)NC(c1cccc(Cl)c1)CNC(c1cnn(CC)c1)=O 4540,C(CC(C)(C)CC(=O)NCCN(C(=O)CCCCc1cnn[nH]1)CC(C)O)OC 4541,N1(C(c2cnn(CC)c2Br)=O)CCOCC(CNC(=O)C(O)C(C)(C)C)C1 4542,N1(CC(=O)NCC#CCNC(CCc2c(C)ncs2)=O)CCC(CN(C)C)CC1 4543,C12(C(N(C(C(=O)N3CC(N(CC=C)C)C3)(C)C)C3CC3)=O)CCCC1C2(F)F 4544,C1(C(=O)O)CC12CN(C(c1cccc(Cl)c1)c1ccccc1)C2 4545,N1(C(C=Cc2cnc(C)s2)=O)CC2CC(NC(c3cc(C#N)c[nH]3)=O)C1C2 4546,Cn1ncc2cccc(C(=O)NC3CCC(NC(=O)C4=NOCC4)CC3)c12 4547,c1(-c2n(C(CCC)CO)ccn2)cc(F)cc(I)c1 4548,n1(C(C)C)nncc1C(=O)NCC(C)NC(=O)C(C)(C)c1ccsc1 4549,C1(NC(=O)Cc2ncc(F)cn2)CCCC12CCN(C(c1ccc(Cl)cc1)=O)C2 4550,C(=O)(C1=C(C)OCCC1)NCC1(CNC(C2C(CC)C2)=O)CCOCC1 4551,N1(C(C(CC)OC)=O)CCC2(C1)CN(C(=O)CC1CN3CCN1CC3)C2 4552,N1(C(CC(CC)OC)=O)CCN(C(=O)CCc2ccc(F)cc2F)C(C(C)C)C1 4553,N1(C(Cc2cn(C)nc2Cl)=O)CCCC(NC(=O)C(C)(C)n2cnnn2)CC1 4554,c1(CNC(C2(C)CCNC2)=O)ccc(O)c(CO)c1 4555,Cc1sc(Cl)c(C(=O)NCC2(O)CC(CNC(=O)CCCC#N)C2)c1C 4556,N1(C(CC(C)SC)=O)CC2CCCC(NC(c3ocnc3C(F)F)=O)C2C1 4557,Cc1ccc(C2(C(=O)NCC(C)(CO)NC(c3cc(Br)n[nH]3)=O)CC2)cc1 4558,C(=O)(C1=NOC2(CCC2)C1)N1CCN(C(C(C)=C(CC)C)=O)CC(O)C1 4559,C1(NC(c2nocc2Cl)=O)CCCC1CNC(C1(C(F)F)CCC1)=O 4560,C(=O)(CS(C)(=O)=O)NCC(C)(N(CC(=O)NCc1ccccc1Cl)C)C1CC1 4561,C(=O)(C1CCc2ccccc21)NC(CCN(C(CC(CC)C)=O)C)C 4562,c1(C2(C)C(C(=O)NCC3(C)CCCS3)C2)cccc(Br)c1 4563,C1(NC(c2c(C)noc2)=O)C=CCCC1C(=O)NCC(F)(F)CO 4564,C1(C(=O)NCC2(O)CN(C(CCC3N(C)CCC3)=O)C2)CCC(NC(N)=O)CC1 4565,CC1(C)CCN(C(C2(C(N)=O)CCC2)=O)CC1CNC(C1CCC=CCCC1)=O 4566,c1(C(=O)NCCC(CNC(C(C(CC)O)C)=O)OC)cc2cnccc2[nH]1 4567,N1(C(C2CCN(C3CC4CCC3C4)CC2)=O)CCN2CCC1C2 4568,c1(NC(C(CO)NC(CC2C(CC)C2)=O)=O)cnc(C)c(C#N)c1 4569,C1(N2CC(C)(C#N)C2)CN(C(c2ccc(Cc3ccccc3)o2)=O)CCC1F 4570,c1(OC)ccc(Cl)c(C)c1C(=O)NC1CCCCN(C(c2ccc(F)o2)=O)C1 4571,c1(OC)cc(CNC(=O)NCC(C2CCCCC2)CO)cc(F)c1F 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4608,C(C(=O)N1CCCO1)NC(=O)OCC.C(CC1C(=O)CCC(=O)N1)=CC 4609,C1(C(=O)NCCNC(=O)C(O)Cn2cncn2)(CC)CCCCO1 4610,CCCC(C(=O)OC)N(C)N1CC(C)CCC1C(=O)OC 4611,N1(C(CC2(CN(C)C)CCC2)=O)CCC(CNC(c2cncc(N)n2)=O)C(C)C1 4612,c1(C(N(CCOCCN(C(=O)CC2CCOC2)C)C2CC2)=O)nonc1N 4613,c1(C(N2C(C(=O)Nc3cc(C)c(Br)cc3F)CSCC2)=O)ccc2c(c1)OCO2 4614,C(CCSC#N)(C(=O)NCc1ccc(F)cc1)N1C(C(C)(C)C)CCC1 4615,c1(C(C(=O)NC2CC(C)(NC(C3CC=CCO3)=O)C2)O)ccc(F)c(F)c1 4616,c1(CNC(c2c(C)n[nH]c2)=O)ccc(CNC(=O)C=Cc2cscn2)cc1 4617,C=C(CNC(c1ccnnc1)=O)CCNC(c1cscc1F)=O 4618,c1(C(N2CCC(CC)C2C(=O)N(C(C)CCC(C)C)C)=O)n[nH]c2ccccc12 4619,N12CC(C(O)C1)c1cn(nn1)CC2.c1(CC(C)(C)C)ccc(NC(=O)CCC)s1 4620,c1(CCC)cc(C(=O)NCCC2CN(C(c3occc3F)=O)CCO2)cc(O)n1 4621,C1(COC(=O)Cc2ccccc2)CN(C(C2CCOC2)=O)CC1CC(F)(F)F 4622,N1(C(c2cc(CC)n(C)n2)=O)CC2CC1CC2NC(=O)C1=CCCC1 4623,c1(C(=O)NC2CCN(CCNC(C(CC)(C)O)=O)CC2)cc(C)cc(O)c1 4624,C(=O)(C1=CCCC1)NC(C1CN(C(C23CCCCC2C3)=O)C1)C 4625,c1(C(=O)NCC(CCC)C(=O)N2CCC2CC2CC2)cc2cccnn2c1 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4644,Cc1cc(C(=O)NCC(C2CC2)N(C(=O)CC(O)C(C)C)C)cnc1C(F)(F)F 4645,c1(C(N2C(C)CC(NC(CCSCCC)=O)C2)=O)nsc2ccccc12 4646,C1(CNC(c2c(N)cc(Br)cn2)=O)CCC2(CCC2)C1NC(=O)C=C1CC1 4647,N1(C(C2(NC(c3ccc(C#C)o3)=O)CCCC2C)=O)CC2OCCOC2C1 4648,C1(C(=O)NC(C)CC2CN(C(=O)C(C)(C)C(C)(C)O)C2)CCC(=O)N2CCCC12 4649,Cc1cccc(C2(NCCNC(=S)NCC(C)(C)[N+](=O)[O-])CC2)c1 4650,CC(C)CC(O)C(=O)NCC1CCCC(CNC(=O)C=Cc2cncc(O)c2)C1 4651,C(=O)(C1=CCN(C(C2C3CCC(C3)C2C)=O)C1)NCCCC(C)CO 4652,C(=O)(C(F)(CNC(c1n[nH]cc1Cl)=O)C(C)C)N1CCCC(CCC#C)C1 4653,N(C1CCOc2ccc(Cl)cc21)C(CC(C)Nc1ccccc1)=O 4654,N1(Cc2c(C)cc(Br)cc2)CCN(C(c2cc(C(N)=O)ccn2)=O)C(C#N)C1 4655,c1(C(N2CC(CC)N(C(=O)C(C)OCCSC)CC2)=O)cc(C)c(OC)c(Cl)c1 4656,Cc1ccc(C(=O)NCCC(C)CCNC(=O)C(=O)C(C)(C)C)nc1O 4657,C1(NC(C2CCCCS2)=O)CCN(C(c2ccc(CO)c(Cl)c2)=O)C12CCC2 4658,C1(C)(NC(CN(C2CC(C#N)C2)C(CCc2cnc(C)o2)=O)=O)CCCC1(C)C 4659,c1(C(=O)NC2CN(C(C(CCSC)O)=O)CC2C)cc(Cl)c2n[nH]cc2c1 4660,CC1(C)CN(C(C2CC(C3CCCCC3)C2)=O)CCCO1.C12CCCN1C1C2C1 4661,c1(C(N2CCCC3(NC(C(N)=O)=O)C2C3)=O)cc2cnccc2[nH]1 4662,C=CC1CCCN1C(=O)CC1(C)CCN1C(c1nc(C)c(C)s1)=O 4663,N1(C(CSCCCC)=O)CC(C(O)C(=O)N(C(C)CCO)CC)C1 4664,S(=O)(=O)(c1[nH]c(=NCc2cccc(F)c2Br)ccc1Br)N(CC)Cc1cn(C)nn1 4665,c1(OCC(=O)N(C)CC2N(C(C(COC)O)=O)CCC2)nc(O)nc(O)n1 4666,c1(C(N2CC(NC(C3CC(CC)(CC)C3)=O)C(SC)C2)=O)nc(C)ccc1C 4667,C(=O)(C1=C(C)C(C)(C)OC1=O)N1CC(CNC(C=C(C)C(F)F)=O)C(C)(C)CC1 4668,C1(C(N(CCCC=C)C)=O)(NC(c2snnc2CC)=O)CC(O)C1 4669,c1(C(=O)NC2CN(C(C3CC(C(C)C)C3)=O)C(C)C2)ccc(N)cc1Cl 4670,C1(F)(C(N(CCNC(C(C)C(=O)OC(C)C)=O)CC)=O)CCS(=O)(=O)C1.C(C)(C)C 4671,C(=O)(CC(C)N(C(=O)C(c1cnn(C)c1)CC)C)NC(CCOCC)C 4672,N1(CC(N2CCN(Cc3ccc(C)cc3)CC2)=O)CCCC2(CCCCO2)CC1 4673,CC1CCC(C(=O)NOCC2CCCC2)CN1C(c1csc(CO)n1)=O 4674,c1(NCc2cc(C)[nH]n2)cccnc1C(=O)NC1CCNC(=O)C1 4675,CC(C)P(=O)(CC(=O)NC1CC2CCC1(NC(=O)CCn1ccnc1)C2)C(C)C 4676,n1(C(CC(N2CCC(N(C(CC)=O)CC)C2)=O)C)nc(C)cc1C 4677,c1(C(N(C(CC)C(=O)OC)CC)=O)cc2sc(C)cc2[nH]1 4678,Cc1cc(C(=O)NCCC2CCCN2C(C2CCCCS2)=O)ccc1C(F)F 4679,Cc1ccc(C(=O)O)c(-n2cc(CNC(C3(CO)CCCO3)=O)nn2)c1 4680,CN1CCCC(C(N2CCCCC2C(=O)NCC(O)CCO)=O)C1 4681,C(C(Cl)C(C)(F)F)N(C(CN(C(C1CCC(N(C)C)C1)=O)CC)=O)C1CC1 4682,N1(C(C(F)OC)=O)CCOC(CN(C(=O)Cc2csc(C(C)(C)C)n2)C)C1 4683,N1(C(C2(C)CCN(C)C2=O)=O)CCN(C(=O)CC2CS(=O)(=O)C2)CC12CCC2 4684,C(=O)(C(C)(C)C(C)(F)F)N1CCN(C)C(CNC(C2CC23CCC3)=O)C1 4685,Cc1cc(CC(=O)NCCC2(NC(C3CCN(C(N)=O)CC3)=O)CCC2)n(C)n1 4686,N1(C(C(C2CN(C(c3cnn(C)c3C#N)=O)C2)OC)=O)CCc2ncccc2C1 4687,n1(CC(=O)N(CCCCCCNC(C2(Cl)CC2)=O)C)nnc2ccccc2c1=O 4688,C(C1=CCN(C(=O)CC(O)CNC(=O)CC2CCOC2C)CC1)OC 4689,N1(C(c2c(OC)csc2)=O)CCC(O)CC1C(N1CCC(CF)C1)=O 4690,c1(C(=O)NC(CC#C)C(=O)NC2CCCN(C)C2C)ccc2[nH]ccc2n1 4691,C1(CC(=O)NCCC2COCCN2C(c2cc(CF)on2)=O)CN2CCN1CC2 4692,c1(C(=O)NC2CCC(N(C(CCCCCC)=O)CC)CC2)cc2cccn2cn1 4693,CCC(C(=O)NCCNC(=O)CC1CCC(C)(O)CC1)C(F)(F)F 4694,C1(C(N2CCC(c3n(C)cnn3)C2)=O)=NOC(C)(C)C1 4695,c1(C(N(C2CCN(C(C3C(OCC)C3)=O)CC2)C)=O)cc(N)c(F)cn1 4696,C12(CCC1)C(=O)N(CCCCCCO)CC2.c1(C(=O)NC2CC2)cnn[nH]1 4697,N1(C(CCN(CC=C)C(c2csc(Cl)c2)=O)=O)CCCC(O)C1C 4698,C1(NC(COc2cccc(C)c2)=O)CCN(C(c2nccs2)=O)C12CCCC2 4699,C1(CC(=O)OC)CS(=O)(=O)C2CN(C(=O)NCC3C(C)(C)CCCC3(C)C)CC12 4700,C1(Cn2cc(C(C)CO)nn2)CN(C(=O)Cn2nccn2)CCO1 4701,CC1CCN(C(=O)CSCC(F)(F)F)CC1N(C(=O)C(C1CC1)C1CC1)C 4702,C(N=c1[nH]c2c(c(=NCC3CC(C)(C)C3)[nH]1)CC(C)CC2)c1c(F)ccc(C)c1 4703,c1(CCC)cc(C(N2CC(O)(CC(N3CCC(C(CC)CC)C3)=O)C2)=O)no1 4704,C1(NC(Cc2c(C)cccc2)=O)CC2CCC(C1)C2NC(=O)C1=CCCOC1 4705,N1(C(c2cnc(C)c(N)c2)=O)CCCC2CN(C(=O)C3=CCN(C)C3)CC12 4706,C(=O)(CC(C)(C)C(=O)OC)N1CCCC(C(N(C2CCN(CCC)C2)C)=O)CC1 4707,C(=O)(C(C)(C)C(C)C)N1CCC(N(C(=O)CN2C(C)CCC2C)CCC)C1 4708,N1(C(c2ccc(C(C)=O)o2)=O)CCC2C(NC(c3cnn(C)c3F)=O)C12 4709,c1(C(=O)NC(CCCNC(c2c(C)ccnc2O)=O)C)cnn2cc[nH]c(=O)c12 4710,C(=O)(C(CC(C)C)C(N)=O)N(CC(=O)NC1CC(C)(CC)C1)CC1CC1 4711,N1(C(c2cc(Cl)cc(Br)c2)=O)CCCC2(CCCN(Cc3ncccc3O)C2)C1 4712,c1(C(N2C(CN(C(=O)CC(C)COC)CC)CCC2)=O)cc(N)nc(Cl)c1 4713,N1(C(CCS(=O)(=O)NC)=O)CC2OCCN(C(=O)Cn3ccc(C)n3)C2C1 4714,c1(CN2CNC(=O)C2C2CCOCC2)nc2cc(Br)ccc2o1 4715,c1(CC(=O)NCC=CCNC(C2(CC=C)COC2)=O)cc(F)cc(F)c1 4716,c1(OCC)nccc(C(=O)NCCCCCCNC(c2cnncc2O)=O)c1F 4717,CC(C)CC(CNC(C1C2CC3C(C2)C13)=O)C(=O)N1CC(C(=O)N(C)C)C1 4718,N1(C(CCNC(=O)OCC)=O)CC(NC(C2C(C)(C)C2(F)F)=O)CC(C)(C)C1 4719,C1(C(N2CCC(CN(C(=O)Cc3ccc(Cl)nc3)C)C2)=O)CCC2CC1C2(C)C 4720,C(C)(C(C(=O)NCC1CCN(CC)C1)C(C)C)NC(c1cn(CCC)nc1)=O 4721,CC1CCN(C(=O)Cc2cn[nH]c2)CC1NC(=O)C=CSc1nc[nH]n1 4722,C12(NC(C(C)OCC(C)C)=O)CCCC1N(Cc1cc(C3CC3)on1)CC2 4723,N1(C(C(CCN(C)C)O)=O)CC2(CCC2)CC1C(=O)NC1CCOC1(C)C 4724,Cc1ccnc2sc(C(N3C4CCC3CC(NC(C3CCCO3)=O)C4)=O)c(C)c12 4725,O=C(CN=c1nc(N2CCC(CO)C(F)(F)C2)c2c([nH]1)COC2)NC1CCOC1 4726,C1(NC(=O)COCCCF)COC2(CCN(C(c3coc(Br)c3)=O)C2)C1 4727,c1(NC(c2nc(C)cs2)CC)nc(C)cc(=NCc2cccc(O)n2)[nH]1 4728,c1(CNC(C2N(C(c3cncc(CC)c3)=O)CCC2CC)=O)cccc(C)c1O 4729,Cc1cc(C)nc(N(C2CCCNC2)C(C2CCC(=O)NC2)=O)n1 4730,N(C1CCOc2c(F)cc(F)cc21)Cc1ccccc1C(C(C)n1cccn1)C 4731,c1(C(N(C2CCCCN(C(C(C)S(N)(=O)=O)=O)C2)C)=O)csc(=NC2CC2)[nH]1 4732,N1(C(C=O)=O)CCCC2(C1)CC2(F)F.c1c(Br)nc2n1CCC2.N12CCN1CC2 4733,C1(NC(Cc2c(C)n[nH]c2C)=O)CC2CC(NC(C3CC(O)C3)=O)CC12 4734,S(=O)(=O)(c1cccc(Cl)n1)NCC(N1CC(c2ccccc2)C1)=O 4735,C1(CNC(C(C)NC(CC)=O)=O)CC2CC2N1C(C1CC1c1ccccc1Br)=O 4736,n1(CC)ncc(C(=O)NC2(CNC(=O)C(C)C#N)CCOC2)c1C 4737,CC(CCCCO)N(C(=O)C(CC1CCC1)NC(=O)CCOCC(F)F)C 4738,Cc1cc(C(N2CCOC(C(N(CCCc3ccccc3)C)=O)C2)=O)nn1C 4739,C(=O)(C1=C(C2CCOCC2)N(CCSC)C(=O)NC1c1cc(C)cc(Cl)c1)OC 4740,C1(C)(CC)CC(NC(=O)Cc2cc(C)[nH]n2)CN1C(C1(NC(N)=O)CC1)=O 4741,n1(CC=C)c(N(CC(C)CC(C)C)C)nnc1C1COc2ccccc21 4742,CC1CC(C(=O)N2CC(C)(NC(C3CC(Cc4ccccc4)=NO3)=O)C2)=NO1 4743,C1(NC(c2c(COC)ncs2)=O)C2CC1N(C(=O)CCc1cccc(Cl)c1)C2C 4744,C(CN=c1cc(F)nc[nH]1)(C1CC1)NC(CC(C(C)C)c1ccccc1)=O 4745,N1(C(c2ccccc2Br)C(=O)Nc2ccc(Cl)cn2)CCC2(C1)OCCO2 4746,C1(C(CC)C)CN(C(=O)C(=O)NC2CC(S)C2)C1.C(C)(C)(C)N 4747,c1(Nc2cccc(-n3cc(CCC(CC)C(=O)O)nn3)c2)onc2ccccc12 4748,C12(NC(C(C)Cn3ccnc3)=O)CCC(F)(F)CC1CN(C(=O)C(C)(C)CF)C2 4749,C1(C(=O)NC(CNC(C=CCC(CC)C)=O)COC)CCC(NC(=O)OC)CC1 4750,c1(NC)ccc(C(N2CC3CCCC23)=O)cc1[N+](=O)[O-] 4751,C(=O)(C1CCc2cc(F)ccc21)NC1(C)CCN(c2cc(CC)nc(Cl)n2)C1 4752,c1(CC(N2CC(NC(c3n[nH]cc3Br)=O)C3C2C3)=O)cccc(F)c1O 4753,c1(C(N2C(CN(C(=O)C(Cl)=CCl)C)CC(F)C2)=O)ccc2c(c1O)CCCC2 4754,C1(CC(=O)NC(C=C)CO)N(C(=O)CC2CCC(C)CO2)CCC1(C)C 4755,N1(C(C(=O)NCC(F)F)=O)CC(O)CC1CNC(C1CC2(CSC2)C1)=O 4756,CC(C)(C)S(=O)(=O)CC(=O)N1CCC(NC(=O)CCCN2C(=O)CCC2=O)C1 4757,C1(CNC(C2CC23CCOC3)=O)CC2(CC2)CN1C(=O)C(F)n1cccn1 4758,CC1(C(=O)NCC2CC3(CC(NC(=O)CC(F)F)C3)C2)CCCC1(F)F 4759,N1(C(c2n[nH]c(C)c2C)=O)CC(NC(=O)C(CC2CC2)CC2CC2)CCC1C 4760,Cc1cc(CNC2(C)CCCN2C(C23CC(c4ccccc4)C2C3)=O)ccc1F 4761,N1(C(C(SC)SC)=O)CCCCC(N(C)C(c2ccc(F)c(F)c2)=O)C1 4762,c1(OC)cc(C(=O)NCCNC(c2c(C3CC3)cnn2C)=O)cc2cn(C)nc12 4763,C(CCCCC(=O)N(C)C)c1cn(CC(=O)NC2CSC2)nn1 4764,N1(C(N)=O)CCC2(CC1)CSC2.CC1(C)C2CC1CNC(=O)CCCN2 4765,C1(Cc2nc(-c3ncn(CCC)c3)on2)CCCN(CC(=O)OC(C)C)C1=O 4766,c1(OC)ccc(CNCCCCC2CC2C)cc1C#N 4767,C=C(C)CCCC(=O)N(CCC(C(C)(C)C)NC(=O)CSCc1ccccn1)C 4768,C1(C(=O)NCC(=O)N(C(C)CO)CC2CCC2)C2CN(C)CC12 4769,c1(OC)cccc2[nH]cc(CC(=O)N(C)CC3(O)CCC(F)(F)CC3)c12 4770,C(=O)(C(F)(F)CO)N1CC(CNC(c2ccn(C(C)(C)C)n2)=O)C1 4771,C=CCC(C)(C)CNC(=O)C(C1CCN(C(=O)CP(C)(C)=O)C1)F 4772,CC1C(NC(c2cnnc(Cl)c2)=O)CC2CCC1N2C(=O)C1=CCCC(C)(C)C1 4773,N1(C(c2c(C)nc[nH]2)=O)CCN(C(=O)CSCC(C)C)CC1CCO 4774,N1(C(C(C)Cc2cnc[nH]2)=O)CC2CCCCC2(NC(c2cc(Cl)ccn2)=O)C1 4775,c1(C(N2CCOCC2C2CCOC2)C(=O)NCC)cc(OC(C)C)cc(CC)c1 4776,c1(C(=O)OCC)c[nH]c(=N)nc1NC(C1CC1CNC(C1(OC)CCCC1)=O)=O 4777,C(c1cc(Cl)ccc1Cl)=CC(N1CCN(C(C(C)(C)OC)=O)CC1)=O 4778,C1(C(=O)NC2(CN(C(CCc3c(C)ncs3)=O)C)CC2)CCC2(CC1)CC2(F)F 4779,c1(CNC(C(CO)NC(C2C(C)CC2)=O)=O)ccc2c(c1)CC2 4780,c1(C(=O)NC(C)CNC(=O)C=CCOCC(F)(F)F)snc(Cl)c1Cl 4781,C(C(C(=O)NC1CC1)N(C1CCCC1)CCCC)(CC(C)C)OC 4782,CCC(C)CC(=O)C(=O)NC1(CN(C)C(c2ccc(CN(C)C)o2)=O)CC1 4783,C1(CNC(C(C(C)(C)C)SC)=O)CC12CCN(C(c1csc(CO)n1)=O)CC2 4784,c1(N(C(C)=O)C)ccccc1C(=O)N(CC(C)CNC(C1CC(N=[N+]=[N-])C1)=O)C 4785,CCCCC(C)CCC(=O)NC1COCC1NC(c1cc(Br)cs1)=O 4786,CC1CN(C(=O)CSc2cnn(C)c2)CCC1NC(=O)CC1CCC(=O)C1C 4787,C(c1ccc(Cl)c([N+](=O)[O-])c1)=CC(N1C2CC(OC)C(C2)C1)=O 4788,C(CCCCC(=O)N1CCN(C(c2cnc(C)nc2)=O)C(C2CC2)C1)NC(C)=O 4789,c1(C(=O)NCC2N(C(C(C)SCc3ccccc3)=O)CCC2)c(O)cccc1F 4790,C(c1cncn1C)=CC(=O)N(CCC(=O)N(CC(O)C1CCC1)C)CC 4791,N1(C(CC(=O)N(CC#C)CC)=O)CCC2CC1CN2C(c1cccc(C)n1)=O 4792,c1(SC)ccc(C=CC(=O)NCC2CC(NC(C3(c4ccsc4)CC3)=O)C2)s1 4793,C1(N(c2cccc3c2OCC3)C(C2OCC(C)C2)=O)CCC2(CCNC2)CC1 4794,CC(C)C(CC(=O)N(CCCNC(c1nccc(Cl)c1F)=O)C)c1ccccc1 4795,C1(NC(c2cn(CC=C)nn2)=O)CC2(C1)CC2C(=O)NCC1CC(F)C1 4796,Cc1cccc(NC(=O)NCC(c2ccc(C3CC3)cc2)(C)C)c1F 4797,C12CN(C(C)(C)C1)C(=O)N1C(C(C)(C)CC1)CCN2.C(C)(C)(C)OC(C)=O 4798,C1(C(=O)NC(C(=O)NC)C)CN(C(C2CC(C)=NO2)=O)CC12CC2 4799,c1(CNC(CC2(CC)CCC2)=O)cc(C(=O)N(C2CC2(C)C)C)on1 4800,CCCCC(C(=O)NC1(CO)CC(C)C1)NC(c1cc(C)c(CC)o1)=O 4801,c1(CCNC(C=CC(C)(C)NC(c2cc(O)cs2)=O)=O)ccncc1F 4802,C1(CC)CCC(C)N(C(=O)CCCN(C(=O)C(C)(COC)OC)CC)C1 4803,CCC(C)CC(CO)NC(=O)CC(CC)N(C(=O)CC1CC(=O)NC1=O)C 4804,Cc1nc2ccc(-n3cc(C4CCN4C(c4cccc(O)c4)=O)nn3)cc2o1 4805,C(=O)(C(F)CCC(C)C)N1C(C)CCC(NC(c2c(C)n(C3CC3)cc2)=O)C1 4806,Cc1n[nH]c(=NC2CCCC(NC(c3cnn(C4CCC4)c3C)=O)C2)s1 4807,c1(C(N(CCC2N(C(c3c(CC)c[nH]n3)=O)CCCC2)C)=O)c[nH]cc(C)c1=O 4808,N1(CC)CCCCC1C(N1CC=CC(NC(C2(C(F)(F)F)CCCC2)=O)C1)=O 4809,C1(NC(CCCC(C)C)=O)CCN(C(=O)Cc2ccon2)C12CCCC2 4810,C1(CNC(C2(CCC)CC2)=O)CC2(CCN(C(C3(C)C=CCC3)=O)CC2)C1 4811,c1(C(N2CCOC(C3CCOCC3)C2)=O)[nH]cc2c1CCC2 4812,c1(C(=O)NCC2C3CN(C(CCCCCC)=O)CC32)cc2n(n1)C(C)CCC2 4813,c1(OC)c(C(=O)NC(CN(C)C)C(=O)NCC2CC(F)C2)cnn1C 4814,c1(CN(C)NC)cc(OC)c(OCCO)cc1-c1ccc(CC(C)CC(=O)O)cc1 4815,N1(C(CC(C)SC)=O)CCC(F)(F)C(CNC(C2(C)CC(C)(C)C2)=O)C1 4816,C1(NC(=O)CN2CCCS2(=O)=O)CC2CCC1N(C(C1CC(C(F)(F)F)C1)=O)C2 4817,C1(CNC(c2c(C)cco2)=O)CC2COCC2N1C(c1cc2cccnn2n1)=O 4818,C12(C(=O)NCC3OCCN(C(C=CCOC)=O)C3)CC(C)(C1)OC2C 4819,N1(C(C(CCCC)O)=O)CC(NC(c2ccncc2)=O)C2CCCC12 4820,c1(C(N(C2CCN(C(=O)CC3CCCO3)C2)C)=O)ccnc2c1CCC2 4821,c1(C(=O)NC2C(NC(Cc3ccc(OC)cc3)=O)CCC2)cc(O)nc(O)n1 4822,C=CCC(C(=O)N1CCC(OCC)C1)C(C)C.C12(CCCCO1)OC2 4823,C(CC(C)C(=O)NCC1CCN1C(=O)CN1CCCCC1)OC 4824,C1(CC(=O)NCc2occc2C(=O)NCCCCC2CCCC2)OCCCO1 4825,CC1CN(C(c2c(F)cccc2Cl)=O)CCN1C(c1ccc(C2CC2)cc1)=O 4826,N1(C(C2CN(C)C2)=O)CCOCC12COCCN(C(C1C3CCCCCCC13)=O)C2 4827,N1(C(C=Cc2ccc(C)nc2)=O)CC2(CCN(C(=O)CC3CCOC3C)C2)C1 4828,C(CCCCC(=O)NC1CCC(C(=O)NCC(C)CC2CCC2)C1)SC 4829,c1(CNC(C=C(C)CNC(=O)CN(CC(C)(C)C)C)=O)cnc(C)c(C)c1 4830,CC(C(F)(F)C(F)(F)F)NC(=O)Nc1ccc(Br)c(Cl)c1F 4831,S(=O)(=O)(c1ccc(SCCNC(c2ccc(CC(=O)O)cc2)=O)cc1)NC(C)C 4832,c1(OC)ncc(C(=O)N(C2CCCCC2)CCOC(C2(C(C)C)COC2)=O)cc1Cl 4833,CC(C)CCCCCC(=O)NCC12CCCCC1N(C(=O)C=CI)CC2 4834,n1(CC(=O)NC(C(=O)N(C)Cc2cnn(C)c2)C2(O)CCC2)[nH]cnc1=N 4835,C(=O)(CCCC(N)=O)NC(C)CCNC(=O)C(=O)NCC(F)F 4836,CCCCCC(O)C(=O)NCC1CC1CC(N1CC(c2ncc[nH]2)C1)=O 4837,c1(OCC)cc(C(=O)NC(C(=O)NCc2csc(C)c2)C2(O)CCC2)[nH]n1 4838,c1(N(C)Cc2nc(C)[nH]n2)nc(NCCN2CCNC2=O)c2ncn(C(C)C)c2n1 4839,C(=O)(C(O)C(F)(F)F)NCC(C)(C)NC(c1cn(C)c(O)n1)=O 4840,c1(N2CCC(C=C)CC2)nc2c(c(=NCC3CCC=CCCC3)[nH]1)CCC2 4841,c1(C(N2CCCC(C(c3c(C)nc(C)s3)=O)C2)=O)c(C#N)c(C(C)(C)C)nn1C 4842,C1(n2c(C(CCC=C)NCc3cc(Br)no3)nnn2)CCC(F)(F)CC1 4843,c1(C(N2CCCC(NS(CC)(=O)=O)CC2)C)cccc2ccccc12 4844,C(=O)(CC1OCc2ccccc21)NCC(C)NC(c1n(CC)nnc1)=O 4845,C1(C(=O)OC)CC2CC(NC(=O)Cc3cnc(C)nc3O)C2C1 4846,C(CC(=O)NC1CCC(CNC(=O)C(C)CC2CCC2)C1)(OCC)OCC 4847,N1(C(C2C(C)(C)CO2)=O)CC2CC(NC(=O)CCCC3CCCCC3)CC2C1 4848,c1(C(=O)NCCN(C(c2[nH]nnc2C(F)F)=O)CC)cnc(O)n1CC 4849,N1(C(CCN(CC)CC)=O)CCC(C(C)(C)C)(CNC(=O)Cc2sccc2C)C1 4850,Cc1noc(N)c1C(N1CCC(NC(c2csc(C(F)(F)F)c2)=O)C1)=O 4851,c1(C(=O)NCC(C)NC(c2ccc(Oc3cccnc3)cn2)=O)nnc(S)n1C 4852,N1(C(CC(CC)C2CC2)=O)CC(NC(C2CCN(OC)CC2)=O)C2(CC2)C1 4853,CC1(C)C(CC(N2CC(CC(N3CCC(O)CC3)=O)C2)=O)CCN1CCO 4854,C1(C(N2CCC(NC(Cc3cccc(C#N)c3)=O)CC2)=O)CCc2ncnn2C1 4855,S(=O)(=O)(c1cccc(N(C)Cc2ccc3ccccc3c2)n1)NC1C(C)CSC1 4856,C12(CCOC)CN(C(=O)C(c3ccnc(C(F)(F)F)c3)(C)C)CC(CO)(C1)C2.C(C)(=O)O 4857,N1(C(C(CC)(C)OC)=O)CCCC(CC)(NC(=O)CCc2ccccc2F)C1 4858,CC(C)S(=O)c1ccc(C(=O)NC2CN(C(C3CCCC3)=O)CCC2CO)cc1 4859,N1(C(c2ccc(-c3c(C(=O)O)snc3O)cc2)=O)CCC(C2CC2)CC1 4860,n1(CC(=O)N(C)CC2COCCN2C(=O)Cn2ncnn2)cc([N+](=O)[O-])cn1 4861,c1(C(=O)OC)ccc(S(=O)(=O)NC2CCCN(C(c3cncs3)=O)C2)cc1 4862,C1(CC=C)(NC(=O)CC(O)CCSC)CCCN(C(c2ccc(CSC)o2)=O)C1 4863,N1(C(C=CC=CCC)=O)CC2OCC(NC(=O)CCCCCCC)C2C1 4864,c1(C(=O)NC2CN(C(c3ccc(C(N)=O)s3)=O)C3C2C3)nccc2cc[nH]c12 4865,CC1CN(C(=O)C(CC(N)=O)NC(c2cnc(O)o2)=O)C(C)CO1 4866,c1(NC(C2(CCl)CN(C(=O)CC3CCCCO3)C2)=O)cccc2cccnc12 4867,c1(C(=O)O)ccnc(N(C2CCCC2)C(C2CCCO2)=O)c1I 4868,c1(C(N2CCCCC(NC(C(CC)(F)F)=O)C2)=O)cc2c(cn1)NC(=O)CO2 4869,C(CC)(CCCC(=O)NCC(C)(F)C(C)(C)F)NC(CC(=O)NCC#C)=O 4870,c1(C(N2CCCN(S(=O)(=O)c3nccs3)CC2)=O)noc2c1CCCC2 4871,C(CC(C(=O)NCC1CC=CC1)NC(=O)C1=NOCC1)OCC 4872,Cn1cc(C(=O)NC2CCCN(C(=O)CCC3CCCCC3)C2)c(O)nc1=O 4873,c1(OC)cc(C)ccc1C(N1CC2CC1CN2C(C1C2CCC(F)(F)C12)=O)=O 4874,CC1CCC(C)(C(N2CC(NC(=O)CC(C)F)CC(O)C2)=O)CC1 4875,c1(NC(CC)=O)ccc(C(=O)NC2CCN(C(=O)C(C)(O)C3CC3)C2)cc1 4876,c1(C(N2CC(OC)C(NC(=O)C=CS(C)=O)C2)=O)ccc(C)c(C(F)(F)F)c1 4877,C1(C(=O)NC2CCN(C(C(CC)(C)O)=O)C2)CC(C(C)C)=NO1 4878,c1(-c2n(C(C=C)C)nc(C(C)CC)n2)ccc(C)c(Br)c1 4879,Cc1c(Cl)cc(NC(=O)CC2CC(NC(=O)Oc3c(Br)ccnc3Br)C2)cc1Cl 4880,CCS(=O)(=O)c1ccc(C(N2CCC(C(F)F)C2)=O)cc1 4881,C12(C(=O)NC(c3ccn(C)n3)CC)CC1CCN2C(=O)CC1CC(C)=NO1 4882,N1(C(c2ccc(SC)cc2)=O)CCC12CN(C(C1(C)CCC(C)C1)=O)C2 4883,c1(NC(CCS(N2CC(OC)C(CO)CC2)(=O)=O)=O)ncc2sccc2n1 4884,c12ccc(cc1)C(CCC)(C)NC2.C1(SCC)CC1(Br)Br 4885,CCCCC(CC(=O)N(C(C)CC(C)CC)C)NC(=O)CC1(C)CC1 4886,N1(C(C2(C)CC(OC)(OC)C2)=O)CC2(CCC(CNC(=O)C(O)C(C)C)O2)C1 4887,c1(OC)cc(C(=O)Nc2c(Cl)c(C)nn2C)cnc1-c1[nH]c(C)nc1C 4888,C1(N(C)C(c2cnc(S)n2C)=O)CCCCN(C(=O)CC2CCCC(C)(C)O2)C1 4889,c1(C(=O)NCC2N(C(C(CC)(C)O)=O)CCCC2)ccc(C)n(C)c1=O 4890,c1(C(N2CCCC(CN(C)C)C2)C(=O)NCCCF)cc(Br)ccc1F 4891,c1(OCC(N2CC(F)(CNC(c3c(C)con3)=O)C2)=O)c(C)cccc1Cl 4892,C1(C(=O)NCC2CC(CNC(C3CC4C=CC3C4)=O)C2)CCCCCC1(F)F 4893,C1(F)(C(=O)NC2C(OCC)CC2)CCCN(C(=O)C(C)CC2CCC2)C1 4894,N1(C(C(C)C#N)=O)CCC(c2cc(CNC(C3CCN3C(C)(C)C)=O)on2)CC1 4895,CN1CCN(C)C(CN(C2CCC2C(F)(F)F)C(=O)CC)C1 4896,c1(C(=O)NC(C(C)NC(C2CCS(=O)(=O)C2)=O)(C)C)ccnn(C)c1=O 4897,CC1(C(N2CCCC(NC(c3coc(CC4CC4)n3)=O)C2)=O)CC2(CCC2)C1 4898,N1(C(C2(C)ON=C(C)C2)=O)CCN(C(c2cnc(O)n2C)=O)C(CC2CC2)C1 4899,N1(C(C(C=C=C)C)=O)CC2CCN(C(=O)Nc3cc(SC(F)F)oc3C)CC2C1 4900,c1(C(N2CC3C(NC(c4n(C(C)C)cnc4)=O)C3C2)=O)c[nH]c2cccnc12 4901,N1(C(c2cccc(CNC(c3ncc(O)cn3)=O)c2)=O)CC2CCC(C1)O2 4902,Cn1c(C(N2CC(F)(F)CC2CCNC(C2CC3(CC3)C2)=O)=O)cccc1=O 4903,c1(NC(C2CC(F)CN(CC3CCC(F)(F)CC3)C2)=O)ccc(C(F)(F)F)cc1O 4904,C(=O)(C(O)CC[S+](C)C)N1CCC(NC(c2c(C)oc(C(C)(C)C)c2)=O)C(O)C1 4905,C#CCC(C(=O)N1CCC(N(C(=O)CN2CCC(C)(O)C2)CC#C)CC1)C1CC1 4906,C1(CNC(CCCNC(C2SCC(=O)C2)=O)=O)CC(O)C12CCC2 4907,C1(C(=O)NCC=CCNC(C(N2CCC(O)CC2)C)=O)CCCC(CF)C1 4908,Cc1cc(C(=O)NC2(c3ccccc3)CN(C(=O)C=C3CCOCC3)C2)n[nH]1 4909,C1(C(=O)NCC2(C(=O)NC(c3ccncc3)C)CC(C)(C)C2)CCC(C#N)CC1 4910,C1(C(N2C(CN(C(=O)CC3CCC34CCC4)C)CCC2)=O)CCC2(CC1)CC2 4911,N1(C(CS(=O)(=O)NCC)=O)CCCC(NC(c2cnc(C)s2)=O)CC1 4912,C(=O)(CCCCCOCC)N(CCC)CCNC(=O)CSc1n[nH]c(O)n1 4913,Cc1nn(C)c(C)c1CC(C)C(=O)NCC(CO)NC(=O)CN1CCCCCC1 4914,c1(CC)conc1C(=O)NCC=CCNC(C1(O)CC(c2ccccc2)C1)=O 4915,n1(CC)cc(C(=O)NC(C)C(C)NC(c2cc(C(F)(F)F)ns2)=O)nn1 4916,c1(C(=O)NCCOCCN(C(c2c(CC)onc2)=O)C)cc2n(c1)CCC2 4917,c1(C(=O)NCC2(NC(c3cc(SC)oc3)=O)CC2)c(F)cc(Cl)cc1Cl 4918,N1(C(C2CN(C(c3cc(C)c(F)cc3)=O)CC(F)C2)=O)CCCC(S(C)(=O)=O)C1 4919,CCCCC(O)C(=O)NCC(C1CCC1)NC(=O)Cc1ccc(OC)cc1F 4920,N1(C(CCC)=O)CCOC(CNC(C2CC(C(F)F)C2)=O)C1 4921,c1(C(N)=O)ccc(NC(=O)Cc2cccnc2F)cc1Cl 4922,Cc1cc(C)c(C(=O)NC(C)C(C)NC(c2coc(N(C)C)n2)=O)cc1N 4923,CC(O)CC(=O)N1CC(NC(=O)CC2CC(N(C)C)C2)C1 4924,C12(NC(CC3(C)CC3)=O)CC3CC(C1)CC(NC(C1CCCC(O)C1)=O)(C3)C2 4925,Cc1cc(O)cc(C)c1C(=O)N(C1CCN(C(c2cccc(F)c2F)=O)CC1)C 4926,c1(-c2onc(CNCCC(c3ccc(N(C)C)cc3)OC)n2)cccc(F)c1 4927,CC1CCCCC1(CNC(=O)CCn1ncn(C)c1=O)NC(C1CC(=O)N1)=O 4928,c1(C(=O)NCCN(CC(=O)NCC2CCCS2)CC)cccnc1 4929,N1(CC(=O)N(CCCN=[N+]=[N-])C(C)CO)CC(=O)NCC1C(C)C.CS 4930,N1(C(C(CC=C)C)=O)CCCCC(NC(c2ccc(N3CCCC3)cc2)=O)CC1 4931,C1(NC(C2N(C)CCC2)=O)CN(C(=O)CCc2ccc(=N)[nH]c2)CC12CCC2 4932,N1(C(c2ccc(C#C)nc2)=O)CCC2CCN(C(c3scnc3Cl)=O)C2C1 4933,c1(C(=O)NCCN(C(C(CC)C(=O)OC)=O)CCOC)cc2cncn2c(O)n1 4934,CCCCS(=O)(=O)NC(C)C(N1CC(N(C)C(c2[nH]ccc2C)=O)C(O)C1)=O 4935,N1(C(CNC(CCCCC)=O)=O)CCN(C(=O)C(C)CO)CC1C(F)F 4936,C(=O)(CC(C)(C)C(F)F)N1C(CC(N2CCC(N(C)C)CC2)=O)C2CCCC21 4937,C1(C(N2C(CC(=O)NC(COC)COC)CC(F)C2)=O)CCOC(C)(C)C1 4938,C1(C(=O)NCc2nc(C)sc2)C=CCN(C(=O)C(F)CC2CCOC2)C1 4939,N1(C2CN(C(=O)OC(C)(C)C)C2)CC(NC(C2CC2(C)C(F)(F)F)=O)CC1=O 4940,N1(C(C2(CCC=C)CN(C(=O)CC=CC)C2)=O)CC2CCC1C(O)C2O 4941,c1(C(=O)NC(C2CCOC2)CNC(c2c(C)ccs2)=O)nc2c(s1)COCC2 4942,C(=O)(C1CCC(NC(=O)NCCc2cc(Cl)cc(Cl)c2)c2ccccc21)OC 4943,Cc1ccc(O)cc1C(N1CC2CC(C1)N2C(c1nc(Cl)ccc1F)=O)=O 4944,N1(C(C(C#C)(C)C)=O)CCC2C(C1)CN2C(C1CC2(CCOCC2)C1)=O 4945,N1(C(CCN(C(=O)COC2CCOC2)CCCO)=O)CCCC2(CCCO2)C1 4946,CCCCC(C)C(=O)NCC12CC(CNC(=O)CC3COC(C)(C)CO3)(CO1)C2 4947,C1(CC)(NC(=O)C=CSCc2ccco2)CN(C(=O)CNC(c2ccoc2)=O)C1 4948,c1(CN2CC(NC(c3cccc(O)c3Br)=O)C(F)C2)ccc(Br)c2nsnc12 4949,c1(C(N2C3(C(=O)NC4C(OC)C(O)C4)CC3CC2)=O)cccc(F)c1F 4950,c1(CNC(C2(COC)CC2C)=O)cc(O)nc(C2CCC2)n1.C(=O)(CO)NCC1CC1 4951,c1(OCC)ccc(C(=O)N(CCCNC(c2cn(C)nc2Cl)=O)C2CC2)cc1 4952,N1(C(C(C)(C)OC)=O)CCCC(O)(CNC(=O)C(F)(F)CN2CCCC2)C1 4953,c1(C(=O)NC(C)Cc2nccn2C)n[nH]c2c1CN(C(=O)CCOC1COC1)C2 4954,CC1CC2(CCN(C(=O)C(C)n3cncn3)CC2)CN1C(=O)Cc1ccncc1 4955,c1(C(=O)NC(C(CO)NC(c2c(Cl)nc(OC)s2)=O)C)ccc(=O)n2c1CCC2 4956,C(=O)(C1=C(C)N(C2CCC2)C(=S)NC1c1cc(I)c(Br)c(F)c1F)NC(C)=O 4957,C1(C(=O)NCCC(CCC)C2CC2)CC2(CCC2)CN1C(=O)C1=NOCC1 4958,C(C)(CCN=c1c(Cl)c[nH]cc1[N+](=O)[O-])NC(CCCc1cc(C)no1)=O 4959,c1(C(=O)OC)ncccc1CNC(=O)NCc1ncc(C)n1C 4960,c1(C(=O)NC2(CF)CCN(C(C(C=C)(C)O)=O)C2)cc(C)nc2c1nc(C)n2C 4961,C(=O)(C1CCCn2nccc21)N1CCC(C)C1CNC(=O)CCCC1CCCC1 4962,N1(C(c2nc(C(C)OC)sc2)=O)CCCCCC1CNC(C1CC=CC1)=O 4963,C(C)(CCC(C)C)OC(CC1ON=C(C)C1)=O 4964,N1(C(C(C)CNC(C2CC2(F)F)=O)=O)CC2CN(C)CC2C1 4965,c1(CNC(CC2OCCN(C(CCCOC)=O)C2)=O)ccc(F)c(O)c1 4966,c1(NCCCCC#CC)[nH]c(=NC2CSc3ccc(F)cc32)nc2sccc12 4967,CC(CN(C)C)CC(=O)N1CCC(NC(c2cccc(C(=O)NC3CC3)c2)=O)C1 4968,C1(C2CCN(C(=O)C=Cc3ccc([N+](=O)[O-])s3)C2)(NC(CCSC)=O)CC1 4969,CC(=O)CCCC(=O)NC1(C(N(C)C(C2CCC(C3CC3)O2)=O)C2CC2)CC1 4970,C1(NC(=O)NC2CCC3(C(=O)OC)C2C3)CCC2OCCC2C1 4971,C12(NC(c3ccncc3Cl)=O)CCCCC1N(C(c1cncc(Cl)c1)=O)CC2 4972,CN1CCOC2CN(C(C3(CNC(=O)COC4CCC4)CC=CC3)=O)CC12 4973,C1(C(=O)NCCCNC(=O)CC2CCC3(CCC3)OC2)CC2C=CCC(C1)C2 4974,c1(C(=O)NCC2CN(C(CCC(C)C)=O)CC2O)cn2c(n1)C(C)CCC2 4975,C1(C)(NC(CC2(NC(c3cc(OC)no3)=O)CCC2)=O)CCCC1C 4976,C1(C2CCC2)(C(=O)NC(C2CNCCO2)C)CC1 4977,Cc1cc(C(=O)NCCN(C(=O)C(c2ccc(Br)cc2)=O)C)nnc1C 4978,C1(CC=C)(NC(=O)C(F)=CC)CCCN(C(=O)Cc2cc(Br)cs2)C1 4979,Cc1cncc(C(N2CCCCC2CC(=O)NCCC(C(C)C)N(C)C)=O)n1 4980,c1(C(N2C(CNC(CC(C=C)CC)=O)C(C)CCC2)=O)ccnc2c1CCC2 4981,C1(NC(C2(CC)CC2)=O)COCCN(C(c2cccc(OC)c2Cl)=O)C1 4982,c1(C(N(C)OC2CCCC2)=O)cc2c(cc1[N+](=O)[O-])C(=O)NC2=O 4983,C1(O)(C(C)NC(=O)C=CC2CC2)CCN(C(c2cc(C3CC3)no2)=O)C1 4984,C1(CC(=O)NC(CNC(C2C(C)(C)C2)=O)(C)CO)CCC2(CCC2)O1 4985,Cc1cnoc1Cn1cc(CCCNC(c2[nH]nnc2-c2ccccc2)=O)nn1 4986,C1(C(=O)N(C)Cc2n[nH]c(C)n2)(OCCCCC)CC1(C)C.C1C(=O)N1 4987,C12(NC(c3cc(N4CCCCC4)ccn3)=O)COC(CNC(C3COC3)=O)(C1)C2 4988,N(S(=O)(=O)N(C)C)CC(=O)N(C)CC1N(C(C2CCN(C)C2)=O)CCC1 4989,C1(CNC(c2nc(C(C)NC(C3(SC)CC3)=O)oc2)=O)CC(O)C(O)C1 4990,C(=O)(CC(C(F)(F)F)NC(=O)CNc1ccccn1)N(C1CCN(C(C)=O)C1)C 4991,c1(C(=O)NCC(C(=O)NCCSCCO)N(C)C)cccc(F)c1N 4992,C(=O)(CC(O)c1cnc(Cl)s1)N(C(CNC(C1(CCC=C)CC1)=O)C)C 4993,C(C(C(=O)NOC(CO)C(C)C)NC(C1CC2(CCO1)CC2)=O)OC 4994,CC1(C(=O)NCC(CO)NC(C2CCCCO2)=O)Cc2ccccc2C1 4995,C1(NCC2CCCC(C(=O)OC)CC2)CCC2(CCCNC2)C1 4996,c1(OC)ccc2[nH]nc(CNS(=O)(=O)Cc3cccc(Cl)c3OC)c2c1 4997,c1(C(=O)NCC(CC)NC(C2CCS(=O)CC2)=O)cccc(C(C)(F)F)c1 4998,C1(CNC(c2cccc(C3(C)CC3)c2)=O)CC2(C1)CN(C(=O)C#CC1CCC1)C2 4999,N1(C(=O)Nc2cc(C)sc2)CC(C)OC2(CCC2)C1 5000,C1(NC(CCCc2onc(CC)n2)=O)CCC(C)(CNC(=O)Cc2ccco2)C1 5001,c1(C(=O)NC2CC(N(C(=O)Cn3cccn3)C)C2)cc(Cl)cc2ccccc12 5002,N1(C(C=C=C(C)C)=O)CCC(CNC(=O)CC2CCCO2)C(C2CC2)C1 5003,C(=O)(C(C)C(F)F)NCC(N(C(Cc1cc(C)no1)=O)C)C1CC1 5004,C(=O)(C(F)C(C)CC(C)(C)C)NCC(C)(C)NC(C1CCC(C(=O)OCC)C1)=O 5005,c1(C(N2CC(CNC(CC(=O)OC)=O)C3(C2)CC3)=O)ccccc1N=S(C)(C)=O 5006,c1(C(C)C)ccccc1C(=O)NC(C)(C)CN(C(=O)CC1CCN(C)C1)C 5007,c1(C(=O)NC(C)CC2CCOC2)ncoc1CNC(=O)COc1ccsc1Cl 5008,c1(C(=O)NC(CC=CC)C(=O)N2CCC(C)(CC)C2)ccc(C)cc1C 5009,C1(COC)(CNC(=O)C(C)(C)c2ccc(Cl)s2)CN(C(c2cnc(C)s2)=O)C1 5010,c1(C(C(=O)NC2CCN(C(C(C)N3CCC3)=O)C2)=O)ccc(O)cc1 5011,N1(C(CC2CCC(=O)NC2=O)=O)CCC(C2(NC(=O)CN3CCCCC3)CC2)C1 5012,C(=O)(C1CCc2c[nH]nc21)N1C(C(C)NC(c2cccc3nccn23)=O)CCC1 5013,C1(NC(CN(C(C)C)C(c2ncsc2N)=O)=O)CCCCCC1(C)C 5014,c1(NC(=O)NC2CCN(CCC)CC2)cc(I)nc(C)c1C 5015,C12(OC)CCC(C(=O)NC3CCC(C)N(C(c4ccon4)=O)C3)(CC1)CC2 5016,C1(NC(C(C)OCCCC)=O)CN(C(=O)C(c2ccccc2)C)CC(C)(C)C1 5017,CC(C)CC(C)(O)CNC(=O)CNC(=O)Cc1ccc(C#N)cc1 5018,N1(c2ncc(C)c(C)n2)CCCC(C)(C)C1CNC(=O)C(C)(C)N(C)C 5019,CCCCCCC(=O)NC1CC2(C1)CN(C(=O)C(C)C(C)c1ccc(F)cc1)C2 5020,c1(N(CC)CC)ccc(C(=O)NC2CC(NC(c3ccoc3Br)=O)C2)cc1 5021,C(=O)(C1c2ccccc2CN1Cc1snc(Cl)c1Cl)N1CC(c2n(C)cnn2)C1 5022,C1(CNC(c2c(OC)cncc2)=O)CCCCN(c2cc(C)nc(CO)n2)C1 5023,c1(C(=O)NC2CC(C)(CNC(C3C(C#C)C3)=O)C2)cccc(Cl)c1C(F)(F)F 5024,C(N=c1[nH]c(C)cc(=NCC(C)N2CCC(C)CC2)[nH]1)C1CC(OC)C1 5025,c1(OCC)cc(C(=O)N(C2CCN(C(C3CC34CCC4)=O)C2)C)cc(Cl)c1O 5026,C(=O)(CC(C)CN(C)C)C(CC=CC(N1C(CCCC)CCC1)=O)(C)C 5027,CCC(C(=O)NCCCCN(C(=O)Cn1ccc(Br)n1)C)N(C)C 5028,c1(C(=O)NCC(C)(O)CNC(C2CCS(=O)CC2)=O)cccc(F)c1O 5029,Cc1cc(O)nc(NC(=O)C(=O)NC(c2ccncc2)C2CCCCC2)n1 5030,C1(C(=O)NC2C=CC(CNC(CC3(C)CCC3)=O)C2)CCC12CCC2 5031,Cc1cc(CN2CCCC(CC3CCNC3)C2)cc(C)c1 5032,C1(NC(c2nc(C(C)C)sc2)=O)CN(C(C23CSC(C2)C3)=O)CC1(C)C 5033,N1(C(c2cn(C)nn2)=O)CCN(C(c2ncc(Br)cc2Cl)=O)C2CC12 5034,n1(C(C(=O)NCC(CCOC)NC(c2cnn(C)c2C)=O)C)nc(C)cc1C 5035,C(CC(=C)Cl)(C(=O)NCCC1CCOCC1)NC(C(CC=C)NC(C)=O)=O 5036,C(=O)(C1=NN(C2CC2)C(=O)CC1)N1C(CNC(C(CCCCC)O)=O)CCCC1 5037,CCCCC1CN1.c12ccc(cc1)C(=O)NCCO2.C(=O)(C(C)C)NCC 5038,C(=O)(CC(C)(F)F)NC(CNC(C1C(COC)C1)=O)C1CC1.c1ccc(F)cc1 5039,CCCC(C)(CC)C(=O)NCC1(F)CCC(CNC(=O)CNS(=O)(=O)N(C)C)C1 5040,CCCCC(C)CCC(=O)NC(C)C(C)(C)NC(c1nc(CC)c[nH]1)=O 5041,c1(C(=O)NC(CCSC)C(=O)NO)ccc2c(c1)OCO2 5042,CCCC(CNC(=O)C(C)(C)c1ccno1)C(=O)N(C)CC1CC1(C)C 5043,c1(C(N(CC(C)NC(=O)Cc2cn(CC)nn2)CC)=O)cc2c(C)cccc2o1 5044,C1(NC(C=NOC)=O)(CO)CCN(C(c2c[nH]nc2-c2cnn(C)c2)=O)CC1 5045,C(CCC)(C(=O)N(C1CCCC(NC(=O)CCC2CC(OC)C2)C1)C)=CCC 5046,C1(NC(CC2C(CN)C2)=O)CCCCC1CNC(=O)CC1CC2CCC1C2 5047,C(=O)(C1Cc2ccc(Cl)cc21)N(CCNC(c1cc(C(C)C)nc(O)c1)=O)CC 5048,N1(C(COCc2cccc(C)c2)=O)CCCC12CCN(C(c1ncoc1C)=O)C2 5049,C1(NC(=O)C(c2ccccc2)F)CCN(C(=O)CC(O)c2cnc(Cl)s2)CC1 5050,O=C1NC2(NC(N3CCC(Cc4ccccc4)C34CCC4)=O)CC3CC1C2C3 5051,C(=O)(CC(C)C(F)(F)C(F)(F)F)N1CC(NC(COCC)=O)C(F)CC1 5052,CCC(C)C(C(=O)NC(CC(C)C)C(=O)N1CC(C)C(C)C1C)N(C)C 5053,Cc1n[nH]c(C)c1C(=O)NCC1CN(C(=O)C(C)Oc2ccccc2F)CCO1 5054,C1(C#CC(=O)N2CCN(CCNC(=O)CCCF)CC2)(CC)CC1 5055,C1(N(C)C)CCC(C(=O)NCC2(O)CCN(C(c3cccnc3)=O)C2)CC1 5056,c1(C(=O)NC(C2CN(C(=O)CC(O)C3CCCC3)C2)C)cc(O)ccc1F 5057,c1(C(C(=O)NCC2(OC)CCN(C(COCCC=C)=O)C2)C)cc(F)cc(F)c1 5058,c1(CCOC)nc(=NC(C)C2CN(C(C3(C)CC=CCC3)=O)CCO2)s[nH]1 5059,c1(CC)ccc(C(=O)NC2CN(C(=O)C(CC)SC)CC2(C)C)cc1C#N 5060,Cc1nc2c(C(=O)N(C)CC3CCCN(C(=O)C(C)(C)CC#N)C3)cccc2o1 5061,C1(NC(c2c(C)nc(Cl)s2)=O)CC2(CCN(C(c3cc(O)n(C)n3)=O)CC2)C1 5062,C1(CNC(c2cc[nH]n2)=O)CCCCN(C(=O)CN2CCCCCCC2=O)CC1 5063,CCCCC(O)C(=O)NC(CN(C)C(c1ccc(F)cc1CC)=O)CC 5064,C1(CNC(CCC2CC(NC(c3cc(C)ns3)=O)C2)=O)CC2(CC2)C(=O)O1 5065,Cn1ncc2ncnc(N3CC4CCCN(C(c5cc(C(N)=O)no5)=O)C4C3)c12 5066,CC1CCCN(C(c2ccn(CCF)n2)=O)C1CNC(=O)C(c1ccc(Cl)s1)=O 5067,C1(CN2C(CC(=O)NC3CCc4ccccc4N3)CCCC2)CC2(CC2)C(=O)O1 5068,C=C1CC(C(=O)N(C)C(C)C2CC2)(CNC(=O)C(C)Cn2cccn2)C1 5069,C(=O)(C1CCCc2ccccc21)NCC1(CNC(c2coc(C(F)F)n2)=O)CC1 5070,CN1CC(C)(C)CC1C(=O)NC1CC12CC(NC(c1cc(O)nn1C)=O)C2 5071,Cc1cccc2c1CCOC2C(=O)NCCN(C(C1CCCSC1)=O)CC1CC1 5072,C(Cc1cn[nH]c1)(C(=O)NCC1COC(=O)N1)NC(CC=CCC)=O 5073,n1(CC(N2CCC(CNC(CCC)=O)C2)=O)ccc2cc([N+](=O)[O-])ccc12 5074,C1(O)(CN(C(=O)C(C2CCOCC2)F)C)CN(C(c2scnc2C(F)F)=O)C1 5075,c1(C(=O)NC(CNC(c2ccc(C#C)o2)=O)(C)C)cc2cc(C)cc(C)c2[nH]1 5076,CCCC(CCC)C(=O)N1CCC(NC(=O)C(c2ccc(C#N)cc2)O)C1 5077,CC1CN(C)CCCN1C(C1(C)CCCN(C(=O)CC2=CCCC2)C1)=O 5078,C1(C#N)(OC)CC(C(N2CC(F)CC2CNC(=O)C=CCCC(C)C)=O)C1 5079,c1(C(=O)NCCN2CCN(C(c3cc(C)sc3C)=O)CC2)cc(C)c(F)c(C)c1 5080,C1(Nc2nc(C)nc(N3CCCN(C(C)=O)CC3)c2)CC2(COC(C)C2)C1 5081,C(=O)(C(CC(C)(C)C)NC(=O)C(F)OC(F)(F)F)NCc1c(O)ncc(C)c1 5082,C1(CC=C)(NC(c2c(-c3ccsc3)noc2C)=O)CCN(C(C2CCCO2)=O)C1 5083,Cc1nn2cc[nH]c(=O)c2c1C(N1CCOC2(CCOCC2)C1)C(=O)Cc1ccccc1 5084,N1(C(C(CC)CN(C)C)=O)CC(C(N2CCCCC2CN(C)C)=O)C2(CCC2)C1 5085,Cc1nc(NC2CCCC(NC(=O)Cc3ccc(C)nc3)C2)c2scc(C)c2n1 5086,N1(C(CS(CC)=O)=O)CCOC2(C1)CN(C(=O)C(C)Cn1ccnc1)C2 5087,c1(C(N2CCCCC(NC(C3(COC)COC3)=O)C2)=O)cc([N+](=O)[O-])ccn1 5088,c1(N2C(CC3(c4ccccn4)CC3)CC2)nc[nH]c(=NCCc2c(C)ccs2)c1C 5089,C=CC1(C(=O)NCC2CN(C(=O)CCCC3CCC3)CCN2C)CCOCC1 5090,c1(C(N2CC(C)N(C(C3COC(=O)N3)=O)CC2)=O)nn(C)c2ccccc2c1=O 5091,C1(C)(C(N2CCC(CN(C)CC)C2)=O)CCCN(C(c2cnsn2)=O)C1 5092,Cc1ccccc1C=CC(=O)NC(C(=O)N1CC(c2ccccc2)C1)C1CCC1 5093,N1(C(C(CNC(C)=O)(C)C)=O)CCN(C(c2cc(C)cc(C)c2)=O)C2CCCC12 5094,C(C)(C)(CCCCC(=O)NCC(C1CC1)NC(=O)CC1CCCN1C(C)=O)OC 5095,c1(C(N(CCNC(C2CC(C(C)(C)C)C2)=O)CC)=O)cccc2ccnn12 5096,C1(CNC(C2(C=C)CCC2)=O)CCC(C(=O)NCCN(C)CC)CC1 5097,CCCCC(CC)CC(=O)N1CC(F)(F)CC1CCNC(=O)CCOC1CCC1 5098,CCC(C)(C)CC(=O)NC(C)CC(=O)N1CC(CC(F)(F)F)C1 5099,C(CC(=O)N(C(C)C(C)C)C)N(C(CC1(CC(=O)OC)CC1)=O)C1CC1 5100,c1(C(N2CC(C)C(NC(c3cc(Cl)cs3)=O)C2)=O)cc(N)c(F)c(F)c1F 5101,C1(Cl)(C(=O)NCC(C)NC(c2cnnn2C)=O)CC12CCC2 5102,c1(OC)ccccc1CNCc1cc(C(=O)Nc2cc(O)ccn2)ccn1 5103,Cc1ccc(Oc2ccc(SC(C3CC=CCC3)=O)cc2)cc1C 5104,c1(C(c2nnnn2CC2CCOCC2)NCC2(CCO)CC2)cc(Cl)no1 5105,C12(C(=O)NCC3C(NC(c4cc(CC)n(C)n4)=O)CCCC3)CC(C)(C1)OC2C 5106,C1(C)(CNC(CN2CCN(C)CC2)=O)CN(C(C2CC(C)(O)C2)=O)C(C)(C)C1 5107,C12CCCCC1C(=O)NCCCCO2.C12(C(=O)NOC)COCC1C2.C1CCO1.O 5108,C1(CNC(c2cccc(NC(CC)=O)c2)=O)Cc2ccccc2N(C)C1 5109,CC(C)C(CNC(c1cc(C2CCC2)on1)=O)NC(=O)Cc1ccco1 5110,O(NC(=O)C(O)CNC(=O)C(F)(F)CC)CC#C 5111,C(=O)(C1CCCn2ccnc21)N1CCC2(C(NC(C3C4(CC4)C34CC4)=O)C2)C1 5112,C12(C(N3CC4C(C)(C)C4C3)=O)CCC(CC1)N(C(=O)C1=CCCCO1)C2 5113,N1(CC2CN(C(=O)OC(C)(C)C)C2)CCN2C(=O)NCC2C1 5114,C1(CC(=O)NC(COC)C(=O)NCCCC2CCCC2)COCC(C)O1 5115,N1(CC(=C)Cl)CC2CCC(NC(c3ncn(CC)n3)=O)CC2C1 5116,c1(CN2CC(C(=O)NC(c3ccc(C(N)=O)cc3)=O)OCC2)cc2n(n1)CCC2 5117,C=CCC(C(=O)NC(CO)C(C)NC(=O)CCC(N)=O)c1ccccc1 5118,C(CC(C(=O)NCCC1CCN(C)C1)NC(=O)Cn1ccc(C)c1)OC 5119,C1(C(=O)NC2CC(C)(NC(C(c3ccc(C)o3)C)=O)C2)CN(C)CCO1 5120,N1(C(C=C(C)c2ccccc2)=O)CC(C)CN(C(=O)C=Cc2cncs2)C(C)C1 5121,c1(C(=O)NCC(CNC(C(C)OCCOC)=O)OC)cc2c(nc1O)CCC2 5122,c1(C(=O)NCC2(F)CN(C(CCC)=O)C2)ccc(F)cc1OC(C)C 5123,Cc1cc(C)c(C(N2CCC(O)C2C(=O)N(C)Cc2cccnc2)=O)cc1Br 5124,n1(CCNC(C=C(C)C)=O)ccc(C(N2CCC(C(C)(C)C)C2)=O)c1 5125,C1(CC(=O)NC2CC(=C)C2)N(C(=O)Cc2csc(C)c2)CCC1(C)C 5126,N1(C(c2nccc(Cl)c2F)C(=O)NCC)CC(C(=O)OC)OC(C)(C)C1 5127,N1(C(CNC(=O)OCC=C)=O)CC(OC)CC(NC(=O)Cc2ccon2)C1.C1(C)CC1 5128,C12(c3nnc(C)o3)CCC1CCN2C(c1c(-n2cnnc2)sc(C)c1C)=O 5129,C1(NC(CC(C=C)CC)=O)(CNC(c2nn(CC)nc2C)=O)CC2CCC1CC2 5130,N1(C(c2ccc(NS(CCC)(=O)=O)nc2)=O)CC2CN(C(=O)C(O)CCl)CC12 5131,C1(NC(=O)C=Cc2ncc[nH]2)CC2CCC1CC2NC(c1ccc(Cl)cc1F)=O 5132,c1(C(=O)NCC(CNC(CC2CCN(C(C)C)CC2)=O)O)nsc2ccccc12 5133,Cn1ccc(C(=O)NCC2CCCC2NC(=O)CCc2cncn2C)cc1=O 5134,N1(C(C(C2CC(F)(F)C2)OCC)=O)CCC(CN(C)C(C2CN(CC)C2)=O)CC1 5135,Cc1cc(C)nc(SCC(=O)NC2CC(O)(CNC(c3cnccc3Cl)=O)C2)n1 5136,c1(C(N)=O)c[nH]c(C(N2CCC(CCNC(=O)C=C3CCCC3)C2)=O)c1 5137,c1(CN(CC(N2CC(CF)C2)=O)CCOC)ccncc1OC 5138,c1(C(=O)NCCN(CCC)CCOC2(C)CC(SCC)C2)ccc(OC)c(N)c1 5139,C1(CNC(C(C)=C2CCC2)=O)(CO)CC12CCN(C(=O)CC(C)(C)O)CC2 5140,N1(C(C(C)OC)=O)CCN(C(=O)CCCCCc2cccs2)CC1CF 5141,N1(CC)CCCC1C(=O)NC1CCCC1CNC(c1ccc(C2CCOC2)s1)=O 5142,C1(C(N2CCC(OCCNC(c3c(CC)nc[nH]3)=O)C2)=O)CCNC(=O)C1 5143,C1(NC(CC2N(C)CCOC2)=O)CC2(CCN(C(c3cc(N)ccn3)=O)CC2)C1 5144,C1(CNC(C(C2CCCC2)OC)=O)CCCN1C(C1CCS1(=O)=O)=O 5145,Cc1nn(C)c(Cl)c1C(N1CCCC(O)(C(F)(F)F)C1)C(=O)NC(C)C 5146,CC1OC(C)CC1C(=O)NCC1(NC(c2sc(N(C)C)nc2Cl)=O)CC1 5147,Cc1ccc(Cl)c(F)c1C(=O)NCC1CCC(NC(=O)Cc2cccc(F)c2)C1 5148,c1(C(N(C2CCN(C(C(F)=CCC)=O)C2)C)=O)ccc(=O)n(C)n1 5149,C1(Cl)(C(=O)NC2CC(NC(C(C)OCC)=O)C2)CC1(C)C 5150,c1(CNC23CC(NC(c4ccc(C(C)=O)c(Cl)c4)=O)(C2)C3)c(C)ccc(C)c1O 5151,c1(C(=O)Nc2ccc(C)nc2Cl)ccc2c(C(N3CCC(C#N)C3)=O)n[nH]c2c1 5152,c1(OC)ccc(Br)c(CNc2csc(-c3c(O)cccc3F)n2)c1 5153,C1(C(=O)NC(CC=C)CO)CCN(C(=O)C(C)COC)C12CC2 5154,C(C)(CCCCO)NC(C(C)NC(CCN(CCC)C)=O)=O 5155,Cc1ccc(C(=O)NCCN(CC(C)O)C(=O)CC2CC=CCC2)cc1O 5156,N1(CC(=O)N(CCC(C)NC(=O)C=CC(=O)N(C)C)C)CCCC(C(N)=O)C1 5157,S(=O)(=O)(CCC(F)(F)F)Nc1c(C(=O)Nc2c(OC)cccc2)c(F)ccc1 5158,C(=O)(C1CCc2cc(F)ccc21)N1CCC(C2CC2)(NC(CC=C(C)C)=O)C1 5159,N1(C(C(C)=NOCC#N)=O)CC(C)(C)CC1CNC(C1C=CCC1)=O 5160,C(=O)(C1Cc2ccc(F)cc21)N1CC(OCCNC(=O)Cc2sc(O)nc2O)C1 5161,C1(N(C(CSCc2nc(C)sc2)=O)C)CCN(C(=O)Cc2cccnc2)CC1C 5162,CC(C)(CCF)C(=O)N1CCCC(F)(CNC(=O)CCC2CCCO2)C1 5163,C(=O)(C(=O)CC(C)C)N1CC(CC=C)(NC(=O)Cc2cn[nH]c2)C1 5164,CC(C)C(C)(CNC(=O)C(CNC(=O)C=Cc1cncn1C)N(C)C)C(C)C 5165,C1(NC(C(CCN(C)C)OCOC)=O)CC2(CCCO2)C1.C1(C)C(=O)N1 5166,C1(C(=O)N(CC(O)CF)C)(CC)CCCN(C(c2csc(CO)n2)=O)C1 5167,c1(C(=O)NC2CC(NC(c3nc(OC)c(F)cn3)=O)C2)ccc(C#N)cc1F 5168,C1(NC(C2C(C)CCC2)=O)CCOC12CCN(C(=O)C(C)(C)CCCO)CC2 5169,c1(CC(=O)NCCC2(OC)CN(C(C3CC3(C)C)=O)C2)ccc(F)cc1C 5170,c1(C(=O)NC2C(CNC(C(COC)(F)F)=O)C2)c(Br)nc2n1CCCC2 5171,C1(OCC)CCC(CNC(c2cnn(-c3ccc(Cl)cc3)c2C)C(=O)OC)CC1 5172,Cc1ccc(C(=O)NC(CO)C(C)NC(=O)CC2(CO)CC2)c(N)c1Br 5173,c1(N2CC(C)OC(CO)C2)ncc(S(=O)(=O)N(C)Cc2ccns2)cc1Cl 5174,Cc1cnn(C)c1CN(C(=O)CCC(C)N(C)C)C.C1(=O)C(C)C(=O)O1 5175,c1(C(N2CCC(NCc3c(C)cccc3O)C2)=O)ccc2cnccc2c1 5176,C(=O)(C1CCCn2c(C)nnc21)NCC(n1cc(Cn2c(C)cc(C)n2)nn1)C 5177,C1(C(=O)NCC(C(C)(C)C)NC(C=Cc2c(C)ccs2)=O)CCc2nc[nH]c2C1 5178,C(CC(C)(C)CC(=O)NCC1CCCCN(C(=O)CC2CC(=O)C2)C1)OC 5179,CC1CCC(C)N1CC(=O)NCC1(F)CCN(C(=O)OCc2ccccc2)C1 5180,N1(C(c2cccnc2Br)=O)CC2CN(C(c3c(Cl)cncc3Cl)=O)C2C1 5181,N1(C(CCSCC)=O)CCC(C2CC2)C1CNC(=O)C(F)=C(C)C 5182,Cc1c(C(=O)N(CC(O)CN(C(=O)CC2COCCN2C)C)C)nc2sccn12 5183,c1(C(=O)O)ccc2c(c1)C(NC(=O)N1CCC1)CCO2.N1(C)CCC2COCC1C2 5184,CCCC(C)(O)C(=O)NCCn1ccc(C(=O)NCCC2CC(F)(F)C2)c1 5185,c1(OC)ccc(C=CC(=O)NC(Cc2ccc([N+](=O)[O-])cc2)C(=O)O)cc1F 5186,C12(C(=O)NCC3(OC)CCOC3)COCC1CN(C(C1CCC1C#N)=O)C2 5187,c1(NC(CN2CCN(C(c3c(C)nc[nH]3)=O)CC2)=O)cc(Cl)cc(Cl)c1Br 5188,CON1CC(C(N2CCC(NC(C3CC=CCO3)=O)CC2)=O)CC1=O 5189,C=CCCCC(C(=O)NCCc1ccncn1)NC(C1C2CCCCCC12)=O 5190,N#CC12CCCCCC1CN(C(=O)C(NC1=CCCCC1)=O)C2 5191,N1(C(c2n(C=C)ncc2)=O)CCC(C)CC1CNC(=O)CC 5192,Cc1cccn2cc(C(N3CC(CNC(=O)CSC(C)C)C(F)C3)=O)cc12 5193,Cc1sncc1C(=O)NC(C)C=CC(=O)N(CCS(C)(=O)=O)C 5194,c1(CNc2c(C(=O)NCCC(C)CO)n[nH]c2)cccc(Br)c1OC(F)(F)F 5195,C(=O)(CCCCC(C)(C)C)N1CCC(F)(CNC(c2c(C)con2)=O)CC1 5196,CC1(NC(=O)CC2CC=CCC2)CCN(C(C2CCC3CCC2O3)=O)CC1 5197,C(CC1CC1)(C(=O)NCC(CO)C1CCC1)NC(=O)Cc1cc[nH]n1 5198,N1(C(c2ccc(CCC)cc2)=O)CC(C)CCC1CNC(C1CN(C(C)C)C1)=O 5199,c1(C(=O)NCC2(C)CCC(NC(c3cnc(COC)s3)=O)C2)cc(C)ccc1O 5200,c1(C(C(=O)N(CCCCCNC(C(CCC)F)=O)C)O)ccc(F)cc1C 5201,Cc1cnccc1C(N1CCCC1C(C)NC(c1cnn(CC(F)F)c1C)=O)=O 5202,C1(C(=O)OC)C(F)(F)C12CC(C(N1CCN(C(c3ccsn3)=O)C(C)C1)=O)C2 5203,C(CC(C)C)(C(=O)NCCCCCN(C)C(C1CC12CC(C)(C)C2)=O)NC(C)=O 5204,C(=O)(C1=CC2CCCCCCC12)N1CCCC(C)(CNC(c2nncs2)=O)C1 5205,C1(C(N(CC(C)(C)CNC(C2CCCCC2F)=O)C)=O)CCC(=C(F)F)CC1 5206,c1(C(c2nnnn2C(C)CC)NCCn2c(CC)ncc2)cc(C)c(C)cc1C 5207,CC1OC2(C(=O)NCCCN(C(=O)CC#N)Cc3ccccc3)CC1C2 5208,CC(C)(C)CC(=O)NCC(=O)NCCC(O)CNC(=O)CCNC(N)=O 5209,CCCC(CC)C(c1nnnn1C1CCC1)NCc1nnnn1CC 5210,CC1c2ccccc2OC1C(N1CC(NC(=O)COCCF)C(C)C1)=O 5211,N(C(=NCc1cccc(F)c1)NCC12CC(C1)C(C)O2)C(C)C1CC1 5212,CC(C)C#CC(=O)NCC1CCCN(C(=O)CCCc2ccccn2)C1 5213,N1(C(C(C)OC2CCOC2)=O)CCC2CN(C(c3cnn(C)c(=O)c3)=O)CCC12 5214,c1(CO)cccc(OC)c1O.n1(CC)cc(CC(=O)N(CCNC(C)=O)C2CC2)cn1 5215,CN1CCC(C(=O)NC2CCN(C(c3oc(C(F)(F)F)nc3C(F)F)=O)C2)CC1 5216,C1(C(=O)NCCS(CC)=O)CCC2(CC2)N1C(c1cc(C#N)[nH]c1C)=O 5217,c1(C(N2CCC(C3C(C(N)=O)CCN3)CC2)=O)ccnc2c(O)cccc12 5218,C1(CNC(=O)Nc2cnn(C(C)(C)C)c2Cl)(CSC)CC12CCOCC2 5219,C1(CNC(CC(C)(C)SC)=O)CCC(C)N(C(c2ccc(F)s2)=O)C1 5220,C(=O)(CC(C)CC(C)(C)C)NCC(CC)(CC)NC(c1cc(C)c(O)c(C)c1)=O 5221,CCC(C)(C)C(O)C(=O)NC1CN(C(c2cc(Cl)cc(C)c2O)=O)CC1OC 5222,C1(C(=O)NC(c2ccoc2)C)CC=CCN1C(c1cccc(CO)c1)=O 5223,c1(C(N2CCC(C)(CNC(Cc3c(C)nsc3)=O)C2)=O)ncc(C2CC2)cc1F 5224,N1(C(C(CC)OCC)=O)CC2(CCN(C(=O)C(CC)C(C)(F)F)CC2)C1 5225,CC1SCCN(C(C23CC(CN2C(=O)C(C)(C)CN(C)C)C3)=O)C1C 5226,c1(OCCOC(c2cn(C)nc2C2CC2)=O)ccccc1[N+](=O)[O-] 5227,N1(C(CC=C=C)=O)CCC2CN(C(c3ccn4nncc4c3)=O)CCC2C1 5228,N1(C(C=CC(CC)C)=O)CC2CCOC2(CNC(c2cc(CC)cc(C)c2)=O)C1 5229,N1(C(C(C(=C)C)(C)O)=O)CCC2(CC1)CC(CNC(=O)CCC(C)C)C2 5230,c1(C(=O)Nc2scc(C(=O)NCCNC(C)=O)n2)c(O)ccc(F)c1F 5231,C(=O)(C(CC(C)C)N(C)C)NCCN(C(=O)Cc1c(C)cnn1C)CCC 5232,Nc1ccccc1OCNC(CO)=O.C1(O)(C)CCNC1 5233,S(=O)(=O)(c1cc([N+](=O)[O-])c(N)cc1Br)NC(C1CN(C)S(=O)(=O)CC1)=O 5234,C1(NC(CN(CCC)C)=O)CN(C(=O)C(c2ccn(C)c2)C)C(C)(C)C1 5235,C1(CNC(C=C(CC)C)=O)COCCN(C(=O)C(c2cccc(C#N)c2)(C)C)C1 5236,Cc1cc(C(=O)NCCC(O)CNC(C2CC2F)=O)nn1CC(F)(F)F 5237,N1(C(=O)CC2CCCCN2C(=O)C(O)C2CCCC2)CC2(CCOCC2)C1 5238,CCCCC(CC(=O)NCC1CCCCC1O)NC(=O)CCC(C)OCC 5239,C(C(CC)(CC)NC(=O)Cc1ncc(C)s1)NC(C(CC)F)=O 5240,C1(CC=C)(NC(C2C=CCC2)=O)CC2CCC(C1)N2C(c1sccc1Cl)=O 5241,C(=O)(CC(C)CC(=O)N(CC(O)CN(C)C(C1(Br)CC1)=O)C)OC 5242,C1(OC)CC(CNC(=O)CCC(=O)N(C)C)CN(C(=O)Cn2ccnn2)C1 5243,C1(CC=C)(NC(=O)CC(C)C=C)CC2CCC(C1)N2C(=O)Cc1cc[nH]n1 5244,C(=O)(CS(=O)(=O)CC(C)C)NC1CC(CNC(CCCC(C)=O)=O)C1 5245,CC1CCN(C(=O)Cn2ccnn2)C(CNC(C2CCOC2(C)C)=O)C1 5246,c1(OCC)nc(Cl)cc(=NC(=O)c2cc(-c3ccc(CC(=O)OC)s3)ccn2)[nH]1 5247,N1(C(c2ccc(CSC)cc2)=O)CCC2(CNC(C3CC3(C)C)=O)CCCC12 5248,C1(CNC(Cc2ccc(OC)cn2)=O)CC12CCN(C(=O)C(C)(O)C(C)C)CC2 5249,C(CCCC(=O)N(C)CC1CCC(=O)N1)N(C(=O)Cn1cnc(C#N)n1)C 5250,CCC(C)(C)C(C)(O)c1nc(C(c2ccccc2)C)no1 5251,c1(NC(N2CCN(CC(=O)Nc3ncc(C)s3)CC2)=O)ccc(C(C)C)c(F)c1 5252,C(=O)(C(C)CC(N)=O)N1CC(O)(C(C)NC(C(C)Oc2cccc(N)c2)=O)C1 5253,C1(NC(CCN(CCC)C)=O)C(C)(C)CN(C(=O)C(C)CC(C)CC)CC1(C)C 5254,N(C1c2ccccc2CC1C)C(C#CCC)c1nnnn1CCCOC 5255,N1(C(CC(C=C)C)=O)CCC(C(=O)NC(c2nc(=O)o[nH]2)C)C1(C)C 5256,N1(C(=O)Cc2ccccc2F)CC2CC(C1)N2C(c1cc(F)ccc1I)=O 5257,c1(C(=O)NCC2CC(F)(CNC(C3CCC(C)O3)=O)C2)cnc(O)c2ccsc12 5258,c1(C(N(C2CCCN(C(C3CCS3(=O)=O)=O)C2)CC)=O)ccnc2c1nnn2C 5259,c1(C(=O)NCC(C)(CO)NC(CC2CN(C)CC2O)=O)ccc2c(n1)OCCO2 5260,C1(C2CC2)(CNC(CCC(C)(F)F)=O)CCN(C(c2cncc3ccsc23)=O)C1 5261,c1(CC)cnn(CC(=O)NCCCN2CCC(NC(C3CCC4CC34)=O)C2)c1 5262,C(=O)(C(C(C)CC)NC(=O)C(C#N)C(C)C)NCC=CC 5263,Cc1nn(C)c(Cl)c1CC(=O)NCC1(C)CCCN1C(c1cnc(O)c(Cl)c1)=O 5264,CCC1=C(C(=O)NCC2CC(NC(c3cc4cscc4s3)=O)C2)CCCO1 5265,N1(C(CCC=C(C)C)=O)CC(CN(C(=O)C(O)C(C)(C)C)C)C2(CC2)C1 5266,CCC(CCOC)C(=O)N1CC(OC)CC1CNC(C1(CF)CCOCC1)=O 5267,c1(C(C(=O)N(C)CCNC(=O)CCOC2COC2)(F)F)ccc(Br)nc1 5268,CC1CC(NC(=O)C(CCOCCO)NC(c2ccncc2)=O)CC(C)C1 5269,CC1CC(C)CN(C(=O)CN2CCC(C(=O)N(C)CC=Cc3ccco3)CC2)C1 5270,N1(C(COCCC(C)C)=O)CC2CC(C1)C2NC(c1ncoc1-c1ccon1)=O 5271,c1(C(=O)NCC(CO)NC(c2ccc(C)n2C)=O)cc2n(c1)CCOC2 5272,c1(OC)ccnc(C(=O)NC2CC(CNC(=O)CC3CC(C)=NO3)C2)c1 5273,C1(C(N2C(NC)CCC2c2ccc(C)cc2)=O)CCN(CCN)CC1 5274,c1(Cn2cc(CNC(c3cccc(Cl)c3)CCO)nn2)c(F)ccc(Br)c1Cl 5275,C1(CCC)CCCN1C(=O)C(O)CNC(=O)CC(C1CC1)C1CC1 5276,C1(CNC(C2C(C=C(C)C)C2(C)C)=O)(NC(c2nnn(C)c2N)=O)CCCCC1 5277,c1(CC)ncncc1C(=O)NC(CC1CCCC1)C(=O)NCCN1CCCC1C 5278,c1(SCC)cccc(C(N2CCCC2C2CCCN(C(C3CCCC3)=O)C2)=O)c1 5279,c1(CC2(C(N(C)OCC(C)Sc3ccccc3)=O)CCOC2)ccccc1 5280,c1(OCCCC)cc(C(N2CCCC2N(CC)CC2CC(COCC)C2)=O)ccn1 5281,O=C(C1=CCCC1)NCC1CCCN1C(=O)CCc1cnc(C2CCC2)o1 5282,CC1CN(C)CC(C(=O)N(C(CNC(=O)COc2cccc(O)c2)C2CC2)C)O1 5283,c1(C(=O)NCC2C(NC(CC3(N(C)C)CCC3)=O)CC2O)cccc2[nH]ncc12 5284,c1(C(N2CC3C(NC(C(CCC)(C)C)=O)(C3)C2)=O)c(Br)ccc(F)c1OC 5285,Cc1cccc(C2(CNC(C3CCCCC3N3CCOCC3)=O)CC2)c1I 5286,N(C(=NCc1cc(CN2CCCC2)on1)N1CCC(COC)C1)C(C=C)C 5287,C1(C)(C(N(C)CC2N(C(c3ncc(C)cc3C)=O)CCC2)=O)CCC(F)(F)CC1 5288,N1(C(C(C)CN(C)C)=O)CC(CCNC(=O)CCC2CCOCC2)C(C)C1 5289,CC1CN(S(=O)(=O)N(C)CC2CC2)CCN1C(=O)CC(F)(F)F 5290,N1(C(c2ccc(OC)nc2)=O)CC2(C1)CN(C(C1CCCC(=O)N1)=O)C2.C(C)(C)(C)O 5291,c1(SCNC(=O)C(C2CC3CCC2C3)C)ccc(Cl)cc1.c1(CC)ccncc1 5292,c1(CC)cccc(C)c1C(N1CCN(C)C(CNC(C2CC(OC)C2)=O)C1)=O 5293,c1(OC)cc(CC(=O)NCC(C)(C)CNC(c2c[nH]c(=N)cc2C)=O)ccc1F 5294,Cc1cnc(C#N)nc1N1CCC(NC(=O)C2=NOC(C(C)(C)C)C2)C(O)C1 5295,CC(C)(C)C(C#N)C(=O)N1CC2CCC1CC2NC(=O)Cc1ccoc1 5296,c1(C(=O)NCC=CCNC(c2cnc(CC(C)C)s2)=O)ccc(Br)nc1O 5297,C(=O)(CC(F)(F)Br)N(C1CCN(C(C2CCN(C)C2C)=O)C1)CC 5298,C(=O)(C1=CCC(C)(C)CC1)N1C(CNC(c2c(C)oc(C)c2Br)=O)C=CC1 5299,C1(C(=O)NC2CCN(C(=O)C(O)C3CCC3)CC2)CCCc2ccccc2C1 5300,Cc1cnc(C(=O)NCCCCC2CCCC2)c(S(=O)(=O)N2CCC(CF)C2)c1 5301,CC1(C)COCCC1NC(N1CC2(CC2)CC1CO)=O 5302,C(C#Cc1cccnc1)NC(C(CCOCC)NC(C1CN(C)CCN1C)=O)=O 5303,N1(C(C2CC(C)(F)C2)=O)CCCC12CCCN(C(c1cccc3c1CCN3)=O)C2 5304,N1(C(CNS(CC)(=O)=O)=O)CCN(C(c2ccnn2CC#N)=O)C(CCO)C1 5305,C1(C(N(C)Cc2ccoc2)=O)COCCN(C(=O)CNC(C2CC(F)C2)=O)C1 5306,c1(C(N2CCC(C)(CNC(=O)Cc3ccoc3)CC2)=O)ccc2nc[nH]c2n1 5307,c1(C(N(C2CCN(C(=O)CC3(OC)CC3)C2)CCC)=O)ccnc(C(C)(F)F)c1 5308,c1(NC(COCCOC)=O)cccc(CNC(=O)C(N2C(=O)CCC2=O)(C)C)c1 5309,C1(CNC(c2ccnc(SCC3CS(=O)C3)c2)=O)CC12CCCOC2 5310,CCC(CC(C)C)C(=O)NCCC(C)N(C)C(c1ccsc1C#N)=O 5311,Cc1nc2n(c1CC(N1CC(C3CCCN3C(C3CC3CF)=O)C1)=O)CCCC2 5312,n1(C(C)C)cc(C(=O)NCC(C)NC(C2CCN(c3nccn3C)C2)=O)cn1 5313,C1(NC(=O)C(N2CCC(CO)C2)=O)CCC2CN(CC(F)F)CC2C1 5314,c1(CN2CC3N(c4ncc(CCC)cn4)C(C3)C2)cc(OC)c(O)c(I)c1 5315,N1(C(CN(C2CCCC2)C)=O)CCC1CNC(C1CC(n2ccnc2)C1)=O 5316,c1(C(N(C2CCNCC2)CC(C)C)=O)noc2c1CC(C)(C)CC2 5317,CCC(C)C(CN(C)C)NC(=O)CCN(C(c1cccc(Cl)c1)=O)C(C)C 5318,C(=O)(C(C)C(O)CC(C)C)N1CC(F)(C(=O)NC(CCC=C)(C)C)C1 5319,CCCCCCC(F)C(=O)NC(CNC(c1cnccc1Cl)=O)C(C)C 5320,c1(OC)ccc(Cl)cc1CC(N1CCC(C(=O)Nc2cccnc2Cl)C(O)C1)=O 5321,C=CCC(CNC(C1CC(CC)(CC)C1)=O)C(=O)NCC1CC12CCC2 5322,c1(C(C)=O)csc(C(=O)NCC(C)(C)CN(C(=O)C(F)(F)c2ccncc2)C)c1 5323,N1(C(CCCC#C)=O)CC(C)N(C(C2CC2C(=O)OCC)=O)CC1C 5324,N1(C(C)=O)CCC(c2nc(CC(CN)C(C)C)n(-c3ccnc(F)c3)n2)CC1 5325,C#CCC(CC(=O)OC)NC(C1CCCCC1NC(=O)CNC(=O)C=C(C)C)=O 5326,C1(C(N2CC(n3ccnc3)C2)=O)(CC)CCN(C(c2n[nH]c(C)c2Cl)=O)C1 5327,Cc1cnc(C(N2CCC(NC(C3CCCOC3)=O)C(O)C2)=O)cc1C#N 5328,C1(C(N(CCC#C)CCO)=O)CN(C(c2ccc(F)c(C)c2)=O)C(C)(C)C1 5329,Cc1cc(C(C)NC(N2CCC(C(=O)O)C2)=O)cc(C)c1F 5330,c1(C(N2CC3CC(CNC(c4n(C)c(S)nn4)=O)C3C2)=O)cc2cccnc2[nH]1 5331,c1(C(N(C(C)CNC(c2ccoc2C(C)C)=O)CC)=O)csc2nccn12 5332,N12CCCN(CC1)C(=O)C=CC=C1C(=NCCCC(CCCO)CCNC1=O)N2 5333,c1(NCC2(C(=O)NCC3C(C(N)=O)C3)CC2)cnc2ccccn12 5334,Cc1nn(C(C)C)cc1C(=O)NCC(C)(C1CC1)NC(C1CCC(=O)N1)=O 5335,c1(N2CC(C(C)NC(C(C)C3CC3)=O)OCC2)c(Br)cncc1[N+](=O)[O-] 5336,c1(C(=O)NCC(C)NC(C2(c3ccccc3)CCOC2)=O)ncccc1Br 5337,c1(C(N(C)CC2N(C(c3c(CC)ncnc3)=O)CCC2)=O)cn2ccccc2n1 5338,CC(CNC(=O)C=C=C(F)F)C(F)C(=O)NCc1ccncc1 5339,c1(OC)cc(C)ccc1OC(=O)Cn1ccc(C)n1 5340,C1(C(N2C(C(N3CCC(OC(C)C)CC3)=O)CC(F)C2)=O)CC2(CCO1)CC2 5341,C(=O)(C(O)CC(=O)OC(C)(C)C)N(C1CCCN(C(=O)Nc2cc(Cl)no2)C1)C 5342,C1(F)(CNC(C(C)(C)F)=O)CCN(C(C2CC(c3cccnc3)C2)=O)C1 5343,c1(N2CC3(CCN(C(c4c(CC)nco4)=O)C3)C2)nccc2c1C(=O)OC2(C)C 5344,c1(C(N(CC(CNC(c2c(C)ccc(C)n2)=O)O)C)=O)cc2cc(F)ccc2o1 5345,C1(C(C(=O)N(C)CC2CCCC2)NC(=O)CCc2ccco2)CCCOC1 5346,C(=O)(C1c2ccccc2C2(CC2)CN1C(=O)C(C1CCCCC1)F)OCC 5347,N1(C(c2c(C(C)=O)cco2)=O)CCC2(CCN(C(c3c(Cl)nn(C)c3C)=O)C2)C1 5348,CCCCCC(CC)C(=O)NC1(C)CCN(c2cc(O)nc(COC)n2)C1 5349,c1(C(=O)NCC(C)(CO)NC(C2C(c3cn(C)nc3)C2)=O)ccnc2ncnn12 5350,CC1CC(C(N2CCC(O)C2C(C)(C)C)=O)N(C(c2cc(CO)ccn2)=O)C1 5351,C1(C(N2CCCC(CNC(c3ccc(C)cn3)=O)CC2)=O)Cc2cccnc2C1 5352,C1(C(=O)NC(CC(=O)OCC)C)(C(C)C)CCN(C(=O)C=Cc2cocn2)C1 5353,C(C1=CCCCC1)(c1nnnn1Cc1ccc(F)cc1)NC(C(=O)NCC)CC 5354,C1(F)(CNC(c2cnc[nH]2)=O)CC2CCC(C1)N2C(c1noc2ncccc12)=O 5355,C(=O)(C(F)C(C)C)NC(C(=O)N(CC(C)C)CCN(CC)CC)(C)C1CCC1 5356,CC(C(C(=O)NCCSC1CC1)N1CCC(Oc2cccc(F)c2)C1)C1CC1 5357,C1(N(C(C(c2ccc(OC)cc2)O)=O)Cc2ccsc2)CCNCC12CC2 5358,c1(OC)cc(C(=O)N(C2CC(CC(=O)NOCC(C)C)C2)C)ccn1 5359,C1(NC(C2CCCC3CCCN23)=O)CN(c2nnc(C(F)F)o2)CC2(CC2)C1 5360,C1(CNC(c2c(C(C)C)ncnc2)=O)CCCCN(C(C2COC(=O)N2C)=O)C1 5361,N1(C(C2C(OCC)C2)=O)CCN(C(=O)C(C)(C)CNC(C)=O)CC(C)(F)C1 5362,c1(NCCCCCC)ccccc1NC(=O)NCC(C)(C)NC(=O)OC(C)(C)C 5363,N1(C(C2CC(OCC)C2)=O)CC2CC2(CNC(=O)CC2CCC(=O)N2)C1 5364,CC1CC(NCc2cccc(F)c2)CN(C(c2ccc([N+](=O)[O-])o2)=O)C1 5365,N1(C(CCC2(SC)CCC2)=O)CC=CCC1C(=O)NOCC(F)F 5366,n1(CC(OC)OC)cc(C(=O)NC2CCC(CNC(c3ccc(SC)o3)=O)C2)nn1 5367,CC(F)(F)CC(=O)NC1CC1NC(=O)CNc1ncccc1C(F)(F)F 5368,N1(C(COCCOCC)=O)CC(O)CCC1C(=O)NCc1[nH]cnc1C 5369,Cc1cnc2n1CCC(C(C1N(C3CCNC3C(C)(C)C)C1)NC1CCC(C(F)(F)F)CC1)C2.C(S(C)(=O)=O)S 5370,c1(CC(=O)NC2C(NC(CCN3CCN(C)CC3)=O)C2)ccc(C(N)=O)cc1Cl 5371,c1(CC)cc(C(=O)NCC2CCN2C(c2c(NC(C)=O)c[nH]c2C)=O)cc(O)n1 5372,CCCCC(C(=O)NCCCN(C(c1cnn(C)c1CC)=O)CC)N(C)C 5373,c1(CC(=O)NC2C(NC(CC3(CC(=O)OC)CC3)=O)C2)cncnc1 5374,N1(C(c2cc3cnn(C)c(=O)n3n2)=O)CCN(C(=O)C(Cl)=CCl)C2CCCCC12 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5463,c1(C(=O)NC(CC)CNC(c2cc(C(C)(C)C)n[nH]2)=O)cc2c(cn1)CCCC2 5464,CCCS(=O)(=O)CC(=O)N1CCN(CCCCCNC(=O)C(CC)C(C)O)CC1 5465,C(=O)(C(F)(F)C1(N(C)C)CCC1)N(CC(C)NC(=O)CCc1n[nH]c(=N)s1)C 5466,C1(C(N2C(CN(C(c3c(COC)noc3)=O)C)CC(F)C2)=O)CCC(F)(F)CO1 5467,C1(CNC(c2ccc(CO)s2)=O)CCCCCN1C(=O)C(F)CC1CCC1 5468,S(=O)(=O)(c1ccc(C#N)cc1)N1C2CN(Cc3c(Br)ccc(C#N)c3)CC21 5469,c1(SCC(=O)NCC=CCNC(C2=C(C#N)CCC2)=O)ccc2c(c1)OCCCO2 5470,N1(C(CN2CC(CC)C2)=O)CCCC(O)(CNC(C2CC3C=CC2O3)=O)C1 5471,CC1CCCc2c(NC(N(C3C(c4c[nH]nc4)NC(=O)CC3)C)=S)cnn21.C1CC1 5472,N1(C(Cc2cccc(CC)c2)=O)C2CCC1C(C)C(NC(c1nc(C)no1)=O)C2 5473,C(=O)(CCCS(N)(=O)=O)NCC1(CNC(CCC2N(C)CCC2)=O)CC12CCC2 5474,C(=O)(C(O)CNC(=O)CC1CC1)N(CCC)CC1CC1 5475,Cc1ccccc1-n1nccc1CNC(c1ccc(OC(F)F)cc1)C(F)(F)F 5476,C1(NC(CCCNC)=O)CC2CCC(C1)N2C(c1cccc(Cl)c1F)=O 5477,c1(C(=O)NCC2N(C(=O)CNC=O)CCC(C)C2)cc([N+](=O)[O-])cnc1N 5478,c1(C(=O)NC2CCCC(NC(=O)CCc3cocn3)C2)cc2cccnc2[nH]1 5479,Cc1nn(C)c2sc(C(=O)NCC3CC3NC(C3CNC(=O)CC3(C)C)=O)cc12 5480,c1(C(=O)NCC(CN(C(c2c(C)con2)=O)C)O)cc2c(C3CC3)cccc2[nH]1 5481,C(N=C(NCC1CCCS1)N1CCC(O)CC(C)(C)C1)c1n(C)ncc1 5482,Cc1nnc2n1CCCC2C(=O)N1CCCC(CN=c2[nH]cncc2Br)C1 5483,N1(C(C(CC)(C)OC)=O)CC(NC(=O)C(F)(F)CCn2cccn2)CC(C)C1 5484,C(=O)(CC(C)(C)C(=O)OC)NC1(CNC(c2c(Cl)cnc(CC)n2)=O)CCOC1 5485,c1(C(C)C)cc(=NCCCCNC(=O)Cc2ccc3c(c2)CCO3)[nH]cn1 5486,C(=O)(CCCCCNC(=O)C(c1nc(C)sc1C)N(CC(=O)NC1CC1)C)OC 5487,CN1CCN(CC(N2CC3CC2C3NC(c2ccc(Cl)o2)=O)=O)CC1 5488,Cc1cc(F)cnc1C(=O)NC1COCCN(C(=O)CCC2(C)CC2(F)F)C1 5489,N1(C(C2C(C)(C)C2C#N)=O)CC23CCCC2(C1)CN(C(=O)CCOC1CC1)C3 5490,N1(C(C(=O)NCCOC)=O)CCCN(C(c2ccnc(OC)c2)=O)CC1CO 5491,C12(CNC(C(C)N(C)C(C3CC(CC4CC4)C3)=O)=O)CCCCC1C2 5492,C(C(C(=O)NCCNC(=O)CO)NC(c1ccco1)C(=O)OC)SC 5493,N1(C(C2CCCCNC(=O)CC2)C)CCC(C2CCC2)CC1 5494,N1(C(COCC)=O)CCC(CCNC(=O)CNC(=O)OCC)C(F)(F)C1 5495,C(=O)(C(F)(F)C1CCOCC1)NCCCN(C(C1C(CCC)C1)=O)C 5496,c1(C(N2CCCC(NC(=O)CC3CCC3)C2)=O)ccc(Br)cc1C(F)(F)F 5497,C(=O)(C(Cl)=CCl)NCCN(C(C)C)C(c1cn(C2CCCCC2)nn1)=O 5498,C1(CNC(CC(=C)C)=O)(CO)CC12CCN(C(=O)COCP(C)(C)=O)CC2 5499,c1(C2(C(=O)NCC(C3CC3)NC(CC(C)(C)C)=O)CCC2)ccc(F)cc1Br 5500,c1(C(N2C(CN(C(=O)C(C)(O)c3ccccn3)C)CCC2)=O)ncccc1Cl 5501,N1(C(CN2CCC(N(C(C(C)CC3CC3)=O)C)CC2)=O)CCc2ccccc21 5502,N(C(=NCc1cc(C2CC2)on1)NC(C)COc1cccc(F)c1)C(C=C)C 5503,c1(CC)c(C(N2CCCCC2CCc2ccccn2)=O)ccn1C 5504,c1(CN(c2ncccc2S(=O)(=O)N(C2CCOC2)C)C)cc2ccccc2n1C 5505,c1(C(N(C2CCN(C(=O)CC3COCC3O)C2)CCC)=O)ccoc1Br 5506,C1(NC(c2ccc(C(C)=O)[nH]2)=O)CCCCC1CCO.C1(C)(C)C(=O)N1 5507,c1(C(=O)NC2CC3CN(C(c4c(C)nn(C)c4)=O)CC32)cncc2nc[nH]c12 5508,N1(C(CC(=O)NCCC(C)C)=O)CC(C(F)(F)F)OC(C)C1 5509,N1(C(C(c2cc(F)cc(F)c2)C)=O)CC2CCC1CN2C(C12CC3CC1C2C3O)=O 5510,C(=O)(C1=NOC(C)(C)C1)NCC(CNC(c1cc(CC)[nH]n1)=O)OC 5511,CCC(C)C(O)CC(=O)N(CCC(=O)NCCC1CC(=O)N(C)C1=O)C1CC1 5512,N1(C(C=C(C)C(F)F)=O)CC2CCC1C(NC(=O)CC1CC3CCC(C1)N3C)C2 5513,C=CC(C)(C)CCCNC(c1cccc(Br)c1Cl)C 5514,CC1CCN(C(=O)COCC(c2ccccc2)=O)CCN1C(c1cc[nH]n1)=O 5515,C1(CNC(C=CCC)=O)CN(C(C2(C3(O)CCOCC3)CC2)=O)CCC12CCC2 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5534,N1(CC)CCN(CC(N2CCC3C(NC(=O)C(C)C4CCC4)C23)=O)CC1 5535,C1(C(N(c2nc(N3CCC(COC)CC3)nc(C)c2)C)=O)Cc2ccncc2C1 5536,c1(C(=O)NCCOCCOCCNC(C2C(=C)CC2)=O)ccoc1C(F)(F)F 5537,C=C1CC(C(N2CC(C)(OCC(=O)N(C(COC)CO)C)C2)=O)(C(F)F)C1 5538,C1(C(=O)NCC2(CC#C)CC2)C2CC1N(C(c1cc(C(C)C)[nH]n1)=O)C2 5539,C1(NC(c2c(OC)cc(O)nc2)=O)C(C)(C)C(NC(=O)C=CC(=O)N(C)C)C1(C)C 5540,c1(C(=O)NCC(CCNC(CCSCC)=O)O)ccc2cnc(C)n2c1 5541,CCC(C)(O)C(=O)N1CC(CNC(=O)C(O)Cc2cnc[nH]2)C(O)C1 5542,c1(OCC)ccc(Cl)nc1C(=O)NCC1CCCC1NC(=O)C(C)c1ccco1 5543,c1(C(=O)NC(C)C(N2CC(C)(C(=O)NCC=CC(C)(C)C)C2)=O)cncc(O)c1 5544,C(=O)(C1CCc2c(F)cccc21)NC(c1ccc(OC)cc1Br)C 5545,c1(C(=O)NC(CC(C)NC(c2ncoc2C2CC2)=O)C)ccnc(NC(N)=O)c1 5546,c1(C(=O)NC2C(CNC(CN3CC(C)(C)C3)=O)CC2)oc2ccccc2c1Cl 5547,C1(CNC(CC(CCC)O)=O)CCN(C(c2csc(Cl)c2OC)=O)CC1(F)F 5548,c1(C(N(C(CCNC(Cc2ccn(C(C)C)n2)=O)C)C)=O)cnc2[nH]ncc2c1 5549,N1(C(C(CC)N(C)C)=O)CC2CCCC(CNC(=O)CCCN(C)C(C)C)(C2)C1 5550,C(CC(CC)C(=O)NC1COCC1NC(=O)CCc1ccc(F)cc1)=CC 5551,C1(NC(=O)Cc2ccccc2O)CC2CC1N(C(=O)COc1ccc(F)cc1)C2 5552,N1(C(Cn2ncc(C#C)c2)=O)CCC2CN(C(=O)CCC3CC(F)(F)C3)CCC12 5553,c1(C(=O)NCC2N(C(CCC#C)=O)CCC(C)C2)cc(OC)c2c(c1)CC(C)O2 5554,c1(COC)ccoc1C(=O)NC1CCCC1CNC(=O)CC(=O)N(C)C 5555,Cc1ccc(C(=O)NCC2C3CN(C(C4CC(n5cccn5)C4)=O)CC23)cc1 5556,N1(C(c2c(C)cns2)=O)CCN(C(=O)C#CC(C)(C)C)CC(O)C1 5557,N1(Cc2cc(OC(C)C)c(I)cc2)Cc2[nH][nH]c(=NC(=O)c3cnn(C)c3)c2C1 5558,C1(NC(C2C(OC)CCC2)=O)(CO)CCN(C(c2ccc(C)[nH]2)=O)CC1 5559,CC1CCC(C)CN1C(=O)C(=O)NC(c1ccccc1F)c1nnc(CO)s1 5560,C(=O)(CC(CN(C)C)C(F)(F)F)N1CC(O)(CNC(C(C)n2ccnc2)=O)C1 5561,C(C(CC(C)C)C(=O)NC(CC(F)F)C(=O)N1C2COCC1C2)OC 5562,N1(C(c2cccnc2O)=O)CC2CC(C1)N2C(=O)CC(O)C1CCCC1 5563,c1(C(=O)NC2CC(C)(C)N(C(c3coc(O)n3)=O)C2)cccc2cnsc12 5564,C(CC(F)F)(C(=O)N1CC(O)(C(F)(F)F)C1)NC(C1C(=C)C1)=O 5565,c1(C(=O)OC(c2ccc(C(=O)O)cc2Br)C(F)(F)F)cc2c(Br)cncc2s1 5566,Cc1cccc(C(N2CC=CC2CNC(=O)CC2CC(c3ccccc3)C2)=O)n1 5567,n1(CCOC)ncc(C(=O)NCC2CN(C(c3sc(C)nc3C)=O)C3CC23)c1C 5568,c1(C(C(N2CC(C)C(NC(=O)COC3CC3)CC2)=O)(C)C)c[nH]c2ccccc12 5569,N1(C(C2(C(C)NC(C34CCC(C3)C4(C)C)=O)CC2)=O)CCC12CCN(C)C2 5570,N1(C(C2C(C=C)C2)=O)CCCC2CN(C(=O)CCS(=O)(=O)NC)CCC12 5571,CC(C(=O)NC1CCC(CNC(c2cnc(N)c(N)c2)=O)C1)C(C)(F)F 5572,N1(C(c2ccc(OC)s2)=O)CCCCC(NC(=O)C(C)Cc2ccco2)C1 5573,N1(C(CC(C)n2ccnc2)=O)CCC2(COC(CNC(c3cnn(C)n3)=O)C2)C1 5574,c1(OC)nc(NC2CS(=O)(=O)CC2NC(c2c[nH]nc2C(C)C)=O)nc(C)c1F 5575,N1(C(c2cc(COC)[nH]n2)=O)CC(C)CN(C(=O)Cc2c(C)noc2C)C(C)C1 5576,Cc1cc(NC(=O)Cc2cn[nH]c2)ccc1NC(=O)CN1CCC(F)(F)C1 5577,C1(CNC(CCCC(=C)C)=O)CN(C(=O)CSc2nncs2)CCC12CCOC2 5578,N1(C(c2c(OC)cncn2)=O)CC(O)CCC1C(=O)NCC1(CCO)CC1 5579,C(=O)(CCN(C)C(=O)OCC)NCCC1(NC(COCC)=O)CC1 5580,C12(CNC(C(CC)=CC)=O)CC1CN(C(c1csc(CC3CC3)n1)=O)C2 5581,c12ccc(C(=O)C3CC3)c(c1)NC(=O)N2.C1(CC(=O)OC)OCCCO1 5582,c1(C(N2CC3(CC2CO)OCCO3)=O)nn2c(c1Br)OCCC2 5583,C1(OC)(OC)CCC(C2(CNC(=O)CC(C)c3ccccc3)CCO2)C1 5584,C(N=c1[nH]c(N2CC(=O)NC(=O)C2)nc2c1CCC2)C1C(C)(C)OCC1 5585,C(=O)(C1CCCc2nccn21)NC(CCCC)CNC(c1cc(C)oc1C)=O 5586,c1(C(c2nnnn2CCOC)NC2(C=C)CCC2)c(C)c(Br)c(C)n1C 5587,C(=O)(C(C)CNC(=O)C1CC1)N(C(CSC)C)C 5588,CC1CC2(CCO1)CC2C(=O)NCC1CCN(C(c2c[nH]ccc2=O)=O)CC1C 5589,N12CCC(F)(C1)C2=O.C1(NC(C(N2CC(C)C2)C)=O)C2CC3C(C2)C13 5590,O=C1CCCC(c2ccccc2)(CNc2ncccc2I)N1 5591,N1(C(=O)C=CC2CC2)CC2(CCN(C(C3CCC4CCC(=O)N34)=O)CC2)C1 5592,C(C(O)C(=O)NC(c1cnn(C)c1)C(N1CC(C)(CSC)C1)=O)SC 5593,C12(CNC(C3CCC34CCCO4)=O)CCCC1N(C(c1cnsn1)=O)CC2 5594,c1(C(=O)NC2CC(N(C(=O)CN3CCCNS3(=O)=O)C)C2)ccc(Cl)c(N)c1Cl 5595,C1(C(=O)NCC2(F)CN(C(CC=CC(C)(C)C)=O)C2)CC2C=CC1C2 5596,C1(NC(c2c(CNC(C(CC)C#N)=O)nnn2C)=O)CC2OC(=O)CC12 5597,C(=O)(C(=O)CC(C)C)N1CC(NC(c2nn(CC)c(O)c2)=O)C1 5598,c1(C(=O)NCC(C)(C2CCC2)NC(C(CC#C)C)=O)cncc(Cl)c1C 5599,C1(N(C(C=C(C)C)=O)C)CCCC(NC(=O)CCn2ccnc2)C1 5600,c1(C(N2C(C(C)(C)NC(CC(C)OC)=O)CCC2)=O)ccnc(C(F)(F)F)c1 5601,c1(C(=O)NCC(=O)NCC2(O)CN(CCCC)C2)ccc2c(=O)cc(C)oc2c1 5602,Cc1nc2nc(=S)[nH]n2c(C)c1CC(=O)NC(C)C(C)NC(=O)C(C)O 5603,C12(NC(C(C(CC)C)NC(N)=O)=O)CCC(CNC(=O)CC(F)F)(CC1)OC2 5604,N1(C(Cc2cc(C)no2)=O)CCC(NC(C2CCCOC2)=O)C(O)C1 5605,c1(CC(=O)NC2CCCC2CNC(=O)C(O)CF)ccc(C(F)(F)F)nc1 5606,c1(CNC(C(C2CCCN(C(CCSC)=O)C2)(C)C)=O)cnc(F)cc1C 5607,C(=O)(C1=C(Cl)CCC1)N1CCC(C(C)(C)NC(c2c(OCC#C)nccc2)=O)C1 5608,Cn1nnnc1SCCC(=O)NC1CC(F)(CNC(c2cc(CCO)on2)=O)C1 5609,CC(CC(N)=O)C(=O)N1CC(CNC(=O)C2CC2)C2(CC2)C1 5610,N1(C(c2ccc(OCC)cc2)=O)CC2(CCC2NC(c2ccc(CO)s2)=O)C1 5611,C1(NC(c2nn(CC)c(C)c2)=O)CC(C)CN(C(c2cc(Br)n[nH]2)=O)C1 5612,N1(C(C(C)C2CCC2)=O)CCOCC(NC(c2occc2-c2cnn(C)c2)=O)C1 5613,N1(C(C(=O)NCCC2CC(O)C(O)C2O)=O)CCCCCC1CO 5614,C1(F)(CNC(C2CCC(CNC(c3cnc(CC)o3)=O)O2)=O)CCOCC1 5615,C(C(=O)N(C)CC1CCCC1NC(=O)COC1(C)CCCC1)(C(C)(C)C)OC 5616,C1(NC(c2c(C)cc(CO)o2)=O)CCN(C(c2ccc(N)c(Cl)n2)=O)CC1F 5617,Cc1c(C(=O)NC(C(N2CC[Si](C)(C)C2)=O)C2CCCC2)ccn1C 5618,C1(NC(C=CCC2(NC(C(C(CC)C)=O)=O)CCC2)=O)CC(C2CCCC2)C1 5619,C(=O)(C1=CC2(CCN(C(c3ncc4ccccn34)=O)C2)C1)NCC(C)CCO 5620,N1(C(C2C(C)(C)CC2)=O)CC(NC(c2cc(O)cc(Cl)c2)=O)CC(O)C1 5621,CC1(C)CC(O)(CC(=O)NCC(C2CC2)NC(C23CC(C)(CO2)C3)=O)CO1 5622,CNS(=O)(=O)N1CCC(C(=O)N(CCCN(C(=O)CCNC(=O)CO)C)C)CC1 5623,C1(C)(CC)CC(NC(=O)Cc2ccc(C)s2)CN1C(=O)CCCCOC 5624,c1(NCCOCCN(C(C2C(CC)CCC2)=O)C)ncnn2c(Br)ccc12 5625,c1(NCCCc2nc[nH]n2)ccc(Cc2ccccc2)cn1 5626,c1(NC(=O)NC(CC)COCC2CC2)ccc(S(C)(=O)=O)nc1 5627,c1(CC=C)ccccc1C(=O)NCC1CN(C(C2CCOC(C)C2)=O)CC1C 5628,n1(CC(=O)NC(C(C)NC(c2cnc(C)o2)=O)C(C)C)ccc(=O)cc1C 5629,CC(C)CC(C)CC(=O)NC1CCN(C(=O)C2=CS(=O)CCC2)CC1O 5630,c1(C(N2CCC(OCCNC(C3CNC(=O)N3)=O)C2)=O)cc2ccccc2[nH]1 5631,C(=O)(C#CC(C)(C)CNC(=O)C=C(C1CC1)C1CC1)NCC1C(C)C1 5632,c1(C(C)C)ccccc1C(N1CCOC(C(=O)NCCC2CCO2)C1)=O 5633,C1(C(=O)NCC2N(C(C=CC=CC)=O)CCN(C)C2)Cn2c(C)nnc2CN1 5634,C1(CCNC(C2C(C)C2)=O)CCN(C(=O)CCSC2CCOCC2)C(C)C1 5635,c1(C(=O)OCC)cnc(NC(=O)N(C(C)C)Cc2coc(-c3ccccc3)n2)[nH]1 5636,Cc1ccc(NC(C2CCCC(NC(c3ccc(Br)cc3Br)=O)C2)=O)c(I)n1 5637,c1(C(=O)NCC2(NC(c3cncc(C=C)c3)=O)CCC2)nnc(O)c(Br)c1O 5638,N1(C(c2ncc(C)s2)=O)CCc2c(Br)ccc(NC(c3ccnnc3)=O)c2C1 5639,C12(c3onc(-c4c(OC)ccc(F)c4F)n3)CCCN(C1)S(=O)(=O)C2 5640,CC#CCCCC(=O)NC1CC(CNC(C2CCCCO2)=O)C1 5641,C(N=c1[nH]c(N2CCC(C(C)C)C2)nc2c1CCCCC2)C1(OC)CC1 5642,C(c1ccc(F)c(F)c1)=CC(N1CCC(C)(NC(C(CSC)O)=O)C1)=O 5643,C1(NC(C=C(CC)CC)=O)CC2CC(C1)N(C(C1CCC(C#N)CC1)=O)C2 5644,c1(OC)cc(C(N2CCC(N(C(=O)Cc3coc(C)n3)C)C(C)C2)=O)ccc1Cl 5645,c1(C(=O)NCC(CC)NC(C2CCC2c2nc[nH]n2)=O)nc2cccnc2s1 5646,c1(C(N(C(CNC(CC2C(C)CCO2)=O)C)C)=O)nn(C)c2c1CCCC2 5647,N1(CC(=O)NCCC(O)CNC(c2cccnc2)=O)CCOC1=O 5648,c1(C(=O)NCC(C)NC(=O)C#CC2CCOC2)cc(S(=O)(=O)N(C)C)cn1C 5649,N1(CCC(=O)OCCCCCCC)CCCc2cc(OC)ccc21 5650,CCN=c1[nH]c(C(N2CCCC2C(C)NC(=O)CN(C2CC2)CC)=O)cs1 5651,c1(C(N2CCC(NC(C(C3CCC3)OCC)=O)C2)=O)ccc(OC)cc1OC 5652,C(=O)(C(C)CC(C)C)NC(c1cnn(C)c1)C(=O)NCC(C(=O)OC)(F)F 5653,c1(C(=O)NC(CCNC(c2cccc(C)c2F)=O)C)cc2c(o1)CCCC2 5654,C(=O)(C(Cc1cn[nH]c1)NC(=O)C(Cl)Cl)N(CCCC)C 5655,C1(C(=O)NC2CCN(Cc3nc(-c4ccccc4)no3)C2)CC2CCC1O2 5656,C(=O)(C(C#N)C(C)C)NCC(CN(C(=O)CCC1CC1(C)C)CC)(C)C 5657,c1(SCC)cncc(C(=O)NCCNC(C2CC(O)CN2)=O)n1 5658,c1(C(C(=O)NCCOCC)N(C)CC2CCC(C)CC2)ncc2ccccn12 5659,C(=O)(C(C)(CC)CCCCCC)NCC1CC(F)(CNC(C(CC#C)C)=O)C1 5660,c1(OC(=O)CNC(=O)OCCOCCOC)c(SC)cccc1Cl 5661,c1(NC(C(CC=CC)NC(c2ncnc(O)c2F)=O)=O)ccc2n[nH]cc2c1 5662,C1(C#CC(=O)NCCCC(C)(C)NC(=O)C(O)CC(C)(C)C)(CC)COC1 5663,N1(CC=CC(=O)NC(CNC(=O)C2CC2)CC2CCCS2)CCOCC1 5664,N1(C(C2(CC=C)CCCN2C(c2ccc(C3CC3)o2)=O)=O)CC(=O)N(C)CC1C 5665,C(CCN=C(NCC1(C2CC2)CC1)N1CCN(c2snc(C)c2C#N)CC1)OC 5666,N1(C(CC(C)c2cnn(C)c2)=O)C2CCC1C(CNC(c1ccon1)=O)C2 5667,N1(C(C(C2CC2)SC)=O)CC=C(C(=O)NC2COCCC2O)C1 5668,c1(C(=O)NCC23C(CN(C(C(CC)SC)=O)C2)CC3)ccc2c(n1)CCC2 5669,N1(CC(=O)NCC(C)(C)OCCNC(=O)C(O)c2ccsc2)CCNC1=O 5670,n1(CC)ncn(NC(=O)C(Cn2cncn2)NC(=O)CC2CCOC2)c1=O 5671,N1(C(CCc2ncn(C)c2)=O)C2CCC1C(NC(=O)CCN1CCOC1=O)C2 5672,C1(CNC(=O)Nc2cncc(SC)c2)CC2(C1)OCCO2 5673,C1(O)(C(C)NC(CCn2ncc(C)c2)=O)CCN(C(c2sc(F)cc2C)=O)CC1 5674,C1(O)(CC(=O)NCCN(C)C)CCN(C(c2ccc(C#N)cc2)=O)CC1 5675,c1(CCC)sc(C(N2CCC(C(=O)C(F)Cl)CC2)=O)cc1CC 5676,c1(C(=O)NCC2(NC(c3cc(C(C)C)no3)=O)CCCC2)cc(N)cc(F)c1 5677,C(=O)(C(C)(O)C(F)(F)F)N(CCCNC(c1c(F)ccc(CC)c1)=O)CC 5678,C(=O)(CC(O)C(C)C)NC(CCC(N1CC2C(C(=O)NC)C2C1)=O)C 5679,CC1(C(=O)NCC2(CNC(=O)CCF)CCC2)COC(=O)OC1 5680,c1(C2CN(CCNC(CCC#C)=O)C2)ccc([N+](=O)[O-])cc1Cl 5681,C(CC)(c1ccc(C)cc1)=CC(N1CCC(CC=C)(NC(=O)CN2CC=CC2)C1)=O 5682,c1(C(=O)NC(C(C)C)CNC(C2CCS(=O)(=O)CC2)=O)cc2cccnn2c1 5683,Cc1nccc(=NCC2CCN(C(=O)CC3(C)CCS(=O)(=O)N3)C2)[nH]1 5684,C12(CCCCC1)C(=O)N2.C1(C(=O)NOCC(=O)N(C)C)(CC#C)CC2(CC2)C1 5685,N1(C(c2c(COC)noc2)=O)CC2CC(C1)CN(C(=O)C(C)(C)C1CCC1)C2 5686,c1(C(=O)NC(c2cnc(C)s2)C)cc(S(=O)(=O)CC2CC2)ccc1F 5687,c1(OC)ccc(CN2CCCC2C(=O)Nc2ccccn2)c(C)c1C 5688,CC(C)(C)CC(C(=O)NC1(C)CC2(CCC2)C1)NC(C1CC1c1ccco1)=O 5689,c1(OCC(=O)NC2CCCC2CNC(c2ccnc(O)c2)=O)ccc(Cl)cc1F 5690,Cn1cc(S(=O)(=O)NCC(=O)NC2CC(CC3CC3)C2)cn1.C12CCCN1C2=O 5691,C#Cc1ccc(C(=O)NC(CCC)C(=O)NCC(O)C(N)=O)nc1 5692,c1(N(CC(C)NC(C(C2CCOCC2)C)=O)C)c(Br)cccc1[N+](=O)[O-] 5693,C(=O)(CCCCC(C)CC)NCCC(=C)CNC(c1csc(Cl)c1)=O 5694,CCCC(C)(CC)C(=O)NC1CCCC(NC(=O)Cc2ccc(O)c(C)c2)C1 5695,N1(C(c2cc(OCC)ns2)=O)CCN(C(C2CC=CCO2)=O)CC1CO 5696,N1(C(C(C(C(C)C)O)C)=O)CCC2(CC1)CN(C(C1C3CC4C(C3=O)C14)=O)C2 5697,C1(NC(=O)CCc2ccncc2)CCCCC1NC(=O)Cn1cc(Br)cn1 5698,C(=O)(C1CCc2ccccc21)N1C(CN(C)C(C2CC(N=[N+]=[N-])C2)=O)CCCC1 5699,CCCCC(CC)CC(=O)N1CC2CC1CN(C(c1cn(CCCF)nn1)=O)C2 5700,CC(C(=O)NC1CC(NC(=O)COCc2nnc(S)n2C)CC1O)C(F)F 5701,CCC(CCO)NC(=O)CCC1(NC(=O)C=Cc2cc[nH]c2)CCC1 5702,C12(C(=O)OCC)CCC(CC1)CN2C(=O)C(N1CCCC1c1ccnc(C)n1)=O 5703,CCCCC(CN=c1nc(C(C)C)[nH]s1)NC(c1n[nH]c2ccccc12)=O 5704,N1(C(c2c(CC)nc[nH]2)=O)CC(NC(C2CC2c2cnn(C)c2)=O)C2(CCC2)C1 5705,C1(CC=C)(C(=O)NCC(F)C2CCC2)CCN(C(=O)C(C)C(C)C)C1 5706,C1(C(=O)NCCN(C(CSCCCC)=O)CC2CC2)CNC(=O)N1C 5707,c1(OC)cccc(Br)c1C(N1CCC(NC(=O)CSC)C(C)C1)=O 5708,Cc1cc2ncc(C(=O)NCC3CC(C)CCN3C(C3CC3(Cl)Cl)=O)c(C)n2n1 5709,N1(C(CC=C)=O)CCN(C(=O)CN2CCc3ccccc32)C2CCCCC2C1 5710,Cn1cc(C(N2CC3(NC(=O)CCF)CCCC3(F)C2)=O)c(=O)c2cnn(C)c12 5711,Cc1nc(C(F)(F)F)ccc1C(=O)NCC1(NC(=O)Cc2cnc[nH]2)CC1 5712,C(c1cc(F)c(F)c(F)c1)=CC(N1CCCN(C(C2(OC)CC2)=O)CC1C)=O 5713,CCC(C(=O)NC1(CNC(=O)CC2(C#N)CC2)CCCC1)n1ccnc1 5714,c1(NS(Cc2cn(C)nc2)(=O)=O)ccc(S(=O)(=O)NC2CC2)cc1 5715,c1(OC)ccc(CNC(N2CCOCC2C(=O)NCC2CCCO2)=O)cc1OC 5716,c1(OC)ccc(F)cc1-c1nc(Cc2ccccc2)nn1C1CCCC1(C)C 5717,c1(CNC(c2ccc(Cl)c(F)c2)C(=O)O)cc2cc(F)ccc2nc1Cl 5718,c1(C(=O)NCC2(C)CCN(C(c3ccc(O)nn3)=O)C2)ccc(C#N)c(Cl)c1 5719,N1(C(c2c(C(C)C)scn2)=O)CCC(C)(C)C(NC(=O)CC2C=CCCC2)C1 5720,CC1(C)Oc2ccc(C(N3CCC4C(CCN4C(=O)C(O)C(F)F)C3)=O)cc2O1 5721,N1(C(c2c(C)oc(Br)c2)=O)CC(NC(c2ccnn2C)=O)CC(C)C1 5722,C1(C(=O)NCc2nc(C)sc2)CCN(Cc2ccc(F)c(Cl)c2)CC1O 5723,c1(CC(=O)NCC2CC(NC(=O)C=CC(N3CCOCC3)=O)C2)cncc(O)c1 5724,C(CC(C)C(=O)NC1CCC(N(C)CCn2nccn2)CC1)=CC 5725,C1(NC(=O)NCC2(C)CC2(F)F)CN(Cc2ccccc2)CC1C#N 5726,C(CNC(=O)C=CCCC=C(C)C)(C(C)C(C)C)NC(c1c(C)oc(CO)c1)=O 5727,c1(C(=O)NC2CCN(C(C(COC)OCC3CC3)=O)CC2)cccn2nccc12 5728,c1(C(N2CC(NC(CC=CCC)=O)C(OC)C2)=O)cn2c(n1)CC(C)CC2 5729,Cc1ccc(Br)c(S(=O)(=O)N2CC(CO)CC2C)c1 5730,c1(C(=O)NC(C2N(C(CCc3n[nH]c(=N)s3)=O)CCC2)(C)C)cc(Cl)nnc1Cl 5731,c1(CC)cccc(CNC(c2[nH]ccc2CNC(C2COCC(C)O2)=O)=O)c1.CN 5732,C(=O)(CC(C)C(=O)N1CCC(C)C(NC(C2CCCC2)=O)C1)OC 5733,Cn1cc(C(N2CCC(NC(c3cc(CO)[nH]n3)=O)C(F)C2)=O)c2cccnc12 5734,C(CCCS(=O)(=O)CCCCO)NC(=O)NC(CC(=O)OC)(C)c1ccccn1 5735,C(=O)(C(C)(C)CC(C)C)NC(CC(C)NC(c1c(CC)ncnc1CC)=O)C 5736,C1(NC(C2CCOC2)=O)CN(C(c2ccc(C(F)(F)F)cn2)=O)C2(CCC2)C1 5737,N1(C(Cc2c(COC)cccc2)=O)CC(NC(C2CCOCC2)=O)CC12CCC2 5738,C1(O)(C(N(CCCCNC(CCNC(C)=O)=O)C)=O)CC1(C)C 5739,N1(C(C2CCC(CC)O2)=O)CC2(C)CN(C(C3CNC(=O)N3)=O)CC2(C)C1 5740,c1(C(=O)NCCOc2cc(Cl)c(Cl)cc2Cl)cc([N+](=O)[O-])c(F)c(F)c1Br 5741,c1(C(N2CCN(C(=O)CCc3cncs3)C3CCCC23)=O)n[nH]c2ccccc12 5742,N1(C(CCCC#CC)=O)CC2CC(F)(F)CCC2(NC(=O)COCC)C1 5743,S(=O)(=O)(c1cnn(C)c1)NC(C(=O)NCCC(C)NC(=O)COC(F)(F)F)C 5744,c1(C(=O)OCC)ncoc1C(N1CCC1CNC(=O)CN(C1CCSC1)C)=O 5745,C(c1cccc([N+](=O)[O-])c1)=CC(=O)NCCOCCCNC(C1CCCCS1)=O 5746,C(c1ccn(C)c1)=CC(=O)NC1(CCNC(C(C)OCCCC)=O)CCC1 5747,N1(C(COC2CC(NC(C3C(C)CCOC3)=O)C2)=O)CC(F)CC(F)C1 5748,c1(OC)cc(N)c(Cl)cc1C(N1CCCC1CNC(=O)C1=CC2CCC1C2)=O 5749,c1(OCC)cccc(CC(=O)NCC2CCC(NC(C3(CO)CCC3)=O)CC2)c1 5750,C(C(=O)NCC1CC(F)CN1C(c1cc(C(F)(F)F)n[nH]1)=O)(C(C)C)OC 5751,C12CCCCCCN1C(=O)CNC2=O.C(COCCOCCO)OCC 5752,c1(NC(C)=O)ccc(Cl)cc1C(N1CC(c2ocnc2CNC(=O)C(C)C#N)C1)=O 5753,C1(O)(CC(=O)NCCCCN(C(=O)CS(=O)(=O)N(C)C)C)CCCCCC1 5754,N1(C(c2nc(CCCC)sc2)=O)CCCN(C(c2cc(C)ncn2)=O)CCC1 5755,c1(NC(c2ccn(CCNC(CC3(C)CCCC3)=O)c2)=O)cnn2c1CCCC2 5756,N1(C(COC(C)=O)=O)CCN(C(=O)C(F)C2CCC2)C(C2CC2)C1 5757,CCC(C(=O)Nc1nc(COc2ccc(F)cc2)cs1)C(=O)O 5758,Cc1ccc(C(C)(C)C(=O)N(C(C)CC(F)F)CCO)c(C)c1 5759,c1(CC)noc2ncc(C(=O)N(CCN(c3nnc(C)s3)C)CC)cc12 5760,c1(CC(=O)NC2C=CCN(C(CCC#C)=O)C2)c[nH]c2cc(C)ccc12 5761,N1(C(=O)NCCc2nc(CC)sc2)CCCN2CCCC12 5762,CC(C(C)(C)NC(=O)Cc1csc(Cl)n1)NC(=O)C=C1CCCC1 5763,C(C(COC)CC(=O)N1CC(CCNC(C2(Br)CC2(C)C)=O)C1)OC 5764,C(=O)(CC(CCC)NC(=O)C=Cc1ccncn1)NCC(=C)Br 5765,N1(C(C(c2ccc(OC)cc2)CC)=O)CC2CN(C(c3ccc(C)o3)=O)CCC12 5766,C#Cc1ccc(Br)c(C(=O)NC2CC(C)CN(C(c3[nH]cnc3CC)=O)C2)c1 5767,C1(NC(C(F)=C(C)C)=O)CC2CC1CN(C(=O)C(c1c(C)noc1C)(C)C)C2 5768,c1(NC2(CC(=O)Nc3ccc(Cl)cc3F)CCC2)ncnc2[nH]ccc12 5769,Cc1cc([N+](=O)[O-])cc(C(=O)NC2CN(C(c3c(C)cnn3C)=O)C(C)(C)C2)n1 5770,c1(NC(=O)C(=O)NC2CC(N3CCC3)C2)ccccc1 5771,N1(C(c2cc(OC)c(Cl)cc2)=O)CC2CCC(C1)N2C(=O)C(C)(C)CCl 5772,C1(C2CCCCC2)(C(=O)NC2CC(NC(C3(C#N)CCOC3)=O)C2)CC1 5773,C1(NC(C=CCOC)=O)CCN(C(C2CCC(=O)N2C(C)C)=O)CC1O 5774,N1(C(CCN(CC#C)C(C2CCCC2)=O)=O)CCOC(CN(C)C)C1 5775,c1(OC(C)C#N)ccc(C(=O)NCC2CC2NC(c2cc(CO)ccn2)=O)cc1 5776,c1(CC(=O)NC2C(C(N(C3CCSC3)CC)=O)CC2)ccc2occc2c1 5777,C(=O)(C(CC)CC(C)C)N1CC(C2CC2)(C(n2cc(C3COCC(C)O3)nn2)C)C1 5778,c1(C(=O)NC2CC3CN(C(C(CC)(C)O)=O)C(C2)C3)n[nH]c2c(C)cccc12 5779,N1(C(c2c(C)scn2)=O)CC2OCC(NC(C3CC4(C3)CC(C)C4)=O)C2C1 5780,c1(NC)cnc(C(=O)NCC2CCCN2C(C2CCN(C)C2)=O)cn1 5781,N1(C(C(CC)(C)OC)=O)CCOCC(F)(CNC(c2nnc(C(C)(C)C)s2)=O)C1 5782,CCCCCCC(C)C(=O)NCC12CCC(C1)N(C(=O)CN1CC(=O)NC1=O)C2 5783,C1(C(N(C2CCN(C(=O)C(C)(C)OC)CC2)CC#C)=O)C2CC2C2CC12 5784,N1(C(N2C(C)(C)CCC2)=O)CCC12CCC(C)CC2 5785,C(CC(=O)N1CCN(CC2CC2)CC1)(C(F)(F)F)NC(c1cccc(C)n1)=O 5786,C(C)(C1=CCN(C)CC1)NC(C1C(CC)OCCC1)=O 5787,C1(CC(N2CCC(C)(CCO)C2)=O)CC2(C1)CN(C(C1(CCCF)CC1)=O)C2 5788,N1(C(c2cn(CCO)nc2C)C(=O)NCCCOC)CCc2c(F)cc(F)cc2C1 5789,c1(C(=O)NCC2(O)CCN(C(COC(CC)(C)C)=O)C2)ccc2c(c1)CC2 5790,c1(OC)nn(C)cc1NC(=O)CC1C=CC(NC(=O)COCOC)C1 5791,CCCC(C)(C)C(=O)NCCC(O)CNC(C1CCC(=O)N(C)C1)=O 5792,CCC(C)(F)C(=O)N(CC(C)OC)CC1(N2CCSCC2)CCCCC1 5793,C1(N(C(CS(CC)=O)=O)C)CCCC2CN(C(c3ccc(N)c(Cl)c3)=O)CC12 5794,c1(OC)ccc2c(c1)NC(=O)C2CC(=O)NCC(F)CNC(=O)C=C(C)C 5795,S(=O)(=O)(c1ccc(NC(c2cc(C)ccc2F)CO)nc1)N1CCC=C(C)C1 5796,C12(NC(c3c(C)ocn3)=O)CC1CN(C(=O)Cn1nc(C(F)F)cc1C(F)F)C2 5797,c1(C(=O)NCc2scc(CNC(CCC=C=C)=O)n2)cccc(F)c1C 5798,N1(C(c2c(C)scc2)=O)CCC(NC(=O)C(C(C)C)N(C)C)C(O)C1 5799,Cc1cc(C(=O)NC(CCNC(C2CCCSC2C)=O)C(C)C)cnc1C(F)F 5800,c1(C(N2CCC(CCNC(C(CC)(C)C#N)=O)C2)=O)cc(S(N)(=O)=O)cn1C 5801,N1(C(C2N(C(C)=O)CSC2)=O)CC2CN(Cc3ccc(Cl)cc3C(F)(F)F)C2C1 5802,c1(C(=O)NC2CCN(CC)CC2)sc(C=O)c(Br)c1Br.C12(C)CN(C1)CC(=O)C2 5803,CC(C)CS(=O)(=O)CC(=O)NC1CC2CC(NC(c3coc(C(F)F)c3)=O)C2C1 5804,C(CS(=O)(=O)C1=NOC(C)(C)C1)OC(CCc1ccc(OC)cc1)=O 5805,O(NS(=O)(=O)c1ccc(F)cc1)CC(=O)NC1CCC(NC(CCOC)=O)CC1 5806,c1(C(=O)OC)ccc(C(C(=O)NCC2CC2)N(C2(C)CCC2)C)cc1Cl 5807,C1(CC(=O)NC(C)C(C2CCCCC2)NC(=O)OC(C)(C)C)CCCC2CC12 5808,C(=O)(CC1=NNC(=O)C1)NC1CCC(NC(CN(CC)CC)=O)C1 5809,c1(C(=O)NCCN(C(C=CC)=O)CC)cccc(C2CCCOC2)c1 5810,N1(C(c2ccc(C)n2C)=O)CC2CCC1CN2C(c1ccc(F)cn1)=O 5811,C1(CCNC(CCSCC(C)C)=O)CN(C(c2cc(CO)[nH]n2)=O)CCO1 5812,C12(C(=O)NCC3(OCC)CCCC3)CC(CO1)N(C(C1CCC1C)=O)C2 5813,Cc1cccc(C(N2CC(C(C)NCCCS(N)(=O)=O)C2)=O)c1 5814,c1(OC)n[nH]c(C(=O)NCC2CC(OC)CN2C(=O)C=C(C)c2ccco2)c1Cl 5815,S(=O)(=O)(c1cccc(=NCc2cc[nH]c(=N)c2)[nH]1)N(CC(C)OC)CC 5816,Cc1cc(S(=O)(=O)NC(=O)C(C(=O)N(C)C)C(C)C)sc1C 5817,C1(C(=O)NC(C#C)C(C)(C)C)CCC2(CC2)N1C(=O)C(C)NC=O 5818,C1(NC(CC2(C)CC2F)=O)CCC2(CC1)CN(C(=O)CCCCC#N)C2 5819,C1(S(N)(=O)=O)(C(=O)NC2CCC(N(C(=O)C=C(Cl)Cl)C)CC2)CCC1 5820,c1(C(=O)NC2CCN(C(CCC(C)OCC)=O)CC2)ccc2nc(S)oc2c1 5821,CC(C)(F)C(C)(F)CNC(c1cccnc1CNC(=O)CCC1CCCOC1)=O 5822,C1(C(C)(C)C)CCC(C(=O)NOCc2cncc(CC3CC3)n2)CC1 5823,c1(NC(c2c(C)nns2)C)[nH]c(=NC2CC=CCC2C)nc2scnc12 5824,c1(CCC(=O)N(C(C2CCN(C(CC)C)C2)=O)C2CC2)ccc(C(F)(F)F)nc1 5825,O=S(=O)(c1ccc(F)cc1F)NCC1CN(Cc2cnc(Br)c(F)c2)C1 5826,C1(NC(CN(C2CC2)CC)=O)CCCC(NC(c2ccnc(C3CCC3)c2)=O)C1 5827,C(=O)(C(C#N)C(C)C)N1C2C(C(=O)NCC(CSC)(C)O)C(C2)C1 5828,C1(CNC(CSCC(=O)OC)=O)COCCN(C(=O)Cn2cnc([N+](=O)[O-])n2)C1 5829,C(=O)(C1=COCCO1)NCC1(CNC(C(C(C)C)C)=O)CC1 5830,C1(NC(C2(CCC=C)CC2)=O)CS(=O)(=O)CC1NC(c1cc(C(C)=O)cs1)=O 5831,C1(NC(c2cc(C3CC3)cs2)=O)CC12CCN(C(=O)CC1CC1(Cl)Cl)C2 5832,c1(C(N2CC(SC)C(NC(C3CC3C3CC3)=O)C2)=O)ccc2c(C)cc(O)nc2c1 5833,c1(C(N2C(C)(C)CC(CNC(C3CC4(CC4)C3)=O)C2)=O)ccn2cccc2c1 5834,N1(C(C2CC=C(C)CC2)=O)CCC2CN(C(C3CCC(=O)N3)=O)C2C1 5835,n1(CC(N2CCCC(CN(C)C(c3cccn3C)=O)C2)=O)cc(Cl)c(O)nc1=O 5836,C1(C(N(C2COC(C)(C)C2)C)=O)CN(C(=O)Cn2cncn2)CC12CC2 5837,c1(C(=O)NC(C)(C)CNC(c2ccc(N)cn2)=O)ncc2cc(Br)ccc2n1 5838,CCC(C)C(O)C(=O)NCC1CC(C)(C)CN1C(C1CC1(F)F)=O 5839,C(=O)(CC(CCCC)NC(C1(C#C)CC1)=O)N1C(C#C)CCC1 5840,c1(C(=O)NC(CN(C(=O)C=C(C)C(C)C)CC)C)ccc(O)c(C(C)(C)C)c1 5841,Cc1c(F)ccc2[nH]c(C(N3CC(NC(=O)C(O)C(C)C)C4(CCC4)C3)=O)cc12 5842,c1(CC(C)NC(c2ccc(C(F)(F)F)c(Br)n2)=O)coc2ccccc12 5843,C12(C(N(c3ccc(Cl)c(C(F)(F)F)c3)C)=O)CCOC1CC(=O)NC2 5844,c1(SCCC(=O)NCC2C(NC(Cc3cn(CC)nn3)=O)C2)ccccc1Cl 5845,C1(C(N2CCC(CNC(C3C(=C)C3)=O)CC2)=O)OC2CCC1CC2 5846,C1(C(=O)NCC2(COC)CCN(C(=O)OC(C)(C)C)C2)OCCCC1(C)C 5847,c1(C(c2n(CCCC)nnn2)NCC=C)cccc(OCC#N)c1 5848,CC1CN(C(c2occc2Cl)=O)CC1CNC(=O)CCOCC1CCC1 5849,n1(CCC(=O)NCC2(C(N)=O)CN(c3cc(O)ncn3)C2)cc([N+](=O)[O-])cn1 5850,CC(C)CCCCC(=O)NCC1CCC1C(N1CCC(n2cncn2)C1)=O 5851,C12(OC)CCC(C(=O)NCC3CCC(NC(=O)CCCC4CC4)C3)(CC1)C2 5852,C=CC(C)CCN=c1[nH]c(=NCC2(C)CC2(F)F)c2cc(Cl)ccc2[nH]1 5853,N1(C(C(COC)C)=O)CCC(CC(C)NC(=O)CN2CCNC(=O)C2)CC1 5854,CCCCC(CNC(=O)CC=CCOC)NC(=O)CCC(=O)NC 5855,C(C(C)C(C)C(=O)NCC(C)CN(C(=O)CC=Cc1ccc(F)cc1)C)OC 5856,C1(COC)N(C(C23CC2CN(C(c2cc(C4CC4)no2)=O)C3)=O)CC1(C)C 5857,N1(C(c2c(C)cnnc2)=O)CC(O)CCC1C(=O)NC(c1nncs1)C 5858,Clc1cccc2ncc(-c3nc(C4CC45CCC5)no3)cc12 5859,N1(C(C(CC=C)c2ccccc2)=O)CCN(CCNC(C2CC2Cl)=O)C(=O)C1 5860,C1(C(=O)Oc2cccc3c2OCCO3)COc2c(cc(Cl)cc2[N+](=O)[O-])C1 5861,C1(C(N(CCN=[N+]=[N-])C)=O)CC(O)CCN1C(C1CCCC(C#N)C1)=O 5862,CCCC(O)CC(=O)NC(C)(C)CCCNC(c1cc(-c2ccc(C)o2)[nH]n1)=O 5863,N1(C(c2c(C)n(C(C)C)nc2)=O)CC2CC1CN(C(=O)CC1CC3(COC3)C1)C2 5864,c1(C(C(=O)NCC=CCNC(C2CCC(F)C2)=O)(F)F)c(F)cccc1F 5865,N1(C(C(=O)NCCc2c(OC)cccc2)CC(C)C)CCCNC(=O)C12CCC2 5866,c1(NC(C(Br)=C(C)C)=O)nccc(C(C)(C)C)n1.C12CCCC1CNC2=O 5867,C1(C(=O)NC(C)CNC(=O)C=Cc2cnc(C)s2)(CC)CCC(O)CC1 5868,C1=CCCC(Nc2ncc(-c3ccccn3)s2)CCC1 5869,C(CC(C)(C)CC(=O)N1CCCN(C(=O)Cc2c[nH]c(=N)nc2O)CC1)OC 5870,N1(C(CN(C(C2(CC=C)COC2)=O)C)=O)CCN(C(c2cscc2F)=O)CC1 5871,C1(NC(C(C)Oc2ccccn2)=O)(CF)CCN(C(c2coc(C3CC3)n2)=O)C1 5872,C1(NC(c2nc(COC)sc2)=O)CC2CN(C(=O)COC3CCC3)CC12.CCC 5873,N1(C(Cn2nnc(C)n2)=O)CCC(C)(C)C(CNC(=O)CC2(C)CCOC2)C1 5874,c1(CC(N2C(C(C(=O)Nc3nc(C)c(C)[nH]3)(C)C)CCC2)=O)cc(Cl)ccc1F 5875,C1(C(C)NC(C2CCCN(C(C)C)C2)C)CN(C)CCN1C 5876,CCCCCC(O)C(=O)N1CCN(C(c2cnc3occc3c2)=O)C(C(C)C)C1 5877,c1(N2CCC(O)(C(=O)NCC(C)(C)O)C2)ncnn2cccc12 5878,c1(C(N2CCC(NC(C3(C)CCCS3(=O)=O)=O)C2)=O)cc2c(Cl)nccc2o1 5879,c1(C(=O)NC2C3CN(C(C4(OCC)CC4)=O)C2C(O)C3)sc2cccnc2c1Cl 5880,C1(CNC(c2cnoc2)=O)CCN(C(c2cn3ccccc3n2)=O)CC1(F)F 5881,Cc1ccc(C(N2CC(C(F)Cn3cc(C4CCCC4O)nn3)C2)=O)o1 5882,CC1(C)C(CO)CCN1C(=O)CC1CCN(C(C2CCCOCC2)=O)CC1 5883,N1(C(=O)OC(C)(C)C)C2CCC1CN(C(=O)OCC1CCCN(S(C)(=O)=O)C1)C2 5884,N1(C(C=C(CCC)C)=O)CCC2CN(C(c3cnn(C(C)(C)C)c3)=O)CCC2C1 5885,C1(C(=O)NC2C3CN(C(c4ccc(SC(C)C)cc4)=O)C2C3)CCC(C)NC1=O 5886,C=Cc1cc(C(=O)NCC2CCC(C)CN2C(c2nnc(CC)s2)=O)cc(F)c1 5887,N1(C(Cc2cnc(C)[nH]2)=O)CCCC2(C1)CN(C(c1cccc(O)n1)=O)C2 5888,CCCCC(C(=O)NCCC(C)NC(=O)CCCc1cccs1)NC(N)=O 5889,c1(N2CCN(CC)CC2)cccc(NC(c2nc(C3CC3)oc2C)=O)c1C 5890,N1(C(c2cc(N)c(N)nc2)=O)CCN(C(=O)C2=CCOCC2)C2CCCCC12 5891,c1(CC)nc(=NC2CC(C)N(C(c3cncc(F)c3)=O)C2)s[nH]1 5892,N(C(=NCCc1nn(C)cc1C)N1CCCC(CSC)C1)C(COC)C 5893,c1(CN(C(c2c(CC)ccs2)=O)C)cnn2c1CN(C(c1c[nH]c(=N)s1)=O)CC2 5894,C(=O)(CCCCC(F)(F)F)NC(CN(C(c1c(C)nn(CCC)c1C)=O)CC)C 5895,N1(C(CCSCCC)=O)CCCCC1C(=O)NC1CCNC(=O)C1 5896,c1(OC)nscc1C(=O)NC1COCC1NC(C1CC1(C)C)=O 5897,C(=O)(C(CC)CCOC)NCC(CC=C)NC(=O)Cc1conc1C 5898,c1(C(N(CC(C)NC(c2cnc(CC)o2)=O)CC)=O)ccc(C(F)F)cn1 5899,N1(C(C(C)(C)C2CCCC2)=O)CCN(C(c2cn3ccnc3s2)=O)C(C(F)F)C1 5900,CC(=O)CCCC(=O)NC(C(=O)NCCOC1CCCC1)C(C)C 5901,C(=O)(C(O)CC(C)C)NCCN(C(COCc1onc(CC)n1)=O)C1CC1 5902,N1(C(c2snc(C)c2N)=O)CCC(N=[N+]=[N-])(C(=O)NCC(O)CF)C1 5903,CCC(CC)C(C(=O)N(C(C)C(=O)NC(C)(C)CC(C)(C)C)C)OC 5904,O=S(=O)(c1cccc(N2CCC(OCCO)CC2)n1)NCc1cc(C(F)F)on1 5905,N1(C(C2CC(=C)C2)=O)CC2CC2(NC(=O)Cn2ccnn2)C1 5906,C1(C(=O)NC2(SC3C(OC)CC3)CCCC2)CCCN(C(=O)COC(C)(C)C)C1 5907,Cc1ccc(O)c(CNC(=O)C(c2ccnn2C)NC(C2CCN(C)CC2)=O)n1 5908,N1(C(=O)Cc2cn[nH]c2)CC(C2CN(C(=O)CCSc3ccc(F)c(F)c3)C2)C1 5909,C1(C(N(CCCn2cc(CN3CC4CC4C3)nn2)C)=O)CCC(=O)C(C)C1(C)C 5910,C1(CC(C)NC(C2(C)CCCS2)=O)CCN(C(=O)CC2CCC(=O)N2C)CC1 5911,N1(C(CC(=O)OC)=O)CCCC(O)(CNC(c2cc(Cl)ncc2OC(F)F)=O)C1 5912,C1(CN=C(NC(c2cccs2)C)NCCOCCS)CCCCC1(F)F.C(C)(C)C 5913,N1(C(C(c2cncnc2)C)=O)CCC(C)CC1CNC(=O)CCCc1cccnc1 5914,S(=O)(=O)(c1ccc(N2CCCC(NCC(F)Cl)C2)c(Cl)c1)CNS(C)(=O)=O 5915,C12(CNC(=O)Cc3csnn3)CCCC1CCN2C(c1ncccn1)=O 5916,n1(CC(=O)NC(CNC(c2cc(C)c(C)s2)=O)(C)CO)ncn2nccc2c1=O 5917,C(=O)(CC(C)C(=O)N1CCC(NC(=O)CC2(C)CC2(Cl)Cl)C1C(C)C)OC 5918,c1(C(N2CC(NC(c3cc(O)cs3)=O)C2)=O)nc(CF)cs1 5919,CC(C#N)CN=C(NCCSc1ccccc1)NCc1cnccc1Cl 5920,Cc1c(C(=O)NCC2(NC(c3csc(C(F)(F)F)c3)=O)CCC2)cnn1C 5921,C(CC(C(=O)NCCOC(F)F)NC(=O)CCn1cnnn1)OC 5922,CC12CCC(C)(CN1CCC1CCNC1)C2 5923,N(C1c2ccccc2CC1C)C(C1CN(c2c(OC)cccc2)C(=O)C1)=O 5924,c1(C(=O)NN2C(Cc3c(CSC)cco3)COCC2)cc2n(c1)CCCNC2=O 5925,C(N=c1nc(N(C)CCN(C)C)c2c([nH]1)CCOC2)C1(CC)CCC(=O)N1 5926,S(=O)(=O)(c1cnccc1N(C)CC1(CO)CCOC1)N(C)CCC1N(C)CCC1 5927,c1(CNCC2CCN(C(C)=O)C2)cc2ncncc2s1 5928,c1(OC)cc(F)c(F)cc1C(=O)NCC1(CNC(C23CC4CC2C3C4)=O)CCC1 5929,C(=O)(C(Cc1cn[nH]c1)NC(c1cnc(O)o1)=O)N(CCOC)CC 5930,C1(C2CCN(C(=O)CCC(F)(F)F)CC2)(NC(C2CC(C)(C)OC2)=O)CC1 5931,C1(NC(COC)=O)CCCOC12CCN(C(=O)CC1CC1C(F)(F)F)CC2 5932,c1(CC)ccc(Br)cc1C(=O)NC(C)CCN(C)C(C1C(C)(C)C1(C)C)=O 5933,CN1CC(CNC(=O)NC2(CO)CCS(=O)(=O)C2)Cc2ccccc21 5934,c1(C(=O)Nc2nnc(Br)s2)nc2n(c1Cl)CCN(C(c1cc(Cl)ccc1Br)=O)C2 5935,C1(C)(NC(CN(CC(C)C)C(c2ccn(CCC)n2)=O)=O)CCC(C)(C)C1 5936,c1(-n2c(CCC3SC(=N)NC3=O)nc(COC(C)C)n2)ccc(Cl)c(F)c1 5937,C1(NC(c2c(C)scc2)=O)CN(C(c2cc3n(n2)CCC3)=O)CC12CCC2 5938,N#Cc1cncc(C(=O)NC2(CO)CCN(C(=O)Cc3sccc3Cl)C2)c1 5939,c1(CC(=O)NC2CC(F)CN(C(=O)Nc3ccsc3)C2)ccc(F)cc1[N+](=O)[O-] 5940,Cc1ncc(Cl)cc1C(=O)NCCC(C)(C)NC(=O)CC1CC(O)C1(C)C 5941,N1(C(CCc2n(C)ncc2)=O)CCC(C(N2CC(O)(C(F)F)C2)=O)C12CC2 5942,S1(=O)(=O)C2=CC=CC(=NCCCOC3CCN1C3)N2.C=CCOC(C)C 5943,c1(CC)cnoc1C(=O)N(CCC(C)NC(=O)C(C)OCC1CCOC1)C 5944,c1(NC(=O)NC2CCN(C(=O)OCC)C2)ccc(S(N)(=O)=O)c(OC)c1 5945,c1(C(N2CCC(C(C)(C)NC(CCOC(C)=O)=O)C2)=O)cn(C(C)C)nc1C 5946,c1(OC)cc(C(N2CCC(F)(C(=O)Nc3ccc(F)cc3Cl)C2)=O)cc(Br)c1 5947,c1(C(=O)NCC2CCCN(C(C3C(C#C)C3)=O)C2)cc2sc(Cl)cc2s1 5948,N1(C(CCC)=O)CCC(NC(C2CC2C2CCCN2C(=O)CC2(C)CC2)=O)C1 5949,CC(C(C)C(=O)NC(c1ccccc1)CNC(=O)CCS(C)(=O)=O)C(C)(C)C 5950,C1(NC(C(CC)n2cncn2)=O)CCC(C(=O)Nc2cnn(CCOC)c2)CC1 5951,c1(OC)ncnc(N2CCN(C(c3ccc(C(F)(F)F)nc3O)=O)C(C)C2)c1C 5952,O(NC(=O)C(CNC(C1CCCSC1C)=O)N(C)C)CCCOCC 5953,C1(C(=O)NCc2cc(NC(C)=O)sc2)CCN(C#N)C1 5954,c1(-n2c(C3C(C)C3C)nc(CSC)n2)ccc(F)c(F)c1 5955,CC1CCN(C(=O)CC(C2CCC2)C2CCC2)C1CNC(=O)CC1OCCCO1 5956,C1(C)(C(N2CCC(O)(CN(C(=O)C3=CCOC3)C)CC2)=O)CC(C(C)(C)C)=NO1 5957,C12(SCC(=O)OCc3nnc(CC(C)C)s3)CC(c3ccccc3)(CO1)C2 5958,c1(C(=O)NC2CC(NC(=O)CCc3nccs3)C2)ccc(CO)nc1 5959,c1(C(=O)NC(CNC(C2(CC=C)CCCC2)=O)CO)ccc(-n2cnnc2)cc1 5960,c1(CNC(C(C)C2CC2)=O)ccc(CN(C)C(C2CCCOCC2)=O)cc1 5961,c1(C(=O)Nc2n(CN3CC(SCC)C3)nc(C3CC3)c2)cccc2c1C(=O)NC2 5962,C1(NC(c2n(CC=C)nnn2)CC2CCC(C)(C)O2)CN(S(C)(=O)=O)CCC1C 5963,S(=O)(=O)(c1cnn(C)c1)NCC(=O)N(C1CCN(C(C2CCC(=O)NC2)=O)C1)C 5964,CC1CC(C(=O)NCC(C)(C)NC(=O)CCc2ccc(F)cc2)=NO1 5965,c1(CCCN(C(C)CNC(=O)C(C)N2CCCC2)C)ncccn1 5966,CC#CCCCC(=O)OCC1CN(C(C2CCCN2C(=O)C(F)(F)F)=O)CC1C 5967,c1(C(=O)NCC2C(NC(Cc3c(C)non3)=O)CC2)ccc(N)c2ccncc12 5968,C1(C(N(CCNC(C(C)CF)=O)CC2CC2)=O)CCc2ccccc2C1 5969,C(=O)(C(F)(F)CCn1cccn1)NCC(C)N(C(C1CC=C(C)CC1)=O)C 5970,c1(-n2cc(CN(C(CC)=O)C)nn2)c(C)cccc1[N+](=O)[O-] 5971,C(=O)(C(CC(F)F)C1CCC1)N(C)CC1CCN(C(=O)CCF)C1 5972,C1(C(N2CC(CNC(=O)CC3(C4CCCO4)CCOCC3)C2)=O)(CO)CCOCC1 5973,c1(OC)ccc2c(c1)C(=O)N2.C1(OC(C)=O)CCN(C(c2ccoc2Cl)=O)CC1O 5974,CC(C(=O)NCCOC(C)(C)CNC(C1CC(=O)NC(=O)N1)=O)C(C)S(C)(=O)=O 5975,n1(CC)cccc1C(=O)NCC(CCNC(c1ccc(SC)o1)=O)OC 5976,C(=O)(C1=CS(=O)CCC1)NCC(CC)NC(C(CC=C)C)=O 5977,c1(C(N2CC(NC(CC(CC)CC)=O)C(C)C2)=O)ccc2c(c1)N(C)CC2 5978,C(C(=O)N1Cc2ccccc2CO1)C1(NC(COC)=O)CCC1 5979,Cc1ccc(N(C(=O)CC2CCCN2C(C2CC3CC3C2)=O)C)c(C)c1 5980,c1(NC(C2CCC(Cc3ccc(COC(C)=O)o3)C2)=O)cc(Br)cc(F)c1C#N 5981,c1(C(=O)NC2(CC)CN(C(=O)CN3CCCCC3=O)C2)ncncc1C 5982,N1(C(C(CO)OC)=O)CCC(C(=O)NCC2CCN(C3CC3)C2)CC1(C)C 5983,N1(C(CNC(=O)OC)=O)CCOCC1CC(N1CC(F)(F)C1C1CC1)=O 5984,c1(CC(=O)OCC)c[nH]c2ccc(-c3cc(C)c(OC)c(OC)c3C)cc12 5985,C(=O)(C1=NN(C(C)C)C(=O)CC1)NCCCC(C)NC(C=C(COC)C)=O 5986,C(=O)(C1CCCn2nccc21)N1CC2N(C(c3cc(C)cc(Cl)c3)=O)C(CC2)C1 5987,C(N=c1[nH]c(N(C)CCC2CCC2)nc2ccc(Br)cc12)c1n(CC)cnc1 5988,Cc1cc(CNC(C2CC(C)N2C(=O)CCC2(C)CC2)=O)ccc1F 5989,CC(C)CC(C(=O)O)NC(C1CCCN(C(c2ccnn2C)=O)C1)=O 5990,c1(CNC(C=CC(=O)OCC)=O)nc(CNC(C2CC2Cl)=O)cc(O)n1 5991,c1(C(C(=O)NC)N(C)Cc2cc(C)c(C)c(Br)c2)cc2c(nc1O)CCC2 5992,c1(C(=O)NC2C(CNC(C(C)SC)=O)C2)ccc(-n2cccc2)nc1 5993,N1(C(C(COC)OC)=O)C2CCC1CC(NC(c1ccccc1SC(C)C)=O)C2 5994,C1(NC(C(CSC)C)=O)COCCN(C(=O)C(c2ccc(F)c(F)c2)(C)C)C1 5995,CCC(O)C(C)(C)C(=O)NCC1CC1NC(=O)COc1ccc(C(C)C)cc1 5996,c1(C(N2CCCOCC2)C(=O)NCCCC(=O)OCC)nc(C)c(Br)s1 5997,C1(CC(=O)NCc2cn[nH]c2)CCN(C(C2CCO2)=O)CC1 5998,N1(C(CCSCCC)=O)CC(NC(c2c(C)csc2Cl)=O)CC1(C)CC 5999,C1(=O)CCCC(=O)O1.N1(C(c2c(C)ccs2)C(=O)NC2CC2)CCC2CCCC12 6000,C1(C(=O)NCCCCNC(=O)C=Cc2cccnc2)CCC(=O)N2CCCC12 6001,N1(C(C2CC23CCC3)=O)CC2CCC(C1)N2C(=O)C(O)CC1CCCCC1 6002,CCC(C)(O)CNC(=O)CCCN(C(=O)CCOCCOC(C)=O)C 6003,Cc1nc(C(N2CC3CC2CN3C(C2CCN2S(C)(=O)=O)=O)=O)c2ccccn12 6004,C1(C)(C(=O)NC2CC(NC(CCCSC)=O)CC2O)CC=C(C)CC1 6005,c1(N(CCCCCOC)C)cccc(S(=O)(=O)N2CCSC(C)C2C)n1 6006,CCCCC(CN=c1nnn(C)[nH]1)NC(=O)CCCC(N)=O 6007,C(CCCCC(=O)NCC1(O)CCCN(C(=O)CC2CC(F)C2)C1)OCC 6008,C1(NC(c2c(C)n(C(C)C)cc2)=O)CCCN(C(=O)Cc2cc[nH]n2)CC1 6009,c1(C(=O)NC(C(=O)NC(C=C)CO)c2ccco2)cnccn1 6010,S(=O)(=O)(c1c(F)cc(F)cc1F)NCc1scc(C(=O)Nc2cccc(Br)n2)n1 6011,CCCCC(C(=O)NCC1OCCC1(C)C)NC(c1cc(C2CC2)[nH]n1)=O 6012,n1(C(C(=O)OCCOc2cccc(C(=O)OC)c2Cl)CCO)c(C)cc(C)nc1=O 6013,c1(C(=O)NC2CN(C(CS(C)(=O)=O)=O)CC2(F)F)cn2ccc(Br)cc2n1 6014,C1(O)(CNC(CCSCC(N)=O)=O)CCN(C(c2n[nH]c(C3CC3)c2Cl)=O)C1 6015,C=CCC(CC)C(=O)N1CCN(C(=O)CNC(=O)COC)CC1CCO 6016,C1(c2nc(CC(C)C)nn2CC(N)=O)CC(O)C(O)CO1 6017,N1(CC(C)C)CCC(C(N2CCCC(C(C)NC(C3(CO)CC3)=O)C2)=O)CC1 6018,Cc1cc(C(N2CC(C)(NC(C3CCC4(CCC4)O3)=O)C2)=O)c2scnc2c1C 6019,N1(C(C2CC(O)CN2c2ncnc3cc[nH]c23)=O)Cc2cccc(F)c2C1 6020,Cc1nc(C(=O)NCCC2CCCN2C(=O)CO)ccc1Br 6021,c1(N2CCC(C(C)(C)NC(C3C(C(=O)OC)C3)=O)CC2)ncc2ccccc2n1 6022,c1(C(N2CCCC2CNC(C2CC(F)(CO)C2)=O)=O)coc2ccccc12 6023,C1(C(=O)NCC2=CCN(C(CN3CC(=O)NC3=O)=O)CC2)CCn2ncnc2C1 6024,N1(C(CC2(C=C)CC2)=O)CCCC2(NC(C3CCC(C(N)=O)CC3)=O)CC2C1 6025,c1(C(N(CC(C)NC(=O)CC2CCNC2=O)C)=O)cc2sccc2[nH]1 6026,C1(C(=O)NC2CC(NC(=O)CCC3CCCCC3)C2)CCCN(C(=O)C2CC2)C1 6027,c1(CC(=O)NC2C(NC(C(C(C)C)NC(N)=O)=O)COC2)nn(C)cc1[N+](=O)[O-] 6028,CCCCC(CNC(=O)CC(O)Cc1ccccc1)NC(=O)CC1CCC(C)C1 6029,C(N=c1nc(N2CCC(F)(c3ccccc3Cl)C2)c2[nH]ccc2[nH]1)C1(C#N)CC1 6030,c1(C(C(=O)N2CC(SC(F)F)C2)NC(CCNC(=O)OCC)=O)c(C)cccc1Br 6031,N1(C(C(CC)F)=O)CCCC2(CCCCC2NC(=O)C(N2C(C)CCC2C)C)C1 6032,Nc1c(F)c(F)cc(C(N2CCN(C(=O)CSC(F)F)C3COCC23)=O)c1Cl 6033,CC(CCC(=O)Nc1cncnc1C(C)C)NC(c1nnc(S)n1C)=O 6034,c1(OCC)ccc(C)nc1C(=O)NC(C)CCNC(c1cc([N+](=O)[O-])c[nH]1)=O 6035,c1(C(=O)NC(CC(C)NC(C=NOC)=O)C)cc2ccc(F)cc2s1 6036,Cc1cc(F)c(C(=O)NC2CC(CCNC(C3CCOC3C)=O)C2)cc1F 6037,C1(C2CC2)(C(=O)NCCCCNC(=O)C=CCN2CCOCC2)CCC1 6038,C(=O)(C1SCCc2sccc21)N1CCC2(CC(NC(=O)CC=C(Cl)Cl)C2)C1 6039,c1(C(=O)NC2C(NC(=O)OC(C)(C)C)CCC2)ncc(Br)cc1O 6040,C1(C(=O)NC2CC(CNC(c3ccc4nncn4c3)=O)C2)CCc2nnnn2C1 6041,O=C(C(F)C1=CCCCC1)NCC1CCCN1C(C1CC2(CCCC2)CO1)=O 6042,c1(NC2(C(C)NC(=O)CCCc3cnn[nH]3)CC2)ncc(Cl)c(C)c1C#N 6043,c1(OC)nccc(C(=O)NCCC2CCCN2C(c2cc(Cl)ns2)=O)c1F 6044,Cc1nc(C(C)C)ncc1C(N1CCC(NC(C2CCCC(F)C2)=O)C(C)C1)=O 6045,c1(C(N2CCC(C#N)(NC(C(C(C)C)=O)=O)C2)=O)cnc2ccccn12 6046,C(=O)(C1=CC2(CCOCC2)C1)NCC1CC(C)N(C(=O)C(=C2CCCCC2)F)C1 6047,S(=O)(=O)(c1cccnc1N(C1(C)CC1)C)NCC 6048,C1(C)(CNC(C(c2ccnn2C)NC(Cc2cnc(C)s2)=O)=O)CCN(C)C1 6049,C1(C(N2CC(NC(c3nc(C(C)=O)sc3)=O)C2)=O)CCN(CCO)C(=O)C1 6050,C=CCCCCCCCC(=O)N1CCC2(CC1)CC2NC(=O)CC(CC)CC 6051,N1(C(c2n(C)nc(Cl)c2)=O)C2CCC1CC(CNC(=O)C=CCF)C2 6052,c1(C(=O)NC(C(C)NC(Cc2c(C)n[nH]c2C)=O)(C)C)cnn2c1OCC(C)C2 6053,c1(N(CCC)C)cccc(S(=O)(=O)NC(=O)C(C)OCCOCCNC(C)=O)c1 6054,N1(C(C(c2cn(C)nc2)=O)=O)CCC(C(=O)NC2CC=CC2)C1C(C)(C)C 6055,C(=O)(C(CC(F)F)NC(=O)Cc1cn[nH]c1)N1CCN(C(C)(C)C)CC1 6056,C1(CNC(COC)=O)CC2CC1CN2C(c1ccc(-c2ccsc2)nc1)=O 6057,Cc1nn(CC(N2CC(NC(c3ncc(F)cn3)=O)C(C)C2)=O)cc1Br 6058,C1(NC(C(n2ncc(C)c2)C)=O)CCCCC1NC(=O)C=Cc1ccoc1 6059,C(=O)(C(F)(CNC(c1cccc(=O)o1)=O)C(C)C)NC1(C(=O)OCC)CC1 6060,N1(C(C=C(CC)C)=O)CCN(C(=O)COC2CC(F)(F)C2)CC1CC 6061,N1(c2cc(N(C)CC3CCN(C)C3)ncn2)CCOC(C)(c2ccccc2)C1 6062,C(=O)(C(C)(C)C(=O)Nc1ccc(F)c(F)c1)NC1CC(C)N(C(=O)CC(F)F)C1 6063,c1(C(CC)C)ccc(C(=O)NC2CCC2CNC(C2(O)CC2)=O)c(O)n1 6064,c1(NCC2(NC(=O)OC(C)(C)C)CC2)n[nH]c(=N)[nH]1 6065,C1(C2CC2)(NC(CC(CNC(C2N(CC)CC2)=O)C)=O)CCCC1 6066,c1(NC(c2ccc(OC=C(F)F)cc2)=O)cccc(-c2nc(O)n[nH]2)c1 6067,c1(COC)cc(N(CC(C)CNC(C2CCCOCC2)=O)C)nc(SC)n1 6068,CCCCC(CN1CCCC(C(N2CCCC(CO)C2)=O)CC1)CC 6069,C=CC(CC)C(=O)N1CC(=O)CC1C(=O)NC(c1cnccc1C)C 6070,N1(C(C(CC2CCC2)NC(C2CN(C3CCC3)C2)=O)=O)CC2(CCC2)C1 6071,N1(C(c2c(C)snc2)=O)CCC2(CCCN2C(c2cc(N(C)C)ccc2N)=O)CC1 6072,C1(NC(CCC(C)OC)=O)CC2CCC(C1C)N2C(=O)C1=CCCCO1 6073,C1(C(=O)NCCCN(C(C2CS(=O)(=O)C2)=O)CC)CCC1(F)F 6074,CC1=CCSC1C(=O)NC(C1CCN(C(=O)CCC2CC(F)(F)C2)C1)C 6075,C1(OC)(CNC(c2nc(Cl)oc2C)=O)CCN(C(c2cnc(C(N)=O)s2)=O)C1 6076,C1(NC(C(=O)N(C)Cc2cn(-c3nccs3)nn2)=O)CS(=O)(=O)C12CCOCC2 6077,N(C1c2ccccc2CC1NC(C12CCC(CC1)CC2)=O)C(C(C)C1CCC1)=O 6078,CCCC(CC)C(=O)NCCC1(NC(=O)C2=NNC(=O)C2)CCCC1 6079,C1(NC(C(CC)CO)=O)CC2CN(C(=O)C(c3ccccc3F)(F)F)CC2C1 6080,N1(C(C=CC(C)NC(C2CC(C(C)=O)C2)=O)=O)CCOC2COCC12 6081,C1(NC(C(CC=C)C)=O)CC(OC)CN(C(c2cc(C)n(CC)n2)=O)C1 6082,C=CCCC(C(=O)N1CC(OC)CC(F)C1)NC(=O)C(C(C)(C)C)N(C)C 6083,C1(NC(c2c(OC)csc2)=O)CC2CN(C(c3ccc(CO)s3)=O)CC2C1 6084,N1(C(COCC=C)=O)CCC(NC(=O)COc2cccc(C)c2)C12CCC2 6085,CC1(C)C2CN(C(C3CCC(NCc4ccc(I)c(O)c4)CC3)=O)CC12 6086,C1(CNC(Cc2c(C)con2)=O)(CNC(c2cc(C)n(CC)n2)=O)CC12CCC2 6087,S(=O)(=O)(CC(=O)OC(C)(C)C)NC(=O)NCC1(CCF)CCN(CCOC)C1 6088,C1(CNC(=O)CCC2CCCCCC2)C2CCCC1N(c1cc(Cl)c(O)nn1)C2 6089,C1(C(N(CCCC)CCOC)=O)CCC2(CN(C(c3cnccn3)=O)C2)O1 6090,N1(C(c2onc(CC)n2)=O)CC=CC(NC(=O)CC(c2cccc(F)c2)C)C1 6091,Cc1ccnc(C(N2CC(C(N)=O)(CNC(=O)CN3CCCCCC3)C2)=O)c1N 6092,Cc1cncc(C)c1-c1noc(-c2ccc(OCC(F)(F)F)cn2)n1 6093,C(CCCCCN(C(=O)CCn1ncn(C)c1=O)C)NC(C1(CC)CC1(F)F)=O 6094,C(=O)(CCN1C(=O)CSc2ccccc21)N1C(C)CCCC1C 6095,n1(CCC(=O)NCC(CC)(CC)NC(C2CCO2)=O)c(C)c(C)sc1=O 6096,N1(C(C2CC(OC)C2)=O)CCOC2CN(C(c3nccc(Cl)c3O)=O)CC12 6097,N1(C(C(C)n2cccc2)=O)CCC2(CC2)CC1C(=O)NCCN1CC=CC1 6098,O(NC(=O)C(O)C1CN(C(c2ccc(=N)[nH]n2)=O)C1)CC1CC(=C)C1 6099,C(=O)(N=c1[nH]n(-c2ncccn2)cc1I)c1ccc(-c2n(C)cnc2)cc1 6100,C#CCC(C(=O)NN1CCN(C(=O)OC(C)(C)C)CC1)NCCSC(F)F 6101,n1(CCC)c(=O)nc(O)c2cc(C(=O)NCCc3cn(CC)nn3)cnc12 6102,N1(C(C(CC)NC(=O)C(=O)NCC2CC2)=O)CCOC(C)(C)C1C 6103,Cc1sc(-c2nc[nH]n2)nc1C(N1CC(O)(CCNC(C2(F)CC2)=O)C1)=O 6104,N1(C(c2coc(C3CC3)n2)=O)CC2CN(Cc3ccnc(Br)c3)CC2C1 6105,c1(OC)ncc(Cl)cc1C(=O)NC1CN(C(C2CC(=C3CC3)C2)=O)CCC1C 6106,C=CC(C)(CCOC)C(=O)NCC1COCCN(C(c2ccc(CC)s2)=O)C1 6107,c1(C(c2nnnn2C)NCCc2c(C)noc2C)ccc2c(c1)OC(C)(C)O2 6108,C1(C)(C(N(C)CC2CCN(C(C3(C)CCCO3)=O)C2)=O)CCCNC1=O 6109,n1(CC)ncc2c(C(=O)OC(C3CCCCC3)C(=O)OC)cc(C)nc12 6110,c1(CNC(N2C(C(=O)NC3(OC)CCOC3)CCC2)=O)cnc(C)cn1 6111,C=CC(C)(C)CC(=O)NC1CC(C)N(C(=O)C(O)Cc2cnc[nH]2)C1 6112,Cc1cc(OCc2ncc3c(C)cccn23)n2ncc(C(F)(F)F)c2n1 6113,Cc1cc(NC(=O)C(=O)NC2CCCC23CNC3)cc(Br)n1 6114,c1(C(=O)NCC#CCNC(c2cc(OC(C)C)ncc2)=O)cc(F)c(N)cc1F 6115,Cc1nccc(NCC2CCCN(C(=O)CCc3ccc(C(C)(C)C)cc3)C2)n1 6116,C12(CNC(=O)Cc3cc[nH]n3)CC1CN(C(=O)Cc1cc(Cl)sc1Cl)C2 6117,C1(NC(C=CC=CC)=O)CC2CC1CN(C(=O)C(C(C)C)n1cncn1)C2 6118,c1(N2CCN(C(C3CCCS3(=O)=O)=O)CC2)ncnc2ccc(O)cc12 6119,C(CC(C(=O)N1CCC1C1CCCC1)NC(=O)CCc1ccsc1)=CC 6120,CC1CCCC=C1C(=O)N1CCCC(F)(C(=O)NC(c2cncn2C)CO)C1 6121,CCCCCS(=O)(=O)CC(=O)NCC1(C)CCCN(C(=O)CC(=O)N(C)C)C1 6122,C1(NC(c2cc(OC(C)C)no2)=O)CCN(C(c2ccc(Cl)cc2)C)C(C)C1 6123,c1(C(C)C(=O)OCC2CCCC(F)C2)ccc(Cl)c(Cl)c1 6124,N1(C(C2C(CC)CN(C(=O)C(C)(C)CO)C2)=O)CC2CC(CO)C(C2)C1 6125,C1(C)(C(=O)NCCCNC(C(C)=C2CCC2)=O)CC2CCC(C1)S2 6126,N1(C(C(C)c2cccs2)=O)CC2(CO)CC1(C(N1CCCC(CC3CC3)C1)=O)C2 6127,C1(CNC(CCCNC(C)=O)=O)CN(C(C23CCC(CC2)C3)=O)C2CCN1C2 6128,CC1(CNC(=O)OC2(C(C)(C)C)CC2)CC12CCN(Cc1ccco1)CC2.C 6129,C1(CC(=O)NCCC(F)(F)CO)CCCC(NC(c2cscc2Cl)=O)C1 6130,C1(NC(C(COC)(C)C)=O)CC2CC(NC(=O)Cn3ncccc3=O)C2C1 6131,C1(CNC(C(CC(C)C)F)=O)CN(C(c2cc3scnc3[nH]2)=O)CCC1(F)F 6132,N1(C(=O)CCOc2ccccc2Br)CCCC2(CCN2)C1 6133,N1(C(c2ccc(NS(NC)(=O)=O)s2)=O)CCN(CCNC(=O)CNC(N)=O)CC1 6134,CN1CC=C(CC(=O)NC2CCC2NC(c2cc(Cl)c(Br)[nH]2)=O)CC1 6135,C1(OC)CN(C(=O)C=CCO)CCC1NC(=O)C(C)(C)c1ccncc1 6136,CC(C)(C(=O)NC(CNC(=O)CCCC1CC1)CC(F)(F)F)C1=CCSCC1 6137,N1(C(CS(CC)(=O)=O)=O)CC2CCCC(NC(=O)CSCCC#N)C2C1 6138,CCC(O)C(C)(C)C(=O)N(C)CCN(C)C(c1cccc(OC)c1O)=O 6139,C1(CNC(CCCCC)=O)CCN(C(c2nocc2Br)=O)CCC1(F)F 6140,CC(C(=O)NCc1noc(C(C)C)n1)(C1CCC1)NC(=O)CCc1cnn[nH]1 6141,C#Cc1cncc(CN2CCCC(N3CC(C)(C)OC3=O)CC2)c1 6142,CN1C(=O)CCCC1Cn1cc(-c2cc(Cl)ncc2N)nn1 6143,Cc1cc(C(N2C(C(=O)NCc3cocn3)CC2C)=O)c(C)n1C 6144,C1(CNC(C23CC(NC(C4CC(C)OC4)=O)(C2)C3)=O)COCC1(C)C 6145,C(C1C(C(=O)NC2CC3CN(C(=O)Cc4ccncc4Cl)CC23)C1(C)C)=C(C)C 6146,C1(NC(c2c(CCC)n[nH]c2)=O)CN(C(=O)CC#N)CCC12CCC2 6147,n1(CC(=O)NC2CC(C)(NC(CC=C=C)=O)C2)nc(C)c([N+](=O)[O-])c1C 6148,Cc1cnc(F)cc1CNCCC1CCC(C(F)(F)F)O1 6149,C(CCCCCC(=O)O)N1CC(CC)OC(C)C1.c1ccc(-c2nn[nH]n2)cc1 6150,Cc1ccc(C(=O)NCC(O)CNC(=O)C2=C(Cl)CCOC2)c2cccnc12 6151,c1(C(C)Nc2nc(C(=O)N(C(C)CC(=O)NC3CC3)C)co2)ccc(F)cn1 6152,C(=O)(CC(CC)CCCCC)NCC(CCC)NC(=O)C=CC(C)C 6153,N1(C(COCCC(C)C)=O)CC2CCN(C(c3cn(C)c(O)n3)=O)C(C2)C1 6154,c1(C(N2CC3C(CNC(C(N)=O)=O)(CC3)C2)=O)c[nH]ccc1=NC(=O)C(F)(F)F 6155,C#Cc1cc(C(N2CCC2CNC(c2sc(Br)c(C)c2C)=O)=O)cc(F)c1 6156,CCCCCCNC(C1CCCC1CNC(C1CNC(=O)C1)=O)=O 6157,CCCCC(O)C(C)C(=O)NCC(CC(C)C)C(=O)NCCC(C)C(F)F 6158,c1(CCNC(=O)C(N2CCC(N3CCCNC3=O)CC2)=O)ccc2c(c1)CCOC2 6159,C(=O)(CC(F)(F)C(F)(F)F)NCCOCCN.C(CCS(=O)(=O)NCCSC)OC 6160,c1(NC(=O)NCCCNC2CNC(CO)C2)ccccn1 6161,c1(CCC(=O)N(C)CC2CCN(C(CC(=O)OC)=O)C2)cc(C)cc(C)c1 6162,C(=O)(C(O)CCC(C)C)NC12CCC(NC(c3cnc(C)[nH]3)=O)(CC1)C2 6163,N1(C(c2c(SC)snn2)=O)CCC(C)N(C(=O)C=Cc2ccsc2)CC1 6164,c1(OC)c(C)csc1C(N1CCC(CCNC(=O)CC(C)n2cccc2)C1)=O 6165,C(C(C)(O)CC(=O)N1CC2(C)CCC2(C)C1)NC(C(CCC1CC1)OC)=O 6166,C12(NC(c3cnc(CC)o3)=O)CCCN(C(c3cccc(C#N)c3C)=O)CC1C2 6167,n1(C(CC)C)nnnc1C1(NCCc2cnco2)CC(c2nc(C)no2)C1 6168,N1(C(c2ccc(CNC(C3CN(C4CCC4)C3)=O)nc2)=O)CCC2CCCCC2C1 6169,CC(C)CC(CN(C)C)CC(=O)N1CCCC1CCN(C)C 6170,Cc1c(C(=O)N(C2CC2)CC2CCOC2)sc2cc(F)ccc12 6171,N1(C(C2C(=C)C2)=O)Cc2n[nH]cc2C1C(=O)NCCC1CCC1 6172,Cc1cc(C)n(C2CCCN(C(c3nnc(CCO)s3)C(=O)NCC(C)C)C2)n1 6173,CCCCCCC(=O)NC(c1nc(C(=O)NC(CC)CC(F)(F)F)co1)C 6174,Cn1ccnc1CC(=O)NCC(C)(C)n1ccnc1.C12(CC1)CC(=O)NC2 6175,c1(NC(CNC(Cc2ccc(C)nc2)=O)C)ncc([N+](=O)[O-])cc1C#N 6176,c1(CN2CC(CC)N(C(C3CCCCN3C(C)=O)=O)CC2)coc2ccccc12 6177,C1(C(N2CC3(CCC3NC(C3C=CCC3)=O)C2)=O)(CC)CCC(F)(F)CC1 6178,Cc1noc(C)c1C(N1CC2(NC(C3CCC3C)=O)CC1C2)=O 6179,N1(CC(N2CCC(CCNC(c3cc(C)on3)=O)C2)=O)CCC(F)(F)C1 6180,Cc1ccc(C(=O)N(CCN(C)C(c2coc(Cl)n2)=O)C(C)C)nc1 6181,Cc1cccc(F)c1CC(=O)NC1CC(N(C)C(c2c(C)ncn2C)=O)C1 6182,Cc1noc2ncnc(NC(C3CCCN(C(=O)CCn4cnnn4)C3)C)c12 6183,C1(C(=O)NCCOCCOCCO)CC2(CC(NC(=O)CCC(N)=O)C2)C1 6184,c1(C(=O)OC)cc(C(=O)NC(C)(C)CCCNC(=O)C=C2CCC2)ccc1F 6185,C1(C)(CNC(c2c(C)ncs2)=O)CCCN(C(=O)Cc2csc(NC=O)n2)C1 6186,Cc1cncc2nc(CC(=O)NCCCN(C(=O)CC(O)C(C)C)CCO)cn12 6187,N1(C(c2snc(C)c2N)=O)CCCN(CCNC(C2CN(C)C2)=O)CC1 6188,O=C1CCC(C(=O)N2CCC(NC(c3cc(C(F)F)cc(Cl)c3)=O)C2)=NN1 6189,C1(NC(=O)C=CCO)COC2(CNC(CNC(CN(C)C)=O)=O)CC1C2 6190,N1(C(C(F)=C(C)C)=O)CCC2CN(C(c3cc(Br)n(C)n3)=O)CC2C1 6191,C1(NC(c2cc3occc3[nH]2)=O)CCCCN(C(C2CC3(C2)CC3F)=O)C1 6192,N1(C(c2c(N)cccn2)=O)CCC2(CCOC2)C(CNC(=O)Cc2csnn2)C1 6193,N1(C(C(CCCOC)C)=O)CCC2(CCCN2C(=O)C(C(C)C)c2cccnc2)C1 6194,C1(C(N2CC(CNC(C(C)C)=O)C2)=O)(N(C)C)CCCCC1 6195,C(=O)(C(CC(C)(C)C)NC(=O)C(C1(O)CCCC1)F)N1CC(CC(C)C)C1 6196,C(CCCCNC(=O)COCC(C)(C)C)N(C(CCC1CC(C)C1)=O)C 6197,c1(C(=O)NCCN(C(=O)C(n2ccc(C3CC3)n2)C)CC)ccc(C)c(C)c1N 6198,c1(CNC(c2c(C(C)(C)NC(=O)C=CCO)noc2)=O)ccccc1F 6199,C1(C(=O)NOCCCOCCO)CC(O)CN1C(=O)Cn1ncccc1=O 6200,N1(C(CCN(C(CCn2ccc(C)n2)=O)C(C2CC2)=O)=O)CCC(C(C)C)(CO)C1 6201,C=CCCC(=O)NC(CNC(C1CN(C2CCOC2)C1)=O)C1CCC1 6202,CCCCCCC(C)C(=O)NC1CN(C(c2c[nH]c(=NC)s2)=O)CC1O 6203,C(=O)(C#CC1CCCO1)NCC1(CN(C(c2c(C)nn(C(C)C)c2C)=O)C)CC1 6204,c1(C(N2CC(OCCOC)C(O)C2)=O)cc(C)ccc1Br 6205,C1(C(N(C2CCN(C)C2)C)=O)CCCC(NC(c2cnn(C3CC3)c2)=O)CC1 6206,c1(C(=O)NC(C(C)C)C(=O)N(C2CCCCC2)CC)cc2c(O)cc(Cl)cc2[nH]1 6207,C(=O)(C(CO)C(C)C)NC(c1c(-n2c(C)cc(C)n2)cncc1)c1ccccc1 6208,C(CC(C(C)C)NC(c1cscc1C(=O)OC)=O)N(C(C=C(CCC)C)=O)C 6209,N1(C(c2cc(SCc3cccc(OC(C)(C)C)c3)sc2)=O)CCCC2(CCC2)C1 6210,c1(C(=O)NC2CC3CC(NC(C(C)SCCCC)=O)C3C2)cc2nccnc2[nH]1 6211,C1(C(=O)N(CC(C)C(=O)NC)C)(CNC(CC2CC(=C)C2)=O)CCCC1 6212,N1(C(C2(CSC)CC2)=O)CC(C)CN(C(=O)Cc2nsc3ccccc23)C(C)C1 6213,c1(CCC(=O)NC2(CN(C)C(C3CC(N(C)C)C3)=O)CC2)cccnc1 6214,C1(NC(c2nc(CC)oc2)=O)CC12CCN(C(=O)Cc1ccoc1C)CC2 6215,N1(C(C(CCN(C)C)NC(CC2C(C)C(=O)CC2)=O)=O)CC2CSCC2C1 6216,c1(NC(CN(C(=O)CSCC(N)=O)CCC)=O)ccc(CC)o1 6217,N1(C(CN(CC)CC)=O)CCN(C(=O)CCc2cccc(C)c2)CC1C1CC1 6218,C(=O)(C1=CCCCC1P(C)(C)=O)N(CC(C)CNC(=O)CCC#N)C 6219,CCCCCC(C)(CC)C(=O)NC(C)CN(CCC)C(=O)C=C(C)C(C)C 6220,N1(C(CCC(C)OC)=O)CCC(C)C(CNC(c2cccc(F)n2)=O)C1 6221,S(=O)(=O)(c1cnc(NCc2csc(C(C)(C)C)n2)cc1C)NC(COC)CCO 6222,C(CC(=O)N(C1CC1)Cc1ccccc1)(C(F)(F)F)NC(C(C)n1ccnc1)=O 6223,CCC(C)(COC)C(=O)N1CCC1CNC(=O)C(C)(C)C(F)F 6224,C1(C(=O)NCC(C)(CO)NC(Cc2c(Cl)cn(C)n2)=O)CCCCC(F)(F)C1 6225,C(=O)(C(O)CC1CCCCC1)N(CCN(C(=O)CCN(C)CCO)C(C)C)C 6226,Cn1nncc1C(=O)NCC1(NC(=O)CCN2CCCC2=O)CCOC1 6227,c1(C(=O)NCCN(CCC)C2CC2)cc(Cl)ncc1F 6228,c1(C(=O)NCC(CC(C)C)NC(c2ccc(=O)n(C)n2)=O)cc2ccsc2s1 6229,N1(CC)CC(C(=O)NC2CC3(C2)CC3Nc2cc(C(N)=O)ncn2)CCC1=O 6230,c1(C(=O)NC2C(NC(CC(CC)CC)=O)CC2)cnc2ccoc2c1 6231,C=CCCCCC(=O)N(C(CC(F)F)C(=O)NCCC(O)CC)C 6232,N1(C(c2c(OC)cccc2)=O)CCCC2C1CCN2C(c1c[nH]c(=N)nc1C)=O 6233,c1(C(=O)NCC(CNC(c2ccn(C)n2)=O)(C)O)cccc2oncc12 6234,CC(CCF)N=c1nc(N(C)CP(C)(C)=O)c2cc(N(CCO)CCO)ccc2[nH]1 6235,C=C(C)CN=C(NCC(C)CCCCO)N(C)Cc1ccc(F)c(Cl)c1 6236,Cc1cc(OC2CCOC2)ccc1F.C12CN(CC1C)C(=O)CONC(=O)C2 6237,c1(C(=O)OC)c(C)[nH]c(C(N2CCC(F)C(NC(=O)C(=O)NC(C)C)C2)=O)c1C 6238,N1(C(CC=CC)=O)CCCC1C(C)(C)C(=O)NCCCC(=O)NC 6239,O=S(=O)(c1c(Cl)ccc(Br)c1Cl)Nc1cc(CO)cc(Br)c1 6240,c1(C(=O)NC(C)C(C)NC(c2ncccn2)=O)ccc(N2CCCC2=O)cc1 6241,CCC(CC)C(C)C(=O)N1CCC(CC(C)NC(c2nc(C)ncc2Cl)=O)CC1 6242,C1(C(N2CCC(NC(C3CC(F)(F)C34CCC4)=O)C2)=O)Cc2ccccc2C1 6243,Cc1ccnc(C=CCNC(C2CCN(CC3CN(C)C3)C2)=O)c1 6244,N1(C(C2C(C)C2C)=O)CCCC(C2CCN(C(C3(O)CCCCC3)=O)C2)C1 6245,c1(C(=O)NCC2(F)CN(C(C3CC4CC3CO4)=O)C2)ccc(Cl)cc1C(F)F 6246,N1(C(C(C)CN(C)C(C2(CO)CCC2)=O)=O)CCS(=O)C(C)C1 6247,C(=O)(CC=C(Cl)Cl)NCCC(C)NC(c1ccccc1OCCF)=O 6248,C(C(N=c1cc(Cl)nc(S(C)(=O)=O)[nH]1)C1CCC1)NC(C1=C(C)OCC1)=O 6249,N1(C(CC)=O)CCCC(C2CCCN(C(c3cc(OC(C)C)ccn3)=O)C2)C1 6250,N1(C(C(C)CN(C)C)=O)CC2CCC1C(CNC(C1(C3CC3)CCCO1)=O)C2 6251,c1(C(N2CCC(n3cccn3)C2)C(=O)NC(CC)C)cc2ccc(OC)cc2o1 6252,C(=O)(C(C(F)(F)F)C(F)(F)F)N1CC2(OCC(NC(C(C)(C)CCF)=O)C2)C1 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6271,C1(NC(c2cc(C(C)(C)C)no2)=O)CCN(C(C2C3COCC23)=O)C1(C)C 6272,C1(C(N(CC(CC)NC(=O)COCCOCCO)C)=O)CCCCN(C)C1 6273,C1(NC(C=CC=CCC)=O)CC2CC(NC(=O)CC(c3ccccc3F)C)CC12 6274,c1(OCC(N2CC(CNC(C3CCCN(C(N)=O)C3)=O)C2)=O)ccc(Cl)cc1Cl 6275,c1(C(N2CCC(CC(=O)NCCc3ccco3)C2)=O)ccc(F)c(F)c1 6276,CCC(CC)(CC(=O)OC)C(=O)NCC1CCCN(C(=O)CCC2CC2C)CC1 6277,c1(C(=O)NCC2CCCN2C(c2ccc(CO)cn2)=O)cn2cccc(Br)c2n1 6278,c1(CCC(=O)NC(C)(CC2C(c3n(C)ncc3)C2)CO)nnc(S)nc1O 6279,CC1(NC(=O)CCc2ccc(F)cc2)CCN(C(=O)C(F)C2CC2)CC1 6280,c1(C(N2CCN(C(C3(CO)CCCO3)=O)CC2)=O)ncc(F)cc1F 6281,Cc1cc(Cl)c(C(=O)NC2CCC(CNC(C3CNC(=O)N3C)=O)C2)cc1N 6282,C(=O)(C(C)C(=O)N1CCC(C)(CNC(=O)C(F)(F)Sc2cnn(C)c2)C1)OC 6283,N1(C(CC(C)c2ccncc2)=O)CCC2(CC1)CC2CNC(=O)Cn1ccnn1 6284,C1(CC)(NC(c2ccnnc2)=O)CCCN(C(c2cc(C3CC3)n(C)n2)=O)C1 6285,N1(C(C2CC(CNC(CCc3n(C)ncn3)=O)C2)=O)CCC(CCO)CC1 6286,CC(F)(F)CCC(=O)NC1CC2(C1)CC2C(=O)NC(C(=O)OC(C)(C)C)C1CC1 6287,C1(CC(=O)NCC2N(C(C(N=S(C)(C)=O)=O)=O)CC=C2)C2CC3CC(C2)CC1C3 6288,C(=O)(CCS(C)(=O)=O)NCC1C(CC(=O)NCCC=C=C)C1 6289,N1(C(C(C)=C2CCC2)=O)CCN(C(=O)C(=O)NC2CC2)CC1c1ccccc1Cl 6290,c1(CO)cccc(Br)c1.c1(C(N2CC(CC)NC2=O)=O)cnn(C(F)(F)F)c1 6291,C(C1=NOC2(CCC2)C1)N(C(C=C1CCN(C)C1)=O)C1CC1 6292,Cc1cccc(OCC(=O)NCC(O)CCNC(=O)CN2CCCNC2=O)c1F 6293,C1(CC)(NC(=O)C=CC2CCCO2)CCN(C(c2cn(C)nc2OC)=O)CC1 6294,N1(C(C(C)C)=O)CCC2(CC1)CC2CNC(C1CCn2cncc2C1)=O 6295,C1(CC(=O)NCC(C2CC2)NC(C=C(CC)CC)=O)CCCOC1 6296,c1(C(=O)NC(c2ccc(C)cc2)C2C3CNCC23)cnc2n1CCS2 6297,C12(CCSCC1)CCNC(=N)NCCS2.C(c1cn(C)cn1)=CC(=O)OC 6298,N1(C(C(C)(C)C2CCC2)=O)CC2CC(C1)N(C(c1cc(S(N)(=O)=O)cs1)=O)C2 6299,Cc1cncc(C(=O)NCCC2(C)CCN(C(C3(Cl)CC3(F)F)=O)C2)n1 6300,C1(C(=O)NCCc2ccc(C)cc2)CN(C(c2ncnc(O)c2F)=O)C(C)(C)C1 6301,C(=O)(C(F)(F)c1ncccn1)NC(CNC(c1ccoc1)=O)C1CC1 6302,C1(NC(c2cnc(C(C)O)s2)=O)CN(C(=O)C(C)S(N)(=O)=O)CC(C)(C)C1 6303,CC1CCN(C(=O)CC2CCC(=O)N2)C(CNC(C2CC(NS(C)(=O)=O)C2)=O)C1 6304,c1(C(=O)NCCCN(CCCNC(C(C=C)O)=O)C)cc(OC)cnn1 6305,C1(NC(c2cc(COC)on2)=O)CCCN(C(c2n[nH]c(C)c2F)=O)C1 6306,C(CCN(C(=O)COC1(C)CCC1)C)(C(C)C)NC(CC1(OC)CCCC1)=O 6307,N1(C(C(CCC)C)=O)CC2CCC1C1CN(C(C3CC(C(C)C)C3)=O)CC21 6308,Cc1ccc(C(N2CCC(CN(C)C(C3CC(=O)NC3(C)C)=O)C2)=O)cc1CO 6309,CCCCC(F)C(=O)NC1CCCCC1C(=O)NCc1cc(C)nn1C 6310,C1(OC)CC(F)CN(C(C2CCC(C)N2C(=O)Cn2cnccc2=O)=O)C1 6311,C1(NC(C(N2C(c3n(C)ccn3)CCC2)=O)=O)CCC(F)(F)CC1 6312,c1(NC2(CNC(C3C(C)CCCC3)=O)CCOCC2)cc(CCO)nc(CO)n1 6313,C(=O)(CC(C)(C)CC(F)F)N1C2CC(N(C)C(C3CC(O)C3)=O)CC1CC2 6314,C(C(C)(C)CC(=O)NCC(CNC(C1CC(=O)N(C)C1)=O)C(F)(F)F)OC(C)=O 6315,C1(CC=C)(NC(C2CCC(N(C)C)CC2)=O)CCN(C(=O)C(O)CC)C1 6316,Cc1c(C(N2CC(CNC(C3CCCC34CC4)=O)C2)=O)ccn1C 6317,c1(C(=O)NC2C(NC(c3c(COC)cc[nH]3)=O)CC2)ccc2c(c1)NC(=O)CS2 6318,N1(C(C(C)OC(C)=O)=O)CCC(C)(CC(=O)NCC(C)CC2CCC2)C1 6319,N1(C(C=CCC)=O)CC(O)C(O)C1CNC(=O)CCc1cccs1 6320,CC1(C)COc2cc(Br)ccc2C1NC(=O)NC1CCN(c2ccccc2Cl)C1=O 6321,c1(NCC2CN(C(Cn3c(C)cnc3)=O)C2)ncnc(N(C)C)c1[N+](=O)[O-] 6322,c1(OC(CC)=O)ccc(OC(C)C(=O)N(CCC)C(C2CCCC2)C)cc1 6323,N1(C(=O)Cn2cnc(Br)n2)CC(NC(C2CC(F)(CO)C2)=O)CC(O)C1 6324,C(=O)(C(C)(C)CCC#N)NC(C)CN(C)C(c1cn(-c2ncccn2)cn1)=O 6325,N1(C(C=CC(C)=O)=O)CCCC(CO)(NC(=O)C(C)Cc2ccc(F)cc2)C1 6326,CCCCCC(F)C(=O)NCC1CN(C(=O)COC2CCCCC2)CC12CCC2 6327,N1(C(C2N(CC)CC2)=O)CCN(C(C2CCN(C)CC2)=O)CC1CC(F)F 6328,C1(O)(CNC(Cc2cc(C)[nH]n2)=O)CCN(C(C2CC2c2ccccc2)=O)CC1 6329,C1(NC(C(CC(C)C)OC)=O)CC2CCC(C1)N2C(=O)C(C)C1CCCO1 6330,C1(CC(=O)OC)CCCN(C(c2cn(C3C=CCCC3)nn2)=O)C1 6331,c1(C(N(CCN(C(c2c(OC)n[nH]c2)=O)C)C(C)C)=O)cn2cc(C)ccc2n1 6332,c1(C(=O)NCC(C)NC(=O)CCc2ccccn2)cc(F)c(F)c(N)c1Cl 6333,N1(C(c2c(COC)noc2)=O)CC2(CCN(C(c3ccc(CN(C)C)[nH]3)=O)C2)C1 6334,N1(C(=O)Nc2ccc(OC(C)C)cn2)CC2(CC2)c2ccc(Br)cc21 6335,N1(C(=O)COC2CC3CCC2C3)CCC(F)(CN(C(=O)C(F)(F)C(F)F)CC)CC1 6336,c1(N2C3CC(CN(C(c4ccc(SCC)cc4)=O)C3)C2)nc2ccc(F)cc2o1 6337,C1(NC(=O)CN(C(=O)CCC2OCCO2)C2CCC2)CCC2CC12 6338,C1(NC(C(C2CCCCC2)OC)=O)CCNC(=O)CC1 6339,CN1CCc2cc(C(N3CCN(C(=O)C(O)C(C)(C)C)CC(C)(F)C3)=O)sc2C1 6340,c1(C(=O)NC2(CC=C)CN(c3ncns3)C2)cn(C2CC2)c(C)cc1=O 6341,Cc1ncnc(C)c1C(=O)NC1C(C(=O)NCCc2cnn[nH]2)C1(C)C 6342,c1(C(=O)NC2CN(Cc3ccc(OC)nc3)CC2O)ccc2cccc(Br)c2n1 6343,c1(C(N(CC(CN(C(CSCCCC)=O)C)O)C)=O)oc(C2CC2)nc1C 6344,CC1CCC=C1C(=O)NC1(C(=O)NC(CCO)C2CC2)CCSC1 6345,CC1CN(C(c2nccnc2C(N)=O)=O)CC1NC(C1C2CC(=O)CC12)=O 6346,c1(N(C(c2ccc(C(=O)OC)[nH]2)=O)C2CC2)ccc(NCc2ccco2)c(F)c1 6347,Cc1cc(C(N2CC(C(=O)Nc3cc(-c4ccccc4)nn3C)C2)=O)ccc1F 6348,Cc1cc(CCCNS(=O)(=O)Cc2ncsc2Br)no1 6349,N1(C(=O)C(c2cccc(C(F)(F)F)n2)(F)F)C2CCCC1CC(O)C2.O=C 6350,C1(C(C)CO)CCN(C(=O)CC2CNC(=O)O2)CC1.c12coc(c1)CC2=O 6351,C1(NC(C(COCC)C)=O)CC2(CCCN(C(=O)C(C)(Cl)Cl)C2)C1 6352,N1(C(c2n(CC)ccn2)=O)CC2N(C(C3CCC(C4CC4)CC3)=O)CCC2(C)C1 6353,CCCCC(O)CC(=O)NC(C)CCN(C)C(c1ccc(N(C)C)cc1C)=O 6354,C1(CC#C)(C(=O)NCC=CCCCNC(=O)COCC(F)F)CCOC1 6355,c1(C(N(C(C)C(C)C)CC)=O)cc(CNC(=O)C(SC)OC)no1 6356,c1(C(N2CCC(C)(CNC(C3C(C)CCCC3)=O)CC2)=O)ccccc1N=[N+]=[N-] 6357,N1(C(CCN(CC)CC)=O)CCC(F)C(NC(c2cn(C)nc2OC(C)C)=O)C1 6358,C=CC(O)(C(=O)NC1CC2CCC1N(C(=O)CCn1cncn1)C2)C(F)(F)F 6359,N1(C(C2(CC=C)CN(C(c3cnc(C)cc3C)=O)C2)=O)CCC2CCCC2CC1 6360,N1(C(C=COCC)=O)CCCC(C)(CNC(c2ccc(Br)nc2N)=O)C1 6361,c1(CNCc2ncc(-c3cccc(Cl)c3)cn2)ccc2cnccc2c1 6362,CC(CCCCNC(=O)CN1CC=CC1)NC(=O)CCN(C)CCO 6363,C1(OC)(CNC(C2C=CCC2)=O)CCN(C(C2COCC(C)(C)O2)=O)CC1 6364,C(=O)(CCC(C)(C)[N+](=O)[O-])NC1CCN(C(C(C)(C)SC)=O)CC1F 6365,c1(OC)cc(CN2CC(C)(C(=O)Nc3cccc(SC)n3)C2)cc(F)c1 6366,C12(C(=O)NC(CC)(CNC(c3cc(C#N)c[nH]3)=O)CC)CC(C)(C1)OC2C 6367,N1(C(C2C(C(=O)OC)C=C2)=O)CCC2(CC1)CC(NC(c1cc(O)ncn1)=O)C2 6368,C(CC(C(=O)NC1(C)CC(O)C1)NC(C1CC2CCC2C1)=O)OC 6369,C(CCC(C)C)(C(=O)NCC12CC(CCO1)C2)NC(c1cccc(CC)n1)=O 6370,c1(C(=O)NC(C)CCNC(c2scnc2Cl)=O)ccnc(O)c1 6371,c1(NC(C)=O)ccc(C(=O)N(CCCNC(=O)Cc2c[nH]nc2O)CCO)nc1 6372,CS(=O)(=O)C1(C(=O)NCCN2CCC(NC(=O)CC3C=CCCC3)CC2)CCC1 6373,CCCCC(C)C(=O)NC1COCCC1NC(C12CSCC1C2)=O 6374,Cc1nccnc1C(=O)NC1CC(C(=O)NCCCC2CCCO2)C1 6375,C1(C(C)C)CC=C(C(C(=O)NC2CC2)N(C)CC2CCC3(CC2)CC3(F)F)CC1 6376,N1(C(CC(=O)N(C)C)=O)CCC(NC(=O)CN(C)S(=O)(=O)N(C)C)C(CO)C1 6377,N1(C(C(C)C(F)F)=O)CCC(CC(=O)N(CCC(F)(F)F)C)(C(=O)NC)CC1 6378,c1(C(=O)NCC2CN(C(C(CC3CC3)OC)=O)C2)c(Br)ccc(F)c1C 6379,CC1SCCCC1NC(=O)Cc1ccc(CNC(C2CCCCC2)=O)cc1 6380,C#CC1(F)CN(C(c2ncoc2CNC(=O)C(C(C)C)OC)=O)C1 6381,C1(CNC(=O)C2=CCCC2)CN(C(=O)C2=CSCCO2)CCCO1 6382,C(=O)(CCC(C)(C)C)N1C(C)CC(CNC(Cc2ccc(C)cc2)=O)C1 6383,C12CCCN(C1)C(=O)C2.C1(COC(C)=O)CCN(C(=O)CC2CC3(CC3)C2)C1 6384,C1(C(=O)NC2CCCCN(C(C(C(CC)O)C)=O)C2)CCc2nccn2C1 6385,c1(CN2CCC(CC(=O)N(c3ccc(Cl)cc3)CC)CC2)cccc(OC)c1Cl 6386,C1(F)(C(=O)OC(CC#CC)C)CCCN(C(=O)C(CC)CCOC)C1 6387,C1(NC(C=CC=CC)=O)CN(C(=O)Cc2ncc(C)[nH]2)C2CCCC12 6388,C1(NC(C(C)(C2CC2)OC)=O)CCCCC1C(=O)NC12CC(C)(C1)C2 6389,C(=O)(C(C)(C)CC(F)F)NC1C(NC(c2n(CC)cc(Br)c2)=O)CC1 6390,c1(CCNC(c2c(Br)cc(C)c(C)n2)=O)ccc2c(n1)OCCO2 6391,C1(C(=O)NCCN(C(=O)CC2(C#N)CCC2)C)CCCC(NC(C)(C)C)CC1 6392,C1(CNC(C=C(C)Cl)=O)CN(C(C2CC2c2cncn2C)=O)CCCO1 6393,c1(CNC(CC2N(C(C(C)n3cccc3)=O)CCC2)=O)ccc2nc[nH]c2c1 6394,C(N=C(NC1CC1)N1CCCC(C)(C#N)C1)c1nnc(SC)s1 6395,C(=O)(C(C)(C)CSC)NCC(c1ccc(OC)cc1)NC(=O)Cn1ccc(C)n1 6396,Cc1cc(CC2CC2)sc1C(N1CCC(O)(C(Cl)(Cl)Cl)C1)C(=O)NCCCF 6397,O(N=C1CCCCCC1)CC(=O)NC1CC(O)(CNC(CN(C2CC2)CC)=O)C1 6398,N#CC1=C(C(=O)NC(CO)C(=O)NCCOC2CCC2)CCC1 6399,C(C(O)CC(=O)NC1CCCC(C(=O)NCc2nc[nH]n2)C1)N(C)C 6400,N1(C(C2OCCN(CC)C2)=O)CC2CC3CC2C1C3NC(c1cc(Cl)cnn1)=O 6401,Cc1[nH]c(C#N)cc1C(=O)NC(C1CCOC1)CNC(c1ccc(O)nn1)=O 6402,C(=O)(C(C)C(C)NC(=O)CCc1cc(C)no1)NC(C#C)CC1CCCC1 6403,C1(C(N2CC(CNC(C3CCN3C3CCCC3)=O)C2)=O)CCC2(CCCC2)CC1 6404,CC(CC(=O)NCCc1ocnc1CNC(=O)C#CC1CCOC1)C(C)(C)C 6405,S(=O)(=O)(c1cc2c(C(=O)OC)cccc2s1)N(CC=C)CC=C(C)Cl 6406,N1(C(=O)C=CCO)CCCCCCC1C(N1CC2(CO)CC2(CO)C1)=O 6407,C=CC1OCCCC1C(=O)NCCCC1CCCN1C(C1CCC=CCCC1)=O 6408,C(=O)(CS(=O)(=O)CC(=O)N(C)CCNC(C1CCCC2(CCC2)C1)=O)OC 6409,N1(C(c2c(OC)ccs2)=O)CCCC(C2CCN(C(=O)Cc3nnc(C)o3)C2)C1 6410,C1(CNC(CCC(=C)C)=O)C(C)CCCN1C(=O)CC(C)(C)C1CC1 6411,C1(NC(c2cc(-c3ccco3)c[nH]2)=O)CCCN(C(=O)CC(F)(F)Cl)C1 6412,C1(C)(C(=O)NCC(c2ccc(O)cc2)OC)COCCO1 6413,C(CCS(C)(=O)=O)(C(=O)NCC=CCNC(=O)CCC1CCCOC1)OC 6414,CC(CN=c1cc[nH]cc1S(=O)(=O)NCC1CCCC12CCOCC2)S(N)(=O)=O 6415,c1(C(=O)NC2C(N(C(C(CC)O)=O)C)CCCC2)cc(C(N)=O)ccc1F 6416,CC1=CCN(C(=O)C(C2CCCCC2)NC(=O)Cc2cc[nH]c2)CC1 6417,N1(CC)CCC=C(c2cc(C(N3CCc4nncn4CC3)=O)cc3c[nH]nc23)C1 6418,C(CCCCC(=O)NC1CCC(C)(CNC(c2[nH]ccc2CC)=O)CC1)=CC 6419,C1(CC)C(C(=O)NC2CC(NC(=O)C=CCNC(=O)OC(C)(C)C)C2)CCN1C 6420,N1(c2cc(Nc3cc(P(C)(C)=O)cs3)nc(C)n2)CCC2(C1)C(=O)NC(=O)N2C 6421,c1(OC)ccc(C(=O)N(C2C3CN(C(=O)C(F)CC4CCC4)CC23)CC)c(C)c1 6422,C(=O)(CC(C)(C)NC(C1CCC(=O)O1)=O)NC(c1ncn(C)n1)C 6423,c1(C(=O)NC(C(C)NC(c2cccc(C(C)C)n2)=O)CO)cc(Cl)c(F)cc1O 6424,c1(C(=O)NCCN(C(c2cn(C3CCC3)nn2)=O)CC)csc(I)c1 6425,Cc1ccc(F)c(C(N2C(CNC(=O)C(F)C(C)(F)F)CC3CC23)=O)c1 6426,CC#CCCC(=O)NC(C)(CNC(=O)C(Cc1ccccc1)N(C)C)C(C)C 6427,C(C(CC1CC1)C(=O)NCc1ccncn1)NC(C1(C)CC(=O)C1)=O 6428,N1(C(c2c(O)cc(C)nn2)=O)CC(NC(=O)CCc2ncc[nH]2)CC12CCCC2 6429,c1(C(=O)NC(CCNC(C)=O)C(C)C)cc(O)nc2c(Br)cccc12 6430,C(=O)(C(O)C(F)(F)F)NC(CCNC(C1CN(C2CCN(C)CC2)C1)=O)C1CC1 6431,N1(C(c2ccc(N(C)C)nn2)=O)CC2OCCN(C(=O)Cc3cn(C)nn3)C2C1 6432,C(=O)C(C)C(O)CC.C(=O)(CC(OCC)OCC)NCC 6433,N1(C(c2c(C)ocn2)=O)CCC(C)C(CC(=O)N(C2CNC(=O)C23CC3)C)C1 6434,C(=O)(CC1COCc2ccccc21)Nc1snc(-c2cccc(C)c2)n1 6435,C#Cc1ccc(F)c(C(=O)N(CC)CC2CCCN2C(C2CC(F)C2)=O)c1 6436,C1(NC(Cc2ccc(C)s2)=O)CC2(NC(=O)CCC3CCC3)COC1C2 6437,C1(C)(CNC(CC(=C=C)C)=O)CCN(C(=O)CCC2CCCC(O)C2)CC1 6438,c1(C(=O)Nc2nc(C)nc(O)c2)cnc2n1CCN(C(C1CCCS1)=O)C2 6439,c1(C(C)(C)C)cccc(CNC(C2CC(F)CN2C(C2CNC(=O)O2)=O)=O)c1 6440,N1(C(c2c(C)nccn2)=O)CCN(C(C2OCCCC2(C)C)=O)C2CC12 6441,C1(C(=O)NCC2(C)N(C(C(C)=C(C)C)=O)CCC2)CC2(C1)CC(C)(C)C2 6442,CN1CCOc2c(C(N3CCC(NC(C4(C)CCCO4)=O)C3(C)C)=O)cccc21 6443,CC1CN(C(C23CCN(CC2)C3)=O)CCN1C(C1COCCN1C)=O 6444,c1(CNc2cc(OCC)ncn2)cc(C(F)F)cc(F)c1 6445,c1(C(N2CC3C(C2)C3(F)F)=O)cn2cc(-c3c[nH]c4ccccc34)ccc2n1 6446,CC1CC(C(=O)NCC2(C(=O)N(C3(c4cc[nH]n4)CC3)C)CC2)CN1C 6447,N1(C(C2(CC#C)CCOCC2)=O)CCC2CN(C(=O)C(C)SCCCC)C2C1 6448,N1(C(CCC=CC)=O)CCC(C)C(NC(c2ccc(O)c(C(N)=O)c2)=O)C1 6449,C12(C(=O)NC3C(C)CN(C(=O)C=Cc4ncc[nH]4)C3)CCCN1S(=O)(=O)CC2 6450,c1(C(=O)NC2CCCN(c3ccccc3F)C2=O)cc2cccc(F)c2s1 6451,C1(C(=O)NC(CNC(c2c(CC)nccn2)=O)CCOC)CC2(CCC2OC)C1 6452,c1(C(=O)NC2CC(NC(c3cccc(C4CC4)c3)=O)C2)cnn2cccc(Cl)c12 6453,Cc1cnccc1C(N1CC(=C(F)CNC(c2csc(Cl)c2Cl)=O)C1)=O 6454,c1(C(C)CNC(=O)Cc2ncnn2C)noc(CC2CCCC2)n1 6455,C1(OC)CN(C(=NCCCSC)NCC2CCN(C(C)=O)CC2)CC1OC 6456,C(=O)(CCCCCn1cnnn1)NCCC(C)(C)NC(C1(C)CC1)=O 6457,CCCC(C)(O)CC(=O)NCCCC(CCC)NC(c1ccc(Br)cc1)=O 6458,C1(CC)CCN(C(=O)OC(C)(C)C)CC1(c1nn[nH]n1)N(CCO)CC 6459,C1(C(=O)NCC(=CC(=O)NC(CC#C)C)C)CC12CCC2 6460,C(CCC(C)C(=O)NC1(CC(=O)NC2(CCCOC)CC2)CCC1)OC 6461,N#Cc1cc(S(=O)(=O)NC2CCCCN(C(=O)C(F)F)C2)ccc1Br 6462,C(=O)(C1=CC2CCC1C2)NC1CCN(C(c2ccc(C)c(O)c2)=O)C1 6463,C12(NC(Cc3cn(CCOC)nn3)=O)CCCC(CN(C(C3(C#N)CC3)=O)C1)C2 6464,Cc1cc(N)c(C(=O)N(C2CN(C(C3CCN3C)=O)CC23CC3)C)cc1C 6465,c1(C(=O)NC2C(NC(c3cncnc3)=O)CC2)ccc(F)c2occc12 6466,c1(C(N2C(CN=c3[nH]nc(CCOC)o3)CCCC2)=O)nsc2ccc(C)cc12 6467,CN(Cc1c(OCCO)cccc1F)N1CC(Nc2ccc(N3CCCC3)cc2)C1 6468,CC1CCCC(C)N(C(C2CCCN2C(C23CC2CNC3=O)=O)=O)C1 6469,C(=O)(C(O)C(C)(C)C)NC1(CNC(c2nccc(CC)c2)=O)CCCC1 6470,c1(CC)nnc2cc(NC3CCN(C(=O)C(C)CCOC)CC3CC)ncn12 6471,N1(C(c2c(Cc3ccc(C)c(Cl)c3)nccc2)=O)CCC2(CC1)CNC(=O)OC2 6472,N1(C(C2N(C(CC=CC=C)=O)CCCC2)=O)CCOC(C(=C)C)C1 6473,Clc1ccc2[nH]c(=NCc3cnsc3)nc(N3CCC(OCC4CC4)CC3)c2c1 6474,CON(CC(C)C)C(=O)C(F)C(F)(F)F.C1(=O)CCC=N1 6475,Cc1cc(C#N)sc1C(=O)NCC1CC(CNC(c2nc(Cl)cs2)=O)CO1 6476,C1(C(N)=O)CCC(C(N2CCCC2CNC(=O)C(CC#N)c2ccccc2)=O)CC1 6477,C1(NC(c2scc(OC)c2)=O)CCS(=O)(=O)C12CN(C(C1(C)CC=CCO1)=O)C2 6478,C(=O)(CCC(C)N(C)C)NCCN1CCC(NC(c2cc(CCC)on2)=O)C1 6479,C1(C(=O)NCc2cc(C(NOCC(=O)N(C)C)=O)sc2)CC(N=[N+]=[N-])C1 6480,c1(OC(=O)CCOC(C)=O)c(Cl)cc(Cl)cc1Cl.C=C1CCN2C(C1)C2=O 6481,C1(CC=C)CCN(C(=O)C(CN(C)C)NC(=O)Cn2nccc2C)C1 6482,C1(F)(C(N2CC(C(=O)Nc3cc(C)cc(F)c3)C2)=O)CCCCC1(F)F 6483,C1(CNC(C2(CC=C)CC2)=O)C(C)CCN1C(c1nn(C)nc1Br)=O 6484,Cc1oc(C#N)cc1C(N1CCC(C)(C)C1C(N1CCCC(CO)CC1)=O)=O 6485,c1(OC)ccnc(C(N2CCC(N(C)C(c3cc(Cl)cs3)=O)C(C)C2)=O)c1N 6486,c1(C(=O)NCC2C(CNC(c3c(CC)[nH]c(=N)s3)=O)C2)cscc1S(C)(=O)=O 6487,C(CNC(=O)CN1CCCCC1=O)(C(C)C(C)C)NC(c1c(C)csc1)=O 6488,c1(CC(=O)NCCOCCCNC(CC(CCC)C)=O)ccc2c(c1)CCOC2 6489,C1(C(N(CCCNC(=O)CCc2ncnn2C)CC)=O)CCc2ncccc2C1 6490,N1(C(c2c(C(C)C)occ2)=O)CCC(C)C1CNC(c1nccnc1Cl)=O 6491,c1(OC)c(NC(=O)CN2CCN(C(C3(O)CC3)=O)CC2)cc(Cl)cc1Cl 6492,C=CCC(C)(C)C(=O)NCC(C)(C1CC1)NC(c1nccnc1N)=O 6493,N1(C(c2cc(C)sc2C)=O)CC2CCC1(CNC(c1n[nH]cc1C)=O)CC2 6494,N1(C(c2cc(C)nn2C)=O)CCOC2CN(C(c3conc3C(C)(C)C)=O)CC12 6495,c1(C(N2CC(CCNC(=O)COc3cccnc3)C2)=O)ccnc2ccncc12 6496,c1(C(=O)NCC(CNC(C(CC)n2cncn2)=O)(C)C)cn(C)nc1COC 6497,c1(CNC(=O)CSCC2CCC2NCc2cnn[nH]2)nc2ccccc2[nH]1 6498,CCC(C)C(CC(=O)NCC(C)(F)C(C)(C)F)NC(c1cccc2ccnn12)=O 6499,c1(CN2CCC(N(CCC)C(c3ncccc3F)=O)C2)ccccc1[N+](=O)[O-] 6500,N1(C(CCC(=O)N(C)C)=O)CC2CCCN(C(c3cccc4c3CCC4)=O)C2C1 6501,Cc1noc(C)c1C(=O)NCC(F)CNC(C1(C)CC(C)(C)C1)=O 6502,c1(C(=O)NCC2N(C(C3CC(C)N(C)CC3)=O)CC(O)C2)ccc2cccnn12 6503,C(C)(C)(C(=O)NCC(F)CNC(c1coc(C(C)C)n1)=O)OC(C)=O 6504,N1(C(C(C)C)C(=O)NCC2CCCO2)CCCCCC(N)C1 6505,c1(C(=O)NC2CN(C(Cc3c(C(=O)OC)csc3)=O)CC2C)ccc(N)c(O)c1 6506,c1(Nc2c(SC)cccn2)nnc(C2CC2)cc1CS(N)(=O)=O 6507,c1(C(=O)NCC2N(C(C(C=CCCC)O)=O)CCC2)cccc2ccc(O)nc12 6508,c1(CNC(=O)CC2CCCN(C(=O)CC3CSC3)CC2)ccc2cc[nH]c2c1 6509,c1(SC(Cn2c(C#C)cc(C3CCCCC3)n2)=O)sc2c(c1F)CCCC2 6510,C(C(C)C(=O)Nn1cccn1)NC(C(=Cc1ccccc1)C)=O 6511,C(=O)(C=C1SCC(=O)N1C)N1C(CN(C(C(CN(C)C)O)=O)C)COCC1 6512,N1(C(Cn2ncc(C#C)c2)=O)CC(C)CN(C(=O)CCCCC=C)C(C)C1 6513,CCCC(CCC)=CC(=O)NC1CC(NC(=O)CCCn2cccn2)C(O)C1 6514,C1(C#N)(C(=O)OCC)CN(C(=O)Nc2ccc(OC3CC3)cc2)C1 6515,c1(C(=O)NC(CC)CNC(=O)CC(C)CC(C)C)cc2c(OC)cc(OC)nc2[nH]1 6516,N1(C(C(CC=C)NC(C)=O)=O)CCC2(CCCC2NC(=O)CC(F)(F)F)CC1 6517,c1(CC(=O)NCC(CCNC(CC(=O)OC)=O)O)coc2ccccc12 6518,c1(NCC)ccc(C(=O)NC2CCCC(NC(c3cnnn3C3CC3)=O)C2)nc1 6519,C1(CNC(C(C)NC(c2ccoc2)=O)=O)C2CC1N(C(=O)Cc1ccno1)C2 6520,C1(C(N2CCCN(C(c3ccc(N)cc3O)=O)CC2)=O)CC12CCS(=O)(=O)CC2 6521,CC1CC(C(=O)NC2(c3ccccc3)CN(C(C3CCC(=O)N3)=O)C2)CC(=O)N1 6522,c1(CC)cc(=NCC2CCCC(NC(C3CC(N(C)C)C3)=O)C2)[nH]cn1 6523,C12(CNC(CCCCC)=O)CCCC1N(C(=O)C(F)=C(C)C)CCC2 6524,C(=O)(C1=Cc2ccccc2C1O)NC1(C)CC(NC(c2ccc(NC)cc2)=O)C1 6525,N1(C(c2ccc(C(=O)NC)cc2)=O)CCC(NC(c2n[nH]cc2Br)=O)CC1C 6526,C12(NC(c3cnc4n3CCS4)=O)CCCC1N(C(C1CCCSS1)=O)CCC2 6527,N1(C(c2ccc(F)cc2Br)C(=O)NC(C(=O)OC)C)CCOC2(CCSC2)CC1 6528,c1(C(=O)NCC(CNC(=O)CC2(N3CCCC3)CC2)OC)ncccc1O 6529,Cc1c(Br)ccnc1C(=O)NCC1CC1NC(c1snnc1C1CC1)=O 6530,c1(NC(c2cccnc2F)=O)ccc(=NCc2cccc3sccc23)[nH]c1 6531,Cc1c(NC(=O)C(N2CC(F)C(F)C2)=O)cccc1Cc1ccccc1 6532,N1(CC)CC2(CCC(CNC(=O)CN(C)C(N)=O)O2)C1.n1(C=O)cc(C2CC2)cn1 6533,Cc1cnc(C(=O)NC(C)CCN(C)C(C2CC2(C)C(F)F)=O)c(Br)c1 6534,Cc1ccc(C)c(C(=O)NC(CNC(c2cn[nH]c2)=O)C(C)C(C)C)c1 6535,C1(O)(CCNC(CN2CC(C)(C)C2)=O)CCCN(C(c2cnc3n2CCC3)=O)C1 6536,N1(CCN(C(C2(OC)CCCC2)=O)C)CCN(C(=O)CCS(C)=O)CC1 6537,c1(C(=O)NC2CCN(C(CCCCCOCC)=O)C2)ccc2c(c1)COC2 6538,C1(CCC)CN(C(=O)Cc2nocc2C)CCN1C(c1cc(C)n(CCO)n1)=O 6539,c1(NC(C2C(C(=O)NC3CC(c4ccccc4)C3)C2)=O)ncc(Cl)cc1Cl 6540,c1(N(C2(C#N)CCNC2)Cc2c(C)noc2C)ncnc2cnn(C)c12 6541,C(=O)(C(CCS(C)=O)N(C)C)NCCC(C)N(C(c1c(CCC)occ1)=O)C 6542,O=C(C1=NOC2(CCC2)C1)NCC1(CO)CC12CCN(C(=O)CC1CCOC1)CC2 6543,C1(C(N2CC(C3(NC(c4c[nH]nc4C4CC4)=O)CC3)C2)=O)CCC2CCC(=O)N12 6544,C1(O)(CNC(c2cc(I)c(Cl)cn2)=O)COCCC1O 6545,C12(C(N(CCNC(=O)C(C)O)CC)=O)CC(C(C)C)(CO1)C2 6546,c1(C(=O)NC2CC(O)(CNC(C(C)(C)CO)=O)C2)cccc2c1OCC2 6547,N1(C(C2C(NC(C=CC=CC)=O)CCC2)=O)CCCC(CCO)C1 6548,Cc1csc(C(C)C(=O)NC(CNC(c2ccc(C(C)C)s2)=O)C(C)C)n1 6549,N1(C(Cc2cc(C)on2)=O)CC(C(=O)NCCc2ncc(C)o2)OC(C)C1 6550,C1(CNC(c2c(C)cn(C)c2)=O)CC2(CC2)CN1C(c1cc(F)n(C)n1)=O 6551,N1(C(C(=O)Cc2ccccc2)=O)CCC2(C1)CN(C(C1CC=CCC1)=O)C2 6552,C12(C(N3CCC(C)(CCNC(c4nnc(C)s4)=O)CC3)=O)CCC(CC1)C(C)O2 6553,N1(C(C(=O)N(CC(C)S(C)=O)C)=O)CCC(C(=O)OC(C)(C)C)C(F)C1 6554,c1(OC)ncc(C(N2CCC(NC(C3CC3C(C)(C)C)=O)CC2)=O)cc1Cl 6555,C1(CNC(C=CCN(CC)CC)=O)CN(C(C2(COC)CCCC2)=O)CC1C 6556,CC1(C(=O)NC2CCN(C(c3csc(CO)n3)=O)CC2)COC(=O)OC1 6557,N1(C(c2ccnc(C)n2)=O)CCN(C(C2(c3cccnc3)CC2)=O)C(C2CC2)C1 6558,c1(C(N(C2CN(C(=O)CC=CC(C)(C)C)C2)C)=O)ccc2c(c1)OC(F)(F)O2 6559,N1(C(Cc2c(CC)cccn2)=O)CCC2(COC(CNC(=O)CCC(C)O)C2)C1 6560,CCCCC(F)C(=O)NCC1CC1CC(=O)NC(C)C(=O)N1CCCC1 6561,C1(c2n(CCC3(C)CC3)nnn2)(NCCC(O)C2CCC2)CC2CSCC2C1 6562,Cc1ccc(C(=O)NC(CNC(=O)Cc2ccoc2)CC(C)C)nc1C 6563,c1(NCC2C(NC(CC(OCC)OC)=O)CCCC2)ccc(Br)cc1[N+](=O)[O-] 6564,C1(NC(C(C)N(C(c2c(COC)noc2)=O)C2CC2)=O)CCS(=O)CC1 6565,CC1(NC(=O)C2=CCOC2)CCCN(C(=O)CC2CCNC(=O)C2)C1 6566,C(CC(C)(C)C)(C(=O)N1CCCCC1CCC(C)(C)NC(c1cocn1)=O)OC 6567,C(=O)(CC(O)CC(C)(C)C)NC1(COC)CCN(C(=O)CNS(=O)(=O)NC)CC1 6568,c1(SC)cccc(C(F)(F)F)c1.C12(CCC1)C(=O)NCCCOCCCNC2=O 6569,CCCC(C)(C)CC(=O)N1CC2OCC(NC(=O)C(C)(C)CN3CCOCC3)C2C1 6570,c1(C(N2C(C)(C(N(CC(C)(C)O)C)=O)C=CC2)=O)n[nH]c2c1CCC2 6571,CCC(C(=O)N1CCCCC1CCCNC(=O)CSCC(F)F)C(F)(F)F 6572,Cc1cc(C(=O)NCC2CN(CCNC(C3CC(C)CO3)=O)C2)ccc1F 6573,CCCCCC(CC)C(=O)NC1CN(C(c2ccc(N)c(SC)c2)=O)CCC1C 6574,c1(OC)ccc(C(=O)NCC2(F)CN(C(=O)C(F)C3CCOC3)C2)c(F)c1 6575,c1(C(N2C(CN(C(=O)CCC3CCOC3)C)CCC2)=O)cc2cccn2cn1 6576,C(C)(C(C)(C)C)=CC(=O)NCC(c1ccccc1)NC(C(c1cccs1)SC)=O 6577,C1(C)(CNC(c2cnc(OC)s2)=O)CCC(NC(=O)CN(C)C(N)=O)CC1 6578,CC1(C)OC(C)(C)C1C(=O)NCC1CN(C(=O)Cc2nc[nH]n2)CC1(C)C 6579,c1(-n2cc(C3(O)CN(C(=O)Cc4ccc(C5CC5)cc4)C3)nn2)ncc(Br)cn1 6580,N1(C(CC2C(C)CCCC2)=O)CC2CCCC(NC(c3cc(CO)[nH]n3)=O)C2C1 6581,C#CCCCCCCCC(=O)NC12CCC(CC1n1cc(-c3cnsc3)nn1)C2 6582,c1(CC(=O)NC2(CNC(=O)CC3C=CCCC3)CCOC2)nc(F)c(F)cc1F 6583,N1(C(c2cncc(NC(c3cc(C)cc(C)c3)=O)c2)=O)CCC(C)(CO)C(O)C1 6584,C#CCCCCCC(=O)NC(CNC(c1nn(C)c(CC)c1Br)=O)CO 6585,CC(CCC(C)(C)C)C(=O)N(C1CCCN(C(=O)CS(=O)(=O)C2CC2)C1)C 6586,c12ccc(F)cc1Cn1cc(nn1)CC1CCN1C2=O.S(C)(=O)(=O)N(C)C 6587,N1(C(CC)=O)CCC(C(N2CC(N(CCO)C(C3CCS3(=O)=O)=O)C2)=O)C1 6588,Cc1n[nH]cc1CC(=O)NCCOC1CN(C(C2(CC3CC3)CCCC2)=O)C1 6589,c1(C(c2n(CC(=C)C)nnn2)NCc2ccnn2CCC)ccnc(SC)c1 6590,CCCC(C)(C)C(=O)N1C2CCC(C2)C1CC(=O)NCCOC(F)F 6591,N1(C(C(=O)N(CCCN2CCCC2)C)=O)CC2(CO)CCCC2(CO)C1 6592,CC1CN(C(c2ncccc2F)=O)CCCN1C(=O)Cc1cc(F)c(F)cc1F 6593,C1(N(C2CCN(C)CC2)CC(C)=CCN(C2CC(C#N)C2)CC)CCCOCC1 6594,N1(C(c2cncc(OC)n2)=O)CC(O)C(O)C1CNC(=O)CSCc1cscn1 6595,c1(C(c2n(CCCSCC)nnn2)NCCCS(C)=O)ccnc(N(C)C)c1 6596,C(=O)(CCCCC(C)(C)C)N1CCC2(CC(NC(C(CCC(C)C)O)=O)C2)C1 6597,C1(C(=O)NC(c2ccc(C)cc2)CC)CN(C(=O)Cc2ncn(C)c2C)CC1OC 6598,C1(C)(CN(Cc2cccc(COC)c2)CCS)COc2ccccc2O1 6599,N1(C(CC2CC(OC)C2)=O)CCCN(C(C2C(C#N)C2(C)C)=O)C(C)C1 6600,Cc1nn(CC(F)F)cc1C(N1CCC(O)(CNC(C2COC(=O)N2C)=O)C1)=O 6601,c1(C(N(CCCNC(C(CC)O)=O)CC2CC2)=O)ccc(-n2cnnc2)cc1 6602,c1(CCC(C(=O)C(F)(F)CO)=O)cccc(F)c1.N1CCCCC1c1cn(CO)nn1 6603,C1(C(N(CCOCC)C)=O)CCn2c(cnc2Br)C1.C(=O)C=CCF 6604,c1(COC)cc(C(=O)NC(C)(C)C=CC(=O)NCCCS(C)=O)no1 6605,c1(OC)cc(C(N2CC3OCCOC3C2)=O)cc(OC)c1Br 6606,c1(OCC)cc(NC(C2(C(N3CC(SC)C3)=O)CC2C)=O)on1 6607,N1(C(C(C)N(C(C)=O)C)=O)CC(CNC(c2cn(C3COC3)nn2)=O)C(C)(C)C1 6608,N1(C(CN(CC)CC)=O)CC(C2CN(C(c3sc(C(C)C)nc3C)=O)C2)C1 6609,C(C(N=c1cc(C(N)=O)nc(Cl)[nH]1)c1ccc(F)cc1)NC(CC(C)SC)=O 6610,c1(CN(CC(=O)NC(C)(C)C)CC)cc(CCN(C2COCC2O)C)ccc1Br 6611,C1(C(=O)NCCN(C(=O)C(C)CO)CCC)CC2(F)CC1C2 6612,c1(C(=O)NCCN(CC(C)O)C(C2CCC3(CC3)C2)=O)ccnnc1S 6613,N1(C(C)=O)CC2(CC2)CC1CNC(C1OCCOC1C1(C(=C)F)CCC1)=O 6614,C12(C(=O)NC(CNC(c3ccc(SC)o3)=O)C(C)C)CC(CO)(C1)OC21COC1 6615,C1(NC(C2C(C)(C)C2(C)C)=O)CCN(C(C2Cc3nccn3C2)=O)CC1F 6616,Cc1cc(C)n(Cc2cn(CCCCNC(C3(F)CCOC3)=O)nn2)n1 6617,C1(C(=O)NCc2nnn(CC)n2)(CC)CCCN1C(=O)CC1NC(=O)NC1=O 6618,Cc1nc(-c2cnn(C)c2)oc1C(=O)NC1CCC1NC(C1CC1C(C)(C)C)=O 6619,N1(C(C2C(C)C2C)=O)CCN(C(=O)C2=CCC2)CC1c1ccccc1Cl 6620,c1(N2CC(C)(CC(C)C)OCC2)nc2cccnc2c(=NCCCSC(F)F)[nH]1 6621,N1(C(C2N(C(C3(CC)CCC3)=O)CCSC2)=O)CCc2oc(C)nc2C1 6622,c1(C(=O)NCC2CN(C(CCc3c(C)ncs3)=O)C2)cc(F)cc2ccncc12 6623,Cc1nc(C(C)C)nc(O)c1C(N1CC2CC1(CNC(C1(C)CCCO1)=O)C2)=O 6624,CCC(C)C(O)C(C)C(=O)NCc1cc(C)c(C(=O)NCCC(F)(F)F)o1 6625,C#CCC(CC(=O)NC(C)(COC)C1CC1)NC(c1cc(O)n(C)n1)=O 6626,C1(C(=O)OCC)C2CC(CN(C(=O)C(=O)C(C)C)C2)N1C(=O)C(C)OC 6627,C(C)(CCC(=O)NC(C)(CO)C(=O)N1CC(c2cc(CO)no2)C1)OC 6628,n1(CC(N2CC(N(C(=O)C=Cc3ccoc3)C)C(F)C2)=O)ccc2ccccc12 6629,C1(CC(=O)NCCCOCCNC(C(CC)C)=O)CS(=O)(=O)CCN1C 6630,c1(C(=O)NCCC(C)NC(C2NC(=O)C3CCC23)=O)c(F)ccc2occc12 6631,CC1(C)CCN(C(c2cc(F)ccc2F)C(=O)NCc2ccco2)CCS1=O 6632,CCCCC(CCCC)C(=O)N1CCCC2(C1)CN(C(=O)C(F)CN(CC)CC)C2 6633,Cc1oc2ccccc2c1CC(=O)N(C)CCN(C)C(C1(C)CC1(F)F)=O.C 6634,C=CCC(CC(F)F)NC(C12CC1CN(C(c1ccn(C)c1)=O)C2)=O 6635,CCC(Cc1ccccc1)CC(=O)NC(C)CNC(=O)Cc1c(C)nn(C)c1C 6636,C(=O)(CCCCCSC)NC(CN(C(c1cnn(C2CC2)c1)=O)CC)C 6637,c1(C(N2C(CNC(c3cccc(SC)c3)=O)CC2)=O)cc2c(cn1)OCCC2 6638,CCCC(C(=O)NCC1CCN(C(c2nc(C)no2)=O)CC1C)C(C)C 6639,S(=O)(=O)(CC(=O)N(C1CCC(NC(=O)C(C)OCC2CC2)CC1)C)NC 6640,N1(C(C(C)OCC)=O)CCCC1CCNC(=O)C(C)n1cccn1 6641,C1(CC(=O)NC(CNC(CCOCC)=O)CO)CCC2(CC1)CCC2O 6642,N1(C(c2cc(C)nc(Cl)c2)=O)CCC=C(C(=O)Nc2c(F)ccc(F)c2F)C1 6643,CN1CCc2[nH]nc(C(=O)NCC3CN(C(C4CC5CC4CC5(F)F)=O)C3)c2C1 6644,CCC(C)CCCC(=O)NCCNC(=O)C(C)(O)C1CC1 6645,C1(NC(=O)CCC2CCCCN2C(c2cncnc2)=O)CC2CCC1(CO)C2 6646,c1(OC)ccc(CN2CCC(O)(C(=O)Nc3nc(Cl)ccc3I)C2)c(Br)c1 6647,Cc1ccn(CC(=O)NCCC(C)N(C(=O)C(C)SC(C)C)C)n1 6648,Cc1ccc(C)c(SCC(N2CCC23CN(C(=O)Cc2ccccc2O)C3)=O)c1 6649,c1(C(=O)NCCCN(C(=O)C=Cc2cc[nH]n2)CC)cc(CO)oc1C 6650,c1(NC(C2CCN(C(C3CCC(CO)CC3)=O)CC2O)=O)cc(O)ccc1Cl 6651,c1(C(N2CC3CC(NC(CC=C)=O)CC3C2)=O)ccc2cnc(C)n2c1 6652,c1(OC)ccc(Br)cc1OCC(=O)NC(c1ccc(OC(F)F)cc1)C 6653,C1(OC(C2CCC(C(C)(C)C)CC2)=O)CC2(CNC(=O)N2)C1 6654,C(CCCC(=O)N1CC2CCC2C1)NC(c1cnccn1)=O 6655,N1(C(c2c(F)cc(NC(=O)OC(C)(C)C)c(F)c2)=O)CCCC2(CCCCO2)C1 6656,Cn1ncc2cc(C(=O)NC(C3CCOC3)CNC(=O)C3CC3)cc(O)c12 6657,C1(CNC(CN(C(=O)CCOC2CCCC2)CC)=O)CCCC(C)(C)C1 6658,N1(C(c2c(C)sc(O)n2)=O)CC2(CCN(C(C3(F)CC3C)=O)C2)C1 6659,CC(CC(=O)NC1CC2(C1)CC(CNC(c1cnc(O)n1C)=O)C2)CC(C)(C)C 6660,c1(C(=O)NCC(CCCC)NC(=O)CCCCOC)c(C)nc(COC)nc1C 6661,C(=O)(C#Cc1ccccc1Cl)NC(c1ccc(OC)cc1)C(=O)OC 6662,C(CC(O)CNC(c1csc(-c2ccoc2)n1)=O)NC(C1(C)CSC1)=O 6663,N1(C(CC2CCN(C(C)C)C2)=O)CCC2COC(NC(=O)C(Cl)(Cl)Cl)C2C1 6664,C1(NC(C(CC)(C)CO)=O)CN(C(c2ccc(SC)s2)=O)CC1S(C)(=O)=O 6665,c1(CC(N2CCC(NC(=O)C(O)C3CCC3)C2)=O)ccc(F)cn1 6666,CC1(C)CC(CNC(=O)CC2(C)OCCO2)N(C(=O)CCC2OCCO2)C1 6667,CC1CC=C(C(=O)N2CC(CCNC(=O)C(C)(C)c3ccn(C)n3)C2)CC1 6668,c1(C(=O)NC(CCNC(CCc2ccc(C)nc2)=O)C)[nH]c(=N)ccc1C 6669,CCCC(CCCO)C(=O)NC(C1CCN(C(c2[nH]c(C)c(C)c2C)=O)C1)C 6670,C1(NC(C(C)CC2CC2)=O)CN(C(=O)CC2CCOC(C)(C)C2)CC2(CC2)C1 6671,c1(N(C(C23CC(C(=O)NCC)(C2)C3)=O)C)ccc2cnccc2c1 6672,C(=O)(C(F)(F)CN(C)C)NCC(c1cccc(C)c1)NC(C1C(C=C)C1)=O 6673,c1(C(COC)(C)O)cn(CC(C)NC(=O)C(CN(C)C)N(C)C)nn1 6674,CN1CCC(CC(=O)NC(Cc2ccccc2Br)C(=O)NC2CC3CC3C2)CC1 6675,N1(C(CC2(OCC)CCC2)=O)CCN(C(=O)C(C)(O)C2CC2)CC1CC(=O)NC 6676,C1=CC(=O)N2CCC1CC2.O(C=CC(=O)OC)CC 6677,Cc1cc(C)nc(SC2CC2)n1.C12(F)CC(C1)NC(=O)C2.C12CC(C1)CNC2=O 6678,CCC(CN(C)C)C(=O)N(CCCNC(C1(c2cccs2)CC1)=O)CCO 6679,c1(C(=O)OC)cccc(-c2ncc(C(=O)NCCc3cc(Br)c(Br)s3)s2)c1 6680,c1(C(N(CC(C)N(C)C(C2CCC(C)(C)O2)=O)C)=O)cc2cnccc2o1 6681,C1(C)(CC(=O)N(C2CCC(C)C2)C)CCN(C(=O)CCn2cccc2)C1 6682,C1(CC(N2C(C(=O)NCc3cn[nH]c3)CCC2)=O)CCC2(CCC2)O1 6683,N1(C(=O)NCC)CCC(C(=O)NCCCCC(C)NC(=O)Cc2cncs2)CC1 6684,Cc1cc(C(=O)NCCCCNC(=O)C(C(C)C)N(C)C)cc(C)c1N 6685,N1(C(C(CC)C)=O)CC2CCC(C1)C2NC(=O)C(C)OCc1ccc(F)cc1 6686,c1(C(=O)NC2C(CC)CN(C(=O)C(F)C(C)C)CC2)cc(C)c(F)cc1N 6687,C1(NC(=O)CCc2ccnc(Cl)c2)COC2(C1)CN(C(c1cn(CCO)nn1)=O)C2 6688,c1(C(N(CCN(C(=O)CC2CC2(Cl)Cl)C(C)C)C)=O)cc(Cl)ccn1 6689,c1(N2CCN(C(=O)NCC3CCCCC3C(F)(F)F)CC2)cccc([N+](=O)[O-])c1 6690,Cc1c(C(N2CCC3(C2)CN(C(=O)C(CCO)N(C)C)C3)=O)nn2c1CCCC2 6691,C(=O)(C1COc2ccccc21)N1C(C)CCN(C(Cc2c(C)scc2)=O)CC1 6692,C(C(C(=O)N(C(C)C(=O)NCc1occc1C)C)N(C)C)OC 6693,c1(C(N)=O)ccnn1CC(N1CCC(COC(F)F)C1)=O 6694,C12(CNC(c3cc(C)no3)=O)CN(C(C3CCS(=O)CC3)=O)CC1CCO2 6695,c1(C(=O)NC(C)C(C)C(=O)NCCCC(O)CO)nccc2[nH]ccc12 6696,N1(C(C=CCN)=O)CC=CCC1C(F)(F)F 6697,C(=O)(CCC(C(=O)Nc1cccc(Cl)c1C)N1CCSCC1C(C)(C)C)OCC 6698,CC(C)(C)CCCC(=O)N1CC(CNC(C2(Cc3ccncc3)CC2)=O)C1 6699,N1(C(C(CC)NC(c2cc(C)[nH]c2C)=O)=O)CC2CC=CCC2C1 6700,CN1CC(NC(=O)C(=O)N(C2CCCN(C3CS(=O)(=O)C3(C)C)C2)C)C(C)(C)C1 6701,N1(C(CC(C(C)C)O)=O)CCC(O)(C2(NC(=O)CC3CCC(=O)NC3)CC2)CC1 6702,c1(NC(CC=C)=O)ccc(=NCc2cccc(OC(F)(F)F)c2O)[nH]c1 6703,c1(CC)c(C(=O)NCCCNC(C2COC(C)C2)=O)cccc1F 6704,C(CCCC(=O)NCC(C)C(=O)NC(c1cncs1)C)OCC 6705,C1(CSC)CCN(c2cc(N(CC(c3ccsc3)C)C)ncn2)CC1 6706,C1(NC(Cc2c(CC)cccc2)=O)(CNC(=O)CCP(C)(C)=O)CCCCC1C 6707,N1(C(CC(CCC)C)=O)CCCCC(C2CN(C(=O)CCSCC)C2)C1 6708,C(CN=c1[nH]nc(O)s1)NC(c1ccc(C(C)(C)C#N)cc1)=O 6709,c1(CN2CCC(c3nc(C)on3)CC2)ccc2cc(F)cc(Br)c2n1 6710,c1(C(=O)NCCC2N(C(c3nc(COC)oc3)=O)CCC2)ccc(C)c(C)c1Cl 6711,CCCCC(O)CC(=O)NC1CCN(C(c2cnc(C3CCOC3)s2)=O)CC1 6712,C12(C(N3CC(NC(c4ccc(Cl)o4)=O)C(C(F)F)C3)=O)CCCN1S(=O)(=O)CC2 6713,C1(C(N(C2CCN(C(=O)Cc3cc(C)no3)C2)CC#C)=O)CC(C)(F)C1 6714,C1(C(N(C2CCCC2)CC#CC)=O)CCCC(NC(=O)C(O)C(F)(F)F)CC1 6715,C1(NC(c2cncc(C)c2)=O)CCC2CCN(C(=O)Cn3nnc(=N)[nH]3)C1C2 6716,C(C(=O)O)(C(F)(F)F)NC(C1CNCCN1Cc1ccccc1)C 6717,N1(C(C=CC(=O)N(C)C)=O)Cc2ccccc2C(NC(C2CC2C2CC2)=O)C1 6718,C1(CC(=O)N(CCOC)CCNC(c2ccnn2C2CC2)=O)CCCCC1(C)C 6719,C=C1CCC(C(=O)NC(C)(CNC(c2cnn(C(C)C)c2F)=O)C(C)C)CC1 6720,N1(C(c2c(CC)ccs2)=O)C2CCC1(CNC(=O)C=CS(C)=O)CC2 6721,c1(C(N(C)CC2COCCN2C(=O)CC2CCCOC2)=O)nnc(O)cc1O 6722,N1(C(C(CN)N)=O)CC2COCC2(C(=O)NCCCN2CCCCC2)C1 6723,C1(OC)CN(C(c2cnn[nH]2)=O)CC1NC(=O)C(C)(C)C1(C)CC1(F)F 6724,Cc1cn2cc(C(N3CCC(NC(=O)CN(CC(C)(C)C)C)CC3C)=O)nc2s1 6725,N1(C(CCCn2c(C)cc(C)n2)=O)CCCCC(N(C(=O)C=CCF)C)C1 6726,C(C(=O)NCC(c1ccccc1F)F)(C(C)(C)C)NC(C(C)(C)C)=O 6727,N1(C(C=CCCC)=O)CCN(C(=O)Cc2ccsn2)C2CS(=O)(=O)CC12 6728,c1(NCCSc2nnc(C)n2C)[nH]c(=NCC2COC(=O)O2)nc2scnc12 6729,N1(C(CC(OCC)OCC)=O)CC(C)(C)CC1NC(=O)Cc1cc(O)nnc1O 6730,N1(C(C(C2(OC)CCCC2)(F)F)=O)CC2CCC1C(CNc1ccnc(C)n1)C2 6731,c1(OCC(N2C(CNC(c3c[nH]ccc3=O)=O)C=CC2)=O)cccc(Cl)c1 6732,n1(CC(C)C)ccc(=NC(=O)C(=O)NCc2ccnc3cc(Cl)ccc23)[nH]1 6733,C(=O)(C1=NNC(=O)CC1)N1CC(O)(CNC(c2cnn(C)n2)=O)C1 6734,c1(C(C)C)cc(C(=O)NC(C)(CNC(=O)C(F)CC2CC2)Cn2cccn2)on1 6735,c1(CC(N2C(CNC(C(C)NC(C)=O)=O)CC2)=O)nnnn1C 6736,c1(C(=O)NCCNC(Cc2c(C)con2)=O)cc2c(cc1[N+](=O)[O-])N(C)CCO2 6737,Cc1[nH]nc2ccc(C(=O)NCC(C)CNC(=O)CCOC3CCOC3)c(Cl)c12 6738,C1(C(=O)NC2CCCN(C(c3cnn(C4CC4)c3)=O)C2)Cc2nncn2C1 6739,N1(C(c2coc3c2COC3)=O)CCCC(N=c2c(Cl)c[nH]cc2[N+](=O)[O-])C1 6740,C(=O)(C(C)(F)C(C)(C)F)N(CC=CC(=O)NC(C12CCC(CC1)C2)C)C 6741,CC(C)CC(C(=O)NC1CC(C)N(C(c2cc(C(N)=O)c[nH]2)=O)C1)C(N)=O 6742,N1(C(=O)CC2(O)CCOC2)CCCC1C1CCC1 6743,Cc1ccc(F)c(C(N2CC3CCC(C2)N3C(c2c(F)ccnc2Cl)=O)=O)c1F 6744,CC(C#N)C(=O)NCC(C1CCCCC1)NC(=O)CC1CSCCO1 6745,CN1CCN(C(c2ccnn2CCF)=O)CC1CNC(C12COCC1C2(F)F)=O 6746,C(C)(CCC(=O)NC12CC(C(C)(C)NC(=O)CC3CCC3)(C1)C2)OC 6747,C1(CC(c2ccc(-c3ccccc3)s2)=O)CCCCN1 6748,C(C(=O)N1CCC(C(=O)Nc2cncnc2N(C)C)C1)(C(C)C)NC(C)=O 6749,c1(N(c2ncnc(OC)c2C)C(c2ccccn2)=O)ccc2c(c1)CCNC2 6750,Cc1ccc(C(F)F)c(C(=O)NCC2CC(NC(C3(C)CC4CC4C3)=O)C2)c1 6751,CC(CCC(C)(C)C)C(=O)N1CC2CC1C2NC(=O)CNC(=O)CC(F)(F)F 6752,C12(C(N3CCC(N(C(c4cnc(C)nc4C)=O)C)CC3)=O)CC(C3COC3)(C1)C2 6753,C1(C(N2CCC(O)(CCNC(c3cc(Cl)cn3C)=O)C2)=O)(OC)CCS(=O)(=O)C1 6754,C1(C(=O)NC(CCNC(C(CC)(C)C)=O)Cc2ccccc2)CCOC(C)(C)C1 6755,c1(CN(C(C(=O)NC2CCN(C)C2)=O)CCC(N)=O)ccc(NC2CC2)cc1 6756,C1(C(N2CCC(NC(CC3CCC(C)C3)=O)C(F)C2)=O)Cc2ccccc2C1 6757,C1(CNC(C(C)=C2CC2)=O)CC(NC(c2cnn(CCC(F)(F)F)c2)=O)CC1O 6758,N1(C(CCN(CCOC)C(c2nc(C)ccc2C)=O)=O)CCC2(CCCN2C)C1 6759,c1(N(C)C)ccc(F)c(C(=O)NCCC2CCC(NC(C3C4COCC34)=O)C2)c1 6760,c1(CC=CC(C)NC(C(=O)N(CC(C)N(C(C)=O)C)C)=O)ccccc1 6761,CCC(C)C(C(=O)N1CCCCC1C1CCC1)N(C(=O)C(C1(O)CCCC1)F)C 6762,C(=O)(C1=CC2C=CC(C1)C2)NC1CC2(C(NC(c3n(C)cc(Br)c3)=O)C2)C1 6763,C(CC(=O)N1CC=CC1C(=O)NCC1(OC(C)C)CCC1)(C(N)=O)NC(C)=O 6764,C=CCCCCC(O)CNC(c1nc(CC)sc1Br)=O 6765,Cc1ccc(OCCCC(=O)NCC2CN(C(c3cocn3)=O)CC2O)cc1C 6766,c1(C(=O)NCC(CC)NC(c2cc(Cl)no2)=O)ccc(O)cc1F 6767,c1(C(N(CC(O)CNC(C2(CO)CCCO2)=O)C)=O)ccc(S(C)(=O)=O)o1 6768,C=CC(O)C(=O)N1CCC1CNC(c1cc(C2(C)CC2)n[nH]1)=O 6769,c1(C(=O)OC)ccc(S(=O)(=O)N2CCC(N)C2)cc1.c12ccc(cc1)c(=O)[nH]2 6770,N1(C(COC(CNC(CCC=C)=O)(C)C)=O)CC(COC)CC1(C)C 6771,C(CCN=c1[nH]ncs1)NC(C1CC(=O)N(Cc2cccc(Cl)c2)C1)=O 6772,C(=O)(C(C)(C)CC(C)(C)C)N1CC(CC)N(C(=O)Cc2cc(Cl)cc(Cl)c2)CC1 6773,C(CN=C(NCC(=O)N(C(C)C)C(C)C)NC1CCC(C)C1)c1ccc(C)cc1 6774,N1(C(C2C(C(N)=O)C2)=O)CCC(C2CC2NC(=O)CCc2ccccn2)CC1 6775,Cc1oc2ccccc2c1CC(N1CCC(NC(C2(CCF)CC2)=O)C(F)C1)=O 6776,C(=O)(CS(=O)(=O)CCC(F)(F)F)N1CCCC(NC(C(N2CC(C)C2)C)=O)C1 6777,C(=O)(NNc1ncnc2[nH]cnc12)c1[nH]cc(OC)c(=O)c1 6778,n1(CC(=O)NCCC(C(C)C)NC(C2CCC(C)(C)C2)=O)cc([N+](=O)[O-])cn1 6779,CC(CNC(=O)CSc1ccccc1)(CO)NC(c1cscc1C(F)F)=O 6780,c1(OC)cc(C(=O)NC(C)CN(C)C(c2ccnnc2O)=O)ccc1Br 6781,N1(C(CCOCCNC(=O)C=Cc2cc[nH]n2)=O)CCC(O)C(F)(F)C1 6782,CC(C(=O)N(CC(=O)NC1CCCN(C(=O)CCCCC2CC2)C1)C)S(N)(=O)=O 6783,CCCCCCC(=O)NC1CC(CCNC(c2cc(Br)n(C)c2)=O)C1 6784,C1(C(C)C)CCC(C)CC1C(=O)NC(CNC(C1(CCO)CC1)=O)C(C)(C)C 6785,N1(C(C2(OC)CN(C(=O)C(C)NC(=O)NC3CC3)C2)=O)CCC(O)C(F)(F)C1 6786,C(=O)(C1=NOC(C)C1C)N(C)CC1(O)CCN(C(c2c(OC)cncc2)=O)C1 6787,CCC(C)C(C(=O)NC1(C(C)O)CC1)N(C)C(C1CCCCN1C)=O 6788,c1(CN2CCC(CC(=O)Nc3cc(I)ncn3)C2)csc2ccccc12 6789,C=CCCC(C)NC(C1(CNC(c2occc2CSC)=O)CCC1)=O 6790,c1(OC)ccc(C(=O)NCC2(NC(=O)Cc3c[nH]nc3O)CCOC2)cc1OC 6791,C(CCCCC(=O)NCCCN(C)C(C1(NC(N)=O)CCCCC1)=O)=CC 6792,C1(C(=O)NC2(CCCNC(c3n(C=C)ncc3)=O)CC2)OCC2CCCCC12 6793,C1(C(N2C(C)CCCC2)=O)N(C(c2ccco2)=O)CCCC1(C)C 6794,c1(OC)ccccc1C1CC1C(N1CC(NC(C2COCCOC2)=O)C(C)C1)=O 6795,CC1(C)OC(=O)NC1C(N1CCC(CCNC(c2cnccn2)=O)C1)=O 6796,C1(C(N2CCN(C(C)=O)CC2C)=O)CCC2(CC1)CC2(F)F 6797,C1(NC(C(CC=CCC)C)=O)CC2(C1)CC(C(=O)NCC1CC1Cl)C2 6798,Cc1cc2ccc(C(=O)N(CC(C)N(C(=O)CCc3ccco3)C)C)cc2o1 6799,c1(C(C(=O)NCC2N(C(CCc3c(C)nn(C)c3)=O)CC2)O)ccc(Cl)cc1F 6800,c1(C(=O)NCCC2CN(C(=O)CC3CCCOC3)C2)cc2cccc(Cl)c2o1 6801,c1(CC(C)(C)CO)nc(C(C2CCCNC2)O)n(CCCO)n1.C1CC1 6802,CCC(CC(=O)NC1CC(CNC(c2ccn(C3CCOCC3)n2)=O)C1)C1CC1 6803,c1(C(=O)NC2CC(O)(CNC(C3CC3F)=O)C2)coc2c1C(=O)NCC2 6804,C1(NC(C(C2CCC2)NC(CC)=O)=O)CCCCN(C(=O)CCC=CC(C)C)C1 6805,C1(C)(NC(C(CCC)OC)=O)CCCN(C(c2c[nH]cc(Br)c2=N)=O)C1 6806,C(=O)(C1=C(C)OCCC1)N1C(CCCC)CN(C(=O)CC2CC3(CCC3)C2)CC1 6807,c1(CC(=O)NCCCN(C(=O)CSCc2ccccc2Cl)C)ccc(O)nc1 6808,CC1CCN(C(=O)CCOC2CN(C(c3ccc(C(N)=O)[nH]3)=O)C2)CCS1 6809,c1(CNC2(C)C(NC(=O)OCC)CCC2)cc(C)nc(C)c1.C123CC(C1)(C2)C(=O)N3 6810,c1(C(N2C(C(=O)NCCc3c(C)[nH]nc3O)CCC2)=O)ccc([N+](=O)[O-])cc1Br 6811,N1(C(C=CC2(C)CCOC2)=O)CCC(NC(c2cnn(C3CCC3)c2)=O)C12CC2 6812,CCCCCCCCCC(=O)N1CC(CNC(=O)CC(C)(C)COC(C)=O)C(C)C1 6813,C12CCCCN1Cc1cn2nn1.C1(NC(=O)Nc2cnccn2)COC2CC1C2 6814,C1(NC(c2c(OC)noc2C)=O)CCCCN(C(=O)CC(C)c2cccnc2)C1 6815,C(C1C(C(=O)NCC2(F)CC(NC(c3cnsn3)=O)C2)C1(C)C)=C(C)C 6816,C12(F)CCCN(C1)C2=O.c1(NC(Cc2ccc(C)nc2)=O)ccc(Cl)nc1C 6817,C1(CC(=O)Nc2cccc(CNC(=O)C(F)(F)C(F)F)c2)CCS(=O)(=O)CC1 6818,C1(O)(CC(=O)NCC(CNC(c2c(C)nc(C3CC3)[nH]2)=O)(C)C)CCCCCC1 6819,C1(N(C(c2cnc[nH]c2=N)=O)CC)(CO)CCN(C(C)=O)C1.C(=O)C1CC1 6820,c1(OCC(=O)NCC2CCCN2C(=O)CC23CCCC2C3)ccc(C(F)F)nc1 6821,c1(SCCC)ccc(C(=O)NC2CCC(NC(C3CC(CC(F)F)C3)=O)C2)cc1 6822,C(=O)(C1=CCCCC1P(C)(C)=O)NCCC1N(C(COCC=C)=O)CCOC1 6823,CCC(CC(=O)N1CCC(C)(NC(=O)CCc2ccc(Br)cc2)C1)OC 6824,N1(C(c2cccc(CC)n2)=O)CC2CC1CC2N1CC(C(N)=O)(C(N)=O)C1 6825,CC1COC(C(=O)N(C2CN(C(=O)C=CC(=O)NC3CC3)CC2O)C)CO1 6826,c1(C(=O)NC2CCC(NC(CC=C(C)C)=O)C2)ccc2c(Br)n[nH]c2c1 6827,c1(C(=O)NCc2cccc(C(N(CC(C)C)CC)=O)n2)cccc2ccoc12 6828,n1(CC(N2C(C)C(NC(C3CC3(Cl)Cl)=O)CC2)=O)ncc(O)nc1=O 6829,c1(NC2(NCCNC(=O)C=O)CC2)ccc(Cl)cc1.c1(CSC)ccccn1 6830,C(=O)(CCCCC(C)(C)C)N(CC(CC)NC(=O)CCc1cncc(O)c1)CC 6831,n1(CCC(=O)NC2C(CNC(c3c(C)ocn3)=O)CCC2)c(C)cc(O)cc1=O 6832,CCCCCC(C)(C)C(=O)NCC(C)NC(=O)Cc1cccc(F)c1 6833,c1(N2CCC(CC(=O)NCCC=C)C2)cc(OC)nc(OC)n1 6834,C1(NC(CNC(=O)OC)=O)C=CCN(C(C2CNC(=O)N2)=O)C1 6835,N1(C(COC)=O)CCC2(CCCN2C)C1.C1(C)C(=O)N(C)C2CC(C2)O1 6836,C1(CCNC(c2ccc(Cl)o2)=O)CCCN(C(c2cc(O)ncn2)=O)CC1 6837,C1(COC)(NC(c2cc(Cl)c[nH]2)=O)CCN(C(=O)Cc2ccc(F)cn2)CC1 6838,c1(CC(=O)N(CC(C)(C)NC(C(C)NC(=O)NC)=O)C)ccc2c(c1)CCCS2 6839,N1(C(C(C)OCCC=C)=O)CC(NC(C2(O)CCSCC2)=O)CC2(CC2)C1 6840,N1(CC(=O)NC(C(=O)Nc2cccc(C)c2)C)C(=O)c2cc(Cl)c(Cl)cc2C1=O 6841,C(=O)(CS(=O)(=O)C(C)(C)C)NC1C2CN(C(Cc3cccc(OC)c3Cl)=O)CC21 6842,c1(C(=O)OC)ccc(S(=O)(=O)N2CCC(O)(C(C)NC(=O)C(C)CO)C2)c(F)c1 6843,C1(CCN(C)C)C(=O)N2CC(C(C)C2)CN1.n1(CC(=O)C(C)C)cc(C2CC2)cn1 6844,N1(C(CNC(CNC(C)=O)=O)=O)C2CCC1CC(NC(=O)CC1CCCOC1)C2 6845,N1(C(C(=O)N(C)CC)C)CCC(C(=O)Nc2nccn2C)CC1 6846,c1(C(CNC(=O)C(C)O)NC(c2ccsc2)C)ccc2ccccc2c1 6847,C1(CC)CN(C(=O)C(CCOC)OC)CC1NC(=O)CC=C(C)C.OC 6848,c1(C(=O)NCC2OCC(CNC(CC(=C=C)C)=O)C2)ccc(Cl)c(CCC)c1 6849,C1(CC(=O)NC(C(=O)NCc2nc(CC)sc2)C2(O)CCC2)C=NN(C)C1=O 6850,N1(C(C2(C#N)CC=CC2)=O)CC(NC(C2CC(F)(CO)C2)=O)C(N=[N+]=[N-])C1 6851,CCC(CCO)NC(=O)CN(C(=O)C(c1cnn(C)c1)O)C 6852,c1(OCC(CN2C(C(=O)NCc3cn(CCC)nn3)CCC2)O)cccc(C)c1 6853,N1(C(c2cc(CC)on2)=O)CCOCC2CN(C(C3CC3(F)Cl)=O)CCC12 6854,C1(C(=O)NCC(=O)OCC=C)CC2CCC1N2C(C1CC(=O)C1)=O 6855,N1(C(c2cc(OC)no2)=O)CCCN(C(=O)C2=CCC(C)CC2)CC1CO 6856,C(=O)(C1=CCN(C)C1)N(CC(CNC(C=Cc1c(C)n[nH]c1)=O)(C)C)C 6857,C(=O)(CC(C)CC(C)(C)C)N1C2CC(NC(CC(C)C)=O)C(CC2)C1 6858,c1(CCC(=O)Nc2cnn(C(F)(F)F)c2)nnc(COCCO)o1 6859,C1(C)(NC(CC(C(C)C)O)=O)COCCN(C(=O)CSc2nncn2C2CC2)C1 6860,C(C(CNC(c1ccc([N+](=O)[O-])[nH]1)=O)C(F)(F)F)NC(C1N(CC)CC1)=O 6861,Cc1ccc(C(C)(C)F)cc1NC(c1cc(F)ncc1F)CCl 6862,C(=O)(C(C)C(C)(F)F)NC1CCN(C(c2ccn(C(C)C)n2)=O)C1 6863,C1(C(N(C)CCNC(c2ccn(C(F)(F)F)n2)=O)=O)CC2(C1)CC(F)C2 6864,Cc1ccc(C(=O)NC(C2CCCC2)CNC(c2cnsn2)=O)c(C2CC2)n1 6865,NS(=O)(=O)C1(C(=O)NC2CC(NC(=O)C=Cc3cocn3)C23CCC3)CCC1 6866,CN1C(=O)CCC1C(=O)NCC1CCCCC1NC(c1cccc(C2CC2)c1)=O 6867,CC(CCCCN=c1[nH]c2cc(Br)cnc2s1)NC(c1cnc2c[nH]nc2c1)=O 6868,N1(C(C2CN(C(=O)OC3CC3)C2)=O)CCC(C(=O)NN2CC3(CCC3)C2)CC1 6869,CC1CCCC1N=c1[nH]c(N2C3CCC2COC3)nc2c1CCCC2 6870,C12C3C4CC5C1C3C45NC2=O.Cc1ccc(CN(C)CCN(C)C)cc1 6871,C(=O)(CCC(C)(F)F)N1CC(CN(C(=O)CSC(C)(C)C)C)OCC1 6872,C12CCN(CC1)C2.N1(CC=CC(=O)NC(N)=O)CCOCC1 6873,c1(C(N2CCC(C(=O)Nc3c(C#N)ccs3)CC2)=O)cccn2c(O)nnc12 6874,N1(C(CC(C)F)=O)CCC2(CC(C(=O)Nc3ccccc3C3CC3)C2)C1 6875,C1(C(=O)NCC2(CC)CC2)(NC(=O)CC2(C)CC2)CCC(C)(C)C1 6876,c1(C(=O)NC(CNC(C(C(=O)OC)C)=O)(C)C(C)C)cccc2ncnn12 6877,C(C(=O)NCC1CCN(c2cc(C)nc(C(F)(F)F)n2)CC1C)(C(C)(C)C)OC 6878,CC1(C)C(C)(C(=O)NC2CCC(NC(=O)CC(=O)NC3CC3)C2)C1(C)C 6879,Cc1cc(=NCC2CC(NC(=O)C3COc4ccccc43)C2)[nH]c(S(C)(=O)=O)n1 6880,C(C(F)C=O)C1CN(C(N)=O)C1.C(CC(C)C)NC(C1(OC)CC1)=O 6881,C1(NC(C2C(C)OCC2)=O)CN(C(=O)C=Cc2ccc(O)cc2)CC1(C)C 6882,C(CC(N)=O)(C(=O)N1CCNC(=O)C1)NC(C1OCCN(C)C1)=O 6883,C1(C)(C(=O)NCC2CCC(F)(CNC(c3cc(OC)no3)=O)C2)CC2CCC1C2 6884,CC1COCC(C(=O)NC2(C(N3CCN(CC(N)=O)CC3)=O)CCN(C)C2)O1 6885,N(C1CCC2(CC2)Oc2ccccc21)C(=O)NCCN(C)Cc1cccc(C)c1 6886,c1(SCC)cc(Cl)ccc1C(=O)NC1CCC(NC(=O)C(C)n2cccc2)CC1 6887,N1(C(C2(c3cccc(-c4cccc(C5CC5)c4)c3)CCCC2)=O)CC(O)C(O)C1 6888,CC1(C)CC(CC(=O)NC2CN(C(=O)CCF)CC2(C)C)NC1=O 6889,N1(C(c2c(CC)nn(C)c2)=O)CC(F)(F)CC1(C)CNC(c1ccnn1CC)=O 6890,C1(NC(c2c(C)nccn2)=O)CCCC12CCN(C(=O)C1=CCS(=O)(=O)C1)C2 6891,Cc1nc(S(=O)(=O)CCN(CCC(F)(F)F)CCOC(=O)C(C)CCO)cn1C 6892,C(=O)(C1=CCCCCC1)NC1CC(F)(CNC(=O)CC2CCCNC2=O)C1 6893,CCCCCC(O)CC(=O)NCC(C)N(C)C(c1ccnc(F)c1Cl)=O 6894,C1(NC(C2N(C)CCC2)=O)CCC2CC1CN2C(c1cnn(C)c1)=O 6895,C(CC(C)(C)CNC(=O)CCC1CCN(C(=O)C(CO)NC(N)=O)C1)OC 6896,N1(C(c2c(C(N(C)CC)=O)cccc2)=O)CCCC2(CCCO2)C1 6897,c1(NC)ccc(Cl)c(C(=O)NCCN(C(=O)Cn2nc(C)cc2C)C)c1 6898,CC(C)(CCC(=O)NC1CCC(NC(c2cnc(N)cn2)=O)CC1)[N+](=O)[O-] 6899,CC1(C)CCC(CNC(=O)C(CNC(=O)C(F)=CC2CC2)CC2CC2)O1 6900,N1(C(C=CCCC)=O)CCCC2(C1)CN(C(=O)Cc1nc(C)c(C)[nH]1)C2 6901,C1(NC(C2(C)CCCN(C)C2)=O)CCCCCN(C(c2ccsn2)=O)C1 6902,c1(C(N(CCNC(C(CC)(C)OC)=O)C)=O)cc(N)cc(C)c1F 6903,c1(CC(=O)NCC(C)NC(c2c(CC)nccn2)=O)c(C)nn(C)c1C 6904,N1(C(C2(C(C)NC(C(C)SCC)=O)CC2)=O)Cc2c[nH]nc2C1 6905,C12(NC(C3CCCCC3)=O)CCCC1N(Cc1cscn1)CC2 6906,c1(C(N2CCC(NC(c3ccc(Cl)cn3)=O)C(F)C2)=O)cccc2c1OCC2 6907,C1(C(=O)NC(CCN(C(COCC)=O)C)C(C)C)CC2(C1)C(F)(F)C21CC1 6908,N1(C(C(C2CCCC2)OC)=O)CCC(NC(=O)C(N)=O)C(C)(C)C1 6909,C1(NC(c2c(COC)ncs2)=O)CN(C(C2COCCN2C)=O)CCC1O 6910,C1(C2CC2)(NS(N(C)CCOC)(=O)=O)CCCCCC1 6911,C1(CNC(c2n(C=C)nnc2)=O)CCN(C(c2ccc(F)cc2C)=O)CC1C 6912,N1(C(c2n(CC)ncc2)=O)CCOC(C)C1C(N1CC2(CO)CC2(CO)C1)=O 6913,C(CC(=O)NOCCCOC)(C(F)(F)F)NC(C1(CC)CCOCC1)=O 6914,c1(C(=O)NCC(CC(C)C)F)ccccc1S(=O)(=O)C(C)C 6915,N1(C(c2c(C)nn[nH]2)=O)CCN(C(=O)Cc2ccc(Cl)s2)C(C)C1C 6916,CC1CCN(C(=O)C(O)Cc2cn(C)cn2)C(CNC(c2cn(C)nn2)=O)C1 6917,N1(C(c2ccc(C3CC3)cc2)C(=O)O)CCN(CC2(c3nn[nH]n3)CCOC2)CC1 6918,CC1(C)CCC(NC(C2CC2CNC(=O)CC2CC3C=CC2C3)=O)CC1 6919,C1(NC(C2C(C)C2C)=O)CN(C(=O)CC2CC3(CCO2)CC3)C2(CCCC2)C1 6920,Cc1ccc(Br)cc1NC(Cc1cnn(C)c1)C(=O)O.C1(C)C(=O)N1 6921,C(=O)(C(C)(C)COC)NCC(CC)NC(c1cccc(F)n1)=O 6922,C(=O)(CN=c1cc[nH]cc1)N(CCOCCC(=O)NC(C)CCn1cncn1)C 6923,Cc1cnc(O)c(NC(C2(O)CCN(Cc3ccc(Br)c(O)c3)C2)=O)c1 6924,N1(C(CCCC(C)c2cn(CC)nn2)=O)CCC2COC(=O)NC2C1 6925,C(=O)(CC1CCOc2ccccc21)N(C(CCNC(CC(=O)NCC)=O)C)C 6926,c1(OC)cc(C(=O)NCC=CCNC(=O)CCc2cnccn2)n(C)n1 6927,CC1CN(C(c2cn3cccnc3n2)C(=O)NCC2CCCO2)CC(C)(C)S1 6928,N1(C(CCCCOCCC=C)=O)CCN(C(=O)CCC(C)SC)CC1CC(F)(F)F 6929,C1(COC)(CN(CC(=O)NC2(C)CCOC2)C)CCCC1 6930,N1(C(C(CCNC(Cc2c(C)noc2C)=O)(C)C)=O)CCC2(CCC2)C(O)C1 6931,C(C)(C(=O)N1CC(C(C(=O)N(C2(CCCCO)CC2)C(C)C)OC)C1)SCC 6932,C1(F)(C(=O)NCC2(CNC(c3c[nH]nc3F)=O)CC2)CCOCC1 6933,CN1CC(NC(C2CCC3(CC3)N2C(=O)CC2C=CCC2)=O)C2(CC2)C1 6934,Cc1cccc(OCC(=O)NC2(CO)CCN(C(c3nc(=O)n(C)[nH]3)=O)C2)c1F 6935,CN(C1CCCc2ccc(Br)cc21)CCCCCNC(c1cnn(C)c1C#N)=O 6936,S(=O)(=O)(c1cccc(F)c1)N1C(C(N2CCCN(C(=O)CO)CC2)=O)CC(F)C1 6937,CC1(C)CCN(C(C2(O)CCCCC2)=O)CC1CNC(c1c[nH]nc1F)=O 6938,C1(CN(C(=O)C(O)COC)CC)CCCN1C(c1cnn(C(F)F)c1)=O 6939,N1(C(CCOCCOC(C)(C)C)=O)CCC(NC(=O)C=CC(F)(F)F)C1 6940,c1(Cc2nc(CCC)nn2-c2ccnc(C(F)(F)F)c2)ccnc(O)c1Br 6941,c1(OC)c(Cl)cc(NC(C2CC(O)CN2S(=O)(=O)c2cccs2)=O)cc1Cl 6942,Cc1cnc2n1CCCC2C(=O)N1CCN(C(C2C=CC=CC=C2)=O)C(CO)C1 6943,CC(C)C(N=[N+]=[N-])C(=O)N1CCC(C)(NC(c2ncn3ccccc23)=O)C1 6944,C(C)(CNC(=O)CCc1cscn1)(CO)NC(C(C)C1CCCC1)=O 6945,Cc1nc(Cl)[nH]c(=NCC2CCC(NC(=O)CC3COCC(C)(C)O3)C2)c1F 6946,c1(C(C(=O)N(CCNC(c2csc(S)n2)=O)CC)C)c(C)n[nH]c1C 6947,N1(C(C(C2CCN(C(c3ccnc(Br)c3)=O)CC2)C)=O)CCc2ncccc2C1 6948,C1(O)(CCNC(C(CC=C)C)=O)CCCN(C(c2cc(C(N)=O)[nH]n2)=O)C1 6949,C(=O)(CCC(C)(F)F)NC(CC(=O)NC1(C#C)CC1)COC 6950,CC(C)(C(=O)NCC=CC(=O)N(C1CC(C#N)C1)CC1CC1)C1CCCC1 6951,c1(NC(C)CNC(=O)C(F)(F)c2cncs2)ncc(F)cn1 6952,Cc1[nH]nc(C(N2CCC(N(C(=O)C(C)CO)CCO)CC2)=O)c1[N+](=O)[O-] 6953,n1(CCCC(C)O)cc(C#CCNC(=O)CNC(=O)OC(C)(C)C)nn1.C1CO1 6954,N1(C(C(C)(C)c2cnsc2)=O)CCC(F)(CNC(C2CCC(F)CC2)=O)CC1 6955,C1(NC(=O)NCC2(CCOC)CCC2)CCC(C)c2ccccc2C1 6956,CC1CC(F)(F)CN1C(C1(NC(=O)C(O)C2CCCC2)CCSC1)=O 6957,CC(C)C(F)(CNC(=O)C1=CCCC1C)C(=O)NC(C)(C)C(=O)NC(C)(C)C 6958,c1(OC)cc(N2CCC(NC(C3(C4CCOCC4)CC3)=O)C2)c(F)cc1[N+](=O)[O-] 6959,C1(C(=O)NCC2(OC)CCCCC2)CN(C)CCN1C(c1cc(C)n(C)c1C)=O 6960,C1(C(=O)NC2(CC#N)COC2)CC(C)(C(=O)NC2CC2)C1 6961,C1(NC(C#CC(=O)N(C)C)=O)CC(F)(F)CC1NC(=O)CC1CCCC1 6962,N1(C(c2ccc(C#C)cn2)=O)CC2(CCN(C(=O)C(C)(CC)CO)CC2)C1 6963,Cc1ccc(F)cc1CNC(=O)C(F)C1CC(NC(c2cc(=O)n(C)cn2)=O)C1 6964,O=C(CCC(=O)NC1C(NC(c2ccns2)=O)CCOC1)Nc1cccs1 6965,N1(C(c2c(C)nns2)=O)CC(NC(c2occc2F)=O)CC(O)C1 6966,Cc1cc(C(=O)NC2(CNC(=O)CCN3CCCC(C(N)=O)C3)CC2)sc1Cl 6967,c1(OC)c(C(=O)NC(C)(C)CCCNC(C2CCC(=O)O2)=O)cc(F)cc1F 6968,C1(C)(CNC(C(C)SCc2cccc(C)c2)=O)CN(C(=O)C(C)(F)F)CCO1 6969,Cc1c(F)ccc(F)c1CN1CCC(O)(CC(N2CCC(C)CC2)=O)CC1 6970,N1(Cc2ccc(C(=O)OC)[nH]2)CCC(CO)(NC(c2cccc(=O)n2C)=O)CC1 6971,Cc1c(Cl)ccnc1NNC(=O)CN1CCCCC1 6972,n1(CC)nc(C)cc1C(=O)NC1C=CCN(C(c2ncoc2Br)=O)C1 6973,c1(CCC)c(C(N2CCCC2CNC(c2nccnc2N)=O)=O)nnn1CC 6974,C1(CNC(=O)NC2C3(CCN(CC(=O)N(C)C)CC3)C2)CCC2(CCCC2)CC1 6975,n1(C(C(=O)NCC(C)NC(=O)CC2C=CCCC2)C)ccc(Br)n1 6976,c1(C(N2CC(NC(CCOC(C)=O)=O)C2)=O)cc(F)c(Br)cc1F 6977,N1(C(CC2(OC)CCCC2)=O)CCN(C)CC1CNC(=O)CC(C)CN(C)C 6978,C1(C(=O)NC(C2CCCC2)CC)CN(C(c2[nH]ccc2C2CC2)=O)CCN1C 6979,c1(CC(=O)NCC(C)(O)CNC(C2CC(=O)NC2=O)=O)c[nH]c2c(F)cccc12 6980,Cn1cc(Br)cc1C(N1CC2CC2C1CNC(=O)CCn1cncn1)=O 6981,C1(c2n(-c3c(SC)cccc3)nc(-c3cncnc3)n2)CC(=O)NC1(C)C 6982,c1(C2(NC(=O)NCC(F)C3CCC3)CCC2)ccccc1 6983,C1(CNC(C=CCOC)=O)CCN(C(c2ccc(F)cc2Br)=O)C1(C)C 6984,C(C(CC(=O)NCC(O)CNC(c1ccc2ccnn2c1)=O)C(F)F)N(C)C 6985,C1(N(C)C)CCC(C(=O)NC2CC(F)(CNC(=O)CC3COCCO3)C2)CC1 6986,C1(NC(Cc2cc(C)c(Cl)cc2)=O)COC2C(NC(C3(C)CCCC3)=O)COC12 6987,c1(OC)cc(CN=[N+]=[N-])ccc1Nc1ccc(N2CCCC(C)C2)nn1 6988,N1(CC=C)CC2(COC(CN(C(=O)CC3(c4c(C)noc4C)CC3)CC)C2)C1 6989,C(=O)(C(O)CCCNC(C1CCCSC1C)=O)NCc1cc(C)ns1 6990,CC(CCP(C)(C)=O)(c1nnnn1C1CCCC1)NCC(CO)SC(F)F 6991,N1(C(CC(C)C)=O)CCCC(NC(=O)C(F)(F)C2(N(C)C)CCC2)CCC1 6992,c1(CC(C(=O)O)NC(C(N2CC3CC3C2)C)=O)ccc(Cl)nc1 6993,N(C(=NCC1(CC)CCCC1)N1CCC(n2cc3cc(F)ccc3n2)C1)CCC 6994,C(C)(CCCC(=O)NC(c1cn(C)nn1)C)NC(c1c(C)cccc1)=O 6995,C1(CC(N)=O)CCCN1C(=O)CCC1CCN(C(=O)CC2CCCSC2)C1 6996,C=C1CC2CCC(C1)N2C(=O)C(C(C)CC)N(C)C(c1ncc(F)cc1F)=O 6997,c1(C(N(C)CC2N(C(c3c(C)ncnc3)=O)CCOC2)=O)cc(O)cc(O)n1 6998,CC1CC(NC(c2ccccc2C2CC2)=O)CN1C(=O)CC1CCOCC1 6999,Nc1cc(C(N2CC(F)(CNC(C3C(F)(F)C34CC4)=O)C2)=O)c(F)cc1F 7000,C1(CNC(CC(CC)OC)=O)CCC2(CCC2)CN1C(C1CC1C1CCC1)=O 7001,C1(NC(C(C)C(C)(C)C)=O)CCN(C(c2cnc3[nH]cncc2-3)=O)CC(C)(C)C1 7002,N1(C(C2N(CC)CCC2)=O)CCN(C(c2c(Cl)cnn2C)=O)CC1CC(=O)NC 7003,c1(C(N(c2ncc(C(F)(F)F)cn2)C2C(C)CNC2)=O)ccc2sccc2c1 7004,c1(C(N2C3CCC2CC3)=O)cc(NC(c2scc(C(=O)OC)n2)=O)n(C)n1 7005,CC1(C)CN(C(c2cccc(C3CC3)c2)=O)CC1CO.C12C=CC(C1)CNC2=O 7006,C(=O)(C(C1=NOC2CC12)N(C)Cc1ccc2c(c1)CCO2)NCCCOC 7007,N1(C(C2CC3(CC(NC(CC)=O)C3)C2)=O)CC2(CCC2)CC1CO 7008,Cc1cnoc1C(=O)NCC(C1CCCN1C(=O)CCSCC(C)C)(C)C 7009,N1(C(CC(CC)SC)=O)CCC(CNC(c2cnc(O)c(F)c2)=O)C(O)C1 7010,C12(NC(C(C)CN(C)C)=O)CCOC(CNC(c3ncccc3C(F)F)=O)(C1)C2 7011,c1(C(=O)NCCC2CCN(C(c3cnns3)=O)C2)csc(Cl)c1Cl 7012,c1(CNC(c2c(NC(CC(=O)OC)=O)ccs2)=O)ccc2c(c1)COC2 7013,C(CS(=O)(=O)CC(=O)NC1CCCN(C(c2cc(C)co2)=O)C1C)OC 7014,N1(C(CN2CCC(C)(O)C2)=O)CCN(C(=O)C(C)(C)O)CC12CCC2 7015,c1(CC(=O)N(C)CC2N(C(CCCCSC)=O)CCC2)cccc(F)c1O 7016,C(CNC(C1C2COCC12)=O)(CC(F)(F)F)NC(c1c(SCC)nccn1)=O 7017,C(=O)(C(C)CS(C)(=O)=O)N1CCC(NC(c2sc(CC)c(C)c2)=O)C1 7018,CC(C)(C(=O)NCCCCNC(C1(c2ccc(Cl)nc2)CC1)=O)C(F)(F)F 7019,N1(C(CSCCCC)=O)CCOCC(F)(CNC(=O)C=Cc2cnc[nH]2)C1 7020,CCC(C)(C#N)C(=O)NC1(CNC(=O)Cc2cnn(C(F)F)c2)CCC1 7021,S(=O)(=O)(c1ccc(C(C)(C)C)cc1)NC(C(=O)Nc1cc(C)c(F)cc1)C 7022,C1(C)(NCCCC(=O)NC(C(C)C)CNC(c2cn(C)nc2O)=O)CC=CCC1 7023,C1(CNC(c2cnc(SC)s2)=O)CCCN(c2cc(-c3ccccc3)ncn2)C1 7024,N1(C(CC(C)OC)=O)CCC2(CC1)CN(Cc1ccc(Cl)cc1C)CCO2 7025,c1(NCC(=O)OCc2ncccc2Cl)ccccc1Cl 7026,C1(NC(C2CCCS2)=O)CCSC12CN(C(=O)CCc1nc3ncccn3n1)C2 7027,CC#CCCCC(=O)NCC1C=CCN1C(c1ccc(CCC)c(N)c1)=O 7028,c1(N(C)Cc2cccc(OC)c2)nc(N2CCC(S(C)(=O)=O)C2)c2c(n1)COC2 7029,Cc1cc(=NCc2nnnn2-c2cc(C)n(C)n2)[nH]c(N2CCC(CO)C2C)n1 7030,n1(CC)cc(CC(=O)NC2CCCC2)cn1.C12CC(C1)CCNC2=O.C(C)C 7031,c1(CN2CCC(C(=O)NC(C(=O)OC(C)C)C)C2)cc(Br)ccc1F 7032,Cc1onc(C(=O)NC2CC2c2cnc(N(C3CCCC3)C(C)(C)C)nc2)c1Br 7033,C1(CNC(C(=O)NC(C)C)=O)COC(C)(C)CN1C(=O)Cn1cccnc1=O 7034,c1(-c2n(CCCCC)nc(CC(C)(C)CO)n2)ccnc2cc(Br)ccc12 7035,C(=O)(CC(CC)C(C)C)N.CCC(CCc1ccccc1)n1cc(-c2cn[nH]c2)nn1 7036,Cc1oc(C)c(C(=O)NC2CC2CNC(=O)C(c2cccc(O)c2)C)c1C 7037,C1(C(=O)NC2CC(N(C(CSCCCC)=O)C)C2)CCc2nc(O)[nH]c2C1 7038,c1(OCC(=O)NCC2(NC(c3cc(C4CC4)cs3)=O)CCOC2)cccnc1 7039,Cc1nn(C)c(C)c1OCC(=O)NC1CC(CO)N(C(=O)CC2(C(F)F)CC2)C1 7040,C1(CC=C)(NC(C2CCCC2)=O)CCCN(C(c2cc(C(=O)OC)c[nH]2)=O)C1 7041,C12CN(CCC1(F)F)C2=O.c1(C(=O)OCC)cnc(Nc2sccc2I)nc1 7042,c1(CN2C(C(N3CCC(F)(F)C3)=O)CSCC2)cnc(Cl)cc1Cl 7043,C1(NC(CCNC(=O)CCN2CCC(O)CC2)=O)CCCC2NCCC12 7044,C1(Cn2cc(-c3n(C)ncc3)nn2)CN(C(c2nc(Br)cs2)=O)CCO1 7045,Cc1cnncc1C(=O)NCC(C)(C)CN(C(=O)COCC(=O)N(C)C)C 7046,N1(C(Cn2c(C)cnc2)=O)CCOC(C(C)NC(c2ccc(Cl)cn2)=O)C1 7047,c1(CCNC(=O)NC(CC(=O)OC)C2CCCCC2)nccc(C(F)(F)F)n1 7048,N1(CC)CC(C(=O)N(C)CCC2CCCCN2C(=O)CCSC)CC1=O 7049,C(=O)(CC(C(=O)NC1(C)CN(C(c2scnc2C(C)C)=O)C1)N(C)C)OC 7050,C1(C(N2CCC(NC(C=NOC)=O)C2(C)C)=O)CCc2nccn2C1 7051,N1(C(CCOCCC)=O)CCC2C(NC(C3CCC(NC(=O)N(C)C)CC3)=O)C12 7052,C#Cc1ccc(C(N2CCC(c3n[nH]c(CNC(=O)C(O)C(C)C)n3)C2)=O)nc1 7053,C(=O)(C1CCc2c[nH]nc21)N1CC(C(C(=O)NCc2cnccc2Cl)OC)C1 7054,C1(CCCCC)CCC(C(N2CCN(C(=O)CC3CCCCO3)CC2)=O)CC1 7055,CN1CCN(C(C2C3CNC(=O)C23)=O)C(CNC(=O)COC(F)F)C1 7056,C(CCCC(=O)NCC(C)(C)C1CCCO1)N(C(=O)CNC(N)=O)C 7057,C1(CCNC(C(C)OCOC)=O)CCN(C(c2ccncc2)=O)CC1 7058,Cc1cc(C)c(C(N2CC(CNC(c3ccon3)=O)C(C)C2)=O)cn1 7059,C1(C(=O)NC(C)(C(=O)NC2COC3(CCC3)C2)C2CCC2)CC(=O)CC(=O)N1 7060,CCC(C)(CNC(C1CN(S(=O)(=O)CC)C1)=O)NC(=O)C(C)(C)c1csc(C)c1 7061,c1(OC)cc(CC(N2CCOC(CNC(c3ccc(C#N)s3)=O)C2)=O)ccc1C 7062,N1(C(C(C)OC)=O)CC2CN(C(C)=O)CC12.c12ccc-1cc2 7063,c1(C(=O)NC2CN(C(c3cc(C)cc(O)n3)=O)C(C)CC2)[nH]cc2c1CCCC2 7064,C1(C(=O)NCC2C(C(N3C(C#C)CCC3)=O)C2(C)C)CC2COCC2C1 7065,c1(CNC(C(CC)C)(C)c2nnnn2CC2CC2)cn2c(C)cccc2n1 7066,C(=O)(C(F)(F)C(F)(F)F)NCC(C)(C(C)C)NC(c1ccnc(C)c1C)=O 7067,c1(C(=O)NC2CC(CCNC(C(CC)NC(C)=O)=O)C2)[nH]c(=N)ccc1C 7068,N1(C(C23CN(C(c4nncc(OC)c4)=O)C(C2)CO3)=O)CCCCCCC1C 7069,N1(C(C(C)OCOC)=O)CC(C)(C)OCC1CNC(c1cnsc1)=O 7070,c1(NCCC(N2CC(OCC)(CO)C2)=O)c(F)cccc1Cl.C12(CC1)C(=O)NC2 7071,O(NC(=O)C(c1cccs1)NC(c1coc(SC)c1)=O)CCCC#C 7072,C(C)(CO)(C(=O)NCc1nc(C)c(C)s1)NC(c1[nH]cc(C(C)=O)c1)=O 7073,N1(C(c2nc(NC)sc2)=O)CCC2(CCCN2C(C2(O)CCC(C)(C)CC2)=O)C1 7074,c1(OC)nccc(CNC(C2COCC2NC(c2csc(C)c2C)=O)=O)n1 7075,N1(C(C(C2CCN(C(c3cnc(C#N)s3)=O)C2)C)=O)CCOC(C2CCC2)C1 7076,c1(C(C(N2CCC(NC(C(C)OC(C)(C)C)=O)C2)=O)(C)C)cc(Cl)cc(Cl)c1 7077,C(CN=C(NCc1c(F)cccc1Br)NCC1CCN(C)C(=O)C1)SC 7078,c1(C(N2CC(NC(CCc3n(C)cnn3)=O)C3C2C3)=O)cc2sc(Cl)cc2s1 7079,N1(C(c2n(C)ncc2)=O)CCC(NC(=O)Cc2c(O)ncnc2O)CC(C)(C)C1 7080,CCC(O)C(C)(C)C(=O)NC1CCCC(CC(=O)NCC(O)(COC)CO)C1 7081,N1(C(CN(CCC#C)C)=O)CCCOC(CNC(=O)Cn2ccc(C)n2)C1 7082,Cc1c(C(C)NC(C2(c3ccccc3)CCOC2)C)cnn1-c1ccccc1 7083,C(=O)(C1=CS(=O)CCC1)NC1CN(C(C2CN(CCCCC)C(=O)C2)=O)CC1C 7084,c1(OC(C)C)cc(-c2cncnc2C(N2CCOC(C(F)(F)F)C2)=O)ccc1C 7085,CCC(C)(C)CCCC(=O)NCC1CCN1C(c1cc(C)cc(OC)c1N)=O 7086,c1(CC(=O)N(CC(C)CNC(C2CC2C2CC2C)=O)C)noc2ccccc12 7087,N1(C(CCOCCC)=O)CCC2CCCC12C(=O)NC(CO)C(C)(C)CO 7088,C1(C(=O)NCC2N(C(C3N(C(CC)=O)CSC3)=O)CC2)CC(S(C)(=O)=O)C1 7089,S(=O)(=O)(c1ccn(-c2ccc(F)cc2)n1)NC1C([N+](=O)[O-])CC1 7090,O=C(N=c1ccn(CCC(=O)N2CCC2C(F)(F)F)[nH]1)c1ccnc(F)c1 7091,C1(N(C(CN(C(=O)CCOC(C)C)CC)=O)C)CC2CCC1O2 7092,n1(C(C)C)cnc(C(=O)N(CCNC(=O)C(c2cnn(C)c2)C)C2CC2)n1 7093,C(=O)(C(CCC1CCC1)NC(=O)CN1CCOCC1)NC1CC(C)(C)C1 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7164,N1(C(C(C(C)C)C2CCC2)=O)CCC(NC(=O)CCC2(C)CC2(F)F)C12CC2 7165,n1(CC(N2CC3(C2)C(=O)N3)=O)cccnc1=O.C1(COC)CCC(CO)C1 7166,C(=O)(C(C#N)C(C)(C)C)NC(CCC(=O)NC1CC(OCC)C1)C 7167,C(C(C)N=c1[nH]c2c(c(=NCC=CCl)[nH]1)COC2)c1cc(C)[nH]n1 7168,n1(C(C(=O)C(=O)C(N2CCSCC2)C)C)cc(-c2ncccn2)nn1.CCC(C)(C)N 7169,CCCCS(=O)(=O)NC(C)C(=O)OCCc1ccnc(C)c1 7170,CCC(C)(CO)C(=O)N1CCC(C(C)NC(c2cccc(C3CC3(F)F)c2)=O)C1 7171,C1(CCOC)(C(=O)N(C2CCCN(C)C2)C)CCN(C(=O)C(F)C(C)C)C1 7172,c1(C(=O)NCC2N(C(CC(CC)CN(C)C)=O)CC2)ccn2ncnc2c1 7173,C1(NC(CC=C(C)C)=O)CCCCN(C(=O)CCc2cccc(OC(F)F)c2)C1 7174,C1(C)(OC)CCC(NC(C2C3CC4C(C3NC(C3CCNC(=O)C3)=O)C24)=O)CC1 7175,CCCCC(C)(F)C(=O)NC1CCC(C(=O)NCC(CO)N(C)C)C1 7176,C1(NC(c2ccc(C)o2)=O)CC12CCN(C(=O)C(CC1CC1)CC1CC1)C2 7177,n1(CCN(C(C2CCCC2n2cccn2)=O)CC)cc(C2(N(C)C)CCC2)nn1 7178,c1(C(=O)NCC(CCCC)NC(c2c(C)cnn2C)=O)nnc(Cl)cc1N 7179,C1(NC(=O)C=CCO)COCCC1NC(=O)Cn1nc(C2CC2)cc1C(F)F 7180,c1(SC)ccc(C)c(C(=O)NCC=C2CCN(C(=O)C=Cc3cc[nH]c3)CC2)c1 7181,c1(C(=O)OC)ccnc(C(N2CC(OCCNC(=O)C(C)O)C2)=O)c1 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7200,N1(C(COCC=C)=O)CCC(CCCNC(=O)C(c2cccnc2)C)CC1 7201,c1(NC(=O)Nc2nc(C(=O)OC)sc2)cccc(N(S(C)(=O)=O)C)c1 7202,N1(n2cc(-c3ccc(C)cn3)nn2)CCOC(CCN2CC3CCC2C3)CC1 7203,C(=O)(CC(C)CCC=C(C)C)NC1C2CN(C(C3(COCC)CC3)=O)CC21 7204,C1(CNC(c2n(C)nc(C(F)(F)F)c2)=O)CC2CCC1N2C(=O)CN1CCC1C 7205,N1(C(C2CC(CC)(CC)C2)=O)CCCC2C1CCCN2C(C1CCC1)=O 7206,C1(C(N(CCC)CCC)=O)CC12CCN(C(=O)C(C)n1ccnn1)CC2 7207,N1(CCCCC)CCC2(C1)c1ncn(C)c1CCN2C(=O)C(C1CCC(=O)N1)C 7208,Cc1ccc(CNCC2CCN(C(C3CNC(=O)N3C)=O)C2)cn1 7209,c1(C(C(=O)NC)N(CCOC)C(c2ccc(C)cc2)C)csc2ccc(C)cc12 7210,C1(NC(C(C)n2ccnc2)=O)CN(C(=O)COC2(C)CCOCC2)CC1C1CC1 7211,N1(C(c2ccc(OC)o2)=O)CC(C2CC2C(=O)NCCc2nncs2)C1 7212,c1(C(=O)NCCCN(C(=O)CCc2ccncc2)C)ccnc(OC(F)(F)F)c1 7213,C1(NC(C2(C(C)C)COC2)=O)CN(C(=O)C(O)c2cnc[nH]2)CC1(C)C 7214,N1(C(CC=CCC)=O)CC(NC(c2c(C)noc2CC)=O)CC12CCCCC2 7215,C1(C)(C(N(CC(C)(C)NC(=O)CSC(C)(C)C)C)=O)CC(C#N)C1 7216,c1(C(N2C(CN(C)C(C3CC4CC3C4)=O)CCCC2)=O)cnc2cccnc2c1 7217,N1(C(C(CCOC)(C)C)=O)CCC2CCN(C(c3nccs3)=O)CC2C1 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7237,c1(OC)nc(N2CC(C(C)NC(c3snnc3C(C)C)=O)C2)cc(C)n1 7238,N1(C(c2c(C)c(C#N)[nH]c2)=O)CCOC2CN(C(=O)CC(C)C(C)(C)C)CC12 7239,CCC(C)C(C(=O)NCCC1CC(NC(C2(C)CC(F)C2)=O)C1)NC(C)=O 7240,c1(C(=O)NC(c2ccccc2)C(=O)NCC2CCCC3CC23)nc(C)c(CC)o1 7241,c1(NC(N2CCCC(n3cc(COC)nn3)C2)=O)oc2ccccc2c(=O)c1C 7242,c1(OC)ccc2c(=NCCC#N)[nH]c(N3CCC(n4cc(CO)nn4)C3)nc2c1 7243,CC1CC(NC(c2ccnc(C3CC3)n2)=O)CN1C(c1cnn(C)c1Br)=O 7244,CC1(C)CCCOC1CNC(=O)CC12CCC1CN(C(=O)CC(Cl)Cl)C2 7245,c1(C(C(=O)NCCOC)N(C2CCN(CC(O)COCC)C2)C)cnc(C2CC2)s1 7246,C1(CNC(C(CC)OCC)=O)(CO)CCN(C(c2csc(SC)n2)=O)CC1 7247,c1(-n2cc(C3CCN(C(CCOC)=O)C3)nn2)cc(Br)ccc1Cl 7248,Cc1ccc(N)c(C(=O)NC2CC(NC(=O)CC3CCCC4(CC4)C3)C2)c1 7249,c1(C(N2CC(C)N(C(=O)CCc3cc(Cl)no3)CC2)=O)cccc2oc(=N)[nH]c12 7250,N1(CC)CC2CN(C(=O)CC3CCCCC3NC(C3CC(C)(C)CO3)=O)CC2C1 7251,c1(NC(C(c2ccccc2F)(C)NC(C)=O)=O)cnc(CN)nc1.C1(C)C(=O)N1 7252,C(CO)(C(C)(C)CO)NC(CCNC(C1(C)CC1(F)F)=O)=O 7253,C1(C(=O)OC)CCCN1C1CCC(CN(C(CC)C)Cc2ccccc2)C1 7254,c1(CC)cc(C(=O)N(CC(C)O)CCNC(=O)CC2CC3CCC2O3)sc1C 7255,C(=O)(C(CC(C)C)C(N)=O)NC(c1c(C(N2C(C(C)C)C(C)(C)C2)=O)con1)C 7256,c1(N2Cc3c(C)cnn3CC2)nc(=NCC2CCO2)[nH]c2c1CCCCCC2 7257,C1(NC(C2C(C(=O)OC)C2)=O)CCC(NC(=O)Cc2ccccc2C)CC1 7258,C(C(=O)NC1CC2CCC1(C(N1CC3(CCC3)C1)=O)C2)(C(C)(C)C)OC 7259,C(=O)(C(CCO)N(C)C)NCC(CC)NC(c1sc(C)nc1CC(C)C)=O 7260,C=CC1(NC(C2CC2NC(=O)COCC(=C)C)=O)CCCCC1 7261,c1(CNC(CCN(C(=O)C=Cc2ccccc2)CC)=O)cc2ccccc2[nH]1 7262,C(=O)(C1CCCc2scnc21)NC1CCN(C(C2(CN(C)C)CC2)=O)CC1F 7263,C(=O)(C1=C(C)OCCS1)NC(COCC)C(=O)Nc1ccc(C)c(CC)c1 7264,C1(NC(CCSC)=O)CN(C(C2CCSC2)=O)CCC1C 7265,C1(Nc2c(OC)noc2C2CC2)CCN(C(=O)OC(C)(C)C)CC1O 7266,c1(OC)ccc2[nH]c(C(N3CC4CC4(NC(=O)C(C)CF)C3)=O)cc2n1 7267,NS(=O)(=O)c1cc(C(=O)NCC2CCC(NC(=O)Cc3ccco3)C2)co1 7268,C1(C2(O)CCN(C(C3CCCC3S(C)(=O)=O)=O)CC2)(NC(C(CC)C)=O)CC1 7269,C=CC1(CC(=O)NC2CCCCC2NC(=O)C(O)C(F)(F)F)CCCCC1 7270,CC(C)(C)C1=NOC(C(=O)NC2CCN(C(=O)COC(F)(F)F)C23CC3)C1 7271,c1(C(=O)NC(C)CC2CN(C(c3cnccc3Cl)=O)C2)cc2cncn2c(O)n1 7272,Nc1cc(C(=O)NC2CC(C(=O)O)C(C(=O)O)C2)sc1C(=O)O 7273,N(C1CN(C(=O)C2=C(CC)OCCS2)Cc2ccccc21)C(C(CC#C)C)=O 7274,C1(c2ccccc2)(NC(=O)CCc2cccs2)CCN(C(C2COC(=O)N2)=O)C1 7275,C(C(C)(C)C(=O)NCC1(F)CCC(NC(C2CCCC(=O)N2)=O)C1)N(C)C 7276,C1(C(=O)NC(C(=O)OC)C2CCC2)CN(C(c2cscc2C2CC2)=O)CC12CC2 7277,C1(NC(C2(C#N)CC2)=O)(CF)CCN(C(=O)Cc2ccccn2)C1 7278,C#CCC(C)(C)C(=O)NCCOC1CCN(C(=O)CC2CCOC(CC)C2)C1 7279,S(=O)(=O)(c1cc(C(F)(F)F)ccn1)N(CC(Cc1ccccc1)SC)C 7280,Cc1cccc2[nH]cc(C(N3CCC(C)(CNC(C45CSCC4C5)=O)CC3)=O)c12 7281,N1(C(C2CC(C)N2C(c2ccn(C)n2)=O)=O)CCc2cnccc2C1 7282,C1(C(C)NC(=O)C=CCN(C)C)CCCN(C(C2(c3cccnc3)CCCC2)=O)C1 7283,C1(C(N(CC(=O)NC2CC2(C)C(C)C)CC#C)=O)CCC(C)N1C 7284,C(=O)(C(=O)N=c1[nH]occ1C1CCC1)NC(C)C(C)(O)Cc1ccccc1 7285,c1(C(N(CCN(C)C(=O)OC(C)(C)C)C)=O)cnn(CC2CC2)c1 7286,C(=O)(C(C)O)OC.C12(CC1)CC(=O)N(CCCN(C)C)CCSCCO2 7287,c1(C(N2CCC3(NC(C(C(=O)OCC)CC)=O)C(C2)C3)=O)cn2cccnc2n1 7288,c1(C(=O)NCC2C(NC(CCOCC)=O)C2)ccc(N(C)C)nc1 7289,S(=O)(=O)(c1cnc(NC(c2nccnc2C)C)c(Cl)c1)NCC=CCCC 7290,N1(C(CN(CC(C)C)C(c2cnn[nH]2)=O)=O)CC(C)C(F)(F)C1 7291,C(=O)(C(C)C(F)(F)F)NCCCCCNC(C(c1cccc(C)c1)F)=O 7292,C1(NC(C(c2cccnc2)OC)=O)COC2(C1)CN(C(c1csnn1)=O)C2 7293,n1(CC)c(C(N2CC(CCNC(c3ccnnc3O)=O)C2)=O)cc2ccccc12 7294,Cc1ccc(C)c(C(=O)NC2CCC(NC(=O)C(O)CC(C)C)C2)c1 7295,Cc1cc(C)c(C(=O)NCC2CCC(C)CN2C(C23CC(C2)C3)=O)c(C)c1 7296,Cc1cccc(Br)c1S(=O)(=O)NC(Cc1ccoc1)C(=O)O 7297,C1(C(=O)NC2(C)CN(C(CCN(C)CC)=O)C2)CCc2ncnn2C1 7298,N1(C(CSCC)=O)CCN(C(=O)CC2C(=O)NN=C2C)C(CS(C)(=O)=O)C1 7299,O=C(CC(CNC(C1CC(F)C(=O)N1)=O)C1CCC1)NOCC1CCCO1 7300,C1(CNC(CCN(C(C)=O)C)=O)CN(C(c2coc(Cl)n2)=O)C2CCN1C2 7301,Cc1cc(NC(C2CCN(C(=O)CCC3CC3)C2)=O)cc(O)c1 7302,C(=O)(C(O)CC(F)(F)F)N1C(C2(NC(Cc3c(C)con3)=O)CC2)CCCC1 7303,N1(C(c2c(C)nc(Br)cc2)=O)CCN(C(=O)CCc2ncc[nH]2)C2(CC2)C1 7304,N1(C(CC2CCN(C)CC2)=O)CCN(C(=O)CSC(F)(F)F)CC1C1CC1 7305,C12(C(=O)NCC3N(C(c4c(CC(N)=O)occ4)=O)CC(F)C3)CC1COC2(C)C 7306,C1(=C)CCN(C(c2ncsc2C)=O)CC1.C1(C(N(C)CC2CCC2)=O)(CSC)CC1 7307,C=CC(C)(CC)C(=O)NC(c1ccccc1F)CNC(=O)CCc1ccc(C)s1 7308,c1(C(=O)NCC(C(C)(C)C)NC(CN(C)CCO)=O)ncc(Cl)cc1Cl 7309,c1(C(=O)NC(C(=O)NCCCCC#C)CC(F)F)ccc2cc[nH]c2c1 7310,N1(C(C(C)(C)OC(C)=O)=O)CC(CNC(c2cc[nH]c2)=O)C(C)(C)C1 7311,C(C)(C(C(=O)NC(c1cccnc1C)C)NC(=O)C(C)OCCOC)OC 7312,CC1CCC(C)N(C(=O)CC2CN(C(c3cocc3C(N)=O)=O)CCO2)C1 7313,C12(NC(C3CCN(C(=O)NC)C3)=O)CCCN(C(c3c[nH]c(=O)cn3)=O)CC1C2 7314,Cc1cc(N)c(C(N2CC3=C(C2)CN(C(C2(C)CC(F)(F)C2)=O)C3)=O)cc1C 7315,C1(=CCNC(CC(C)N(C)C)=O)CCN(C(=O)C=CC(C)(C)SC)CC1 7316,N1(C(C2(OC)CCOC2)=O)CCCC(C)(NC(c2csc(-c3ccco3)n2)=O)C1 7317,C1(C(=O)NC(C(=O)NCCNC(C(C)(C)C)=O)Cc2cn[nH]c2)CC12CCCC2 7318,N1(C(c2cc(OC)n[nH]2)=O)CC2(COC(CNC(c3ccc(C(F)F)o3)=O)C2)C1 7319,Cc1nccn1C(C)C(=O)NC1CC(CCNC(c2cnc(C3CC3)o2)=O)C1 7320,N1(C(C(CC)NC(c2ccco2)=O)=O)CCC(CNC(=O)C(C)OC)C(C)C1 7321,C(=O)(C1=Cc2ccccc2C1)N(CC(C)NC(=O)CCP(C)(C)=O)CC 7322,O=C1CCC(CC(N2CCCC(CCNC(c3cc(=O)cc[nH]3)=O)C2)=O)CN1 7323,c1(CC)ncccc1C(=O)NCCN(C(=O)CC12COCC(C1)C2)C1CC1 7324,C1(N(CCC(F)(F)F)C(C(N2C(C)CCCC2)=O)=O)CCNC(=O)CC1 7325,Cn1cc(S(N)(=O)=O)c(CNC(C2(c3nncs3)CC2)=O)n1 7326,C1(C(=O)NCC(C2CCOC2)NC(=O)Cc2cncc(O)c2)CC2(CCCO2)C1 7327,C(=O)(C1CCCn2cnnc21)NCC1(CN(C)C(c2cn(C3CC3)cn2)=O)CC1 7328,CC1(C)CCC(C(=O)NC2CCC(NC(=O)CC=C(Cl)Cl)CC2)CO1 7329,C(CC#CC)(C(=O)NC1CCCC(O)C1O)NC(C1CC(O)(CC#C)C1)=O 7330,c1(C(N(CC(C)NC(C2(NC(C)=O)CC2)=O)CC)=O)ccc2c(c1)CCS2(=O)=O 7331,c1(NC2CCN(C(C(CC)(C)C)=O)C2)ncnc2c1c(Br)cn2C 7332,N1(C(C2CC(C)OC2=O)=O)C2CCCC1CN(C(=O)C=CC1CCC1)C2 7333,c1(C=O)[nH]c2ccccc2c1CC.C#CCCCNC.C1C(=O)NC(C)CO1 7334,O=S(=O)(c1cccc(F)c1)Nc1ccc(F)cc1OC(F)F 7335,C(=O)(C1=C(Cl)CCOC1)NCC(CC)NC(c1cccc2sncc12)=O 7336,c1(-c2c(C)ccc([N+](=O)[O-])c2C)ccc2c(c1)N(C)C(=O)C(C)O2 7337,N(C1CCCc2cc(F)ccc21)C(Cc1ccc(CN)nc1)=O 7338,CC1(C)C2CC(C(=O)NCC3(F)CCN(C(c4cncnc4)=O)CC3)CC12 7339,C1(CNC(c2nc(OC)oc2)=O)CCC(NC(C23CCC(OC)C2C3)=O)CC1 7340,N1(C(C2C(CNC(Cn3c(=N)nc[nH]3)=O)CCO2)=O)CC2CCCC2C12CC2 7341,N1(C(C(CC)OC)=O)CCN(C(C2(C#N)CC2(C)C)=O)CC1C 7342,C(=O)(C(Cc1ccccc1)S(C)(=O)=O)NC1CCC(C#C)CC1 7343,C1(C(=O)NC(C(C)C)(C)CNC(=O)C(O)Cn2cncn2)SC2C=CC1CC2 7344,Cc1ccc2ncc(C#N)c(N3CCN(C4CC4)C(C)C3)c2c1 7345,CCS(=O)c1ccccc1C(=O)NC1CN(C(c2cncnc2)=O)CC1C1CC1 7346,C1(CC)CN(C(=O)CO[Si](C)(C)C)CCN1C(=O)CC1(CO)CC1 7347,CCCCC(C)CCC(=O)NOCC(N1CC2(CCCCCC2)C1)=O 7348,c1(C(=O)NCCC(C)NC(C(CC)CC2CCCC2)=O)cc(OC)cc(C)c1 7349,N1(C(CC2C(C)CCO2)=O)CCC(CNC(=O)CCCC(N)=O)C(O)C1 7350,c1(C(C)NC(=O)NC2(c3ccccc3)CC2C(F)(F)F)cnc2ccccn12 7351,C=CC(C)(C)CC(=O)N1CCCC1C1CCCN(C(=O)CCN(CC)CC)C1 7352,C1(n2cc(-c3c(C)n[nH]c3)nn2)CCC(NC(c2ccc[nH]2)=O)CC1 7353,c1(CC(N2C(C(=O)NCCCC3CC3(F)F)CCC2)=O)ccc(O)nc1 7354,N1(C(C(c2ccccc2)OC)=O)CC2CN(C(c3ccc(C#N)cn3)=O)CC2C1 7355,N1(C(C(=O)NCC(F)(F)C2(O)CNC2)=O)CCN2C(=O)OCCC2C1 7356,S(=O)(=O)(c1ccc2[nH]c(=NCC3(C)CC3(C)C)ccc2c1)NCC1(OC)CCC1 7357,C1(CC#C)(C(=O)NC2CC(F)(CNC(=O)Cc3ccno3)C2)CCCC1 7358,C(=O)(C1CCCc2cc(O)ccc21)N1CC2CCN(C(C=CCCC)=O)C2C1C 7359,C(=O)(N=c1[nH]n(CCOc2nncs2)nc1C1CCOCC1)C1(F)C(C)C1 7360,N1(C(COCCOCC#C)=O)CCCC(C)C1CCNC(=O)Cn1ccnc1C 7361,c1(C(C(N2CC(CC)C(NC(=O)COCCOC)C2)=O)C)cc(C)ccc1F 7362,C1(C(N(CC(N)=O)C)=O)C2CC3C(C2NC(C2CCC(=O)O2)=O)C13 7363,CC(CC(C)NC(=O)C(C)Cn1ccnc1)N=c1[nH]c(Cl)ncc1[N+](=O)[O-] 7364,CCCCCCC(=O)NC(Cc1cn[nH]c1)C(=O)NCCC1CCCO1 7365,c1(CC(=O)NCCNC(C(c2cscn2)N(C)C)=O)ccnc(C(F)(F)F)c1 7366,C(=O)(C(C)(F)C(C)(C)F)NC1C(CNC(C(CC)(F)F)=O)CC1 7367,c1(C(=O)NC(CCNC(C(C(CC)O)C)=O)C)cc(=O)c(OC)cn1C 7368,C1(CNC(c2c(CC)con2)=O)CN(C(c2ccc(Cl)cn2)=O)CC12CCC2 7369,C1(N(C(=O)COC2CCCOC2)C)CCN(C(=O)CCc2cnn[nH]2)C1 7370,N1(C(CN(CCOC)C)=O)CC2CC(NC(c3c(C)nn(C)c3Cl)=O)C(C2)C1 7371,N1(c2cc(C)c(Br)cc2)C(=S)NC(c2cccc(Br)c2Br)C2=C1C(C)(C)NC2=O 7372,Cn1ccnc1C(F)(F)C(=O)NCC1CC(CNC(=O)CSC(F)(F)F)CO1 7373,N1(C(C=C(C)C(C)C)=O)CC(C)CCC1CNC(c1cccc(F)c1F)=O 7374,C(=O)(C1=CCCN(C(c2cc(O)nc(O)n2)=O)C1)NC(c1cncs1)C 7375,C1(NC(C2(C)CC(F)(F)C2)=O)CCN(C(=O)CSC2CC2)C(C2CC2)C1 7376,c1(C(=O)NCC(=O)NC(C)CC2CCCCO2)ccc2cc[nH]c2n1 7377,N1(C(c2nc(=O)cc(N)[nH]2)=O)CCC2(CC1)CN(C(c1cc(Cl)ncc1F)=O)C2 7378,C1(C(C)NC(c2ccsc2-n2cnnn2)=O)CCCCN1C(c1nocc1Cl)=O 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7575,c1(C(=O)NC(CNC(C(Cc2c(C)noc2C)C)=O)C)ccc(C#N)nc1 7576,N1(C(C2(CC)CCCC2)=O)CCN(C(=O)COCCSC)C(C2CC2)C1 7577,c1(SCC(=O)NCCC(C)NC(C2COC3(CCC3)C2)=O)ccsc1[N+](=O)[O-] 7578,S(=O)(=O)(c1cnn2ccc(=NCC3CC3Cl)[nH]c12)N1C2CC(N(C)C)CC1CCC2 7579,C12(CNC(CNS(N)(=O)=O)=O)CCCC1N(C(=O)CC1CCNC(=O)C1)CC2 7580,N1(C(CC(=O)N(C)C)=O)CC(NC(c2cccc(CS(C)=O)c2)=O)C2(CCC2)C1 7581,c1(C(=O)NC2CCN(C(C(CCC)C)=O)CC2O)cc2c(Cl)ccnc2s1 7582,C12(NC(CSCCNC(C3N(CCC)CCC3)=O)=O)COC(C1)C(O)C2 7583,C1(C(=O)NCC2CN(C(c3ncc(C)nc3)=O)C2)CC(C)CC(C)(C)C1 7584,n1(CCC(N2C(CCNC(C(N)=O)=O)CCC2)=O)ncc2c1CCCC2 7585,C(=O)(C(C)S(C)(=O)=O)NCC(c1ccccc1)CNC(c1cc(C)ncn1)=O 7586,C1(S(C)(=O)=O)(C(=O)NC2C(CNC(c3[nH]cc(CC)c3)=O)C2)CCCC1 7587,C12(COC)CC(NC(=O)Cc3cn[nH]c3)(CO1)C2.C(CCC(=O)N(C)C)N 7588,CC(C)CC(C(=O)N1CCCC1CS(N)(=O)=O)C(N)=O 7589,N1(CC)N=C(C(=O)N2CCCC(C)C2CNC(=O)CSC2CC2)CCC1=O 7590,C1(CC(=O)NCC2CCC(N(C(CC)=O)C)CC2)C(=O)N(C)N=C1C 7591,N(C(=NC1CCS(=O)(=O)C1)N1CCC2(CC1)CC(O)C2)C(C#C)CC 7592,N1(C(c2cnc(C)nc2)=O)CC(NC(=O)CCC(N)=O)C2(CC2)C1 7593,N1(c2ncc(C)cc2Cl)CCCc2sccc2C1 7594,c1(NC(C2(CC=C)CN(C(=O)CSC3CCCC3)C2)=O)cccc(C(C)O)c1 7595,c1(CNC2CCC(CNC(c3c(C)cc(Br)cn3)=O)CC2)cc2ccncc2[nH]1 7596,CCC(C(=O)NC1CCN(C(=O)Cc2cc[nH]c2)C12CCC2)C(F)(F)F 7597,N1(C(C(CCC2CC2)NC(c2c(C)ocn2)=O)=O)CCC2CN(C)CC2C1 7598,C(=O)(C(CNC(=O)CC(O)C1CCCC1)C(C)(C)C)NCCC=CCCC 7599,C(=O)(C1=CCCN(C(=O)CCCCC(N)=O)C1)NCC1C(C)CCC1 7600,Cc1ccc(C(N2CCC(C(C)Nc3ncnc(Cl)c3F)C2)=O)cc1C 7601,CCN=c1[nH]c(CNC(=O)NCC2CC(O)C2(C)C)cs1 7602,Cc1cccc(C(=O)NCC2(CN(C)C(C3CCCC34CC4)=O)CC2)n1 7603,N1(C(c2ccnc(C)n2)=O)CC2CC(NC(c3ccc(C)c(F)n3)=O)C2C1 7604,C(=O)(C(CC)CC(C)C)NC1(CN(C(c2cc(CC)c(F)cc2)=O)C)CC1 7605,Cc1cc(C(=O)NC2CC(NC(C3(Br)CC3)=O)C2)[nH]c1C 7606,C(CSC)(C(=O)NOCCc1ccccc1)NC(C(C(C)C)SC)=O 7607,c1(C2C(Cc3cn(C4C(OC)CCCC4)nn3)C2)c(C)cccc1[N+](=O)[O-] 7608,n1(CC(=O)NC(C2(CNC(C3OCCCO3)=O)CC2)C)cnc(Br)n1 7609,CC1(C)CCC(CNC2CN(C(=O)C(=O)N(C)C)C(C)(C)C2)OC1 7610,N1(C(c2c(C)cncc2)=O)CCC2(CCC2)C(NC(C2CC3(CSC3)C2)=O)C1 7611,c1(C(C)=O)ncccc1C(=O)NCCC1CC(N(C(=O)CCc2ccon2)C2CC2)C1 7612,c1(C(N(C(C)C(=O)O)CC2CCOC2)=O)cc[nH]c(=N)n1.c12cn(nn1)C(C)CS2 7613,CC1C(C)N(C(=O)CCCSC(C)(C)C)CCN1C(C1C2CCC1CC2)=O 7614,c1(C(=O)NC2CCCC(NC(C3(C)C(C)(C)C3(C)C)=O)C2)cnc2cc[nH]c2c1 7615,C1(CN(C(c2n[nH]cc2Br)C(=O)NCC(F)F)C)CCC=CO1 7616,C(=O)(C(C(C)(C)C)c1ccccc1)N1CC(NC(CCCSC)=O)C(C)C1 7617,Cc1nc(N2CCCC2C2CCN(C(=O)CCC(C)(C)F)C2)c(Cl)cc1C#N 7618,c1(C(=O)NCC(C)(CO)NC(CCSCC)=O)cn(C)nc1C(C)C 7619,CC1C(NC(=O)CCn2ccnc2)CCN1C(c1cnc(C(C)(C)CF)o1)=O 7620,C(C1CCOCC1)=CC(=O)OCC1CS(=O)(=O)C1 7621,CCCC(O)CCNC(=O)CNC(=O)CCCOC(C)C 7622,Cn1ccc(=O)c(C(N2CCC(O)(CNC(=O)C(F)n3ccnc3)CC2)=O)c1 7623,N1(C(CCc2c(C)noc2C)=O)C2CCC1CN(C(c1ncoc1C)=O)C2 7624,N1(C(C2CCCN(C)C2)C(=O)NC2CC(F)(F)C2)CCc2cccc(F)c2C1 7625,C1(C(C)C(=O)NCCn2cnnn2)CCCN(C(C2SCCS2)=O)C1 7626,c1(CC)cc2c(cc1OC)CN(C(C1CCN(C3CCN(C)CC3)CC1)=O)CC2 7627,c1(OC)cc(Br)cc(CN2CCCC2(C)C(=O)Nc2cnc3cc[nH]c3c2)c1O 7628,C=C(Cl)CC(C(=O)NCC(C)(C)C1CC1)NC(C1CC(=O)OC1(C)C)=O 7629,c1(CC)noc(C(N2CCSCC2CCNC(c2cnc(C)nc2)=O)=O)c1C 7630,N1(C(CC2CN(C(c3c(C)ccc(OC)c3)=O)C2)=O)CCC2(CC1)CC2(F)F 7631,c1(C(N2CCNCC2c2ccccn2)=O)cnc2c(Br)n[nH]c2c1C 7632,c1(N2CCCC(C(C)NC(CCOCC#C)=O)C2)cc(-c2ccco2)nc(C)n1 7633,C1(NC(c2n(C)nnn2)(C)CCOCCBr)CCN(c2ccccc2I)CC1 7634,C(=O)(CC(F)(F)C(F)(F)F)NC1CCCN(C(C(CCC)c2nn[nH]n2)=O)C1C 7635,C1(NC(C(CC)Cc2ccccc2)=O)C(C)CCN(c2cncc(Cl)n2)C1C 7636,c1(CNc2cc(CO)c(OC(F)(F)F)cc2)cc(F)c(F)cc1Br 7637,C1(NC(N2CCC(N3CCc4ccccc43)CC2)=O)CC2CC(CCCC2)C1 7638,C1(NC(Cc2cccc(OCC)c2)=O)CCSC12CN(C(=O)C(O)C(F)(F)F)C2 7639,c1(NC(C2N(C(C3C(C(=O)OC)C3)=O)CCOC2)=O)ccc(F)c(C(N)=O)c1 7640,n1(CC(=O)OCC)nc(-c2cccc(F)c2)nc1-c1c[nH]c(=O)cn1 7641,c1(C(=O)NCC=CCNC(C2C(C=C(C)C)C2(C)C)=O)cc(N)c(Cl)c(O)c1 7642,c1(CNC(c2cc(CC)on2)C)cc(Br)ccc1C(F)(F)F 7643,C(CC(=O)NCC1CC(NC(=O)C(C)n2ccnc2)C1)OCCCOC 7644,CC1(C)CCC(C(=O)NCCC2CCCN2C(c2cc(O)cs2)=O)C1 7645,c1(OC)ccc(C(=O)NCC2(F)CC(NC(=O)C(O)C(C)OC)C2)c(OC)n1 7646,Cc1ccc(C(N2CC3(C2)CN(C(=O)C(=O)N(C)C)CC3CO)=O)c(N=[N+]=[N-])c1 7647,c1(OC)cncc(C(=O)N(C(C)CNC(=O)CC2CCC(=O)O2)C)c1C 7648,Cc1c(C(=O)NC2(CO)CCN(C(=O)C(C)CS(C)(=O)=O)C2)nn2c1CCCC2 7649,CCCCCC(F)C(=O)N1CCC(C)C1C(=O)NCCc1nc[nH]n1 7650,c1(NC(C)C)ccc(C(N2CC(CC(C)NC(=O)C(F)C(C)C)C2)=O)cc1 7651,C1(NC(CC(=C)C)=O)CCC2(CC1)CN(C(=O)C1=COCCC1)CCO2 7652,c1(C(=O)NCCN(CC(C)O)C(C2CCC2(C)C)=O)sc([N+](=O)[O-])cc1Cl 7653,c1(-c2nc(CC(CC)C)nn2C(C)C(F)(F)F)cc2nccnc2cc1C 7654,CC(C)CS(=O)(=O)CCC(=O)NC1COC2CN(C(C3(C)CNC(=O)C3)=O)CC12 7655,c1(CCC(N2CCC(CCNC(CCC(C)OC)=O)C2)=O)ccc(Cl)c(C)c1 7656,N(C1CCCc2c(Br)cccc21)C(c1n(CC)nnn1)c1cccc(C(C)C)c1 7657,N1(C(c2cccc(NC(C3C(C(=O)OC)C3)=O)c2F)=O)CCC(O)C(C)(CO)C1 7658,C1(CC)CCN(C(=O)Cc2ccc(C)s2)C(C(=O)NC(CC)C(C)C)C1 7659,CC(C)CC(O)C(C)C(=O)NC(Cc1ccco1)C(=O)NCCCC(C)CO 7660,C1(NC(c2c(CCC(=O)OC)cccc2)=O)CN(C(=O)CC2CC2)CCC1(C)C 7661,C(N=c1cc(C(F)F)nc[nH]1)C1(NC(=O)CCCc2cnn[nH]2)CCOCC1 7662,C(=O)(C(C)(O)CC(C)C)NC1CCCC(NC(COCC=C)=O)C1 7663,N1(C(C(COC)OC)=O)CCC(O)(C(N2CCC(C)(O)C2)=O)C1 7664,C(=O)(C1CCCc2nn(C)cc21)NC(C)CC(=O)NNC(=O)C1CC1.C(C)(C)(C)O 7665,C1(C(N2CCC(CCOC)(NC(=O)Cn3cnnc3)C2)=O)C2CCC(C2)C1(C)C 7666,N1(C(c2ccc(C#C)cc2)=O)CCCC2CN(C(=O)C(n3ccnc3C)C)CC12 7667,N1(C(CSCCNC(COC(CC)(C)C)=O)=O)C2CCC1CC(=O)NC2 7668,c1(N2CCC=C(C(=O)OC)C2)ncnc2c1ncn2C1CCC(CO)O1 7669,N1(C(c2c(CC)occ2C)=O)CC(NC(=O)CP(C)(C)=O)CC(O)C1 7670,C=CCCCC(C)(C)C(=O)NC1CCOCC1NC(=O)C(c1ccnn1C)O 7671,Cc1cc2[nH]c(C(N3CCC4C(C3)CN4C(=O)COC3CCCCC3)=O)cc2s1 7672,Cc1c(C(N2C3CCC2CN(C(=O)C(O)C(C)C)C3)=O)sc2ccnc(O)c12 7673,CCC(CN(C)C)CC(=O)NC(C(=O)NC1CCS(=O)CC1)C1CCC1 7674,c1(CC(=O)N(CCCN(C)C(C2CC2(F)F)=O)C)ncccc1Br 7675,C1(NC(C2CC23CCC3)=O)COCCC1NC(C1CCS(=O)CC1)=O 7676,N1(C(c2cc(CCC)on2)=O)CC(NC(c2ccc(O)nn2)=O)C2CC12 7677,C(C1CCOC1)=CC(=O)NCCCCNC(C1CC(F)C1)=O 7678,Cc1cc(F)sc1C(=O)NCC1CCCC1C(=O)NCC(O)CC(C)C 7679,c1(C(=O)NC(CNC(C(C2CCC2)OC)=O)C)cc(O)c2cnn(C)c2c1 7680,N1(C(C(C)NC(COC)=O)=O)CCCCC1C(N1CC2CC2(CO)C1)=O 7681,CCC(CC(=O)NCC1CCCCCN1C(=O)COCc1nnc(C)s1)C(C)C 7682,c1(C(=O)NC(C)CCS(C)=O)ccc(Br)c(C#N)c1 7683,C(=O)(C1=CC2(CN(C(=O)C(C)(C)n3cccn3)C2)OC1)NC(COC)C(C)C 7684,C1(CN(C(=O)CC2CCOCC2)CC)CCN(C(c2cnn(CC)c2)=O)CC1 7685,C1(CNC(c2cc[nH]n2)=O)(NC(c2ccc(-c3ccccc3)o2)=O)CCCCC1 7686,C1(NC(c2[nH]nnc2C2CC2)=O)CN(C(=O)Cc2cncc(F)c2)C2CC12 7687,c1(C(=O)NC(CC)CN(C)C(C2(CC)CCOCC2)=O)ncc(C)cc1Br 7688,C(C(C(C)(C)C)CC(=O)O)NC(C1CC(COCCOC)C1)=O 7689,C(=O)(C1(C)CCn2c(C)nnc21)NCC1CN(C(COCC)=O)CC(C)(C)C1 7690,Cc1cccc2[nH]c(=NC3CCC4CN(C(C5CC5F)=O)CC34)sc12 7691,CC1(C(F)F)CC1COC(=O)CCc1ccc[nH]1 7692,c1(C(N2CCC(NC(C3(C=C)CC3)=O)C(C)C2)=O)ccc2c(=O)cc[nH]c2c1 7693,C1(OC)CC2(C1)CC(C(=O)NC1CC(CNC(=O)CSC(C)C)C1(C)C)C2 7694,C1(CNC(c2cc(C)n(C)n2)=O)CCC(C)CN1C(=O)CC(C)(C)N(C)C 7695,C(=O)(C(C)C(C)C(C)(C)C)NCC(C(C)C)(C)NC(c1ccc2c(c1)NCC2)=O 7696,CC(C)CCC(c1nnnn1Cc1ccccc1)NCC1(C)CC1(Cl)Cl 7697,N1(C(c2c(CC)n[nH]c2)=O)CC2CN(C(=O)C(n3nccc3C)C)CCC12 7698,c1(OCC(N2CC(C)C(NC(=O)COc3ns[nH]c3=O)C2)=O)ccccc1C#N 7699,C(=O)(C1=CC(O)C(NC(C2(F)CCC2)=O)C1)NC1(CC=C)CCC1 7700,c1(C(N2CCC(NC(C(CC)C)=O)C(F)C2)=O)nn(C)c2ccc(Br)cc12 7701,c1(C(=O)NC2CN(C(C3(OCC)CCOC3)=O)C2)cc(F)cc(C)c1N 7702,c1(C(=O)NCC=CCNC(=O)CC2CC(F)C2)ccccc1C#CC1CC1 7703,Cc1[nH]cc(C(=O)NC2CC(CO)N(C(=O)CCCN(C)C(C)C)C2)c(=O)c1Cl 7704,c1(OC)ccc2c(=NCc3sccc3C)[nH]c(=NC(C)COC)[nH]c2c1 7705,N1(C(C(CC=C)C)=O)CCCCC(C2CN(C(c3ccc(O)c(N)c3)=O)C2)C1 7706,C1(NC(CC(CC)C)=O)CCN(C(=O)C(C)NC(=O)CC(C)(C)C)C1(C)C 7707,N1(C(C(C(C)O)NC(C(CC#C)O)=O)=O)CCCCC1C#C 7708,c1(N)ccc(-c2ccns2)cc1.Cc1csc(C)n1.C12(CC1)C(=O)N2 7709,C1(NC(C2(C(N(C)C)=O)CC2)=O)CC2CCC1N2C(C1CCOC1(C)C)=O 7710,C1(C2CCCO2)(C(=O)NC(=O)CC(=O)NC(C2CC23CCCC3)C)CCOCC1 7711,n1(CC(C)(C)C)cccc(-c2nc(-c3cncc(F)c3)nn2CCCCO)c1=O 7712,c1(C(N2CCC(CNC(c3c(C)nc(C)s3)=O)C2)=O)oc(P(C)(C)=O)cc1C 7713,c1(NC(C(N2CCC(O)CC2)C)=O)cncc(-c2ccc(F)cc2)c1 7714,C1(C)(CC(=O)NC2CC(CCNC(C(c3cncn3C)N(C)C)=O)C2)CCCO1 7715,c1(CN(C)C)cccc(C(=O)NCC=C2CCN(c3ncc(Br)cn3)CC2)c1 7716,C1(C(N(CCCCCNC(=O)Cc2nn(C)cc2Cl)C)=O)COCC(C)(C)O1 7717,C1(CC(C)C)(C(=O)NC2(C(=O)OC)CCC2c2ccccc2)CCNC1=O 7718,CCC(C(F)C(=O)NC1CC(=O)N(O)C1)NC(=O)CC1CCCC(C)O1 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7844,N1(C(C2(SCC)CC2)=O)CCCC2(C1)CN(C(=O)C(C)Oc1cccnc1)C2 7845,C(CC(C)(C)CC(=O)NCCCNC(c1ncc2ccccn12)=O)OC.C1CN1 7846,C1(N(C(=O)CN2CCCCC2=O)CC)CCN(C(=O)C(=O)Nc2ncc[nH]2)CC1 7847,CC1CCCCC1Cc1nc(-c2cccc(N)n2)nn1C1C2CCC1CC2 7848,C=CC(C)(CCOC)C(=O)NCC1(NC(=O)CNC(C)=O)CCCC1 7849,Cc1c[nH]nc1C(=O)N(C(CNC(=O)C(F)C1CCC1)C1CC1)C 7850,N1(C(CCCc2n(C)cnn2)=O)CCCC(C(C)(O)CNC(C2(SC)CC2)=O)C1 7851,C1(NC(c2nncs2)=O)CC2CC(NC(C34CCCC(CO3)C4)=O)C1C2 7852,Cc1cc(Cl)ncc1CNC1C2CN(C(C3CCN(C)CC3)=O)CC12 7853,CCC1=NOC(CNC(=O)Nc2ccnc(OC(C)C)c2)C1 7854,Cc1nc(C)n(CC(=O)NC(CCN(C)C)C(=O)NCCCN=[N+]=[N-])n1 7855,c1(C(N2CCC(CC(C)NC(C3(C=C)CC3)=O)CC2)=O)ccc(F)c(Cl)c1N 7856,C1(NC(CC(CCC)C)=O)CN(C(c2nc(Cl)ccc2Cl)=O)C2CCCCC12 7857,C1(C)(C(=O)NC(C)CCCCNC(=O)Cc2nc[nH]n2)COc2ccccc2O1 7858,C12(c3ccccc3)C(CF)CC1CNC2.N1(CC)CCN(C(=O)OC(C)(C)C)CC1 7859,c1(C(=O)NCC2N(C(CC(C=C)CCC)=O)CCCC2)cccn2cc(C)nc12 7860,N1(C(C(n2c(C)ncc2)C)=O)CC(NC(=O)CC(F)(F)C(F)F)CC12CCC2 7861,C1(CN(C(CC(=C)Br)=O)C)CCN(C(C2CCCC(OC)C2)=O)CC1 7862,c1(C(=O)NC2C(C)CN(C(=O)C=C3CCOCC3)CC2)cc(F)cc2nc[nH]c12 7863,Cn1c(O)nc2cc(C(=O)N(C3(C)CCOC3)C(C3CCCO3)=O)ccc12 7864,c1(C(=O)NC(CCC)CNC(=O)C(C)NC(=O)NC)ccsc1C#N 7865,N1(C(CC2(OC)CCC2)=O)C2CCCC1CN(C(C1CC(O)C1)=O)C2 7866,n1(C(CC)CC)nccc1C(=O)NCC(C)(C1CC1)NC(=O)C(CO)N(C)C 7867,C1(C(=O)OC)CCN(Cc2ccc(CCN(C)C)cc2)CC1OC(F)F 7868,C1(CC(=O)N(CC(C)N(C)C(c2cc3sccc3s2)=O)C)CCC(C)(C)CO1 7869,c1(COC)cccc(C(=O)NC2CN(C(=O)C=CC(C)(C)C)CC2O)n1 7870,c1(C(NNCC=C)=O)sc2cc(Cl)ccc2c1Cl 7871,C=CCC(C)C(=O)NCC(CCCC)NC(=O)C(C)NC(C1CCCCC1)=O 7872,Cc1c(F)ccc(C(=O)NCC2CN(C(c3cc[nH]n3)=O)CCO2)c1Cl 7873,N1(C(COC)=O)CCN(C(=O)CP(C)(C)=O)C(CO)C1 7874,Cc1cc2[nH]c(C(=O)NC3CC4CC3N(C(c3ccsc3)=O)C4)cc2o1 7875,N1(C(=O)OC(C)(C)C)C2CCC1C(C(N1CCC1CC1CC3CNC1C3)=O)C2 7876,C(CCN=c1ccc(C(F)(F)F)c[nH]1)N(C)C(c1cccc(Br)c1Br)=O 7877,Cc1nc(F)ccc1NC(=O)CCC1CCC(NC(=O)CCCC#N)C1 7878,N1(C(C2(NC(c3nccc(C)c3N)=O)CC2(C)C)=O)CC(C)OCC(C)(C)C1 7879,c1(N(CCCNC(c2ccc(O)nc2)=O)C)ncnc2c1cnn2C 7880,C1(C(C)(CNCCCOCCO)NC)CCOCC1 7881,CC(C)CCC(CO)NC(C1CC(NC(=O)CC2CCC(C)(C)C2)C(O)C1)=O 7882,N1(C(CC2C(C)CCN(C(C(CC=CCC)C)=O)C2)=O)CC(C)(CO)CC1(C)C 7883,C1(CNC(=O)Cc2cccc(F)c2)CN(C(C2CCCC(F)(F)C2)=O)CC12CC2 7884,N1(Cc2c(C#C)cccc2)CC2CCC1CN(C(c1cc(C)n(CC)n1)=O)C2 7885,C1(CNC(C(c2ccccc2F)C)=O)CCN(C(C23CC(C)(CO2)C3)=O)CC1C 7886,C(=O)(C(C)CC(F)F)NCC(CC=C)NC(c1ccnc(OCC)c1)=O 7887,Cn1c(C(N2CC(O)(C(F)C(=O)NC3CC(=O)N(O)C3)C2)=O)ccc1C#N 7888,CC1CCCC1CC(N1CC(CCCCNC(=O)CNC(c2ccsc2)=O)C1)=O 7889,c1(C(N(C2CCN(C(C3CN(CC)C(=O)C3)=O)C2)C)=O)ccc2c(c1)CCCN2 7890,C1(OC)CCC12CC(C(=O)NC13CC(NC(=O)CC4CCOC4)(C1)C3)C2 7891,C(c1ccc(F)cc1)=C(C)C(=O)N1CCC1n1cc(COCC(=O)O)nn1 7892,C(=O)(C(C)S(N)(=O)=O)N1C(C(N2CC(CO)C2)=O)(COC)C=CC1 7893,N(C(=NCCC(=C)C)NC1CCN(Cc2cccnc2)CC1)CC(C#C)OC 7894,N1(C(CC(C(C)C)c2ccon2)=O)CC2CCC1C(CNC(C1(CO)CC1)=O)C2 7895,c1(C(N2CC(C)C(CNC(=O)Cc3ccno3)C2)=O)ccc2c(O)ncnc2c1 7896,C(=O)(C1=CC2(CCOC2)C1)NCCN(C(=O)CCc1cnc[nH]1)C 7897,c1(CNC(C(CC)SC)=O)nc(CNC(C2CCC3CC2CO3)=O)cc(O)n1 7898,c1(CC)cnc(C(=O)NC2CCC(C(=O)N(C(C)CC(C)C)C)C2)nc1 7899,Cc1cc(=NC(=O)C(=O)NCC2(NC(=O)C(O)C3CCCC3)CCC2)[nH]o1 7900,c1(C(=O)NC2C(NC(C3(CC)CCOCC3)=O)CC2)cncc(C)c1C 7901,C1(NC(C2(C)CC=CC2)=O)CC2CCCC(C1)N2C(c1cnc(Cl)s1)=O 7902,O=S(=O)(c1cnc(NC2COCC2O)c(Cl)c1)NC1CCC=CCC1 7903,N1(C2CCN(C(C3CN(C)C3)=O)CC2)Cc2cccnc2N2CCCC2C1 7904,C1(C(C)NC(c2c(Cl)cnn2C(C)C)=O)CN(C(=O)CSc2cnn(C)c2)CCO1 7905,c1(N2CCN(CC(=O)NC(C3CC(=O)NC3=O)C)CC2)ccccc1[N+](=O)[O-] 7906,N1(C(c2cnc(CCC)s2)=O)CCCC(C)(NC(=O)CC(C)(C)OC)C1 7907,c1(C(=O)NC2CCN(C3CCN(C(CCCC)=O)C3)CC2)cc(F)ccc1Cl 7908,c1(SCC(=O)NCC(C)(C)NC(C(CO)N(C)C)=O)nc2ccccc2o1 7909,N1(CC)CC(NC(=O)C(C(C)(C)C)NC(=O)C(=CC2CCCC2)C)CCC1=O 7910,C1(CC)CCC(C(=O)NC2CC23CC(NC(=O)COCc2ccncc2)C3)CC1 7911,C(=O)(C(CCNC(c1cccn1C1CC1)=O)OC)N(C)CC1CC(=C)C1 7912,N1(C(C2C(CNC(C3C(CC)C3)=O)CCCC2)=O)CC(=O)NC(C)C1 7913,N1(C(C2C(OC(C)(C)C)C2)=O)CCC2C(NC(=O)COC(F)(F)F)C2C1 7914,N1(C(C2(CC)CCCCC2)=O)CC(CN(C)C(c2ccoc2)=O)C2(CC2)C1 7915,C(=O)(C(CC(C)C)NC(=O)C(C#N)C(C)C)N(c1ccc(C)cc1)CC 7916,c1(NCCCC(=O)c2ccc(Cl)s2)nc(F)c(I)cc1F 7917,C1(O)(C(N2CCCC(CNC(=O)CC3CC4CC3C4)C2)=O)CCCCCC1 7918,C1(N(C(C(F)OC)=O)C)CCCC2CN(C(c3ccncc3F)=O)CC12 7919,CC1(C(=O)NCC(C2CC2)NC(c2csc(C3CCCCC3)c2)=O)CC1(F)Cl 7920,c1(CC)ccc(F)cc1C(=O)NCC(C)(CO)NC(c1cc(F)ccc1O)=O 7921,N1(C(C(C)SCC)=O)CCN(C(=O)CCOC(C)=O)CC1CC(F)F 7922,C12(C(N3CC(CNC(COCCOC)=O)C(C)C3)=O)CCC(C1)C(C)(C)O2 7923,c1(C(N2CC(CCNC(C(C)OC)=O)C2)=O)ccc2nc(O)[nH]c2n1 7924,N1(C(Cc2cn(C(C)C)nc2)=O)CC=CC(NC(C2CC2c2ccsc2)=O)C1 7925,C(CC(C(C)(C)C)NC(C1CCCN1C1CCCCC1)=O)N(C(=O)CCF)C 7926,N1(C(CCOCC(C)C)=O)CC2(CCCC2)C1C(=O)NC(C1(O)CCC1)C 7927,N1(C(c2cnc(=N)[nH]c2)=O)CCC(C2CCC2)(CNC(=O)CC2C=CCC2)CC1 7928,C1(NC(C(C)n2cncn2)=O)COCC1CNC(c1csc(C(F)F)n1)=O 7929,C1(NC(COCCC=C)=O)C2CN(C(c3cc[nH]c3CCC)=O)CC12 7930,c1(C(=O)NC(C2CN(C(CCC3C(C)=NOC3=O)=O)C2)C)nc(O)nc(O)c1N 7931,Cc1cc(C(N2CCC(NC(=O)CC(C)CF)CC2)=O)c(Br)cc1F 7932,CCC(C)C(O)CC(=O)NC(CNC(=O)CCCCN(C)C)CC(F)(F)F 7933,C1(OC)CCC(NC(=O)C(C)NC(c2ccc(C)o2)=O)C1 7934,c1(OC)ccc2cc(C(N3CCC(NC(=O)Cc4cnc(C)o4)C3C)=O)[nH]c2c1 7935,C=CC(O)C(=O)NC(Cn1cccn1)C(=O)N1CC(C)(C(N)=O)C1 7936,N1(CC)CC(C(=O)NCC2CCCC2NC(=O)CC2CCCOCC2)CCC1=O 7937,N1(C(C(C(C)C)F)=O)CCC12CN(C(C1(c3ccc(O)cc3)CC1)=O)C2 7938,C1(C)(CNC(c2nc(C(=O)OC)oc2)=O)CCCN1C(c1cnn(C)c1F)=O 7939,Nc1ccc(C(=O)NCC2CCN2C(=O)CC2CCCS(=O)(=O)C2)nc1N 7940,C(=O)(CC(P(C)(C)=O)P(C)(C)=O)NC1CC(NC(c2cc(C)nn2C)=O)C1 7941,C(=O)(C1=CC(C)(C)C1)N1CCC(C)(CCNC(c2cnc(C)n2C)=O)C1 7942,C(=O)(C(C)(C)C(=O)NCC1CN(C(c2cn(C)nc2C)=O)C1)OCC 7943,CC1(C(N2CCC(O)(c3ccc(F)cc3)CC2)=O)CCCNC1=O 7944,c1(CNC(c2cnc(C)s2)=O)ccc(C(=O)NCC2(F)CCOCC2)nc1 7945,C1(O)(CNC(C2C(c3n(C)ncc3)C2)=O)CCN(C(c2ccccc2)=O)C1 7946,C(C1=CCN(C(c2cnc(-c3ccco3)s2)=O)CC1)NC(C1(C=C)CCC1)=O 7947,C1(C(N(C)Cc2c(C)cco2)=O)C2CC3C(C2NC(C2CCC(F)C2)=O)C13 7948,C(=O)(C1=CC2CCCC12)N.O=C(CCc1ccco1)NCC1(C)CC1 7949,CC(CC(N)=O)C(=O)N(C)CCC1CCCCN1C(C1C=CCS1)=O 7950,c1(C(=O)NC2CCCC(NC(c3ccnc(S)c3)=O)CC2)ccn2cccc2c1 7951,N1(C(CC2(OC)CN(C(=O)C(F)(F)C(C)(C)O)C2)=O)CC2OCC(CO)C2C1 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8150,Cn1c(O)ncc(C(=O)NCC2(NC(C3CNC(=O)N3)=O)CCOC2)c1=O 8151,CCCC(C)NC(C)=O.C1CC(=O)N1CC1CCCS1 8152,C12(NC(C3CC(C)OC3)=O)CCCCCC1N(C(c1cc(O)ccc1N)=O)CC2 8153,c1(C(N(CC(C)NC(=O)Cc2cncnc2O)C)=O)ccnc(Cl)c1Cl 8154,N1(C(CC2(C=C)CCCCC2)=O)CC2CCN(C(C3SCCS3)=O)C2C1 8155,c1(-c2cn(CC(N3CCC(N4CCCC4)C3)=O)nn2)ccc(CCO)cc1 8156,C(=O)(C(CC)C(C)(C)CC)N1CCC(CNC(C(CC)Sc2ccccc2)=O)CC1 8157,N1(C(CCc2nnc(C)o2)=O)CCN(C(C)CNC(c2cnsn2)=O)CC1 8158,c1(C(=O)NC23CN(C(C=C(C)C(C)(C)C)=O)C(CC2)C3)c[nH]c2c(F)cccc12 8159,C1(C(N(C)CC2CC(OC)C2)=O)C2CC3C(C2NC(c2cc(C)nnc2C)=O)C13 8160,N1(C(CN(C2CC2)CC)=O)CC2(C1)CN(C(=O)CCC1CCCO1)C2 8161,Cc1c[nH]c2ncc(C(=O)NCC3(CNC(=O)CN4CC5CCC4C5)CC3)cc12 8162,C=CC(C)(C)C(=O)N(CC(O)CN(C)C(C1(CC)CCOC1)=O)C 8163,C12(NC(=O)CCF)CCCC1CN(C(c1ccc(-c3ccsc3)nc1)=O)C2 8164,c12cccnc1C(=O)NC1CCC(C1)NC2=O.C1(CCC)(C(=O)C2CC2)CC1.O 8165,c1(C(=O)NC2C(CNC(=O)CCF)COC2)ncccc1C1CC1 8166,c1(OC)ncc(C(=O)NCC(CNC(=O)CCc2csc(=N)[nH]2)OC)cc1C 8167,C1(C)(C(=O)NCC2CC(NC(c3n(CC)ccc3)=O)C2)CCC(=O)N(C)C1 8168,CC1CN(C(=O)COC2CCC2)CCCN1C(C1C2COCC12)=O 8169,C1(C(=O)NCc2nc(=N)[nH][nH]2)CCN(C(C2C=CCS2)=O)CC1 8170,c12nc(cc(C)n1)N2.C12CN(C1)C(=O)CC1(CC1)OC(C)C2.CCO 8171,C1(NC(c2coc(Cl)n2)=O)CCC2(CC1)CCN(C(c1ccc(I)c(O)c1)=O)C2 8172,C(C)(N=c1[nH]c(=N)[nH]c(=NCC(C)C)[nH]1)c1c(C(c2ccccc2)C)cc(F)cc1 8173,c1(C(=O)NC2C(NC(C(C)Sc3nc[nH]n3)=O)CCC2)cccc(C(F)(F)F)c1 8174,C1(C(=O)NCc2c(CCNC(C(C)(C)F)=O)ocn2)CC1C1CC(F)(F)C1 8175,N1(C(c2cnc(CCC)s2)=O)CC(NC(=O)C(C)(CC)CO)C(C2CC2)C1 8176,CC1(C)COCCN(C(C2CC(O)CN2C(=O)CC2CC2C2CC2)=O)C1 8177,Cc1nnc2ccc(C(=O)N(CC(C)CNC(=O)C=Cc3ccc(Cl)s3)C)cn12 8178,C1(C(=O)NC(C(=O)NCC)CC)CN(C(=O)CC2(C)CCCC2)CC12CC2 8179,C1(NC(C=CCCC)=O)CCC2(CCN(C(C3(C)CCCC3O)=O)C2)C1 8180,C1(O)(CNC(c2n(C(CC)C)ncc2)=O)CCN(C(C2CCCOCC2)=O)CC1 8181,Cc1cnn(C)c1CC(=O)NCC1CCCN(C(c2cnn(C3CCC3)c2)=O)C1 8182,C1(NC(=O)CBr)CCC(CNC(C2(n3cccn3)CC2)=O)C1 8183,C(C(C(=O)NCc1cc(C)no1)C(C)(C)C)NC(C(C)(C)SC)=O 8184,c1(OC)nc(C)cc(C)c1NC(C1CCCN1C(C)=O)=O 8185,C(=O)(C1CCCn2cnnc21)N1CC(NC(=O)CSc2nc[nH]n2)(CO)C1 8186,C12(C(=O)NC3CCN(C(CC(C=C)C)=O)C3C)CCC(CC1)C(C)O2 8187,C1(NC(=O)CN2CCCC2=O)CC2CC1N(C(c1nccc(F)c1Cl)=O)C2 8188,c1(SCC(=O)NCCCCCCNC(c2ccc(C#C)o2)=O)ccc2c(c1)CCC2 8189,N1(C(C2C(=C)CC2)=O)CCC2(CC1)C(NC(=O)CCC(C)SC)CS2(=O)=O 8190,N1(C(=O)N(C2CCCCC2)C2CCCC2)CCC(C2CCCC23OCCO3)C1 8191,c1(CC)c(C(C(=O)NCc2nnn(C)n2)N(CC(C)C#N)C)cccc1C 8192,N1(c2ccnc(NC(c3ccncc3Cl)C)n2)CC2CC1CS2=O 8193,N1(C(C(Cn2cccn2)NC(COCCSC)=O)=O)CCCN(C(C)C)CC1 8194,Cc1cc(C(N2CCCC2CCCNC(=O)Cc2ccsc2C)=O)[nH]c1C 8195,CC(C)(C#CC(=O)N1CC(O)C(O)C1CO)CNC(c1coc(CO)c1)=O 8196,Cc1cc(C(=O)NC(C2CCN(C(c3ccccc3Br)=O)C2)C)ccn1 8197,c1(C(N2CCC(C)C(NC(C3CSC3)=O)C2C)=O)c[nH]c2cccc(F)c12 8198,N1(C(c2cc(CC)on2)=O)CCN(CCCNC(=O)CC(C)CC)CC1 8199,c1(CCC)cc(C(N2CC=CC2C(=O)NC2(C(=O)NC)CCOC2)=O)n[nH]1 8200,C12(CCCC)CN(C1)C(=O)C1CCC1C(=O)C(=O)C1CCN(C1)C2=O.OC.OC 8201,c1(C(=O)NCC2CCC(CNC(=O)C(F)F)CC2)cc2cccc(Br)n2c1 8202,C1(C(=O)NC(C)CC(=O)N(C)CCOCCCO)CC2CC(=O)C1O2 8203,C1(C(N(c2nccs2)CC)=O)CCN(Cc2ccc(F)s2)C1 8204,c1(NC(C2COCCN2C(C2C3COCC23)=O)=O)ccc(Cl)c2cc[nH]c12 8205,C1(CC(=O)NCC(C)(CNC(C2CCC3(CCC3)O2)=O)OC)CCC2(CCC2)O1 8206,C(=O)(CCC(=O)NCCC1COCCN1C(=O)Cn1cc(C2CCC2)nn1)NC 8207,C(C(C)(O)CC(=O)NCC(CC(F)(F)F)NC(c1ccn(CC)c(=O)c1)=O)OC 8208,C12(Cc3ccco3)CCCC1CNC2.C1(CO)CC2(CO1)CC2OC 8209,N1(C(C(=O)NCCOC)=O)CCC2(CNC(=O)CN(C)S(N)(=O)=O)CCCC12 8210,c1(C(=O)OC)cc(C)cnc1NC1CC(C)N(C(c2cnn(C3CCC3)c2)=O)C1 8211,C(CC(C)C)(C(=O)N1CCC(C(C)CO)CC1)N(C(CSCCC(C)C)=O)C 8212,N1(C(N2CCCC(O)(CC(=O)OC)C2)=O)CCC2(CC1)COc1ccccc12 8213,C1(C(=O)NCCCC(=O)NCCCOCC=C)CC(=O)OC1(C)C 8214,C(=O)(C1CCCc2n[nH]cc21)N1C(CNC(C(C)(C)CF)=O)CCC1 8215,c1(C(C)=O)cc(C(=O)NC2COCCN(c3ccnc(C)n3)C2)ccc1[N+](=O)[O-] 8216,c1(OC(C)C)cc2ccc1NC(=O)O2.c1(CC(C)N(CC)CC)n[nH]c(=N)s1 8217,C1(N(C(C2CCN(CC(C)C)C2)=O)C)CN(C(=O)CCCC2CC2)CC1O 8218,C1(CNC(Cn2c(C)cc(C)n2)=O)CCC12CCN(C(=O)Cc1csnn1)CC2 8219,N1(C(c2cc([N+](=O)[O-])sn2)C(=O)NCC2CC2)CCOc2cccc(F)c2C1 8220,N1CC=CC1(C(N1CC(OC)C1)=O)C(=O)NC(COCC)=O.C1(SC)CCC2(CC2)C1 8221,c1(C(N(CC(CC)NC(c2sc(C)cc2OC(C)C)=O)C)=O)cnc(OC)cn1 8222,Cc1ccc(-n2cc(CC3CCN(C(=O)CC(C)n4cccc4)C3)nn2)cc1Cl 8223,c1(C(N2CC(CNC(CN(C)CC)=O)(OC)C2)=O)cc(C2CC2)n(C)n1 8224,Cc1c[nH]nc1C(=O)NC(C)CC(C)NC(=O)C(c1cncnc1)C 8225,C(=O)(C1=CCCCO1)NCCN(C(C1(O)CCN(C(=O)OC(C)(C)C)C1)=O)C1CC1 8226,c1(C(NNC(C2C(c3cn(C)nc3)OCCC2)=O)=O)c(F)ccc(Br)c1F 8227,C1(CCC(=O)NC2CCCC2CNC(C2CC(=O)N2)=O)CCCCO1 8228,C(=O)(CC(C)CNC(C1C=CCCN1C(=O)CSCCC#N)=O)NC 8229,c1(C(N2C(CN(C(=O)C3=CCN(C)C3)C)CCC2)=O)cnc2nccn2c1 8230,Cc1cn(C)nc1C(N1CCC(CNC(=O)CC2CCC(C(F)(F)F)O2)CC1)=O 8231,C(=O)(C(C)(C)c1cccnc1)NC(c1nocc1NC(C1CCC(=O)N1)=O)C 8232,C1(NC(c2c(OC)csc2)=O)C2CC(O)C1N(C(=O)C=CC1C(C)C1(Cl)Cl)C2 8233,c1(NC(COCCOCC)C)[nH]c(=NCC2(F)CCC2)nc2c1cnn2C(C)C 8234,CN1CCN(C)C(CN(C=O)Cc2ccc(-c3cccc(Cl)c3)o2)C1 8235,C1(C(N2CC(NC(=O)CCc3cnccn3)C3(C2)CC3)=O)CC2CC1CC2(F)F 8236,N1(C(c2c(CC)con2)=O)CC=CC(C(=O)NCC#CC2CC2)C1 8237,c1(CCC(=O)NCC2CCN(C(C(CC#C)C)=O)C2)ccc(Cl)c(F)c1 8238,c1(-n2cc(C3N(C(CSC(C)(C)C)=O)CCC3)nn2)ncc(Cl)cc1Cl 8239,CC1COCC(C(=O)NC(C)(C(=O)NC2CCN(CCF)C2)C2CCC2)O1 8240,C1(C(N2CC(CNC(c3ccccc3)=O)OCC2)=O)C2Cc3ccc(Br)cc3C12 8241,c1(C(CO)NC(c2c(C(C)C)c[nH]n2)=O)ccc(Cl)cc1Cl 8242,C(=O)(C(CNC(C1OCC2CCCC12)=O)CC(C)C)NCc1c(C)nsc1 8243,C(=O)(CCCC(C)(C)NC(=O)C(C#N)C(C)C)NCC(CC)(C)CC 8244,c1(NC2N(C(=O)NC(C(=O)OC)C)CC(F)C2)ncnc2cc(Br)ccc12 8245,C=CCC(CC=C)C(=O)NC(C)(C)CCNC(c1cn(C)nc1C(F)(F)F)=O 8246,Cc1ccc(C(C)NC(=O)CCOCCN(C)C(C2CC2(F)Cl)=O)nc1 8247,CC1CCC(CNC(=O)CCCC2CC2)CN1C(=O)C=CCN1CCCC1 8248,O=S(=O)(CCN1Cc2ccccc2C1=O)c1ccccc1 8249,C1(CC(=O)NC(COC)C2CC2)CC(NC(c2coc(C(F)F)c2)=O)C1(C)C 8250,C(CC(C)(C)C(=O)NCC(c1ccccc1)CNC(C1(F)CC1C)=O)SC 8251,NC(CCOc1ccccc1)C(=O)NNc1nc(Cl)ncc1F 8252,C(CCCNC(C1(Br)CC1)=O)N(C(=O)CNC(c1cscn1)=O)C 8253,C(CS(=O)(=O)CC(=O)NC(C1CC(NC(=O)CN2CSCC2=O)C1)C)OC 8254,N1(C(c2nccc(=NC(C)Cc3ccnn3C)[nH]2)C)CCN(C)C2(CCOC2)C1 8255,C(C(=O)NOC1CC2CCC1C2)(c1ccco1)NC(C1CC1(Cl)Cl)=O 8256,C1(NC(C=CC)=O)CC2CCCC(C1)N2c1cc(C(C)=O)ncn1 8257,C1(NC(CC2CC(SC)C2)=O)C=CCN(C(=O)Cc2ccc(C)cn2)C1 8258,CCCCC(C(=O)NCC1CCC(C(N2CCCC(CCC)C2)=O)CC1)C(C)C 8259,C(CCCCCCCO)=CC(=O)NC1CN(C(C(CN(C)C)(C)C)=O)CC2C1C2 8260,C1(NC(C2(CC#C)CCC2)=O)CN(C(c2ccc(C(F)(F)F)cn2)=O)CC1C 8261,c1(C(N2CCCC(O)(CNC(C(C(C)C)C#N)=O)C2)=O)sc2cccnc2c1Cl 8262,N1(C(C(C)O)=O)CCCC(C2CCCN(CCCOc3cccc(Cl)c3)C2)C1 8263,C1(C(=O)NCC(CN(C(C2(CC=C)CCOC2)=O)C)O)CC2(C1)CC(C)C2 8264,C1(CCNC(c2ccco2)=O)(C(=O)NCC2COCCO2)CCCC1 8265,c1(NCC2(C)CC(NC(CCOCCCOC)=O)C2)cccnc1C(=O)OC 8266,c1(OC)cc(OC)cc(C(=O)NCCCCNC(=O)CCC2CCN(C)CC2)c1 8267,C1(NC(CN(C(COC)=O)C)=O)CC(F)CN(C(=O)C(F)(F)CO)C1 8268,c1(CCNC(C(N2CCC(N(C)C)CC2)C2CC(=C)C2)=O)cccc(F)c1 8269,C1(CNC(C2(CCC=C)CC2)=O)CC2CC1CN2C(=O)COC(C)(C)C 8270,c1(C(=O)NC2CC3CN(C(C45CC4C5)=O)CC3C2)cc2cccc(F)c2s1 8271,CN1CCC(=CC(=O)NCCC2CCN(C(=O)CC3CCC(=O)N3)C2)CC1 8272,C(=O)(C(C)(C)C(F)F)NCC1CCN(C(CCCCN(c2ccccc2)C)=O)C1 8273,c1(C(N2C(C)CN(C(C3(C)CCC(=O)N3)=O)CC2)=O)ccc2ccccc2n1 8274,N1(C(C2CCCN(C(c3c(C)nsc3C)=O)C2)=O)CCCc2occc2C1 8275,C1(CC(=O)NCC2C(C(=O)NCC(COC)(F)F)CCO2)C(=O)NN=C1C 8276,C12(C(N(CC(=O)OC(C)C)C)=O)CC(NC(C3SCC=C3C)=O)(C1)C2.C1C(=O)N1 8277,C1(CNC(c2cccc(O)n2)=O)CC2(C1)CC(O)C2.CC1CC2CN1C2=O 8278,Cc1ccsc1C(=O)NCC1C=CC(NC(=O)C(O)CC2CCCC2)C1 8279,c1(OC(C)C)ccc(-c2nc(C3CCCC(CF)C3)n(CCn3cccn3)n2)cn1 8280,C(C(CC(F)(F)F)NC(C1(O)CC1)=O)NC(c1nc(CC(C)C)sc1)=O 8281,N1(C(C2(COC)CCCO2)=O)CCC(n2cc(C3CCCCC3O)nn2)CC1 8282,N1(C(CN(C2CCC2)C)=O)CC2CCC2(CCNC(=O)C=Cc2nccs2)C1 8283,c1(C(=O)NC2(CC=C)CN(C(c3ccnnc3O)=O)C2)cncc(C(F)F)c1 8284,N(C(=NCCC(C)N(C)C(=O)OC(C)(C)C)NCCF)C1CC(N(CC(C)C)C)C1 8285,Cc1ccc(CCC(=O)NCC23CC(CO2)N(C(C2CCC(C)C2)=O)C3)cc1C 8286,C1(C#N)(C(=O)NCCCCCNC(C2N(C(C)=O)CCC2)=O)CCCOC1 8287,C1(CC(=O)N(CCC(C)C)C2CC2)C(NC(c2cncs2)=O)CC1O 8288,N1(C(c2n(CC#C)cnn2)=O)CCC(C)C1C(=O)NC(C)(C)C#CCC 8289,c1(CC)ccc(C)c(C(N2CCC(CCNC(C3SCC=C3C)=O)CC2)=O)c1 8290,c1(C(=O)NC2C(CNC(c3ccc(O)cc3)=O)C2)cccc(Cl)c1[N+](=O)[O-] 8291,C1(CC(=O)NC2(CC=C)CCC2)CCCN1C(=O)OC(C)(C)C 8292,c1(OC)ncc(Cn2nnnc2N2CCOCC2C(C)(C)O)cc1F 8293,N1(C(CCCc2c(C)ccs2)=O)CCC(C)C1CNC(c1ccccc1CO)=O 8294,Cc1cnc(-c2cn(CCNC(C3C4CC5C(C4=O)C35)=O)nn2)c(C)c1 8295,c1(C(=O)NCC2C(C)CCN2C(=O)C2CC2)ccc2nnn(C(C)(C)C)c2c1 8296,N1(C(C2(OC)CCC2)=O)CCC(C(C)CNC(C2CC(OC)C2)=O)CC1 8297,N1(C(CCOCC)=O)CCC(O)C1C(=O)N(CC(C)(C)OC)C 8298,C(CC(CC)(CC)NC(=O)CC(C)C(C)C)NC(CNC(=O)OCC)=O 8299,N1(C(c2ccc(CNC(C(CCCC)F)=O)nc2)=O)CCC2(CCCOC2)C1 8300,c1(C(=O)OC)cnc2c(=NC(=O)N(c3ccc(F)c(C)c3)C(C)C)nc[nH]n12 8301,C1(CNC(=O)NC(C(C)c2ccccc2)(C)C)CC(C)(C)CO1 8302,C12(CNC(C(c3ccn(C)n3)C)=O)CC(CCO1)N(C(=O)CN1CCSCC1)C2 8303,C(=O)(C(C(=O)N1CCC(NC(=O)C=CCOCCOC)C12CC2)C(C)C)NCC 8304,c1(C(N(C2CCCC(NC(=O)CC=C(Cl)Cl)C2)C)=O)ccnc(-n2cccc2)c1 8305,c1(C(=O)NCC2C3CN(C(CCC(=O)NCC)=O)C(C3)C2)csc2c1CCCC2 8306,N1(C(C2(OC)CC(C)C2)=O)CCN(C(=O)CCn2nc(C)cc2C)CC12CCC2 8307,C(=O)(C(=O)CCc1ccccc1)NC(C)CCN(C)C(c1ccno1)=O 8308,C1(CNC(CC2(C)CC2(Cl)Cl)=O)C2CN(C(c3ccc(N(C)C)nc3)=O)CC12 8309,N1(C(CCC2N(C(=O)CNc3ccncc3)CCCC2)=O)CCC2(CCC2)C(O)C1 8310,c1(OC)c(C(=O)NCC2CCN2C(=O)C#CC2CC2)cccc1C#N 8311,C1(C(N(CC(c2nn[nH]n2)C)C)=O)CC(NC(=O)CC2CNC(=O)O2)C(O)C1 8312,c1(C(=O)NC2CCN(C(CCCCNC(N)=O)=O)C2)ccc(N)cc1C(F)(F)F 8313,C1(C(=O)NCCOc2ccccc2)CN(C(c2csnc2Cl)=O)CCC1(F)F 8314,C(=O)(CC(C)(C)C#N)N1CCC(CNC(C2N(S(CCCC)(=O)=O)CCC2)=O)C1 8315,N1(C(CCCCN(C)C)=O)CC2(CCCN(C(=O)C(C)(C)C3CC3)C2)C1 8316,N1(C(C2(N)CC(C)C2)=O)CCCOC(CN)C1 8317,C1(NC(C(C)N(C(=O)CC2CCOC2)CCC)=O)CCc2n[nH]cc2C1 8318,C(=O)(CC(C)(C)CC(=O)NCC(F)CNC(c1ccc(C)nc1OC)=O)OCC 8319,N1CC2(CCN(C=O)C2)C1.c1(-n2ccc(C)n2)cccc(-c2cn[nH]c2)c1 8320,CC(C)C(O)(C(=O)N1CC(N(C)C(c2cc(O)nc(C3CC3)n2)=O)C1)C(F)(F)F 8321,CC(C)CC(O)C(C)C(=O)N(C)CCOCCNC(=O)CCC[N+](=O)[O-] 8322,C(=O)(C#CC(C)(C)CCC(c1n(CCC)ncn1)=O)NC(c1c[nH]cc1C1CC1)=O 8323,N1(C(C(C)c2ccsc2)=O)CCCC(CO)(NC(=O)CO)C1 8324,C1(CNC(CNC(C(CC)CC)=O)=O)CN(C(c2ns[nH]c2=O)=O)C2(CCC2)C1 8325,CC(C(=O)NCC1OCCC1C(N1CCN(C)CC1C1CC1)=O)C(C)(C)C 8326,C(=O)(CN=c1cc[nH]cc1)N(C1(C(N2CC[Si](C)(C)CC2)=O)CC1)C 8327,c1(C(N2CC(NC(=O)NC(C(=O)OC)C)C(F)(F)C2)=O)cc2ccc(Br)cc2s1 8328,Cc1cc(Br)cc(C(=O)NC2CC(NC(=O)CCS(C)=O)C2)c1F 8329,C1(C(=O)NCC(C2CCN(C(=O)CCn3ccnc3)CC2)(C)C)CC2(CC2)CO1 8330,Cc1onc(Br)c1C(=O)NC1CCC1NC(=O)CC1CCN(C)C1=O 8331,N1(C(C(=O)NC2CC2)=O)CC2CN(C(=O)C(=O)Nc3nccs3)C2C1 8332,N1(C(=O)CC2CC(C(F)(F)F)C2)CCCC2(C1)CN(C(C1(Cl)CC1)=O)C2 8333,c1(C(C)=O)ccc(NC(=O)CC2CC(NC(c3c(Cl)cccc3Cl)=O)C2)c(Br)c1 8334,C1(C(N2CC(C(CC)C)C2)=O)CCC(NC(=O)C(C)O)CC1 8335,CC1CN(C(c2cc(C(N)=O)cs2)=O)CC(C)CN1C(c1ccc(N)c(N)n1)=O 8336,CCCCCC(C)CC(=O)NC1CCN(C(c2cccc3c2CCC3)=O)C1(C)C 8337,C1(C(N2CC(C(N3CC(COC(C)=O)C3)=O)OCC2)=O)CC2(CCC2O)C1 8338,NC1CCC2(CC1)CN(C(=O)Nc1cccn(C3CCOC3)c1=O)C2 8339,CCCCC(CC)CC(=O)NCCCC(C)(C)C(=O)NCC(C)(O)COC 8340,c1(OC)cc(OC)cc(CC(=O)NC2(CN(C)C(C3COC(C)C3)=O)CC2)c1 8341,c1(C(=O)OCC(C=C)(F)F)ccncc1-c1cccc(C(=O)NCC)c1 8342,c1(C(=O)NCCC2CCCN2C(=O)CSc2cnc[nH]2)ccc(C(F)(F)F)cn1 8343,CN1CCC2CN(C(C3CCN(C(=O)CCc4nc(=N)[nH][nH]4)CC3O)=O)CC12 8344,c1(C(=O)NC2CC(C(=O)NC(CCCC)CO)OCC2)ccc(=NC)[nH]c1 8345,CCC(O)C(C)C(=O)NCCC1(OC)CN(C(C2CC2F)=O)C1 8346,CC1(C)Cc2[nH]nc(C(N3CCC(O)(CNC(=O)C4=NOCC4)C3)=O)c2C1 8347,CCC(C(=O)NCCCCCN(C(=O)C(C)c1cccs1)C(C)C)C(C)C 8348,N1(C(=O)OC(C)(C)C)C(CCN(C=O)Cc2c[nH]nc2C2CC2)COC1(C)C 8349,C1(C(=O)NCC2CCCN2C(c2nn(CC)c(C3CC3)c2)=O)CC(C2CCC2)C1 8350,C1(OC)CC2(C1)CC(C(=O)NCC1(O)CC(CNC(=O)C(O)C(C)C)C1)C2 8351,n1(CC)cc(C(=O)N(C2CC(NC(C3CC3C3CC3)=O)C2)C)c(C(F)(F)F)n1 8352,c1(C(C(=O)NCC2(NC(C(c3n(C)ncc3)(C)C)=O)CC2)(F)F)c(F)cccc1F 8353,c1(C(N(CCCCCNC(C(COCC)C)=O)C)=O)cc(OC(F)F)n(C)n1 8354,Cc1cc(C(=O)NC2CC(CCNC(C3(O)CCC(C)CC3)=O)C2)nc(C)n1 8355,c1(C(N2C(CNC(C(C)(C)N(C)C)=O)CC3CC32)=O)cc2n(n1)CC1(CC1)C2 8356,N(C(=NCC(CO)c1ccc(Cl)cc1)NCC(F)F)CC(CN(C)C)(C)C 8357,C(=O)(C1OCCc2c(Br)cccc21)NC1(CNC(c2cocn2)=O)CC1 8358,O=C(C1CCc2ccccc21)N1C2CC1CN(C(C1(F)CC1c1ccccc1)=O)C2 8359,Cc1cc(C(=O)N(CC(C)O)CCNC(=O)CCC2CCCN(C)C2)cc(Cl)c1 8360,c1(CC)occc1C(=O)NC(C(=O)NCCC(O)C1CC1)C1(C)CC1 8361,C1(CNC(COCCCC(C)C)=O)(NC(=O)C(F)n2cccn2)CCCCCC1 8362,Cc1cc(N(C)C)nc(C)c1.c12cnc(cc1C)n(C1CCNCC13CC3)c2=O 8363,N1(C(C2C=C(C)CS2)=O)CCC2(CC2CNC(c2cc(Cl)n[nH]2)=O)C1 8364,N1(C(c2c(CC)nc(C)nc2)=O)CC2CC(NC(=O)C(F)CC3CC3)CC2C1 8365,c1(C(N2CC(CCC)C(C(=O)OC)C2)=O)cc(Br)c(F)cc1F 8366,c1(C(N2CC(NC(C(C)O)=O)CC3(C2)CC3)=O)cc2ccc(Cl)cc2c(O)n1 8367,c1(C(=O)NCC(C23CCC(CC2)C3)NC(CC(C)O)=O)cnn2c1OCCC2 8368,CCC(=O)CCC(=O)N1CC=CC1(C)C(=O)NC1CNC(=O)C1(C)C 8369,C=CC1(CC(N2CCC(C)C2CNC(c2cc(C)cc(C)c2)=O)=O)CCCCC1 8370,C1(CC(=O)NCC2(C=C)CCC2)CN(C(C2CCC2(F)F)=O)CC12CC2 8371,C1(C(=O)Nc2cnccc2C(F)(F)F)CC12CCN(C(C1CC(O)CN1)=O)C2 8372,O=C1CCC(C(=O)NCC2(CO)CCN(C(=O)CCc3cncnc3O)C2)CN1 8373,Cc1ccc(Cl)cc1NC(C1CC(C)(C)CN1C(=O)C(C)N=[N+]=[N-])=O 8374,C1(C(N(CCNC(CC(C=C)C)=O)C2CC2)=O)CC1C1CCOCC1 8375,CCCC(C)(CC)C(=O)NCC(C1CCC1)NC(c1cn(C)cc1C)=O 8376,CC(CS(C)(=O)=O)NC(c1ccc(CNC(C2CCN(C)C2)=O)nc1)=O 8377,c1(C(N2CCC(CC)C2C(=O)NCCN2CCOC2=O)=O)cnc2cc[nH]c2c1 8378,C1(C2CCN(C(C3CC34CC(C)(C)C4)=O)C2)(NC(C(C)OC)=O)CC1 8379,N1(C(C(C(C)C)C)=O)CC2(CCCCN(C(=O)C(C)(C)C(C)(F)F)C2)C1 8380,Cc1cc(O)ccc1C(=O)NCC(C1CC1)N(C(=O)C=Cc1cscn1)C 8381,N1(C(c2cn(CCC)nc2C)=O)CCC(NC(c2cncc(C)c2)=O)CC1C 8382,CC(C)(C)C(C#N)C(=O)NCCOCCNC(C1Cc2ccccc2C1)=O 8383,c1(OC)ccc(NC(=O)C(C2CN(C(C3CNC(=O)O3)=O)C2)SC)cc1C 8384,c1(-c2nc(NC(c3c(OC)c(Cl)c(Cl)cc3)=O)sc2)ccc(Br)c2cccnc12 8385,Cc1cc(C(=O)NC(C(=O)N(C)CCC2OCCO2)C2(C)CC2)nn1C 8386,N1(C(C2(NC(c3cc(O)cc(F)c3)=O)CC(O)C2)=O)CCC2(CNC(=O)O2)C1 8387,C1(NC(C(c2c(C)noc2C)CC)=O)CCCCCN(C(=O)Cc2csnn2)C1 8388,CCCCCCCCCCCC(=O)NCC1CC1CNC(C1CC(F)C1)=O 8389,c1(CC)cc(C(=O)NC(c2cccnc2)C(=O)NCC(C2CCCO2)O)n[nH]1 8390,C1(NC(C2(COC)CCOC2)=O)CCC2CN(C(c3cc(O)cs3)=O)CCC2C1 8391,c1(OC)cnc(C(N2CC(F)(C(=O)NCc3ccc(C)cc3OC)C2)=O)c(F)c1 8392,C(CCCCNC(=O)CC(C1CC1)NC(c1coc(CO)c1)=O)N(C)C 8393,C=CCC(CC=C)C(=O)NCC1CCC1NC(C12CCC(CC1)CO2)=O 8394,c1(C(C)C)cncc(C(N2CCC(F)CC2)C(=O)NC2CCOCC2)c1 8395,c1(NC(N(C)Cc2ccc(N(C(=O)NC(C)=O)C)cc2)=O)ccc(S(C)=O)cc1 8396,C1(C(=O)OC)C2COC(C(=O)NCCN(C(=O)C(C)NC(C)=O)C(C)C)CC12 8397,C(=O)(C1CS(=O)(=O)c2ccccc21)N(CCN(C(C(CC)C#N)=O)C)C 8398,C1(=CCNC(C2CC=CCC2)=O)CCN(C(c2cccnc2C(F)(F)F)=O)CC1 8399,C(=O)(C1=C(Cl)CCOC1)NCC1C(C)CN(C(=O)C=Cc2cccn2C)C1 8400,C12(C(=O)NCCC3(OC)CN(C(C4(C5CCC5)CC4)=O)C3)CCC(CC1)C(C)O2 8401,C(C(O)C(=O)NCCCN(C(=O)CCC1(C)CC1)CC1CCCC1)=CC 8402,CC(C)CC(C)(O)c1cn(C2CC(N(C(=O)CC3CCCC3(F)F)CCO)C2)nn1 8403,N#CC1(C(N2CCC(CNC3CC(N4CCCCC4)C3)CC2)=O)CCCOC1 8404,C1(NCCc2cccc(OC)c2C)CCNCC(C)(C)C1 8405,C(=O)(C1=CC2C=CC(C1)C2)NCC(CC(C)C)NC(c1ccccc1C(F)F)=O 8406,c1(C(=O)NCC2(C(F)F)CCN(C(C(CC)OC)=O)C2)cnc2c(c1)CCCO2 8407,CCCC(C(O)C(=O)NCCC(C)C(=O)OC)NC(C1CC1C(F)(F)F)=O 8408,Cc1noc(N)c1C(=O)NCC#CC(=O)NC(c1cncc(F)c1)C 8409,c1(C(C(=O)NCC(=O)OC)=O)c(OCC2CCOC2C)cccc1Cl.C1CO1 8410,c1(CCCNC(N2CCOCC(CC3(CO)CC3)C2)=O)nc2ccccc2s1 8411,c1(C(=O)NC(CCNC(C(C)SC)=O)C(C)C)cc(C)cc(O)n1 8412,N12CC(C3(CC3)C1)NC2=O.n1(CC#C)cccc1C(=O)OCC1CCCCC1 8413,c1(OC)ccccc1C(C)C(=O)N(CC(C)CNC(c1nocc1C)=O)C 8414,N1(C(C(=O)NCC=C)CC2CC(C(=O)OC)C2)CCC(N2CCCC2)CC1 8415,C1(=O)CS(=O)(=O)CCOCCOCCCN1.CCC(C)C(=O)C(=O)NCC 8416,N1(C(COCCCCC)=O)CC(NC(=O)C(C)Sc2ccccc2)C(O)C1 8417,C12CCN(CC1)CCn1cc2nn1.CC1(C)CC1(Cl)C(=O)NCC1CCOC1=O 8418,C12(NC(Cc3cn(CC)nc3C)=O)CCCC1CN(C(C1(CC)CCCC1)=O)C2 8419,C1(NC(C(C2CCC2)N(CC(=O)NCC2CC2)C)=O)CCC(=O)NC1 8420,C1(CNC(C2CC3C=CC2C3)=O)CC2(CC2)CN1C(=O)COc1ccc(Cl)nc1 8421,Cc1cc(S(=O)(=O)NCCCN2C(=O)CNC2=O)sc1C 8422,CCCCCC(F)C(=O)NC1(CCCC(=O)N2CC(N3CCOCC3)C2)CCC1 8423,C(=O)(CC(C)P(C)(C)=O)NC(=O)CCN1CCCCC1=O.C12CN(C1)C(=O)C2C 8424,O=S(=O)(N(c1ccccc1)C1CC1)N1CCN(CC(F)C(F)(F)F)CC1 8425,N1(C(c2snc(SC)n2)=O)CC(NC(=O)C(C(C)C)N2CCCCC2)C(C)C1 8426,c1(C(N2CCCC(F)(CNC(C(C)(C)OC)=O)C2)=O)ccc2ccoc2c1 8427,N1(C(C=NOC)=O)CCN(C(=O)CCc2ccc(Cl)nc2)CC1CC(F)(F)F 8428,N1(C(C(C)OCC)=O)CC2CN(C(=O)C=Cc3cccc(Br)c3)CC2C1 8429,c1(C(CNC(C=CC(C)NC(=O)CN(C)C(=O)C2CC2)=O)C)ccccc1 8430,N1(C(C(CC(N)=O)NC(c2cc(CC)ncn2)=O)=O)CCCC2(C)CCCC12 8431,c1(C(=O)NCC2CN(C(c3cc(C)c(C)[nH]3)=O)CC2O)ccc2nnnn2c1 8432,C1(CC)C(C(N2CC(CCCCNC(c3ccc(SC)o3)=O)C2)=O)CCN1C 8433,Cc1ccc(C)c(C(=O)NC2CN(C(c3nnn(C)c3C)=O)CCC2F)n1 8434,C1(CCOC)CCCCC1.C=C1CC(C2CN2)C1.C1(=O)CCN1.C(=O)(COC)N 8435,CC#CCCCC(=O)N(C1CCN(C(=O)C(C)C2(O)CCC2)C1)CC 8436,C(CCCCN=c1[nH]c(=N)[nH]c(=NC2CCCN(CC)C2)[nH]1)OC 8437,C(=O)(C#CC1CCC1)N(C1CCN(C(C2CC2CNC(=O)OC(C)(C)C)=O)C1)C 8438,C1(CC=C)(NC(=O)C(C)CN2CCCCC2)CN(C(C2(OC)CCC2)=O)C1 8439,c1(C(=O)NC(C)CN(C(=O)Cc2cncs2)C)cc(Cl)ccc1OCC#N 8440,N1(C(CCCSC)=O)CC2(CCC2)CC1CNC(C1CCCCC1N=[N+]=[N-])=O 8441,N1(C(c2ncc(N)nc2)=O)C2CCC1CN(C(=O)COC1CCCCC1)C2 8442,c1(C(C)=O)ccc(C(=O)NC2CC2C(=O)NCc2c(F)cccc2F)cc1O 8443,C1(C(N(CC(C)NC(=O)CCSC(F)(F)F)C)=O)CCC2(CCCC2)C1 8444,Cc1cc(C(=O)NCC2CCC(NC(C3CCCCCC3)=O)C2)oc1C 8445,N1(C(c2scc(C(=O)NCc3ccc(C)cc3)n2)=O)CCc2ccncc2C1 8446,C1(O)(CC(=O)NCCC(CNC(CN(c2ccc(O)cc2)C)=O)O)CCCOC1 8447,C1(NC(c2c(C)oc(Cl)n2)=O)C2CCC1CN(C(c1ccc3nccn3n1)=O)C2 8448,N12CC3CN(CC3C1)C(=O)C2C.c1(C(=O)N(CCCCC)C(C)C)ncc(Cl)cc1Cl 8449,C1(C(=O)NCC(c2ccccc2)CNC(c2cc[nH]n2)=O)(CC)CC1(F)F 8450,N#Cc1c(NC(=O)CC2CCCN2Cc2cccc(F)c2Br)cc(Br)cc1F 8451,c1(C(=O)NC(C(N2CCC(C(F)F)CC2)=O)Cc2ccoc2)c(O)cccc1Cl 8452,c1(CC(N2CCC(NC(CC=C=C)=O)C2(C)C)=O)ccc2oc(O)nc2c1 8453,C1(C)(NC(Cc2cc(C(C)=O)c(C)o2)=O)CCCN(C(c2ccc(CF)cc2)=O)C1 8454,C1(=CC(=O)NCCC(CCNC(C(C)OCC=C)=O)C)CC2CCC(C1)N2C 8455,N1(C(C)=O)CCc2cc(CC)ccc21.N1(C(C=O)=O)C2CCC1CC2 8456,C1(C(=O)NC(C(C)CO)C)(CCO)CCN(C(=O)CN(C)C)C1 8457,N1(C2CN(C(CC3(OC(=O)OC(C)(C)C)CC3C)=O)C2)CC2CC2(NC=O)C1 8458,Cc1ccc2c(=NC3COCCOC3)[nH]c(=NCc3nc(C)c(C)[nH]3)[nH]c2c1 8459,N1(C(C(CCSC)O)=O)CC2CC(N(C)C(c3cccc(SCC#N)c3)=O)C1C2 8460,C(CCCCC(=O)NC1COCC1NC(C1CC1c1ccn(C)n1)=O)NC(C)=O 8461,CC(C)CC(CNC(=O)CCSC(F)(F)F)NC(=O)CNC(=O)C1CC1 8462,C12CC3CCCC(C1)N3C(=O)CCOC1(CC1)C(=O)N2.C1CCC1.CC(=O)OC 8463,C(=O)(CC(CC(C)C)NC(=O)CC1CC2CC2C1)NCCc1cc(CC)no1 8464,Cc1c(C(N2CCCC2CN(C)C(c2cc(C(F)(F)F)on2)=O)=O)c(Cl)nn1C 8465,N1(C(C2C(NC(C(C)CC(N)=O)=O)CCO2)=O)CC(C)(C)OCC1C 8466,C(=O)(CP(C)(C)=O)NCC1C(NC(CCN(C(C)=O)C)=O)COC1 8467,N1(C(COCC(=O)OC)=O)CCOCC1CNC(C1(C)CNC(=O)C1)=O 8468,N1(C(c2c(CC)c[nH]c2)=O)CCC2C(CCCN2C(c2ccc(N)cc2Cl)=O)C1 8469,c1(N(C(=O)NCCOC)C)coc(OCCCCO)n1.c1(O)ccccc1 8470,c1(CN(C(C(=O)NC2CCC(C(=O)OC)C2)C2CC2(Br)Br)C)cc(Br)ccn1 8471,C=CC(CC(=O)OC)C1CN(C(COC(F)F)CO)C1 8472,c1(-c2c(CCOC)cccc2)cccc2c1CN(Cc1ccc(F)nc1Br)CC2 8473,Cc1cc([N+](=O)[O-])cnc1C(N1CC2C(CNC(=O)CC3CC=CCC3)C2C1)=O 8474,C(=O)(CCCS(C)(=O)=O)NC1(C)CC(NC(C2(O)CC(C)(C)C2)=O)C1 8475,N1(C(C2N(C(c3cc(OC)n[nH]3)=O)CC(F)C2)=O)CCC2(CCN(C)C2)C1 8476,c1(CNC(c2nnnn2C(C)CC)CCOCC)ccc(OC)c(C)c1 8477,Cc1cc(N2CCC(N(C(=O)C(F)CC3CCCCC3)C)CC2)ncc1C#N 8478,C1(CC)CN(C)CCN1C(=O)CC(CNC(=O)CS(C)(=O)=O)OC 8479,N1(CC#C)CCCC1C(=O)NC(C(=O)OC1CCCC1)C 8480,N1(C(c2c(C(C)C)nn(C)c2)=O)CC(N(C)C(C2CCOCC2)=O)C2(CC2)C1 8481,C1(C(N2CCCC(CC3CC3)C2)=O)(OC)CCN(C(c2c[nH]ccc2=O)=O)C1 8482,C(=O)(C(C(C)C)N1CCCC1=O)NC1C(CNC(C2CN(C(C)=O)C2)=O)CC1 8483,c1(NCC2(CNC(=O)CS(=O)(=O)NC3CC3)CC2)nc(Cl)nc2[nH]c(O)nc12 8484,C1(C(=O)NCC2C(CC(=O)NC(C#C)C3CC3)C2)CC2(CCC2)C1 8485,C1(C(=O)NCCCNC(C(C(C)C)n2ccc(C)c2)=O)CC2OC1C1CC21 8486,Cc1cc(C)c(C(N2CCC(C3CC3)C2CNC(=O)CP(C)(C)=O)=O)cc1C 8487,CCCCC(O)C(C)C(=O)NCC#CC(=O)NCC1(CSC)CC1 8488,C1(NC(CC(CC)(C)C)=O)CCN(C(=O)C(C)(O)C(C)(C)C)CC(C)(C)C1 8489,c1(CCCC2N(C=O)CCC2)cccc(C2(N3CCCC3)CCC2)c1 8490,c1(C(=O)NCC(c2cccc(Cl)c2)NC(C=CCCC)=O)ccccc1C1CC1 8491,N1(C(CN(S(CC)(=O)=O)C)=O)CCC(C)(C)C1CNC(C1CC2(C1)CC(O)C2)=O 8492,N1(C(C(C)OC)=O)CCCN(C(c2ccc(SCC(N)=O)cc2)=O)C(C(C)C)C1 8493,c1(CNC2C(C(=O)NCc3ccc(C)cc3C)C2)ccc(F)c(F)c1C 8494,N1(CCC(=O)N(C)C2CC2)CCCCC(NC(=O)CC=CCc2ccccc2)C1 8495,CC(C)(C)C(C)(O)C(=O)NCC1(C)CCCN1C(c1cnc2n1CCS2)=O 8496,C(=O)(CC1=NN(C)C(=O)C1)NC1CN(C(C(C)n2ccnc2)=O)CC1C 8497,C(C)(C)(CCCF)NC(c1c(CNC(C2(C(C)C)COC2)=O)ccs1)=O 8498,c1(NC(=O)NC2(c3ccccc3)CC(F)C2)ncc(C(F)(F)F)cc1Cl 8499,CCC(CNC(=O)Cc1cn(C)nc1C(F)(F)F)(CC)NC(C1CSCCS1)=O 8500,CC(C)(F)CCC(=O)NCc1cc(C(=O)NCCc2ccns2)no1 8501,N1(C(=O)C2=COCCC2)CCOC2(C1)CN(C(c1cscn1)=O)C2 8502,S(=O)(=O)(c1ccc(=NCC2CC23CCC(F)(F)CC3)[nH]c1)N(CCOCC)C 8503,CCCC(CNC(=O)CC(C)C)C(=O)N1CC(=O)NC(CC)C1 8504,C(C)(C(=O)NCc1ncnn1CC)(C1CCC1)NC(C(C)OCCC=C)=O 8505,C1(NC(CC(CC)OC)=O)CCC2CN(c3nnc(-c4ccon4)s3)CC12 8506,Cc1c(C(N2CCC3(C=CCOC3)CC2)=O)cccc1S(C)(=O)=O 8507,C#Cc1cnc(C(=O)NCc2ccc(C(=O)N(C)Cc3cocn3)s2)c(C)c1 8508,c1(OC)ccc2cc(C(=O)NCC(C)(C(C)C)NC(=O)COC(F)F)[nH]c2c1 8509,C1(NC(C2(C(CC)(F)F)CC2)=O)C2CC(NC(=O)CCC3CCN(C)C3)CC12 8510,CCCCCC(O)CC(=O)N1CC2CC1CN2C(C1CCc2nccn2CC1)=O 8511,c1(C2(C(=O)NC(CN(C(c3n[nH]c(C)n3)=O)CC)C)CCC2)ccccc1C 8512,Cc1cc(C(C)C)ccc1C(=O)NCC1CN(C(=O)CC(O)C2CCCC2)CC1C 8513,C1(OC)CC(C(=O)NCCC2CCN(C(c3cnc(O)n3C)=O)C2)CC1OC 8514,N1(C(c2cc(C)sn2)=O)CCC(C(C)(C)C)(CNC(C2CC2C#N)=O)C1 8515,N1(C(c2c(C)csc2)=O)CCC2(CCN(C(C3CN4CCN3C(C)C4)=O)C2)C1 8516,c1(C(N2CC3CN(C(CCc4scc(C)c4)=O)C3C2)=O)ccc2ccoc2c1 8517,c1(-c2cccc(CN3C(CO)CSCC3)c2)ccnc2c1CCC2.c1ccccc1 8518,c1(CNC(C(CC)(F)F)=O)nnc2n1CCN(C(c1nocc1Br)=O)C2 8519,C1(NC(CONC(CCOC(C)C)=O)=O)Cc2ccccc2C1C 8520,Cc1c(C(N2CCC(NC(=O)Cc3cnoc3)C2C)=O)c(O)nc2ccccc12 8521,C12(C(=O)OC)CC3CC1C2C3N(C)CCc1ccccn1 8522,C(=O)(C(O)(CN(C)C)C(F)(F)F)NCC1C(NC(C2(OCC)CC2)=O)C1 8523,C1(CNC(c2ccn(C(CC)C)n2)=O)(NC(=O)C=C(C)C(F)F)CCCCC1C 8524,C1(C(C)C)CCN(C(C2CC3(C2)CC3F)=O)C(CNC(C2CCOCC2)=O)C1 8525,C(=O)(C1=CCCCCC1)C1(C)CN(C(N2CCCC23CC3)=O)C1 8526,N1(C(C(c2ccc(OC)cn2)(F)F)=O)CCC(CNC(c2cocn2)=O)CC1C 8527,N1(CCNC(=O)NCCN(C(CC)COC(C)(C)C)C(C)C)CCC(C)CC1 8528,c1(C(N(C2CCCN(C(=O)CCOCC(F)F)C2)CC)=O)cnc2nccn2c1 8529,N1(C(C(C)O)=O)CCN(C)C(CNC(c2cc(C3CCC3)nn2C)=O)C1 8530,C1(OCC(=O)OC(C)(C)C)CCN(C(=O)C(F)(F)C=Cc2ccccc2)CC1 8531,N1(C(c2c(C)[nH]c(=N)s2)=O)CC(CNC(=O)C(C)CC(C)(C)C)CC(C)(C)C1 8532,c1(CNC(C2C3(CCN(CC(=O)NCC)CC3)C2)=O)cc2cc(C)ccc2s1 8533,N1(C(CN2CCN(C)CC2)=O)CCN(C(c2nc(=O)n(C)[nH]2)=O)CC1CC1CC1 8534,C(CC(=O)NCCC(C)(C)F)(C(F)(F)F)NC(c1ccc(C#C)cc1)=O 8535,c1(C(C)NCc2ccsc2C(F)(F)F)cc2ccccc2oc1=O 8536,C=CCCCC(C)(C)C(=O)NC1CC(N(C)C(c2ccc(C(=O)OC)n2C)=O)C1 8537,c1(OC)ccc(C(N2CC(NC(=O)CCNC(C)=O)C(F)C2)=O)c(F)c1F 8538,c1(C(C(=O)NC)N(C(CCC)C(=O)NC(C)C)C)cc(CO)cc2ccccc12 8539,C1(C)(OC)CCCN(C(=O)CCCC(C)NC(=O)C(C)=CC2CC2)C1 8540,c1(CN(C(=O)C(O)CSC)CC#C)ccc(C(F)F)cn1 8541,CCC(C)(C)CC(=O)NC(CCN(C)C)C(=O)N1CC(N(CC(C)C)C)C1 8542,c1(CC(=O)NC2CCN(C(C3C(C(=O)OC)C3)=O)C23CC3)csc2ccccc12 8543,CC1(C)CC(NC(=O)CN(C(=O)CCCn2cccn2)C2CCCSC2)C(=O)O1 8544,C1(CC(=O)O)CCCCC1C(=O)NCc1cc(C)ns1 8545,C1(C(=O)OCC)(C(=O)NCC2(O)CN(C(=O)CCC3CC3)C2)CC12CC2 8546,CC1CC(C(=O)NC2CN(C(=O)C=Cc3cc[nH]n3)CC2n2ccnn2)CN1C 8547,N1(C(C=CSC)=O)CCC2(CCC2)C(CNC(c2nc(C(F)(F)F)oc2C)=O)C1 8548,C1(C#N)(C(=O)NCC2(C)CCN(C(c3c(COC)cccc3)=O)C2)CC2CC2C1 8549,Cc1cc(C(=O)NCC(C)(F)CNC(=O)C(C)C(C)(F)F)cc(C)c1F 8550,S(=O)(=O)(c1[nH]cnc1C)C(N1C(c2occ(C)n2)CCC1)=O 8551,C(C(C(C)(C)C)NC(=O)Cc1cccc(C(F)(F)F)c1)NC(C(C=C)O)=O 8552,c1(C(N(C)CC2(NC(C3CC3c3cnc[nH]3)=O)CC2)=O)ccc2nccn2c1 8553,CCC(C)(CC)C(=O)NCCCCC(=O)Nc1cn(C)nc1Cl 8554,N1(C(CC(C)(C)O)=O)CCN(C(c2ccnn2CC(F)(F)F)=O)CC(O)C1 8555,Cc1cc(C)c(C(=O)NCCC2CN(C(C3CC(C)C3)=O)CCS2(=O)=O)cc1C 8556,c1(CNC(c2c(CNC(C(CO)OC)=O)n[nH]c2)=O)cccc(C)n1 8557,c1(COC)cc(C(=O)NCC2C3COCC23)on1.n12cc(nn1)C(=O)N1CC2C1 8558,CC1CCCN(C(=O)C=CC=C(Cl)Cl)C1CCNC(=O)CCC(N)=O 8559,C(=O)(CC(=O)NC1CCCC1CNC(c1coc(Br)n1)=O)NCC 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8651,C1(CCC(=O)NCC(CSC)OC)CCCCN1C(=O)CCCC1CC1 8652,CCC(C)C(O)CC(=O)NC1CCC(CC(N2CC(F)(F)CC2C)=O)CC1 8653,n1(CC(=O)NC2C(C)CCN(C(C34CCC(C3)C4)=O)C2)ccc(=O)c([N+](=O)[O-])c1 8654,C1(CNC(c2ccc(Cl)nc2)=O)CN(Cc2cc(Br)c[nH]2)CCO1 8655,S(=O)(=O)(c1ccc2nc(O)sc2c1)N(CC)CC1CC1 8656,C(CCC(C)(C)C)NC(c1c(CNC(C(C)=C(C)C)=O)n[nH]c1)=O 8657,Cc1ccc(C(=O)NC2CC3CC2N(C(=O)CN2CCC(C)CC2)C3)c(O)n1 8658,N1(C(C(CC)C(C)C)=O)CCCC2(NC(=O)Cc3cc[nH]n3)CC2C1 8659,c1(C(C)=O)c(C)[nH]c(C(=O)NCC2(O)CC(CNC(=O)CCC3CC3)C2)c1C 8660,c1(OC(C)C(=O)NC(=O)NCC(=C2CCCC2)F)ccc(F)cc1F 8661,c1(C(N2CC(F)(CNC(c3ccc(CO)o3)=O)C2)=O)cc(F)c(Br)cc1F 8662,N1(C(CSCC=C)=O)CCc2sc(CNC(=O)CCOCC(C)C(C)C)nc2C1 8663,CC1CNC(C(c2ccccc2)NC(=O)C(=O)NCC2CCCCC2)C1 8664,c1(CSCC(=O)N(CC(C)NC(CNC(C)=O)=O)C)coc(-c2ccccc2)n1 8665,C1(C(N2C(CCNC(COC)=O)CCC2)=O)CCC(F)(F)CC1 8666,C#CCCCC(C)C(=O)NCC(C(=O)NC1CC(O)C(F)C1)N(C)C 8667,CCCS(=O)(=O)c1ccc(C(=O)NCC2CCC(C)CN2C(=O)C(N)=O)cc1 8668,c1(CN2CCC(CC(=O)Nc3c(OC)ccnc3)C2)ccnc(Cl)c1Cl 8669,C(CCN=c1[nH]c2cc(Br)cnc2s1)N(C(C(C)CSC(F)(F)F)=O)C 8670,C1(CC)CC(CC(N2CCN(C(=O)C(F)=C3CCC3)CC2)=O)C1(C)C 8671,C1(CNC(Cc2c(SC)cccc2)=O)CCC2(CN(C(=O)CC3CN(C)C3)C2)O1 8672,CC(C)(CC(=O)N1CCC(CNC(C2C3CCCC23)=O)CC1)CC(F)F 8673,C1(C(=O)NCCN(C(C)C)C)CCCCN1C(C1CC1(F)F)=O 8674,CCCCC(C)C(=O)OCC1(F)CCCN(C(=O)OC(C)(C)C)C1 8675,C12(C(N3CC(N(C)CC)C3)=O)CC1CN(C(=O)CCC(=O)OC)C2 8676,C(=O)(CS(=O)C(F)(F)F)N(CC(C)N(C(CNC(C)=O)=O)C)C 8677,C(N=c1[nH]c(=NCCCc2nccs2)[nH]c2cccc(F)c12)c1cc(CC)on1 8678,n1(CC(=O)NCC(CNC(C2(C)CCOCC2)=O)O)cnc([N+](=O)[O-])c1 8679,C1(C(=O)NC(C(C)NC(C2(CF)CC(F)(F)C2)=O)C)CC(=O)NC(=O)C1 8680,C1(C(N2CCC(C)(CNC(c3cnc(NC)s3)=O)C2)=O)CC(C)CC(C)C1 8681,N1(C(COCCCC(C)C)=O)Cc2nccn2CC(NC(C2CCC2)=O)C1 8682,C12(CNC(C(CSC)OC)=O)CC(NC(=O)C(C)Cc3ccccc3)(C1)C(C)O2 8683,C(=O)(C1CCc2c[nH]nc21)NC1CC2CN(C(c3n(CC)nc(C)c3)=O)CC21 8684,N1(C(CC=CCC)=O)CC2COCCC2(NC(c2ccc3c(c2)CCC3=O)=O)C1 8685,C1(C(=O)NC(c2cccc(Br)c2)C)CC12CCN(C(c1cncc(Br)c1)=O)C2 8686,C1(CC(=O)N(C2CN(C(C3CCSCC3)=O)CC2O)C)CCCC(C)(C)O1 8687,N1(C(c2c(OCC)ccc(Cl)c2)=O)CCN(C(=O)N=CC(F)(F)F)C(C)CC1C 8688,C(CN=c1[nH]cnc2c(Cl)cc(Cl)cc12)C1CCC(NC(c2c[nH]c(Br)c2)=O)C1 8689,N1(C(c2c(C)cn(C)c2)=O)CCN(C(=O)C(C)C2=CCCC2)CC1C(C)C 8690,C1(C(N(C2CCC2)CC#C)=O)CC2CCC(C1)N2C(=O)Cc1ccon1 8691,c1(C(=O)NCC(CC=C)NC(=O)C(n2ccnc2C)C)nc(C)ccc1OC 8692,c1(C(N2C(CC=C)(C(=O)NCC3(CCC)CC3)CCC2)=O)cnn(C)c(=O)c1 8693,CC1=C(C(=O)NCC2CCCCN2C(c2cccc3nonc23)=O)CCCC1 8694,c1(C2C(C(=O)NCC(C)NC(=O)C=C3CCCC3)CCC2)nnc(S)n1C.C1(C)CC1 8695,C1(CC(=O)NCC(C)(C)OC(C)C)CC(F)CN1C(=O)Cc1cnns1 8696,C#CCCCCCC(=O)NCC1(CNC(C2CC2(Cl)Cl)=O)CC1(F)F 8697,C12(C(N3CCC(C(C)NC(C4COC(=O)N4)=O)CC3)=O)CCC(CO)(CC1)CC2 8698,c1(C(N2CCC(NC(C(C=CCCC)O)=O)C(O)C2)=O)cnc2n1CCOC2 8699,O=S(=O)(c1ccc2c(c1)CC2)NC1CCc2ccccc21.c12ccccc1O2 8700,N1(C(C2C(c3c(C)ccs3)C2)=O)CC(NC(c2cncc(N)c2)=O)C(C(F)F)C1 8701,c1(CN2C(C(=O)NC3CCN(CCC)CC3)CC3(CC3)C2)cc(OC)c(O)c(Br)c1 8702,c1(OC)ccc(C(=O)NC(C)CC(C)NC(c2cncnc2)=O)cc1C(F)F 8703,N1(C(C(C)=C(CC)C)=O)CCC2(NC(C3CS(=O)(=O)C3)=O)CCCCCC12 8704,N(C(=NCCOCC)NCc1ccc(CSC)cc1)c1ccc(OCC=C)cc1 8705,C1(N(C(C2CN(C)C2)=O)C)CCCCC1N(C)C(c1ccccc1OCCF)=O 8706,N1(C(C2N(CC)CC2)=O)CCC2CN(C(=O)Cc3ccc4c(c3)CC4)CC12 8707,C12(NC(C3N(CC)CC3)=O)CC(C1)N(C(=O)CCn1cc(Cl)cn1)C2 8708,C1(NC(C2(C(=O)NC)CCC2)=O)CC2CC(C1)N(C(=O)Cn1cc(Cl)c(C)n1)C2 8709,c1(-n2cc(C(=O)NC(C)CCN(C)C(C3CC(C#N)C3)=O)nn2)ccccc1Cl 8710,c1(OC)cnc(C(N2CCCCC2CCCNC(=O)Cc2c[nH]nc2C)=O)cn1 8711,C1(NC(CC2(CSC)CC2)=O)CN(C(=O)C(F)(F)COC)CCC1C(F)(F)F 8712,C1(C2CCCN(C(C3CC(F)C3)=O)C2)(NC(C(C)NC(=O)CC(C)(C)C)=O)CC1 8713,c1(-c2ccc(OCC)cc2)ccc(=NCc2ccc(OC(C)C)cc2)[nH]c1 8714,c1(OCCN(C)C)ccccc1S.C1(C(=O)N)C2CC1N(C(=O)CN1CCSCC1)C2 8715,c1(N(C)CCO)ccc(-c2csc(CC(N3CCC(=O)NC3=O)=O)n2)c(O)c1 8716,C=C1CCC(C(N2CCCCC2CNC(=O)C(C)CCO)=O)CC1 8717,C1(OCCNC(CCOC(C)=O)=O)CC(NC(=O)CNS(N)(=O)=O)C1 8718,C1(C(=O)NCCN(C2CCCCCC2)C(=O)CN2CC=CC2)CC2CCC(C1)O2 8719,N1(C(C23N(C(Cc4ccc(C)cc4)=O)CC(C)(C2)C3)=O)CCC2(CC1)CSC2 8720,c1(OCC(=O)NCC2CC(CNC(=O)CCF)CO2)ccc2c(c1)CCCC2 8721,N1(C(CCCC(C)NC(C(CC)N(C)C)=O)=O)Cc2ccccc2C1 8722,c1(OC)cc(C(=O)NCCC(O)CNC(=O)C(C)(C)C)ccc1[N+](=O)[O-] 8723,C(=O)(C1=CS(=O)CCC1)NCC1(C(=O)NC(c2cocn2)C)CC1 8724,CC(N=c1cccc(S(=O)(=O)NCC23CCCC2C3(F)F)[nH]1)c1cn[nH]c1 8725,C1(O)(CCNC(CC=C(C)C)=O)CCN(C(=O)C(C(C)(C)C)C2CCC2)CC1 8726,N1(SCNC(N(C)CCc2ccccc2S(C)(=O)=O)=O)CCc2cc(F)cc(F)c2C1 8727,N1(C(CNC(=O)C2CC2)=O)CCN(C(=O)C(O)C2CC2)CC2(CC2)C1 8728,C(CN=c1[nH]c2c(c(=NC(C)c3cncc(F)c3)[nH]1)CCC2)(C1CCCC1)OC 8729,c1(C(=O)NCC23CN(C(c4n(C)nnc4)=O)C(CC2)C3)c(S(C)(=O)=O)cnn1C 8730,N1(C(C2(C)CCCCC2)=O)CCS(=O)(=O)CC1.n12cc(nn1)NC(=O)N(C)C(C)C2 8731,c1(CCC)noc(CCC(=O)NC2CCCC2NC(C2CC2C)=O)n1 8732,N1(C(C(F)=C(C)C)=O)CC2CC(C1)CN(C(C1CC(=O)N(C3CC3)C1)=O)C2 8733,C(CCCCC(=O)NCC1CC2CN(C(c3c(C)nn(C)c3F)=O)CC12)SC 8734,c1(C(c2n(CCCOC)nnn2)NCC(C)CC(C)C)cn(C)c(C)cc1=O 8735,c1(C(=O)NC(C)CCN(C(=O)CC(F)(F)C(F)F)C)cc2c(nn1)CCCO2 8736,c1(C(N2CCC(NC(=O)CC3(CO)CC3)C2)=O)cc(-n2ccnc2)ccn1 8737,c1(CC)cc2cc(Br)ccc2c(OC)c1C.C12CCC(CC1)NC2=O 8738,C1(C(=O)NC2(CCCC)CCC2)CCCN(C(=O)Cn2cc(C#N)cn2)C1CC 8739,C(=O)(C1=CCCCC1)N1CC2C(CN(C(=O)C(F)(F)C3(O)CCC3)C)C2C1 8740,C1(NC(=O)CSC(F)(F)F)COC2(CCN(C(C3CC34CCSCC4)=O)CC2)C1 8741,CC(CC(F)(F)F)C(=O)NCCCCN(C)C(C1(C)CCNC1=O)=O 8742,Cc1ccc(F)c(C(=O)NCC(C)CN(C)C(C23CCC(C2)OC3C)=O)c1 8743,c1(C(C)=O)ccc(NC(C2CCC(CNC(=O)C3CC3)CO2)=O)cc1Cl 8744,c1(N(C)C)ccc(C(=O)NC2CC(CNC(=O)Cc3cnn(C4CC4)c3)C2)cc1 8745,Cc1nc(O)c(Br)cc1C(=O)NCCCNC(=O)Cc1ccc(O)nc1 8746,C(=O)(C(F)(CC)C(=O)OC)N1CCC(N(C(c2c(CC)occ2C)=O)CC)C1 8747,c1(CC)ccc(C(=O)NCC(C(C)C)NC(=O)C(c2cnccn2)C)c(Cl)c1 8748,N1(C(c2nc(CC)sc2)C(=O)NCc2nnn(C)n2)CCOC(C2(C)N=N2)C1 8749,CCCCC(CNC(=O)C(C1CCOC1)OC)NC(=O)CSCC(N)=O 8750,N1(C(CCCCOC)=O)CC=C(CNC(=O)CCCCC2CCCCC2)CC1 8751,c1(NC2CCN(C(C=CCC)=O)CC2CC)c(Cl)cccc1[N+](=O)[O-] 8752,c1(N2CCCC(OCCOC)C2)nc(=N)[nH]c(=NCC(=O)NC2CC2)[nH]1 8753,Cc1sncc1C(=O)N(C(C)CCNC(=O)CC1(C)CC1)C 8754,N1(C(C2=CCN(C(C3CN(C)C(=O)CC3)=O)C2)=O)CC2(C1)NC(=O)NC2=O 8755,N1(C(c2c(C)occ2)=O)CCN(C(c2ccc(N=[N+]=[N-])cc2)=O)CCC1C 8756,c1(N2CC(CC)SCC2)nc(=NCC(C)C(C)(C)C)[nH]c2c1CSC2 8757,Cc1nnccc1C(=O)N(C)CC1CCCN(C(C2CC(C)(C)O2)=O)C1 8758,c1(C(=O)NCC(C)CNC(C2CCC(C(F)(F)F)O2)=O)nsc2c(Cl)cccc12 8759,C1(CCNC(C2C(C)(C(C)C)C2)=O)COCCN1C(C12CC(C1)C2)=O 8760,c1(C(=O)NC(C(C)C)CNC(C2CC(CCN(C)C)C2)=O)ccc(Cl)nc1 8761,c1(N(c2ccccc2Cl)CCCOCC)cc(Cl)nn(C)c1=O 8762,Cc1ccnc(C(=O)NC(C2CCOC2)CNC(=O)C(F)(F)c2ccccn2)n1 8763,C(=O)(C1=NNC(=O)CC1)Nc1ncc(CNCCn2c(C)ncc2)s1 8764,N1(C(c2ncc(I)s2)C(=O)NC(C2CCCO2)C)CCC(N(C2CC2)CC)CC1 8765,CCC(CC(F)F)C(=O)NCC(C)CNC(c1c[nH]c(=N)o1)=O 8766,CC(O)CCCCCC(=O)N1CCC(CN=c2[nH]nc(C3CC3)s2)C(C)C1 8767,CC(C)CCC(N)C(=O)NCC(c1ccco1)N1CCCC1 8768,C#CCCC(O)C(=O)N1CCCCC1CNC(c1cnccc1C)=O 8769,C1(NC(C#CC(C)C)=O)CN(C(=O)C(C)(C)c2ccc(C(F)(F)F)s2)CC12CCC2 8770,C1(C(N(CC(C)(C)NC(c2c(CC)nco2)=O)C)=O)CCCCC1(F)F 8771,C1(CNC(=O)Cn2cnnn2)CN(C(c2cccc(-c3nc[nH]n3)c2)=O)CCO1 8772,C(=O)(CC1=CCCC1)NCC(CC)NC(c1ccccc1NC(C)(C)C)=O.C(N)(=O)N 8773,C1(COC)(CNC(=O)CCNC(=O)NC2CCC(=O)C2)CCCO1 8774,CC(C)(C)C(O)CC(=O)N1CC(CNC(c2ccc(C(F)(F)F)[nH]2)=O)C1 8775,C(=O)(C1Cc2c(Cl)cccc21)NC1CCCN(C(c2nnc(CC)o2)C)CC1 8776,C1(NC(c2c(CCC)nns2)=O)CCCCCC1NC(=O)C(C)(C(C)C)OC 8777,CN1CCCCC1C(N1CCCC1(C)CNC(c1cc(C2CC2)ncn1)=O)=O 8778,C1(NC(c2c(C)csc2)c2nnnn2C2CCCCC2)CC(C)OC(C)C1 8779,c1(C(N(CCNC(C2(C)CCN(C)C2)=O)CC)=O)c(Cl)ccc(O)c1N 8780,Cc1cc(F)cc2c1N(C(c1cnc(C)n1-c1ccccc1)=O)CC2 8781,Cc1ccn(C(C)(C)C(=O)NC2(C)CC(NC(=O)C(N3CCOCC3)C)C2)n1 8782,c1(N)nc(C)ccc1OC.C1(C)(CC(=O)N(CCC)CCNC(=O)COC)CCCC1 8783,c1(CC(N2C(CNC(C3C(CC)OCC3)=O)CC2)=O)cccc(F)c1O 8784,Cc1cnc(NCc2c(C)cccc2C)c(S(=O)(=O)N2CCC(C3CCC3)C2)c1 8785,C(=O)(C#CC1(C)CCCO1)NCCC1(CNC(c2c(C)nn(C)c2N)=O)CC1 8786,c1(CC)nn[nH]c1C(=O)N(C)CCNC(C1(COC)CCOC1)=O 8787,C1(C(=O)NC(C(N2CCCC(OCC)C2)=O)C)CCC2(CCC2)C1 8788,N1(C(C2C(C(N)=O)COC2)=O)CC(F)CC1CO.C1(O)CCOCC1.C1(=O)NCCO1 8789,C(=O)(C1SCCc2ccccc21)N1CC(NC(CSC)=O)C(F)CC1 8790,C1(N(C(=O)CCCCO)C)CCCN(C(c2cccc(F)c2N)=O)CC1 8791,c1(C(N2CC3C(CNC(C(C)c4cccs4)=O)C3C2)=O)coc2cccc(O)c12 8792,c1(C(N2CCCC3(NC(C=CCCC)=O)C(C2)C3)=O)cc2c(cc1O)CCCC2 8793,CC(C)C(O)C(C)C(=O)N(C(C)(C)CC(=O)NC12CCC(C1)OC2C)C 8794,CN1CCNNS(=O)(=O)c2cc([N+](=O)[O-])ccc2C(=O)N(C2CC2)C2(Cl)CCC12 8795,c1(C(N(CC(=O)N(C(C(N)=O)C2CC2)C)CCC)=O)ccc(N)cn1 8796,C1(c2cn(CCCSC)nn2)(NC(c2cn(CCC)nc2)=O)CCCOC1 8797,N1(CCC)CCN(C(=O)NCC2(C)CCCC2O)CC1 8798,c1(C(=O)NC(C2OCCN(C(C(C=C)CC)=O)C2)C)cc(N)cc(F)c1 8799,Cc1ncc(NC(C2CC(C)(NC(=O)CC3COCCO3)C2)=O)c(C)c1C 8800,c1(CC(=O)NC2C(C)CN(C(=O)C3=CCSC3)C2)cccc2cnccc12 8801,c1(CC(=O)NCCOCCOCCNC(=O)CC2(O)CCC2)ccc2c(c1)CCO2 8802,C1(CC(=O)NCC(Cn2cc(CN(C(C)=O)C)nn2)(F)F)CC2CCC1O2 8803,c1(C(=O)NC2C(NC(CNC(=O)NC)=O)C2)cccc2ccn(C)c12 8804,N1(C(c2c(C)cno2)=O)CCCCC(CNC(=O)Cc2cn(C)nc2C)C1 8805,c1(NCc2c(C(=O)Nc3c(C)cnc(Cl)c3)cccn2)ccc2ncccc2c1 8806,C(=O)(C(O)CCC(F)(F)F)NCC1CC(NC(CC(=O)NCC)=O)C1(C)C 8807,C1(C(=O)NC(CC)CNC(C2CCOC2=O)=O)CC2(C1)CC(C)(C)C2 8808,c1(N(C2N(C(C)=O)C3C(C2)C3)Cc2ccc(C(=O)O)s2)nc2cncnc2s1 8809,Cc1nc(C2CCN(CC3COC(c4ccccc4)C3)CC2)nc2c1CCCC2 8810,C1(C(=O)NC(c2n(CC#C)cnn2)C)CCCN(C(=O)CCNC(C)=O)C1 8811,Cc1onc(C2CC2)c1C(=O)NCC1CCN1C(C1CC(C)(CN(C)C)C1)=O 8812,C1(SCCN2C(=O)CN(C(=O)OC(C)(C)C)CC2(C)C)CCC2(CCCCC2)O1 8813,C1(C(=O)NC(C)C)CCCC(C(=O)Nc2cc(C3CCOCC3)nn2C)C1 8814,C(=O)(C1Cc2c(Cl)cccc21)NCCN(C)C(c1cnc(CCC(F)(F)F)s1)=O 8815,c1(C(N(CC(C)(C)NC(CCNC(C)=O)=O)C)=O)ccnc2[nH]ncc12 8816,c1(C(N(CCC)CCNC(C2CC2(F)Cl)=O)=O)nc(C)c(C)nc1C 8817,N1(C(C(C)(C)C2CCOCC2)=O)CCC(O)(CNC(=O)CCC2CCCOC2)C1 8818,CC(C)CC(CC(=O)NC(CN1CCCC1)CO)NC(=O)C(C)C(C)(C)C 8819,N1(C(CCSc2n(C)nnn2)=O)CCN(C(C2(C)COC2)=O)CC1CCO 8820,N1(C(C=C(C(=O)NCCOCCC)F)=O)CCC(C)C1CC 8821,c1(C(N(CCCC(=O)NC2CCSCC2)C)=O)ccc2[nH]nc(Cl)c2c1 8822,N1(C(C(COC)C)=O)CCC(CC(=O)NC2CCCN(CCO)C2)CC1 8823,c1(COC)cc(NC(C2CC(O)CN2Cc2cscc2Br)=O)cc(Br)c1 8824,c1(C(=O)NCC(CC)(C)NC(c2cnns2)=O)cnc(C)nc1 8825,C12(C(N)=O)CCCC1(C(=O)NCC1(O)CCN(C(=O)COc3ccccc3)C1)C2 8826,N1(Cc2cccc(C(=O)NCC(C)C#N)c2)C(=O)CN(C)C1=O 8827,c1(C(=O)NC(CC(=O)NCC(C=C)O)CC2CC2)cccc(C)c1F 8828,c1(C(N2CCC(NC(c3cnc(C)nc3)=O)C2C)=O)cc2c(Cl)cccc2[nH]1 8829,C1(C(N2CCC(NC(CC(C)n3cccc3)=O)CC2)=O)CC2CCC(C1)C2F 8830,C(C(=O)NOCCCCC)C1C(NC(CN(CCC#C)C)=O)CCC1 8831,C(C1CCN(C(c2nnn(C)c2N)=O)CC1)=CC(=O)NC(c1cnc[nH]1)C 8832,C(=O)(CC(C)CC(=O)SC)NCC#CC(=O)NCC(CC)NC(=O)OC(C)(C)C 8833,n1(CCC=C)c(N(C)Cc2cnccc2Cl)nnc1CC1(c2cccc(F)c2)CC1 8834,c1(C(=O)NCCN(C(c2cncc(OC)c2)=O)C)cc(O)nc2c1c(C)nn2C 8835,C(C(=O)N1OC2CCC1CC2)(N(C)C(c1c[nH]nc1[N+](=O)[O-])=O)C1CC1 8836,Cc1cccc(F)c1C(=O)NCCNC(=O)C(C)(C)N(S(C)(=O)=O)C.C12CC1N2 8837,C1(O)(C(C(=O)OCC)(F)F)CCN(CC(C)C(C)(F)F)CC1 8838,c1(N(C)C(=O)Nc2scc(C(=O)OC(C)(C)C)c2)ccc(C(F)(F)F)cc1 8839,C(=O)(C(F)CC(C)(C)NC(c1ncccc1O)=O)NCC(C=C)(C)C 8840,C1(C(N2CCN(C(CC)=O)CC2CC(F)F)=O)CCc2cnc(C)n2C1 8841,C(=O)(C1=Cc2ccccc2C1)NCC1(C)CN(C(c2cnc(O)s2)=O)CCO1 8842,C1(NC(C2C(OC(C)(C)C)C2)=O)C=CCC(C(=O)NC2CC2)C1.C12(CC1)C(=O)N2 8843,c1(C(=O)NC2CN(C(C=COCC)=O)CC(O)C2)[nH]c2c(c1C)CCC2 8844,C=CC(C)(C)CC(=O)N1CCN(C(c2[nH]ccc2C2CC2)=O)CC1CF 8845,c1(C(=O)NCCCN(C(COCC(=O)NC)=O)C2CC2)cscc1SC 8846,C1(CNC(CCc2ccc(C)s2)=O)COCCN1C(C1CCCC1)=O 8847,Cc1cc(C(=O)NCCN(C)C(c2cc(C(=O)C(C)C)c[nH]2)=O)nn1C(F)F 8848,c1(NC2C(F)CCN(C(c3ccc(OC)c(C)c3)=O)C2)ncc2sccc2n1 8849,C(=O)(C1=CC2CCC=CCCC12)N1CC2(C(CO)CN(C(C(C)=C(C)C)=O)C2)C1 8850,C(=O)(C(CC(C)C)NC(N)=O)NC(C(=O)NCC(C(=O)OC)(F)F)C1CC1 8851,c1(C(N2C(C(=O)NCC34CC(CCO3)C4)CC2)=O)coc2ccccc12 8852,n1(CC)ccc(C(=O)NCC2(F)CCN(C(=O)C(c3ccnn3C)O)C2)cc1=O 8853,Cc1cc(C(=O)N(C)CCN(C(=O)C(C)C(F)F)C)cc([N+](=O)[O-])c1Cl 8854,c1(C(N2C(C)CC(CNC(C=C(C)C)=O)C2)=O)ccc2c(c1)C(=O)NCC2 8855,C1(CN(C(CNC(CC)=O)=O)C)CCN(C(c2coc(C(C)C)n2)=O)C1 8856,C(=O)(C1CSc2ccccc21)NC1CCC(CNC(c2ncncc2F)=O)CC1 8857,c1(C2C(C(=O)NCCCN(C(c3cnc(C(C)O)s3)=O)C)C2)ccc(F)cc1F 8858,n1(CC(=O)NCCC2(NC(C3N(CC)CC3)=O)CC2)ccc(C(F)(F)F)n1 8859,Nc1cccn(CC(N2CCCCC(CNC(=O)CC3CCCOC3)C2)=O)c1=O 8860,N1(C(C2CC(CCC)C2)=O)CCN(C(c2n[nH]c(CC)n2)=O)CC1C 8861,C1(C(=O)NC(CNC(CCOCC#C)=O)C)CNC(=O)CC1C 8862,n1(CC)nnc(C(N2CCC2CNC(=O)CNc2nccs2)=O)c1C 8863,c1(NC(COCC)Cc2ccc(Oc3cccc(F)c3)cc2)c(C)cccc1C#N 8864,C(=O)(C(CC)C(C)O)N(CCNC(c1cccc(C(=O)NCCC)c1)=O)C 8865,CC1CN(C(=O)CC2CC3(CCC3)C2)CC(C)N(C(c2cc3scnc3[nH]2)=O)C1 8866,C1(O)(C(=O)NC(C2CC(NC(C(c3ccccc3F)C)=O)C2)C)CCCCC1 8867,CN1CCN(C(C2C=CC=CC=C2)=O)CC1C(N1CCC2CC12)=O 8868,C(=O)(CCCCC(C)C)N1C(CNC(c2c(C)cco2)=O)CCC1 8869,C1(NC(CCC(CC)OC)=O)(CNC(C2CCCN2N=O)=O)CCC(F)(F)CC1 8870,c1(C(N2CCN(C(c3[nH]cc(C#N)c3)=O)CC2CCO)=O)nccc2nn[nH]c12 8871,c1(C(=O)NC2C(CNC(c3c(C)nns3)=O)CCC2)ccc(F)c(F)c1N 8872,C1(NC(C=CCCC)=O)CCCN(C(C2CC3(CSC3)C2)=O)C1 8873,c1(NC(C2CC(C)CN2Cc2ccc3ccsc3c2)=O)nc(Cl)cc(Cl)c1[N+](=O)[O-] 8874,C1(CNC(C(CC=C)CC)=O)CN(C(=O)CCC(=O)OCC)C2COCC2O1 8875,C1(NC2CC(OCC)C2SC)CCCCCC1C 8876,c1(-c2scc(CN3CCN(CCCCC)CC3)n2)ccc(F)c(OC)c1 8877,c1(C(N2CC(NC(C(C)n3ccnc3)=O)C(F)C2)=O)ccc2sccc2c1O 8878,C1(CC)C(NC(C2CC3=NOC(C)C3N2)=O)CCCN1C(C1CC1C(=O)NC)=O 8879,C1(CNC(C(C)NC(=O)NC)=O)N(C(=O)CCCC(C)(F)F)CCCC1(C)C 8880,C1(N(CCNCC(=O)NC2(COC)CC2)C)CCCC1 8881,C1(C(=O)NC(C)C2CC2)CCN(C(=O)C2=NOCC2)C(C)(C)C1 8882,c1(C(N2CC(OC)(CNC(=O)CC3CCOC3C)C2)=O)c[nH]nc1[N+](=O)[O-] 8883,c1(C(C)OC)nc(C2CC(F)(CO)C2)n(-c2cncc(Br)c2)n1 8884,N1(C(C(C)=C(CC)C)=O)CC(C(=O)NCCC2(C)CC2(F)F)C(C(C)C)C1 8885,C1(OC)CCCC12CCCN(C(C1CCC(n3ccnn3)CC1)=O)C2 8886,C(C(C)(C)C#CC(=O)NCCSC(C)C)NC(Cc1ccc(OC)cc1)=O 8887,O=C1OC(C(=O)NCC2CCN2C(=O)Cc2cn[nH]c2)Cc2ccc(Cl)cc21 8888,Cc1ccc(C)c(CC(=O)N(C(CNC(c2cncc(C)c2C)=O)C2CC2)C)c1 8889,c1(CCCC)c(CSC2CCOC2)oc2ccccc12.C12CCCCC1OC2=O 8890,N1(C(CSCC(N)=O)=O)CC(S(=O)(=O)N2CCN(C(C3CCCSS3)=O)CC2)C1 8891,C1(C(N(CCC(=O)NCCCc2ccsc2)CC)=O)CCCC(=O)N1 8892,S(=O)(=O)(c1ccc([N+](=O)[O-])c(Br)c1)N1CCN(C(C2(C)CCC2)=O)CC1 8893,C(C(C(C)(C)C)NC(c1c[nH]nc1C1CCCCC1)=O)NC(CC1(C)CC1)=O 8894,c1(CCC(=O)NCCCN(C)C(C2CC2(Br)Br)=O)cncnc1 8895,c1(CC(=O)NCC2CNCCOC2)ccc(Br)c(O)c1 8896,N1(C(CCOCCOC)=O)CCC(CNC(=O)C(COC)CC)C(C)(C)C1 8897,C(=O)(C(CO)C(C)(C)C)N(CC(C(N1C2(CC(COC)C2)CC1)=O)C)C 8898,N1(C(CN(CC)CC)=O)CCC(CC)C1CNC(=O)COCCN(C)C 8899,CCCC(C(=O)NCCn1cc(C(N2CCC(N3CCC3)CC2)=O)cn1)OC 8900,N1(C(c2c(OCC)cccc2)=O)CCC2(CCCCN(C(C3CCCO3)=O)C2)C1 8901,N1(C(c2cc(CC)nc(O)c2)=O)CC2CN(C(=O)CN(C)S(N)(=O)=O)CC2C1 8902,C1(CC(=O)N(C)CCNC(=O)CC2(C)CCC2)COCC1(C)C 8903,C1(CC(=O)NCCCOC=C)CCN(C(=O)Cc2ccc3c(c2)CC3)C1(C)C 8904,Cc1nnc2c(C(N3CCC(CNC(C4CCC4)=O)C34CCC4)=O)cccn12 8905,CC(C)(CCC(=O)NCC1CCN(C(c2sccc2Cl)=O)C1)[N+](=O)[O-] 8906,C=CCCCC(=O)NCC(CC(=O)NCC(C1CCCCC1)O)C1CCC1 8907,C1(O)(CCNC(CCc2ccn(C)n2)=O)CCCN(C(C23CCC2C3)=O)C1 8908,C(c1c(F)ccc(Cl)c1F)=CC(N1CC2C(NC(CC(C)C(F)F)=O)(C2)C1)=O 8909,c1(C(N(C(CNC(C=C(C)c2ccccc2)=O)C)C)=O)cc(S(N)(=O)=O)c(C)o1 8910,N1(C(CCCC(CC)CC)=O)CCOC2(CCN(C(=O)C)CC2)C1.S(C(F)F)CC 8911,C(=O)(C(O)CC(F)(F)F)N1CCC(O)(CNC(c2c(C)nccn2)=O)CC1 8912,Cc1cncc(C(N2CC(NC(C3CNC(=O)O3)=O)C(C)C2)=O)c1 8913,N1(C(C(CCC)C)=O)CCN(C(c2n[nH]c(C)c2F)=O)C(CC(C)(C)C)C1 8914,C(=O)(C1CCCn2ncnc21)NC(C)CC1CN(CC2CC3CCCCN3C2)C1 8915,N1(C(C2CC(C)=C(C)CC2)=O)CCC(C)N(C(=O)C(c2cnn(C)c2)C)CC1 8916,C1(CC(=O)N(CC(C)NC(c2c(C)ncnc2C)=O)CC)CCC(F)(F)CO1 8917,C1(C(=O)NCC2C(CCC)C2)CCN(C(=O)Cc2ncn(C)c2C)CC1 8918,c1(C(N2CCC(CN(C)C(C3(F)CC=CCC3)=O)C2)=O)cnccc1Cl 8919,C1(O)(CC(=O)NCC2CC(C(=O)NCC(=C)CC)C2)CCCOC1 8920,C1(F)(CNC(C2CCC(CC)O2)=O)CCN(C(c2sc(C)cc2OC)=O)C1 8921,C(C1CCOCC1)=CC(=O)N(C(C)C(=O)Nc1cnn(CC)c1C)CC 8922,C1(C)(C(=O)NCC2CN(C(c3c(CC)onc3)=O)CC2O)CCCCC1(F)F 8923,C1(CC(N2CC(C)(NC(C(C)OCCOC)=O)C2)=O)COc2ccccc2O1 8924,CC(C)(C)C(C)(C)C(=O)N1CCC(CCNC2CCCCC2F)CC1 8925,CC(C)CC(CNC(=O)CC1CCC(C(F)(F)F)O1)NC(C1(C)CCOCC1)=O 8926,c1(C(CNC(=O)NCc2cc(C)no2)(C)O)cccc(S(N)(=O)=O)c1 8927,N1(C(C2C(OC)CC2)=O)CC2CCC1CN2C(C1(CO)CC(C)(C)C1)=O 8928,c1(C(=O)NC2COCC2NC(C2CCCOC2)=O)ccnnc1S 8929,N1(C(c2nc(CC)sc2)=O)CC2CCC1C(CNC(=O)C(CO)N(C)C)C2 8930,C1(O)(CNC(=O)CC2CCOC2)CCN(C(c2coc(CO)c2)=O)CC1 8931,C1(C(=O)NC(C(NOCCCCC)=O)c2cccnc2)C2CCC(C2)C1C 8932,c1(CC(=O)N(CC(O)CNC(c2ccc(C#N)[nH]2)=O)C)ccc([N+](=O)[O-])cc1F 8933,C1(CC(=O)NCCCCCN(CC)CC)CN(C(=O)C(C)OC)CC1C 8934,N1(C(C2CC(=O)CC2C(F)(F)F)=O)CCn2cccc2C1CC 8935,N1(C(C(n2cc(Cl)cn2)C)=O)CCC(CCNC(C2CN(C3COC3)C2)=O)C1 8936,c1(C(=O)NCCC2N(C(Cc3cnc(C)s3)=O)CCC2)ccccc1F 8937,C1(NC(CN2CCN(C(CC(=O)NCC)=O)CC2)=O)CCC(C2CC2)CC1 8938,N1(C(c2c(CC)cco2)=O)CCCC(C(=O)NC(c2ccc(F)cc2)CO)C1 8939,c1(C(=O)Nc2c(CC)nn(C)c2)coc2c1CN(C(=O)CC1CCCC3CC13)C2 8940,c1(C(=O)NC2CC3(CN(C(C4(C)CCCC4O)=O)C3)C2)cc(Cl)cc2c1CCC2 8941,c1(N(CCC(=O)N(CCCC(=O)OC)C(C)(C)C)C(C)(C)C)c(Cl)cnn1C 8942,CCC(CC(F)F)C(=O)N1CCC(NC(c2cc3ccccc3s2)=O)C1C 8943,c1(C(=O)NCc2csc(CNC(c3ccnn3CCF)=O)n2)cnncc1O 8944,N1(C(C2(C#N)C(C)C2)=O)CCC2(CC1)CN(C(=O)CCNC(=O)C=CCl)C2 8945,C(CC)(C(C)(C)O)NC(CCCN(C(CC=C)=O)C)=O 8946,C(CC(O)C(F)(F)F)NC(C(CCN(C)C)NC(C=CCOC)=O)=O 8947,c1(C(=O)NCC(C)C(=O)O)ccc(S(=O)(=O)NCCC2CCCCN2C)cc1 8948,C1(C(=O)NCC2(NC(C(C)C3CCOC3)=O)CC2)CC(=O)c2ccccc2O1 8949,C1(NC(C(CC2CCOCC2)NC(C(C)N=[N+]=[N-])=O)=O)CC12CCOCC2 8950,c1(CNC(C2CC23CN(Cc2ccnc(Cl)c2)C3)=O)cc(Br)ccc1O 8951,C1(C(N2CC(NC(C3N(CCC)CCC3)=O)C(SC)C2)=O)CC=C(C(C)C)CC1 8952,CCC(C)(COC)C(=O)NC1CC2CCC1(NC(=O)CCCc1cccnc1)C2 8953,c1(C(=O)NCCCN(C(=O)CN(C)C(N)=O)CCC)c(C)c(C)cc(C)c1C 8954,N1(C(CSCC#C)=O)CCC(CC(=O)NCC2CCCCO2)C1 8955,C1(CN)(CO)CCN(C(=O)COCc2ccco2)C1 8956,N1(C(C2N(C(CNC(=O)OCC)=O)CCC2)=O)CC2CCCC2(C(N)=O)C1 8957,N1(C(C2C(OCC)CC2)=O)CC2CCC(C1)N2C(=O)CCc1ccon1 8958,Cc1cc(=O)ccn1CC(N1CCC(NC(=O)Cn2nnc(=N)[nH]2)C(C)C1)=O 8959,C(C)(CCCCCO)NC(C(CSC)(C)NC(C1CC=CCO1)=O)=O 8960,C12(C(=O)NC3C(NC(C=C(C)c4cccs4)=O)COC3)CCN(CC1)S(=O)(=O)C2 8961,N1(C(C(c2cncc(OC)c2)(F)F)=O)CC2CC(NC(c3cnn[nH]3)=O)CC1C2 8962,C(=O)(CCCC(F)(F)F)NCC(C(C(C)C)C)NC(c1ccc(N)c(F)c1F)=O 8963,CCC(C)C(C(=O)NC1CCOCC1C)N(C(=O)CCC1CC(OC)C1)C 8964,Cc1[nH]nc2ncc(C(=O)NCC3(F)CCN(C(C4CC(N(C)C)C4)=O)C3)cc12 8965,N1(C(C(CC)(CC)OC)=O)CCC2C(C1)CN2C(=O)C(C#N)C(C)(C)C 8966,CC1(C)CC(CNC(C2CCN(C3CC3)CC2)=O)CN1C(=O)CCS(C)(=O)=O 8967,c1(C(=O)NC(C(C)C)CNC(c2ccc(Cl)nc2O)=O)cccc(S(N)(=O)=O)c1 8968,C1(NC(c2ncn(CC)n2)=O)COCCC1C(=O)N(CCO)CCO 8969,c1(C(N(CC)CC2CCN(C(=O)CCC3CC3C)CC2)=O)ccc([N+](=O)[O-])cn1 8970,c1(C(=O)NC2CN(C(C(C)=C(CC)C)=O)C3C2C3)cc(Cl)cc(Cl)c1OC 8971,CCC(C)C(C(=O)NCc1nnc(O)o1)N(C)C(c1nc(O)sc1C)=O 8972,CC(F)(F)CC(=O)NCc1n[nH]cc1C(=O)NCCCCCCC1CC1 8973,C1(C(N2CCCC2)=O)CC(O)CCN1Cc1cnccc1Cl.CC12CCN(C1)C2 8974,CC(CO)(CO)C(=O)N(c1ncncc1-c1ccccc1)Cc1ncc(Br)cc1F 8975,c1(CS(Cc2ccc(-c3ccc(CC(C)C)cc3)cc2)=O)cccc(F)c1Br 8976,C(=O)(C(C)CC(=O)N(CCC(N1CC(N=[N+]=[N-])C1)=O)C)OC 8977,C1(CC(=O)NC2C(CC)N(C(c3cc4n(n3)CCC4)=O)CC2)CCS(=O)(=O)CC1 8978,C1(NC(=O)NC(CC(=C)Cl)CO)CCOC2(CCCC2)C1 8979,c1(C(N2CCC(NC(c3cnc(O)c(F)c3)=O)C2)=O)ccc(C(F)F)cc1F 8980,c1(CCC(=O)NCC(COC)(C)CO)ccc(F)cc1C(=O)OC(C)(C)C 8981,CC1(C(=O)NC2CN(C(=O)C(F)(F)C3CC3)CC2CC2CC2)CCCS1(=O)=O 8982,C1(NC(C(Cn2ccc(C)n2)C)=O)CN(C(C23CC(CO2)C3)=O)CC1(C)C 8983,C1(COC)CN(C(c2[nH]c(C)nc2C)=O)CCN1C(c1cc(COC)cn1C)=O 8984,C=CC(C)(CC)C(=O)NCCOC(C)(C)CNC(c1cc(O)cc(F)c1)=O 8985,C(=O)(C(C)C(O)CC(C)C)NC1(C)CN(C(C2(C#C)CCCCC2)=O)C1 8986,c1(CC)ccc(OC)cc1C(=O)NCC1C(CC)CCN1C(c1n[nH]cc1C)=O 8987,C(=O)(CC1OCc2ncccc21)NC(C)CNC(C1C2(CC2)C12CC2)=O 8988,C1(CC=C)(NC(C2CC2Br)=O)CCCN(C(c2ccc(Cl)cc2)=O)C1 8989,Cc1ccc(S(=O)(=O)NC2CCS(=O)(=O)C2)cc1Cl.N12CCCC1CC2=O 8990,C1(C)(NC=O)CCN(C(=O)CC(C)(C)C2CC2)C1.C1(N(C)CC)CC1CC 8991,c1(CC(N2CCCC2=O)C)nc(-c2cc(Cl)ccn2)nn1CC(N)=O 8992,C1(NC(CCNC(=O)OC)=O)COC2(CNC3CCCC3)CC1C2 8993,Cn1nccc1C=CC(=O)NCC1CCC(C(N2CC(O)C(O)C2)=O)CC1 8994,C1(CC=C)(NC(=O)CC2CC2C(F)(F)F)CCOC1.C12CC(C1)C(=O)NC2 8995,CC(=O)CCCC(C)C(=O)N1CC(NC(=O)CCC(CF)CF)C(O)C1 8996,C1(NC(Cc2occ(C)c2)=O)CCN(C(C)(C)C)C2(CC2)C1 8997,C1(CC)CN(C(=O)COCC(=O)N(C)C)CCN1C(=O)CCC1CCCCN1C 8998,CCC(CC(=O)NC(CNC(c1nc(C)sc1Br)=O)CCOC)C1CC1 8999,C(=O)(CCS(=O)(=O)C1CCCC1)NCC(CC)NC(C1CC(OC)C(OC)C1)=O 9000,C1(CNC(c2n(CC)cc(Br)c2)=O)CCN(C(c2ncn(C)n2)=O)C12CC2 9001,Cc1nc2ncccc2cc1C(=O)NCCCCN(C)C(c1nsnc1O)=O 9002,c1(C(N2CC(=C(C(=O)OCC)F)C2)=O)ccc2[nH]c(C(F)(F)F)cc2c1 9003,Cc1coc(C(=O)NCC2CC(NC(=O)Cc3csnn3)C2)c1 9004,C=C(C)C(O)CC(=O)N1CC=C(CNC(=O)C(CO)NC(N)=O)CC1 9005,c1(NS(CC2OCCN(C)C2)(=O)=O)c(Cl)nn2ccccc12 9006,C1(NC(c2ccc(OC)s2)=O)CC2CCCC(C1)N2C(C1(C)COC1)=O 9007,c1(C(N2CC(C)C(NC(c3cccc(Cl)c3)=O)C2)=O)ccc2c(c1)CCCCS2 9008,C#CCCC(C(=O)N1CCC(C)(CCO)C1)NC(c1cnc(S)nc1)=O 9009,C1(C(N2C(CNC(c3c(C)cccc3Cl)=O)CCC2)=O)CC2CCCN2C(=O)N1 9010,N1(C(CCNC(CC(C)C)=O)=O)CCC2CCC(NC(=O)CC(C)C3CC3)C12 9011,c1(C(=O)NCC(CCNC(C(C)NC(CC)(C)C)=O)O)ccnc2[nH]c(O)nc12 9012,C1(CC(=O)NCCC2CN(C(CC(C)c3cnn(C)c3)=O)C2)NC(=O)CNC1=O 9013,C(C)(CN=C(NC1CCCCC1)N1CCC(NC(N)=O)CC1)C1C(C)CCCC1 9014,c1(C(N2CC(CNC(CCN(C(C)=O)C)=O)C2)=O)cnc2cc(Br)ccn12 9015,c1(C(N2CC(CNC(c3ccc(C(C)=O)[nH]3)=O)C2)=O)oc(S(N)(=O)=O)cc1C 9016,C1(C(=O)NC2C(C)(C)C(=O)NC2)CCN(C(=O)C(F)(F)c2ccno2)O1 9017,Cc1nc2cc(C(F)(F)F)cnc2[nH]c1=NCCCn1cccc1 9018,c1(C(=O)NC2CN(C(CC#C)=O)CC2F)cc(C(F)(F)F)cc(Br)c1 9019,c1(C(N(C(CNC(C2CC(O)(CC#C)C2)=O)C)CC)=O)nc(C)ccc1F 9020,C1(C(=O)NC(C(=O)NC(CN(C(C)C)C)C)Cn2cncn2)CCCSC1C 9021,c1(CC(=O)NCC2(F)CN(C(CSC(C)C)=O)C2)ccc(OC(C)C#N)cc1 9022,C(CC(CNC(=O)C=CCOCCOC)OC)NC(CC=CCC)=O 9023,C1(NC(c2cc(C(=O)OC)nn2C)=O)CN(C(c2ncncc2F)=O)CC12CC2 9024,N1(C(C2(C)CCOC2)=O)CC(NC(=O)C(=O)NCC(F)F)C(F)C1 9025,c1(C(N2CCC(C3N(C(COC)=O)CC3(C)C)CC2)=O)cc(F)cnc1O 9026,c1(COCC)nc(C)c(C(=O)NCC(C2CC2)N(C(=O)CCCC2(C)N=N2)C)s1 9027,Cc1ccc(NC(=O)C(F)CC2CN(C(=O)Cn3[nH]cnc3=N)C2)cn1 9028,C12(C(=O)NCC(C#C)OC)CC(CN(C(=O)C(C)NC3CC3)C1)C2 9029,C(CCC(=O)N1CCC(N(C(=O)CCC=C)CCO)C1)=CCC=C 9030,N(C(=NCC)N1CCN(C(C)=O)C(C)(C)C1)C(C#C)(CC)CC 9031,C1(F)(CNC(CNS(CC)(=O)=O)=O)CCCN(C(C2CC3CC3C2)=O)C1 9032,C(=O)(C(F)C(F)(F)F)N(CC(=O)N(C(C)CCO)C)CCOC 9033,c1(C(=O)NC(CC(C)NC(C2CCCC(C(N)=O)C2)=O)C)cc(N)ccn1 9034,Cc1cccc2[nH]cc(C(=O)NC3CCCC(NC(C4CC(F)C4)=O)CC3)c12 9035,c1(CC)ccc(S(=O)(=O)NCc2nnnn2-c2cc(Cl)c(Cl)cc2OC)o1 9036,Cc1nc2cc(C(N3CC4CC(NC(c5cccc(Cl)c5F)=O)C4C3)=O)[nH]c2s1 9037,S(=O)(=O)(c1ccc(C(=O)NC2CCN(C(C34COC(C3)C4)=O)C2)cc1)NC 9038,C(c1c(C)nn(C)c1Cl)=CC(N1CCCC(NC(CC)=O)(CO)C1)=O 9039,C(N=c1[nH]c(=NCC2(CF)CCC2)c2ccccc2[nH]1)C1CC(=O)N(C2CC2)C1 9040,c1(C(=O)NC(C2CN(C(Cc3c(SC)cccc3)=O)C2)C)cc2cccnn2n1 9041,C1(O)(CC(=O)N(C)C)CCN(C(=O)C(N2CCN(C3CCNCC3)CC2)=O)CC1 9042,c1(C(N(C(CCNC(Cc2c(C)ccc(C)c2)=O)C)C)=O)ncc(Cl)c(N)c1Cl 9043,c1(C(N2CC(CCNC(=O)C(Cl)=CCl)(OC)C2)=O)cccc(=O)o1 9044,c1(C(N(C2CCN(C(=O)CO)CC2)CC#C)=O)ccc(CO)cc1OC 9045,N1(C(C(C)=CC2CC2)=O)CC2CC(NC(C3C4CNC(=O)C34)=O)CC1C2 9046,C1(C(=O)NCC2(O)CC(NC(CCCc3n(C)cnn3)=O)C2)C2CCN1CC2 9047,C1(NC(CC2CCC(C)(O)CC2)=O)CN(C(=O)C(C)(Cl)Cl)CCC12CCC2 9048,c1(C(C)C)ccc(O)c(C(=O)N(C2CN(C(C3CC4C(C3)C4(F)F)=O)C2)C)c1 9049,Cc1cc(NC(=O)CN2C(=O)CNC2=O)ccc1NC(=O)C(C)C1CCC1 9050,CC1CN(C(=O)CC2CCCN(C)C2)CCCN1C(=O)CC(C)(C)CN(C)C 9051,C1(CC)CCN(C(=O)C=Cc2cnn(C)c2)C1C(=O)NCc1sccc1C 9052,C1(CNC(C2CCN(CC(F)(F)F)C2)=O)CC2CC2N1C(=O)CCc1ccccc1 9053,c1(N2CC(c3ccccc3)(CO)OCC2)nc(=NCc2ccoc2)[nH]c2cc[nH]c12 9054,c1(C(=O)NC2C(CNC(=O)C=Cc3ccncc3)CCC2)ncc(Cl)cc1Cl 9055,C#Cc1ccc(F)c(CN(c2ccncc2)C(C2CCCCC2(C)C)=O)c1 9056,n1(CC(N2CCOCC(CNC(C3C4COCC34)=O)C2)=O)cc2ccccc2n1 9057,C(C(CC(=O)N1CCC(O)(CCNC(c2coc(O)n2)=O)C1)C(F)F)N(C)C 9058,C1(CNC(C(C)OCCOCC)=O)CCCC1NC(=O)Cn1cc(CO)nn1 9059,c1(C(N2C(CNC(CCNC(COC)=O)=O)CCCC2)=O)ccnc2[nH]nnc12 9060,C1(C(=O)NC(C2OCCN(C(c3c(C)cno3)=O)C2)C)CC2C=CC1CC2 9061,C1(NC(c2c(CC)scc2)=O)C2CC3CN(C(c4c[nH]c(Br)c4)=O)C1C3C2 9062,N12CCC(CC1)CCC2=O.N1(C(c2nnc(C(C)(C)C)o2)=O)CCCCCC1 9063,CN1C(=O)CCCC1C(N1CC(C2CC2C(N2CC(NC(=O)C3CC3)C2)=O)C1)=O 9064,C1(OC)CC2(C1)CC(C(=O)NCC(C)(CC(C)C)NC(c1nc(C)oc1C)=O)C2 9065,n1(CC)nnnc1C(c1cccn1C)NC(COC)C1CC1 9066,CC1(CNC(=O)CCCCC2CC2)CN(C(C2NC(=O)OC2C)=O)CCO1 9067,c1(OC)c(C(=O)NCC2CCN(C(C3C(C)C3C)=O)C23CC3)[nH]c2ccccc12 9068,N1(C(C(C)N(C(c2cccc(C)n2)=O)C2CC2)=O)Cc2cnn(C)c2C1 9069,C(C(C(=O)N(CC(C)(C)C)C)NC(=O)C=NOC)OCC 9070,C(=O)(CC(C)C(C)C(C)C)N(CC(C)(C)NC(Cn1nc(C)oc1=O)=O)C 9071,N1(C(C2CN(C)C2)=O)CCC(NC(c2cnc(C(F)F)nc2)=O)C(F)C1 9072,c1(C(=O)NCC2(CNC(C(C)=C3CCC3)=O)CC2)nc2cccnc2s1 9073,C1(NC(C(C2CCC2)OCC)=O)CN(C(C2CC(O)CN2C)=O)CC1SC 9074,c1(OCCC)ccc(CCCC(=O)NC2(COC)CCCCC2)cc1 9075,c1(CNC(c2ccnc(Cl)c2F)c2n(CCSC)nnn2)c(C)oc(C)c1C 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9094,Cc1cc[nH]c(=NCCCC(C)NC(=O)CCCc2ccc(C)s2)n1 9095,N1(C(COC2CN(C(C)=O)C2)=O)CCC(CCCNC(c2cnc(Cl)s2)=O)CC1 9096,c1(C(=O)NCc2nnc(C)o2)ccc(CNC(=O)CCc2nccs2)cc1 9097,Cc1scc(C(=O)NC2CCOCC2C(=O)N(C2CCOCC2O)C(C)C)c1C 9098,C(=O)(C(CC(C)C)NC(C)=O)NCCNC(c1ccc(CC)o1)=O 9099,c1(CNC(C2N(Cc3nc(C)sc3C)CC2)=O)cc(Cl)ccc1C 9100,CC(C)(CC(F)F)C(=O)N1CCCC(O)(CNC(C2(C)CC2(F)F)=O)CC1 9101,O=C1CCN(Cc2ccc(Cl)cc2)C(=O)C(CCc2nn[nH]n2)N1 9102,C1(NC(C(CC)(CC)CC)=O)C2CC3CN(C(C4CC5CC4CO5)=O)C1C3C2 9103,C(CC(C(=O)N1CC(O)(C(C)C)C1)NC(=O)C(CN(C)C)CC)OCC 9104,c1(N(CC)CC)ccc(NC(=O)NC(C)C(C)=C(C)C)c(F)c1F 9105,C(=O)(CC(C)C(C)(C)NC(c1ccnn1C)=O)NC(C)CCC1CCCO1 9106,n1(CC(=O)NCC(CN(C)C(c2ccon2)=O)O)nnc2ccccc2c1=O 9107,C1(NCCOCC#C)CCN(C(=O)CN(C)CCc2ccccn2)CC1 9108,C1(C(=O)NCc2occ(C(=O)NC3CCN(C)C3)c2)CCC2(CC2)C1 9109,c1(CNC(=O)NC(CO)CCO)csc(O)n1.C1C(=O)N1 9110,Cc1c(C(=O)NCCCN(CCO)C(C2COCCN2C)=O)c[nH]c1C#N 9111,C(=O)(CC(O)CC(C)C)N1C(C(N2CCC(C(C)OC)C2)=O)CC(OC)C1 9112,C1(CCNC(c2ccc(OCC)cc2)=O)C(C)CCCN1C(c1cnns1)=O 9113,C1(C#N)(C(N2CC(C)C(NC(C3(CF)CCC3)=O)C2)=O)CC2C=CC1C2 9114,C1(CC(=O)NCC(C)NC(=O)C(C)C2CCC2)CC1(Cl)Cl 9115,C(=O)(CCCCN=[N+]=[N-])NC(C(=O)NCC(C#C)CC)COC(C)C 9116,CCCN=C(NCC(CC(F)(F)F)F)N1CCC(CC(=O)OC)C(c2ccccc2)C1 9117,c1(C(=O)NCC2CN(C(COC(C)=O)=O)C2)ccnc(N(C)C)c1 9118,N1(c2nc(C)nc(O)c2)CCC2(CCOC2)C(CNC(=O)COC(F)F)C1 9119,C1(C(=O)OCCN(C)C2CC2)(CNc2cncn2C)CCCO1 9120,C1(C(=O)NCCCN(C(C(C)c2cncs2)=O)C)Cc2nccnc2C1 9121,C1(C(=O)OC)CCN(C(=O)C(CCSC)NC(c2cnsc2)=O)C1C 9122,N(C(=NCCCCl)NCCNc1c(C)cc(C(F)(F)F)cc1)Cc1ccccc1 9123,C(N=c1[nH]c(=NCC(F)F)[nH]c2cccnc12)c1c(Cl)cccc1 9124,Cc1ccc(C(N2CCOC(CC(N3CCN(CCO)C(C)C3)=O)C2)=O)nc1C 9125,Cn1ccc2cnc(N3CCNCC3C(=O)Nc3nc(Cl)ccc3F)nc12 9126,CC1(C)CN(C(=O)C(F)(F)CO)CC1C(=O)NCCOC1CCCC1 9127,C1(N(C(C(C)NC(C)(C)C)=O)C)CCC(NC(=O)CN2CCC(C)(O)C2)CC1 9128,CCC(CNC(C1CCCCC1(C)NC(=O)CCn1cnc(=N)[nH]1)=O)CC(C)C 9129,CC1(C(=O)NCC2CCCCN(C(c3cncc(Cl)c3)=O)C2)CCCCNC1=O 9130,C1(S(C)(=O)=O)(CNC(=NCCc2nnc(C)s2)NCC2CCOC2)CCC1 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9149,CC(CNC(c1ccnn1C1CCC1)=O)(CO)NC(=O)CC1(c2ccccc2)CC1 9150,N1(C(CC(CC)C(C)C)=O)CCC2CCN(C(C3CCOC3C(C)C)=O)CC12 9151,c1(NC(C2C(NC(c3cnc(OC)c(C)c3)=O)CCC2)=O)nc(Cl)c(Cl)cc1Cl 9152,C=C(C)CC(C(=O)NCC=Cc1cccnc1)NC(C1CCOC(C)(C)C1)=O 9153,c1(NCC=C=C)ncccc1S(=O)(=O)N1CC2CC3CC2C1C3 9154,c1(C(=O)NCCC(C)NC(C2CC2C2CCC2)=O)ccnn(C)c1=O 9155,N1(C(CSC)=O)CC(O)CC(O)C1.N12CCC(C1)C2=O 9156,N1(C(C2C(=C)CC2)=O)CCN(C(c2ccnc(Cl)c2)=O)C(C)C1 9157,c1(C(=O)NC(CC(C)NC(Cc2c(C)cc(F)cc2)=O)C)cc2n(n1)CCCO2 9158,C1(CCNC(=O)Cc2cc[nH]n2)CC(F)(F)CN1C(c1cc(Cl)c(Cl)s1)=O 9159,C12(NC(c3c(C)occ3)=O)CCCC1N(C(c1ccc(C3CCC3)cc1)=O)CC2 9160,C(=O)(CN=c1cc[nH]cc1)NCC(c1ccccc1)NC(c1c(C)cnn1C)=O 9161,C12(CNC(C3CC34CCCC4)=O)CCC(CC1)CN2C(=O)COCC1CCCO1 9162,c1(C(C)=O)ccc(C(N2CCN(C(=O)CCCF)C(C)C2)=O)cc1C 9163,C#CCC(CC#C)C(=O)NCC(F)CNC(C1(O)CCCCC1)=O 9164,c1(N(C)C)ccccc1C(c1nnnn1C1CC1)NC1C2COCC12 9165,Cn1cnnc1CC(=O)N(C1CCN(C(=O)COc2cccnc2)C1)CC1CC1 9166,c1(C(N(CC(C)(C)NC(c2c(C)ccnn2)=O)C)=O)[nH]c2cc(F)ccc2c1C 9167,c1(C(=O)NCC2C(C(=O)NCc3c(OC)cccc3)CCC2)ccc(C)cc1O 9168,C1(C(N2CCCC2C(F)(F)F)=O)(NC(C2CC2F)=O)CCCCC1 9169,N1(C(C(C)Cc2ccnn2C)=O)CCC(O)(C(C)NC(c2coc(Cl)n2)=O)CC1 9170,c1(C(N2CC(SCCSCC)OCC2)=O)cnc(OC)c(Br)c1 9171,c1(C(=O)NC2C(CNC(C3(CC=C)CC=CC3)=O)CC2)nsc2ccc(C)cc12 9172,c1(C(N2CCC(N(C)CC3CCCC3(C)C)C2)=O)ncc(F)cn1 9173,Cc1cc(C(=O)NCC2CC(C)CN(C(C3(C)SCCCS3)=O)C2)c(O)nn1 9174,c1(C(=O)NCC2(NC(CC3N(C)CCCC3)=O)CCC2)cc[nH]c(=N)c1[N+](=O)[O-] 9175,N1(C(CC2(C)N(C(C(CC)SC)=O)CCC2)=O)CC2CC1CN2CC 9176,c1(C(=O)NC(CNC(c2nc(C)oc2C)=O)C)ccc(F)c2cccnc12 9177,c1(C(=O)NCCN(CCOC)C(c2scnc2C(C)(C)C)=O)cc(SC)nn1C 9178,c1(NCC(c2cc(F)ccc2F)OC)ccc(NS(C)(=O)=O)c(Cl)c1 9179,c1(C(=O)NCC(N(C)C(C2CC23CCOC3)=O)C2CC2)c(F)cc(N)cc1F 9180,N1(C(c2c(Cl)cc(C)s2)=O)CCC2(CCCC2NC(c2coc(C#N)c2)=O)C1 9181,c1(OC)cccc(C(=O)NC2CN(C(=O)C(C)n3ccnc3)CC2C)c1 9182,Cc1ccn(C)c(=O)c1NC(C12CCCC(CO1)C2)=O 9183,C(=O)(CCC(=O)NC1(CF)CCN(C(c2cnoc2CSC)=O)C1)NCCC 9184,C1(NC(C(COC)N(C)C)=O)CCCCCN(C(=O)CCN2CCCC2=O)C1 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9578,C1(OC)CC2CCC1CC2C(=O)NCC1(CNC(C2CCCOC2)=O)CCC1 9579,C(C(C(=O)NC1CC(NC(C2CC(=O)N(OC)C2)=O)C1)C(C)(C)C)OCC=C 9580,N1(C(CCN(C)CC)=O)CCOCC(NC(=O)CCCOc2ccccc2)C1 9581,C(=O)(CS(=O)(=O)C(C)C)N1CCC(NC(c2cccc(C(=O)NC)c2)=O)C12CC2 9582,n1(CC)cnc2c(NC(C)C(C)NC(=O)CN(C)CCO)nc(Cl)nc12 9583,c1(NC(C2CCN(Cc3c(C)nn(C)c3)CC2)=O)cn2c(F)cccc2n1 9584,C1(CN(C(C(CC)OCC)=O)C)CN(c2nccc(CC#N)n2)CCO1 9585,N1(C(C2(Cl)C(C)(C)C2)=O)CCN(C(=O)Cc2cnsc2)C(CO)C1 9586,Cc1cc(Cl)cc(C(N2CCC3(C2)CN(C(=O)CC2CCOC2=O)C3)=O)c1C 9587,C(=O)(N1CC(O)C(O)CO1)c1cn(CCCOC2CN(S(N)(=O)=O)C2)nn1 9588,C1(NC(c2ccc(CC)cc2)=O)CCCCN(C(=O)CCCC(C)C)C1.C(=O)CS 9589,c1(C(=O)NC2CC(C)(NC(c3ccc(Cl)[nH]3)=O)C2)ccc(N)c(Cl)n1 9590,Cc1ccn(CC(=O)NC(C)CNC(=O)C(C)Cn2cccn2)c(=O)c1 9591,C1(CN(C(C(=Cc2cnc[nH]2)C)=O)C)CCN(C(=O)Cc2sccc2C)CC1 9592,N1(C(=O)CC2(N3CCCC3)CC2)CC2CC1CN2C(C1(C(F)F)CCCO1)=O 9593,C1(CC(=O)N(CCCOC)CCO)CN(C(c2cnc(C)cn2)=O)CCC1C 9594,Cc1ccccc1CCC(N1CCC(CNC(c2cnnn2C)=O)C1)=O 9595,C=C(Cl)CC(C(=O)NC1CCN(C2CCOCC2)C1)NC(=O)CC(C)(O)C=C 9596,Cc1ccc(C(=O)OCCc2nnn(C(C)(C)C)n2)c2cccnc12 9597,C1(C(=O)NC2CN(C(c3cnc(-c4ccc(Cl)cc4)s3)=O)C2)(CC)CCOCC1 9598,c1(N2CCCN(Cc3cnc(C)[nH]3)CC2)nc(C)nc2ccccc12 9599,c1(NC2CC(C)N(C(=O)Nc3cncc(OCC(F)F)c3)C2)ncnc(Cl)c1F 9600,CC(C)(C)CC(C)(C)C(=O)N1CC2CC2(NC(=O)C(c2ccccc2F)O)C1 9601,c1(C(N2CC(NC(C=CC)=O)C(c3ccccc3)CC2)=O)cc(F)c(F)cc1Cl 9602,CC(C)CC(F)C(=O)N(C(C)CNC(=O)CCCN1CCCC1)C 9603,c1(CN(C(c2cccnc2)CC)C)cc(F)c(C(F)(F)F)cc1F 9604,c1(OCC)ncccc1NCc1cn(CCCC(=O)NC)nn1.C1C(=O)N1C 9605,Cc1cccc2c(C(N3CCCC3C(C)(C)NC(C3CC3C)=O)=O)cnn12 9606,Cc1ccc(CCNC(=O)CC2CC(C)N(C(=O)CNC(C3CC3C)=O)C2)cn1 9607,C(=O)(C(F)CCC(C)(C)C)N1C(CN(C)C(c2ccnc3ncnn23)=O)CCC1 9608,N1(C(C2ON=C(C(C)C)C2)=O)CC2(CCC(CNC(=O)CCCCF)O2)C1 9609,C1(O)(CCNC(=O)NCc2ccc(-c3cscn3)cc2)CCCOC1 9610,c1(NC)ccc(C(=O)NC(c2ccccc2)C(C)NC(=O)Cn2nccn2)cn1 9611,N1(C(C(CC#C)C2CC2)=O)CCC2(CCC(CNC(C3(CF)CCC3)=O)O2)CC1 9612,CCCC(C)(O)CC(=O)N1C2CCC1CN(C(=O)CN1C(=O)NC(CC)C1=O)C2 9613,C1(C)(NC(C23C(NC(C(CC)C)=O)C4CC2C3C4)=O)CCC(C)(C)CC1 9614,S(=O)(=O)(c1ccc(NCC2CN(C)C2)c(Cl)c1)NC(CC(C)C)CN(C)C 9615,N1(C(C(CCC=C)(C)C)=O)CCC2CN(C(c3cnc[nH]3)=O)CC2C1 9616,c1(NCC(CC)CO)ccc(S(=O)(=O)N2CCC(C3CCCCC3)C2)cc1Br 9617,C1(C(N(CC(N2CCOCC2)(C)C)C)=O)CCN(C(=O)C2CC3CCC(C2)O3)O1 9618,N1(C(c2cnn(C)c2N)=O)CCC(CO)(NC(=O)CCOCC2CCCC2)CC1 9619,N1(C(c2ccc(CSC)o2)=O)C2CCC1CC(NC(=O)C(O)C(F)(F)F)C2 9620,c1(C(N2C(CC(=O)N(CC(Cl)Cl)C)CCCC2)=O)cc(F)ccc1F 9621,c1(C(N2C3CN(C(c4n(CC)ncc4)=O)CC32)=O)ccc2cc(OC)c(F)cc2n1 9622,Cc1cc(C(=O)NCCOCCNC(c2cnn(C)c2Cl)=O)c2sc(=N)[nH]c2n1 9623,c1(OC)cccc(C(=O)NCC(C2CC2)NC(C2CN(C)CC(C)O2)=O)c1OC 9624,CC(C)C(O)C(C)C(=O)N1CCC(CNC(c2coc(CO)c2)=O)C(O)C1 9625,C1(CC)(NC(=O)C(C)CC2CC2)CCCN(C(c2ccc(C)c(C)n2)=O)C1 9626,c1(OC)cncc(C2CCN(C(C3(CC(F)F)CC3)=O)C2)c1 9627,N#Cc1cc(CNC(C2(F)CCCN(C(=O)CC3CCSC3)C2)=O)ccn1 9628,C1(C(=O)NC2C(CO)CCN(C(c3cc(C)sc3)=O)C2)CN(C)CCN(C)C1 9629,C(=O)(CCN=[N+]=[N-])N1CCC(C(N(C)CC2CCCS2)=O)C1 9630,CCC(C(=O)NC1CN(C(=O)CCCN(C)C)CC2(CC2)C1)C(C)(F)F 9631,C=CCCC(CC(C)C)C(=O)NCC(C(F)(F)F)n1cncn1 9632,C1(NC(C2(F)CCCOC2)c2n(CCSC)nnn2)CCCC2(C1)CC(O)C2 9633,C1(NC(c2cc(CC)[nH]n2)=O)CCC(C)N(C(c2cc(C(=O)OC)n[nH]2)=O)C1 9634,Cc1ncc(Cl)cc1C(N1CC(NC(C2CCCCC2(C)C)=O)C(O)C1)=O 9635,C=C1CCN(C(=O)CN2CCOC2=O)C(C(=O)NC2CCCNC2=O)C1 9636,N1(C(CCn2ncc(C)c2)=O)CCC(N(C(=O)C=Cc2cn(C)nn2)C)CC1 9637,C1(C(=O)NCC2(CN(C)C)CC2)COC2(C1)CN(C(=O)COCCOCCO)C2 9638,c1(C(N2CC(NC(c3ncncc3F)=O)C3C2C3)=O)cc2c(s1)CCCC2 9639,c1(CC)nnc2cc(N3CCN(C(c4ccn(CC)n4)=O)CC3C)ncn12 9640,C(=O)(C(CC(C)CC)NC(C1CCC(=O)O1)=O)N(CC(=O)NCC)C 9641,C1(C(N)=O)COC2(C1)CN(C(=O)CCC=O)C2.N1CC(C(F)(F)F)C1 9642,c1(N(CC(C)NC(C(COC)O)=O)C)cc2nncn2cn1 9643,CC(C)CC(O)C(=O)N1CC=CC1(C)C(=O)NC1(C)CSC1 9644,O=C(Nn1cnc2scc(-c3cccs3)c2c1=O)NCC1CC12CCOC2 9645,C1(C(N(C2CCCCC2)CCNC(C(CN(C)C)O)=O)=O)C2CCCCC12 9646,c1(C(N(C(C)CN(C(=O)COC2CCOC2)C)C)=O)[nH]cc2c1CCC2 9647,CN=c1[nH]cc(C(=O)OCc2cnccc2C(F)(F)F)s1 9648,c1(CCC(=O)NCC2(C(N)=O)CCCO2)nc2ncccn2n1 9649,c1(C(=O)NC2(C)CN(C(Cc3cc(C(C)C)no3)=O)C2)ccc2[nH]ccc2n1 9650,N1(C(c2cc(OCC)no2)=O)CC(C)CC1C(=O)NCC(C)CN(C)C 9651,CCC(CC)(CCNC(c1c[nH]c(=N)s1)=O)NC(=O)C(F)CC1CCCCC1 9652,Cc1cc(C(N2CCN(C(=O)C(N3CCC(N(C)C)C(C)C3)=O)CC2)=O)ccc1F 9653,c1(OC)c(C(N2CC(NC(=O)CCC=CC(C)C)C3(CC3)C2)=O)cc(F)cc1Br 9654,c1(C(=O)NC2CCCN(C(CCC=C=C)=O)C2)ccc(N)c([N+](=O)[O-])c1 9655,C(=O)(C(C)(F)C(F)(F)F)N1CC(CC(CNC(C(C(C)C)OCC)=O)(C)C)C1 9656,N1(C(C2CC(C)(C)C2)=O)CCC(C(N2C3CCC2CC(F)C3)=O)CC1(C)C 9657,Cc1ccc(C(N)=O)cc1C(=O)NC1CC(NC(=O)C(C)(C)CC#N)C1 9658,Cc1ccc(=O)n(CC(N2CCN(C(C3COCCOC3)=O)CC2C2CC2)=O)c1 9659,c1(C(N2CC(CNC(C3(C=C)CCC3)=O)OCCC2)=O)c(C)nc2ccccn12 9660,C(CN=c1cccc(S(=O)(=O)NCCC2SCCS2)[nH]1)c1cccc(OC)c1 9661,Cc1cc(C(=O)NCC2(C)CC(NC(=O)CCc3ccc(C)s3)C2)nc(C)n1 9662,c1(C(=O)NC(CCCCNC(c2cccc(C)c2)=O)C)cc(O)ncc1Br 9663,N1(C(C(CC#C)C)=O)CC2CCCC2(NC(=O)CSc2ccc(C)cc2)C1 9664,c1(C(=O)NC(C(=O)N(CCCCC)CCO)C2CC2)cc(C)nnc1C 9665,C1(C(N(C2CCN(C(CN(CC(C)(C)C)C)=O)C2)C)=O)CCC2(CCCC2)C1 9666,n1(COC)nc(C2OCCc3ccccc32)nc1-c1coc2c(F)cccc12 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9918,C#CCC(C)(CC)C(=O)N1CCC(O)(CNC(c2ccoc2Br)=O)C1 9919,Cc1ncn(C)c(=O)c1C(=O)NCC1(NC(=O)C(C)N2CC(C)C2)CCC1 9920,CN=c1[nH]cc(C(=O)NC2C=CC(C(=O)NCC(CO)OC)C2)o1 9921,C1(NC(c2cccn3ncnc23)=O)CC12CCN(C(c1ccccc1Cl)=O)CC2 9922,N1(CC)CCN(C(=O)C(CNC(=O)C(F)C(C)(F)F)N(C)C)CC1C 9923,CC1=C(C(=O)NC2COCCC2NC(=O)C=Cc2cnc[nH]2)CCC1 9924,C(=O)(CCCCCC(=O)N1CC(NC(=O)C(F)=C2CCC2)C(C2CC2)C1)OCC 9925,c1(C(N(CC(C)NC(=O)CCNC(=O)OC)CC)=O)c(C)ccc(Cl)c1F 9926,N1(C(c2cc(C)nn2CC(F)F)=O)CCC(F)C(NC(C2CCCC2)=O)C1 9927,Cc1c(C(N2CC(CNC(=O)C(C)CCO)CC2C)=O)[nH]c2c1C(=O)CCC2 9928,N1(C(C(C)C)=O)CCC2CCN(C(c3ccc(NC(C4CCC4)=O)cc3)=O)C2C1 9929,C1(CNC(c2ncc[nH]2)=O)CC(F)CN1C(=O)CCC1OCCO1 9930,N1(C(C=CCC)=O)CCN(C(c2cccn(C)c2=O)=O)C(C(C)(C)C)C1 9931,CCCCC(C(=O)NCCNC(=O)C=C1CC1)NC(=O)OC(C)(C)C 9932,C1(C(=O)NCCNC(C(COC)OC)=O)CC2CC1CO2 9933,c1(C(N2C(C)(CNC(=O)C(O)C3CC3)CCC2)=O)cccc(N=[N+]=[N-])c1 9934,Cc1[nH]nc(C(F)(F)F)c1C(=O)NCCOCCNC(=O)C=Cc1ccoc1 9935,C(=O)(CC(C)C(F)F)NC(CC)(C)CCNC(c1ccccc1SC)=O 9936,N1(C(CS(=O)(=O)NC)=O)CC2C3CCC(C2C1)N(C(c1ccc(C)nc1N)=O)C3 9937,S(=O)(=O)(c1ccc(Br)c(OC)c1)Nc1cc(-c2nc(SC)no2)cc(OC)c1Cl 9938,C1(NC(C2(C3CCOCC3)CC2)=O)CC2CN(C(C3CC(F)C3)=O)CC2C1 9939,CC1CCC2CN1C2=O.N1(C(=O)CCc2cnoc2)CC(CO)CC1CO 9940,N1(C(C(C)(C)NC(=O)C(F)(F)F)=O)CCC(NC(=O)CCc2cc[nH]n2)CC1 9941,N1(C(=O)C(O)C(F)F)CCC(C2CCN(C(=O)CCSc3ccccn3)CC2)C1 9942,C1(C(=O)NCC(CNC(c2ccc(C#C)cn2)=O)C)CCc2n[nH]cc2C1C 9943,c1(C(=O)NC2C(NC(C3CC(=O)NC3)=O)C2)csc2nnsc12 9944,C1(NC(C2C(=C)CC2)=O)CCC2CC1CN2C(c1c[nH]ccc1=O)=O 9945,C1(C(=O)NCc2c(CC)n[nH]c2)CCC(C)(C)N(C(C23CCC(C2)C3)=O)C1 9946,C1(CC)CN(C(=O)Cc2ccc(O)c(C)c2)CCC1NC(c1cc(Cl)c[nH]1)=O 9947,N12C3CCC1CN(CC3)C(=O)Nc1c(cccc1)N(CC)C(=O)C2.C(C)(C)OC 9948,C12(CNC(c3cocn3)=O)CCCC1N(C(=O)CN1CCCCC1)CCC2 9949,C=C1Cn2c(C(=O)NCC3(C)CCN(C(=O)C=Cc4c[nH]nc4C)C3)nnc2S1 9950,CCC(C)CC(C(=O)Nc1ccc(OC)cc1C)NC(=O)CC1(O)CCOCC1 9951,C(C)(C(C)(C)CO)NC(C1C(CNC(C2(CC)CCCC2)=O)CCC1)=O 9952,Cc1nn(CC(N2CCC(NC(=O)COCC3CCOC3)C2C)=O)cc1[N+](=O)[O-] 9953,C1(NC(c2cnsc2)=O)CC2CCC1N(C(=O)COc1ccc(F)nc1)C2 9954,c1(C(N(c2cnn(C)c2)C)=O)cccc(CNC(C2CCC3(CC3)C2)=O)n1 9955,C(=O)(C1=CCC(C)(C)CC1)NC1CC(CNC(c2c(C)[nH]nc2C(F)F)=O)C1 9956,N1(C(CCCOCCC)=O)CC(C)CCC1CNC(=O)CNS(=O)(=O)CC 9957,N1(C(C(C)C#N)=O)CC(F)(F)CC1CCNC(c1ccc(C(C)(C)C)cn1)=O 9958,C(CCCC(CO)NC(=O)CCc1cnn(C)c1)NC(C(C1CC1)OCC)=O 9959,N1(C(C2(F)CCN(C(CC(C)n3ccnc3)=O)C2)=O)CC2CCC1C(O)C2O 9960,C=CCN=C(NCC1CN(C)CCO1)N1CCCC(C(=O)N(C)C)C1 9961,Cc1cc(C)n(C(C)CC(=O)NCCC(C)NC(=O)CSCc2ccccc2)n1 9962,C(=O)(CC(=O)NCC1CCC1NC(C1(C2CCCCO2)CC1)=O)NCC 9963,N1(C(c2c(CC)cccc2)=O)CCCC(NC(c2cnc(S)nc2)=O)C1CC 9964,C(=O)(C1=CC2(CCOC2)C1)N.C(=O)(CCCn1cncn1)N(C(c1cnc[nH]1)C)CO 9965,c1(C(N2CC(NC(CCC=CC)=O)C3(C2)CC3)=O)ccc2sncc2c1 9966,CCC(CC(=O)NC(C)(C)C1CC1)NC(=O)C(C)OC1CCCCC1 9967,C(=O)(C1=CC2CCCCCC12)NCC1(CNC(c2ccc(C)o2)=O)CC1 9968,c1(C(=O)O)nccc2c1CCN(CC(c1cc3ccccc3o1)O)C2 9969,Cc1cc(C(=O)NCCC(C)NC(=O)C(C)C#N)n[nH]1 9970,N1(C(CN(C2CCSC2)C)=O)CC(F)(F)CC1(C)CNC(c1csc(Cl)n1)=O 9971,c1(SC(c2ccccc2Cl)C(=O)OCc2cc(C)ncc2)cc(Cl)cc(Br)c1 9972,c1(C(N2CC(CNC(C3(CF)CCC3)=O)C3(CC3)C2)=O)cnc2n1CCCC2 9973,C1(N(C(C(CC)(C)F)=O)C)CN(C(=O)CCCOc2cccc(C)c2)CC1(C)C 9974,CCC(C)(C)C(O)C(=O)N1CCC(NC(=O)Cc2scnc2C)C1 9975,N1(C(C(c2ccc(Cl)cc2)OC)=O)CCCC12CCN(C(C1CCOC1)=O)CC2 9976,c1(NC(C2CCC(CC(=O)NCc3ccsn3)C2)=O)ccc(Br)c(Cl)n1 9977,C(=O)(CC1CCCc2c1[nH]c1ccccc21)Nc1cc(F)cc(OC)c1OC 9978,c1(C(N2CC3(CC(CNC(C4(CC)CC4)=O)OC3)C2)=O)cnc2c(c1)CCCO2 9979,c1(CC(=O)OC2CN(CCOC(C)(C)C)C2)cccc(Br)c1 9980,CC(C(=O)N(C1CN(C(c2nn(CC(F)(F)F)cc2Cl)=O)CC1O)C)C(C)(F)F 9981,CCCC(CCC)C(=O)NC1CCC(C)N(C(C2(c3ccccc3Cl)CC2)=O)C1 9982,C1(NC(c2cc(C(=O)OCC)nn2C)=O)C(OCC)C2CCCCCC12 9983,N1(C(C2OCCC(C)(C)C2)=O)CCC2(C=C(C(=O)N3CC(C4CCOC4)C3)C2)C1 9984,C(CCCC(=O)N1CCC1CNC(C1(F)CCCOC1)=O)N(C)C 9985,c1(CC)c(N2CC(NC(C3CCN(C)CC3)=O)CCC2C)ncnc1Cl.C1(C)CC1 9986,c1(NC(CC2(C)N(c3cc(C(=O)OC)ncn3)CCC2)=O)ccnn2cccc12 9987,N1(C(COC2(C#C)COC2)=O)CC(C(N2CCCCCC2)=O)C(C2CC2)C1 9988,c1(N(C)Cc2ccncc2F)cccc(S(=O)(=O)NC2CSC2)n1 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10041,C(C(C)C(=O)NCC1(C(C)(C)O)CN(C(=O)CCSC2CCCC2)C1)OCC 10042,CCCCC(C)CCC(=O)NCCCN(C(=O)C(c1ccccc1)F)C(C)C 10043,C1(CNC(COCC=C)=O)CCC2CN(C(c3ccncc3CC)=O)CCC2C1 10044,C1(=CC(N2CC(NC(=O)C=C3CCC3)CC(C)C2)=O)CCOc2ccccc21 10045,c1(CC)ccc(C(C)C(=O)NCC(O)CNC(=O)CCc2cncs2)cc1 10046,c1(C(=O)NCC(CNC(c2cc(C(C)=O)oc2)=O)(C)C)cc(C)ccc1Br 10047,c1(C(=O)NC2CN(C(c3cc[nH]n3)=O)C3CC23)ccc2c[nH]nc2c1 10048,N1(C(C2CN(C(C3ON=C(CC)C3)=O)CC2C)=O)C2CCC1CC(F)C2 10049,C#CCCCC(C(=O)N)N1CCC(CCCSC)C1.n1(C)cc(C)cn1 10050,C(CC(F)(F)F)N(C)C(c1noc(C(C)(C)C)n1)=O.C(=O)CCOCCCNN 10051,c1(NC(C(C)C)=O)cccc2c1CCCN2C(C1OCCC1c1ccccc1)=O 10052,C1(NC(C)=O)CCC12CN(C(C1CCC(C(N)=O)CC1)=O)C2 10053,Cc1nc2ccc(C(=O)N(CCC(F)(F)F)C3CCOC3)cc2n(C)c1=O 10054,C1(C)(NC(C(c2ccc(Cl)s2)OC)=O)CCCN(C(c2coc(C(C)=O)c2)=O)C1 10055,c1(-n2cc(CCCC)nn2)cccc(C(=O)OC)c1.C1C(=O)N1CCOCCO 10056,C(=O)(C(C)(C)NC(=O)C(F)(F)F)N(C1CCCCC1)CC(C)NC(=O)CC(C)C 10057,N1(C(c2cc(C)[nH]c2)=O)CC(F)(F)CC1C(=O)NOCCF 10058,N1(C(c2nc(C(N)=O)sc2)=O)CC(CNC(C2CS(=O)C2)=O)N2CCC1C2 10059,CC1(C)CC(NC(c2ccc(C(C)(C)C)o2)=O)CC(O)C1 10060,c1(C(=O)NCC2CCC(CNC(C3CC34CCOC4)=O)CC2)ccc(F)c(Cl)c1 10061,c1(C(N2CC3C(NC(CCNS(C)(=O)=O)=O)(C3)C2)=O)cc2c(Cl)nccc2s1 10062,CN1CCC(O)(C(N2CCC(CC(N3C4CCC3C(N)C4)=O)C2)=O)CC1 10063,C1(NC(CCC2CCCN(C(c3c(CC)occ3)=O)C2)=O)CNC(=O)C12CC2 10064,CCCC(O)CC(=O)NC(CN(C)C(c1nc(C)ccc1F)=O)CC 10065,C1(CC=C)(NC(C2CCOC2C)=O)CCN(C(C2CCN(CC(C)C)CC2)=O)C1 10066,c1(C(=O)NC2CC3(C(N4CC(N5CCC5)C4)=O)COC2C3)cn2ccccc2n1 10067,CC(CCC(C)(C)C)C(=O)NCC(O)C(=O)N1CC(F)(CF)C1 10068,C1(C(N2CCC(N(C(=O)CC3CCC(=O)N3CC)CC)C2)=O)CC2(C1)CC2(F)F 10069,N1(C(C(C)NC(CC)=O)=O)CC2CC1C2NC(=O)C(C)=C1CCC1 10070,c1(C(=O)NC2(CCNC(C(CCCCC)F)=O)CCC2)nc2nc(C)ccn2n1 10071,C#CCC(CC(=O)NC1CCCCCC1)NC(c1cccc(C)c1C)=O 10072,C(C(C)(C)C(=O)N(C(CNC(C1(c2ccccc2)CCCO1)=O)C1CC1)C)SC 10073,c1(OC)ccc(F)c(C(=O)OCC2(c3cc[nH]n3)CC2)c1 10074,N1(C(c2c(C)cc(SC)o2)=O)CCC(C)C(NC(C2CCCS2)=O)C1C 10075,N1(C(c2c(C)oc(C)c2Br)=O)CCN(C(=O)C(C)N(C)C)CC(C)(F)C1 10076,N12CCCC(O)(CC1)c1cn(nn1)CC2=O.c1(SCCC)cnc(OC)c(F)c1 10077,c1(C(N2CC(F)(COC)C2)=O)cccc(CNC2CC(n3cnnc3)C2)c1 10078,C1(C(=O)NC(CC)CNC(C2(OC(C)C)CCCC2)=O)CCC(F)(F)C1 10079,c1(NC(=O)NCc2nc(-c3c(C)ccs3)on2)cc([N+](=O)[O-])cc([N+](=O)[O-])c1C 10080,Cc1ccc2nnc(CCNC(=O)NCC3(C)CCOC3)n2c1 10081,N1(C(CC2CN(C(c3ccc(CC)s3)=O)CC23CC3)=O)CCn2ncc(C)c2C1 10082,C1(C#N)(CC(=O)N(CCCNC(=O)C(C)CC2CC2)CC)CCOCC1 10083,C(=O)(C(CC(C)C)NC)N(CCN(C(=O)C(O)C1CC1)Cc1ccccc1)CC 10084,C1(F)(C(N(CCCCNC(=O)CN(CCC(N)=O)C)C)=O)CCCC1 10085,c1(CC(=O)NCCC(C)NC(CC2N(C(C)C)CCC2)=O)ccnc(Br)c1 10086,N#CC1CN(C(c2cc(Cl)ccc2Cl)=O)CCN1C(c1cnnc(Cl)c1)=O 10087,CCCCC(O)CC(=O)N(CCN(C)C)CC1CCC(C(N)=O)O1 10088,C1(CS(C)(=O)=O)C2CCC1CN(C(=O)COC(=O)CCC1CCC(=O)N1)C2 10089,C(C(F)(F)C(=O)NCC(C1CCN(C(=O)CC2(CO)CCCC2)CC1)F)N(C)C 10090,N1(C(C2(C)CC(C)C2)=O)CCN(CCN(C)C(C2CC2Br)=O)CC1 10091,N1(C(C(COC)(F)F)=O)CCCC(O)(CN(C)C(C2CCCC(C)(C)C2)=O)C1 10092,N1(C(Cn2ccc(C)n2)=O)CC2(C1)CN(C(=O)Cc1ccnc(F)c1)CC2CO 10093,c1(OC)ccc(-c2nc(C)c(C(C)NC(c3nnnn3C3CC3)C3CC3)s2)cc1 10094,c1(OC)cc(C)cnc1C(=O)NC1(C(=O)O)CC(OC)C1 10095,N#Cc1c(F)cc(C(=O)NC2CC(CNC(=O)C3=COCCC3)C(O)C2)cc1F 10096,C12(CNC(C(C)=CC)=O)CC(CO1)N(C(=O)Cc1ccccc1CC(N)=O)C2 10097,C(C(C)(C)CCCc1ccccc1)N(C(C)C)C(C1CC1C(F)(F)F)=O 10098,Cc1ccc(CNC(C2(NC(=O)Cc3ccnc(O)c3)CC2)=O)cc1 10099,N1(C(CCCCSC)=O)CCC2(CC(NC(c3cc(C(N)=O)cs3)=O)CO2)C1 10100,C(=O)(C1=C(CCl)N(c2ccc(Cl)cc2)C(=S)NC1c1ccc(=O)n(C)c1)OCC 10101,C(=O)(C#CC1CCOC1)NCC1C(C(=O)NC2C(C)(C)C2(C)C)CC1 10102,C(=O)(C1=CN(C)S(=O)(=O)N=C1C)N(CC(CNC(C(C(CC)O)(C)C)=O)(C)C)C 10103,C(=O)(C(CN=[N+]=[N-])NC(=O)CN1CCN(C)CC1)NCc1c(C)ccs1 10104,CCCC(C(=O)NCCCN(C(C)C)Cc1csc(C(C)C)n1)OC 10105,N1(C(CC(=C)Br)=O)CC2CCCC2(NC(=O)CCc2ccccc2Cl)C1 10106,Cc1cc(P(C)(C)=O)oc1C(=O)NC(C)CNC(c1cc(C2CC2)cs1)=O 10107,N1(C(C2C(C(=O)OCC)C2)=O)CCC2(C1)CN(C(c1n[nH]c(C)n1)=O)C2 10108,N1(C(C=C(COC)C)=O)CC2ON=C(CNC(c3csnc3Br)=O)C2C1 10109,C1(NC(CCC#CC)=O)CC2(NC(c3scnc3COC)=O)COC1C2 10110,C1(C)(CCNC(C(CC)O)=O)CCN(C(c2ccc(-c3nc(C)no3)cc2)=O)C1 10111,c1(C(=O)OC)cccc(C(N2CCC(NC(=O)CC3CC(SC)C3)C2C)=O)c1 10112,Cc1ccc2c(C(N3CCOCC3CCNC(=O)CCC(C)(C)F)=O)c[nH]c2c1 10113,C1(C)(C(N(C)CC2OCCN(C(CCCC=C)=O)C2)=O)CC2(CCC2)C1 10114,C=C(C)CCC(=O)NCCC1CC(NC(=O)C(F)(F)c2nc(C)cs2)C1 10115,C1(N=[N+]=[N-])(C(=O)Nc2c(COC)nn(C)c2)CCN(C(=O)Cc2csc(C)c2)C1 10116,N1(C(C(C)(C)N2CCOCC2)=O)CC2(C1)CN(C(C13CC(CO1)C3)=O)CC2CO 10117,C1(C(N2CC=C(C)C2)=O)(C(C)C)CCN(C(=O)CCC2CCC2)C1 10118,CC(C)CC(O)C(=O)NCCN(CCCN(C)C)C(C1CCCSC1)=O 10119,c1(C(N2CCCCC2C2CCCC2O)C(=O)NCCC)cc(Br)ccc1F 10120,CC1(C)C(CC(=O)NC(c2nn[nH]n2)=O)CCN1C(=O)Cc1cccc(Cl)c1 10121,c1(C(=O)NC2CC(NC(c3c(CC)nccn3)=O)C2)nc(C2CC2)ncc1Cl 10122,CN1CCCC1(C)C(=O)NCCOCCCNC(C1CCCS1)=O 10123,C1(C(=O)NC2CC(CNC(C(C)CC3CCCC3)=O)C2)Cc2ccc(F)cc2O1 10124,C1(c2ccccc2)(NC(CCN(CCCCC)C)=O)CCN(C(=O)CSC)C1 10125,c1(C(=O)NCCCCCN(C(c2ccc(CC)nc2)=O)C)ccc(C)c(N)c1 10126,c1(NC(=O)NCC(N2CC(C)(C)C(CO)CC2)=O)cnnc2ccccc12 10127,C1(NC(c2c(C)nns2)=O)CCCN(C(=O)CC2CCN(C)C2)C1C 10128,c1(C(=O)NC(C2C3CNCC23)C(=O)OC)csc(Cl)c1OC 10129,c1(OC)ccc(O)cc1C(=O)NCC1CCCC(NC(C2CC(F)C2)=O)C1 10130,c1(C(N2CC(N(C(c3c(C)nccc3)=O)C)C(F)C2)=O)cc(C2CC2)nnc1O 10131,c1(CN(C)C)cncnc1O.c12ccoc1C(=O)N1CCC(C1)CC(=O)N(C)C2 10132,n1(C(CC)C)nc(C(C2CCC2)OC)nc1-c1ccc(OC(F)F)cc1 10133,CC(CCN(C(=O)CCC1OCCO1)C)NC(=O)Cc1nc[nH]n1 10134,Cc1cccc(N2CCC(NC(=O)CC3(C)CCOC3)C2=O)c1 10135,N1(C(c2cnsn2)=O)CCC2CN(C(C3CC(C4CCC4)C3)=O)C2C1 10136,C1(CC)(NC(=O)COCP(C)(C)=O)CCN(C(=O)C=CC(C)(C)C)CC1 10137,c1(C(=O)NCC(CN(C(c2ncc(C)c(C)c2)=O)C)C)ccc2ccnn2c1 10138,C1(C(N2CC(C(=O)NC)(NC)C2)=O)COC(=O)N1C 10139,N1(C(C2CC(SC)C2)=O)CC(NC(c2csnc2C)=O)CC12CCCC2 10140,CC(=O)CCCC(=O)NCC1C(O)C(O)CN1C(c1c[nH]nc1Br)=O 10141,C1(NC(c2c(CC)nns2)=O)CN(C(=O)C2=CSCCO2)CCC1CO 10142,N1(C(c2ncn(C)n2)=O)CC(NC(=O)C(F)(F)C2(O)CCC2)CC12CCCCC2 10143,CCC(C(=O)NCC1(C(C)NC(=O)Cc2ccncc2Cl)CC1)C(F)(F)F 10144,C12(NC(=O)COc3ccon3)CCCN(C(C3(CO)COC3)=O)CC1C2 10145,N1(C(c2n(CC)ccn2)=O)CC2CC1C2NC(=O)CN1C(=O)CCC1=O 10146,C1(C2CN(C(c3ccc(C#N)[nH]3)=O)C2)(NC(CSCCC=C)=O)CC1 10147,c1(C(=O)NC(c2cccc3cc[nH]c23)CC)cnn2cc(CCOC)cnc12 10148,c1(C(N(CC(CN(C(=O)CCC2CC2(C)C)C)O)C)=O)cc(P(C)(C)=O)cs1 10149,CC1CC(C2CN(C(=O)CN(C(C3OCCCC3(C)C)=O)C3CC3)C2)=NO1 10150,c1(C(N(CCC(=O)N(CC(=O)NCCC)C)CC2CC2)=O)cc(C)c[nH]1 10151,c1(C(=O)NCC(CNC(CCCOCC=C)=O)O)ccc(S(=O)(=O)C(F)F)cc1 10152,Cc1cccc2c(=O)c(C(=O)NC3CC(NC(C4COCC4(C)C)=O)C3)c[nH]c12 10153,c1(C(=O)NC2CC(F)(CNC(C3(C4CCCO4)CCC3)=O)C2)cc2cn[nH]c2cn1 10154,c1(CC(=O)NC2CC(NC(CC3C(C)(C)C(O)C3)=O)C2)ccccc1[N+](=O)[O-] 10155,CC1C(=O)CC2CCC1N2C(=O)NNc1nccs1 10156,Cn1cc(C2CC2C(=O)NC2(CNC(=O)C(C3CC3)N(C)C)CCOC2)cn1 10157,c1(OCCNC(C(=O)NC2CC(C(=O)OC)NC2)=O)cccc(Br)c1C 10158,c1(C(N2C(CNC(C(C(C)C)C)=O)CC(O)C2)=O)cc(=O)n(C)cc1Br 10159,c1(NC(c2ccc(-c3ccc(Br)s3)s2)=O)ncccc1OCCF 10160,C(=O)(C(O)C1=CCCCC1)N1C(C2(NC(CC(=O)NCC)=O)CC2)CCC1 10161,CCC(C)(CS(C)(=O)=O)C(=O)NCC(O)CNC(=O)CNC(=O)NC 10162,c1(C(=O)NC2(CN(C(C(CC)OC)=O)C)CC2)cc2c(C#N)cccc2[nH]1 10163,N1(C(COCC#C)=O)CC(C2CCCN(C(C3(CC)CCCO3)=O)C2)C1 10164,N1(C(Cc2c(C)nc[nH]2)=O)CCC(CO)C(NC(C2(C(C)C)CCC2)=O)C1 10165,CN1CCC(C(=O)NC(c2ccc(CO)cc2)CNC(c2cn[nH]c2)=O)CC1=O 10166,c1(C(N(CCC(C)NC(=O)C(C)(C)C)C)=O)ccc2c(c1)OC(C)(C)OC2 10167,CC(C1OCCc2ccccc21)N(S(=O)(=O)Cc1csc(Br)c1)C 10168,O=C(C(O)CNC(c1cccnc1)=O)NC(C1CCCC1)CO 10169,N1(C(c2c(C)scc2)=O)CCC(C(=O)NCC(F)Br)C1(C)C 10170,C1(NC(=O)COc2cccnc2)COCCN(C(C2C3COCC23)=O)C1 10171,C1(NC(CC(CC)CN(C)C)=O)CC2(CCC(NC(=O)CNC(C)=O)CC2)C1 10172,n1(CC)nccc1S(=O)(=O)N1CCC(NC(=O)C(C2CC2)OC)C1 10173,N(C)(S(=O)(=O)N(C)CC1CC1)CC#C 10174,c1(C(C(=O)NCC=CCl)NC(CN(C)CC)=O)cnn(C)c1 10175,C1(Oc2ccc(C)cn2)CCN(N2CCCC(N3CCCCC3)C2)C1 10176,N1(C(c2c(CNC(CC3C(C)(C)C(O)C3)=O)cco2)=O)CCOCC2(CC2)C1 10177,C1(CNC(CCN(CC)CC)=O)CN(C(=O)Cc2csc(NC=O)n2)C2CC12 10178,C(N=c1[nH]c(N2Cc3cnn(C)c3C2)nc2c1CC(C)CC2)C1CCC(C)N1C 10179,C(=O)(CS(=O)(=O)CCO)N(C)CC1CN(C(C2CCOC(C)(C)C2)=O)CCO1 10180,N1(C(C(COC)CC(C)C)=O)CC(C)OC2(CCN(C(=O)CCC(C)C)CC2)C1 10181,C1(C(=O)NC2CC(CNC(c3c(CC)noc3)=O)C2)CCCCC12OCCO2 10182,c1(OC)ccc(C)cc1C=CC(=O)NCC1CCN1c1nc(C2CC2)ns1 10183,c1(NC(C2CCCC2)C=C)ncnc2ccc(NC(=O)C(C)CCC(C)(C)C)cc12 10184,C(CC(C)C(=O)NC1CCC(F)(CNC(c2c[nH]nc2C(C)C)=O)C1)OC 10185,Cc1nsc(NC(=O)C(N2CC(F)CC2c2ccccc2)=O)c1Cl 10186,C(CC(C)C(C)(C)C)NC(C1(CCNC(C=CC)=O)CCC1)=O 10187,C1(CNC(C(CC=C)NC(C)=O)=O)CC(C(=O)NCC2(N(C)C)CCC2)=NO1 10188,N1(C(C(C2CC2)SC)=O)CC(NC(=O)CC2CCSC2)C(C)(C)C1 10189,C1(NC(C(N)=O)=O)CC2(CCN(C(C3CCCOC3)=O)C2)C1 10190,C1(NC(C2(COC)CCOCC2)=O)CCN(C(c2ccsc2)=O)CC1(C)C 10191,c1(C(N2CCC(O)(CNC(C3C(CCOC)C3)=O)C2)=O)ccc([N+](=O)[O-])o1 10192,C(=O)(C(C)(O)C(C)C)NC1CC2C(NC(C(C)OCC(C)C)=O)C2C1 10193,C(C(C)(C)CC(=O)NCC1CCN(Cc2nnnn2C(C)(C)C)C1)OC 10194,C1(NC(C(C)OCC)=O)CCN(C(=O)Cc2ccc(C(C)=O)s2)CC1(C)C 10195,CC(C)C(C(=O)NC(CNC(=O)Cn1cnnn1)C(C)(C)C)NC=O 10196,c1(CC)[nH]nc(Cl)c1C(=O)N(CCN(C1CCCCC1C)C)CC 10197,CCC(CC)C(C)C(=O)NC1COCC1CNC(C1(OC)CCCCC1)=O 10198,N1(C(=O)NCc2ncc(CC)o2)CCCCC1CCNC(C)=O 10199,c1(CN(c2ncnc(OCC)c2OC)C2CCCCNC2)cccc([N+](=O)[O-])c1 10200,N1(C(CCCNC(=O)NC)=O)CCC(CCNC(C2(COC3CC3)CC2)=O)CC1 10201,CC(C(=O)NC1(CNC(C2(C(F)F)CCC2)=O)CCC1)F 10202,Cc1ncc(C(=O)Nc2ccc(-c3cnc(N4CCC4)nc3)nc2)cc1Br 10203,C(=O)(C1CCc2ccccc21)NC1(C(=O)NCC(c2cnc[nH]2)C)CCCC1C 10204,C1(C(=O)NC(c2ccns2)C)(CC)CCCN(C(c2cnn(C(C)C)c2)=O)C1 10205,C#CCCCCCC(=O)N1CCCC2(NC(=O)C(C)Cc3ccccc3)CC2C1 10206,Cc1cc(C(=O)OC(C(=O)Nc2ccc(N(C)C)c(F)c2)C(C)C)ncc1N 10207,c1(NCC(CCC)(C)C)ccc(S(=O)(=O)NCC2C=CCC2)cc1Br 10208,c1(C(=O)NCCC2CCCN(C(C3CC(F)C3)=O)C2)nccc2n[nH]cc12 10209,c1(C(C)=O)cncc(C(=O)NCCCCNC(C2CCC2(F)F)=O)c1 10210,N1(C(CC(C)OC)=O)CC2(CCN(C(=O)C(C)Sc3ccc(N)cc3)C2)C1 10211,c1(C(N2CCCSCC2C)C(=O)Nc2c(OC)cccc2)sc(C)c(Br)c1C 10212,C1(C#N)(NC(CSc2ccc(OC)cc2)=O)CCN(C(C2CCCCC2)=O)C1 10213,N(C1CCCn2cnnc21)C(C1CC(O)(COCC)C1)=O.C1(=O)C2=NOC(C2)N1 10214,c1(C(=O)NCc2cccc(-c3cccc(OCC)n3)c2)ccc2sc(O)nc2c1 10215,c1(C(N2CCC(C)C2CNC(=O)CC(F)(F)F)=O)cnn2c1CCC2 10216,O=C1CC2(CCCN(C(=O)C3=NOC(CO)C3)CC2)N1 10217,CC(CN(C)C)C(=O)N1CCCC1C(C)NC(=O)N(C)C 10218,C(=O)(C(CNC(=O)CN1CCCC1=O)C(C)C)N1CCC(C(=O)NC)CC1 10219,C1(NC(C(C)NC(=O)Cc2cc[nH]c2)=O)CN(C(=O)OC(C)(C)C)CC1C 10220,CCCC(CCC)CC(=O)NC1CN(C(C2CCCOCC2)=O)CC1OC 10221,C(C1c2ccccc2CN1C(=O)C(n1nccc1C)C)NC(CC(=O)NC)=O 10222,c1(NC2CCN(C(c3cnc(SC)nc3Cl)=O)C2)ncnc2sc(C(C)C)cc12 10223,S(=O)(=O)(c1ccc(C(=O)NC2CCC(CNC(=O)C(C)C(C)O)C2)cc1)NCC 10224,N1(C(CNC(CSCC(N)=O)=O)=O)CC2(SCCCO)OCC(C(F)(F)F)C2C1 10225,n1(CC(=O)NCC2CCN(C(=O)C(C3CCOCC3)O)C2)ncccc1=O 10226,c1(C(N(C2CCN(C(COC)=O)CC2)CCO)=O)cnn2cc(OC)ccc12 10227,N1(C(C(CC)NC(N)=O)=O)CCN(C)C(CNC(c2cc(Cl)sc2Cl)=O)C1 10228,C1(N(C(C(=O)Oc2ccccc2)=O)CCCO)CC2CC1CN2 10229,c1(CC)cc(C(=O)NCCC(C)NC(c2ccn(C(C)(C)C)n2)=O)oc1CC 10230,CC(CNC(C1(F)CCN(C(c2ccc(CO)cn2)=O)CC1)=O)CC(F)(F)F 10231,C1(C(=O)NCC(CNC(c2c(C)n[nH]c2)=O)C)CCCN(CC(C)C)C1 10232,c1(N2CCOCC(CNC(c3nc(CC)sc3)=O)C2)nnc(C)c(C)c1C#N 10233,c1(N2CC(C)S(=O)CC2)ccc(Br)c(S(=O)(=O)N(CC(O)CF)C)n1 10234,CN1CCCC1C=CC(=O)NC1(C(=O)N(C2CSC2)C)CC(F)C1 10235,C12(CNC(c3c(C(C)C)n[nH]c3)=O)CCC1CN(C(c1ccc(=O)n(C)c1)=O)C2 10236,C1(Nc2nccc(OC)n2)(CO)CCN(C(C2CN(C3CCOCC3)C2)=O)CC1 10237,N1(C(CC2(N(C)C)CC2)=O)CC(NC(=O)Cn2cc(Cl)cn2)C(C(F)F)C1 10238,C1(NC(=O)NCCC2=NN(C)C(=O)C2)CCc2ccccc2C1=O 10239,c1(OC)nsc(OC)c1C(C)NC(C1(n2cc(F)cn2)CC1)=O 10240,C1(C(=O)NC2(C)CCN(C(=O)CS(N)(=O)=O)CC2)CC(O)c2ccccc2O1 10241,C12(OC)CCCN(C1)C(c1n(CCCCCC)nnn1)CC2.C(C)(CC(C)C)SC 10242,C1(C(=O)OC)CCOC1C(=O)NCCN(C)C(C1CC(C(C)C)C1)=O 10243,C(CCCC(=O)N1CC2C(CNC(=O)C(c3ccc(Cl)s3)=O)C2C1)SC 10244,CCS(=O)(=O)CC(=O)NC1(CO)CCN(C(c2cccc(OC)c2OC)=O)C1 10245,c1(C(N2CCCC(CNC(C(C)OCCC=C)=O)C2)=O)cc(Cl)c(OC)cc1C 10246,C(=O)(C(C)(C)CS(C)(=O)=O)NCCCC(C)NC(=O)C(O)CC(N)=O 10247,C(=O)(CC(C(C)C)NC(=O)C(=O)NC1CC1)N1C(CN(CC)CC)CCC1 10248,c1(C(=O)NC(C2CCN(C(c3cc(CO)ccn3)=O)CC2)C)cc(O)cc(=O)o1 10249,Cc1cnc(Cl)[nH]c1=NCC=Cc1ccc(NC(=O)CC2CC(F)C2)cc1 10250,N1(C(CNC(CC)=O)=O)CCC(CCNC(C2(C3CC3)CCC2)=O)CC1C 10251,c1(C(=O)NC(C)C(C)(C)NC(=O)CCC(C)C#N)cc(N(C)C)ccc1F 10252,N1(C(CC2CCN(C(=O)CCc3ccccc3)CC2)=O)CCOCC2(CCC2)C1 10253,c1(CN2C(C(=O)NCc3ncccc3F)CSCC2)cc(Cl)ccc1Cl 10254,N1(C(CCOCC#C)=O)C2CCC1CN(C(c1cscn1)=O)C2 10255,Cc1cc(C(=O)NCC2CN(C(=O)COCCF)CC2C)c2c(C)nn(C)c2n1 10256,c1(C(=O)NCC(C2N(C(C(CC)CC)=O)CCCC2)(C)C)cnc2ccnn2c1 10257,N1(C(=O)CCN(C(c2nsnc2O)=O)CC2CC2)CC23CCC2(COC3)C1 10258,c1(NC(C2(C)CCN(C(c3ccc(CF)cc3)=O)C2)=O)ccc(F)c(O)c1 10259,Cc1nn2cccnc2c1C(=O)NC(C1CCCN1C(=O)CN1CCCC1=O)C 10260,C(CN=C(NCC1Cc2ccccc2C1)N1CCC(C(C)O)C1)c1ncc(C)nc1 10261,C1(=O)C(C(=O)N(CCSC)CC)O1.c1(C(=O)NCC)ccc(CNC(C)=O)cc1 10262,C(=O)(CC(C)C(F)(F)F)NCC1C(CNC(C(NOC)=O)=O)CCC1 10263,C1(CCNC(CCC#CC)=O)CN(C(C2(C3CCCO3)CCC2)=O)CCS1(=O)=O 10264,C1(C(=O)NC2(CCC)CC2)C(C2CC2)CCN1C(=O)COCCCF 10265,C1(N(S(=O)(=O)CC#N)C)CCCN(CCF)C1=O.c12ccc(cc1)[nH]c2=O 10266,N1(C(CCCC#C)=O)CCC(C(=O)NC(CCF)C(=O)OC)C(C)C1 10267,N1(S(C)(=O)=O)CCC(C(=O)NCCC2CN(C(=O)C(F)=CC3CC3)CCO2)CC1 10268,C(=O)(CCC(=O)NCCCCCCNC(C1CC1(Br)Br)=O)NCC 10269,C1(NC(C2CN(C(C)=O)C2)=O)CN(C(c2cc(Cl)ccn2)=O)C2(CCOC2)C1 10270,c1(C(N2C(C)C(NC(=O)CCc3ccnn3C)CC2)=O)cc2ncccc2s1 10271,C1(CC)CNC(=O)CN1C(=O)CCC1CN(C(=O)NC2C(Cl)(Cl)C23CC3)C1 10272,C#Cc1ccc(C(N2CCCC2CCC(N2CCOC(C(N)=O)C2)=O)=O)cc1 10273,c1(CC(N2CCC(Cc3cn(CCCCF)nn3)C2)=O)ccc2c(c1)CCO2 10274,C(=O)(C(CC(C)C)C(C)C)NCCN1CCN(C(c2c(N)ccc(C)c2)=O)CC1 10275,Cc1c(CN2CC3(CCN3C(c3cc(Cl)cc(Cl)n3)=O)C2)[nH]c2ccccc12 10276,N1(CC)CCCCC1C(=O)NC(C)C(=O)O.C12CCN(C1)C2=O 10277,C12CN(CCN1CC(F)F)C2=O.c1(-c2nc(C3(CN)CC3)on2)cccc(Cl)c1 10278,Cc1ccc(C(=O)NCC(=O)NCC(C2CC2)NC(=O)C=CSc2nc[nH]n2)s1 10279,N1(C(c2cnc(C)[nH]2)=O)CCCC12CCN(C(=O)C(C)CC(C)(F)F)C2 10280,CC(CC(=O)N(C)CC1CCCCN1C(C1CCCO1)=O)C(F)(F)F 10281,c1(NC(N2CCC(S(C)(=O)=O)C2)=O)csc2ccc(F)cc12 10282,c1(C(=O)NC2(CNC(C3=CCC(C)(C)CC3)=O)CC2)cc(Cl)cc2c1NCCC2 10283,N1(C(c2cc(CC)nc(O)c2)=O)CC2(CCN(C(=O)C(CO)NC(=O)NC)C2)C1 10284,C1(CNC(c2cn(CCC=C)nn2)=O)C(C)CCCN1C(=O)C#CC(=O)N(C)C 10285,c1(C(=O)O)cnn2c(NC3(n4ncnn4)C4CCCOC4C3C)cccc12 10286,C1(C(N2CCC(COC)(NC(=O)C=Cc3cscn3)C2)=O)CC2COCC2C1 10287,C1(C(=O)NCC(CCC)OC)CCC2CCC1N2C(=O)CNc1ccccn1 10288,N1(C(Cc2c(C)oc(-c3ccsc3)n2)=O)CCc2nncn2CC1 10289,CC(C)C(C(=O)NC1(C)CN(C(C2CCC(=O)C2)=O)C1)c1cccc(Cl)c1 10290,c1(C(=O)NCCNC(CCc2ccc(C)nc2)=O)nc(C)n(C)c1C 10291,c1(C(=O)OC)cc(NC(C2COCCN2Cc2coc(Cl)n2)=O)ccc1F 10292,c1(OC)ccc(CNCC(N)C(C)C)cc1Cl 10293,C12(CNC(c3cncc(SC)c3)=O)CCC(CC1)CN2C(=O)C(C1CC1)C1CC1 10294,c1(COC)ccoc1C(=O)NCCC(C)NC(c1ccc(CN=[N+]=[N-])o1)=O 10295,c1(C(=O)NOCCCCC2CC2)ncnc(O)c1F.C12(CCSC1)C(=O)N2 10296,N1(C(C(C2CCCO2)SC)=O)CCC(N(C(=O)CCOC2CCC2)CCO)CC1 10297,N1(C(C(Cn2cc(-c3nncc(OC)c3)nn2)OC)=O)CCC(C)(O)C(C)(O)C1 10298,N1(C(c2nccc(C)c2O)=O)CCC2(CCC2)C(NC(C2CCCSC2)=O)C1 10299,C1(C(N(C2CC(=C)C2)C)=O)CCC(n2cc(CCc3nn[nH]n3)nn2)CC1 10300,S(=O)(=O)(c1ccc(C(=O)NC2(CO)CN(C(=O)C(F)(F)C3CC3)C2)cn1)N(C)C 10301,N1(C(CCCCCOC)=O)CC(CNC(C2(CCO)CC2)=O)CC12CCC2 10302,N1(C(C(C#N)CO)=O)CC2=C(C1)CN(C(C13C4C5C1C1C3C4C51CO)=O)C2 10303,c1(C(=O)NC(CC2(CC)CCC2)=O)cc(CN2CCCC(NC(C)C)C2)ccn1 10304,C(=O)(C(C)(C)C(C)(C)O)NC(C(=O)N(CC(C)C(C)(C)C)C)CC(F)F 10305,Cn1c(C(=O)NCC2CCN2C(c2cc(CO)on2)=O)cc2cc(Cl)ccc12 10306,C(=O)(CCCC(=O)N1CCC(C(F)(F)F)C(C(=O)C=CC(F)(F)F)C1)N(C)C 10307,C12CN(CC13CCC3)C(=O)c1nc(C)ncc1C(=O)N2.c1(CC)csnc1Cl 10308,N1(C(=O)Nc2cc(C)c(NS(C)(=O)=O)cc2)CCN(C)c2ccc(C(F)(F)F)cc21 10309,Cc1c(C(=O)NCC2CCN2C(c2cc(N(C)C)ccn2)=O)cnn1C(C)(C)C 10310,C(=O)(N=c1[nH][nH]cc1-c1ccc(F)cc1)c1cncnc1.Cc1n[nH]cc1 10311,C1(CC=C)(NC(c2csc(CCCC)n2)=O)CN(C(=O)C(F)CC2CCCC2)C1 10312,N1(c2nc(OC)nc(C)c2)CCOC2(CCCN(C(C3CCCCC3C)=O)C2)C1 10313,Cc1ccc(C(N2CCC(C(=O)Nc3ccc(F)nc3)C(O)C2)=O)c(F)c1 10314,C1(COC)(NC(=O)CN2CCS(=O)CC2)CCN(C(C2(Cl)CC2(F)F)=O)C1 10315,C12(CNCC3C(C)CC=CC3)CC(CO1)N(c1cc(O)ncn1)C2 10316,c1(CCC(N2CC(OC)C(NC(=O)CC3CSCCS3)C2)=O)cccc(F)c1F 10317,c1(C(C(=O)NCc2cn(CCSC)nc2)CC)cccc(Cl)c1 10318,C(=O)(CCCCCc1ccccc1)NC1C(CNC(c2c(CC)cc[nH]2)=O)C1 10319,N1(C(C2CC(N(C)C(C34CC(CO)(C3)C4)=O)C2)=O)CCC([N+](=O)[O-])CC1 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10354,CC1(NC(=O)C(F)CC2CCCC2)CC(NC(=O)Cn2ccc(C(F)(F)F)n2)C1 10355,c1(CC)cc(N)ccc1C(=O)NC(C)(C)CNC(C1(C(F)(F)CC)CC1)=O 10356,N1(C(c2c(C)nn(C(C)C)c2)=O)CCC2(CCC2)C(NC(C2CC(C)(O)C2)=O)C1 10357,n1(CC(=O)NCC(C)(O)CNC(C2CC23CCC3)=O)cnccc1=O 10358,c1(OC)ccnc(O)c1C(=O)NC1CCCCN(C(C2Cc3nncn3C2)=O)C1 10359,N1(C(c2c(C)ccc(C(=O)OC)c2)=O)CC(C)N(C(=O)CC(C)SC)C(C)C1 10360,N1(C(COCC(C)C)=O)CCC(N(C)C(C2CC3(CC(=O)C3)C2)=O)C(C)C1 10361,CC(CC1CCC1)C(=O)NCC1(NC(c2cnnn2C)=O)CCCC1 10362,C1(C(C(C)C)NC(Cc2nnc(C)o2)=O)CCN(C(C2(O)COC2)=O)CC1 10363,C(=O)(C1=CC2CCC1C2)NC1CC2C(NC(c3cn(CCC)nc3C)=O)C2C1 10364,S(=O)(=O)(c1cccs1)CCn1cc(-c2nc(C3(C)CCO3)sc2)nn1 10365,c1(N(CCCN(CC(C)(C)C)C)C(C)C)nc(O)c2ccc(Cl)cc2n1 10366,c1(C2C(C(=O)NC3C(CNC(COC(CC)C)=O)CC3)CC2)ccccc1 10367,C1(NC(CC2(OCC)CC2)=O)CCC2CN(C(C3CCSC(C)C3)=O)CCC2C1 10368,N1(C(CC(CCC)O)=O)CCCC(C)(C)C1CNC(C1(C(C)(F)F)CCC1)=O 10369,c1(OC)c(C(N2CC3CC2CN3C(C2CC(=C3CCC3)C2)=O)=O)c(C)nn1C 10370,C1(NC(CC2ON=C(C)C2)=O)CN(C(c2csc(-c3cn[nH]c3)n2)=O)C(C)(C)C1 10371,N1(C(C)C)C(=O)CCC1C(=O)N(C1CCN(C(=O)CC2(C3CC3)CC2)C1)C 10372,c1(C(=O)NCc2cnc(OCC#C)c(Cl)c2)ccc2c[nH]nc2c1 10373,C(=O)(C(C)(C1CC1)N(C(=O)CCc1cncn1C)C)NCC(CC)O 10374,Cn1cnc2nc(N3CC=CC(NC(c4cc(C5CCCC5)[nH]n4)=O)C3)ncc12 10375,CC(C)(C)C(O)CCC(=O)NCC1CN(C(C2CC2C(F)(F)F)=O)C1 10376,c12ccccc1S2.c1(C(=O)NCC(C)SC2CN(C(N)=O)C2)[nH]nnc1C1CC1 10377,CC(C)(C#N)CC(=O)N1CCC(F)(CNC(C2CC3(CCCC3)C2)=O)C1 10378,c1(C2CC2)ccc2c(c1)CCCN2.C1(N2CCC2)CCCCCC1.CO 10379,c1(C(N2CC3(C2)SCCC3NC(C23CCC2C3)=O)=O)ccc2nsnc2c1 10380,CCC(C)(C)CCCC(=O)N1CCC(N(C)C(C2CC3CCC3C2)=O)C1 10381,CN1CCC(c2ncc(C(N3CC(n4cc(C(=O)O)nn4)C3)=O)[nH]2)CC1 10382,c1(OC)cnc(C(=O)NC(C)CNC(c2n[nH]cc2CC(C)(C)C)=O)c(OC)n1 10383,C(C#Cc1ccccc1)N1CCN(C(=O)CC2CCCNC2=O)CC1 10384,C1(SCCNC(=O)CC2CCCO2)CN(C(=O)C(=O)NCC(F)F)CCC1(F)F 10385,c1(C(=O)NC(CNC(C2(C)CCN(C)C2)=O)(C)CO)cccc2c1OCC2 10386,CC(C)CC(=O)C(=O)NCCC(O)CNC(=O)CCCN(C)C(C)C 10387,N1(C(CCNC(C)=O)=O)CCC2(CC1)OCCCC2NC(=O)CSc1ccoc1 10388,C1(CNC(c2cc(C)on2)=O)C2CN(C(=O)C(C)(C)N3CCOCC3)CC12 10389,C1(OC)CCC12CC(C(=O)NCCC1CCN(C(c3cnc(=N)[nH]c3)=O)CC1)C2 10390,C(CCF)(C(=O)NCCNS(N)(=O)=O)NC(CCC1(C)CC1)=O 10391,C#CCCCCCCC(=O)NC(C(=O)NC1CCC(=O)NC1(C)C)C(C)OC 10392,C(=O)(CC(O)CC(C)C)N(CCC(=O)NCCc1noc(=O)n1C)CC=C 10393,N1(C(CC2(CSC)CC2)=O)CC(NC(c2ccc(-c3csnn3)cc2)=O)C(O)C1 10394,N1(CC)CCOC(C(=O)NCCCN(C(=O)CNC(=O)C(C)(C)C)C2CC2)C1 10395,C1(CC(=O)NCCOC2CC(CNC(CCSCC)=O)C2)CCNC(=O)C1 10396,C(c1ccc(CN(C)C=O)cc1)=CC(=O)OC(c1cc(Br)ccc1Cl)C 10397,CC(C(=O)NCCOCCOCCNC(=O)C=Cc1ncc[nH]1)C(C)O 10398,CCCCS(=O)(=O)CC(=O)NCC1(C2CC2)CCN(C(C2CCS(=O)(=O)C2)=O)C1 10399,c1(CN2CCC(C#N)(C(C)C)C2)cc(Br)cc(F)c1O 10400,S(=O)(=O)(c1c[nH]c(C(N2CC(CNC(=O)CCC3NC(=O)NC3=O)C2)=O)c1)NC 10401,c1(C(=O)NC(COC)C(=O)NCCC(C)(C)N(C)C)ncncc1Cl 10402,N1(Cc2cc(OC)cc(Br)c2)CCC2(CC1)CC2NC(c1ccn(C(C)C)n1)=O 10403,C1(CNC(C=CCC)=O)CC2CN(C(C3CC(OC)C3)=O)CC2C1 10404,C1(CNC(C2(CNC(CS(N)(=O)=O)=O)CC23CCC3)=O)CC(C2CC2)=NO1 10405,C1(O)(CCNC(C(C)C#N)=O)CCN(C(c2cc(C(N)=O)n(C)n2)=O)CC1 10406,c1(C(=O)NCC(C)(CC)NC(CC(CC)C(F)F)=O)c(F)ccc2occc12 10407,c1(-c2cn(C(n3cc(COC)cn3)OC)nn2)ccc2c(c1)CN(C(C)C)C2 10408,C(=O)(C1CCCc2sc(=N)[nH]c21)N1C(CNC(CNC(CC)=O)=O)CC(F)C1 10409,C(=O)(C(CCS(C)(=O)=O)OC)NC1CCN(C(CSCC#C)=O)CC(O)C1 10410,C1(n2c(C(CO)NC3(C(N)=O)CC3)nnn2)CCC(F)(F)CC1 10411,C(CN=c1cc(OCCNCc2ccc(CNC)o2)nc(C(F)(F)F)[nH]1)OC 10412,C12(NC(CNC(N)=O)=O)CC1CN(C(=O)CC(F)(F)Cl)C2 10413,c1(OCC(=O)NCC2CN(c3nnc(C(F)F)s3)CCO2)ccc(Cl)cc1 10414,N1(C(=O)NCC2CCSCC2)CCN(c2ccc(F)cc2F)C(=O)C1 10415,C1(C2(O)CCN(C(=O)C(C)C(C)(C)C)CC2)(NC(CCc2scc(C)n2)=O)CC1 10416,N1(C(C(CNC(C2CCC(=O)N2)=O)CC2CC2)=O)CCSC2(CCC2)C1 10417,C(=O)(C(C(=O)N1CCC(CC(=O)NCCC2CC3C=CC2C3)O1)C(C)(C)C)OC 10418,CC1COC(C)CN1C(c1ccc(Cl)s1)C(=O)NCC1CC1 10419,C=C(Cl)C(C)(C)C(=O)N1CC2CC(NC(C3(F)CCOC3)=O)C1C2 10420,C1(C(=O)NCCCNC(c2ccc(C3(F)CC3(F)F)cc2)=O)CCCC12CC2 10421,C#CCC(CC(=O)Nc1ccc(F)nc1)NC(c1ccoc1C)=O 10422,c1(OC)cc(C(N2CCC(NC(=O)Cc3c(C)cnn3C)C(C)C2)=O)ccc1C 10423,c1(C(=O)NC2CC2CNC(C2CC3COCC3C2)=O)ccc([N+](=O)[O-])cc1Cl 10424,C1(C(=O)NC(CNC(c2cc(C)n(C)c2)=O)(C)C2CC2)CNC(=O)CC1C 10425,Cc1cc(CN2CCC(C(N3CC4CC4(CO)C3)=O)C2)c2cc[nH]c2c1 10426,N1(CC)C(=O)CCC1CC(=O)NC1CC(N(C(=O)Cn2nnc(C3CC3)n2)C)C1 10427,c1(C(=O)NCC2C(NC(C(c3nccc(C)c3)(C)C)=O)CC2)cc(Cl)ccc1N 10428,C(C(=O)NC(C(=O)NC1CCC(C)(C)C1)C1(O)CCC1)(C(C)C)SC 10429,N12CCC(O)C(C1)C(=O)N1CCC2C1.C(COCCO)OCC 10430,c1(C(=O)NC(C)CNC(=O)Cc2cn(C)nn2)ccc2c(c1)CCS2(=O)=O 10431,c1(C(=O)NCc2c[nH]nc2C2CCNC2)cnn2ccc(N(C3CC3)CC)nc12 10432,c1(CCc2cn(CCC(N3CC(C(C)C)SCC3)=O)nn2)cnc2sccn12 10433,N1(C(C=CC)=O)CC2CN(C(C3C4C=CC(C4)C3CO)=O)CC(C1)O2 10434,Cc1cnc(C(=O)NCc2cccc(NC(=O)C(CC#N)c3ccccc3)c2)nc1 10435,C#Cc1ccc(CCCC(=O)NCC(C)CN(CC(C)(C)C)C(=O)C(C)O)cc1 10436,c1(N(C(c2cncc(Cl)c2)C(=O)NC2CSC2)C)ccc(OCC(N)=O)cc1 10437,N1(C(C2(SC)CCC2)=O)CCCCC(N(C(=O)Cn2ncccc2=O)C)C1 10438,N1(C(C(CCC)CCC)=O)CC2(C1)CN(C(C1CCCN1CCC)=O)CCO2 10439,CC1(CNC(C2(c3ccccc3)CC3(CC3)C2)=O)CCCN1C(c1ccsn1)=O 10440,C(CCCCCNC(=O)C(C1CCC(=O)N1)C)n1cc(C(C)OCC)nn1 10441,C(CN=c1nc(OC)cc[nH]1)C1CCC(NC(c2cc(OC)nc(C)c2)=O)C1 10442,Cc1nc(C(N2CC3CC2C3NC(C2(C)CCCOC2)=O)=O)cn1C(F)F 10443,N1(C(C2C3CN(Cc4cc(OCC)ncc4)CC32)=O)CCN2C(C)COCC2C1 10444,c1(CC(=O)NCC2COCC2NC(C2CC(O)C2)=O)csc(-c2ccccc2)n1 10445,C(=O)(C1=CNS(=O)(=O)N=C1C)NC(CNC(CCCCCC)=O)C1CC1 10446,C(=O)(C(O)CC(C)C)N1C(COC)(CNC(=O)C(C)=C2CC2)CCC1 10447,C1(CNC(CCSCCC)=O)CCN(C(=O)C(C)NC(=O)OC(C)(C)C)CC1F 10448,Cc1cc(OCCO)cc(NC(=O)OCCF)c1 10449,C(=O)(C(CC(C)C)C(N)=O)NC(CC)CNC(c1sc(F)cc1Cl)=O 10450,C=CCC(CNC(c1cn2c(n1)CCC2)=O)C(=O)NC(CN(C)C)CO 10451,C(=O)(C(C)C1=CCCC1)NC(CN(C(=O)CCC(CF)CF)CC)C 10452,C1(OCC=C)CCN(C(=O)C(CNC(C2CC2(F)Cl)=O)N(C)C)C1 10453,C1(CNC(C(C)=CC)=O)CCN(C(C2CCn3cc(C)nc3C2)=O)CCC1(F)F 10454,Cc1cccc(C(=O)NCC2(C)CCCN2C(=O)CC2C=CCC2)c1Br 10455,c1(C(c2n(CC=C)nnn2)NCC2(C)CC=CCO2)cc(OC)c(OC)c(Cl)c1 10456,Cc1ncc(CCNC(=O)C(C2CCN(C(c3csc(C)n3)=O)C2)C)s1 10457,c1(C(=O)NC(C2(O)CN(C(=O)CCc3ccc(F)nc3)C2)C)cncc(Cl)n1 10458,N1(C(C(C)(C)Cl)=O)C2CC1CN(C(C1(c3ccccc3F)CC1)=O)C2 10459,c1(C(=O)OC)ccc2c(c1)C(C(=O)N1CC(CC(C)NC(=O)C(C)COC)C1)CC2 10460,N1(CC)CCC(N=c2nc(C3CCCC3)[nH]s2)CC1.C1(CC(C)C)(C=O)COC1 10461,C1(CNC(c2n(CC)ccn2)=O)CN(C(C2(F)CC=CCC2)=O)CCN1C 10462,C(c1ccncc1C)=CC(=O)NC(CN(C(=O)CCCC(C)=O)CC)C 10463,c12cn(nn1)C2.N1(C(CC2(COC)CC2)=O)CC(CC(=O)OC)C1.NC 10464,C(=O)(C1(C)CCn2ccnc21)NCC(C)CN(C)C(c1csnc1Cl)=O 10465,C1(N(C(C)C)C(C2CC(N(C(=O)C(O)CN3CCCC3)C)C2)=O)CCOCC1 10466,C(=O)(CCCS(C)(=O)=O)NC1CC(NC(c2ccnn(C)c2=O)=O)C12CCC2 10467,C=CC1(O)CCN(C(=O)C(C)N(C(c2cc(O)cs2)=O)CC)C1 10468,c1(C(=O)NCC2CCN(C(c3c(C)csc3)=O)C23CC3)c2c(nn1C)CCSC2 10469,c1(C(=O)NC(CCCC)CNC(=O)C(O)c2cnc[nH]2)ccc([N+](=O)[O-])o1 10470,Cc1cc(C(=O)NC2CC(NC(=O)CC3CSC3)C23CCC3)cc(Cl)c1 10471,C1(C(=O)NCC(CNC(C2(CSC)CCC2)=O)CO)CCC(C)(C)C1 10472,C1(C(=O)NC2C3CN(C(c4nc(CCC)sc4)=O)CC32)CCc2nnnn2C1 10473,Cc1cc(=NCC(C)CNC(c2c(F)ccnc2F)=O)[nH]c(C2CC2)n1 10474,C(=O)(C(C)S(=O)(=O)CCC)NCC(CC=C)NC(c1nc2cc(F)ccc2s1)=O 10475,N1(C(c2cccs2)=O)CC=CC(NC(C2CCCN2S(=O)(=O)CC2CCC2)=O)C1 10476,C1(C(=O)NC(C2(C(N3C(C)CC(CO)C3)=O)CC2)=O)(CN(C)C)CC2(CCC2)C1 10477,Cc1nc(C2CC2)ncc1C(N1CCC(CNC(=O)CC2CCCO2)C1(C)C)=O 10478,C#Cc1cnc(C(N2CCOCCC2C(=O)NCC(C2CCC2)OC)=O)c(C)c1 10479,C1(CC(=O)NC2CN(C(=O)CCc3nncs3)C2)COC(=O)C1 10480,C(c1ccc(SC)o1)=CC(=O)NC1(C2NCCC2)CC1.C(CC)(C=O)=CCCC 10481,C(=O)(C1=CCC(C)CC1)N1CCC(C(C)NC(=O)Cn2cnnc2O)C1 10482,c1(N2CCC(NC(CCOc3c(C)ccc(C)c3)=O)C2)nc2cccnc2s1 10483,c1(OC)cncc(C=CCC(=O)Nc2ncccc2C(F)C(F)(F)F)c1 10484,C(=O)(CC(O)CNC(=O)CNc1nc[nH]n1)N(CC(C)(C)C)C 10485,c1(CC)cccc(F)c1C(N1CCCOC(CCNC(=O)C2=CCCC2)C1)=O 10486,c1(C(N(CCN(C)C(c2csc(C3CC3)n2)=O)C)=O)c(N)ccc(F)c1F 10487,c1(C(N(C(C)CNC(=O)C=C2CC2)C)=O)cc(F)c(F)c(O)c1F 10488,C(CCC(C)(C)C(=O)Nc1ccc2c(c1)OCO2)N(C)C 10489,Cc1ccc(C#N)c(C(N2CCC(CN3CC(C)OC(C)C3)CC2)=O)c1 10490,N1(C(C2N(CC)CC2)=O)CC2(CC2)CC1CNC(c1ccccc1COC)=O 10491,Cc1cc(C(=O)N(C2CCN(C(c3c(C)[nH]c(C)c3C)=O)C2)C)ncc1Br 10492,C1(NC(CC(C)(C)NC(CCOCC(C)C)=O)=O)CCCCC1(C)O 10493,N1(C(CC2CCC(C)(C)O2)=O)CCCC2CN(C(=O)Cc3csc(Cl)c3)CCC12 10494,c1(C(N(CCN(CCOC2CCC(CC)CC2)C)C)=O)cc(C)nc(C)n1 10495,N1(C(c2cccc(NC(C)=O)c2)=O)CC2CC(NC(c3scnc3C)=O)C1C2 10496,CCCCC(C(=O)N1CCC(CCO)CC1)NC(c1cn(C)nc1OC)=O 10497,C1(C(N2CC3C(NC(c4ccc[n+]([O-])c4)=O)C3C2)=O)COc2ccc(O)cc2O1 10498,Cn1cnc2[nH]c(=NCC3CCCN(C(=O)CSCC(F)(F)F)C3)nc(O)c12 10499,C(=O)(CCC(O)C(C)(C)C)N1CCC(CCNC(CNC(CN(C)C)=O)=O)CC1 10500,N1(C(c2c(CNC(CC=CC=C)=O)ccs2)=O)CC2CCC(CO)(C2)C1 10501,c1(OC)ccc(C(=O)NCC(CONC2(c3ccccc3)CC(C)C2)O)cc1 10502,c1(C2CCN(C(=O)Nc3ccc(-c4onc(C)n4)nc3)C2)ccc(Cl)c(F)c1 10503,Cn1cc(CC(N2CCCC2C(C)(C)NC(c2cc(C(F)F)[nH]n2)=O)=O)cn1 10504,CCCC(CN=c1cccc(S(=O)(=O)NC2CCc3ncsc3C2)[nH]1)OC 10505,C1(C)(C(=O)NC(CN(C(C2(CSC)CCC2)=O)C)C)CCC(=O)N(C)C1 10506,CCC(CC(F)(F)F)N=c1[nH]c(=NC(C)CC(C)(C)OC)[nH]c2ccsc12 10507,C1(C(=O)NCCOCCCNC(C(C)C2=CCCC2)=O)CCC2(CC1)CC2(F)F 10508,C1(Nc2ccc(-c3nc(C)on3)cc2)CCCC12CCOCC2 10509,CC(C)C(C#N)C(=O)NC(C1CCCCC1)CNC(=O)Cc1cnoc1 10510,CC(CO)C(=O)NCCOCCCN(C)C(c1cnn(C)c1)=O 10511,C(C(CC(C)C)C(=O)N1CCC(N=[N+]=[N-])C1)NCCSCCOCC 10512,C(CCCC(=O)NCC(C)(C)CN(C(=O)CCS(C)=O)C)N(C)C 10513,n1(CC(N2C(C)CCC(NC(CC(=C)C)=O)C2)=O)c(=O)nc(O)c2ccccc12 10514,c1(OC)c(F)cc(F)c(C(=O)Nc2c[nH]nc2C(N2CCN(C)C(C)C2)=O)c1F 10515,c1(C(N2CCC(OCc3ccccc3)C2)C(=O)NCC)cc(Cl)nn1C 10516,c1(CC)nocc1C(=O)N(C)CC1CCCC1NC(=O)CC1CNC(=O)O1 10517,c1(C(N(CC=C)CC=C)=O)ccc(C(c2ccc(C(F)(F)F)cc2)=O)cc1 10518,c1(C(N2CC(NC(C3C(CC(C)C)C3)=O)C(C)C2)=O)ccc(=O)n2c1CCC2 10519,N1(c2c(C)c(NCc3ccc(N)cn3)ncn2)CCC(C2CCCCC2)C1 10520,C1(CC(=O)NC(Cc2cc(C)[nH]n2)C)CN(C(c2ccccc2O)=O)CCC1C 10521,Cc1ccccc1C(F)(F)C(=O)OC(CCN1CCN(C)CC1)C(N)=O 10522,c1(CCNC(NCC(C2CCCCC2)OC)=NCCF)nnc2c(=O)[nH]ccn12 10523,c1(C(N2CCCC2C2CCCC2)C(=O)NCCCOC)ccc(C)c(OCC)n1 10524,CC1CN(C(C2CC23CC(C)(C)C3)=O)CCC1NC(C1CC2(CCCO2)C1)=O 10525,CC1CC=C(C(=O)NCC(C)(CO)NC(=O)CN2CSCC2=O)CC1 10526,c1(OC)nc(CNC2(c3c(F)cccc3F)CCCCC2=O)ncc1F 10527,N1(C(c2nc(C)n(C)c2C)=O)CC2CCCC2(NC(C2CCCC(=O)N2)=O)C1 10528,N1(C(CCOC)=O)CC(NC(=O)C=C(C)Cl)CC12CCC2 10529,c1(OC)ncc(NC(C2(F)CCN(Cc3cc(O)ncc3Br)CC2)=O)cc1F 10530,C1(CNC(Cc2cc(C)[nH]n2)=O)(NC(C2CCSC2)=O)CCCCC1 10531,CC(=NO)C1CC(C(=O)NCC2CCN(C(=O)CCSC(F)(F)F)CC2)C1(C)C 10532,c1(C(=O)NCC2CCCN(C(Cc3c(C)n[nH]c3C)=O)C2)ccc(Br)c(O)c1Br 10533,N1(C(c2c(C)cc[nH]2)=O)CCC2(CC1)CC2CNC(c1cnc(S)[nH]1)=O 10534,c1(C(N2CC(NC(=O)C(F)=C3CCCC3)CC(C)C2)=O)cncc(P(C)(C)=O)c1 10535,N1(C(C(C2CCC2)OC)=O)CCOCCC1C(=O)NCC1(c2ccccc2)CC1 10536,N1(C(C2CCCC(OC)C2)=O)CCCC(NC(c2cc(Cl)cnn2)=O)C1C 10537,C(C)(CN=c1[nH]cncc1C)NC(C(c1ccc(C)cc1)C)=O 10538,c1(C(=O)NCCC(C)NC(c2c(C3CC3)cccc2F)=O)cn2cccnc2n1 10539,C(=O)(C(O)CCS(C)=O)N(CCC)CCNC(c1ncc(F)cc1N)=O 10540,C(C(=O)NCCN(C(C1CCC12CCC2)=O)C(C)C)(C(F)(F)F)OC(C)=O 10541,C#CCC(O)C(=O)N1CC(C(=O)NCCCCC2CC2)C(F)C1 10542,N1(S(CCCC)(=O)=O)CCC(COC)(NC(c2cc(Cl)ccn2)=O)CC1 10543,C1(C(=O)NCC2(CCNC(=O)C3=CCCSC3)CC2)CCc2ccccc2O1 10544,C1(C(=O)OC)CC(C(=O)NC(C)CCNC(C23COCC(C2)C3)=O)C1(C)C 10545,C#Cc1ccc(CC(=O)NCC(CNC(=O)CC(C)(F)F)S(C)(=O)=O)cc1 10546,c1(C(N2C(C(C)NC(c3c(C)nc(C)o3)=O)CCC2)=O)ccc(C)c(Cl)c1 10547,N1(C(C2(C(=O)OC)COC2)=O)CCN(C(=O)CCP(C)(C)=O)CC(O)C1 10548,N1(C(c2ccc(CC)o2)=O)CCC(O)(CC(=O)NCC(c2ccncc2)C)CC1 10549,C1(OCC)COCCC1CC(=O)N(CC(C1CC1)N(C(=O)COCCSC)C)C 10550,Cn1cc2cccc(CN3CCN(CC(=O)Nc4cccc(Br)c4O)CC3)c2n1 10551,CN1CCC(CN(C=O)Cc2cnn(C3CC3(F)F)c2)CC1 10552,CC(C)CC(CNC(c1ccc(Cl)o1)=O)NC(=O)C(C)OCC(F)(F)F 10553,CCC(C)(C)C(O)C(=O)N1CC(C(=O)NCc2nocc2C)C(C2CC2)C1 10554,C1(C)(C(=O)NC(CN(C(c2cc(OCC)n[nH]2)=O)C)C)CC(OCC)CN1C 10555,c1(OC)ccc(F)cc1C(=O)Oc1ncc(CCSC)s1 10556,N1(C(CC(COC)NC(C2(C#N)CCCC2)=O)=O)CC(O)CC(O)C1 10557,N1(C(C2(OC)CCOCC2)=O)CC(=O)NCC1NC(C12CCC(CC1)C2)=O 10558,N1(C(Cc2cc(CC)no2)=O)CCCC(CO)(Nc2nc(C(C)C)ncc2Br)C1 10559,C1(NC(C2C=CCN(C(c3n(C)c(=O)ccc3)=O)C2)=O)CC2(CCCCC2)C1 10560,c1(C(N2CCN(C(=O)Cc3ccc(O)cn3)C3C2C3)=O)cc(Cl)c(Cl)cc1Cl 10561,CCC(CC)C(C)C(=O)N1CC(C)(CNC(c2c(C)cccc2C)=O)CC1(C)C 10562,N1(C(Cc2ccc(OCCCOC)cc2Br)=O)CC2(CCCN2C(C)=O)C1 10563,c1(CNC(=O)C(N2CCOC(C3CCC3)C2)c2ncco2)c(Cl)cc(F)cc1Cl 10564,N1(C(C=Cc2ccc(OC)cc2)=O)C2CCC1CN(C(c1cnncc1C)=O)C2 10565,N1(C(c2c[nH]c(=N)s2)=O)CCCC2C(NC(c3ccc(C4CCC4)cc3)=O)C12 10566,C=CCCCC(C(=O)N1CC(F)C(F)C1)NC(C1CC2CCC2C1)=O 10567,N1(C(C2(F)CC2)=O)CCCC2(CCC(NC(C3(C4CC4)CC3)=O)C2)C1 10568,N1(CCCCNC(C(C(C)C)OC)=O)CCCN(C(c2csc(C)c2)=O)CC1 10569,C(=O)(C(C(C)O)N(C)C)NCC1(NC(C2OCC(C(=O)OC)C2)=O)CC1 10570,C1(C(N(CC#C)CC)=O)CN(C(=O)C(C)(C)CCF)CCN1C 10571,c1(C(N2C(CCNC(C3(N(C)C)CC3)=O)CSCC2)=O)cccc2cnccc12 10572,c1(CNC(C2N(C(Cc3nc(C)on3)=O)CC(C)C2)=O)cc(F)cnc1Cl 10573,Cc1cc(S(C)(=N)=O)cnc1N1CCOCC(C)(C)CC1 10574,C1(C(=O)NC2(C)CC(=C)C2)CCCN(C(=O)C(C)c2ccco2)C1 10575,C(=O)(CC(C)C(F)F)N(CCN(C(CC1N(CC)CCC1)=O)C)C(C)C 10576,C1(C(N2C(CC)CN(C(c3c(Cl)n[nH]c3C)=O)CC2)=O)CCCCCC1(F)F 10577,N1(C(CC)=O)CCOCC(NC(C2C(C)CCN2C(=O)OC(C)(C)C)=O)C1 10578,CN1CCN(C(C2CC3(CCC3)CO2)=O)C(C(=O)NCCC#CCO)C1 10579,C1(NC(c2cnc(C)nc2)=O)CC12CCN(C(=O)CC(C)CF)CC2 10580,c1(C(N2CCC(NC(CC(C)n3cccn3)=O)C2C)=O)[nH]cc2c1CCCC2 10581,CCCCCC(C)CC(=O)NCCC1CCN(C(C2CN(C)CC(C)O2)=O)CC1 10582,CC1CCCC(CC(=O)NCCOC2CN(C(=O)C(C)Cn3ccnc3)C2)C1 10583,c1(C(=O)NCC2C(NC(C3(SC)CC3)=O)CCCC2)c(Br)cc(F)c(F)c1F 10584,N1(C(C(c2scc(C)n2)C)=O)CC2(CCN(C(c3cccc4sccc34)=O)C2)C1 10585,c1(C(=O)NC2(CNC(C(CCOC)OC)=O)CCOCC2)ncc(N)nc1C 10586,C1(C(=O)NCCCCCCN(C(CCCCC=C)=O)C)Cc2ccc(F)cc2C1 10587,C#CC1(C(=O)N(C)CC2CC2(F)F)CCN(C(=O)CS(=O)(=O)CC)CC1 10588,c1(C(=O)NCCC2(NC(c3coc(C(F)(F)F)n3)=O)CC2)ccc2ncnn2c1 10589,CC1C(C)N(C(c2cccnc2CNC(=O)Cn2cc(CO)nn2)=O)CCN1C 10590,N#Cc1ccccc1OCC(N1CCC(CCNC(c2csnc2Cl)=O)CC1)=O 10591,c1(C(=O)NC(c2nn[nH]n2)Cc2c(F)cccc2F)c(O)nnc2c1CCC2 10592,CC(C)CC(CNC(C12CC(F)(C1)C2)=O)C(=O)NC(C)CS(C)(=O)=O 10593,Cc1cc(CN(C(=O)COC2CN(C(C3CCC(C)C3)=O)C2)CC(C)C)on1 10594,CC1CN(C(=O)CSc2nncs2)CC(C)N(C(C2(O)CCOCC2)=O)C1 10595,N1(C(Cc2cc(C)on2)=O)CC(NC(=O)Cn2ccc(C3CC3)n2)CC1CO 10596,N1(C(C(COCC)C)=O)CCCCC(NC(c2cscc2Cl)=O)C1 10597,n1(CC)nc(C)c(C(N2CC(N3CCN(C(c4cnn(C)n4)=O)CC3)C2)=O)c1Cl 10598,c1(OC)cc(CCNC(=O)C(C)Oc2ccc(F)cc2)cc(OC)c1O 10599,C1(C(N2C(C(C)NC(=O)C=C3CCN(C)CC3)CCCC2)=O)CC12CCCCC2 10600,Cc1ccc(S(=O)(=O)NC2(CCc3ccnc(Cl)c3)CCCCC2)cc1 10601,c1(NC(C2CCC(NC(COCC)=O)CC2)=O)cc2nccc(C(F)F)n2n1 10602,Cc1cc(C)c(C(=O)NC(c2ccc(F)cc2)CNC(=O)C(CO)N(C)C)o1 10603,c1(NCC(C)C)nnccc1C(=O)N(C)CC1(CO)CC1.N1(CC=O)CCC(C)C1 10604,c1(C(=O)NCC(CCNC(=O)C(C)n2ccnn2)OC)cc2ccncc2[nH]1 10605,C1(C(=O)NCC2(O)CCN(C(=O)CN3CCC(CO)CC3)C2)CC12CC(F)(F)C2 10606,N1(C(CC(C)SC)=O)CC(NC(c2cccc(C3(F)CC3)c2)=O)C(C)C1 10607,CC(C)(C)C#CC(=O)N1CCN(C(=O)C(=C2CCCCC2)F)C(CO)C1 10608,C1(C(N(C)CC2CCCN2C(=O)CC2CC3C=CC2O3)=O)NC(=O)C2CC12 10609,Cc1nc(C2CC2)[nH]c1C(N1CCC(NC(C2SCCCS2)=O)CC1)=O 10610,C1(CC(=O)NC2CC(NC(C3N(CCC)CCCC3)=O)C2)CCC(=O)NC1=O 10611,CCCCC(O)C(=O)NCCC1CSCCN1C(c1ncc(C(N)=O)cc1Cl)=O 10612,CC1(C)CCC(C(=O)NCCC2(C)CC2(F)F)CN1C(C1CCC(=O)O1)=O 10613,C1(NC(=O)COc2cccc(F)c2)CN(C(C2(CO)CCCO2)=O)CCC1F 10614,Cc1nc(C(C)NC(=O)C(C)NC(=O)C(O)C2CC2)c(C)o1 10615,c1(C(=O)NC(c2cccnc2)CN(C)C)c[nH]nc1C1CCOCC1 10616,N1(C(c2n(CCC)ncc2)C(=O)NC2CC2)CC(C(N)=O)C(C(N)=O)C1 10617,C1(C(N(C(C#C)C)CCCC)=O)CCC2(CC2)N1C(=O)CCc1ccccc1 10618,C(=O)(CCCCC(N)=O)N1C(CC(N2CCCC(C)C2)=O)C(C)(C)CC1 10619,c1(OC(CC)C(=O)NC(C)(C)CNC(=O)COCC2CCC2)cccc(C)c1 10620,C1(C2CCN(C(C3(F)CCOC3)=O)CC2)(NC(C(C)OCCC=C)=O)CC1 10621,c1(C(=O)NC2CC2)cc(C(C)NC(CCN(CCOCCOC)C)=O)no1 10622,c1(C(=O)NCCC2(NC(=O)CC3COCC3O)CC2)cc2c(s1)CCCCCC2 10623,c1(C(=O)NC2(CNC(C3CC(=C4CC4)C3)=O)CCCC2)ccc(Cl)cc1O 10624,C1(C2CN(C(C34CCCC3C4)=O)C2)(NC(CCCn2c(C)ncc2)=O)CC1 10625,C(=O)(C(CC)CC(C)C)NCc1cc(C(=O)NC(CCC(=C)C)C)on1 10626,c1(C(N2CCOC(=O)C2)=O)nn2ccccc2c1CNC(C1N(C)C(=O)OC1)=O 10627,C(=O)(CCN(CCO)C(c1cocn1)=O)NCCN(C)C 10628,C1(NC(c2c(CCC)cccc2)=O)COC2C(NC(=O)CC3CN(C)C3)COC12 10629,C1(C2CCOCC2)(c2onc(C)n2)CCN(C(c2cnc3snnc3c2)=O)C1 10630,Cc1ncnc(C(=O)NC(C)(C)CC(N2CCOC(C)CC2)=O)c1C 10631,c1(C(=O)NC(C)CN(C)C(c2cnn(C(C)(C)C)c2)=O)cnn2c1CN(C)CC2 10632,C1(C(=O)NC2C(C(=O)NCC(C)NC3CC3)CC2)CC=CC(O)C1 10633,c1(C(=O)NCC2(OC)CCOC2)oc(-c2ccccc2C)nc1C 10634,Cc1nc(C)c(CCC(=O)NC2C3CC2N(C(=O)CC2CC(C)(C)C2)C3)c(O)n1 10635,C(=O)(CCC1=NNC(=O)CC1)N1CC(N(C(=O)CCCC(F)F)C)C1 10636,N(C(=NCCNC(c1ccccc1Cl)=O)NC1CC1(c1ccccc1)C)C(C)C 10637,c1(C(C(=O)NCC(=C)CCNC(c2oncc2CC)=O)C)ccc(Cl)c(Cl)c1 10638,Cc1ccc(O)c(CC(=O)NC(C2CCCN(C(=O)CC#N)C2)C)c1 10639,c1(C(=O)NC(C)CCNC(c2c(C(F)F)cccc2F)=O)cc(C#N)ccc1Cl 10640,C1(C(=O)NC2CC(NC(c3cnc(SC)n3C)=O)C(O)C2)CCCCN1N=O 10641,c1(-c2nc(CNC(=O)NCCCc3ccnc(C)n3)on2)c(Cl)cccc1Cl 10642,CC1CN(C(c2cnc(NC3CC3)cn2)=O)CCN1C(=O)CS(N)(=O)=O 10643,C1(CNC(CCC#CC)=O)CC2(CC(NC(=O)C(c3cn(C)nc3C)C)C2)C1 10644,S(=O)(=O)(c1ccc(NCC(C)NC(C)=O)cc1Br)N(C(CC)C)C 10645,N1(C(c2n(C)ncc2)=O)C2CCC1CC(NC(C1(O)CC3(CCOCC3)C1)=O)C2 10646,n1(CC(C(=O)NCCN(CC)Cc2ccc(C)cc2)C)cnc2ccccc12 10647,c1(C(=O)NCC2CCN(C(c3ccc(C)cc3F)=O)C2)ccc(Br)c2cc[nH]c12 10648,S(=O)(=O)(c1occc1C)NC(c1c(C)ccc(C)c1)CCCC(=O)O 10649,C(=O)(C(CC)CC(C)C)Nc1cn(CCNC(COCCCCOCC)=O)nc1 10650,c1(C(N2CCC(NC(C3CC(=O)N3)=O)C23CCC3)=O)ccc2ccccc2c1 10651,C1(C(c2nnnn2C2CC2)(C)NCC23CC4CC(CC2C4)C3)CCOC2(CCC2)C1 10652,c1(C(N2CC3CC3C3CC23)C(=O)NCCCOC)ccc2c(c1)COC2 10653,c1(C(N(C2CC(NC(=O)C(=O)C(C)(C)C)C2)C)=O)cc(F)cc2ccoc12 10654,N1(C(CCC(C)NC(C2(C(C)(F)F)CC2)=O)=O)C(CO)CCC1C(C)(C)C 10655,c1(C(N2C(CCNC(CCC(=C)C)=O)CCC2)=O)c(OC)cnc2ccccc12 10656,c1(CNC(C(C2(O)CCC2)NC(c2cccnc2S)=O)=O)ccc(CO)nc1 10657,C(=O)(CCCCC(=O)NC1CCN(C(=O)CN2CCN(C)C(=O)C2)CC1C)OC 10658,C1(NC(CC(CCC)C)=O)CC2(CCCN(C(c3cnn(C)c3)=O)C2)C1 10659,C12(NC(c3cc(C)c(C)o3)=O)COCCC1CN(C(=O)Cc1[nH]cnc1C)C2 10660,c1(C(N2CCC(Cc3ccccc3Br)C2)=O)ccnc2ncnn12 10661,C=CCC(C)(C)C(=O)N1CCN(C(=O)C(C2CCC2)OC)C(C2CC2)C1 10662,N1(C(c2c(C)cc(F)s2)=O)CCC(C)(C)C1CC(=O)NCC#CC(F)(F)F 10663,CCC(C)(C#N)C(=O)N1CCC(NC(c2cccc(N(C)C)c2)=O)CC1 10664,c1(C(=O)NC(CCCC)CNC(=O)CCCCCO)ccc2c(c1)COC2 10665,Cc1oc(C(=O)NC2C3CC2N(C(=O)CCCN2CCCC2)C3)cc1S(C)(=O)=O 10666,N1(C(C(c2cccnc2)C)=O)CCC2(C1)CN(C(C1(F)CCCOC1)=O)C2 10667,C1(NC(N)=O)CCC(C(N2CCC2C(=O)NCC2(CO)CC2)=O)C1 10668,N1(C(Cc2c(C)ccs2)=O)CCCC2CN(C(=O)C=Cc3ccccc3)CCC12 10669,C12(NC(C3N(C(C)=O)CCC3)=O)CCN(C(c3ccoc3C3CC3)=O)CC1C2 10670,c1(C(=O)NCC2(CCNC(C(C)(C)OCC)=O)CC2)cc(C#N)no1 10671,c1(CN(C=O)CC2(OCC)CCOC2)ccccc1-n1nc(C)cc1C 10672,C1(n2cc(CCC(C)O)nn2)CON(C(=O)C(C)C(F)F)C1 10673,C1(NC(C(C)(C)NC(=O)OC)=O)CCN(C(=O)C(c2ccc(Cl)cc2)O)CC1O 10674,c1(C(CC(=O)NC(C)CNC(C2(C)CC2)=O)=O)cc(-c2ccccc2)no1 10675,Cc1oc([N+](=O)[O-])cc1C(=O)N(C1CCN(C(C2CC(F)C(=O)N2)=O)C1)CCO 10676,N1(C(=O)CCc2nc[nH]n2)C2CCC1C(F)C(NC(C1(CNC=O)CC1)=O)C2 10677,N1(C(Cn2cc(C(=O)OC)nn2)=O)CCCC2(CCN(C(=O)C(C)C3CC3)C2)C1 10678,C(=O)(N=c1[nH][nH]c(C)c1-c1ccccc1)c1c(C)ncs1.N12CC3OCC(C3C1)O2 10679,C(=O)(C(O)C(F)F)NCC(C)N(C)C(c1ccc(NC(C)C)nc1)=O.CCO 10680,c1(OCC)cnc(C(=O)NC(C2CCN(C(=O)C(F)C3CCCC3)C2)(C)C)cn1 10681,C1(NC(C23OCC(C)(C2)C3)=O)CCCC12CCN(C(=O)C(F)C(F)(F)C(F)(F)F)CC2 10682,CCCCCC(O)C(=O)N1CCCC1(C(=O)NCC1(CC)CCCC1)CC 10683,C=CCCC(C(=O)N1CC(C)(C)C1COC)NC(C1(C)CCC2CC2C1)=O 10684,c1(C(N2CC(CN(C(CCCC=C)=O)C)OCC2)=O)cc2ccc(Cl)c(F)c2[nH]1 10685,C1(NC(c2cc(C(F)F)ccn2)=O)CCN(C(C2C(Cl)(Cl)C23CC3)=O)CC1F 10686,c1(SC)nc(N(C)CC2CCN(C(c3cnc(C(N)=O)cn3)=O)CC2)ncc1C 10687,N1(C(c2cncc(C)n2)=O)CCC2CC(C1)CN(C(c1coc(C(N)=O)c1)=O)C2 10688,Cc1onc(C(=O)NCC2CCCC(NC(C3CC=CC3)=O)C2)c1[N+](=O)[O-] 10689,Cc1ccc(C)c(C(c2nnnn2C(C)C)NC2(C(=O)NCC3CCCC3)CC2)n1 10690,CN1CCCC(C)(C(=O)NCCC2(O)CCN(C(c3ccoc3Cl)=O)C2)C1 10691,C(=O)(CCN=C(N)NCC1CCC(C)CO1)CCCCl.c1(CN)ccc(Cl)cc1 10692,OCC(Cc1cccc(F)c1)CN=c1[nH]c2c(F)c(F)c(F)cc2s1 10693,c1(C(=O)NC2CC3CN(C(C(CC)SC)=O)CC32)nccn2ccnc12 10694,N1(C(C(Cn2cccn2)NC(CC2(C)CC2)=O)=O)CCCC(F)(F)CC1 10695,N(C(=NCCCCl)NCCCN1CCCC1=O)N(C1CCOCC1)C 10696,c1(OC)cc([N+](=O)[O-])ccc1CNC(=O)C=Cc1ccc(Cl)cc1F 10697,C(=O)(C(C)(C)CC#N)N1C(CN(C(=O)Cc2cnc[nH]2)C)COCC1 10698,C1(NC(CC=CC=C)=O)(CF)CCN(C(=O)CN2CCCNC2=O)C1 10699,CS(=O)c1ccccc1-c1cccc(CC(N2CCCC(CC3CC3)C2)=O)n1 10700,c1(OC(C)C)ncccc1C(=O)NCC1CCC(C2OCCO2)CC1 10701,C1(NC(N(C)CCc2ccncc2)=O)CCN2CCCCC12 10702,c1(C(N2CCC(NC(c3cncnc3)=O)CC2C2CC2)=O)cc([N+](=O)[O-])ccn1 10703,C=C1CC2(C1)CC(C(=O)NC1CCN(C(=O)C=Cc3cncs3)CC1C)C2 10704,C(=O)(C(C)(C)C1CCN(C(c2cnn(CC)c2)=O)C1)NC(c1ccccc1)CC 10705,C1(OC(C)C)CCN(CC(O)COc2ccc(C(N)=O)c(C)c2)C(C)C1 10706,C1(CNC(Cc2c(SCC)cccc2)=O)CN(C)CCN1C(=O)Cc1ccoc1 10707,C1(O)(CCNC(C(CC)OCC)=O)CCN(C(c2cnccc2Br)=O)C1 10708,c1(C(N2C3CC(CC(NC(c4n(C)ccc4)=O)C3)C2)=O)coc2cc(O)ccc12 10709,CC1CN(C(C2(O)CCSCC2)=O)CCC1CNC(=O)Cc1cnc[nH]1 10710,C(=O)(C1CCCc2ccnn21)N1CC(C2CN(C(CS(C)(=O)=O)=O)C2)C1 10711,Cc1nnc(CNC2CC(F)C2)n1C.N12CCCC(C1)CN(C)CC2=O 10712,C(=O)(C1=CCCN(C(=O)CNc2ccccn2)C1)NCC1N(CC)CCC1 10713,C1(NC(CCN(S(C)(=O)=O)C)=O)CC2CC1CN(C(c1ccncc1F)=O)C2 10714,C(=O)(CCCC(C)(C)C)NCC(CC=C)NC(=O)CCc1nnc(C(F)F)o1 10715,C#Cc1cn(C)nc1C(=O)NC1CCC(CC(N2CCCC2C)=O)C1 10716,CC1(F)CCCCN(C(=O)C(C)(C2CCC2)NC(c2cccnc2O)=O)C1 10717,C#CCCCCC(=O)NC1CCCCCC1NC(c1ccn2ccnc2n1)=O 10718,c1(CNC(c2n(CC(=O)OC)nnn2)c2ccns2)cc(F)c(F)cc1F 10719,N1(C(C2C(CC)C2)=O)CCCC2(C1)CN(C(c1ccc(N)cc1F)=O)C2 10720,c1(N(CC(=O)NCC2C(NC(CSc3cn(C)nc3)=O)C2)C)ccnc(Cl)n1 10721,Cc1cnn(CCCN(C(=O)CCCC2CC2C)C(C2CCC(C)C2)=O)c1 10722,CCC(C)CC(=O)NCCC(=O)Nc1ccc(C(F)C(F)(F)F)cc1 10723,C(=O)(C(O)CCC(F)(F)F)N1CC(CNC(c2c(C)cccn2)=O)N(C)CC1 10724,CCC(CC(C)C)C(=O)N1CCC(F)(CNC(=O)CC2CC(SC)C2)CC1 10725,C1(C)(COC)CC(NC(=O)Cc2cccs2)CN1C(=O)Cn1cnc([N+](=O)[O-])n1 10726,CC1OC2CCC1(NC(C1CC=CCN1C(C1CC(N(C)C)C1)=O)=O)C2 10727,C(CCN=c1[nH]c(=NCCC(C)F)[nH]c2c1COCC2)N(C(C)=O)C 10728,CCCC(CC)C(=O)N1CC(NC(c2cc(Cl)cc(Cl)c2)=O)CC(F)C1 10729,c1(NC(C(=O)NC(c2ccc(Br)s2)C)=O)ccc2ccnc(Cl)c2c1 10730,c1(C(N2C(CNC(c3cc(CCC)on3)=O)C=CC2)=O)n[nH]c2c1COC2 10731,N1(C(C(C(C)C)F)=O)CCCN(C(=O)COC(C)(C)C)C(c2ccccc2)C1 10732,C(CC(C)C)(C(=O)N1CC2CC(C1)C2NC(c1snnc1C)=O)NC(C)=O 10733,CCC(O)C(C)C(=O)NC1CCCN(CC(N2C(C(=O)OCC)CCC2)=O)C1=O 10734,C(=O)(C1=COCCO1)NCC(C(C)(C)C)NC(c1c(Cl)cncc1Cl)=O 10735,C1(NC(C=NOC)=O)CC2(CCCN(C(=O)C3=NOC(C(C)(C)C)C3)C2)C1 10736,N1(C(C2(NC(=O)C(F)C3CCCC3)C(C)(C)C2)=O)C2CCC1COC2 10737,N1(C(=O)Cc2cn[nH]c2)CC2CC(C1)N(C(C1CCCN(c3nccs3)C1)=O)C2 10738,C12(C(=O)NCCC3OCCN(C(C(CCSC)O)=O)C3)CCC(CC1)C2(C)C 10739,Cc1nc(N2CCC3CCC(C2)N3C(=O)C(C)n2ccnc2)c2cc[nH]c2n1 10740,C1(C(=O)NC(C2CCCCN2C(=O)CC2CCCSC2)C)(CC)CCOCC1 10741,N1(C(c2cnc(=N)[nH]c2)=O)CC2COCC(C1)C2NC(c1cc(CO)on1)=O 10742,C1(C(F)F)CC(=O)N1.C(C)(C)(CO)N.CCC(=O)C1CC1C(F)(F)F 10743,c1(CSCC(=O)N(C(CNC(CCC(=C)C)=O)C)C)nc2ccccc2[nH]1 10744,C1(N(C(C(COC)COC)=O)NC(C(C2CCCC2)OC)=O)CCc2nn[nH]c2C1 10745,C1(NC(=O)NCCS(=O)(=O)NC2CCCC2)CCCC1C1CCCC1 10746,c1(N2CC3C(CNC(C(C)Cc4ccco4)=O)C3C2)ncnc(Cl)c1Br 10747,C1(NC(C=C(CC)C)=O)CC2CCC1C1CN(C(=O)C(=CC3CCCC3)C)CC21 10748,N1(C(c2ccc(C)nc2C)C(=O)NCCC)CCCC(O)(C2CC2)C1 10749,C(c1ccc(C)cc1C)=CC(=O)NCC1(C)N(C(C2C(=C)C2)=O)CCC1 10750,N1(C(c2n(CC)cc(Cl)c2)=O)CCCN(C(=O)C(O)CC(F)(F)F)C(C)C1 10751,c1(C(=O)NCC2C(C)CCN2C(c2nnsc2N)=O)ccc(OC(F)F)cc1F 10752,C#CC1(C(=O)NC2CCN(C(C)=O)CC2)CCN(C(=O)Cc2cscn2)C1 10753,Cc1cc(=O)n(CCC(N2CCCC(N(C(=O)CC=C(Cl)Cl)C)CC2)=O)cn1 10754,C1(NC(C2CCSCC2)=O)CC(O)CN(C(c2ccc(CC3CCC3)cc2)=O)C1 10755,N1(C(C(CCOC)OC)=O)C2CC=C(C(=O)NCC(C3CC3)N(C)C)C1CC2 10756,c1(CC(=O)NC(CN2CCN(C(CCC#C)=O)CC2)C)c(F)cccc1Cl 10757,C(C(CC(C)C)C(=O)N1CCOC(CF)C1)OC.c12cc(nn1C)C(=O)N2 10758,S(=O)(=O)(c1ccc(N2CCOC(C)(C(C)(C)C)C2)c(Cl)c1)N(C)CC1CC1(C)C 10759,S(=O)(=O)(c1cc(C)c(CC(CS(CC)(=O)=O)(C)C)o1)N 10760,C1(CC)COCCN(C(=O)C(=O)NCCn2cc(C(C)(C)N(C)C)nn2)C1 10761,c1(C(N2CC(NC(C3(SC)CC3)=O)C(F)C2)=O)ccc2nc(O)[nH]c2n1 10762,C(CCN=c1[nH]c2c(c(=NCCN3CCOCC3C)[nH]1)COC2)OCC(C)C 10763,c1(CC)noc(C)c1C(=O)NC1(C2CCCCN2C(=O)Cc2csc(C)c2)CC1 10764,Cc1nc(N2CC3CC3(CNCc3ccncc3Cl)C2)c2c(n1)CCC2 10765,N1(C(CCCOCC=C)=O)CCN(C(=O)C(O)CC)C(CC(=O)NCC)C1 10766,C1(N(C(=O)CCCC2CCCC2)C)CN(C(C2CC(C)(C)O2)=O)CC12CC2 10767,N1(C(C=C(CCC)C)=O)CCCC(C)(CC(=O)NCc2cc(O)ccc2C)C1 10768,c1(C(=O)NCC(C)CNC(C23CC(C(F)F)(CO2)C3)=O)ncc2ccccn12 10769,C1(CNC(CC(=C)Br)=O)CCCC2(CCN(C(=O)C(C)CN(C)C)CC2)O1 10770,CCCCC(O)C(=O)NC(C1CCN(NC(c2ccccc2)C2CC2)CC1)=O 10771,N1(C(C(C)(C)NC(=O)NCC)=O)CCCC(CNC(=O)C(C)c2ccsc2)CC1 10772,c1(SC)c(C(=O)NC2(C)CN(C(c3ccc(C)nn3)=O)C2)cccc1F 10773,c1(C(N(CCCNC(CC(CC)C)=O)CCO)=O)ncnc2cc[nH]c12 10774,S(=O)(=O)(c1ccc(=NCCc2ccc(OC)c(C)c2)[nH]c1)N(CC=C)CCOC 10775,Cc1cnc(C(N2CCC(NC(C3CCC(C)O3)=O)C23CC3)=O)c(C)c1 10776,CC1=NNC(=O)C1CC(=O)NC(CNC(=O)C(C)c1ccco1)C(C)(C)C 10777,c1(C(=O)NCC(C)NC(c2cccc(C(C)=O)c2)=O)cccc2c(C)cccc12 10778,C(C1CN(C(c2cc(C)c(O)nn2)=O)CC1C(=O)NCCC(O)C1CC1)=CC 10779,c1(C(N(CCCNC(CNC(=O)OC)=O)C)=O)ccc(NC(=O)OC)cc1F 10780,c1(C(C)OCC)noc(CCC(=O)NC(C)(C)CNC(=O)CC23CC(C2)C3)n1 10781,C=CC1(C(=O)N(CC(N)=O)C)CCN(C(=O)CCC(=O)NCC)C1 10782,C=CC(C)(C)CC(=O)NC(C1CCN(C(=O)CCS(C)=O)C1)(C)C 10783,C1(C(C(=O)NC(CC)CNC(c2cccc(CO)n2)=O)O)CCS(=O)(=O)CC1 10784,c1(C(=O)NCCC(C)N(C(CN2C(C)CC2)=O)C)nn(C)cc1N 10785,C1(CC)CCN(C(=O)CC(C)(C)O)C1CNC(c1cc(C)ncn1)=O 10786,C1(CC(=O)NCCC(C)N(C(=O)CCN2CCOCC2)C)CC(F)CN1 10787,c1(COC(c2ccc(OC3CCOCC3)cc2)=O)cc2c(s1)CCOC2 10788,C1(OC)CN(C(=NCCCCl)NCc2ccc(CSC)cc2)CC1O 10789,Cc1c(C(=O)NC2CCC2NC(c2ncoc2C2CC2)=O)n[nH]c1C1CC1 10790,c1(C(C(N2CC(CC=C)(NC(C3CC(C)=NO3)=O)C2)=O)C)nc(F)ccc1Cl 10791,FC(F)C1=NOCC1Oc1ccccc1.c12cccc(c1)NS2 10792,c1(N(CC(=O)NCC(Cn2cc(C(C)OC)nn2)(C)C)C)ccc(Cl)cc1C#N 10793,C1(CNC(=O)CCCn2cccn2)CC2(CC2)CN1C(=O)CN1CCCC1CO 10794,C1(CC)C(NC(c2scnc2COC)=O)CCN1C(c1cnc(C(C)C)n1C)=O 10795,C(=O)(C1=CCCC1C)N1C(CO)CC(NC(c2n(CC)c(O)nc2)=O)C1 10796,C1(C(N2CC(C(C)NC(=O)CCSc3cccc(Cl)c3)C2)=O)CCCC2(CC2)C1 10797,C(=O)(CC(C)CC(C)(C)C)N1CC(NC(c2c(C)ccc(C)c2)=O)C(F)C1 10798,c1(C(=O)NC2C(CC(=O)NC(C#CCC)(C)C)CCC2)c(F)cncc1F 10799,c1(N2CCN(c3ccc(C)cc3C)CC2)ncnc2c(C)cc(Br)cc12 10800,S(=O)(=O)(c1ccc(Cl)cc1)CC(=O)NC(C)CCNC(=O)C(C)OC(C)(C)C 10801,C(=O)(CCN(OC)C(=O)c1coc2c1COC2)N1CC(COC)(OC)C1 10802,c1(C(=O)NCC2C(C)C(=O)CC2)nc(N(C)C)n(-c2ccccc2)c1Cl 10803,c1(COC)csc(C(C)(C)C)n1.C12(COC1)C(=O)NCC2 10804,C1(C(=O)NCCCC#C)CC(NC(c2cn(C)nc2OC)=O)CCO1 10805,c1(C(N2C(C(=O)OC(C)(C)C)C3(C2)CCC3)=O)ccc(F)c2[nH]ccc12 10806,Cc1cccc(OCC(=O)Nc2ccccc2CNC(=O)CC(C)(C)C#N)c1C 10807,c1(OC)c(Cl)ccc(C(=O)NC(C)(CNC(=O)C(C)CSC)C2CCC2)c1F 10808,c1(C(N(CCC(C)NC(c2cnoc2C2CC2)=O)C)=O)cc(F)cc2nn[nH]c12 10809,c1(C(=O)NCCC(C)NC(=O)C(F)(F)c2csc(Cl)c2)cn(C)nc1Cl 10810,Cc1c(C(=O)NCCC2CCCCN2C(C2CN(C)C(=O)N2)=O)cnn1C1CC1 10811,C1(C)(C(=O)NCc2c(CNC(CC3(C)CC3(Cl)Cl)=O)cccc2)COC(=O)OC1 10812,CC(C)(C)C(=O)N1CCCC1C(=O)NCCC1CCCN1C(=O)Cc1cccs1 10813,C(CC(C(=O)NC(c1ncc(F)cn1)C)NC(c1ccoc1Cl)=O)=CC 10814,N1(C(C2(OCC)CCCOC2)=O)CCC(C2(O)COC2)CC1 10815,C1(CNC(c2cc(OC)ns2)=O)CN(C(C2(c3cc[nH]n3)CC2)=O)CCN1 10816,C1(CNC(CCCOC(C)C)=O)CC(C)(C)CN1C(=O)CC1(O)CCCOC1 10817,C1(C(C)C)CN(C(C2CC2(C)C(F)F)=O)CC1C(=O)N(C)Cc1cnn[nH]1 10818,N1(C(c2scc(C)c2)=O)CCC(NC(c2cnc(C3CC3)s2)=O)CC1C1CC1 10819,C1(NC(CC=CCC)=O)CC(O)CN(C(=O)C(=O)Nc2ccccc2)C1 10820,N(C1CCSc2ccc(Br)cc21)C(N1C(COC)COCC1)=O 10821,c1(C(=O)NC2(CO)CCC(NC(C3(COC)CC3)=O)CC2)ccc(OC)c(O)c1 10822,CCCCC(C)CCC(=O)N(C1CC(C(=O)NCC(CC)SC)C1)C 10823,c1(C(=O)NCC2N(C(C)=O)CCC2C)cc([N+](=O)[O-])sn1 10824,CC1CC2CN(C(C3(c4ccc(F)cc4)CC3)=O)CC2N1C(=O)CCC(C)(F)F 10825,CC1CCN(C(=O)CC2COCCN2C(c2cc(Cl)cs2)=O)CC1CO 10826,C1(CNC(COCCOC)=O)CN(C)CCN1c1ncnc(Cl)c1Br 10827,C1(CC(=O)OCC)CCN(S(=O)(=O)NC(C2N(C)CCCC2(C)C)=O)CC1 10828,Cc1ccc(SCC(=O)N(C)CCN(C)C(C23CCC2(C(=O)O)C3)=O)cc1 10829,N#Cc1ccc(COCC(=O)OCCCOc2ncc[nH]2)cc1 10830,C1(NC(C=CS(CC)(=O)=O)=O)CCC2CCN(C(=O)C(=Cc3cnc[nH]3)C)C1C2 10831,C1(N(CCC)C(c2cc(C)co2)=O)CCN(C(=O)CSCC2CCCCO2)CC1 10832,C1(C(N2CC(C(C)OC)C2)=O)CC(C)(C)CCN1C(c1cccc(C)n1)=O 10833,Nc1c(C(=O)NC2CC(CCNC(=O)CN3CCCC3CO)C2)cc(F)cc1Cl 10834,c1(CC(C(=O)C(C(N2CCSCC2)C)=O)O)ccc(F)cc1.C1(N)CC(NC)C1 10835,c1(CN=[N+]=[N-])ccc(NC(=O)Cc2cc(F)cc(Br)c2)cc1F 10836,c1(OC)cc(C)cc(C(=O)NCC=CCNC(c2cnc(C)nc2CO)=O)c1N 10837,C(=O)(CN=S(C)(C)=O)NCC1C(NC(c2nc(CC)oc2)=O)C1 10838,Cc1cc(C(=O)NC(C)(CNC(C2CC2C(N)=O)=O)C(C)C)cc(C)c1C 10839,Cc1cc(C(=O)N(CC(=O)NCC2NC(=O)CC2(C)C)CC2CC2)ncc1F 10840,N1(C(C(CC)=CC)=O)CCC(C)C(NC(c2cc(Cl)cc(Cl)n2)=O)C1 10841,C1(CC(=O)OC)CC(C)(C)CN1C(=O)NC(C1(n2cccn2)CC1)C1CC1 10842,C1(NC(CCNC(N)=O)=O)CCCCC1NC(C1(CO)CC(F)(F)C1)=O 10843,C(=O)(C(=O)CCCC)N1CCC(N(C(CC=CC=C)=O)CC2CCCO2)CC1 10844,C1(N(C)C(c2ncoc2C2CC2)=O)CCCC(NC(=O)C=Cc2cncn2C)C1 10845,c1(NC2(CN(C)C)CCC2)nncc2sccc12 10846,C1(C(N(C2CC3(CCC3)C2)C)=O)CC2CC1CN(C(C1CC1C1(C)COC1)=O)C2 10847,C1(C(=O)OC)CCC2(CCC2)N(C(=O)CCC2CCOC2=O)C1 10848,CC1CN(C(C2CC=CCC2)=O)CC(C)N(C(c2ccc(N3CCC3)nc2)=O)C1 10849,C1(NC(C(C)C)=O)CC(C)CN(C(C2CCN2Cc2ccccc2)=O)C1 10850,c1(SC)nc(C(=O)NCC(F)CNC(=O)C(F)(F)C2(O)CCC2)c2ccccn12 10851,C(=O)(CS(=O)C(F)(F)F)N1CCC(CNC(CCOC)=O)C1(C)C 10852,Cc1cc(OCC(=O)NC2CC(NC(C3CCOC(=O)CC3)=O)C2)ccc1Cl 10853,C(=O)(CCC[N+](=O)[O-])N1CCC(C)(CNC(C(Cc2c(C)noc2C)C)=O)C1 10854,C1(CC(=O)NC(C(=O)NCC(C)C)c2cn[nH]c2)CC2C=CC1C2 10855,Cc1nn(C)c2c(N3CCOc4cc(Br)ccc4C3)nc(=NCC3CC3Cl)[nH]c12 10856,CN1CC(NC(=O)C(CO)NC(=O)CC=CC(C)(C)C)C(=O)N1 10857,c1(-c2nc(C3C(C)(C)CN(C(=O)C(C)(O)C(F)(F)F)C3)on2)ccc2c(c1)CCO2 10858,C1(NC(C(C)NC(=O)NCC)=O)C=CCN(C(c2cc(OCC)n[nH]2)=O)C1 10859,C1(n2cc(CNC(C(C)=C(C)C)=O)nn2)CCN(C(=O)CCc2cccs2)CC1 10860,C1(NC(=O)Cc2ccc(O)cn2)CCCCCCC1NC(=O)CCc1ncc[nH]1 10861,c1(CC(N2C(CNC(C(C(C)C)(C)O)=O)COCC2)=O)cccc2c1OCCO2 10862,N1(C(CC(=O)OCC)=O)CCC(CNC(=O)CCNC(=O)NC2CC2)C(C)C1 10863,N1(C(C(c2c(C)n[nH]c2C)C)=O)CCCN(C(c2cnns2)=O)C(C)C1 10864,C1(C(N2CC(CNC(=O)CSC)C(C(F)(F)F)C2)=O)(COC)CC=CCC1 10865,c1(OC)cc(CCC(=O)NC(C)CN(C)C(c2cc(C(F)(F)F)cs2)=O)on1 10866,Cc1ccsc1C=CC(N1CCC(OCCNC(=O)CC2CCCO2)C1)=O 10867,C12(C(N3CCC(C)(CCNC(c4ccccc4)=O)C3)=O)CC(C)(CCO1)C2 10868,CCC(C)CCC(=O)NCC1COCCN1C(c1cnc(-c2ccccc2)[nH]1)=O 10869,C1(C)(CNC(C(=O)NC(C)C)=O)CCC(NC(=O)C(c2ccccc2)=O)C1 10870,c1(C(=O)NCC2(F)CC(CNC(CN(CC(C)(C)C)C)=O)C2)cc(Cl)ccc1O 10871,C1(C(C)(C)NC(CCNC(COC)=O)=O)CCN(C(=O)CSCC(F)(F)F)C1 10872,Cc1cc(C(=O)NC2CN(C(c3ccc(I)c(C)c3)=O)CC2O)cc(C)c1 10873,C(CCCCC(=O)NCCc1cnc(C)s1)NC(C1(OC)CCC1)=O 10874,N1(C(C(C(C)C)F)=O)CC2CCCC(NC(c3csnc3Cl)=O)C2C1 10875,CC(C)CC(C)(C)C(=O)NCC(C(C)C(C)C)NC(C1(C(C)C)CC1)=O 10876,c1(CN2CC(C(N(CC)Cc3ccncc3)=O)SCC2)cnc(Cl)c(Cl)c1 10877,CCC(F)(F)CC(=O)N1C2CCC(C2)C1CNC(=O)C(C)Oc1ccccc1 10878,C1(C(N2CCC(NC(c3n(C)nnc3)=O)(CF)C2)=O)CCc2nccn2CC1 10879,c1(C(N(C2CCN(C(C3CC3c3ccco3)=O)C2)C)=O)ccc(F)c(F)c1O 10880,c1(CSC(C)C(=O)NCC(C2CC2)NC(=O)CCc2cnccn2)ccccn1 10881,C1(O)(C(N2CCCCC2CCCNC(C2(F)CC=CC2)=O)=O)CCOCC1 10882,c1(N(C)C)ncccc1C(N1CCC1NCC1CC(C(=O)OC(C)(C)C)C1)=O 10883,Cc1ccc(C)c(-c2ncc(C(=O)OCC(C3CC4CC4C3)=O)s2)c1 10884,c1(NC(C(CN(C(=O)CC2CCCS2(=O)=O)CC)SC)=O)ccc2nn[nH]c2n1 10885,N1(C(CC(C)F)=O)CCC(C)(C)CC1C(=O)NCc1cncc(C#N)c1 10886,C(c1ccccc1Cl)=C(C)C(=O)NC1CC(C)N(C(=O)CCn2ccc(=N)[nH]2)C1 10887,c1(C2(C(=O)NCC3C=CC(NC(c4ccsn4)=O)C3)CC2)cc(F)cc(Cl)c1 10888,S(=O)(=O)(c1cc2c(Br)cncc2s1)NCCC1CCN(C(C)=O)CC1 10889,C1(C)(CC)CC(C(=O)NCC2N(C(=O)C3=C(Cl)CC3)CCC2(C)C)CCO1 10890,C12CCN(CC1)C2=O.C1(NC(COCc2nnc(C)s2)=O)CC12CC(O)C2 10891,c1(-c2cc(CC)no2)cnc(N(C)Cc2cc(OC)ccc2OC)c(Cl)c1 10892,c1(OC)cnccc1-c1noc(C2(C3CC3)CC2)n1 10893,C(=O)(CCCCC(=O)N1CC(CNC(=O)CN2CCCCC2)CC1C)OC 10894,c1(C(=O)NCC(CCC)NC(=O)CCN(C)CCC)c(C)coc1CC 10895,c1(CC(=O)NCCOCCNC(=O)Cc2cncs2)ccc(F)cc1Br 10896,CC(C)C(C(=O)NCCC(C)N(C)C(C1CCC(=O)C1)=O)N(C)C 10897,N(C1COc2ccc(Cl)cc21)C1(c2n(CCSC)nnn2)CCC2CCC12 10898,c1(N2CC3CC(NC(c4csc(COC)c4)=O)C3C2)nc(C)nc2scc(C)c12 10899,c1(C(N2C(CC)CN(C(c3cc(Cl)n(C)n3)=O)CC2)=O)cccc2ccncc12 10900,c1(CNC(=O)C(=O)NCc2nc(C(F)(F)F)n[nH]2)cccc(I)c1 10901,C1(C(N2C(CNC(CN(C)CC)=O)CCCC2)=O)CNC(=O)CC12CCOC2 10902,N1(C(c2cnn(C)n2)=O)CCCC(CCC(N2CCCC2C(C)(C)CO)=O)CC1 10903,c1(OC)ccc(C(=O)O)cc1CN1CCC(O)C(C(=O)Nc2nc(C)co2)C1 10904,C12(CNC(c3n(CC)ncc3)=O)CC1CN(C(C1CC(C)(O)C1)=O)C2 10905,c1(CNC(=O)CC(=O)Nc2cc(F)c(F)cc2I)cc(Br)cc2[nH]ccc12 10906,Cc1nc2ccc(C(N3CCC4CN(S(=O)(=O)c5nccs5)CCC34)=O)cc2o1 10907,CCC(C)(COC)C(=O)N1CCN(C(=O)CC2CCC(C)(C)CO2)CC1 10908,C1(CC)(CC)CC(NC(c2cncc(CO)c2)=O)CN1C(C1CC=CC1)=O 10909,C1(CC#C)(C(N2CCCC2CC(=O)NC)=O)CCN(C(=O)C(COC)COC)C1 10910,c1(CC)ncc(C(=O)N(C)CC2CCCC2NC(c2cc(OC)ns2)=O)o1 10911,N1(C(c2c(C)nccc2Cl)=O)CCCC(NC(=O)C=Cc2ccsc2)C(F)C1 10912,N1(C(C(C)C2CCOC2)=O)CCC2CCC(C1)N2C(c1cc(=O)cc[nH]1)=O 10913,c1(CN2CC(NC(c3c(CC)nccc3)=O)C(F)(F)C2)cc(F)cc(F)c1OC 10914,N1(C(CC(=O)NCC#C)=O)CCC(C(=O)NCCCC(C)(C)O)C12CCC2 10915,N1(C(=O)CCc2cnco2)CC=CCC1C(N1CCSCC1C1CC1)=O 10916,N1(C(C2(C)COC2)=O)CCC2(C(=O)Nc3cncc(C(N)=O)c3)CCCC12 10917,c1(OC)ccc(C(=O)NCC(C)CNC(c2ccccc2C(C)=O)=O)cc1OC 10918,c1(CC(C)=O)ccc(CC(C)CO)cc1.CCC=CC#N 10919,CCCCC(F)C(=O)NC1CCCCC1C(N1CCC(CC(N)=O)C1)=O 10920,c1(-c2nnc(N3CCCC(C)(NC(=O)CCCCCF)C3)o2)noc2ccccc12 10921,c1(OC)ccncc1CCC(=O)N(C(C)Cn1cccn1)C(C)C 10922,Cc1cc(C(=O)NC2CC3CN(c4nccc(Cl)n4)CC3C2)cc2nn[nH]c12 10923,CCCC(C(=O)NC(C)CC(C)NC(c1nnn(CC)c1C)=O)NC(N)=O 10924,CN(C)S(=O)(=O)N(C)CC(c1ccco1)NC(N1CCC(N2CCNCC2)CC1)=O 10925,C(=O)(C(O)C1=CCCCC1)N1C(CNC(c2c(C)cnn2C(C)C)=O)CCC1 10926,c1(C(=O)NCC2C(NC(c3cccc(O)n3)=O)C2)cc(Br)ccc1[N+](=O)[O-] 10927,c1(C(N2CCC(O)(CNC(Cc3scc(C)n3)=O)C2)=O)ccc(C(N)=O)c(Cl)c1 10928,c1(C(=O)NC(C(C(C)C)C)CNC(c2ccn(C)n2)=O)cc2ccc(O)cc2[nH]1 10929,C1(CCNC(C2CN(C)C(=O)C2)=O)CN(C(c2cccc(Cl)c2F)=O)CCCO1 10930,c1(C(N2C(C3CCN(C(C(C)NC=O)=O)C3)CCC2)=O)cccc(=O)n1C 10931,n1(CCC)c(C(N2CCC(NC(=O)C(O)C(F)F)C23CC3)=O)cc2ccccc12 10932,c1(NC2C3(CC(OCC)C3)C2)nc(N(CC(C)C2CC2)C)nc2sccc12 10933,C1(C(N(CCSC2CC2)CC)=O)CCN(C(=O)C(O)Cc2ccc(Cl)cc2)CC1 10934,C(=O)(CC=CC(C)(C)C)NCC=CCNC(CC1(C)CC1)=O 10935,c1(C(=O)NC2(CC(=O)NCC(n3cccn3)C)CC2)ccc(=N)[nH]n1 10936,C(N=c1[nH]c(=NCC2CCCSCC2)[nH]c2c1CC(C)CC2)c1[nH]c(=NC)sc1 10937,C1(c2c(C(=O)NCC=C(C)C)c[nH]n2)CCCCN1C(=O)CC1(O)CCCCC1 10938,N1(C(CCOCC#C)=O)CC2CCC1CN2C(C1CCCC(C)CC1)=O 10939,S(=O)(=O)(c1ccc(NC(C)C(c2cccc(C)c2)OCC)cc1Cl)N(CC)CC 10940,C(=O)(CCCCC(N)=O)N1CCC(NC(c2c(C)ccc(OC)c2)=O)(CF)C1 10941,C(=O)(CCCC(C)(F)F)N1CC(N(C(=O)C=Cc2ccncn2)C)C(C)(C)C1 10942,c1(CC(=O)NC2CN(C(C(CC(C)C)C)=O)C2)c[nH]c2cccc(Br)c12 10943,c1(C(N2CC3CN(c4ncc(Cl)c(O)n4)CC3C2)=O)c(F)c(F)cc(F)c1F 10944,C(=O)(CP(C)(C)=O)NC1(CCNC(CCc2n(C)ncc2)=O)CCCC1 10945,c12nnc(-c3ccc(C)nc3)n1CCC(C)CCN2C.c1(O)ccccc1.CS 10946,c1(C(=O)NCCC2(C)CCN(C(c3nocc3Cl)=O)C2)cc2c(s1)CCC2 10947,N1(C(C2(COC)CC(=C)C2)=O)CC=C(C(=O)N2CCC(CC)C2)C1 10948,c1(CC)c(C(=O)NC(C)(CNC(=O)C(O)CC(C)C)CO)cccc1F 10949,C1(NC(C(CCCC)O)=O)Cc2ccccc2C1NC(C1(CC)CC1)=O 10950,C12(O)CCCN(C1)C(=O)CS2.CC(C(=O)N(C)NC(=O)OC(C)(C)C)=CC1CC1 10951,C1(C)(NC(C2(OC)CCN(C(c3cnn[nH]3)=O)C2)=O)CC2(CCC2)C1 10952,N1(C(C(C)(C)SC)=O)CCC2(CC1)COC(CNC(c1cc(=O)n(C)cn1)=O)C2 10953,c1(CCC(=O)NC2(CNC(C(C)C3CCOC3)=O)CCC2)nc(C(C)(C)C)no1 10954,N1(Cc2nn(C)c(OC(F)F)c2)CCC(NC(c2ccsn2)=O)C(O)C1 10955,c1(CC(=O)NCC(C)(C)CNC(C2C=CCC2)=O)cccc2nsnc12 10956,C(=O)(C1Cc2ccccc21)NC(CCC=C)C(=O)NC1(C)CC(N(C)C)C1 10957,Cc1nc(CC(=O)NC2CCC(CNC(C3CCC(=O)N3)=O)C2)co1 10958,N1(CC(=O)NCC2(NC(=O)CCCSC)CC2)CCc2sccc2C1 10959,c1(COC)nc(C)c(C(=O)NCCC(C(C)C)NC(c2n[nH]cc2C(C)C)=O)s1 10960,C1(C(=O)NCCn2nccn2)C2CCC1N(C(=O)CCn1ccc(Br)cc1=O)C2 10961,c1(CNCC2CCC(C)(CC)O2)c(F)cc(CO)cc1Br 10962,n1(CC)cc(C2CCC(NC(=O)N(C3(C)CC3)CCO)C2)cn1 10963,C1(C(=O)NC2(C)CC(NC(c3cc(Cl)ccc3Cl)=O)C2)CCC2(CCC2)O1 10964,c1(SC)ncc(C(F)(F)F)c(N(C(c2cc(C)cc(F)c2)=O)CC2CCNC2)n1 10965,S(=O)(=O)(c1ccc(N(C)CCOc2ccccc2)c(C#N)c1)NCCSCC=C 10966,N1(C(C(C)(C)NC(=O)NCCC)=O)CCC(CNC(C23CC(F)(C2)C3)=O)C(C)C1 10967,c1(C2CC2)ccc(F)nc1.C12CCCN1C2=O.C1(C(=O)NC)CN(C(N)=O)C1 10968,O=C(C#CC1CCCO1)N1CC2(CCN(C(C3(C(F)(F)F)CC=CCO3)=O)C2)C1 10969,Cc1noc(C)c1S(=O)(=O)N1CCOCC1C(=O)NC(C)C.C12CCN(CC1)C2 10970,c1(C(N2CC(n3cccn3)(CN)C2)=O)cc2c(nc1O)CCCC2O 10971,c1(C(=O)NC(CCN(C)C(c2ccsc2)=O)C(C)(C)C)c[nH]c2cc(F)ccc12 10972,c1(CNC2C(C(N3CCC(Br)CC3)=O)CCC2)c(F)ccc(Cl)c1F 10973,C#CC1CN(C(=O)C(c2ccnn2C)NC(=O)C=CCCC(C)C)CCN1C 10974,C(c1ccccc1Cl)=C(C)C(=O)NCC1(CNC(=O)CCCCN(C)C)CC1 10975,c1(CC(N2CC(CNC(C=CC=CC)=O)OCC2)=O)ccc(C)c(OC)c1 10976,C(C)(C)(CCCNC(=O)CO)n1cc(C(COC(C)C)C)nn1 10977,c1(C(N2C3C(NC(c4occc4F)=O)CC(C3)C2)=O)cccc2occc12 10978,C(=O)(CCCCCN=[N+]=[N-])N1CC(C)N(C(Cn2ccc(C)cc2=O)=O)C(C)C1 10979,C1(CNC(CC2N(C(C3CC(C(C)C)C3)=O)CC2)=O)CNC(=O)CO1 10980,c1(C(N2C(C)CC(CNC(=O)C3CC3)C2)=O)ccc(Cl)c(Br)c1 10981,C1(n2cc(OCCOCCOCC)nn2)C(C2CC2)CCN1C(=O)CCCOC 10982,c1(C(=O)NC(CC(C)NC(C(C)=C2CCC2)=O)C)c(C)nc(C(C)C)nc1S 10983,N1(C(C=CC=CCCCCC)=O)CCC2CCC(C1)N2C(=O)COCCCF 10984,C1(O)(CCC)CCN(C(C2CCCN(C(C3OCCCC3(C)C)=O)CC2)=O)CC1 10985,Cc1nccnc1CCNC(c1csc(-c2ccn(C)n2)n1)=O 10986,Cc1nnc2n1CC(C(N1CCC(CNC(C3CCCN3C3CC3)=O)C1)=O)C2 10987,N1(C(c2cnc(CC)[nH]2)=O)CC(CO)CC1CNC(=O)CCCNC(N)=O 10988,C(=O)(C#CC1CCOCC1)NCC(CCNC(c1c(CC)nc(C)o1)=O)(C)C 10989,N1(C(c2cn(CCN(C)C)nc2)=O)CCC2(CC1)CC2NC(c1cscc1F)=O 10990,c1(CC(C(=O)NC(C(C)NC(c2cnc(O)s2)=O)C)O)cccc(Cl)c1 10991,C(C)(C(=O)OC(C)(C)C)(C(=O)NC1CN(C(C2CC3CC3CC2C)=O)C1)OC 10992,c1(C(N(CCCCCNC(=O)C2=COCC2)C)=O)cnn2c1N(C)CC2 10993,c1(C(C(=O)N(C2CCN(C(C)C(=O)NC)CC2)CCC)(F)F)c(C)cccc1Br 10994,C1(C(N2CCC(O)(CCNC(CCc3nc(C)sc3)=O)C2)=O)CC12CC(C)(C)C2 10995,c1(C(=O)NC(C(=O)NCCCCCC)C2CCCO2)n[nH]c(C)c1Cl 10996,N1(C(CSCC)=O)CCC(CNC(C2CC2C2CC2C)=O)C12CC2 10997,C=CC(C)(C)CC(=O)NC1CC2C(NC(C3CCOC(=O)CC3)=O)C2C1 10998,c1(C(N2CC(C)(C(N(C3CN(C(C)C)C3)C)=O)C2)=O)cc2ccccn2n1 10999,N1(C(c2nc(C(C)=O)sc2)=O)CCC(C2CCN(C(=O)COCCO)C2)CC1 11000,c1(CCC(N2C(C)CCC(NC(C=C(C)Cl)=O)C2)=O)ccc2ocnc2c1 11001,c1(CC)ccc(C(=O)NC2CC23CC(NC(C2CC2C(N)=O)=O)C3)cc1CC 11002,N#Cc1cc2c(n(C(c3noc4c3CCCC4)CNc3csnn3)c1=O)CCC2 11003,C1(NC(CC(=O)OC)=O)C2CCCC1CC(NC(C1CN3CCN1CC3C)=O)C2 11004,N1(C(c2ncn(C)n2)=O)CCN(C(C2CCc3nnnn3C2)=O)C2CCC12 11005,C1(n2cc(-c3cn(C(C)(C)C)nc3)nn2)CCCN(C(C2CCC(=O)CC2)=O)C1 11006,c1(NC(C2N(Cc3c(C)noc3)CCC2)=O)cc(Br)ncc1F 11007,C1(c2n(C3(C)CC3)nnn2)(NC2CCCC(O)C2)CCN(c2ncccn2)CC1 11008,c1(N(C)C)ccc(C(=O)NC2(CNC(=O)CC3CC4CC4C3)CC2)nc1O 11009,C1(C(=O)NC2C(NC(c3cccc(C(F)F)c3)=O)COC2)CS(=O)(=O)CC12CC2 11010,C1(CN2CCC(CCCO)CC2)CC2(CCN1)CCOCC2 11011,Cc1c[nH]cc(C(N2CC(NC(=O)CSc3cn[nH]c3)CC(O)C2)=O)c1=O 11012,C1(C(=O)NC(C=C)CO)(CC)CCN(C(=O)CC2CCCCN2C)C1 11013,c1(CC)onc(C)c1C(N1CC(CC(C)NC(=O)Cn2c(C)ncc2)C1)=O 11014,CC1(NC(=O)CCc2nccs2)CCN(C(=O)C(F)CC2CC2)C1 11015,C#CC1(NC(N2CC(C(=O)NC)(CC)C2)=O)CCCCC1 11016,c1(CC)cnoc1C(=O)NCCN(C(c1cc(C(C)(F)F)n[nH]1)=O)CC 11017,c1(C(=O)NCC(CN(C)C(c2ccc(Cl)o2)=O)O)c(N)nn2ccccc12 11018,CC1(O)CCC(CC(=O)NCCNC(c2n[nH]c(C3CC3)c2Cl)=O)CC1 11019,c1(OC)cccc(S(=O)(=O)N2CC3CC2C3C(N2CCN(C)C(=O)C2C)=O)c1 11020,N(C1CCc2c(F)cc(Br)cc21)Cc1nc2ccc(C)cc2[nH]1 11021,c1(CN(C)C)cc(C(=O)NC2CCC(CNC(=O)C(F)CC3CC3)CC2)ccn1 11022,C(CCCC(=O)NCCCCCn1cc(CCN2CCCNCC2)nn1)N(C)C 11023,C1(CNC(c2ccc(SCC)cc2)=O)CC(F)(F)CN1C(=O)C(C)S(N)(=O)=O 11024,C1(C(=O)NCC2CC3CCC(C2)S3)C2CCCCCCC12 11025,Cc1cccc(Cl)c1C(=O)NC1CC(NC(=O)CCC2CCCCC2)C(O)C1 11026,C1(C(N2CCC(C)(O)CC2)=O)CC2(CCC2)CN1C(=O)CSCC(F)F 11027,c1(C(=O)NC2(CO)CCCN(C(C(CCC)(C)C)=O)C2)nc2cc(C)ccc2o1 11028,C1(N(C(c2cccn2CC)=O)CC)CCCN(C(C2CCC2(F)F)=O)CC1 11029,C1(C(=O)NC2(C)CCCN(C(c3cc(O)cc(=O)o3)=O)C2)CCC(C2CC2)CC1 11030,c1(C(CCC(=O)NCc2cnn(C3CCCCC3)c2)O)ccc(Cl)c(Cl)c1 11031,CN1CC=C(CC(=O)N(C)CCOCCNC(C2CC3CCC(C2)S3)=O)CC1 11032,C12(c3onc(C)n3)CCC(CC1)N2C(=O)C(c1cccc(O)c1)C 11033,c1(C(N2CC(N(C)C(C3CC(n4cnnc4)C3)=O)C2)=O)cnc(CC(C)(C)C)s1 11034,c1(C(=O)OCC2(F)CCCN(CCCCCC)C2)cnc2[nH]c(C)nc2c1 11035,C1(C(=O)NC2(CN(CC)CC)CC2)COCCN(C(=O)C=Cc2ccnn2C)C1 11036,c1(CC(C2(C)COCCN2C(C(n2cccnc2=O)C)=O)O)ccc2c(c1)C(=O)NC2 11037,O=C1CCc2cc(C(N3CC(N4CCCC4=O)C3)=O)c(F)cc2N1 11038,c1(OCCC(COC)OC)nc2ccccc2nc1N1CCCC(F)(CO)C1 11039,c1(CC)ncccc1C(=O)NCC=CCC(N1CCCC2CC12)=O 11040,C1(C(N(CC(=C)C)CC)=O)CC=CCN1C(c1csc(C)c1)=O 11041,C12(NC(=O)Cc3sccc3Cl)CCC(CN(C(c3coc(Br)c3)=O)C1)C2 11042,c1(NC(C(N2C(CCn3ncc(C)c3)CCC2)=O)=O)nc(C)n(C)c1C 11043,Cc1cc(Cc2[nH]c(C)nc2C)c(O)nn1.c12ncoc1C1CN(C1)C(=O)N2 11044,CC(C)C(C)(CNC(C1CCCC(C)O1)=O)NC(=O)CO 11045,C1(C)(CNC(C2CCC(CC)O2)=O)CCCN1C(=O)CCc1ccccc1Cl 11046,C1(CNC(C(CC=CC)C)=O)CC2CCCCC2N1C(=O)CCSC(F)(F)F 11047,C1(CNC(C(C=CC)O)=O)CC(C)(C)CN1C(=O)Cn1cc(C(=O)OCC)nn1 11048,c1(C(=O)NC(C#C)CC2CCOC2)ccc(-c2ccc(Br)cc2)n1C 11049,C(=O)(C1Cc2ccc(Cl)cc21)NCC1C2(CC(NC(CSCC(=O)OC)=O)C2)C1 11050,C(c1ccc(Cl)cc1)=CC(=O)NCC1CC(OC)CN1C(=O)CCc1cnoc1 11051,Cc1nc(CN(CC(N2CCC(CCCC3CCCO3)C2)=O)C)cs1 11052,Cc1cc(Cl)c(Cl)cc1C(=O)NC1CCCCC1NC(=O)C(C)(C)F 11053,S(=O)(=O)(c1cccnc1NC1CCN(C)C1)NCc1ccc(C(CC)C)cc1 11054,N1(C(C(C)=C2CC2)=O)CC=CC1C(=O)NC.C1=CCN(CC)CC2(CC2)CNC1=O 11055,c1(C(C)=O)cc(COC(c2ccc(C(F)(F)F)nc2)=O)c(C)o1 11056,c1(C(=O)CNC(c2cccs2)=O)cc(Cl)ccc1OCC1CCCO1 11057,C1(C)(NC(C(CCN(C)C)NC(c2coc(CO)c2)=O)=O)CC2CCC1C2 11058,c1(OC)ncc(C)c(C(N2CCC(NC(c3ccncc3Cl)=O)C(O)C2)=O)c1Cl 11059,C(=O)(CCCN(C)N=O)N1CCC(C)C1CNC(c1cnn(-c2nccs2)c1)=O 11060,N1(C(C(CC)=CC)=O)CCC(N=[N+]=[N-])(C(N2CC(n3cccn3)C2)=O)C1 11061,N(C1CCOc2c(F)cccc21)C(=O)Nc1ccc(S(=O)(=O)CF)cc1 11062,N1(C(c2c(C)[nH]nc2I)=O)CCOC2(CCN(C(=O)C(N)=O)C2)C1 11063,N1(C(CCCC#N)=O)CCN(C(C2CCCS2(=O)=O)=O)CC1CS(=O)(=O)F 11064,C#CCC(C)(C(=O)N1CCN(CC#C)C(=O)C1)NC(=O)CCCCCF 11065,C1(C(N(C2CCOCC2)C)=O)CC2C=CC1N(C(=O)CC(=O)OC(C)(C)C)C2 11066,CC1(C)C(NC(C2CCOCC2)=O)CC1CNC(C1(CC(=O)OC2CC2)CCC1)=O 11067,c1(C(=O)NC2C(CNC(C(COC)N(C)C)=O)CC2)cnn2ccn(C)c12 11068,N1(C(C(C)(C)OCC)=O)C2CCCC1CN(C(c1ccc(C)c(C)c1)=O)C2 11069,CCC(C(=O)N(CC(=O)NCC1(CCO)CN(C)C1)C1CC1)N(C)C 11070,N1(C(CSCCCC)=O)CCC(C(C)(C)NC(=O)CCC2CCC(C)O2)CC1 11071,n1(CC)nc(C(N2CCCC2CC(=O)NC2CCC(O)CC2)=O)c(C)n1 11072,C(=O)(C1=CCCSC1)NC1C(CNC(c2ccc(CNC(C)=O)cc2)=O)CCCC1 11073,C(=O)(CCC(=O)N(CC)CC)N1CC(OCC)(CO)C1.C1(CC(=O)N)CCCN1C 11074,N1(C(CC(CNC(=O)CN(CCCN=[N+]=[N-])C)OC)=O)CCN(C)CC1C 11075,C(=O)(C#CC(C)(C)O)N1CCCC(NC(C(CC)(C)C)=O)C1 11076,C12(C(N3C(CC)CC(C)C3)=O)COCC1CN(C(C1CC1(C)C)=O)C2 11077,C(=O)(C(O)CC(C)C)NC1(CCNC(CNC(CCC(C)C)=O)=O)CCC1 11078,c1(C2N(c3nnc(C4(C)C(=C)OCC4)n3C)CCC2)ccc2snc(Cl)c2c1 11079,N1(C(CCCOCC=C)=O)C2CCC1C(NC(=O)CNC=O)C2 11080,C1(CNC(c2c(C)c(F)ccc2)=O)CCCCN(C(=O)Cc2n[nH]c(=N)s2)CC1 11081,C1(C(=O)NCC(C)OCC#C)C2CC3C(C2NC(C2(CO)CCOC2)=O)C13 11082,C1(NC(c2c(OCC)ccs2)=O)CCN(C(C2CCCCC2)=O)C1C(C)(C)C 11083,N1(C(C2(C)C=CCC2)=O)CCC(CC(=O)NC2CN(C(N)=O)C2)CC1 11084,C(=O)(CN=S(C)(C)=O)N1C(CN(C)C(C2CC2c2ccncc2)=O)COCC1 11085,N1(C(c2cnc(COC)s2)=O)CC=CC(NC(=O)CC2CCCO2)C1 11086,CCC(CO)CCNC(C1C=CCCN1C(=O)Cc1cn[nH]c1)=O 11087,N1(C(c2ccccn2)=O)CCCC(C(N2CCN(S(=O)(=O)CBr)CC2)=O)C1 11088,C1(CNC(c2c(C)cco2)=O)C(C2CC2)CCN1C(c1ncc[nH]c1=O)=O 11089,c1(CC)nnc(CC)s1.C1(C2COC2)C(=O)N1CC 11090,C=CCCCC(C(=O)NC(C=C)C(F)(F)F)NC(=O)CCNC(C)=O 11091,c1(C(N2CCC23CN(Cc2ccncc2)C3)=O)cccc(C(F)(F)F)c1F 11092,C1(CC(=O)N(C(C)C(=O)NC2C3CCCC23)CC)CCCC(C)O1 11093,c1(C(N2CC3CC(NC(C(C)(C)C)=O)C3C2)=O)nccc2cccnc12 11094,C1(NC(C(CC)CC)=O)CCN(C(c2ccc(CC#N)cc2)=O)C(C2CC2)C1 11095,CC(C)(CNC(=O)CCc1cncnc1)CNC(c1nn[nH]c1C(F)(F)F)=O 11096,Cc1cc(-c2ccnc(NC(=O)Nc3cc(C)c(Cl)cn3)c2)cc(C)n1 11097,C1(NC(C(=O)NC2CC(C)OC(C)C2)=O)CCCCC12CCCC2 11098,c1(C(=O)NC2C(C)N(C(=O)Cc3cncnc3)CCC2)cn2ccccc2n1 11099,c1(C(N2CC(C(C)C)C(NC(=O)COC(C)(C)C)CC2)=O)nc2c(s1)COCC2 11100,N1(C(CCN(C(=O)C2=NNC(=O)C2)CC)=O)CC2(CC=CC2)C1 11101,c1(C(=O)NC(CNC(c2ccncc2NC2CCCCC2)=O)CO)ccc(F)cc1 11102,N#CC1CCN(C(C2CCOCC2NC(C2(O)CCOC2)=O)=O)CC1 11103,c1(C(=O)NC2C3CN(C(C4CCCN(C(C)=O)C4)=O)C2C3)cnc(F)c(C)c1 11104,N1(C(C(CC=C)C)=O)CC(NC(=O)Cc2ccoc2)CC(C)C1 11105,CC(CN(C)C)CCC(=O)N1CCN(C(=O)C=Cc2cc[nH]c2)C(C)C1 11106,C(=O)(CCC(=O)NN(C)C)NC(C1(O)CCN(C(C(CC#C)O)=O)CC1)C 11107,c1(C(N(CCNC(=O)COC2CCCCCC2)CC)=O)nc2c(s1)CN(C)CC2 11108,C1(CNC(Cc2c(C)cccc2)=O)CC2(CO1)CN(C(c1c(C)n[nH]c1C)=O)C2 11109,C1(C(=O)NCc2cc(NC(C)=O)n(C)c2)CCC2(CCC2)CO1.C12CCN1C2 11110,c1(C(C)OC)cn(CC(F)CCNC(C2OCC2(C)C)=O)nn1 11111,C1(NC(CC2(C)CCOC2)=O)CCCCC1CC(=O)NCCCc1ccsc1 11112,c1(C2C(C(=O)NCCNC(c3n(C(CC)C)ncc3)=O)C2)ccccc1Cl 11113,N1(C(c2cc(CC)[nH]n2)=O)CCC(CNC(=O)C(C)SC)C(C)C1 11114,c1(OC)ccc(Br)cc1CC(N1C(C(N2CCCC2CC(C)C)=O)CC2CC12)=O 11115,N1(C(C=CCNC(C(C(=O)OC)(C)C)=O)=O)CC2(C1)NC(=O)NC2=O 11116,c1(C(C(=O)NC2CCOCC2)N(CCC(F)(F)F)CC)ccc(C)c(Cl)c1 11117,N1(C(C=Cc2ncn(C)c2)=O)C2CCC1CN(C(c1cc(C3CC3)sn1)=O)CC2 11118,c1(OCC(=O)NCCC2N(C(CC#C)=O)CCCC2)ccc(Br)c(Cl)c1 11119,CCC(C)CC(=O)NC1CC(CNC(=O)CSCc2ccc(Cl)s2)C1 11120,c1(CC)ncccc1C(N1CCC(CC(C)C)CC1)C(=O)NC(C)C(=O)NC 11121,CC1C(=O)NC(=O)CN1C(=O)C=CCC1(NC(=O)Cc2cccn2C)CCC1 11122,c1(C(=O)NCC(C)NC(c2ccccc2N(C)C)=O)cc(C#N)no1 11123,c1(OC)ccc(CC(=O)NCC2C=CCN2C(c2conc2C)=O)cn1 11124,c1(C(=O)NCCC2(OC)CN(C(c3ncsc3C(C)C)=O)C2)occ2c1CCC2 11125,C(=O)(C(C)(C)CS(N)(=O)=O)NC1CN(C(c2c(C)nc(CC)s2)=O)CC(O)C1 11126,Cc1ccc(C(=O)O)c(-n2cc(-c3ccns3)nn2)c1.C12CCCN(C1)C2 11127,N1(C(c2c(C)n[nH]c2C)=O)CCN2C(=O)C(NC(=O)CC(C)(C)C)CC2C1 11128,c1(OC)ccc(NC(c2ccccc2NS(=O)(=O)C2CC2)=O)c(OC)c1OC 11129,C(CC(C)C(=O)NC(C1CCN(C(=O)C(=C2CCCCC2)F)CC1)CO)OC 11130,C1(O)(C(C(=O)NOCCCOC)NC(CN(CCC)C)=O)CCCCC1 11131,c1(C(N2CCC(C)N(C(c3ccco3)=O)CC2)=O)c(S(C)(=O)=O)cnn1C 11132,c1(NC)cc(Cl)ccc1Cl.C1(CC=C)(NC(=O)CSC)CN(C(=O)Cc2cnc[nH]2)C1 11133,c1(C(N2C(C)C(NC(=O)C(=O)N=S(C)(C)=O)CCC2)=O)cn2c(n1)C(C)CCC2 11134,N1(C(C(C=C)CC)=O)CCCCCC(NC(=O)CCNS(C)(=O)=O)C1 11135,Cc1ccc(C2CC2C(=O)N(CCCCCNC(C2(F)CCOC2)=O)C)cc1 11136,C1(CC)CN(C(C2CCN(C(=O)C(C)C(=O)OC)C2C)=O)CCS1 11137,CN1CCCCC1CC(=O)NC1CCCC1(C)CNC(c1c[nH]nc1C(F)F)=O 11138,c1(C(=O)NCC(C)N(C(=O)C(C)C(C)(F)F)CC)cc(OC)c2c(c1)OCCO2 11139,C1(CC(=O)NC(C(C)(C)NC(c2cnc(CCCC)s2)=O)C)CC(=O)NC1=O 11140,N1(C(CCC(C)(C)NC(=O)Cn2cnnc2O)=O)CC2CC(C1)C2(C)C 11141,c1(OC)ccc(C)c(C(=O)NCC2(CCCNC(=O)C=C(C)C)CCCC2)n1 11142,O=S(=O)(c1cccc(F)c1)NC(C1CNCC2(CCOCC2)O1)=O 11143,c1(OC)cc(C(=O)NCC2CCC2NC(c2cc(Br)n(C)n2)=O)ccc1C 11144,c1(OCC)ccc(N)c(C(=O)NC2(CO)CCN(C(=O)C(O)C(F)(F)F)C2)c1 11145,c1(C(=O)NC(C(N2CCC(COC)CC2)=O)CO)ccc2n[nH]cc2c1 11146,c1(CCNC(C2CCCCO2)CF)cccc(Cl)c1Cl 11147,c1(N2CC3CCN(C)C3C2)nc(=NCc2nccc(O)n2)[nH]c2ccsc12 11148,c1(C(=O)NC2C(O)CCN(C(c3nc(C)oc3C)=O)C2)cccc2c1OCC2 11149,C(=O)(C(CC(N)=O)NC(=O)Nc1ccccc1)NC1CCN(C(CCC=C)=O)C1 11150,Cn1cnn(CC(N2CC(CNC(=O)CCc3ccc(Cl)cc3)C2)=O)c1=O 11151,C1(n2c(C)ncn2)COCCN1N1CCC(N)CC1.N1CCCC1 11152,c1(C(N2C(C(=O)NC34CCN(CC3)C4)(CC)CCC2)=O)coc2ccccc12 11153,c1(C(N2C(COC)CN(C(=O)C=CSC)CC2)=O)cnn2ccc(OC)cc12 11154,c1(OCC)cc(OC)nc(NC2CC(NC(C3CC4(CC(=O)N4)C3)=O)C2)n1 11155,C1(C(=O)NC(C)CN2CCCC2)C2CCCC2CN1C(=O)Cn1ccc(Cl)n1 11156,N1(CC)CC(NC(C2(NC(c3ncncc3Cl)=O)CC(O)C2)=O)CC1=O 11157,n1(CC(=O)NC2(CF)CCN(C(C3OCCCO3)=O)C2)nc(O)ccc1=O 11158,CCC(CNC(C1CCS(=O)(=O)CC1)=O)(C(=O)OC)c1ccccc1 11159,Cc1c(C(=O)N(C(C)C(=O)NC(CO)CCF)C2CC2)ccn1C 11160,c1(-c2cn(CC3CCN(C(CN(C)C)=O)C3)nn2)cc(CO)ccn1 11161,CCC(C(=O)NCC(C1CCCCC1)NC(=O)Cc1cnc(Cl)cc1C)C(F)(F)F 11162,c1(CC(=O)NC(C(C)NC(c2c(CC)ocn2)=O)(C)C)ccc(F)c(Cl)c1F 11163,CC1(C)C(CNC(=O)Cc2ccsc2)CCN1C(C1CCCC12CC2)=O 11164,c1(C(=O)NCCC2CC(NC(=O)CC3CC4CCC3O4)C2)nc2ccccc2s1 11165,C(CC(=O)NCCC1CCC(C)(C)O1)(C(C)(C)C)NC(C1CCCN(CC)C1)=O 11166,CN1CCCCC(C(=O)NC(C)(CNC(C2(C)CCC(=O)C2)=O)C2CC2)C1=O 11167,c1(CCC)noc(CCC(=O)N(C2CCN(C(=O)C=C(C)C(F)F)C2)C)n1 11168,C1(CNC(c2occ(C)c2)=O)CC(C)N(C(c2cn(C(C)C)cn2)=O)C1 11169,C(C)(CCC(C)(C)C)NC(c1nnnn1CCCC(=O)OC)(CC)C1CCC1 11170,CC(C)P(=O)(CC(=O)NCC1(C(N)=O)CN(C(=O)C(C)(C)F)C1)C(C)C 11171,C1(O)(CNC(C2(NC(CC3(COC)CC3)=O)CCC2)=O)CCCC1C 11172,CCCCC(CNC(=O)COCCCF)NC(=O)C(C)Oc1cccc(C)c1 11173,CC(=O)C(C)CC(C)C(=O)OCC(N1CCCCC1C(C)CCCl)=O 11174,c1(C(=O)NC2CCN(C(c3c(F)cccc3F)=O)C2)cccc(F)c1C1CC1 11175,c1(C(N(C)CCC2CCN(C(=O)Cn3cccn3)CC2)=O)cccn2nnnc12 11176,c1(C(C)N(C)C(=O)N(C)CC2CCCO2)cnn(C)c1 11177,Cn1nnc2ccc(C(N3CC(NC(c4ccc(=O)oc4)=O)C4(CC4)C3)=O)cc12 11178,N1(C(C2(SC)CCC2)=O)CCN(C(C2CCCCS2)=O)C(c2nccn2C)C1 11179,c1(C(=O)NCCC2(CNC(CN(S(C)(=O)=O)C)=O)CC2)nnc2ccccc2n1 11180,c1(OC)cccc(CNC(=O)NC2(C)CCN(C(c3occc3C)=O)C2)c1 11181,c1(C(C(=O)N(CCN(C(C(C)C2CCC2)=O)C)C)C)ccc(Cl)c(Cl)c1 11182,N1(C(C(C)=CC)=O)CC2CCN(C(c3nc4ncc(C)cn4n3)=O)C(C2)C1 11183,N1(C(C2C(CNC(C3(CCC)CC3)=O)CCO2)=O)CCC(CO)C(C)(C)C1 11184,Cc1cccc(C(CNC(=O)N(C(C)(C)S(C)(=O)=O)C)OCCCN)c1 11185,C(C(CCC)CCC)NC(CCC#CC)=O 11186,N1(C(C=C=C(C)C)=O)CCCC(F)(C(=O)NCC(F)C2CCC2)C1 11187,N1(C(C2CCC(C(=O)OC)C2)=O)CC2CC(C)N(C(c3ccsc3Cl)=O)C2C1 11188,c1(CC)cc(C(=O)NCCC(C)NC(C2(C(F)(F)F)CC(O)C2)=O)c(C)o1 11189,C1(C(=O)NCC2(F)CC(CNC(C3CCCO3)=O)C2)Cc2ccccc2S1 11190,CCCCC(C)C(=O)NC(CNC(c1cnn(CC)c1C1CC1)=O)CC(C)C 11191,C(=O)(CCS(=O)(=O)C(F)(F)F)N1CC(CCNC(Cc2cnn(C)c2CO)=O)C1 11192,CC1COCCC1NC(=O)C(CC1CC1)NC(=O)CC=C(Cl)Cl 11193,C1(NC(c2ncc(C(N)=O)nc2)=O)CN(C(=O)CCOCCF)CCC1C(F)(F)F 11194,CC(C)CC(C(=O)NC1CCCCCN(C(=O)C(=O)NC2CC2)C1)C(N)=O 11195,CC(C)(C)C(CNC(=O)C(O)CC1CCOCC1)NC(C1(CF)CCC1)=O 11196,C1(C(N(C(CC)CNC(c2cnc(C(C)(C)C)o2)=O)C)=O)CCOC(C)(C)C1 11197,N1(C(c2cnc3ncccn23)C(=O)NCC)CCC2(CCN(C)CC2)C1 11198,N1(C(C2C(=C)C2)=O)CCC(CO)(CNC(=O)Cn2cccnc2=O)C1 11199,c1(NC(C2CCCN(C(CC(CC)C)=O)C2)=O)cc(F)c([N+](=O)[O-])cc1F 11200,c1(C(N(CC(CC)NC(C2(O)CCOC2)=O)C)=O)ccsc1SC 11201,c1(NC(N2CCCC(O)(c3ccc(Cl)cc3)C2)=O)ccc(S(=O)(=O)CC2CC2)cc1 11202,N1(C(Cc2c(C)ccnc2)=O)CC2CCC1C(NC(=O)Cn1ccnn1)C2 11203,C1(CNC(c2ncn(C(C)(C)C)n2)=O)CC2CCC1N2C(C1(C)CCC(=O)C1)=O 11204,C(=O)(C1CCCc2ncccc21)NCC(CNC(c1c(C)onc1Cl)=O)C 11205,c1(NC(CCC2N(c3ccnc(N(C)C)n3)CCC2)=O)ccc(Br)cc1F 11206,CC1(NC(=O)C)CC(NC(C2CCOC2)=O)C1.c1(-c2csnn2)ccccc1 11207,C(N=c1cc[nH]cc1S(=O)(=O)NCC1(CO)CC1)c1cnc(C(C)(F)F)s1 11208,N1(C(C(C2CCCC2)NC(C2NC(=O)CC(C)C2)=O)=O)CCC2CCC(C1)N2C 11209,C1(C(=O)NCCC(C)N(C(C(C)OCC#C)=O)C)CC12CCOCC2 11210,CC(CCC(=O)NC1(C2CCN(C(=O)C3=CCOC3)CC2)CC1)S(C)(=O)=O 11211,N1(C(C2CN(C(C3CCCC(C#N)C3)=O)CCC2)=O)CC2(COC(=O)C2)C1 11212,c1(C(=O)NC23CC(NC(C4C(CCC)C4)=O)(C2)C3)ccc(CC)c(C)c1 11213,C(=O)(CCCCCNC(C1CC2(CC2)CO1)=O)NC(c1cn[nH]c1)C 11214,C1(C)(CNC(C(c2cccnc2)C)=O)CCCN1C(c1cccc[n+]1[O-])=O 11215,c1(C(=O)NCC(C)NC(=O)C(c2ccc(Cl)cc2Cl)O)nccc2[nH]ccc12 11216,c1(C(=O)NCCCNC(C(c2cc3ccccc3o2)C)=O)ccc2c(c1)CCO2 11217,C(=O)(CC(O)CNC(=O)CCCN(C)C)NC(C1CSC1)C 11218,Cc1nc(N2CCC(NC(=O)Cn3nnnc3C3CC3)C(O)C2)cc(C#N)n1 11219,N1(C(C2(C)COC2)=O)CC(C(N2CCCCC2C(C)(C)O)=O)C(F)C1 11220,C(=O)(CC1OCc2ccccc21)NCC1CN(C(C(CCOC)C)=O)C(C)C1 11221,Cn1c([N+](=O)[O-])cnc1C(N1CC2CCOC2(CNC(=O)CC2CC(F)C2)C1)=O 11222,C1(CCNC(CC)=O)CCCN1C(c1csc(NC(=O)NC2CC2)n1)=O 11223,c1(NC(C2C(CNC(C3CCC(C4CC4)C3)=O)OCC2)=O)cnc2c(c1)CCC2 11224,c1(C(N(CCCCNC(C2CC2C2CCCO2)=O)C)=O)ccncc1Br 11225,C1(NC(C(CSC)C)=O)CC2CN(C(c3cc(-c4ccncc4)on3)=O)CC12 11226,N1(C(C(Cc2cn[nH]c2)NC(c2cc(OC)no2)=O)=O)CCOCC1CC(C)C 11227,CC1CC(C(N2CC3(CCCO3)C2)=O)CCN1C(C1CCCCNC1=O)=O 11228,N1(C(C(C)(C)NC(=O)C(F)(F)F)=O)CC2CN(C(C3CC(=O)C3)=O)CC2C1 11229,C1(N=[N+]=[N-])(C(N(C2CCCC2C#N)C)=O)CCN(C(=O)CN2CSCC2=O)C1 11230,N1(C(Cc2nc(COC)sc2)=O)CC2CCN(C(c3cccc(Cl)n3)=O)C(C2)C1 11231,c1(CCC(=O)N(CCN2C(C)CCCC2)C(C)=O)nc2cccc(Cl)c2[nH]1 11232,C1(OC)CCN(C(C2CCCCCN2C(=O)CCC(=O)C2CC2)=O)CC1O 11233,c1(C(=O)OC)nccn1CC1CN(C(=O)CC2(NC(=O)C(C)(Cl)Cl)CCC2)C1 11234,N1(C(=O)CCC2OCCO2)CCCC2C1CCN2C(=O)CC1CCC1 11235,C(CC(F)(F)Cn1cc(CCN(C)C)nn1)NC(COCCCC)=O 11236,N1(C(C)CN(C2CC(=CC(C)N(C)C)C2)C=O)CCC2(CC=CCO2)C1 11237,N1(C(c2cncc(C)n2)=O)CCC2CN(C(=O)Cc3nc(C4CC4)cs3)CC2C1 11238,C1(C(=O)NCCCN(C(=O)CC2CCCCO2)C)(CC)CCOCC1 11239,c1(C(N(C2CCN(C(=O)CC3C=CCCC3)CC2)CCOC)=O)ccccc1C 11240,S(=O)(=O)(c1cccs1)NCC(=O)NC(CNC(Cc1c(C)nsc1)=O)C1CC1 11241,N1(C(CC(=C)C)=O)CC(NC(=O)CCc2cc(Cl)no2)CC(C)C1 11242,c1(C(=O)NCC(c2cn(CC)nc2)O)ccc(Br)c2cn[nH]c12 11243,c1(C(=O)NCC2N(C(C3C(C)C3)=O)CC3(CC3)C2)c[nH]c2nccc-2c1 11244,N1(C(C(C)OCCC=C)=O)CCC(C2CCCN2C(=O)C2=CCCC2)CC1 11245,C1(CC(N2CCC(OCCNC(C3C(OCC)C3)=O)C2)=O)CCCS(=O)(=O)C1 11246,c1(NCC(=C)CC)ccc(S(=O)(=O)NCCC(C)(C)F)cc1C#N 11247,Cc1cc(C)cc(C=CC(=O)NC(CNC(=O)CCC(C)(C)F)CC(C)C)c1 11248,CC(C)(CCCF)C(=O)NCc1ncc(C(=O)NOCCCCF)cn1 11249,N1(C(c2c(C)cno2)=O)CCC(CNC(c2cnn(C3CCC3)c2)=O)C12CCC2 11250,N1(C(C(Br)=C(C)C)=O)CC(CNC(=O)COC2CCCCC2)CCC1C 11251,N1(C(c2cnc(C)o2)=O)CC(NC(c2ccc(CC(C)(C)C)cc2)=O)CC1C 11252,C(=O)(CCS(C)(=O)=O)N1CCC(CC)C1CNC(=O)C(=Cc1cccnc1)C 11253,C1(NC(CCCC#CC)=O)CN(C(=O)CC(C)CN(C)C)C2(CCC2)C1 11254,c1(C(C)C)ncc(C=CCNc2conc2C2CC2)s1 11255,C=CC1(CC(=O)NC(c2ccnn2C)CO)CN(C(=O)CCN(C)C)C1 11256,Cc1onc(CO)c1C(=O)NC1CCN(C(c2ccc(C#N)s2)=O)C1 11257,C1(CCNC(N2C(CCN(C)C)C=CC2)=O)CCCCC12CC2 11258,N1(C(c2c(Cl)cn(C)n2)C(=O)NC2CCOC2)CCCC2(CCCNC2=O)C1 11259,CC1CC=C(C(=O)N2CCC(CN(C)C(c3cccc(O)c3F)=O)C2)CC1 11260,Cc1cc2nc[nH]c(=NCC(C(C)(C)C)NC(c3cc(O)nc(C)n3)=O)c2[nH]1 11261,C1(C(N2CCN(C(c3c(Cl)ccc(C)c3)=O)CC2C)=O)CCCC2CCCN12 11262,Cc1cc(-n2cccn2)nc(=NC(C)C2CCCCN2C(=O)CC2CCC2)[nH]1 11263,C1(CNC(C(C)O)=O)CCCN(C(=O)C=CCN2CCC2)C1 11264,c1(C(=O)NCC2CN(C(CNC(C)=O)=O)CC2(C)C)ccc(O)c(F)c1F 11265,c1(NC(C(CNC(=O)CCNC(N)=O)OC)=O)cccc(C(C)F)c1 11266,c1(NC2C(C(=O)Nc3c(OC)cc(F)c(C)c3)C2)ncnc2c(C)cccc12 11267,CC1=C(C(=O)N(CCCCCNC(=O)CC2(CO)CC2)C)SCCO1 11268,N1(C(CC2(O)CCCN(C(C)=O)C2)=O)CC2CN(C(c3c[nH]cc3Br)=O)CC2C1 11269,c1(-c2nc(C(C3CCCO3)C)nn2-c2cnnn2C)cc(CO)nc2oncc12 11270,Cc1cc(O)ccc1CNC(C12CC(NC(=O)OC(C)(C)C)C1C2)=O 11271,c1(C(=O)NC2C(C)CN(C(C34CC3C4)=O)C2)cnc2[nH]cncc1-2 11272,C1(OC)CC(OC(C)(C)C)CN(C(C2CC(CC(F)F)C2)=O)C1 11273,CC(C)C(O)C(C)C(=O)N1CC(C(=O)NC2CNC(=O)C23CC3)CC12CCC2 11274,N1(C(C(COCC)(C)C)=O)CC(NC(=O)COc2ccc(F)c(F)c2)C(C)(C)C1 11275,C1(C)(CNC(C2(CC)CC=CC2)=O)CCCN(C(=O)CCN2CCCCCC2)C1 11276,C#CCC(C)(COCCOC(=O)CCc1cc(C(=O)OC(C)(C)C)c(C)o1)CO 11277,CC(CC(C)(C)C)C(=O)NCC12CCC(CN1C(c1cc(Br)n[nH]1)=O)C2 11278,N1(C(C(C)C2CC2)=O)CCCC(CN2CCN(C(C3(F)CC=CC3)=O)CC2)C1 11279,N1(C(Cc2nc(C)oc2)=O)CC2ON=C(CNC(c3nnc(C)s3)=O)C2C1 11280,C1(NC(C2(F)CCN(C(C=CC(=O)OC)=O)C2)=O)CC2CC(OC)C2C1 11281,C(=O)(C(C(C)(C)C)OCC)N(CCC)CCNC(C12CCCC1C2)=O 11282,N1(CC(=O)N(CCC(N2CCC(n3ccnn3)C2)=O)CCO)CCC(F)CC1 11283,c1(N2CC(C(C)C)OCC2)nc(NC2CC2C(F)(F)F)c2cnn(C)c2n1 11284,c1(CN2CCCC(NC(c3cnc(C)s3)=O)C2)ccc(C(F)(F)F)cc1O 11285,Cc1cc(C(=O)NCC2CC(NC(c3nc[nH]c3C(F)(F)F)=O)C2)cs1 11286,Cc1[nH]c(C(=O)N(C)CC2CCN(C(=O)CC(C)(C)C#N)CC2)c(C)c1C 11287,CC1OC(C)C(C(N2CCCCC2CNC(C2CC(F)(F)C2)=O)=O)C1C 11288,c1(C(=O)NCC2CCCC(NC(CC=CCC)=O)C2)cc(N)cc(O)n1 11289,N1(C(=O)C=CCOC)CCCC(CN(C(=O)COC2CC(OCC)C2)C)C1 11290,CC(C)C(CNC(=O)CC1CSC1)C(=O)N(C)Cc1ccon1 11291,N1(C(CN(C(=O)OCC)C)=O)CC(C)(C(N2CC3(CCCN3C)C2)=O)CC1(C)C 11292,O=C(C#CC1CCCCO1)NC1CCC2CCN(C(=O)CN3CCCC3=O)C12 11293,Cc1cn2c(n1)CCC(C(=O)NC1CC(CNC(c3ccc(C)s3)=O)C1)C2 11294,C1(N(C(CN(CC(C)NC(c2ccon2)=O)C)=O)C)CCCCCC1 11295,N1(C(C(F)OC)=O)CCC(NC(=O)C(Cc2ccsc2)NC=O)CC(C)(C)C1 11296,Cc1ccnc(C(=O)NC2CCCC2NC(C2CC(=O)C2C(C)(C)C)=O)c1F 11297,CC(C)CC(C)C(=O)N1CCOC(C(=O)NCCC(CO)C(C)C)C1 11298,c1(C(=O)OC)ccc2sc(=NC3CC(CNC(=O)Cc4cn(C)nn4)C3)[nH]c2c1 11299,N1CCS(=O)(=O)CC1.C(=O)(C(C#N)C(C)C)NC1C(NC(C(CC)(C)OC)=O)C1 11300,Cn1nc(C(F)F)nc1C(C1CC1)NC(=O)CCn1cc(C2(C)CC2)nn1 11301,C#CC1(C(=O)NCCC2CC(C)=NO2)CCN(C(C2OCCCC2(C)C)=O)CC1 11302,CC1(C)CCN(C(=O)C2=CCCS2)CC1NC(=O)CCC1CC1CC1CC1 11303,C(=O)(CCCCCCC(=O)N1CCC(NC(C2CCC(F)CC2)=O)C(F)C1)OC 11304,C12(NC(Cc3ccc(OCC)cn3)=O)CCCC1CN(C(c1occc1F)=O)C2 11305,n1(CCNC(c2n(C)cc(NC(=O)CO)c2)=O)cnc2ccccc12 11306,c1(C(N2C(C3(NC(CCC=C(C)C)=O)CC3)CCC2)=O)ncc(Cl)cc1O 11307,Cc1cc(C(=O)NNC(=O)N2CC(N3CCC(F)(F)C3)C2)c(C)n1-c1ccccc1 11308,C=CC(C)(O)CC(=O)NCCc1cc(C(=O)NCCN(CCO)CC)no1 11309,C(=O)(C1=C(Cl)CCOC1)NCC1C(NC(CC2CCCC(C)(C)O2)=O)CCCC1 11310,C(=O)(C(CNC(c1c(Cl)cnn1C)=O)C(C)(C)C)NCC1(O)CCN(C)C1 11311,C1(NC(C2N(C(=O)NC)CCC2)=O)CCC2CC1CN2C(c1ncncc1Cl)=O 11312,C(C)(C)(CC(=O)N(C)CCc1ccccn1)N(C(C1C(C)C1C)=O)C 11313,c1(-c2nc(C(C)SCC)nn2-c2ccc(C)cc2)nc2ncccn2n1 11314,N1(C(CN2CCCC(CC)C2)=O)CCC(NC(=O)Cc2ccsc2Cl)C12CC2 11315,N1(C(C2CN(C(N)=O)C2)=O)CCOC2(CCC(NC(C3CC=CC3)=O)CC2)C1 11316,c1(C(N(C)Cc2cn(CC3CC3C3CCOCC3)nn2)=O)ccc([N+](=O)[O-])cc1 11317,CC(C)CC(C)C(=O)NCC(C)NC(c1c(Br)cnn1C)=O 11318,C(=O)(C1=CC2C=CC(C1)C2)NC(C(=O)N(C(C=C)C)C)CO 11319,C1(CNC(C2C3CN(C(=O)CCc4nc[nH]n4)CC23)=O)CCCCCC1 11320,CCC(CNC(c1cscc1C)=O)(CC)NC(c1ccc(C(=O)N(C)C)cc1)=O 11321,N1(C(C2CC(=C)C2)=O)CCC2(COC(CNC(=O)CCS(C)=O)C2)C1 11322,Cc1ccc(C(=O)NC2CN(C(=O)CN3CC4CC4C3)CC2C)n1C(C)C 11323,CCCC(C(=O)NC1(CO)CN(C(c2nc(C)sc2C)=O)C1)N(C)C 11324,N1(C(CCC=CC(C)C)=O)CC2(CCCC2)C1 11325,CCC(COC)C(=O)NCCCN(C(c1cc(C(C)(C)O)ccn1)=O)CC 11326,C1(CCCNC(C2(C)C=CCC2)=O)CCCCN1C(=O)Cc1cnccc1Cl 11327,C(CCS(=O)(=O)NCC(N1CCC(NC(=O)Cc2ccc(Cl)s2)C1C)=O)OC 11328,CCC(CC)C(=O)NCC(=O)NCCCC1(NC(=O)C(C)C(C)O)CC1 11329,c1(C(N2CC(NC(C(CC)CC)=O)C(C)C2)=O)cc(Cl)c(O)c(Cl)c1 11330,n1(CC(C(=O)NCCCNC(c2scc(C(C)=O)c2)=O)(C)O)c(C)cccc1=O 11331,Cc1ncc(F)c(N2CCC(C#N)(NC(c3n[nH]c(C)c3C)=O)C2)n1 11332,C1(NC(c2csc(-c3ccccc3)c2)=O)CC2(C1)CN(C(C1CCCCO1)=O)C2 11333,c1(C(=O)NC2CN(C(=O)C(F)(F)c3nccs3)CCC2F)cccc2nccn12 11334,N1(C(CN(C)CC)=O)CC(O)CC1CNC(=O)C(F)(F)c1cccnc1 11335,c1(CC(=O)NCC(C)(C2CC2)NC(C(CCC)OC)=O)ccc2ocnc2c1 11336,CCC1c2ccsc2CCN1C(c1cccnn1)C(=O)NC1CCCCC1 11337,C(C(C)(C)C(=O)NC(C)CCCNC(=O)C(O)CCSC)OCC 11338,Cc1cc(C(N)=O)cc(C(=O)NNC(c2c(Cl)cncc2Cl)=O)c1 11339,Cc1cc([N+](=O)[O-])cnc1C(N1CCC(C2(NC(c3csc(O)n3)=O)CC2)C1)=O 11340,CN1CCCC1C=CC(=O)NCCN(C(=O)C=Cc1cscn1)C1CC1 11341,c1(CCC(=O)N(C(CC)C)CC)ccc(OC)c(OC(=O)C(C)=CC(C)(C)C)c1 11342,C1(N(C(C(C)(C)NC(C=COC)=O)=O)C)CN(C(C2CCOC2)=O)CC12CC2 11343,C(CO)(C(=O)NC(c1ccn(C)n1)C)NC(C1(COC)CC1)=O 11344,c1(C(N(CC(CC)NC(CC(=C)I)=O)C)=O)n[nH]c(C)c1O 11345,Cc1cc(Cl)cnc1C(N1CC(O)(CCc2cn(C3CCCCC3)nn2)C1)=O 11346,Cc1cc(F)c(CC(N2CCN(c3ccccc3F)C(=O)C2)=O)cc1F 11347,c1(NC(C2CCC(CCCCC)O2)=O)cc(F)ccc1C(C)(F)F 11348,CCC(CC(=O)NCCC1CC(C)C1)N(C)C(c1cnsc1C)=O 11349,c1(CNC(Cc2cn(CC)nn2)=O)ncccc1CNC(C1CNC(=O)C1)=O 11350,c1(OC)cc(CC(=O)NC2CCC2NC(=O)CCc2ncc[nH]2)cc(F)c1 11351,C1(C(=O)NCC(C(=O)NC)C)CC12CCN(C(=O)CC(O)C1CCCC1)C2 11352,C=CC(C)(C)CC(=O)NC1CCC(CNC(c2cc(C3CC3)ccc2F)=O)C1 11353,c1(C(=O)N(C)C)cc(C(=O)OC(c2ccnn2C)C)c2n1CCOC2 11354,C1(F)(C(N(CCC)CCNC(=O)C(c2cccc(F)c2)C)=O)CCN(C)CC1 11355,Cc1ccc(C(=O)NCCN(CC(C)O)C(c2coc(Br)c2)=O)o1 11356,c1(Cn2cc(C(=O)NCC3(F)CC(CNC(=O)CO)C3)nn2)cccc(Cl)c1 11357,C1(C(=O)NCCCC2N(C(C3(C(=O)OC)CCO3)=O)CCC2)COC(C)(C)C1 11358,c1(OC)cc2[nH]ncc2cc1NC(C1CCN(C(C2(C)CCCN2)=O)CC1)=O 11359,c1(NC(=O)OCC)ccc2c(c1)OCCO2.C12CCCC1C(=O)OC2 11360,Cc1oc2ccccc2c1C(=O)N(CC(C)(C)NC(=O)C1Cc2ccccc21)C 11361,c1(C(N2CC(O)(CC3CC(O)C3)C2)=O)ccc(C(=O)NCCn2cncn2)nc1 11362,N1(C(C2N(C=O)CCC2)=O)CC(O)C(O)C1CNC(C1(F)CCCC1)=O 11363,C1(C(N2C(CNC(Cc3cccc(OC)n3)=O)C(C)CC2)=O)CC(=O)CC(=O)C1 11364,N1(C(C2CCC(=C)CC2)=O)CCC2CCN(C(=O)C(C)SC(C)C)CC2C1 11365,c1(C(N2CC(NC(c3ccc(O)nn3)=O)CC(C)C2)=O)cc2c(cn1)OCCO2 11366,c1(C(c2cccnc2)CC(Cc2ccccc2)N(C(C)=O)CC)nc(C)n(C)n1 11367,C(C#CC(F)(F)F)NC1CCN(C(C(=O)N(CC(F)F)C)=O)C1 11368,c1(NC2CCC(SC)C2)ccc(S(=O)(=O)N(C2CCOCC2)C)cc1C#N 11369,c1(C(N(C2CCCN(C(C34CC(O)C3C4)=O)C2)C)=O)ccc2c(c1)C=CS2(=O)=O 11370,c1(CC)cccc(N(Cc2cn(C)nn2)CC2CCC2)c1.c12ncn(n1)[nH]c2=O 11371,Cn1c(C(N2CCOC(C3CN(C(=O)C=CCO)C3)C2)=O)cnc1O 11372,C(N=c1cc(C)nc[nH]1)C1CN(C(C(C)NC(COC)=O)=O)CC1(C)C 11373,C(CCC(C)C)(C(=O)N1CCC(O)C(C)C1)NC(CCN(CC)CC)=O 11374,c1(N(C(N2C(C)CC2CO)=O)C)ccc(-c2ccccc2)c(F)c1 11375,C1(C(=O)NC(CC(=O)N2C(CCC=C)CCC2)CC=C)CC2COCC(C1)C2 11376,c1(C(=O)NCC(CO)NC(c2ccc(C3(C)CC3)cc2)=O)cccc([N+](=O)[O-])c1 11377,Cc1c(Cl)ccnc1C(N1CCC(CF)(NC(=O)CCc2ncc[nH]2)C1)=O 11378,c1(CCC(=O)Nc2cc(C(C)(C)C#N)c(F)cc2)nc(O)c2ccccc2n1 11379,n1(C(C)CNC(C2(Cc3ccccn3)CC2)=O)cc(C(C2CCOC2)O)nn1 11380,Cn1nccc1C1CC1NC(N1CCC(c2nncs2)C1)=O 11381,N1(N2CCC(c3n(C)c(=O)on3)CC2)CCN2C(=O)COCC2C1.C(C)(C)C 11382,C(N=c1[nH]cnc2cc(C)[nH]c12)C1C(NC(Cn2ccc(C)cc2=O)=O)CCC1 11383,N1(C(C(CC)C)=O)C2CCC1C(C(N1CCCC1c1ccncc1)=O)C2 11384,c1(C(=O)NC2CCC(=CC(NOC3CCN(C)CC3)=O)C2)cccc2[nH]ncc12 11385,C12(C(=O)NCC(CC(=O)NCC3(CO)CCN(C)C3)O)CCC(CC1)CO2 11386,C1(NC(C(C)SCCCC)=O)CN(C(c2cc(CCOC)on2)=O)CC1C 11387,Cc1cc(C)c(CC(N2CC3(CC3)CC2C(=O)NCC(F)CO)=O)c(C)c1 11388,C1(NC(COCCCC)=O)C(C)CCN(C(=O)CCc2ccn(C)n2)C1C 11389,N1(C(c2ccc(CC)o2)=O)CCCC2(C1)CN(C(=O)CC1CN3CCN1CC3)C2 11390,Fc1cccc2cccc(CNCc3cc(F)c(F)cc3N)c12 11391,Cc1ccc(NC(C2CC(O)(CNC(=O)C=Cc3ccncn3)C2)=O)cc1F 11392,C(C(C)(C)C(=O)NCc1cccc(F)c1)NC(c1ccc(CC)[nH]1)=O 11393,C(C(C)(O)CC(=O)NCC(C1CCC1)NC(=O)CC1CSC1)OC.C(=O)(C(C)C)N 11394,N1(C(CNC(CCC(C)C)=O)=O)Cc2ccnn2CC(NC(C2CC=CC2)=O)C1 11395,Cn1nc(C(F)(F)F)c(C(=O)NCC2CN(C(C3CC3CF)=O)CCO2)c1C#N 11396,C1(CNC(C2(COC)CCCC2)=O)CC(C)(C)CN1C(=O)C1CC1 11397,c1(C(=O)NCC(CCCC)NC(=O)C2=CCCC2(C)C)ccc(Cl)c(C)c1N 11398,C(=O)(CCC(C)(C)ONC(=O)CCOCCNC(C1(F)CC=CC1)=O)OC 11399,S(=O)(=O)(c1cccc(F)c1C)N1CCN(CC(=O)Nc2ccnc(C)n2)C(=O)C1 11400,C(CCCCCC(=O)N(c1csnc1C)C)NC(C(OC)OC)=O 11401,C1(NC(C(=O)NC2CCCN(C3CCOCC3)C2)=O)CCNC2(CC2)C1 11402,CN1CCCC1C(N1CC(c2cc(C(F)(F)F)on2)C1)=O 11403,c1(C2(C(N(C3CN(C(=O)CCc4cn(C)cn4)C3)C)=O)CC2)ncccc1F 11404,C1(C(C)C(=O)N(C2(C(=O)NC(C)C(=O)NC3CC3)CC2)C)CCC(=O)N1 11405,c1(OC)ncc(Cl)cc1C(=O)NC1CCN(C(=O)C(C)C(F)F)C1 11406,C#Cc1cccc(N(C)CCO)c1.c1(C(c2ccccc2)=O)cccc(C)c1C 11407,N1(C(CCCCOC)=O)CCN(C(=O)C=C2CCSCC2)CC(CO)C1 11408,C#Cc1cc(COC(=O)Cc2ccc(C=O)[nH]2)cc(C(F)(F)F)c1 11409,c1(C(=O)NCCc2ccoc2)ccsc1SCCO 11410,c1(NC(C(C)Nc2ccc(C)nc2)=O)cc(Cl)ccc1C 11411,CN1C(=O)CSC1=CC(=O)NC1CCC(C(=O)Nc2ccccc2N(C)C)OC1 11412,N1(C(Cc2cc(OC)no2)=O)CCC(C2CC2)(CNC(=O)CC2CCC3CC23)C1 11413,c1(OCC)ccccc1NC(=O)C(N1CCC(C)(CNC(C2CC(C)C2)=O)C1)=O 11414,N1(C(CC2N(C)CC=CC2)=O)CC2(CCCC2NC(c2ccc(=N)[nH]n2)=O)C1 11415,c1(NCCC2(CC)CC2)ccc(S(=O)(=O)N)cc1F.C1(C)(NC=O)CCOC1 11416,C(=O)(C(CC)C(=O)OCC)N(CCN(C(c1nccc(CC)c1)=O)C)C 11417,CC1=C(C(=O)NCCCCNC(=O)CN2CCCCC2=O)Cc2ccccc2O1 11418,C12(C)CN(C1)CC(=O)C(=O)N2.c1(CC)cnc(CN)o1.C(C)(C(C)N)(C1CC1)OC 11419,N1(C(COCc2c(C)ncs2)=O)CC2(NC(C3CCC(=O)N3)=O)CC1C2 11420,c1(C(C(=O)NCCC2(NC(C3CC34CCC4)=O)CC2)(F)F)ccccc1F 11421,c1(CNC(C2CC(CNCc3cccc(C(N)=O)c3)C2)=O)c(I)ccnc1Cl 11422,C1(C(=O)NCC(C)(C)N(C)C)CN(C(=O)C(O)CN2CCCC2)CCC1(C)C 11423,N1(C(COCCCOC)=O)CCOCC1CNC(c1conc1C(C)C)=O 11424,C12(C(=O)NCC(CC(=O)OC)C)CCC(CN(C(=O)CCCNC(C)=O)C1)C2 11425,N1(C(C=CCCC=C(C)C)=O)CCOC(CNC(=O)C(C)(C)c2ccccc2)C1 11426,n1(CC=C)cc(C(=O)NCCN(C(c2cn(CC)nn2)=O)CC)nn1 11427,CCC(C(C)(C)C)NC(C1CCOCC1NC(c1ccc(C)cn1)=O)=O 11428,c1(SC)ccc(CC(=O)NC(CO)C(C)NC(C2CCCC2(F)F)=O)cc1 11429,CCC(C)CC(C(=O)NCc1cccnc1)NC(c1cc(C(C)=O)[nH]n1)=O 11430,N1(C(C2(C)CC(=C)C2)=O)CCC(CCCNC(C23CCCC2C3)=O)CC1 11431,N1(C(C(C)(F)F)=O)CCCC2(C1)CN(C(c1ccnc(-c3ccccn3)c1)=O)C2 11432,C(C)(C)(CCCC(=O)N1CC(CC(C)(C)C)C1)NC(c1cc(COC)on1)=O 11433,CCC(C(F)(F)F)NC(=O)C(=O)N(C1CCC1)C 11434,N#CC1CCCCC(n2cc(CS(=O)(=O)CC(O)CN3CCOCC3)nn2)C1 11435,c1(OC)ccc2ccc(C(=O)NC3CCCSC3)nc2c1Br 11436,CC1CN(C(C2(C)CCCO2)=O)CCCN1C(c1cc(Cl)ccn1)=O 11437,C1(C(=O)NC(CC=C)C2CC2)(CO)CCN(C(c2cc(OC)cnn2)=O)C1 11438,C(=O)(C(C)(CC)C(F)F)NC(CN(C(c1coc(C)n1)=O)CC)C 11439,C1(C2(O)CCC2)(C(=O)NCC(c2ccccc2)NC(c2ccc(C#C)o2)=O)CC1 11440,Cc1cc(C(=O)NC2CCCC(NC(c3ccsn3)=O)C2)ncc1S(N)(=O)=O 11441,C1(C(N(C(c2c(Br)cnn2C)=O)Cc2ccccc2)=O)CC(C)CN1CC 11442,N1(C(CNC(CCC(C)C)=O)=O)CCC2(CC1)CCN(C(C1CNC(=O)CC1C)=O)C2 11443,CC1(C)CCc2c1n[nH]c2C(=O)NC1CCSC12CN(C(=O)C1CC1)C2 11444,N1(C(Cn2cc(C(=O)NC)nn2)=O)C2CCCC1CC(NC(C1CCOC1)=O)C2 11445,N1(C(=O)Nc2c(F)cccc2Cl)CC2CCC1C(CO)C2.C123CC(C1)(C2)C(=O)N3 11446,c1(C(=O)NCC2N(C(CCCCC)=O)CC(OC)C2)cc2c(C)cccc2[nH]1 11447,Cc1nc(C#N)c(NC(=O)NC(C)(CNCc2ccccc2)C2CC2)nc1Cl 11448,N1(C(C(CO)NC(N)=O)=O)CCC(F)(C(=O)NCc2ccccc2F)C1 11449,N1(C(C(CNC(c2cncc(CC)c2)=O)CC2CC2)=O)CCCCCC1C 11450,C1(OC)CC(CNC(c2csc(F)c2)=O)(NC(=O)CC(C)C2CCCC2)C1 11451,c1(CC)cc(C(=O)NCCCn2cc(CCCCCCC3CC3)nn2)c(C)nn1 11452,CCC(CC)(CCNC(=O)Cc1c(C)nn(C)c1C)NC(c1cccs1)=O 11453,N12CCC(C(F)C1)C2=O.C(=O)(C1=CCCC1C)NC1C(c2ccc(C)s2)C1 11454,c1(C(N(c2ccc(Br)cc2)C(C)C)=O)cc(Br)c2[nH]c(=N)sc2c1 11455,N1(C(CCC#C)=O)CCC(F)CC1C(N1C(CO)CC1CO)=O 11456,C1(C(N(C2CCCN(C(c3ccc(C(C)=O)[nH]3)=O)C2)CC)=O)CC(=O)N(O)C1 11457,C1(CC)(CO)CCCN1C(C1CC1CNC(=O)C=CC1CC1)=O 11458,C(=O)(C1Cc2ccccc21)N(C)CC1N(C(CCC=C=C)=O)CCOC1 11459,C1(C(=O)NC(C)CF)CN(C(c2cncc(N(C)C)c2)=O)CCC1(F)F 11460,N1(C(c2n[nH]c3c2CN(C(C2C(C)CCO2)=O)C3)=O)CCC2CN(C)CC12 11461,C1(OC)CN(C(=O)C=CC2CCCC2)CC1NC(C1CCN1S(C)(=O)=O)=O 11462,c1(CN(C(C2CC(CNC(=O)CCCc3ncco3)C2)=O)CC)cccnc1 11463,c1(C(N2C3(CNC(C=CCC)=O)CCC2CC3)=O)ccc(Br)c(F)c1C 11464,C#Cc1ccc(C(=O)NC2(C(=O)NC(c3ncn(C)n3)C)CCSC2)cc1 11465,C1(COC)(CNC(c2nocc2C)=O)CCN(C(C2CCC(C)(C)C2)=O)C1 11466,C#Cc1cc(C(=O)NC2(C)CCC(NC(=O)CC3C=CCC3)CC2)cc(Cl)c1 11467,n1(CC(CC)CC)nc(-c2ccc(C(C)C)cc2)nc1C1CCC(=O)N1C1CC1 11468,C(=O)(C(F)C(C)(C)O)N(CCNC(=O)CSCCC#N)CC 11469,C12(CNC(C(C)SC)=O)CCCC(CN1C(=O)CCc1nc(C)c(C)o1)C2 11470,c1(C(=O)OC)sc(C(N2CC=CC(NC(C3(OC)CCCOC3)=O)C2)=O)cc1N 11471,Cc1cc(Br)cc(C)c1NNC(=O)CNc1ccnc(C(N)=O)c1 11472,c1(C(=O)NC2CCCN(C(C3C(CC)CCO3)=O)C2)cncc(C)c1O 11473,Cc1cccc(F)c1C(N1CCC(C)(CNC(=O)CC(F)(F)Cl)CC1)=O 11474,N1(C(CC(C)(C)O)=O)CCC(NC(=O)CCNC(=O)CO)C(F)C1 11475,C1(C(N(CCOC)CCNC(c2coc(C3CC3)n2)=O)=O)CC2OC(C)(C)OC2C1 11476,C1(CNC(=O)NC(Cc2ccc(Cl)nc2)C(=O)O)CCC2(CC1)OCCO2 11477,c1(CC)cc(C(=O)N(CCCNC(=O)CC2CCC(C)C2)C)no1 11478,S(=O)(=O)(c1ccc(NCCc2nc(C)oc2C)cc1Br)NCC(CCCCC)O 11479,C1(CCNC(=O)CCF)(NC(CC2CN(C)C2)=O)CCCC1 11480,C1(CN(C(=O)CS(N)(=O)=O)CCCNC(CC)=O)CCCCC1.N(C)C 11481,c1(C(=O)NCC(CN(C(c2c(CC)nc(C)o2)=O)C)O)cccc(F)c1C 11482,c1(OC)cc(C(=O)N(CCC(C)NC(=O)C(O)Cc2cn(C)cn2)C)[nH]n1 11483,c1(C(=O)NC2COCCN(C(c3cc(Br)ncc3Cl)=O)C2)cc(O)c(Br)c(O)c1 11484,CCCCC(O)CC(=O)N(C1CCCC1)CCCNC(c1cncc(C)c1)=O 11485,c1(OC)c(F)cc(C(=O)NC23CC(C(=O)NCc4nn[nH]n4)(C2)C3)cc1F 11486,C1(N2CCN(CCOC)CC2)COC2(CCN(C(C3CCCO3)=O)CC2)C1 11487,N1(C(CC(=O)OCC)=O)CCC2(C=C(C(=O)N3CCOC(C)CC3)C2)C1 11488,C1(N=[N+]=[N-])(C(=O)NC(CCSC)C)CCN(C(c2oc(C)nc2C)=O)C1 11489,C1(OC)CCCCCCC1OC(c1cnc(-c2nccs2)nc1O)=O 11490,c1(CC)nc(C)c(C(=O)NCCN(C(=O)C(C)C2CCC2)Cc2ccccc2)s1 11491,C1(CC)CC(C(=O)NC(CNC(=O)CC2CCOC2(C)C)C(C)(C)C)CCO1 11492,Cc1cnc(C(N2CC(CNC(c3cc(Cl)cnn3)=O)CC2C)=O)cc1Cl 11493,N1(C(c2ccnc(OC)n2)=O)CCCC2C1CCCN2C(=O)Cc1cc(C)ns1 11494,CCCC(CCC)C(C)NS(=O)(=O)Cc1ccc(F)cc1Cl 11495,N1(C(CN(C)C2CC2)=O)CCCC(O)(CNC(c2ccnnc2O)=O)C1 11496,c1(C(=O)N(C2CC2C(=O)NC(C(O)CO)C2CC2)C2CC2)occc1C1CC1 11497,C1(C)(C(=O)NCC2C(C(N(CC(=O)NC(C)C)C)=O)CCO2)CCC(=O)CC1 11498,N1(CCC)CC(C(=O)NCCCCCCNC(c2ccsc2C)=O)CC1=O 11499,CC1CN(C(C2CC2CF)=O)CC1NC(C1CCC(N2CCCC2=O)CC1)=O 11500,C(=O)(CC1CCCc2ccc(C(=O)N(C)Cc3ccc(C(C)(C)C)o3)cc21)OC 11501,C(C)(CCCCNC(C1CCCC1(F)F)=O)NC(Cn1ccc(C(=O)OC)n1)=O 11502,N1(Cc2c(OC)cccc2)CC(C(=O)Nc2ncc(C(C)=O)cc2C)CC(F)C1 11503,CN1CCN(C(=O)CSc2nnc(S)s2)CC1CNC(=O)C=CCCCC1CC1 11504,N1(C(c2c(COC)cco2)=O)CCCC(F)(C(=O)N(CC)Cc2nc(C)cs2)C1 11505,CC(C(C)(C)NC(c1ccnn1C(C)(C)C)=O)NC(c1cnn(C(F)(F)F)c1)=O 11506,C(CC1=CCN(C(=O)C(N2CCCCCC2)C)CC1)NC(C=CC=CCC)=O 11507,C1(CNC(CC2CCC(=O)NC2)=O)(NC(c2csnn2)=O)CC2CCC1CC2 11508,c1(CC(=O)NCC2C(C)CCCN2C(c2ccoc2)=O)c[nH]c2cnccc12 11509,N1(C(c2c(C)scc2)=O)CC2CC2(NC(=O)CCc2cncc(O)c2)C1 11510,C1(CNC(c2nc(CC)[nH]n2)=O)CCC(CNC(=O)CCc2cccs2)CC1 11511,C12(C(N(C)CC3CCN(C(C4C(C)(C)OC4(C)C)=O)C3)=O)CCCC(C)(C1)OC2 11512,C1(O)(C(=O)NCC2C3CN(c4nccc(C(C)=O)n4)CC32)CCCC(C)(C)CC1 11513,O(NC(=O)CC1(CNC(=O)CN(C(C)C)C(C)C)CC1)CC(C)C 11514,Cc1cn2c(CC(=O)NC(C)C(C)(C)NC(C3CCCCC(=O)N3)=O)csc2n1 11515,N1(C(c2ccc(CC)nc2)=O)CCCC(NC(=O)C(C(C)C)SCC)C1CC 11516,c1(NC(C2CCC(OCC(C)(C)C)CC2)=O)cnc2ncccn12 11517,Cc1ccc2ccccc2c1OC(C1C2CCCCC12)=O 11518,C1(NC(C2CN(C(C)=O)C2)=O)CN(C(C2(C)CC2(C)C)=O)CC1c1ccnn1C 11519,c1(C(=O)NCCC2CSCCN2C(=O)CC2CCOC2)cccc(C2CC2)c1F 11520,c1(C(=O)Nc2c(C)nc(C#N)cc2)n[nH]c2cc(COC(C)(C)C)ccc12.C=O 11521,Cc1ccnc(C)c1CNC(c1coc(CNC(C2C=CCCC2)=O)c1)=O 11522,C(C(C)CC(=O)NC1CC(NC(c2coc(-c3ccccc3C)n2)=O)C1)OC 11523,c1(C(=O)NC(C)CC2CCCCC2)cccc(N2CCOCC2)c1 11524,N1(C(C2CC2[N+](=O)[O-])=O)CCC(C(C)NC(=O)C=CC(c2ccccc2)=O)CC1 11525,c1(C(=O)NCC(CCCC)NC(=O)C(F)C2CCC2)cnc2c(C)cccc2c1 11526,N1(C(Cc2nc(C)[nH]n2)=O)CCC2CCCC12CNC(c1ccc(F)s1)=O 11527,N1(S(=O)(=O)c2ccc(NCCc3ccns3)nc2)C2CCC1c1ccccc12 11528,C1(F)(C(N(CCO)CC)=O)CCN(C(=O)C(C2(O)CCCC2)F)C1 11529,c1(=O)nc2nc([nH]1)NN2C.c1(C(C)OC(C)(C)C)cc(Cl)nc(Cl)c1 11530,C1(NC(C2CCCCC2)=O)CC2(C1)CC(NCc1cc(Cl)c(Cl)cn1)C2 11531,N1(c2cc(C)[nH]c(=NCC3(C(N)=O)CC3)n2)CC2(C)CN(C)CC2(C)C1 11532,C1(CN(C)C(c2cnc(O)n2C)=O)CCC(NC(c2ncoc2Br)=O)CC1 11533,C1(NC(c2cccc(OC(F)F)c2)=O)CCN(C(C23C=CC(CC2)C3)=O)CC1 11534,C1(C(=O)NCCN(C(=O)OC)C)COCCC1NC(c1ccccc1C)=O 11535,N1(C(C=CC)=O)C(CNC(=O)C(c2ccc(Br)cc2)OC)CC2CCCC12 11536,C#Cc1cc(F)c(C(=O)NC2CN(C(=O)CN(C)CC)CC2(C)C)c(F)c1 11537,C(=O)(C1CCCc2sccc21)NCC(CCOC)NC(=O)CCn1ccc(C)n1 11538,Cc1cncc(CC(N2CC=CC2C(=O)NC2C(C)CCC2C)=O)c1 11539,C(C(CC(=O)NCC1CCC1NC(c1cccc(=O)o1)=O)CC(C)C)NC(C)=O 11540,C1(c2nnnn2C2CCCC2)CCCC(=O)N1.c1(CC)cc[nH]c1C(=O)OC 11541,N1(C(c2c(C)ocn2)=O)CCN(C(=O)C(C2CCOCC2)F)CC1C(C)(C)C 11542,c1(OC)cc(C(C(=O)NCC2CC2)N(CC(C)C#N)C)c(F)cn1 11543,N1(Cc2cn(CC)nc2)CCCC2(CCN(C(c3cc([N+](=O)[O-])cs3)=O)C2)C1 11544,C(C)(C(CC(=O)NCC1CC(SC)C1)NC(=O)C(C)NC=O)OC 11545,C12(CNC(C=CC=CC)=O)CCCC1N(C(c1nonc1CC)=O)CC2 11546,c1(N2CC3CCN(C)CC3C2)nc(=NCC2CCC2)[nH]c2cccnc12 11547,CC1(C2(C)CC2C(N2CCCCC2Cn2cccn2)=O)CC1 11548,C12(NC(=O)CC=CCNC(=O)C(O)c3ccsc3)CC(CO)(C1)C2 11549,CC(C)(CCNC(=O)C=C(Cl)Cl)NC(=O)CCNC(N)=O 11550,c1(C(N2C(CNC(c3cnc[nH]3)=O)CCCC2)=O)cc2ccc(Cl)cc2c(=O)o1 11551,C1(COC(=O)CCOC2CCCCC2)CC2(CCC2)CN1C(=O)C1=COCCC1 11552,C(=O)(CCCCCNC(C1CC2CC2N1Cc1sccc1Cl)=O)OC 11553,c1(NC(CCC=C)C)[nH]c(=NC(C)c2ccncc2)nc2c1ncn2CC 11554,Cc1nn(C)c(C(=O)NCC(C)NC(C2CC2c2cnn(CCO)c2)=O)c1Cl 11555,N1(C(C(COCC)n2cc(CN(C(C)=O)CC)nn2)=O)CCC(C(C)(F)F)CC1 11556,c1(OC)cnc(C(F)(F)F)cc1C(=O)OC(C)(C)C.C12CC13CC(C3)CN2C=O 11557,c1(C(N2CC(NC(CCN(CCCCC)CC)=O)C(C)C2)=O)cc(=O)cc(Cl)[nH]1 11558,c1(OC)nccc(C(N2CCN(C(=O)C(Cl)=CCl)C(CS(C)(=O)=O)C2)=O)c1F 11559,CC(C)CC(C(=O)N1CCCC1C(C)(C)C)ONC(c1cnon1)=O 11560,c1(CC)c(C(=O)NCC2(NC(=O)SC)CC2)cnn1-c1ccc(OC)cc1 11561,N1(C(CC2N(C)CCOC2)=O)CCC2CN(C(c3nnn(C)c3N)=O)CC2CC1 11562,Cn1nc(Cl)cc1C(=O)NCC1(CNC(C2CC(F)C2)=O)CCCCC1 11563,C1(C)(NC(Cc2n(C)ccn2)=O)CCCN(C(c2c(Cl)n[nH]c2C2CC2)=O)C1 11564,c1(C(=O)NCCC(C(=O)N(C)CCc2noc(C)n2)OC)ccc(F)c(F)c1 11565,Cc1ccc(C(N2CCC(NC(c3ccns3)=O)CC2C)=O)cc1OC(F)F 11566,CC1(C)CC(=O)OC1CNC(C1C=CCN(C(C2CCSCC2)=O)C1)=O 11567,C(CC(O)CC(=O)NC1C=CCN(C(=O)C(C(C)C)NC(C)=O)C1)SC 11568,c1(C(=O)NCC2C(NC(C3OCCN(CC)C3)=O)C2)ccc(Cl)c2ncccc12 11569,C1(C(=O)NC2C(O)CCN(C(CCNC(=O)NC)=O)C2)CC2CCCCCC12 11570,CCC(C(=O)NC1(C)CC(NC(=O)CCC2CCCOC2)C1)N(CC)CC 11571,Cc1[nH]c(C(=O)NC(c2ccc(F)cc2F)C)c(C)c1C(=O)NCC1CCCO1 11572,N1(C(CC2(C)CC2)=O)CC(C)(C)OCC1Cc1sccc1NCS(C)(=O)=O 11573,N1(S(c2cnc(C(C)=O)s2)(=O)=O)CCC2C1CCCN2C(c1ccsn1)=O 11574,c1(CC)ncc(C(=O)NC2CC(C)CN(C(c3ccn(C4CC4)n3)=O)C2)c(O)n1 11575,N1(C(C=CCNC(C2CCOC2C2CC2)=O)=O)CCCC2CCCCC12 11576,N1(CCNC(c2ccc(S(N)(=O)=O)cc2)C)CCC2(C1)NC(=O)N(C)C2=O 11577,c1(SC)ccc(C(=O)NCCC(C)NC(C2CCN2C2CCCC2)=O)cc1 11578,C1(CC(N2CC(CCNC(c3[nH]c(C)nc3C)=O)(OC)C2)=O)CCCNC(=O)C1 11579,Nc1cc(Cl)nc(Cl)c1C(N1CC2CCN(C(C3CC3(F)F)=O)C2C1)=O 11580,Cc1ccc(C=CC(=O)NC(C2(O)CN(C(c3cnc(Cl)[nH]3)=O)C2)C)cc1Cl 11581,C1(O)(CNC(CC(CC)c2ccccc2)=O)CCN(C(c2ccc(=N)[nH]n2)=O)CC1 11582,C(=O)(C1CCc2ccccc21)N1CC2C(C(=O)NC(CC=C)C)(CCC2)C1 11583,C(=O)(CCCCc1cnc[nH]1)NCC1C(NC(C(CC)O)=O)C1 11584,c1(C(c2nnnn2C)NCC2(OC)CC2)cc(Cl)nc(Cl)c1 11585,C1(OC)CCc2nncn2C1.c12ncnc(c1C)C1CCN2CC1 11586,C1(CC=C)(C(=O)NC(C)CCC(=O)OC)CCN(C(=O)C=C(C)C(C)(C)C)C1 11587,C1(C(N(C(CCOC(=O)OCC)=O)C)C2CC2)CCc2nc(C(F)(F)F)cn2C1 11588,N1(C(c2cnc(CC)o2)=O)CCC2CC12C(=O)NCC(CC)CC 11589,CCC(CC)C(CCNC(c1nnnn1C1CCOC1)c1cn[nH]c1)OC 11590,C(C)(CCC(F)(F)F)(c1n(C)nnn1)NC1(C(=O)O)CC=CC1 11591,c1(C(=O)NC2CC(NC(c3c[nH]c(=NC)s3)=O)C2)cccc(S(=O)(=O)C(F)F)c1 11592,C1(C)(NC(C=CC(C)NC(COC)=O)=O)CCC(C)=C(C)C1 11593,O=CN1CCOCC1C(=O)NCC1(NC(c2cnn[nH]2)=O)CCCC1 11594,c1(C2C(C(N(CCC(=O)NC(c3nncn3C)C)CC)=O)C2)ccc(F)cc1 11595,C(CCCCCCCCCCCO)NC(=O)N(C1CCCC1)CCc1cccs1 11596,C=CC1CN(C(c2n[nH]c(C)c2C)=O)CC1NC(c1ncoc1C1CC1)=O 11597,c1(C(=O)NC2(CCCNC(C(C)n3cnnn3)=O)CC2)ccc(Br)nc1N 11598,N1(S(CC)(=O)=O)CCC(C(=O)NC(C)CCN(C(=O)CN(C)C(C)=O)C)CC1 11599,N#CC1(CC(N2CCCCCC2CNC(=O)C(F)n2cccn2)=O)CCOCC1 11600,CC1(C)CN(C(c2ccc(C#N)o2)=O)CC(CNC(C2CC3C=CC2C3)=O)O1 11601,C(CN(C)N1CCC(NC(=O)NCc2ccco2)CC1)SC 11602,c1(C(N(C2CCNCC23CC3)Cc2ccc(C)s2)=O)ccc(Br)cc1S(C)(=O)=O 11603,N1(C(c2c(CC)occ2)=O)C2CCC1CN(C(C1(CC(=O)OC)CCC1)=O)CC2 11604,c1(CC(=O)NCC(C)CNC(C2CCN2S(C)(=O)=O)=O)ccncc1Cl 11605,c1(CC2(C(=O)NCC(C)N(C(=O)CN(C)C)C)CC2)ccc(Cl)s1 11606,O=C1Nc2ccc(C(=O)NC3(CNC(=O)C4=CC5(CCOC5)C4)CC3)cc2C1=O 11607,C(=O)(C(F)C1=CCCCC1)N1CC(C)N(C(=O)C=Cc2cncnc2O)CCC1 11608,CC(C)CCCCCC(=O)N1CC2CC1C2NC(c1cncc(CN(C)C)c1)=O 11609,C(=O)(CCCCCn1cnnn1)NC(C)(C)CCCNC(=O)CCC1CC1(C)C 11610,c1(C(N2C(CNC(c3cn(CC)nc3)=O)CCC2)=O)cc(Cl)ccc1OC 11611,C(=O)(CC1=CCN(C(C2CC2C2CCCC2)=O)CC1)NC(CC=C)C(=O)OCC 11612,CCCCC(O)CC(=O)NCC1CN(C(=O)CNC(N)=O)CCCO1 11613,c1(CNC(C(C)=CC(C)(C)C)=O)cncc(C(=O)NC2(CCF)CC2)c1 11614,c1(C(N2CC(NC(c3cnc(O)o3)=O)C(O)C2)=O)cnc(O)c2cnccc12 11615,CC12CC(C(=O)NC3CN(C(c4ccc5cnnn5c4)=O)CC3F)(C1)C(C)(C)O2 11616,CCC(O)C(F)(F)C(=O)NCCN(C(c1cccc(S(C)=O)c1)=O)CC 11617,C(=O)(C1CCc2c(Cl)cccc21)NC1CC2(C(NC(c3cc(=N)[nH]cc3)=O)C2)C1 11618,c1(C(=O)NC2C3CCN(C(c4c(C)cc(C)s4)=O)C32)cc2c(Cl)cccn2n1 11619,CCC(C(=O)N(C1C2CN(C(=O)CN3CCN(C)C(=O)C3)CC12)C)C(C)(C)CC 11620,c1(OC)cccc(F)c1C(=O)NCCNC(c1ccc(-n2cnnn2)cc1)=O 11621,N1(CC(CSC)(C)C)CCC(C2CCCCC2)C1.c12ncnc(c1C)N2 11622,C1(c2scc(C)n2)CCC(C)N1C(=O)NCc1ccc(-c2noc(C)n2)cc1 11623,N1(C(c2c(C)coc2)=O)CC(NC(=O)C(F)(F)c2ccccc2)C(O)C1 11624,N1(C(=O)Nc2c(C)ncc(C)c2)CCC2(CC1)OC(C)(C)NC2=O 11625,C(=O)(CC(C)C(F)(F)F)N1CCC(NC(C(COC)(C)C)=O)C(O)C1 11626,c1(C(=O)NC2CN(C(C(C)C)=O)CC2C)cc2ccoc2cc1F 11627,C(N=c1cc[nH]c(=NCCCc2cccc(C)n2)[nH]1)c1c(CC)nn[nH]1 11628,c1(OC)cc(C)cc(C(=O)NCCOCCNC(C2(S(N)(=O)=O)CCCC2)=O)c1O 11629,C(=O)(CC(=O)NCCCN(C(=O)Cc1cnn(C)n1)C)OCC 11630,Cc1nc(C)c(C(N2CCN(C3CCCN(C(=O)C=CC(N)=O)C3)CC2)=O)[nH]1 11631,C1(NC(C(CO)OC)=O)CCOC(CNC(c2ccc(C(F)F)cc2)=O)C1 11632,C(CC1=CCN(C(C2CCCC23CCC3)=O)CC1)NC(C1CCC2CC2C1)=O 11633,N1(C(c2ccoc2C2CC2)=O)CC2(CCN(C(C3(c4cc[nH]n4)CC3)=O)C2)C1 11634,N1(c2ncc(CNC(=O)NCC)cn2)CCC2CC1(c1noc(C(C)C)n1)C2 11635,N1(Cc2cnc(C)nc2)CCN(C(c2cccc(C(F)(F)F)c2)=O)CC1C 11636,Cc1sc(Cl)c(C(N2CCN(C)C(CNC(=O)Cc3nc[nH]n3)C2)=O)c1C 11637,CCC(C)(C(=O)NCCC(Cc1ccccc1)NC(=O)C(CCSC)SC)OC 11638,N(C1CCNc2ccccc21)C(=O)CC1CCc2ccccc2C1 11639,c1(CC(=O)NC2(CO)CCN(C(C=C3CCC(C)C3)=O)C2)cccc(Cl)c1F 11640,Cc1ccc(=N)[nH]c1C(=O)NCC(CO)NC(C1CC(F)C1)=O 11641,C(CC(=O)N1CC(C(C)OC)C1)(CC(C)C)NC(C1ON=C(CC)C1)=O 11642,C(=O)(CC(F)(F)C(C)C)NCC(CCCC)NC(C1CCC(=O)N1C)=O 11643,CP(C)(=O)c1cncc(C(N2CCC3CN(C(c4ccc(=N)[nH]n4)=O)CC23)=O)c1 11644,c1(C(N(CCCN(C(CC2(COC)CCCC2)=O)C)C)=O)ccc(C)n(C)c1=O 11645,C(CCN=C(NC1CSC1(C)C)N1CCC(CC(F)(F)F)CC1)OC 11646,C(=O)(C(C)C(=O)N1CCOCC1)NCc1onc(CC(=O)NC)n1 11647,CC(C)C(C(=O)N(CC(O)CN(C(=O)C(C)Cc1ccccc1)C)C)NC(N)=O 11648,C1(C(=O)NCCNC(c2cc(O)nc(O)n2)=O)CCc2nnc(O)n2C1 11649,c1(CC(=O)NC(CNC(C(C)C#N)=O)CO)ccc(Br)cc1 11650,C1(C(=O)OCC)CC2(CC(NC(C3CCCN(CC(F)F)C3)C)C2)C1 11651,N1(C(c2cc(C)sc2)=O)CC2CC(NC(=O)C(C(C)C)n3cnnc3)CC(C2)C1 11652,c1(NC(=O)NC)cccc(C(=O)NCc2cc(Br)ncc2F)c1C 11653,c1(C(=O)NC2CN(C(C3(C)CCOC3)=O)CC2F)ccc(F)c(O)c1 11654,N1(CCNC(C(COC(C)C)(C)C)=O)CCCN(C(C2COCCN2C)=O)CC1 11655,c1(NC(N(C)Cc2ccc(C(C)(C)OC(F)F)cc2)=O)ccc(OC(F)F)c(F)c1 11656,C1(CNC(CC2(C(C)NC(=O)C=C3CCCCC3)CC2)=O)CC12CCOCC2 11657,c1(C(=O)NC(c2cn(C)nn2)C(=O)N(CC(F)Br)C)ncc(F)cn1 11658,N#Cc1ccc(F)c(CNC(=NCCCF)NCc2cnccn2)c1 11659,CCC(C(=O)NC1(CO)CN(C(C2CC2c2ccncc2)=O)C1)C(C)O 11660,c1(OC)ccc2c(c1C(=O)NC1CN(C(=O)CC=C(C)C)CC(F)(F)C1)CCC2 11661,C(=O)(C(O)CCCNC(C1(F)CCC1)=O)N1CC(OC)(CO)C1 11662,C(C(C(=O)N1CC(CNC(c2ncn(C)n2)=O)(COC)C1)OC)OC 11663,C1(CCOC)COCCN1C(C1(n2cc(CC(C(=O)O)SC)nn2)CC1)=O 11664,C(CC(C)P(C)(C)=O)NC(C(n1cc(-c2ccc(C)nc2)nn1)C)=O.N1CCCC1 11665,C=CCC(C(=C)C)C(=O)NC1CN(C(c2cc(F)c(Br)c(F)c2)=O)C1 11666,C=CC(C)CC(=O)N1CCCC1C1(NC(=O)Cc2csc(C(C)(C)C)n2)CC1 11667,C#CCC(CC(=O)N(CCC(=O)NC1CC1)CCOC)NC(=O)C=C(C)C 11668,c1(C(=O)NC(C(C)NC(c2cc(CCC)[nH]n2)=O)(C)C)c[nH]c2cc(F)ccc12 11669,N1(C(c2cc(C)c(Br)cn2)=O)CC2CCN(C(c3cccnc3N(C)C)=O)C2C1 11670,N1(C(c2cc(C)c(F)cn2)=O)CC(C(=O)NC(C2(O)CCC2)(C)C)CCC1(C)C 11671,C=CCCC(CO)NC(=O)CCC(C)NC(=O)CC=C 11672,c1(-c2ccc(CC)s2)ccc(CNC(C2(CC)CCOCC2)=O)cc1 11673,c1(CC(N2C(CCNC(C3CC3(F)F)=O)CCC2)=O)nsc2ccccc12 11674,Cc1ccccc1NC(C1(NC(c2cncc(N(C)C)c2)=O)CCOCC1)=O 11675,C1(O)(C(N(CCCN(C(C2CC(=C)C2)=O)C)C)=O)CCCC(C)(C)CC1 11676,N1(C(c2c(CC)noc2)=O)CC2(CCCC2NC(=O)C(c2ccccc2)C)C1 11677,CCCC(O)(C(=O)NC1CC1c1cccc(F)c1)C1CC1 11678,c1(C(=O)NCCCC2OCCN(C(C(CC)C)=O)C2)coc2c1COC2 11679,C=CCCC(C(=O)NC1(C)CC2CCC1C2)NC(=O)C(O)CC 11680,Cc1n[nH]c(C)c1CC(N1CC2C(NC(c3ccn(C4CC4)n3)=O)C2C1)=O 11681,Cc1cc(F)ccc1C(c1ccccc1)NC1(C)CCOC1=O 11682,CN=c1nc(C(=O)N(C2CCN(C(=O)C(C)N(C)C)C2)C)cc(C)[nH]1 11683,Cc1ccn2nc(C(=O)OC3CCN(N4CCNCC4)CC3)nc2n1 11684,C(C(=O)NCCN(CCOC)C(c1cccc(C(F)(F)F)c1)=O)(C(C)C)SC 11685,N1(C(CCCC2CCCCO2)=O)CC(OC2CCC2)C(O)C1 11686,C=CCC(CNC(=O)CC1COCC1O)NC(c1cnc[nH]1)=O 11687,N1(C(c2ccc(C)cc2C)=O)CC2CC(C)N(C(=O)C(F)CC3CC3)C2C1 11688,C1(C(N2C(CC(=O)NCCC(C)OC)CCCC2)=O)CC(C)(C)CN1C 11689,C1(NC(C)=O)CC(NC(=O)Cn2cc(C3CC3)cn2)C(O)C1 11690,C1(C(=O)NC(C2CCCCC2)C)CCN(C(=O)CCC2CCCC2)C1 11691,Cc1ccc(OCCC(=O)NCCCCN(C)C(C2CCCS2(=O)=O)=O)cc1C 11692,CN1CCOC2CN(C(C3CC(N(C(=O)CC4CCCOCC4)C)C3)=O)CC12 11693,c1(C(=O)NCC(c2ccc(C(C)C)cc2)NC(CC=C)=O)cccnc1C1CC1 11694,CCC(C)(C#N)C(=O)NCCCCCCNC(=O)C(O)CCN(C)C 11695,CC(CC(=O)NCC1CCC1NC(=O)C=CSCc1ccco1)C(F)(F)F 11696,c1(CC)ccc(C(=O)N(CCC(C)NC(=O)CC=CCc2ccccc2)C)cc1 11697,C1(F)(C(=O)NC(CC(=O)NC)C)CCN(C(c2cscn2)=O)C1 11698,c12nn(C)c(c1Cl)N(C)C2=O.C1(NC(C2C(C)C2)=O)CCN(C(=O)CC)CC1 11699,C(=O)(C1CNC(=O)c2ccccc21)N(C)CCNCc1ccc(F)c2cccnc12 11700,N1(C(C(C(C)(C)C)C2CCCC2)=O)CCCC(NC(=O)CCS(N)(=O)=O)CCC1 11701,N1(c2sc3c(n2)C(C)CCC3)CCC2(CCc3cc(Br)ccc32)C1 11702,CCS(=O)c1ccccc1CC(=O)NCC(OC)OC 11703,C1(C2N(C(c3c(C)csc3)=O)CCC2)CCN(C(C2CC(F)(CO)C2)=O)CC1 11704,C1(C(C)(C)O)(CNC(C2C(C(C)C)C2)=O)CN(C(C2(c3ccccc3)CC2)=O)C1 11705,c1(Oc2c(C(c3ccccc3)OC)c(C3CC3)on2)ccccc1C1CC1 11706,N1(C(Cn2c(C)cc(C)n2)=O)CCC2C(C1)CN2C(C12CC(C)C1C2)=O 11707,N1(C(C(CNC(CN(CCOC)C)=O)(C)C)=O)CCCC2OCCC2C1 11708,c1(CC(=O)NC2CC(NC(C(C)OCCC(C)C)=O)C2)ccc2[nH]ccc2c1 11709,N1(CC(=C(Cl)c2ccccc2F)C)c2ccc(Cl)cc2NC(=O)C1C 11710,N1(C(C2CC(CCNC(C3CC4(CCC4O)C3)=O)C2)=O)CCOCC2(CC2)C1 11711,c1(C(C)C)c(C(N2CCC(O)(CNC(c3cc(C(F)F)no3)=O)C2)=O)cnn1C 11712,c1(CC(=O)NCC(N(C)C(c2ccc(C(N)=O)s2)=O)C2CC2)ccc(O)nc1 11713,CC1CC(O)CCN(C(=O)C(C)N(C(c2cccc[n+]2[O-])=O)C2CC2)C1 11714,C12(C(CNC(c3n(CC)nnc3)=O)NC(c3ccc(CO)o3)=O)CCC(CC1)C2 11715,C1(NC(Cc2nc(C)sc2)=O)C2CC1N(C(=O)CSc1nncn1C(C)C)C2C 11716,C1(C(N(CC(CNC(C(=Cc2cnc[nH]2)C)=O)(C)C)C)=O)CC2(C1)CC1(CC1)C2 11717,C1(C(=O)N)CCC(C2CC2)C1.c1(CN)nc(CNC(C(=O)C(N(C)C)=O)=O)cc(O)n1 11718,c1(NC(c2n(CC)nnn2)C23CCCC2C3)ccc(OC(C)C)cc1 11719,CC1(C)CC(C(=O)NCC2CCCSC2)CN1C(c1cccnc1O)=O 11720,C(=O)(C(C)CC(C)(F)F)NCC(C1CCN(C(C(CC(C)C)O)=O)CC1)(C)C 11721,CC1CCOC1CNC(c1sccc1CNC(=O)CC1COC(=O)C1)=O 11722,c1(C(=O)NC23CCC(NC(c4c(CC)ncs4)=O)(CC2)C3)ccc2sccc2c1 11723,C(=O)(CCCCCO)NCC12N(C(C3C(OC)CCC3)=O)CC(C1)C2 11724,c1(C(N(C2CCN(C(c3cccnc3O)=O)C2)C)=O)ccc2nn[nH]c2c1O 11725,C1(C(=O)OCC)CCCC(Nc2c(C(N3CC(CC(C)(C)OC)C3)=O)scc2)C1 11726,c1(OC)cc(C(N2CC3(C2)CN(C(=O)C(O)CC2CCCC2)C3)=O)c(F)cn1 11727,c1(C(=O)NCC=CCNC(C2CN(CCC)C(=O)C2)=O)ccc(N)c(Cl)c1O 11728,C(CS(=O)(=O)CC(=O)N1CCC(C)N(C(c2n[nH]c(C)c2C)=O)CC1)OC 11729,c1(COC)cc(C(=O)NCCN(CC(C)O)C(c2ccn(CC(C)C)n2)=O)co1 11730,C1(C2CCC2)(C(=O)NCC(CN(C)C(c2ccn(C3CC3(F)F)n2)=O)O)CCC1 11731,C(CCCCC(=O)N1CCOC(C2(C)CC2)C1)NC(C(C(C)O)N(C)C)=O 11732,N1(C(C=CC(c2cccnc2)C)=O)CC2C(CNC(C3CN(C)CCO3)=O)C2C1 11733,N1(C(C=C(C)C)=O)CCCC1C(C)(C)C(=O)NCCC(F)(F)F 11734,C1(=O)C(C(C)C)N(C)CCN1.C(C)=CC 11735,CC12CN(C(c3c(O)cccc3F)=O)CC1(C)CN(C(=O)C1=CC3CCCC13)C2 11736,c1(C(N2C(C)(CNC(C(CCSC)O)=O)CCC2)=O)c[nH]c2cccnc2c1=O 11737,N1(C(c2cc(C)c(C)[nH]2)=O)CC(C2CCCCN(C(c3cnc(O)o3)=O)C2)C1 11738,Cc1ccc2cc(C(=O)NC(C)Cc3cc(Br)ccc3F)cnc2c1 11739,CC(C)(C)CN(CCO)C(C1(CNC(=O)CC2CC=CC2)CC1)=O 11740,C(=O)(CCCCCOC)N1CCC(NC)C1COC.C1=CC(=O)NC1(C)C 11741,N1(C(COCCC#C)=O)CCN(C(c2nnc(C)cc2O)=O)C2CCCCC2C1 11742,c1(CC)nc(=N)[nH]cc1C(N1CCCCCC1CNC(C1CNC(=O)N1C)=O)=O 11743,N1(C(C2(C)CCNC2=O)=O)CCCC(F)(CNC(=O)CP(C)(C)=O)C1 11744,c1(CC(N2CC(NC(C3C(CC)CCO3)=O)C2)=O)cc2ccccc2cc1O 11745,CC(C)CCCC(C)C(=O)N1CCC(CC(=O)NCCC2(CO)CC2)C1 11746,N1(C(CCSCC)=O)CCC(NC(C23CCC(CC2)CO3)=O)C(F)C1 11747,C1(CNC(C=C(C)C)=O)CCN(C(c2n[nH]c(C)c2C)=O)C1(C)C 11748,C(c1ccncc1)=C(C)C(=O)N(C1CCN(C(c2nc(Cl)cs2)=O)CC1)C 11749,c1(CC)cccc(S(=O)(=O)N2CCN(C(c3cc(C)c(Br)s3)=O)C(CC)C2)c1 11750,c1(C(=O)NCC2=CCN(C(C3CC3F)=O)CC2)cc(F)cc2nc[nH]c12 11751,c1(OC)ncnc(C)c1C(=O)NCC1CN(C(C2(OC)CCCC2)=O)CC1C 11752,C12(C(=O)NC3COCCN(C(=O)CC4CSC4)C3)CC=CCN1CCC2 11753,C1(C(=O)NC2CC(NC(CCSCC)=O)CC2O)CCN(C(=O)C2CC2)CC1 11754,c1(NC(C2C(C=C)C2)=O)cccc(C(F)(F)F)c1.C1(CC)CN(C)C(=O)C1=O 11755,C1(C(=O)N(C)CC2(CNC(c3ccc[n+]([O-])c3)=O)CC2)(OC)CCC(C)C1 11756,C1(C(=O)NC2CC(CNC(c3c(C)ncs3)=O)CC2O)CC12CCS(=O)(=O)CC2 11757,CC(C)CC(CO)N(C)C(C1C(C(C)C)CCN1C(=O)CN(CCO)CCOC)=O 11758,O(NC(=O)C(COCC)NC(=O)CCC1CCOCC1)CC(CC)C 11759,c1(C(=O)NCC=CCNC(C2(SC)COC2)=O)ccc(=O)n2c1CCCC2 11760,N1(C(CCN(C)C)=O)CC(C(=O)N(C2CCSC2)C)C(F)(F)C1 11761,Cc1ccc(C(=O)NCC(C)CC(=O)NC(c2ncccc2F)C)cc1O 11762,C(CC(=O)N1CCC(CNC(c2nc(Cl)c(Cl)s2)=O)C1)(C(F)(F)F)OC 11763,CC(C(O)C(F)F)NC(C1CC(OC2CC2)C1)=O.C12(CCCC1)CCC(=O)N2 11764,c1(C(N2CCN(C(C(CCC)=CCC)=O)C3C2C3)=O)ccc(S(N)(=O)=O)c(Cl)c1 11765,N1(C(CC(C)(C)OC)=O)CC2(CCC(CNC(=O)C(C)(C)c3cc[nH]n3)O2)C1 11766,C1(NC(C=CCC)=O)CN(C(c2c(C)ccn2C)=O)CC1O 11767,N1(C(CC2CN(C)C2)=O)CC2(CCN2C(C2CCCC3(CC3)C2)=O)C1 11768,N12CC3(CCC(CC3)C(=O)OC(=O)C(CC)C1=O)C2.C1(CC)CCCO1 11769,C1(NC(C(CO)NC(N)=O)=O)CCCN(Cc2ccccc2)C1 11770,CC1CN(CC(Cl)=CCl)CCC1N(C)C.C12(CCC1)C(=O)N2 11771,c1(C(=O)NCC2CCCN(c3nccc(CO)n3)C2)cnc(O)c(C(F)(F)F)c1 11772,C1(CN)CCN(CC(=O)NC2CCCC2)CC1.N12CCC(C1)C(=O)NCC2 11773,C(=O)(C1=CCN(C(c2cc[nH]n2)=O)C1)NC(c1ncc[nH]1)(C)C 11774,C(=O)(CC(C)(C)N(C)C(C1(C(C)(F)F)CC1)=O)N(CC(CN(C)C)O)C 11775,C1(O)(CC(=O)NC(C)CNc2cc(O)nc(O)n2)CCCN(C)C1 11776,c1(C(=O)NC2CN(C(c3ccc(C(N)=O)cc3)=O)C2)cc2n[nH]cc2cc1Cl 11777,c1(CC)nn(C)c(C(N2CCSC(C(N3CC(SC)C3)=O)C2)=O)c1Cl 11778,C(=O)(CCCN(C)C)N(CC(C)(C)Cn1cc(CCS(N)(=O)=O)nn1)C 11779,C(=O)(C1=CCN(C(C2(F)CCCC2)=O)C1)N(c1cnc(F)nc1)C 11780,N1(C(c2ccc3c(n2)NCC3)=O)CCCC2CN(C(C3CC(O)C3)=O)CCC12 11781,N1(C(C(C)OC)=O)CC(CNC(=O)C(c2ccc(C)cc2)C)C2(CCC2)C1 11782,Cc1cc(C(N2CC(NC(=O)C(F)F)C(F)C2)=O)c(C)n1-c1ccc(Br)cc1 11783,C1(NC(C(C=C)O)=O)CCC(CNC(=O)C(COC)SC)CC1 11784,C(CCCc1cccs1)(c1cccnc1)NC(C(n1cc(C2CCC2)nn1)C)=O 11785,CCC(O)CC(=O)NC(C)(C(=O)N(C)CC1CCCC2CC12)C1CCC1 11786,CCC(C)(O)C(=O)NCC1(F)CCC(CNC(=O)C=C(C)I)C1 11787,c1(C(N2CC(CC(=O)N(CCCCCC)CC)(OC)C2)=O)ncn2c1CCC2 11788,CCC1CC(=O)N(C)C2CCCCC2NCC(=O)N1C.C1(N(C)C)CCC1 11789,C1(NC(c2cnc(O)s2)=O)CCN(C(=O)CC2CC2C2CC2)C1C1CC1 11790,c1(CNC(=O)C(C2CCN(C(C3C4CCOCC34)=O)C2)F)cnccc1C1CC1 11791,c1(CC)cnc(C)nc1N1CCC(CF)(NC(c2cccc(F)c2)=O)C1 11792,N1(C(C(C)(C)OC)=O)CC2(CCCN(C(=O)CC3CCCC(=O)C3)C2)C1 11793,c1(C(=O)NCC(CNC(c2c(C)cc(C)nc2)=O)(C)C)ccc2nc(S)[nH]c2c1 11794,c1(CN(C)C)cccc(C(N2CC3CCC3C2)C(=O)NCC(F)F)c1 11795,c1(CC)cc(F)ccc1C(=O)NC(C)C(C)NC(C1(C2CC2)CC1)=O 11796,c1(C(N2CCCC(NC(C3(C#N)CC3(C)C)=O)C2)=O)cnc(CC(C)=O)nc1C 11797,CC1CCN(C(c2n[nH]cc2Cl)=O)C(CNC(c2cc(-c3ccco3)on2)=O)C1 11798,N1(C(=O)NC2CC3CCC2O3)CCc2sc(-c3cn(CC(O)CO)nn3)cc2C1 11799,N1(CC)CCC(C(=O)NC2CCCCC2CNC(c2cnsc2C)=O)CC1 11800,C(CN=C(NC(C)COC)NC1CC2(CC2)C1)OC 11801,N1(C(c2cc3c(s2)CCC3)=O)CCCN(C(=O)C(F)CC2CCC2)C(CO)C1 11802,N1(C(CNC(=O)NC)=O)CCC2C(CCCN2C(=O)CCn2cc(Br)cn2)C1 11803,C(CNC(c1ccccc1N(C)C)=O)(C(C)C(C)C)NC(Cc1cnc(C)s1)=O 11804,c1(C(=O)NCCCNC(C2CCC3CCC23)=O)nc2c(s1)COCC2 11805,C12CC3(C1)CC3C(=O)N2.N1(C(C(C)(C)N2CCCC2)=O)CCC(O)(C(F)(F)F)C1 11806,c1(C(N2CC(n3cc(CCNC(C)=O)nn3)C2)=O)cc(Cl)cn1C 11807,C(C(=O)NC1CCC1)(C(C)CC1CCC1)N(C1CCOC1)CC 11808,c1(C(=O)NC2C(NC(C(C)CN(C)C)=O)CCCC2)ccc2c(O)ncnc2c1 11809,CC1CCC(NC(=O)Cc2ccc(C(F)F)cc2)CN1C(C1CC(=O)C1)=O 11810,C#Cc1ccccc1CC(N1CCC2C(C(=O)NCCNC(N)=O)C2C1)=O 11811,Cc1cc(CC(N2CC3CC(C2)C3NC(=O)C(c2ccccc2)C)=O)ccc1Cl 11812,Cc1ncsc1CN(C(=O)CCn1cc(-c2ccccc2)nn1)CCO 11813,c1(C(=O)NC2CCCC(NC(c3ncc(C)c(Cl)c3)=O)C2)cc([N+](=O)[O-])cn1C 11814,n1(CC(N2CC(C(C)NC(Cc3c(C)n[nH]c3)=O)C2)=O)nc(C)n(C)c1=O 11815,C(=O)(CCCCCC#N)NCC(CN(C(C1CC12CCOCC2)=O)CC)(C)C 11816,c1(N(C(c2cncnc2)COC)CCO)cnc(C(C)(C)Cl)s1 11817,C1(NC(CSCC(=O)OCC(C)C)=O)CN(C(=O)CCOC(C)C)CCC1C 11818,N1(C(CSCC(C)C)=O)CC2CC(C1)CN(C(=O)C(C)C(C)n1cccn1)C2 11819,C1(C(=O)NC(CNC(C2(CC)CC2)=O)(CC)CC)Cc2ccccc2N1C(C)=O 11820,c1(CNC(=O)NC2(C(=O)O)C(C)C2)cc(Cl)cc(Br)c1 11821,N1(C(CCOC2CN(C(CCCC#C)=O)C2)=O)CCSCC(C)C1 11822,N1(C(c2cc(C)nc(O)c2)=O)CC(CNC(c2nccnc2Cl)=O)OC(C)(C)C1 11823,N1(C(C(C)(C)c2cnco2)=O)CCCC2(C1)CN(C(=O)Cn1ccnn1)C2 11824,Cc1nc(C(=O)NCC2C=CC(NC(=O)C(O)CC3CCOCC3)C2)sc1C 11825,N1(C(CCN(C(CCC)C)C)=O)CCOCC1CNC(C1CCCCCC1)=O 11826,Cc1ccccc1NC(C1COC(=O)C1)=O.N12CCOCC1CC(=O)NCC2=O 11827,N1(C(C2(CCC=C)CN(C(=O)C3=C(C)CCC3)C2)=O)CC2(C1)CC(C)(O)C2 11828,c1(CC)cccc(C(=O)N(CC(C)N(C)C(c2ccc(Br)cc2)=O)C)c1 11829,CCCC(C)CCNC(c1nnnn1CCCF)c1cn[nH]c1 11830,N1(C(C(c2cccnc2)NS(CC)(=O)=O)=O)CC(CN)C(C)C1 11831,Cc1c(F)cc(C(N2CC(NC(c3ccc(CO)cc3)=O)C(C#N)C2)=O)cc1Br 11832,N1(C(C2(CC=C)CCN(C(c3cc(OC)nn3C)=O)C2)=O)CCC(C2CCC2)C1 11833,Cc1ccc(=O)n(CC(N2CC(NC(c3cc(C(C)(C)C)n[nH]3)=O)CC2C)=O)n1 11834,N1(C(c2n(CC=C)ccn2)=O)CC(C2CCN(C(=O)C(C)(F)C(C)(C)F)CC2)C1 11835,CCCCCCC(F)C(=O)NCC(CC(C)C)NC(c1cc(CC)sn1)=O 11836,c1(C(N2C(C(=O)NC)CCC2)=O)ncc(Br)cc1Br 11837,N1(C(c2c(C)nc(OC)s2)=O)CC2CCCC2(NC(c2coc(C(C)C)n2)=O)C1 11838,C#CCCN=C1NCC=C2CN(C2)C(=O)CN1.c1(COC)cc(C(F)(F)F)n[nH]1 11839,C(=O)(C1=CC2CCCC12)NC1CC2(CN(C(c3c(SC)cc(C)cc3)=O)C2)C1 11840,CC(C)CC(=O)C(=O)NC(C)(C)CC=CC(N1CC(CO)CC(C)C1)=O 11841,C(CC(C(=O)N(C1CCNC1=O)C)NC(c1cccn1C)=O)OC 11842,Cc1c(C(=O)NCCn2cc(C(=O)NC(c3ncnn3C)C)nn2)ccn1C 11843,C1(C(N(CCN(C(CC2C(C)=NOC2=O)=O)C)C)=O)SC2C=CC1CC2 11844,n1(CC)nc(C(N2CC3CC3(NC(C3CCC(C(F)(F)F)CC3)=O)C2)=O)cc1O 11845,CCC(c1cccc(Cl)c1)=CC(=O)NC1CCC(NC(=O)CC23CC(C2)C3)CC1 11846,C(=O)(C(CC(C)(C)C)NC(C1CC(=O)N(C)C1)=O)NC1CCC(C)(OC)CC1 11847,C(CN=c1ccc(S(=O)(=O)N2CCCC(C)(F)C2)c[nH]1)c1cncc(OC)n1 11848,C1(CNC(c2c(OC)csc2)=O)CCCC2CN(C(=O)C=CS(C)=O)CC12 11849,N1(C(CSCC)=O)CCCC2(CCCN(C(c3[nH]ccc3C)=O)C2)C1 11850,C1(NC(c2c(CC)nn[nH]2)=O)CC=CCC1C(=O)NC(C(C)C)C1CC1 11851,C1(C(N(C(C)CNC(C2COCCN2CC(F)F)=O)C)=O)CCCCC1(C)C 11852,c1(C(C)NC2CC(CO)CN2)ccc(Cl)cc1 11853,C#CC(C)(C)C(=O)NC(C1CN(C(=O)C=CCN(CC(F)(F)F)C)C1)C 11854,c1(CC(C)C)c[nH]c(C(=O)NCCCCCNC(C2CC2c2cccnc2)=O)c1 11855,c1(C(=O)NC2(CNC(C3CC(CF)C3)=O)CC2)cc(=O)n(-c2ccccc2)[nH]1 11856,N1(C(c2c(C)ncnc2C)=O)CC2OCCN(C(C3CCCC4(CC4)C3)=O)C2C1 11857,Cc1cc(CN2CCC(C)(NC(c3cc(C)n(C)n3)=O)C2)c(C)s1 11858,N1(C(C(C)NC(CC)=O)=O)C2CCC1CN(C(c1c(C)nc(C)n1O)=O)C2 11859,Cn1cc(Br)cc1C(=O)NCC1CC1NC(c1cncnc1C1CC1)=O 11860,c1(C(=O)NC2CC(CNC(C(C)O)=O)C2)ncoc1C1CC1 11861,c1(C(=O)NCCN(c2[nH]cnc3nc(Cl)cc2-3)CCC)cc(F)cc2nn[nH]c12 11862,c1(CN(C(=O)C(N2CCOC(CC(F)F)C2)=O)C)ccc(SC(F)(F)F)cc1 11863,Cc1cc(F)cnc1C(N1CCCC1CCNC(C1(C(F)(F)F)CCC1)=O)=O 11864,N1(Cc2scc(CC(=O)OC(C)(C)C)n2)CCCN(C(C2C=CCC2)=O)CC1 11865,N1(C(=O)C2=CCCO2)CC2CCCN(C(C3C=CCCC3)=O)C2C1 11866,N1(C(C2(O)CCN(Cc3c(OCOC)cccn3)C2)=O)CCCC(S(C)(=O)=O)C1 11867,c1(CCC(N2CCCC(n3nnnc3CC3CC3)C2)=O)ncc(Br)cn1 11868,C(=O)(C1=CCCC1C)NCc1cc(C(=O)NCC(C)OCC=C)on1 11869,N1(C(CC(CCCC)O)=O)CCC2(CCN(C(c3cc[nH]n3)=O)CC2)C1 11870,c1(C(=O)NCCc2cncc(C)n2)cccc(Br)c1N 11871,C1(C(=O)NCCCC(=O)OC)CCCN(Cc2ccc(Cl)cc2C(F)(F)F)CC1 11872,N1(C(C(=O)N(C)C)=O)CCC2CCN(C(c3coc4ccccc34)=O)CC12 11873,CCC(C)(CNC(c1ccc(F)o1)=O)NC(=O)CN(C)CCO 11874,N1(Cc2sc(C)c(Br)c2)Cc2[nH][nH]c(=NC(=O)c3ccn4ccnc4n3)c2C1 11875,C(=O)(C(CC(F)F)c1ccccc1)NCC(CC=C)NC(=O)OC(C)(C)C 11876,C(=O)(C1CCCc2nccn21)Nc1cc(C)c(Br)cn1.C1(OC)CN2CCC12 11877,C(=O)(C1=C(F)CN(C(=O)CN(C)C)CC1)NC1CC2(CC(OC)C2)C1 11878,c1(CC(CC)C)nc(-c2cc(C(C)C)ncn2)n(CSc2ccccc2C)n1 11879,CC(Cc1ccc(Cl)cc1)CC(=O)N(CC(C)CNC(=O)Cc1cnccn1)C 11880,Cc1ccc(C(=O)NC2CC(NC(c3cc(F)cc(Cl)c3)=O)C2)c2ccccc12 11881,N1(C(C(CCC(C)(C)C)F)=O)CCCCC(C2CN(C(C3CCC(=O)N3)=O)C2)C1 11882,c1(C(N2CC(C)(CCNC(C3CNC(=O)C3)=O)C2)=O)ccc(Cl)cc1 11883,N1(C(c2nsnc2O)=O)CC2CCCC2(Nc2cc(O)ncn2)C1 11884,C1(F)(C(=O)NC(C(=O)O)C2CCCC2)CN(C(=O)OC(C)(C)C)CC1C1CC1 11885,CC1COc2c(C(=O)NC3CCC3CNC(c3cnc(Cl)s3)=O)cccc21 11886,C(=O)(CC(=O)NCC(C)(CO)NC(=O)CC(C)NC(N)=O)OC 11887,C12(NC(COC(CC)(C)C)=O)CCCCC1N(C(c1ccncc1NC)=O)CC2 11888,N1(C(C(CC)C(F)(F)F)=O)CCC(C2CCN(C(=O)CCn3cnnn3)CC2)C1 11889,c1(CC(N2CCN(CCNC(C(CO)N(C)C)=O)CC2)=O)ccc(F)cc1Cl 11890,CC1(C)CC(CNC(C2CC2F)=O)CN(C(=O)CN2CC3CC3C2)C1 11891,Cc1ccncc1C(=O)NCc1cn(CCNC(=O)Cc2ccns2)nn1 11892,C=CC(CC)CC(=O)N1CCN(CCCNC(C2(S(C)(=O)=O)CC2)=O)CC1 11893,N(C(=NCCCF)N1CCCC(S(C)(=O)=O)C1)C(C1CCCCC1)Cn1c(C)ncc1 11894,c1(NC(=O)CCc2ccc(C(N3CCSCC3)=O)[nH]2)cc(Br)cc(I)c1 11895,C1(CCNC(CC2(C)OCCO2)=O)CCCN(C(c2cnc(Cl)s2)=O)CC1 11896,c1(C(C(=O)NCCC2CCC(NC(c3cnns3)=O)C2)(F)F)ccc(F)cc1F 11897,C=CCC(CC)C(=O)N1CCN(C)C(C(=O)NC(c2c(C)n[nH]c2C)C)C1 11898,Cc1cncc(C(N2CC(NC(c3cc(-c4cnn(C)c4)[nH]n3)=O)C(F)C2)=O)n1 11899,c1(C(N(CCn2cc(CCOC)nn2)CC)=O)cccc2c1OC(C)(C)CC2 11900,c1(C(N2CCCC(CCNC(C(CC)CO)=O)C2)=O)ccc2nonc2c1 11901,C1(NC(=O)CC(=O)N(CC)CC)CCN(C(=O)CN(c2ccnc(Cl)n2)C)CC1 11902,c1(CNC(C2CC2F)=O)ccc(CNC(=O)Cn2cc(CO)nn2)cc1 11903,N1(C(C(C2CCCCC2)NC(C(=O)NC(C)C)=O)=O)CCS(=O)(=O)CC1 11904,C1(C(=O)NCC2CCN(C(C3CCOC3)=O)CC2(F)F)CCC2(CCCC2)CC1 11905,N1(C(CCCC#CC)=O)CCC2(CCC2NC(=O)CCc2nncn2C)CC1 11906,n1(CC)c(N(Cc2cccc(CO)c2)CC2CC2)nnc1-c1ncc[nH]1 11907,C1(CNC(C(C)NC(N)=O)=O)CCN(CC2(C#N)CCC2)C1 11908,N1(C(CC=C=C)=O)CCC(C2N(C(=O)C(C)NC(=O)C3CC3)CC2(C)C)CC1 11909,C(=O)(C1=C(C)CCCC1)NCC12N(C(C(CCCC)O)=O)C(CC1)CC2 11910,C#CC(C)(C)C(=O)NCC1CN(C(c2cn(C(F)F)cn2)=O)C2CC12 11911,c1(CC)oc2ccccc2c1C(=O)NC(C)CCCNC(C1CCCCS1)=O 11912,N1(CCC)CCc2cc(NC(C)CSCOC(C)C)ccc21 11913,C1(NC(c2c(SC)cn(C)n2)=O)CCN(C(c2cc(F)ccc2F)=O)C1(C)C 11914,CCCC(C(=O)N1CCC(N(C)C(c2ccc(O)c(F)c2F)=O)CC1)S(N)(=O)=O 11915,CC1OC2CCC1(C(N1CC(NC(c3cc(Cl)cs3)=O)C1)=O)C2 11916,c1(OC)ccc(C(=O)N(CC(N2CCCC2CO)=O)CC2CCOCC2)cn1 11917,C1(C#N)(C(=O)NCC(C)NC(C2CC(O)(C(F)(F)F)C2)=O)CCCOC1 11918,C(=O)(CCCCCC(C)(C)C)NCC(CNC(CN1CC(CC)C1)=O)O 11919,C#CCCCC(=O)NCc1ccc(N2CCN(C(=O)CSCCC)CC2)cc1 11920,C1(C(N2C(C(C)(C)NC(=O)CC3CCCC(O)C3)CCC2)=O)CC(S(C)(=O)=O)C1 11921,C12(C(=O)NC)CCCN(CC1)C2.C1(C(C(=O)CN)=O)CCCC1Cc1nc[nH]n1 11922,N1(C(=O)CC2CCCO2)CCN(C(c2cnc(O)o2)=O)C(c2ccccn2)C1 11923,C1(CNC(C2N(CC)CC2)=O)CN(C(=O)Cn2cc(C3CCC3)nn2)CCCO1 11924,c1(OCC=C)ccc(CCNC2CC(=O)N(c3ccccc3Cl)C2)cc1 11925,C1(C(=O)NC(C2(O)CN(C(Cc3cc(C)[nH]n3)=O)C2)C)CCc2nccn2C1 11926,C#CC(CNC(=O)CN(C(=O)C(F)C1CCCC1)CC(C)C)CC(C)(C)C 11927,C1(C(=O)NCC(C(C)C)NC(c2c(C)snc2)=O)CCCN(C(=O)C2CC2)C1 11928,C1(O)(CNC(CCN(CC(F)(F)F)C)=O)CCN(C(=O)C=C2CCCCC2)C1 11929,c1(OC)cc(C(=O)NC(C)C=CC(=O)NCC(=O)OCC2CC2)[nH]n1 11930,c1(CCCN2C(=O)CN(CC3CCCS3(=O)=O)C2=O)ccccc1[N+](=O)[O-] 11931,c1(N2CCC(C(C)NC(C=COCC)=O)C2)ncc2cccnc2n1 11932,N1(CC(c2ccc(OC)cc2)C)CCC(=O)N(Cc2cc(Br)c(F)cc2F)C1=O 11933,C1(NC(CC2ON=C(CC)C2)=O)CC2CCCC(C1)N2C(c1cccn1CC)=O 11934,c1(C(=O)NC2C(CN(C(C3=C(C)CC3)=O)C)CCC2)cc([N+](=O)[O-])n[nH]1 11935,N1(C(CC(C=C)(C)O)=O)CCC2(CC1)CN(C(=O)C=CBr)CC(C)O2 11936,N1(C(C=C(COC)C)=O)Cc2ccccc2CC1CN(CC(C)(C)C)C(=O)CO 11937,C1(C(=O)NCC2(OC)CN(C(C3CC=CCO3)=O)C2)C2(CCC2)C12CCC2 11938,c1(CN(C)C(c2ccon2)=O)ccccc1CNC(c1cc(Cl)ns1)=O 11939,N1(C(C=COCC)=O)CCCC(CN(C(=O)CCCCN2CCCCC2)C)C1 11940,c1(-c2cn(CC(=O)N(CCC)CCN(C)C)nn2)ccc(COC)nc1 11941,c1(CN=C(NC(c2sc(CC)c(C)c2)C)NC(C)CC)c(F)cc(F)c(F)c1F 11942,c1(C(=O)NC2CCN(C(C3CCN(C4COC4)C3)=O)C2)ccc2c(c1)NCC2 11943,N1(C(CCCCC=C)=O)Cc2ccnn2CC(NC(c2ccsc2)=O)C1 11944,N(C1CCc2cc(Br)ccc21)C(c1ccccc1S(=O)(=O)N1CCCCCC1)=O 11945,Cc1ccc(C)c(C(=O)NC2CCN(C(=O)CSc3ccncc3)CC2F)c1C 11946,c1(-c2nc(CO)nn2-c2ccccc2)ccc2ncccc2c1 11947,c1(OC)ccc2c(C(=O)NC(C3CCCCN3C(c3ccns3)=O)C)n[nH]c2c1 11948,C(CCCCC(=O)NC1COCCN(C)C1)NC(c1ccnc(C)n1)=O 11949,C1(N(C2CC(CCC)OCC2)C)CC2CCC(C1)N2C(C1CCOC(C)C1)=O 11950,O(N=C1CCCCCC1)CC(=O)NC1(COC)CN(C(C23CCCC2C3)=O)C1 11951,c1(CN(C(OCC(CCCC)CC)=S)c2ccccc2)ccc(S(=O)(=O)NC)cc1 11952,CC1(C)CC(CO)(CNC(=O)C(C)(C2CCC2)NC(C2CC2(C)C(F)F)=O)C1 11953,c1(OCC(N2C(CNC(C(C)SC)=O)C(C)CC2)=O)ncc(Cl)cc1Cl 11954,CC1(C(=O)NC2CCC(F)(F)C2O)C2Cc3ccccc3C12 11955,CC1(C)CC(CNC(=O)CC2CCC=CCC2)N(c2nc(C(F)(F)F)ns2)C1 11956,C(CCC(=O)NCC1(C(N2CC(CC)C2)=O)CC=CC1)=CCC=C 11957,C1(C(N2C(CNC(CSCC=C)=O)CC(C(F)(F)F)C2)=O)CCn2nnnc2C1 11958,CC(C)CC(F)C(=O)N1CC2CC1(CNC(c1csc3nnsc13)=O)C2 11959,c1(C(N(CC)CC2CCN(C(=O)C(=O)N(C)C)CC2)=O)cc2n(n1)C(C)CCC2 11960,c1(C[SH2]C2(N(C3CCCCC3)C(=O)NCC)CCC2)ccccc1 11961,CCCCC(O)C(=O)NC1CCN(C(=O)C(C)CSC(F)(F)F)CC1 11962,C(=O)(C(C)(C)C1=CCN(C(=O)C(C2CC2)C2CC2)C1)NCC(C(CC)C)CO 11963,n1(CC(=O)NCC(C)(CNC(=O)CCOC2CCCC2)OC)nc(C)nc1C 11964,O=C(C1=CC2(CCOC2)C1)NCC1CCN(C(c2cc(=O)cc(Cl)[nH]2)=O)C12CC2 11965,c1(N2CC(C(C)C)OCC2)nc(N2CCC(CO)CC2)nc2c1SCC2 11966,c12ccc(c3c1NC(=O)C3CC(CC(C)C)OC1CC1)C1=CC=CC=COC2C1C 11967,O=S(=O)(c1cc(Br)c(Br)s1)N1CC2CCCC2(C(F)(F)F)C1 11968,c1(C(=O)NC(CNC(C(CC#C)C)=O)CO)cc(N2CCCC2)cc(Cl)c1 11969,C1(N(C(CCc2ccc(C)s2)=O)C)Cc2cccc(C)c2C1 11970,c1(OCc2nnc(SCC(=C)Br)n2CC(CC)CC)ccc(Cl)cc1 11971,c1(OC)cc(C(=O)NC2CCC(C(=O)Nc3cnc(C)c(F)c3)OC2)ccc1O 11972,c1(C(=O)NC(CNC(C2(C#C)CC2)=O)CC(C)C)ccc(Cl)c(CCC)c1 11973,CC1CCN(C(=O)Cc2cc(Cl)cs2)CC1CNC(c1cnc(Cl)s1)=O 11974,S(=O)(=O)(c1ccc2c(c1)CCCO2)N(CC=C)Cc1cccc(Br)c1 11975,C1(NC(N(C(c2cccnc2)C)C)=O)(CF)CCN(C(=O)OC(C)(C)C)C1 11976,N1(C(=O)Nc2ccc(N=S(C)(C)=O)cc2)Cc2ccccc2C(C(=O)O)C1 11977,Cc1cc2sc(C(=O)NCC(C(C)C)NC(=O)C(C#N)C(C)C)cc2s1 11978,CC(C)(CNC(=O)CN(C(=O)CCNC=O)CCO)CCCO 11979,c1(OC)ccc(O)cc1NC(=O)CCC(C)NC(=O)C(C)(C)C(C)O 11980,CCC(O)(CC)CCNC(c1ccc(CNC(=O)C(C)C2CCCO2)s1)=O 11981,c1(C(N2CCC(NC(C(CC=C)C)=O)(CO)C2)=O)cccn2c(CO)nnc12 11982,C1(C(=O)OC)CCCCC1C(=O)NCCC1(O)CN(C(=O)C2=NOCC2)C1 11983,c1(C(N2CC(CNC(c3nc(C)nn3C)=O)C(C)C2)=O)cc(Cl)cc2c1CCC2 11984,C1(NC(C2CC3CCC2C3)=O)CCCC(CC(N2CCC(F)CC2)=O)C1 11985,CC(C)C(Br)C(=O)c1ccc(C2CCN(C)CC2)s1 11986,C1(c2n(C(CC)C)nnn2)(Nc2cnn(CC(C)C)c2C)CSC(C)(C)C1 11987,N1(C(c2c(N)cncc2)=O)CC2(CCCC2NC(=O)C(=O)Nc2ncc[nH]2)C1 11988,C(=O)(C(C)S(C)(=O)=O)NCC1(CNC(c2n[nH]c(C)c2Cl)=O)CC(F)(F)C1 11989,C12(NC(C(CC#CC)NC(=O)CCCCOCC)=O)CCC(CC1)C2(C)C 11990,c1(C(=O)NC(CN(C(c2ccc(OC)c(F)c2)=O)C)C)csc2c1CCC(C)C2 11991,c1(OCC(=O)OC)cccc(C(=O)NC(C2CCN(C(=O)CCC(C)C)C2)C)c1 11992,C(CC(C(=O)NC1CC1NC(=O)CC1CC(C(F)F)C1)c1ccccc1)=C(C)C 11993,c1(N2CCC(NC(=O)Cc3cccc(Cl)c3)C(O)C2)ncnc2ccc(O)cc12 11994,N1(C(c2cccc(NC)n2)=O)CCC(C)(C)C1C(=O)NOCCC(F)F 11995,c1(C(N2CCC(NC(c3nn(C)c(Cl)c3)=O)C2)=O)c(F)cncc1Cl 11996,C(=O)(C(O)CC(F)(F)F)N1CC(CCCCNC(c2ccc([N+](=O)[O-])o2)=O)C1 11997,c1(CNC(C=NOC)=O)ccccc1CN(C)C(C1CC(=O)N(C2CC2)C1)=O 11998,C(=O)(CCCCCC(C)C)N1CCC(C(C(N2C(CC)CCC(C)C2)=O)F)C1 11999,c1(OCC)nc(N2CCOCC2CN(C)C(C23CCCC(C2)OC3)=O)ncc1Cl 12000,C1(CNc2ccc(F)c(NCc3ccccc3)c2)CCC2(C1)OCCO2 12001,CC1(C)CN(C(=O)CC(F)(F)Cl)CCC1NC(c1ccc(CO)s1)=O 12002,N1(C(C(C)SC)=O)CCC(C2CCN(C(c3cn(C)nc3C(F)(F)F)=O)CC2)C1 12003,CC1(C)COCC1C(=O)NC1CCC(NC(C2(C(F)F)CCCO2)=O)CC1 12004,c1(C(=O)NC2CC3CN(C(c4ccc(Br)cn4)=O)CC23)cccn2cncc12 12005,C(=O)(C1=CCC(C)CC1)N1CCN(C(c2ccc(C)cc2F)=O)CC1 12006,Cc1cc(C)n(CC(=O)NCc2cc(C(=O)NCc3noc(C)n3)co2)n1 12007,c1(C(N(C)CC2N(C(C(C)NC(N)=O)=O)CCC2)=O)ccc(Cl)c(Br)c1 12008,C(=O)(C(C(C)(C)C)NC(C1CC2(CC2)CN1C)=O)NCc1c(CC)cncc1 12009,C1(NC(c2c(SC)cccn2)=O)COC2(CCN(C(C3OCCO3)=O)C2)C1 12010,C(=O)(C1=CSCCO1)N(CCCNC(=O)Cc1sccc1Cl)CCC 12011,C(N=c1cc[nH]cc1[N+](=O)[O-])C1CCCCN(C(c2nc(Cl)ccc2Cl)=O)C1 12012,C12(C(N(CC#C)C)=O)C(NC(=O)C=C(C3CC3)C3CC3)C3CC1C2C3 12013,CC1C(NC(=O)C(C)(C)COCC(F)F)CC2CCC1N2C(=O)Cc1ccsn1 12014,C(C(C(=O)N(C1(C2CC2)CC1)C)NC(C1CCC(=O)O1)=O)N(C)C 12015,C1(C#N)(C(N2CCN(C(Cn3c(C)cc(C)n3)=O)CC2)=O)CCCC(=O)C1 12016,C1(NC(c2cnc[nH]2)=O)CCN(C(=O)CSc2ccccc2O)C2CC12 12017,Cc1[nH]c2ccc(Cl)cc2c1C(=O)NCC1CCCN(C(=O)C2=CSCCO2)C1 12018,C1(C(=O)NC2CCC(NC(CCc3cc(C)on3)=O)C2)CCC2(CCCCC2)C1 12019,c1(C(=O)NCC2CC(NC(CCOCCOC)=O)C2)cc(OC)ccc1N 12020,Cc1ccc(F)c(C(N2CC(CNC(=O)C(C3CCOCC3)C)C(O)C2)=O)c1 12021,C(=O)(C#CC1CCOCC1)N1CCC(C(N2CCCC(CC(C)C)C2)=O)C1C 12022,c1(C(N2C(CNC(c3cc(Cl)cs3)=O)CCCC2)=O)cc([N+](=O)[O-])cnc1O 12023,N#Cc1ccc(N2CCCC(N3CCC(COc4ccccc4)CC3)C2=O)cc1 12024,N1(C(CCCCC)=O)CCCN(C(c2sccc2Br)=O)C(C(C)C)C1 12025,c1(CC)cccc(C(=O)N(C)CC2(NC(c3cc(C4CC4C)on3)=O)CC2)c1F 12026,Cc1cc(CC(N2CC(n3cc(CNC(N)=O)nn3)C2)=O)ccn1 12027,C1(N(C(C(COC)N(C)C)=O)C)CN(C(c2cn(C)nn2)=O)CC1O 12028,C(C(=O)CCC(=O)NNC(=O)C(C)(F)F)c1ccc(OC(C)C)cc1 12029,C#Cc1ccc(CC(N2CC3CC3(CNC(=O)C(c3ccccc3)O)C2)=O)cc1 12030,CCC(C)CCCC(=O)NCC1CN(C)CCN1C(c1cc(C)ccc1C)=O 12031,c1(OC)ccc(CCC(=O)NCCC(C)NC(C2CC2CC(C)C)=O)cc1C 12032,C1(O)(C(C)NC(=O)CCCOC2CCCC2)CCN(C(C2(Cl)CC2)=O)C1 12033,C1(CNc2c(F)ccc(C)c2F)CC2CCC(C1)S2(=O)=O 12034,Cc1cc(=O)n(CCC(=O)NCc2cccc(NC(C34CCCCC3C4)=O)c2)cn1 12035,N1(C(C=C(C)C(F)F)=O)CCOC(CN(C)C(C2CCCN2C=O)=O)C1 12036,c1(C(=O)NC(C)CNC(c2nscc2Br)=O)ccnc(OCCO)c1 12037,c1(CC)c(C(N2CCC(COC)(NC(c3coc(OC)n3)=O)C2)=O)cccc1F 12038,C1(COC)(NC(=O)CCNC(N)=O)CCN(C(c2cc(F)cc(Cl)c2)=O)CC1 12039,c1(OC)cc(C(N2CCC(CN=[N+]=[N-])(C(F)(F)F)C2)=O)cc(OC)c1O 12040,Cn1cc(C(=O)NC2CCC(CNC(C3(C)CCNC3=O)=O)C2)c(=O)n(C)c1=O 12041,N1(C(c2c(CC)cns2)=O)CC(O)CC1C(=O)NC(COC)CC 12042,C1(NC(CCN(CCCCC)C)=O)CC2(CCN(C(=O)C(C(C)C)OC)CC2)C1 12043,c1(CN(C(C2(c3ccccc3)CCNC2)=O)CC)ccc(Cl)c(Cl)c1 12044,CCCCCCCCC(=O)NCC(C1CC1)NC(=O)C(CC)C(=O)OCC 12045,N(C(=NCc1ccc(C)cc1)NC1CCOCC1)CC(CC)NCC(F)(F)F 12046,C1(OC)C(OC)CN(C(=O)C(C)C2CC2)C1CNC(c1nc(Cl)sc1C)=O 12047,C1(NC(c2c(C)snc2)=O)COC2(C1)CN(C(=O)CCCn1ccnn1)C2 12048,C1(OC)CC2(CCC(C(=O)NC3CCCC(CNC(=O)CNC(C)=O)C3)CC2)C1 12049,Cc1ncccc1CC(=O)NC1CC1NC(=O)CCc1cn(C)nn1 12050,C1(OC)CC(CNC(=O)C=Cc2ccnn2C)N(C(c2cc(C)on2)=O)C1 12051,c1(C(=O)NC2(c3ccccc3)CN(C(CC(C)SC)=O)C2)ncnc(C)c1C 12052,C(=O)(C(=O)CC(C)C)N1CCC(CN(C(C2(OCC)CCC2)=O)C)CC1 12053,C1(C(N2CC(N(C)C(c3cc(F)c[nH]3)=O)C2)=O)CC12CCOC2 12054,C12(C(CNC(CC3CC(C)C3)=O)NC(=O)CC3CCCOC3)CCC(CC1)C2 12055,N1(C(C(C)NC(N)=O)=O)CCC(CO)C(NC(C2(CF)CC2)=O)C1 12056,CC(C)(C)CCC(F)C(=O)NCC1CC(F)CN1C(=O)C(O)C(C(C)C)OC 12057,C1(CC2CCC(C(=O)OC)O2)CCCCN1Cc1cccn1CCn1ccnc1 12058,c1(SC)ccc(NC(C2CCN(C(=O)C(C)=C(C)C)C2C(C)C)=O)cc1 12059,c1(NC(CC2CC(OC)C2)=O)cc(C(=O)NCC2(CN(C)C)CC2)ccc1C 12060,C(=O)(C#CC1CCCCC1)N1CCCCC(NC(c2c(SC)cn(C)n2)=O)C1 12061,c1(CN2CCN(C(C)=O)CC2CC(F)F)nn(-c2ccc(F)cc2)c2c1CCC2 12062,c1(CC(=O)NCC(CN(C(=O)Cc2cn[nH]c2)C)O)nc2ncccn2n1 12063,c1(C(N2CCCC(NC(c3ccco3)=O)(CO)C2)=O)c(F)cc(F)c(O)c1F 12064,CC(CC(C)(C)C)C(F)C(=O)NC(c1ccccc1)CNC(C1CNC(=O)N1)=O 12065,C1(C(N2CCN(C(C(c3cncn3C)C)=O)CC2CO)=O)CCC2(CCC2)CO1 12066,c1(OC)ccc(S(=O)(=O)N2CC(NC(=O)CCc3cncnc3)C3(CC3)C2)cc1 12067,CC(CC(=O)NC1(C)CC1)C(C)(C)NC(c1ccc(F)cc1)=O 12068,C(=O)(C1CCc2nccn21)NCC(C)(C)NC(c1cccc(NCC)c1)=O 12069,Cc1cc(C(=O)NC(CNC(c2ccc(CC(N)=O)cc2)=O)C2CC2)ncn1 12070,c1(CNC(c2n(CCOCC)nnn2)c2ccno2)ccc(CC(C)C)cc1 12071,c1(CNC(C=CC(=O)NC2(C)CN(C(C)=O)C2)=O)ccc(F)c(Cl)c1 12072,c1(C(N2CCC(CC=C)(NC(C3CC(C)OC3C)=O)C2)=O)cnc2nccn2c1 12073,Cc1nnccc1C(N1CC2CC1C2C(=O)N(C)CC1(N(C)C)CC1)=O 12074,N1(C(C2=CCCN(C(C3CCC(C)O3)=O)C2)=O)CCCC(C2(C)CC2)C1 12075,c1(OC)ccc2onc(CC(=O)NC(C)C(C)NC(c3c[nH]c(=N)o3)=O)c2c1 12076,C1(CNC(Cn2cnc(=N)[nH]2)=O)CCCN(C(c2ccc(C3CC3)nn2)=O)CC1 12077,c1(C(=O)OCCSc2cc(Cl)ccc2Cl)cc(Cl)c(Cl)cc1F 12078,N1(C(CCCCN(C)C)=O)CCS(=N)(=O)C2(CCC2)C1 12079,c1(C(=O)NCCCOCCNC(c2c(C)ccnc2O)=O)cc2c[nH]cnc-2n1 12080,C1(C(=O)NCC(C)CC(=O)N2CCCC2c2cccnc2)CCC(=O)N(C)C1 12081,C(=O)(C(C(CC)CC)OC)NCCNC(C(C)N(CCCF)CCC)=O 12082,N1(C(c2c(OC)cnnc2OC)=O)CC2ON=C(CNC(c3ccsc3)=O)C2C1 12083,N1(C(c2scc(OC)c2)=O)CC(C(=O)NC2CC(=O)N(O)C2)CC(C)C1 12084,C(C(F)(F)CNC(=O)C(c1ccoc1)NC(=O)CNC=O)OC 12085,n1(CC(=O)NCC(C)N(C(CCC(C)SC)=O)C)c(=O)cnc2ccccc12 12086,c1ccc2nc(-c3nnc(CN4CCC5(CNC(=O)N5)C4)o3)ccc2c1 12087,C1(COC)CN(C(C2CCCC3(CC3)C2)=O)CCN1C(c1cnn(C(C)C)c1)=O 12088,c1(C(=O)NC2C(NC(=O)CSCc3ncc[nH]3)CCC2)cccc[n+]1[O-] 12089,N1(C(CCCC)=O)CCC(CNC(=O)CCNC(=O)OCC)(OC)C1 12090,c1(CC(=O)NCC2C3CN(C(=O)CC4CC(F)(F)C4)CC23)ccc(O)c(Cl)c1 12091,N1(C(C(CCOC)C)=O)CC(NC(=O)CCc2cccnc2Cl)C2(CCC2)C1 12092,C1(NC(C(C(C)C)O)=O)C2CC3C1C3C2C(=O)NCc1ccccc1F 12093,c1(C(=O)NC(C2CCCN2C(c2nn[nH]c2Cl)=O)C)ccc(C(F)F)cn1 12094,c1(CC(=O)NCC(C)CNC(=O)CC2CC3(CC3)C2)c[nH]c2ccccc2c1=O 12095,c1(OC)cccc(C(=O)NCCCCC(C)NC(=O)C(=O)NCC(F)F)c1 12096,N1(C(c2scc(C)c2C)=O)CCCC(n2cc(C(C)Cc3nc(C)sc3)nn2)C1 12097,CC1(C)C2CC=C(C(c3nnnn3C3CCOC3)NCCC3CCC3)C1C2 12098,N1(C(C2CC(NC(C=C(C)C3CC3)=O)C2(C)C)=O)CCN2CCCC2C1 12099,n1(CC(=O)NCC2N(C(C(C#C)(C)C)=O)CC2)c(SC(C)C)nc2ccccc12 12100,c1(C(N(CCCC)CCOC)=O)ccc(CC2CNCCOC2)cc1Cl 12101,C1(O)(C(C(=O)NCc2ccccc2)NC(C2CS(=O)C2)=O)CCCCC1 12102,C1(CC)C(NC(C2CS(=O)C2)=O)CCCN1C(c1ccc(C)c(C)c1)=O 12103,CC1CCc2c(COC(C3CC3c3ccccc3Cl)=O)n[nH]c21 12104,CC(C)C(C(C)NC(c1cscc1Cl)=O)NC(c1ncoc1-c1ccon1)=O 12105,CCCS(=O)(=O)C(C)C(=O)NCC1CN(C)CCN1C(c1cc2occc2[nH]1)=O 12106,c1(C(N2CCC3(NC(CCCN(C(C)=O)C)=O)C(C2)C3)=O)n[nH]c2c1CCCC2 12107,C1(CNC(c2cc(C)oc2)=O)CCN(C(c2cc(Cl)c(Cl)n2C)=O)CC1C 12108,N1(C(Cc2c(C)n[nH]c2C)=O)CC(NC(c2conc2C2CCC2)=O)CC(C)C1 12109,c1(CN(C(=O)C(N2CCOCC2C2CC2)=O)C)cccc([N+](=O)[O-])c1 12110,CCC(CNC(=O)CCC(C)NC(=O)CC(C)(C)OC)CCO 12111,C1(C(N(CCC(c2cccs2)NC(CC=C)=O)C)=O)(CO)CCCO1 12112,C1(NC(C=CCCC)=O)COC2(C1)CN(C(=O)C(C)OCC(F)(F)F)C2 12113,c1(C(N2CCC(O)(CNC(CCC(C)OC)=O)C2)=O)ccnc(C)c1C 12114,C1(NC(C2CCC(O)C2)=O)CC2(CCN(C(C3(F)CC=CCC3)=O)CC2)C1 12115,C(=O)(C1=NN(C2CCCC2)C(=O)CC1)OC.c12c(cccc1F)NC2=O 12116,n1(CCC)cc(C(=O)NCCN(C(=O)CC2OCCC2C)C(C)C)nn1 12117,c1(C(=O)NC(CC)CNC(=O)C(C)SC(F)(F)F)ccc([N+](=O)[O-])s1 12118,N1(C(C(C)(C)N(C)C)=O)CC23CCCCC2(C1)CN(C(=O)C(O)CC(N)=O)C3 12119,C(=O)(C1CCCc2sccc21)N1CC(CNC(c2ccc(C(C)F)cc2)=O)C1 12120,c1(C(N(C2CN(C(CCCN(C(C)=O)C)=O)C2)C)=O)ccc([N+](=O)[O-])s1 12121,C1(NC(c2cn(C)nc2)=O)CC(N(C)C)CN(C(=O)CCC(=O)c2ccc[nH]2)C1 12122,Cc1nc2cc(C(=O)NC(CNC(=O)CN3CCCCC3=O)CO)c(F)cc2[nH]1 12123,C=CCC(C(=O)N1CC(SCC)C1)NC(c1ccnn1CCC)=O 12124,Cc1cc(C(=O)NC2CCCC(CN(C)C(c3oncc3C)=O)C2)c(F)cc1N 12125,c1(C(C)C)cc(C(=O)N(C(C)CN(C)C(c2cc(N)c(F)cn2)=O)C)cc(O)n1 12126,C1(NC(C(=O)NCCOCCCC)=O)CC(F)CN1C(=O)C(C)SCC 12127,C1(C(N2CCC(CC)(NC(C3CC3C3CC3C)=O)CC2)=O)CCC(N=[N+]=[N-])CC1 12128,N#CC1(C2CCN(C(c3cc(C(=O)C4CC4)cs3)=O)CC2)CCCCC1 12129,CC1(C)CC(CNC(C2CSCN2C(=O)CC=C(Cl)Cl)=O)CCO1 12130,C1(C(=O)NC2C3CCN(C(CN(C)C4CC4)=O)CC32)CN2CCC1(C)CC2 12131,C(=O)(C(C)(C)C(C)C)NCC1N(C(C(C)SC)=O)CC(C(F)(F)F)C1 12132,N1(C(c2c(CC)occ2)=O)CCCCC(CCC(=O)NCC2COCC(C)O2)C1 12133,N1(C(CCn2c(C)cc(C)n2)=O)CCC2CC1CN2C(C1CCCS(=O)(=O)C1)=O 12134,Cc1cc(C)c2[nH]c(=NCC(C)NC(=O)C(c3c(F)cccc3F)(C)C)sc2c1 12135,C(CO)(CC(C)CC)NC(CSCCNC(C(C=C)C)=O)=O 12136,c1(CCC(=O)NC(CN(C(=O)C(C)CC(F)F)CC)C)c(C)ncnc1O 12137,N1(C(COCC=C)=O)CC2C=CC1C(C(=O)NCC(CO)C(C)CC)C2 12138,N1(C(=O)CCOc2ccc(F)cc2)CCN(C(=O)Cn2ncnn2)C2CCCC12 12139,c1(C(N(CC(c2conc2C(F)(F)F)=O)CC(F)F)=O)ccc(O)cc1 12140,CN1CCC(C(N2CC(O)(CNC(c3cc(C(C)(C)C)n(C)n3)=O)C2)=O)CC1 12141,C1(CC)CCCC1C(=O)N(CC(C)CNC(c1csc(C)c1)=O)C 12142,Cc1ccc(F)c(N)c1C(=O)NC1CC(C)(CNC(C2CCCN(C)C2)=O)C1 12143,Cc1sc(C)c(C(=O)NCC23CC(CO2)N(C(C2C4CC(=O)CC24)=O)C3)c1C 12144,c1(CC)nc(-n2cccc2)sc1C(=O)NC1CN(C(c2cnoc2C)=O)CC1C 12145,CN=c1[nH]c(=NC(C)c2cccc(S(N)(=O)=O)c2)[nH]c(=NCC(C)N(C)C)[nH]1 12146,c1(C(N2CCC(N(C(COCCOCC#C)=O)C)C2)=O)ccc2c(c1)COC2=O 12147,N1(C(c2[nH]cc(CC)c2)=O)C2CCC1CC(c1cn(CCN3CCCC3)nn1)C2 12148,Cc1occc1C(=O)NCCc1cn(C(c2ccccn2)C)nn1 12149,Cc1[nH][nH]c2ncnc(=NCC3(CNC(C4C(C)C4C)=O)CCC3)c1-2 12150,c1(CCC)nc(C(=O)NCC(C2CCC2)NC(c2cc(C(N)=O)no2)=O)cs1 12151,CS(=O)(=O)c1ccccc1CNCC1CC2CC1CC2(F)F 12152,N1(C(N(c2ccc(Cl)cc2F)CC(=O)OC)=O)CC=C(c2ccc(Br)cc2)CC1 12153,C(=O)(CC1COc2ccccc21)N(CCN(C(CC1(C=C)CCOCC1)=O)C)C 12154,c1(C(=O)NCCCC2(NC(=O)CCNC(N)=O)CC2)cnc(-c2ccco2)s1 12155,c1(-n2cc(C)nn2)cccc2n[nH]cc12.C1(SC)CCCC1C(=O)NO 12156,C(CC(=O)N1CCC(O)CC1C)(C(F)F)NC(c1cnn(CC)c1C)=O 12157,C(=O)(C(=O)C(C)(C)CC)N1C(C)(C(N(C)Cc2ccc(CC)o2)=O)CC(O)C1 12158,N1(C(C(CCSC)O)=O)CCC(CNC(=O)C(c2cnccn2)C)CC1C 12159,c1(C(C(=O)NCc2ccccc2SC)N(CC(=O)OC)C2CC2)ccc(F)cc1Cl 12160,CC1CN(c2cc(C(F)F)ncn2)CCC1NC(C1CCC2CC2CC1)=O 12161,C1(C(N2CC(NC(C3CC(C)(C)C3)=O)C(C(F)F)C2)=O)CCn2c(O)nnc2C1 12162,C1(CC(=O)OC)CS(=O)(=O)CCN1C(=O)C(=O)N=S(C)(C)=O 12163,c1(CC)ccc(C(=O)NC(CN(C(=O)CN2CCNC(=O)C2)CC)CC)c(Cl)c1 12164,C1(C(=O)NC(c2ccccn2)CC)C2CN(C(=O)Cc3ncccn3)CC12 12165,CC1(C(=O)NN(C2CCCC2)Cc2cn(-c3ccccc3F)nn2)CCC(O)CC1 12166,Cc1noc(C)c1CNC(C1CCN(C(C2CCC(O)C2)=O)CC1)=O 12167,C1(NC(C(C2CCN(C(C(n3c(C)cc(C)n3)C)=O)C2)C)=O)CC2CCCC2C1 12168,C1(C(=O)NCC2(OC)CCN(C(C34CSC(C3)C4)=O)C2)CCS(=O)(=O)CC1 12169,C1(CNC(C2C(C)OC(C)C2C)=O)CCC2(CN(CCOC3CCCCC3)C2)O1 12170,C(c1ccc(C(=O)NC2CC2CNC(=O)C(C)(C)CO)o1)=CC(=O)OC 12171,N1(C(CCSC)C(=O)NCCCN2CCCC2)CCN(C)C(C2CC2)C1 12172,CCC(C(=O)OC)C(=O)NC1CC(C(N2CC(F)C(F)C2)=O)C12CCC2 12173,N1(C(c2ccc(Cl)s2)=O)CCC2(C1)CN(C(C1CCc3nn[nH]c3C1)=O)C2 12174,N1(c2nnn(C)n2)CC2CC1CCC2NC(=O)C(C)(C)n1cnnn1 12175,CC1CCCc2nc(C(=O)N(CC(O)CN(C(=O)Cc3csc(S)n3)C)C)cn21 12176,c12ccc(F)c(c1Br)C(=O)N2.N1(C(C)=O)CC(N(C(=O)C=CC2CC2)C)C1 12177,C12(CNC(c3occ4c3CCOC4)=O)CCCC1CCN2C(c1occc1Br)=O 12178,C1(CNC(C(=O)N(c2ccccc2O)C)=O)CC2CN(Cc3nncn3C)CC12 12179,c1(-n2c(C(C)C(C)n3cccn3)nc(-c3nc[nH]n3)n2)ccc(F)c(Cl)c1 12180,C=C(C)C(CC(=O)N1CC(OCCNC(=O)C(c2cnn(C)c2)C)C1)OCC 12181,N1(C(C=C(C)Cl)=O)CCC2(CCC(NC(C3(C4CC4)CC3)=O)C2)CC1 12182,N1(C(C(CCC)C#N)=O)CC2CCC1C1CN(C(=O)COc3cccnc3)CC21 12183,C(=O)(C1=CC2(CCN(C(=O)CCOCC3CC3)C2)C1)N1C(C)CS(=O)CC1 12184,c1(SC2CC2NC(=O)CCN(S(=O)(=O)C(F)F)CCO)cccc(OCCO)n1 12185,N1(C(CC2N(C(c3cnc(C)s3)=O)CCC2)=O)CC(C)CC(C)(C)C1 12186,N1(C(c2c(CNC(c3cnc(CC)s3)=O)ocn2)=O)CCCN(C)CC1 12187,c1(C(=O)NC(CCOC)CNC(=O)C=CC2CCCC2)cnc[nH]c1=N 12188,c1(NC(C=CC=CCC)=O)ccc(NC(=O)C(O)P(C)(C)=O)cc1C 12189,N1(C(c2c(CCC)[nH]cc2)=O)CC2CC(C1)N(C(=O)Cc1cc(O)nnc1O)C2 12190,c1(OCC)nc(Cl)ccc1C(=O)N(C)CC1CCCN1C(c1ccc(O)cn1)=O 12191,N1(C(C(CCC)OCC)=O)CC2CCN(C(c3sc(SC)cc3C)=O)C(C2)C1 12192,c1(C(C)CNCc2cc(CC)cc(F)c2)ccc2cc(OC)ccc2c1 12193,c1(CC(=O)N(CC)CC2CCCN2C(=O)CC2OCCCO2)ccc(F)c(C)c1 12194,CS(=O)(=O)c1ccc(NC(C2CCCC(COc3ccc(F)c(Cl)c3)C2)=O)nc1 12195,C1(NC(CC(C=C)C)=O)CCCCN(C(c2csc(COC)c2)=O)C1 12196,c1(C(=O)NCC2CC(F)(CNC(C(C)SCC)=O)C2)nccn2nccc12 12197,c1(N(C(CSCC#C)=O)CCNC(=O)C(C)(C)OCCC)ccccc1NC 12198,N1(C(c2c(CC)noc2)=O)CCC2(NC(c3occ(C)c3C)=O)CCCCCC12 12199,C1(C(=O)NC2C(C(=O)NCC3(OCC)CN(C)C3)CCOC2)C2CCC(C2)C1C 12200,C12(C(=O)NC3C(NC(c4cnc(C)[nH]4)=O)COC3)CCC(C(F)(F)F)(CC1)C2 12201,C1(NC(=O)CCF)(CNC(C2CCC(N3CCOCC3)CC2)=O)CCCCC1 12202,C1(N(CC#C)C(C2CS(=O)(=O)C2)=O)CCN(C(=O)COC2CCOCC2)CC1 12203,C12CCN(CC1)C(C)(C)NC2=O.C(C)(C)(C(=O)N1CCCC1C1(O)CC1)OCC 12204,Cc1cccc(Br)c1C(=O)NC1CN(C(c2ncoc2C)=O)CC1C#N 12205,c1(NC(C2CN(c3ncnc4ccsc34)CCC2O)=O)ncc2c(n1)CCC2 12206,CC(C(=O)OC(C)(C)C)N(C(C(=O)NCC#N)C1CC1C1CCOC1)C1CC1 12207,C(=O)(C(F)CCC)NCC(c1ccccc1)N(C(CCOCC#C)=O)C 12208,N1(C(C(CC)N(C)C)=O)CCC(NC(c2cccnc2)=O)C1(C)C 12209,CC(C)(C)C#CC(=O)NC1CCCCN(C(=O)COCCCF)C1 12210,c1(OC)ccc(C(=O)NC2CCN(C(=O)CO)CC2C)c(C(F)F)c1.C(=O)C1CC1 12211,c1(C(=O)NC2CCCN(C(CCCCOC)=O)C2)cnc2c(cnn2C)c1 12212,CC1CCN(C(=O)C(c2ccc(F)c(F)c2)(C)C)CCN1C(C1CCCOC1)=O 12213,C(C(C)C(F)F)NC(CCN(C(C(C)=C(CC)C)=O)CCO)=O 12214,N1(C(CCC(C)C)=O)CC(O)(C2(CNC(c3cccc4ccnn34)=O)CC2)C1 12215,Cc1c(C(=O)NCC(C)(C(C)C)NC(c2nn(C)cc2Cl)=O)[nH]c2c1CCCC2 12216,C(=O)(CC1=NNC(=O)C1)N1CCN(C(c2c(C)oc(CC(C)C)c2)=O)CC1CO 12217,CCC(CCC(=O)NCCC(C)CCNC(c1cnn(C2CCC2)n1)=O)OC 12218,CC(CF)CC(=O)NCCCC1(NC(c2nccnc2N)=O)CC1 12219,Cc1nscc1C(=O)NC(C1CCN(C(=O)CC2CCCN2C(C)C)C1)(C)C 12220,CC1CC2CN(C(C3CCC(NC(=O)CC4CCCO4)C3)=O)CCN2C1 12221,Cc1nc(=NCc2cc(C(=O)NCc3cscn3)ccn2)[nH]cc1Br 12222,c1(OCC)nc(NC(C(C)NC(c2cc(C3CC3)cs2)=O)C(C)C)ncc1Cl 12223,C1(C(=O)NC2(CO)CN(C(c3ccc(C)c(Br)c3)=O)C2)CCn2ccnc2C1 12224,Cc1cnc2n1CCC(C(=O)N(CCNC(=O)C=Cc1cn(C)cn1)C1CC1)C2 12225,CC(CC(=O)NCC1(C(C)(C)O)CN(C(=O)C(C2CCCCC2)O)C1)P(C)(C)=O 12226,[N-]=[N+]=NC1CCN(C(c2coc(CNC(=O)C(=O)NCCF)c2)=O)CC1O 12227,c1(OCC)ccc(CN(c2ccc(C(=O)N(C)C)c(C)c2)C)cc1OC 12228,C(=O)(CCN(OC)C(=O)C(CC1CC1)NC(=O)CCCC1CCC1)OC 12229,N1(C(c2ccc(C)c(C)n2)=O)CCC2(CCCN(C(c3cnc(S)n3C)=O)C2)C1 12230,C12(NC(C(c3cccc(Cl)c3)CC)=O)COC(C)(C1)C2 12231,C(=O)(C1=Cc2cc(Cl)ccc2OC1)N1CC(C)N(C(=O)C(N)=O)CC1C 12232,C1(N(C(=O)CC2(NC(N)=O)CC2)C)CCC(NC(=O)Cc2ccccc2Br)CC1 12233,C1(NC(C2CN(C(C)=O)C2)=O)(CO)CCCN(C(=O)C=Cc2cccc(Cl)c2)C1 12234,C1(NC(CCCCC)=O)CCCCCC1C(=O)NC(CC)C(=O)OC 12235,C=C(Br)CC(C)(C)C(=O)NC1CCN(C(C2(C#N)CCOC2)=O)CC1O 12236,C1(OC)CCC(CC(=O)NCC2CC(C)N(C(c3nc(Cl)sc3C)=O)C2)CC1 12237,C1(C(=O)NC(CCNC(C2(C)CCC(OC)CC2)=O)C)CCC2(CC1)CC2(F)F 12238,N1(C(CC(CCC)C)=O)CC(C(=O)NC(C)CSC)C(C2CC2)C1 12239,c1(CC)cnc(C)c(NC(=O)C(CCNC(=O)CP(C)(C)=O)OC)c1 12240,c1(NC(c2c(C)cccn2)C)ncccc1S(=O)(=O)NC1CCCC(O)C1 12241,c1(C(N2CC3(CCCCN3C(c3ccns3)=O)C2)=O)cc2cc(F)cc(F)c2[nH]1 12242,C(=O)(N=c1cc2ccccn2[nH]1)C1N(Cc2c(C)n[nH]c2)CCSC1 12243,C(CCN=c1ccnc(Cl)[nH]1)NC(c1coc(C2CCOCC2)n1)=O 12244,CCC(C)(C)C(=O)N(C)CC1CCN(C(c2cnc(SC)nc2)=O)C1 12245,c1(C(=O)NCC2CN(C(c3nc(C)[nH]n3)C)C2)ccc(F)c(C(F)(F)F)c1F 12246,N1(C(CC#N)=O)CCC2CCN(C(=O)CCn3ccnc3)CC2C1 12247,C1(C(N2C(C)C(NC(c3cc(O)nn3C)=O)CCC2)=O)CCc2cnn(C)c2C1 12248,N1(C(CC(C)NC(=O)CCc2ccnn2C)=O)CCOCC1CCO 12249,C(CC(F)F)(C(=O)N1CC(C)C(C)(CO)C1)N(C(C1CN(CC)C(=O)C1)=O)C 12250,c1(-c2cn(C3(CCN4CCC(OCC)C4)CC3)nn2)ncc(N)cc1C 12251,N1(C(C(c2ccccc2)OC(C)=O)=O)CCC(C)(NC(=O)CC2(O)CCC2)C1 12252,Cc1oc(Cl)nc1C(=O)N(C(C)CCNC(=O)Cc1ccccc1O)C 12253,C12(C3(C4CCCCO4)CC3)C(C(=O)OC)C3CC1C2C3 12254,C1(C)(CC)CCC(C(=O)NC(CN(C)C)C(=O)NC(C)CC(C)(C)O)O1 12255,C1(CC(C)(C)C)COCCN1C(N1CCC(=O)C1)=O.c1(C)ncsn1 12256,CN1CC(C(N2CCCC(NC(=O)CCCc3ccsc3)C2)=O)CC1=O 12257,C(=O)(C1Cc2c(Cl)cccc21)NCC(C)(CO)NC(c1c(C)ncc(N)c1)=O 12258,c1(OC)ccc(C#N)cc1NC(C1CCCN(Cc2sccc2C)C1)=O 12259,C1(NC(c2c(C(C)C)nn(C)c2)=O)C2CC3CN(C(=O)CC4CN(C)C4)C1C3C2 12260,c1(C(N(CCOC)CCNC(c2cccnn2)=O)=O)c(O)ncc(Br)c1C 12261,N1(C(C2C(C)(C)OCC2)=O)CCOC(C(N2CC(c3ncccn3)C2)=O)CC1 12262,C(C(=O)N(CCC(=O)N1CCC(F)(F)C(OC)C1)OC)(C1CC1)OC 12263,Cc1cc(C(=O)NC(C(N2CCCC2CO)=O)C2CC2)sc1C 12264,C1(N(C(c2cc(CC)on2)=O)C)CCCN(C(c2ccn(CC(C)C)n2)=O)CC1 12265,C1(NC(C(c2ccccc2F)(C)C)=O)CCN(c2nnc(C(F)F)o2)CC(O)C1 12266,N1(C(c2ccn(C(C)C)n2)=O)CCCC(NC(=O)CC2COCCN2C)C1 12267,Cc1ccc(OCC2(F)CN(C(=O)CCn3ncccc3=O)C2)c(C)c1.CC=O 12268,c1(CSC)cc(C(=O)NCCC(C)(C)NC(=O)C=NOC)sc1C 12269,C1(OCCC(=O)NN2C(=O)C(=O)NCCC2)CCOCC1.C(C=O)N(C)C.C1CC1 12270,C1(CNC(COC)=O)CC2CCC1N2C(c1cc(C)cc(C)n1)=O 12271,N1(C(C2(CC)CCC2)=O)CCOC(C)(CNC(=O)CC2CC(=O)NC2=O)C1 12272,Cn1c(CO)nnc1C1CCCN(C(c2cc(-c3cccnn3)[nH]n2)=O)C1 12273,N1(C(C(=O)NCC(F)C2CCC2)=O)CCC(O)C(F)C1 12274,CCCCC(C(=O)N1CC(C(C)CC)C1)NC(c1cn[nH]c1)=O 12275,S(=O)(=O)(c1cnc(NCC(c2ccncc2)O)cc1C)NC1CC(CC)OCC1 12276,CCCC(CC)CCC(=O)NCC#CCNC(=O)C(CC)(CC)c1ccccc1 12277,c1(C(=O)NC(CCCCNC(c2cccc(CC)n2)=O)C)cccc2occc12 12278,Cc1cc(C(=O)N(C2CC(C(=O)NC(C(F)(F)F)C3CC3)C2)C)n[nH]1 12279,N1(C(N(C2CCNCC2)C)=O)CC2(CCN2C(c2ccc([N+](=O)[O-])[nH]2)=O)C1 12280,CC12CCN(C1)C2=O.c1(NC(=O)COc2cn[nH]c2)c(Br)cnn1C1CC1 12281,S(=O)(=O)(c1ccc2[nH]c(=NCCC#CBr)sc2c1)NCC(C(C)C)O 12282,C1(NC(C2(CSC)CCC2)=O)CCC2CN(C(=O)C(C)OCCC(C)C)CC2C1 12283,C1(NC(CC(CC)C)=O)CC12CCC(NC(=O)CCc1cccnc1C)CC2 12284,c1(C(=O)NC2(C)CC(NC(C(CCC)O)=O)C2)cccc2ccc(C)nc12 12285,c1(C(N2CC(O)(C3CC3)C2)=O)cc2c(F)c(Cl)ccc2[nH]1 12286,c1(NCc2cc(Br)co2)ccccc1.O=C1C(F)C2CC(C2)N1 12287,N1(C(C2CC(C)(CC)C2)=O)CCCC(CC(=O)NCc2ccc(C#N)o2)C1 12288,N1(C(C(CCCC=C)NC(C2CC3(CC3)C2)=O)=O)CCN2C(=O)NCC2C1 12289,c1(CC)nc(C)n(C)c1C(=O)NCCOCCNC(C1CCC2(CCC2)C1)=O 12290,C1(CCC)CN(C(c2cnns2)=O)CCN1C(=O)CNC(=O)Nc1cccs1 12291,Cc1ccc2nc(SCC(N3CC4CCN(C(=O)C(C)CO)CC4C3)=O)[nH]c2c1 12292,c1(COC)nc(OC)cc(NC23CCC(CC2NC(C)=O)C3)n1 12293,C(CCC(=O)N(C1CC(NC(c2cc[nH]c2C2CCC2)=O)C1)C)OCC 12294,N1(C(C(C)COc2ccccc2)=O)CCC(C)(C)C1CNC(=O)C(C)(C)F 12295,C1(CCNC(CC2(OC)CC2)=O)(NC(=O)CCCc2cccs2)CCCC1 12296,N1(CCC(=O)NCC2(CN(C(C(CC)C)=O)C)CC2)CCCCC1C 12297,N#Cc1ccccc1CCC(=O)NC1CCCN(C(c2ccc(Br)cc2F)=O)C1 12298,N1(C(C2CC(OC(C)(C)C)C2)=O)CCC(O)(CCNC(C2CCSC2)=O)CC1 12299,C(c1cc2ccccc2o1)=CC(=O)NCC1CC(NC(CC=CC)=O)C1 12300,c1(CN2CCC(CNC(C(c3ccc(OC)cc3)O)=O)C2)ccc(F)c(F)c1 12301,CC1CCOCC1C(=O)NC(C1(N2CCOCC2)CCCCC1)c1ccccc1 12302,c1(CC(=O)NCc2ccc(CNC(C3C4CCC(F)C34)=O)cc2)ccccc1Cl 12303,c1(OC)cc(N)c(Cl)cc1C(N1CC2CC(NC(c3ccc(F)cc3)=O)C1C2)=O 12304,CCC(C(=O)NCCOCCNC(c1ccc(N)c(Br)n1)=O)C(C)(F)F 12305,C(=O)(CC(O)CC(C)C)N1CCC(C(C(=O)NC(C(=O)OC)(C)CO)F)C1 12306,c1(C(=O)NC2CCN(C(=O)C3=COCCC3)CC2O)cnc2ccc(F)cc2c1 12307,c1(C(=O)NCC2(CNC(=O)Cc3nc[nH]n3)CCC2)nc2cnccc2s1 12308,CCC(C)(C)C(O)C(=O)NC1(CCNC(=O)CC2CCC(C)(C)C2)CCC1 12309,CCC(C)C(O)C(=O)N1CCCC(C)(CNC(=O)C(C2CCCCC2)C)C1 12310,c1(C(N2CCC(NC(C3C(F)(F)C34CC4)=O)C2)=O)cc2cc(F)cc(F)c2[nH]1 12311,C1(C(=O)N(C(c2onc(C)n2)CO)CCO)CN(C(=O)C(C)CC2CCC2)CC1F 12312,CCC(CC(=O)N(C1CC(NC(c2cc(Cl)ns2)=O)C1)C)C(C)(C)C 12313,C(=O)(C(CC)(CC)C(=O)O)N1CCC(Oc2cc(C(=O)OCC)c(OC)cc2)C1 12314,c1(C(=O)NC(CNC(c2cc(C)nnc2)=O)C2CC2)cc([N+](=O)[O-])ccc1N 12315,CCC(CC(F)F)C(=O)N1CC(OC)CC(NC(=O)CCNC(N)=O)C1 12316,N1(C(CC=CC=CCCCCC)=O)CC(CNC(c2cccs2)=O)C(O)C1 12317,N1(Cc2c(C)ncs2)CCN2C(=O)COCC2C1.C12COC(C1)C(=O)NC2 12318,c1(C(=O)NC2C(C)(C)N(C(C3CC4CC4C3)=O)CC2)cccc2[nH]nc(O)c12 12319,c1(C(=O)NC2C(CNC(C(CCC)CC)=O)CC2)cc(C)c(Br)c(C)c1 12320,C(=O)(C(F)C(F)(F)F)NC1(CC(=O)NC2CCC(C(N)=O)CC2)CCOCC1 12321,C1(NC(C(Cc2c(C)nc[nH]2)O)=O)CC2CC1N(C(c1csc3nnsc13)=O)C2 12322,c1(C(N2CC(C(=O)NCc3ncccn3)C(F)(F)C2)=O)ccc2nccn2c1 12323,C1(C2CCN(C(C3CCCCCS3(=O)=O)=O)CC2)(NC(C2CCCC2)=O)CCC1 12324,N#CC1(c2nnc(N3CCC(CC(F)F)C3)n2CCOCC(F)(F)F)CCCC1 12325,N1(C(Cn2ccc(C)n2)=O)CC2C(CNC(c3ccc(CF)cc3)=O)C2C1 12326,N1(C(c2c(COC)cc[nH]2)=O)CCOC(C)(CNC(=O)C(c2nc(C)cs2)C)C1 12327,N1(C(C(C)CC2CC2)=O)Cc2ccccc2CC1CNC(=O)C(C)C(C)(F)F 12328,N1(C(C2C(C#C)C2)=O)CC2(CCC2)CC1CNC(c1cnn(C(C)C)n1)=O 12329,C1(C(=O)NC2CCCN(C(C=C(C)CN3CCOCC3)=O)C2)CC2CCC(C1)S2 12330,C1(CN(C(C2(CC)CN(C(=O)CCc3ccc[nH]3)C2)=O)C)CCCCC1O 12331,C1(OC)CC2CC(NC(=O)C(CCNC(C3C4(CC4)C34CC4)=O)OC)CC12 12332,C1(OC)CCC(C(=O)N(C(C)(C(=O)NC(C)CC(C)C)C2CC2)C)CC1 12333,N1(C(C#CC(C)C)=O)CCC(C)C(NC(c2cc(C(N)=O)ccc2F)=O)C1 12334,O=C(C(O)C(F)(F)F)N1CC(O)(C2CCCN2C(C23CC2CCO3)=O)C1 12335,C#Cc1ccc(CC(N2CCN(C(C)=O)C(CS(C)(=O)=O)C2)=O)c(F)c1 12336,C=CC1(C(=O)NC(C)CN2CCCC2)CCN(C(C2OCCC2(C)C)=O)CC1 12337,N1(C(CCC#CC)=O)CC(NC(=O)C=CC(c2ccc(F)cc2)=O)CC12CCCC2 12338,N1(C(COCCOC)=O)CCC2(CC1)OCCC2NC(c1cc(C)nc(C)c1)=O 12339,C1(C(=O)NCC(C(=O)NC(C2CCOC2)(C)C)CC2CC2)CC2(CC(=O)C2)C1 12340,c1(C(=O)NCC(CNC(C2C(C=C)C2)=O)F)cc(N)c(F)cc1F 12341,N1(C(CCC=C=C)=O)CCCC(O)(CCNC(=O)CCN2CCC(F)C2)C1 12342,C1(NC(c2ccn(CCC)n2)=O)CCC12CN(C(=O)CCOCC)C2 12343,CCCC(C(=O)NC(C)CC(C)(C)CO)NC(C1CC(F)(CF)C1)=O 12344,C(=O)(C1=CCCC1C)NC(C(=O)NCC1CCCN(C(C)=O)C1)CO 12345,C12(NC(c3c(C)n(C)cn3)=O)CCCC1CN(C(=O)CN(C1CCCC1)C)C2 12346,CCC(CC)C(C)C(=O)N1CCC(NC(c2cc(O)ccc2F)=O)CC1C 12347,N1(C(C(C)=C2CC2)=O)CCN(CCCNC(=O)CCNS(C)(=O)=O)CC1 12348,N1(C(C(C2CCC(=O)N2)C)=O)CC(C)(NC(C2(CC3CCC3)CC2)=O)C1 12349,N1(CC2(C(=O)NC(c3ccn(C)n3)C)CCC2)CCN(C(N)=O)CC1 12350,N1(C(c2cc(C)no2)C(=O)NCC(F)F)CCc2cc(C#N)ccc2C1 12351,c1(Cn2c(C)ncc2)ccc(OC(C)Cc2nccn2C)cc1 12352,Cc1nc(Br)cnc1NC(=O)C(=O)Nc1c(NC(=O)CCC(C)C)cccc1F 12353,N1(C(CC=CCC)=O)CCC(C2CCN(C(c3n[nH]c(C4CC4)n3)=O)C2)C1 12354,c1(N(C)C)cc(CC(N2CCC(NC(=O)C(Cl)=CCl)CC2C)=O)ccc1[N+](=O)[O-] 12355,N1(C(CC=CCC)=O)CCN(C(=O)CN(CC)Cc2ccc(C)cc2)C(CC)C1 12356,C=C(C)CN=C(NCC(C1CCCCCC1)(C)O)NCC1CCC(C2CC2)O1 12357,n1(CC)ncc2cc(C(=O)NC(c3ccccc3)C3CC3)c(C)nc12 12358,C(=O)(C(CC(C)(C)C)OC)N1CCCC(CC)C1C(=O)NCc1sc(C)nc1C 12359,N1(CC(N2C(CCNC(CCCC(N)=O)=O)CCC2)=O)CCCCCCC1=O 12360,C1(NC(C2C(CC)C2)=O)CCCCCCC1NC(=O)CCc1cnc[nH]1 12361,c1(CC)nc(C)[nH]c1C(N1CCC(N(C(=O)CC2C=CCC2)C)C1)=O 12362,C(=O)(C(O)C(CCC)NC(c1sncc1C)=O)N(CCC)CCN(C)C 12363,C(N=c1[nH]c(C2CC2)nc2[nH]ccc12)C1CC(NC(c2cc(C)cc(Cl)n2)=O)C1 12364,C1(F)(C(N2C(C)(CCO)CCC2)=O)CC2CCC1C2.C1CCCCN1C 12365,C1(N(C(c2c(C)nccc2)=O)C)CN(C(C2CC3C=CC2C3)=O)CC1(C)C 12366,c1(N2C(C(N3CC(C(=O)OC)C4C3C4)=O)CC=CC2)nc(C)cc(C)c1CSC 12367,Cc1ccsc1CCCC(=O)NCCN(C(=O)C(C)Cc1ccco1)CC(C)O 12368,C12(CNC(CS(=O)(=O)NC)=O)CCCC1CN(C(c1cc(C)co1)=O)C2 12369,Cc1csc(=O)n1CC(=O)NC1C2CC1N(C(c1sccc1SC(F)F)=O)C2 12370,c1(C(=O)NCC2N(C(C(C=C)(C)C)=O)CCC2)ccc2cnccc2c1 12371,C(CCC(=O)NC(=O)NC(C1CCCC1)Cc1cnn(C2CC2)c1)OCCOC 12372,Cc1cnn(C)c1C(=O)NC(C)C(C1CCCCC1)NC(c1ccsc1)=O 12373,C1(CNC(C(=O)NC(C)C)=O)CC12CCc1ccccc12.c12cc(on1)C2N(C)C 12374,N1(C(c2ccc(OC)s2)=O)CC(NC(C2CC(N(C)C)C2)=O)CC12CCCC2 12375,N1(C(CC2(C)CCCC2)=O)CCCC(C)(O)CC1.c12cccc(c1)-n1cc-2nn1 12376,c1(C(CC(=O)NCC2CN(C(COC)=O)C(C)(C)C2)=O)c[nH]c2ccccc12 12377,C(=O)(C1=NNC(=O)C1)NCCCC(C)NC(C(C)c1ccon1)=O 12378,O=C(C1=CC2(CCN(C(c3ccco3)=O)C2)C1)NCCc1ncccc1F 12379,CC1CC(NC(=O)CCc2cccc(O)n2)CN1C(c1cscc1C#N)=O 12380,N#CCCCCCC(=O)NC1CC2CCC1CC2NC(C1CCS(=O)(=O)CC1)=O 12381,C=CC1CCCC(NC(C2CC(C)(NC(=O)C=CC(C)CC)C2)=O)C1 12382,N1(C(CCC(=O)OC)=O)CCNCC1C1CC1.c1(C(C)C)ccc(Cl)cc1F 12383,C(=O)(CCCC(=O)N1CCC(C(C)NC(=O)CC2CCC(C)(C)CC2)C1)OCC 12384,c1(C2CCN(C(CSCCOC)=O)CC2)ccccc1NC(=O)C(C)C1CC1C 12385,N1(C(C(COCC)NC(C)=O)=O)C2CCC(C2)C1C(=O)NC1CN(C)CCC1O 12386,C1(CNC(=NCC)NCCC(C)(C)C)CC2(CC2)S(=O)(=O)N1 12387,Cc1ccc(C=CC(N2CCC3(CC3NC(=O)CSC(F)F)C2)=O)cc1 12388,C(=O)(C1CCOc2c(F)cccc21)NC(CC(C)NC(C1CC2C=CC1C2)=O)C 12389,C1(NC(COCCC#C)=O)CCCOC12CCN(C(C1(O)CC1(C)C)=O)CC2 12390,Cc1cccc2c1c(CNC1CC(NC(=O)C(O)C(C)C)C1)cn2C 12391,N1(C(C2CC(=C)C2)=O)CCN(C)C(C(=O)NC2(C(=O)OC)CCCO2)C1 12392,c1(C(N(C2CCN(C(=O)COc3ccccc3)C2)C)=O)c(N)cnn1C 12393,c1(N(CCOC)C)nc2c(c(=NC3CC(Sc4cccnc4)C3)[nH]1)CC(C)CC2 12394,C(=O)(CCCCC(C)C)NC1C2(CN(C(C3CN(CCC)C(=O)C3)=O)C2)CC1 12395,C(N=c1nc2c(ncn2C)c(NCc2ccoc2C)[nH]1)C1(CCC)CC1 12396,c1(C(=O)NCCCNC(CC(CCC)(C)O)=O)cc(S(=O)(=O)CC)cnc1O 12397,Cn1cc(C(N2CCC(C(=O)NCC3(CO)CCC3)C2)=O)cn1 12398,c1(OC)cc(C)ccc1OCC(=O)N(CCC(C)NC(=O)C(C)S(N)(=O)=O)C 12399,CC(C)C(C(C)NC(c1c[nH]nc1-c1ccncc1)=O)NC(=O)CSCC(N)=O 12400,N1(c2nnc(C)s2)CC2(C1)SCCC2NC(C1CCc2c[nH]nc2C1)=O 12401,CC1NC(=O)CCC1CNC(=O)CCN(C(=O)C1=NOC(C)C1)C 12402,C1(C(=O)NCC(=C)CCNC(=O)C(C)n2cccn2)CCC(=O)N(CC)C1 12403,C12(NC(CN(S(CC)(=O)=O)C)=O)CCN(C(c3ncn4c3CCC4)=O)CC1C2 12404,c1(CC(=O)N(CC(C)N(C(C(CCC)OCC)=O)C)C)cc(F)cc(Cl)c1 12405,N1(c2c(OC)cc(C)cc2)N=C(C(=O)N(c2cccc(O)c2)C)CCC1=O 12406,N#CC1(C(=O)NC2CC(CCNC(=O)C=C(Cl)Cl)C2)CC2(CC2)C1 12407,Cc1c(C(N2CCC(C)(NC(=O)CN3CCC3C)C2)=O)[nH]c2ccccc12 12408,Cc1cnc(C=CC(=O)NCC2CCC(NC(c3sc(C)nc3C)=O)C2)[nH]1 12409,N1(C(c2ccnc(F)c2)=O)CCC(F)(F)C(CNC(C23CCCC2C3(F)F)=O)C1 12410,Cn1nc(C(N2CC(O)CC2(C)C(N2CCC2C2CCCCC2)=O)=O)ccc1=O 12411,C1(CNC(C2(C)CC=CCC2)=O)CC12CCN(C(C13CC(CO)(C1)C3)=O)CC2 12412,c1(C(=O)NC2C(C)CCN(C(C=Cc3c(C)ncs3)=O)C2)ccc2n[nH]cc2c1 12413,c1(OC)cccc(N2CC3CCC2C(NC(C2CC(=O)N2)=O)C3)c1[N+](=O)[O-] 12414,CP(C)(=O)c1ccnc(C(N2CCCN(C(c3cccnn3)=O)C(CO)C2)=O)c1 12415,c1(C(=O)NC2C(NC(C)=O)CC2)cccc(C(C)C)c1C.C12CC(O)CN1C2 12416,C1(NC(COCCOCC#C)=O)CCCC1NC(=O)CCC1CCN(C)C1 12417,Cn1cc(C(N2CC3CC3(C(=O)NC3CNC(=O)C3)C2)=O)n(C)c1=O 12418,CCC(C)C(C)(O)CNC(=O)CC1(NC(c2cc(O)nc(O)n2)=O)CC1 12419,c1(C(C(=O)NCC(c2ccccc2)N(C)C(c2cnco2)=O)O)ccccc1Cl 12420,N1(C(CCSc2ccc(C)cc2)=O)CC2(CCC2NC(=O)CC2CNC(=O)C2)C1 12421,CC(=O)CCCC(=O)N(C)CC1CCN(C(=O)COCc2ccnc(O)c2)C1 12422,N1(C(=O)COC2CCCCC2)CCC(CNC(C2(F)CC2)=O)C12CCC2 12423,C12(C(=O)NCC(CNC(=O)C(C)SC(F)(F)F)OC)CC(CC(F)F)(C1)C2 12424,C1(O)(CN(C(CC)=O)C)CCN(C(=O)C(C)c2ccsn2)C1 12425,c12cccc(c1)NC(=O)NC2.N1(CC(C)C)CCC(NC2CC2)C1 12426,C1(CC(=O)NC(CC2CC2)C(=O)N(CC2CC2)CC2CC2)CNC(=O)O1 12427,CC#CCC(C(=O)NC(c1nc[nH]n1)CO)NC(=O)C(CC1CCC1)OC 12428,C(=O)(C(F)C(=O)NC1CN(C(=O)Cc2nncn2C(C)C)CC1C(F)F)OCC 12429,C(=O)(N=c1[nH]oc2cc(Br)ccc12)C1CCN(CCC)C1 12430,N1(C(CC(C)C2CC2)=O)CCN(C(=O)C(C(C)O)NC(c2ccccc2)=O)C(C)C1 12431,C1(CC=C)(NC(c2cc(COC)on2)=O)CCN(C(C2CSCCS2)=O)C1 12432,C1(CC)C(NC(=O)C=Cc2cncc(OC)c2)CCCN1C(C1C2CCCC12)=O 12433,c1(C(N2C(Cn3cc(CC(C)(C)O)nn3)CC2)=O)ccc(-c2nccnc2Cl)cc1 12434,C1(NC(CSc2n(C)ccn2)=O)CCC2(CC1)CCN(C(=O)CC1CC1(C)C)C2 12435,N1(C(C(CN=[N+]=[N-])NC(C2CCCCC2O)=O)=O)CCn2nncc2C1 12436,CC1OC2(C(=O)NC3C=CCN(C(c4c(F)cccc4F)=O)C3)CCC1CC2 12437,c1(C(N2CC(C)C(CNC(c3cc(Cl)no3)=O)CC2)=O)ccc2ncccn12 12438,C1(CC(=O)NCCCN(C(=O)C(c2cccnc2)O)C(C)C)CC1C1CC1 12439,c1(NC2CN(C(C)C)C2)ncccc1S(=O)(=O)N1CCCCC2(CCCC2)C1 12440,c1(NC(N(C2(COC)CCSC2)C)=O)c(OCC2CC2)cccc1Cl 12441,N1(CC(C)(C)NC(C(CC2CC2)OC)=O)CCN(C(C23CCCC2C3)=O)CC1 12442,C=CC1(CC(=O)N(C)Cc2scnc2C)CN(C(C2CC(C)(C)CO2)=O)C1 12443,C1(C(=O)Nc2scc(C(=O)OC)n2)CC2CC2N1C(=O)Cc1ccccn1 12444,C(CCOC)(C(=O)NCCN(C(=O)C1=CCCC1)CCOC)OC.C1CO1 12445,C=CC1(C(=O)NC(c2nn[nH]n2)C2CC2)CCN(C(=O)C=CCC)C1 12446,c1(C(N(CCCNC(CC(N2CCCCC2=O)C)=O)C)=O)ncccc1Br 12447,CC1CCC(C)(C(=O)N(CC(C)CNC(=O)C(O)Cc2ccccc2)C)C1 12448,c1(C(N(CCNC(CCC(=O)NCC)=O)CC)=O)ccc(N)cc1Cl 12449,CC1C(C(=O)N(C)CC2CC(F)C2)CCCN1C(=O)Cc1ccccn1 12450,c1(Sc2cccc(F)c2)cc(Br)ccc1N(C1CNCC(N)C1)C 12451,C1(NC(C(CCC)O)=O)CC2CCC(C1C)N2C(=O)C(C)S(=O)CC 12452,c1(C(N2CC3C(CCNC(=O)CSC(F)(F)F)(CC3)C2)=O)cnc2cc[nH]c2c1 12453,N1(C(c2c(CC)nccc2)=O)CCCC(C)(C(=O)Nc2cc(Br)cnc2Br)C1 12454,CON(C)C(=O)CN(C)NC(=O)Cn1nc(C)c(C)c1C 12455,c1(OC)cccc(C(=O)NC(C(=O)NC(C(O)CO)C2CC2)c2ccoc2)n1 12456,CC1CSCCN(C(c2cnn(CCNC(=O)CC3CC(F)C3)c2)=O)C1 12457,CC1CC(CNC(C2(O)CCSCC2)=O)CN1C(=O)CN1CCCNC1=O 12458,C(CC(O)C(=O)N1CCCC(NC(c2ccnc(C(N)=O)c2)=O)C1)N(C)C 12459,c1(NC(c2nccs2)CC)ccnc(N(C)Cc2sccc2C)n1 12460,C1(C(N2C(C(C)NC(c3ccc(Cl)cn3)=O)CCC2)=O)OCC2COCCC12 12461,C1(C(N2CC(c3cn(CC=C)nn3)(C(=O)OC)C2)=O)CC2C=CC1C2 12462,C1(N(C(C=C(CC)C)=O)C)CC2CCC(C1)N2C(=O)C(C(CC)CC)OC 12463,CC(C)C(CN(C)C)C(=O)N1CCCC1CNC(=O)C(F)(F)C1CC1 12464,C(CNC(C1(Cl)CC1C(C)=O)=O)(CC(=O)N(C)CC1CN(C)CCO1)OC 12465,C(CC(C)(C)C(=O)NCC1CCN(C(=O)C(C)Oc2ccc(Cl)cc2C)C1)OC 12466,N1(C(C(C(C)C)SC)=O)CCC(C)C(NC(c2cc(C(C)(C)C)n[nH]2)=O)C1 12467,N1(C(CCc2cn(C)nc2)=O)CCC2(CC1)CN(C(C1CCC(C)(C)CO1)=O)C2 12468,C1(NC(c2ccc(CC)cc2O)=O)CC(NC(c2ccoc2)=O)C12CCOCC2 12469,CC1COC2(CCC2)CN1C(C1CC2CC1CC2NC(c1cccn1C)=O)=O 12470,C1(CC(=O)NC(C(=O)OCC=C)(C)C)C2CCCC2N1C(=O)CCc1cnoc1 12471,N1(C(=O)CCc2nc[nH]n2)CCC2(CC1)CN(C(C1C3COCC13)=O)CC2CO 12472,C(CC(C)C)(C(=O)N1CCCC(C)(C(N2CC(O)C(O)C2)=O)C1)NC(=O)OC 12473,C(C(C)(C)CNC(C1(OC(C)C)CCC1)=O)N(C(=O)CCc1conc1C)CC 12474,c1(-c2cc(OC)ncc2)nc(C(N2CCC(C(F)(F)F)C2)=O)ccc1F 12475,CCC(C)(CNC(C1(CNC(=O)Cc2ccnn2C)CC2(CC2)C1)=O)C(N)=O 12476,O=C1CN(CC(N2CCC3CC23C(=O)Nc2cnccc2CO)=O)CCN1 12477,CC(C)C(O)C(C)C(=O)N1CC=CC1(C)C(=O)NC1(C2CC2)CC1 12478,Cn1nc(C(=O)NC2CC(CNC(=O)C(c3ccccc3)F)C2)ccc1=O 12479,c1(CNC(C)=O)n[nH]cc1C(=O)NCCC1CCNC1=O 12480,Cc1cccc(N)c1C(=O)NC1CCC(N(C(=O)CCC2CNC(=O)N2)C)CC1 12481,N1(C(c2n[nH]c(CC)c2Cl)=O)CCC2(C1)CN(C(=O)C(c1ccc(Cl)s1)C)C2 12482,C=CCC(C(=O)N1CCCC(CNC(c2cc(CCCO)on2)=O)C1)NC(C)=O 12483,CC1CC(NC(c2cscc2C#N)=O)CCN1C(C1CN2CCC1CC2)=O 12484,C1(C)(CNC(C2(SC)CN(C(COC)=O)C2)=O)CC(F)(F)C1 12485,c1(C(=O)NCC2CC(NC(CC3C(C)(C)C(O)C3)=O)C2)ccnc2ccnn12 12486,c1(C(c2nnnn2CCCF)NCC2(C)CCC(=O)N2)cc(Cl)cc([N+](=O)[O-])c1 12487,c1(C(=O)NCCCC2N(C(c3c(C)ccs3)=O)CCC2)ccccc1OC1CC1 12488,CC1=C(CNC(=O)C(C(C)O)NC(=O)CC2CCCCO2)COCC1 12489,C1(C2CCN(C(=O)CCNC(c3ccc(F)cc3N)=O)C2)(NS(N)(=O)=O)CC1 12490,CC(C)CC(CNC(=O)CSc1ccccc1)C(=O)OCC(c1cn[nH]c1)C 12491,C1(N(C(c2cc(CC)on2)=O)C)CCCN(C(=O)CC2C=CCC2)C1 12492,c1(C(=O)NC2C(CNC(Cc3cnc(C)s3)=O)CC2)cc(F)c(C)cc1O 12493,C1(C)(C(N2CCC(CCNC(C3C(=C)C3C(=O)OC)=O)C2)=O)CCCCO1 12494,N1(C(CCSCCC)=O)CCC2(CC(C(=O)N(CC)Cc3ccc(F)cc3)C2)C1 12495,N1(C(C2C(C)C2)=O)CCC(CN(c2nn(C)cc2Br)CC2CC2)CC1 12496,c1(OC)c(C)cc(C(=O)N(CC)CC2CCCN2C(=O)C(O)P(C)(C)=O)cc1C 12497,CC1CCc2nc(Cl)nc(N3CCCCC(NC(c4coc(Cl)c4)=O)C3)c2C1 12498,N1(C(C2N(C(C)=O)CSC2)=O)CCC12CN(C(=O)CN(C1CCCC1)C)C2 12499,C1(CC)CN(C)CCCN1C(c1cncc(CNC(=O)C(F)C(F)(F)F)c1)=O 12500,CC(C)CC(=O)NC(c1nocc1C(=O)NCCCC1CCN1C(C)(C)C)C 12501,Cc1cc(C(F)(F)F)n2ncc(C(=O)NC3CC3NC(=O)C3=CCCC3)c2n1 12502,C1(C(N(C)CC2CC(F)C2)=O)CC2C=CC1N(C(C1CC=CC1)=O)C2 12503,C1(C(N(CCNC(=O)CNC=O)CC)=O)CCn2ncnc2C1 12504,N1(C(C2NCCCCC2)=O)CCCC2(CCC2)C1.CC1=C(C=O)CCC1 12505,c1(SC)c(C(=O)NC2CCC(NC(=O)C(N3CCCCCC3)C)C2)cccc1F 12506,c1(SC(C)CCNC(N2CCC(CS(C)(=O)=O)C2)=O)ccccc1Cl 12507,C(=O)(C1CCc2snnc21)NCC1CCN(C(C(CCC)NC(N)=O)=O)C12CC2 12508,N1(C(Cc2c(C)ocn2)=O)CCCC(C)(C)C1CNC(c1cnc(O)o1)=O 12509,N1(C(CCS(=O)(=O)NC)=O)CC2(C1)CN(C(C1CCC3(CC1)CC3)=O)CCO2 12510,C1(NC(C2C3COCC23)=O)CN(C(=O)C=CCF)C2(CCC2)C1 12511,c1(CCNC(C=C(CNC(CCCOC)=O)C)=O)cccc(C)n1 12512,C1(NC(Cc2ncc(CC)[nH]2)=O)CN(C(=O)Cn2cnccc2=O)CC1CC 12513,c1(OC)c(Cl)cc(C(=O)NCCC(C)NC(c2cc(C)oc2C)=O)cc1Cl 12514,N1(C(C(c2ccc(OC)cc2)CC)=O)CC(NC(c2occc2C)=O)CC(C)C1 12515,C(=O)(C(C)(C)C)NC(C)C(=O)NC1CC1NC(=O)C=Cc1ncco1 12516,c1(N(C)Cc2ccns2)ccc(S(=O)(=O)N2CCC3(CCOC3)C2)cc1Cl 12517,CC1CC(NC(c2cc(N)ccc2Cl)=O)CCN1C(=O)C=Cc1ncc[nH]1 12518,C(c1ccc(C)c(Cl)c1)=CC(C(=O)C=C(C)C)=O.C1(CC=C)(N)CCNCC1 12519,N1(CC(=O)NCC2(C(=O)NC(C(O)CO)C3CC3)CCCO2)CCCNC1=O 12520,c1(C(=O)NCC2CN(C(C3CC4(CCC4O)C3)=O)C2)ccc([N+](=O)[O-])cc1C(F)F 12521,CC(CCc1ccncc1)N=c1[nH]c2c(c(=NCCCCN(C)C)[nH]1)COC2 12522,N1(C(CCOC)=O)CCCCC(C(=O)NC(c2ccccc2)C(C)C)C1 12523,CCCCCCCCC(=O)NC1CC1NC(c1ccc(C(C)(C)C)s1)=O 12524,C(=O)(C1=C(Cl)CCOC1)N1CC(NC(Cc2c(C)nccc2)=O)C(SC)C1 12525,N1(C(CC(C)O)=O)CC(CNC(=O)CC2C=CCC2)C(F)(CO)C1 12526,C1(NC(CCC(C)OC)=O)C2CCC(C2)C1C(=O)NCC(O)C(N)=O 12527,N1(C(C(CCC)(C)C)=O)CCC2OCCN(C(C3CC4CC4C3)=O)C2C1 12528,n1(CCCC)nnnc1C(c1ccncc1)NCCSCC1CCCC1 12529,N1(C(c2c(CCC)n[nH]c2)=O)CC(CNC(c2ccn(CCF)n2)=O)CC1(C)C 12530,c1(CN2CCC(C(C)C(=O)N3CC(n4cnnc4)C3)CC2)cc(Cl)ccn1 12531,N1(C(C=C(CCC)C)=O)CCC(CNC(C2(OC)CCCOC2)=O)C(F)(F)CC1 12532,c1(C(N2CC(C)N(C(c3csc4cncn34)=O)CC2)=O)ccnc(P(C)(C)=O)c1 12533,c1(OC(C)C(=O)NC(C)CC2CN(C(C3CSCN3C)=O)C2)ccc(F)nc1 12534,N1(C(c2cc(C)oc2C)=O)CCC(NC(=O)Cn2ccnn2)C(CO)CC1 12535,c1(C(=O)NCC2CC(NC(C(C)Sc3ccccn3)=O)C2)cc2ccccc2o1 12536,C1(C(N(C)Cc2c(CNC(CSC)=O)cccc2)=O)CCOCC1(C)C 12537,C1(NC(c2ccc(SC)s2)=O)CC2CN(C(c3ccc4[nH]ccc4n3)=O)CC2C1 12538,c1(NC2C3CN(C(C4CC=C(C)CC4)=O)CC32)nc2cc(C)ccc2o1 12539,CC(C)(CCNC(c1c[nH]nc1Cl)=O)C(=O)NC1C2CCC1CC2 12540,C1(OC)CC(NC(=O)C=C(Cl)Cl)CN(C(C2CCS(=O)CC2)=O)C1 12541,C(=O)(CCCC(=O)NC(=O)C=Cc1ccsc1)NC1C(CC(=O)OCC)CCC1 12542,Cc1cc(F)sc1C(=O)N(CCCCCCNC(c1ccn(C)c1)=O)C 12543,CC1(C(=O)NCC2CC(NC(c3cccc(CF)c3)=O)C2)CC2CC2C1 12544,Cc1ccc(C(=O)NCC(C2CCC2)NC(=O)C(C)(C)c2ccns2)s1 12545,N1(C(CCc2c(C)cccn2)=O)CCC(CNC(C2CCCOC2)=O)C(C)C1 12546,C=CCC(CC(C)C)C(=O)N(CC(O)CNC(=O)COc1ccc(F)c(F)c1)C 12547,C#Cc1ccc(C(=O)NC2CC(NC(C3(C)CC=C(C)CC3)=O)C2)nc1 12548,N1(C(C(COC)N(C)C)=O)CCCC(CC(=O)NCCC2CC(C)(C)CO2)CC1 12549,C(C1=NOC2C3CCC(C3)C12)NC1CC(OCC)C1(CC)CC 12550,CC1CN(C(=O)Cn2ncnn2)CC(CCNC(=O)CC=CC(C)(C)C)O1 12551,C(=O)(C(C)(C)C(C)(F)F)NCC1N(C(CC(CC)SC)=O)CCOC1 12552,c1(C(=O)NCC#CCNC(c2cc(CC)nnc2C)=O)cnc2ccnn2c1C 12553,N1(C(c2ccc(C)nc2C2CC2)=O)CCOC2(CCN(CC3CCC3)CC2)C1 12554,C1(C(=O)NC2CC(CNC(C3CC4(CCC4)C3)=O)C2)CC12CCCOC2 12555,C1(NC(=O)C=C2CCOCC2)CC2CC1CN(C(C1CCCCC1)=O)C2 12556,CC1(C#N)CCN(C(=O)CCC2(NC(=O)C(=O)NC3CC3)CCCC2)C1 12557,N1(Cc2ccc(C(CC)C)cc2)CCCCCC1N=c1ccc(C#N)n[nH]1 12558,CC1CN(C(=O)Cc2nc(C3CC3)n[nH]2)CC1NC(=O)CC1CC1 12559,CON1CCC(C(=O)NC(CN(C)C)C(=O)NCC2(F)CCOCC2)CC1 12560,C1(C(=O)NC2CC3(C(NC(c4c(C)nc(CO)s4)=O)C3)C2)COC2CCCCC12 12561,C(=O)(C(C)(C)C(C)O)NCCn1cc(C(N(CCCC)CCOC)=O)nn1 12562,c1(COCC)ccc(C(=O)NCC2(C)CCCN2C(C2CC(C)=NO2)=O)cc1 12563,N1(C(C(c2n(C)ncc2)NC(=O)C(O)C2CCCC2)=O)CC2CCC(C1)C2C#N 12564,C#CCC(C(=O)NCCCSC)NC(=O)C(=Cc1cn[nH]c1)C 12565,C1(SC)CCN(C(=O)CCOCCN(C(=O)C(C)Cc2cnc[nH]2)C)C1 12566,CN1CCN(C(c2sccc2CNC(=O)CNC2CCCC2)=O)C(C2CCC2)C1 12567,C(=O)(C(C)S(=O)(=O)C(C)C)NCC(CNC(C(CC)(CC)CC)=O)C 12568,C1(c2nnnn2CC(c2ccccc2)OC)(CC2(COC)CC2)CCCSC1 12569,c1(CC(=O)NCC(C(C)(C)C)NC(c2c(CC)ccs2)=O)ccc(OC)c(C)c1 12570,C1(C)(COC)CCCN(C(=O)C(c2ccnn2C)NC(=O)C(C)n2ccnc2)C1 12571,N1(C(C2N(C(C(=Cc3cn[nH]c3)C)=O)CCOC2)=O)C2CCC1COC2 12572,CC1CCCC(O)(C(=O)NCC2(F)CN(C(c3ccc4cc[nH]c4n3)=O)C2)CC1 12573,c1(C(=O)NC2C(NC(c3c(C)cco3)=O)CC2)cc(F)c(F)c(O)c1F 12574,c1(C(=O)NCC(C)NC(C(CC)n2cncn2)=O)cnc(C)n1C 12575,CCCCC(S(=O)(=O)NC(=O)C(c1ccc(Br)nc1)(C)C)c1ccccc1 12576,CC(C)CC(C)(CNC(c1cc(Br)n[nH]1)=O)NC(=O)Cc1cccn1C 12577,Cn1cc(C(F)=CC(=O)NCC2C=CCN2C(=O)CC2CCCC2)cn1 12578,c1(C(=O)NCC2N(C(c3c(C)cncc3)=O)CCOC2)nc(C2CC2)ncc1Cl 12579,N#Cc1ccc(C(N2CCC(C3(NC(=O)CCCCC(N)=O)CC3)C2)=O)cc1F 12580,c1(C(N2CCN(C(=O)Nc3cccc(C)c3)C3C2C3)=O)nncc2c1CCCC2 12581,N1(C(C(C)O)=O)C2CCC1CC(NC(c1ncsc1Br)=O)C2 12582,c1(CNC(C#C)=O)nc2c(s1)CCN(C(=O)CS(=O)(=O)N1CCCCC1)C2 12583,C1(F)(C(=O)NCCC2CC(NC(Cc3cnc(C)o3)=O)C2)CCCOC1 12584,C(CCC(=O)NC1C(NC(=O)C(C)OC(C)=O)CC1)SC 12585,c1(OC)nc(Cl)ccc1C(N1CCC(NC(c2ncccc2C)=O)CC1C)=O 12586,N1(C(CCCn2cc(CC(C)(C)CO)nn2)=O)CC2CC2(CN2CCCC2)C1 12587,CCCCCC(CC)C(=O)NCCOCCNC(c1c[nH]c2cccc(C)c12)=O 12588,N12CCC3(CC3C1)C2=O.c1(OC)cc(CNC(=O)COc2cc(C)on2)ccn1 12589,N1(CC(=O)NC2C3CC2N(C(c2snc(O)c2Cl)=O)C3)CCCCCCC1=O 12590,c1(C2(C(=O)NCC(C)CN(C)C)CCCC2)ccc(Cl)cc1 12591,C(C(CC(F)(F)F)NC(C1CC1C#N)=O)NC(c1cnc(C(C)C)[nH]1)=O 12592,N1(C(C(CC)OC)=O)C2CCC1CC(CC(C)NC(=O)CCc1ccnn1C)C2 12593,C(=O)(N1CCCc2nncn21)C1C2(CCN(C(c3cc(OCC)no3)=O)C2)C1 12594,CC(C)CC(C)(CNC(C1CN(C)CC(C)O1)=O)NC(c1c[nH]cc(Cl)c1=O)=O 12595,C(N=c1nc2c(cnn2C(C)C)c(NCC2CC=CC2)[nH]1)c1ccc(C)cc1Br 12596,C1(NC(C=C(C)C2CC2)=O)CN(C(C23CCCC(C2)OC3)=O)C2CCCCC12 12597,C(CCS(=O)(=O)c1ccc(F)cc1)NC1C(C)CN(C(=O)C(=O)NC2CC2)CC1 12598,c1(SC)cccc(N2CC(c3nc(C4CCCC4)nn3C3CCOC3)CC2=O)c1 12599,C=C1CC2CCC(C1)N2C(=O)C(CCCC)NC(c1coc(C(F)F)c1)=O 12600,C1(NC(C=CSC)=O)CS(=O)(=O)C2CN(C(c3cc(Cl)no3)=O)CC12 12601,Cc1nn(CCC(=O)NC2CCCC2CNC(c2cncc(N)n2)=O)cc1Br 12602,C1(C(N2CCC(O)(C(C)NC(=O)COCCF)C2)=O)CS(=O)(=O)CC(=O)N1 12603,c1(NCC2C(C)CCN(C(=O)CC3(C)CC3)C2)ncnc2cnccc12 12604,C1(C(N(C)CCNC(c2ccc3c(c2)OCC3)=O)=O)C2C3CC4C1C1C2CC3C41 12605,N1(C(c2c(C)cnnc2)=O)CCC2(CC2)CC1C(=O)NCCCc1ncn(C)n1 12606,C1(C)(CNC(CC=C)=O)CN(C(c2coc(COC)n2)=O)CC1C 12607,N1(C(c2ccn(CC)c2C)=O)CC2(C1)CN(C(c1cc(C3CCC3)[nH]n1)=O)C2 12608,C(=O)(C(F)(F)CCCn1cc(CCO)nn1)NC(c1cnc2n1CCCC2)C 12609,CC(CC(F)(F)F)C(=O)N1CC2(CC2)CC1C(=O)N(C1CC1(C)C)C 12610,C1(C)(CCCC(=O)N(CCCCN(C(CN(C)C)=O)C)C)NC(=O)NC1=O 12611,c1(C(N2CC3(N(c4nccc(C#N)n4)CC3)C2)=O)cccc2c1OC(F)(F)O2 12612,Cc1csc(=O)n1CC(N1CCC(C)(NC(=O)C(C)Cn2cccn2)C1)=O 12613,c1(CC(=O)OC(C)C(=O)N2CC(n3cnnn3)C2)cc(Br)cs1 12614,N1(C(C(c2ccc(C#N)cc2)C)=O)CCCC2(CNC(=O)C=Cc3cccs3)CC12 12615,N1(C(C(c2cccc(C)c2)O)=O)CCC(C)N(C(c2ccn(C3CC3)n2)=O)CC1 12616,C1(C(CN(C(C)=O)C)(C)O)CCCN(C(=O)Cc2cnc(C(C)C)[nH]2)C1.C1C(=O)N1 12617,c1(C(N2CC(C)(NC(CCC)=O)C2)=O)cc2c(F)ccc(Br)c2[nH]1 12618,C12(CNC(Cc3c(C)nsc3)=O)CCC(CC1)N2C(C1C2CC3C(C2=O)C13)=O 12619,C1(C(N2C(CNC(C3(CC)CCC3)=O)CCCC2)=O)CCOC(=O)CC1 12620,Cc1ccn2ncc(C(N3CCN(C(=O)CCC4CCC4)CC3C(C)C)=O)c2n1 12621,N=c1[nH]c2c(s1)CCCC2C(=O)NCC1(O)CCCN(C(=O)C(O)C(F)F)C1 12622,CC(C)(CCCO)NC(C1CSCCN1C(C1CCCCC1)=O)=O 12623,c1(C(=O)Nc2nc(-c3ccc(OCOC)c(Cl)c3)sc2)cc2n[nH]cc2cc1Cl 12624,C1(C(=O)NC2(CC(=O)N(CC(C)N(C(C)=O)C)C)CC2)CCCC(F)C1 12625,c1(C(=O)NC2(N3CCCC3)CCC2)ccnc(C(=O)NC2CC(N(C)C)C2)c1 12626,c1(NC(CC)=O)cncc(C(N2CC(=C(F)CNC(=O)C=C(C)C)C2)=O)c1 12627,CN1CC(CNC(=O)CCN(CCCO)C(=O)CC2CCC(C#N)C2)CC1=O 12628,C12(NC(C3OCCN(C(C)C)C3)=O)CC(CNC(=O)C(C)(C)CF)(C1)OC2C 12629,N1(C(C(OC)OC)=O)CC2C(CNC(=O)CNS(=O)(=O)N(C)C)C2C1 12630,C1(NC(N2CCOC(CO)CC2)=O)CCC2(CCOCC2)C1 12631,C(=O)(CC1=CCOCC1)NC(COC)CC(=O)NCC1(OC)CCCCC1 12632,C(C(=O)NCCC1(C)CCOC1)(C(C)(C)O)NC(C1CCC(CC)O1)=O 12633,c1(CC)cc(CC(=O)NCCN(C(=O)CCCc2cnccn2)CC)on1 12634,CCCCCCCN(C(=O)CCCn1cc(C(C)(C)CO)nn1)C(=O)OCC 12635,C12CCN(C1)CC(=O)N2.CCC(CC)N(C1CCC1)C(C1CC(N(C)CC)C1)=O 12636,N1(C(C2CNC(=O)N2)=O)CC(NC(=O)COC2CC2)C(c2ccc(F)cc2)C1 12637,C1(C(=O)NCc2n(C(C)C)ncn2)CCN(c2nc(C(C)(C)C)co2)CC1 12638,C(C(O)CC(=O)NCC(=O)NC(C)C)NC(c1c(COC)cc[nH]1)=O 12639,O=C1CCC(C(=O)NCCOC2CN(C(c3ccccc3C(F)F)=O)C2)CN1 12640,c1(CC(=O)NCC2(OC)CCN(C(=O)Cc3cnsc3)C2)cccc(C)c1Cl 12641,Cc1cc(F)sc1C(=O)NC(C1CCN(C(C2CC2(C)C)=O)C1)C 12642,N1(Cc2cccc(OC)c2)CCN(C(=O)C(F)(F)F)CC(C)(C)C1 12643,c1(C(N(C2CN(C(c3cnc(CCC)s3)=O)CC2O)C)=O)nccc2ccsc12 12644,Cc1cc(Cl)c(NC(C2CSCCS2)=O)cc1O 12645,CC(C)(C#CC(=O)NCC(C)(O)C1CC1)CNC(=O)CN1CCOC1=O 12646,C1(CC)CCc2sc(C(=O)NCC3CC(NC(=O)CC4(C5CC5)CC4)C3)cc2C1 12647,CC1COc2ccc(C(N3CC4CN(C(=O)CC5=CCCC5)CC4(C)C3)=O)cc21 12648,N#Cc1cncc(NC2(CNC(=O)C=CC(=O)NC3CC3)CCOCC2)n1 12649,C(=O)(CCCCCC(C)O)N(CC(CN(C(C(C)N(C(C)=O)C)=O)C)O)C 12650,Cc1cc(Cl)c(Cl)cc1NCc1nc(-c2ccoc2C)no1 12651,C(N=c1[nH]c(C(F)F)nc2ccccc12)C1N(C(C2=C(C)OCCS2)=O)CCC1 12652,S(=O)(=O)(c1cnccc1NC(=O)Nc1cccc(C(C)C)c1)N(CCOC)CC 12653,c1(C2C(CNC(=O)Nc3sncc3Br)CC2)ccccc1 12654,N1(C(C2C(CC)CCCC2)=O)CC2(C1)CN(C(c1nc(F)ccc1Cl)=O)CCO2 12655,c1(C(=O)NC2(CC=C)CCN(C(=O)CC(C)OC)C2)cc(C)cc(Br)c1 12656,C1(C(N(C)CC2(O)CN(C(=O)C=Cc3cc[nH]n3)C2)=O)COCCN1C 12657,c1(NC(C(C)NC(CC)CNC(C2CC=C(C)CC2)=O)=O)cccc(C)c1F 12658,N1(C(C(c2ccn(C)c2)C)=O)CC2CCCC(N(C(=O)CSC(C)(C)C)C)C2C1 12659,c1(C(=O)NCC2CCN(CCOC)C2)c[nH]c(C)c1Cl 12660,CN1CCCC2CN(c3cc(C(=O)O)c4c(c3)CCCC4)CCC12 12661,CCN=c1[nH]cc(C(=O)NC2CC(CCn3cc(C(C4CCCC4)C)nn3)C2)s1 12662,N1(C(Cn2ccc(C)cc2=O)=O)CCC(C)N(C(=O)CC2CN(C)CC2O)CC1 12663,C(=O)(C1=C(Cl)CCOC1)NC1(CC=C)CCN(C(C2CCCCC2O)=O)CC1 12664,N1(C(c2nn(C)c(O)c2)=O)CCN(C(c2cc(N)c(Cl)cn2)=O)C(CC(F)F)C1 12665,c1(CNC(C(C)NC(=O)CCCc2cnn[nH]2)=O)c(O)cccc1F 12666,c1(C(=O)NC(C)(C)CNC(c2ccc(N)cc2)=O)cc2ccc(O)nc2s1 12667,N1(C(c2cccc(N)c2Br)=O)CCOCC(F)(CNC(c2cnc[nH]2)=O)C1 12668,CCC(CN=c1cc(NCCCCN2CCCCC2C)nc[nH]1)OC 12669,CC#CCCC(=O)NCC(C1CCOC1)NC(=O)Cc1cnn(C)c1C(F)F 12670,C1(NC(C(C)=CC)=O)CN(C(C2(C3CC3)CCCC2)=O)CC1c1ccccc1Cl 12671,c1(C(N2CCC(CCNC(C(CC)N(C)C)=O)CC2)=O)cc2ccc(O)nc2s1 12672,CC(C)CCC(C(=O)NCC(C)(O)CO)NC(c1cn(C)cn1)=O 12673,c1(NC(CC)=O)ccc(C)c(C(=O)NC(c2ncc(Br)cn2)C2CC2)c1 12674,C1(NC(=O)C=CC2CCOC2)CCCC12CCN(C(C13CC(C1)C3)=O)CC2 12675,c1(C(=O)NC2(CNC(CCN(CC)CC)=O)CC2)nnc(S)n1C 12676,N1(C(c2ccc(OC)c(O)c2)=O)CCC2(C1)CN(C(c1ncsc1C1CC1)=O)C2 12677,c1(C(N2CCN(C(C3CC(=C)C3)=O)C(C)C2)=O)cc2ccccc2nc1O 12678,c1(NCC2OCCN(C(CCC(=O)N(CC)CC)=O)C2)ncn(C)c(=O)c1Br 12679,Cc1cnn2ccc(C(N3CCC(C(C)NC(=O)CP(C)(C)=O)C3)=O)nc12 12680,C1(SC)CN(C(c2cc(C)ccc2Cl)C(=O)NC2CCCC2)C2(CCC2)C1 12681,N1(C(CSCc2ccc(C)cc2)=O)CCC(C2(NC(=O)C(C)O)CC2)C1 12682,C(=O)(C(O)P(C)(C)=O)NCC(CN(C)C(c1cncc(C(C)(C)C)c1)=O)(C)C 12683,N1(C(C(CCOC)OC)=O)CC(CO)C2(C1)CN(C(=O)CN1CCS(=O)CC1)C2 12684,C(=O)(C(CNC(=O)CC(F)(F)F)C(C)(C)C)NCCc1cn(CC)nn1 12685,CC(C)S(=O)(=O)c1ccccc1C(=O)NC1CCN(C(C2CC(F)C2)=O)C1 12686,c1(C(=O)NC23CC(CNC(CC4CCCN(C)C4)=O)(C2)C3)ccc(F)cc1Cl 12687,C(=O)(C(F)(CNC(C12CCC(C1)C2)=O)C(C)C)N(C(c1ncc(C)[nH]1)CC)CC 12688,Cn1cc(-c2n[nH]cc2C(=O)Nc2nc(C3CC3)cs2)cn1 12689,C(CCCCC(C(=O)NCCCC1CC1)OC(c1cccc(CSC)c1)=O)OC 12690,O=S(=O)(c1ccccc1N1CC(O)CC(F)C1)NCCOC1CC1 12691,C(=O)(CCCC(F)(F)F)NCCOCCN(C)C(c1nccnc1-n1ccnc1)=O 12692,C1(COC)CN(C(=O)CC2(CO)CC2)CCN1C(C1CC1n1ccnc1)=O 12693,c1(C(N(C(CCNC(C(CCCC)C)=O)C)C)=O)cccc(S(=O)(=O)CF)c1 12694,C12(C(=O)NC3CCCCN(C(Cc4c(Cl)cc(C)s4)=O)C3)CC1Cc1c[nH]nc12 12695,C(N=c1[nH]c(=NC)[nH]c(=NCC2C=CCCC2)[nH]1)c1ccc(N(CCC)CC)cc1 12696,c1(N(C)CCOC(F)F)nc(=NCc2cc(Br)ccc2C)[nH]c2c1CSC2 12697,Cn1cc(C=CC(=O)NCC2(C(=O)NCCC3CC3C3CC3)CC2)nn1 12698,C1(C(C)NC(C(CC)NC(N)=O)=O)CCN(C(=O)CCCC2CC2)CC1 12699,C1(COC)(CNC(=O)CCC2CCOCC2)CCN(C(C2CC(=O)N(C)C2)=O)C1 12700,C#CCC(C)(C)C(=O)NC(CNC(=O)C(C)n1ccnc1)CCOC 12701,C1(C(C)=O)CC(CC(=O)NC2(CN)CC2)C1(C)C.C(=O)(CCC(=O)c1cccs1)N 12702,C=C(F)CN=c1[nH]c2c(c(=NC3CC(=O)N(CCC)C3)[nH]1)SCC2 12703,N1(Cc2cn(CC(N3CC(C)C(C(F)(F)F)C3)=O)nn2)CCCCC2(CCC2)C1 12704,c1(C(=O)OC)c(NC(=O)CCC(C)(C)OC)sc2c1CCC(C)C2 12705,C(=O)(C(C(F)(F)F)C(F)(F)F)N1CCCC(C(N2CC(C)(C)n3c2ccc3)=O)C1 12706,C(=O)(C(C)(C)C(O)C(C)C)N1CCCC(C)(C(=O)NCc2ccc(OC)cc2)C1 12707,S(=O)(=O)(c1ccncc1)NCc1c(NC(c2ccco2)C)cccc1 12708,C1(n2c(C3CCCN(C(C)C)C3)nc(-c3ccc(Cl)cn3)n2)CCCS(=O)(=O)C1 12709,CCC(C(=O)NC(CNC(c1cc(C2CC2)ns1)=O)Cc1ccccc1)NC(N)=O 12710,C1(C2CN(C(=O)C=C(C)Cl)C2)(NC(C2ON=C(CC)C2)=O)CC1 12711,c1(C(N2CCC(C)C2CNC(=O)C(F)(F)c2ccsc2Cl)=O)ncc(N)cc1Cl 12712,c1(N(C(=O)C(C)c2ccon2)C(C)CN(C(=O)Cc2ccccc2)C)cccnc1O 12713,c1(C(c2nnnn2C2(C)CC2)N(CCCC#C)CC)nc(CCCOC(C)=O)cs1 12714,C1(NC(C2C(C)N(C)CC2)=O)CCC12CN(C(=O)CCCc1ccccc1)C2 12715,C(CC(=O)N=c1cc[nH]c(CO)c1)C1N(C(c2cc(OC)cc(Cl)c2)=O)CCC1 12716,C1(CCNC(c2cnn(CCC)c2C)=O)CCN(C(=O)CN(C)CCO)C(C)C1 12717,C1(NC(C2OCCC(NC(C3NC(=O)CC(C)C3)=O)C2)=O)CCCCC1N=[N+]=[N-] 12718,CCCC(C)(C)CC(=O)N1CC2CCC2(CC(=O)NCc2cc(C)ncn2)C1 12719,c1(C(=O)NC(CNC(C(F)=CC)=O)CC(F)(F)F)cc(=O)n2nccc2[nH]1 12720,CN=c1ncc(-c2nc(C(N3CC4CCC(C3)O4)=O)cs2)c[nH]1 12721,C1(NC(c2cnn(C3CCC3)c2)=O)CN(C(c2ccsc2Cl)=O)CCC1CO 12722,N1(C(Cc2scc(C)c2)=O)CCC(C)(NC(c2scnc2C)=O)C1 12723,C1(NC(C2CC(C)(C)C2)=O)CC(NC(c2coc(Br)n2)=O)C12CCOCC2 12724,N1(CC2OCC(CN)C2)CCc2cc(C(F)(F)F)ccc2C1 12725,C(=O)(CC(O)CC(C)C)NCC(CCC)C(=O)NC1C=CC(C(=O)OC)C1 12726,C(=O)(C1c2c[nH]nc2CN1C(=O)CCCn1ccnc1)NCC(N1CCCC1)C 12727,c1(C(=O)NCCOCCC(=O)NCC=C)ccc(CC)o1 12728,c1(NC(C)=O)ccc(Cl)c(C(=O)NCC(C)NC(=O)C(c2ccccc2Cl)O)c1 12729,c1(CC)cc(C(=O)NCc2n[nH]cc2C(=O)NC2CCCC2C#N)ncn1 12730,c1(C(=O)NCC2N(C(C3C(C=C)C3)=O)CCC2)cc(F)cc(Br)c1Cl 12731,C(=O)(C1=CCC(NC(C2CCCCS2)=O)C1)N1CC(C)(O)C1 12732,C1(CNC(=O)NCC2CCC(C(=O)OC)C2)CCCC(C)(C)CC1 12733,N1(C(C(CCC)O)=O)CCC(C(C)C)CC1CNC(=O)Cn1nnnc1C 12734,Cn1ccn2ncc(C(N3CC4C(NC(=O)C=Cc5cc[nH]c5)C4C3)=O)c12 12735,C1(NC(C(CSC)O)=O)CC2CC1CC2C(=O)NC(CCO)C(C)(C)C 12736,C=CC(CC)CC(=O)NCc1ccc(C(=O)NC2CN(C)CC2(F)F)cc1 12737,c1(C(N(C2CCN(C(C3(C#N)CC3(C)C)=O)C2)C)=O)cn2c(Br)cnc2s1 12738,Cc1nn(C)c2ncc(C(=O)NCC(C3CC3)N(C)C(c3coc(O)n3)=O)cc12 12739,C(=O)(C1Cc2ccc(Cl)cc21)NC(CCCC)CNC(c1cc(C2CC2)[nH]n1)=O 12740,C(=O)(C(C)(C)N(C)C)NCCC(C)N(C)C(c1ccc(Br)o1)=O 12741,c1(C(N2C(C)(CNC(c3ccsc3C(F)F)=O)CCC2)=O)ccc2nonc2c1 12742,c1(CCC(=O)NC(C)CNC(C2(CC3CCC3)CC2)=O)ccc(Br)s1 12743,c1(CCC(=O)NC(CC2CCS(=O)(=O)C2)C(=O)O)cccc2cn[nH]c12 12744,c1(C(C(=O)OC)N(CCCCO)CC2CCNCC2)ccc(Br)cc1Cl 12745,C(=O)(C(C(=O)N1CC(CC(C)NC(c2cc(OC)cnn2)=O)C1)OC)OC 12746,N1(C(CC2(N(C)C)COC2)=O)CCC2(CC1)CC2NC(=O)CC1CC=CC1 12747,c1(C(=O)NCC2CCC(NC(c3c(CC)non3)=O)C2)nccc2c1NCCC2 12748,N1(C(C(C)Nc2cc(Br)ccn2)=O)CCOC(C(=O)NOC(C)(C)C)C1 12749,C(=O)(C1=Cc2ccccc2C1O)N1CC(O)(CNC(c2cncc(CC)c2)=O)C1 12750,c1(CC)c(N2CCC(NC(C3CC34CCC4)=O)CC2)ncnc1Cl 12751,C(=O)(C(C)C(F)(F)F)NCCC(C)(C)NC(c1c(C)nc(CCCC)s1)=O 12752,CC1(C)NC(=O)N(CC(N2CCCC(O)(CNC(=O)C(=O)NC3CC3)C2)=O)C1=O 12753,CCC(CC)CC(=O)N1CC(O)(CNc2nccc(-c3cnccn3)n2)C1 12754,C#Cc1ccc(C(=O)NC(CCN(C)C)C(=O)NCCc2nnc(C)n2C)cc1 12755,C=C(Br)CC(=O)NC(C(CO)NC(C1CC1(Cl)Cl)=O)C1CCCC1 12756,c1(OC)cscc1C(=O)NC(CNC(=O)C(C)Sc1ccccc1)C(C)C 12757,CCCC(CCCNC(C1CC1(F)F)=O)NC(=O)CCCCc1ccccc1 12758,c1(C(=O)NC2CCC(NC(CCSCCCC)=O)C2)nccnc1C(F)(F)F 12759,C1(F)(C(N(CCn2cc(COc3cc(Cl)ccc3Br)nn2)CC)=O)CCS(=O)(=O)C1 12760,CCCC(CC)CCC(=O)NCCC(C)(C)NC(C1CCCCC1OC)=O 12761,CC1=NN(C)C(=O)C1CC(=O)NC12CC1CN(C(=O)CC1CCOCC1)C2 12762,N1(C(CSCC#C)=O)CCC(CNC(=O)C(O)Cn2cncn2)(OC)C1 12763,C1(NC(c2nc(CC)oc2C)=O)COC2(CNC(=O)C(C(C)C)SC)CC1C2 12764,C1(CCN(C(=O)C(O)Cn2cncn2)C)CCCCN1C(=O)CCC#N 12765,c1(C(N2CC(OC)C(NC(=O)COC(C)=O)C2)=O)cccc2c1OC(C)(C)C2 12766,Cc1cccnc1CC(=O)NC1CCC1CNC(=O)C(c1cccn1C)=O 12767,c1(OCCCC)ccc(Nc2cc(CN(C)C)nn2C)c2cccnc12 12768,C1(O)(CNC(c2cc(OCC)n[nH]2)=O)CCN(C(=O)CCC2CC(F)(F)C2)C1 12769,C1(C(=O)NCc2ncc(C)[nH]2)CC12CCN(C(=O)C(F)C1CCCC1)CC2 12770,C1(NC(c2ccc(Cl)cc2)=O)CN(C(=O)C(O)Cc2cnc[nH]2)CC1CC1CC1 12771,CCC(CC(=O)NC1CCN(C(C2CC23CCCCC3)=O)C1(C)C)CC(C)C 12772,c1(C(=O)NC(C)C(C)NC(c2c(F)cncc2Cl)=O)cc(F)cc2cc[nH]c12 12773,C1(CN(C(CC)=O)CC)C2CN(C(=O)CC3(C(F)(F)F)CNC(=O)C3)CC12 12774,N1(CC)CCN(CC(=O)NCC(CO)NC(=O)Cc2ccco2)CC1 12775,N1(C(Cn2cc(Cn3c(C)ncn3)nn2)=O)CCC2CC2C1 12776,c1(C(N(C2CCN(C(=O)C(C)C(C)O)C2)CC)=O)cnc(C)cc1C 12777,C(=O)(C(C)CCC(C)(C)C)NC1(CCC(=O)Nc2ccc(C)cc2)CCCC1 12778,c1(N(C)Cc2c(C)ccnc2)nc(N(C)CC2CC(F)C2)nc2ncn(C)c12 12779,c1(C(=O)NC2(C)CC2)cn2c(n1)CCN(C(=O)Cn1cc(S(C)(=O)=O)cn1)CC2 12780,C(=O)(C1=CS(=O)CCC1)NCCC(C)NC(c1nnc(Cl)cc1N)=O 12781,C1(CCC(=O)NCCN2CC3CC3C2)CCCCN1C(=O)C=Cc1ccco1 12782,C(=O)(CCC(=O)NC1CCCC1CNC(=O)C=CS(C)=O)NC(C)=O 12783,Cc1cnc(C)c(C(=O)NCC(C)CN(C)C(c2sc(F)cc2Cl)=O)c1 12784,C(=O)(C1=CC2CCC1C2)N1CCCC(N(C)C(c2cccc(Cl)c2)=O)C1 12785,c1(NC(C2N(C(c3n(C)nc(CC)c3Br)=O)C(C)CC2)=O)c(C)ccc(I)c1C 12786,c1(N(C)CC2CCN(C(=O)CC3CCCCO3)C2)nccnc1C#N 12787,C1(NC(c2n(CCOC)ncc2)=O)CCCC(NC(C2OCCCO2)=O)CC1 12788,C1(NC(CCn2c(C)ccc2C)=O)CCN(C(c2ccncc2N)=O)C12CCC2 12789,c1(N(C)CCc2ccc(F)cc2)nc2cc[nH]c2c(=NCC2(C)CC3(CC3)C2)[nH]1 12790,O=C(C1=C(Cl)CCCC1)NC(C12CCC(CC1)C2)CNC(C1CS(=O)(=O)C1)=O 12791,C(C)(CCCCNC(c1onc(C)c1C)=O)NC(c1n(CCC)ncc1)=O 12792,C1(NC(CCc2c(C)noc2Cl)=O)CC1C1CCN(C(=O)C(C)C2CCC2)CC1 12793,C1(O)(CNC(C2(N(C)C)CC2)=O)CCN(C(c2cc(Cl)ccc2F)=O)CC1 12794,c1(C(=O)NC2(CNCC3(C(CC)=O)CC3)CCOCC2)cccc2oc(C)cc12 12795,CCC(C)(CNC(c1cccn1C(C)C)=O)C(=O)NCC1OCCCC1(C)C 12796,CC(CNC(=O)CC=CCNC(=O)CCn1ccnc1)Cn1cccn1 12797,C(=O)(C(C)(C)C(F)(F)F)N1CC(CNC(Cc2cccc(SCC)c2)=O)OCC1 12798,CCS(=O)(=O)CCNC(C1(CNC(C2CC2(F)Cl)=O)CC(=C)C1)=O 12799,c1(C(=O)NCC2CN(C(CS(=O)(=O)NC)=O)C(C)C2)nn(C)c(Cl)c1Cl 12800,c1(CNC(C(CCOC)NC(=O)CSC(F)F)=O)cccc(F)c1F 12801,C1(NC(CC2(NC(C)=O)CCCCC2)=O)CC(F)CN(C(=O)CCS(C)(=O)=O)C1 12802,c1(NCc2ccc(CC(=O)NC3(F)CCNCC3)cc2)ncnc2ccccc12 12803,N1(C(C(N2CCOCC2)C)=O)CC2CC(NC(=O)C=Cc3cccnc3)CC1C2 12804,c1(C(N2CC(CCNC(C3CCC(C)O3)=O)C2)=O)cccnc1OCC(F)(F)F 12805,C1(C(N(C)Cc2snc(C)n2)=O)CN(C)CCN1C(c1cccc(O)c1)=O 12806,C1(OC)CC2CC(NC(c3cccnn3)c3nnnn3CCOCC3CC3)CC12 12807,c1(C(N2CCC(NC(c3ccc(OC)nc3)=O)C2C)=O)cc(Cl)cc2c1OCC2 12808,C1(C(=O)OC)CCN(C(=O)COC2CN(C(C3COCC(C)O3)=O)C2)C1C 12809,C1(NC(CCCCC=C)=O)CN(C(=O)C(C)(C)C2CCOC2)CC(F)(F)C1 12810,N1(C(CCC(=O)NCCC)=O)CCC2CCCN(C(=O)CCCC(C)CC)C2C1 12811,C1(C)(C(N(CCS(C)(=O)=O)C)=O)CCN(C(C2CC2c2ccco2)=O)CC1 12812,C(C(C)N=c1nc(N(C)Cc2cc(F)ccc2F)c2sccc2[nH]1)c1ccc(C)s1 12813,N1(C(C(C(C)NC(C(CC2CC2)OC)=O)C(C)C)=O)CCCC12CCOC2=O 12814,N1(C(C(C)OCC=C)=O)CC(C(=O)N(c2ncccn2)CC)CC(F)C1 12815,CC1CCCCC1(CNC(c1ccc(=O)oc1)=O)NC(C1CC2CCC1C2)=O 12816,C(CN=C(NCC(=O)NC(C)C)N1CCCC(OC)C1)C1(OC)CCC1 12817,N1(C(c2cc(F)cnc2O)=O)CC2=C(C1)CN(C(c1ocnc1C1CC1)=O)C2 12818,N1(C(C(CC)C)=O)CC(C)CN(C(C2CCc3c[nH]nc3C2)=O)C(C)C1 12819,C1(C(=O)OC)(OC)CCN(C(=O)C(CN)Oc2ccccc2)C1 12820,C(=O)(C#CC1(C)CCCO1)N(CCCCN(C)C(C1(C)CC1Br)=O)C 12821,c1(C(N(C)CC2CCN(C(Cc3c(C)ccs3)=O)CC2)=O)csc2ccncc12 12822,N1(C(c2cc(CC)oc2C)=O)CC2CCC1CN2C(=O)CCC1CCN(C)C1 12823,Cc1nnc2n1CC(C(=O)NCCC(C(C)C)NC(=O)CCCNC(N)=O)CC2 12824,Cn1cc(Cl)c(C(=O)NCC2CC2NC(c2ccc(OCC(F)(F)F)cn2)=O)n1 12825,CC1(C)CC(C(=O)NC2CC3CCCC3C2)CN(C(=O)CCN2CCCCC2)C1 12826,C1(NC(=O)CCCn2cccn2)CS(=O)(=O)CC1NC(C12CCCN1CCC2)=O 12827,N1(C(C2(SC)CN(C(C3CCCC(C)C3)=O)C2)=O)CCn2nccc21 12828,C(=O)(C(F)CCC(C)(C)C)NCc1c(C(=O)Nc2c(C)csc2)nco1 12829,CC1ON=C(C(=O)NC(C2CCCN2C(c2csnn2)=O)(C)C)C1C 12830,CCCCCC(O)CC(=O)NC1CCCC1NC(C1(C(F)F)CC1)=O 12831,C1(C)(C(=O)NC(CC)C(=O)NC)CCN(C(c2c[nH]nc2OC)=O)CC1 12832,CCC(CC)CCCC(=O)N1CC(C)CCC1CNC(=O)CCOC(C)C 12833,c1(C(N2CCCC(NC(C(CC3CC3)OC)=O)C2)=O)ccc(C)c2c1CCC2 12834,N1(C(C(C)Oc2ccccn2)=O)CCN(C(=O)CC2(CSC)CC2)C(C2CC2)C1 12835,c1(OC)ccc(C(CNC(=O)Cc2nnc(C)n2C)NC(=O)C(O)C(C)C)cc1 12836,C1(O)(COC)CN(C(C2CCC2CNC(=O)C(C)c2ccco2)=O)C1 12837,CCC(C(=O)Nc1cc(C(=O)Nc2nn[nH]n2)cs1)n1cccn1 12838,Cn1nc(CC(N2CCC3CC(C2)CN(C(=O)C(O)CF)C3)=O)c2ccccc12 12839,C12CCCCN1CC2.C1(N(C(C=CC=CC)=O)C)CCCN1CCCC 12840,C(C1CCCCCC1)=CC(=O)NCC1(F)CN(C(CCC(=C)Cl)=O)C1 12841,C=CC1CN(C(c2cnc(C)c(CC(C)C)c2)=O)CC1NC(=O)C#CC1CC1 12842,CC(C)CC(O)C(C)C(=O)N1CCCC1CC(=O)Nc1cn(C)nc1O 12843,CC1CCCC=C1C(=O)NCC1CCC1NC(c1ccn(C(C)(C)C)c1)=O 12844,c1(C(N2CCC(C(C)(C)NC(Cc3c(C)con3)=O)C2)=O)c(C)coc1C 12845,C(=O)(C1=NOC(CNC(=O)CCOC(F)F)C1)NCC(n1cccn1)C 12846,N1(C(C)C(=O)NCCC2CC(NC(C3(C4CC4)CC3)=O)C2)CCCCC1=O 12847,c1(C(C)C)ccoc1C(=O)NC12CC(NC(=O)CC3CC3C)(C1)C2 12848,c1(CNC(C(C)O)=O)ccc(CNC(C2CCCN2Cc2cccnc2)=O)cc1 12849,c1(CC)nc(Cl)c(F)c(=NCCCCNC(=O)C(Cc2ccccc2C)CC)[nH]1 12850,c1(C(N2C(CNC(C(CSC)O)=O)CC(C)(C)C2)=O)ccc2oc(=N)[nH]c2c1 12851,N1(C(CCCCN(C(=O)C(O)c2ccco2)C)=O)CCC2(CCC(N(C)C)C2)C1 12852,C=CCCC(CC(C)C)C(=O)N(CC(C)NC(C1CCOC(C)C1)=O)C 12853,c1(C(=O)NC(CCCC=C)c2ccccc2)[nH]cc2c1CCCC2 12854,N1(C(C=C2CCN(C(c3c(Cl)cccc3I)=O)CC2)=O)Cc2ccc(O)cc2C1 12855,c1(C(=O)NC(C)CNC(c2sc3sccc3c2Cl)=O)cc(O)c2ccoc2c1 12856,C(=O)(C#CC1(C)CC1)NC(CNC(C(C)NC(=O)C(C)(C)C)=O)C1CC1 12857,c1(C(=O)NC2CC3CCC2(NC(c2ccon2)=O)C3)cc2ccccn2c1 12858,c1(C(N(CC(C)O)CCNC(c2c(OC)csc2)=O)=O)c(NC(C)=O)c[nH]c1C 12859,C1(S(C)(=O)=O)(NC(Cc2c(C(C)C)con2)=O)CC1C(F)(F)F 12860,CC(C)(C)CCCC(=O)C(=O)N1CCC2(CC1)CC(NC(C1CC13CCC3)=O)C2 12861,C1(C(N(CC)CC)=O)CC2CC2N1C(=O)CCOC1CC1 12862,N1(C2C3CCCC32)CCC(N=c2[nH]c(N3CCSC(C4CC4)C3)nc3c2COC3)C1 12863,c1(COC)nn[nH]c1C(=O)NC(C)C(C)NC(=O)CN(C)CCO 12864,c1(SC)cccnc1C(=O)NCC1CC2CC2N1C(=O)CCc1cscn1 12865,C1(NC(C#CC(C)(C)C)=O)CC(N=c2ccnc(Cl)[nH]2)C1(C)C 12866,c1(CNC(C2(CC)COC2)=O)nnc2n1CCN(C(C1(S(C)(=O)=O)CCC1)=O)C2 12867,N1(C(CCCN(C(C)C)C)=O)CCN(C(C2COC(=O)N2C)=O)C(C)C1 12868,N1(C(C(C)OCC(C)C)=O)CCC(C2CCN(C(C3CCCCN3C)=O)CC2)C1 12869,C1(CCC(=O)N(C(C#C)C)C)CCCN(C(=O)CCC(C)OC(C)=O)C1 12870,N1(C(c2n(CC)nnc2)=O)C2CCC1CC(N(C(=O)CN(C1CCSC1)C)C)C2 12871,c1(C(CNC(C2CCCO2)=O)NC(c2cc(C(N)=O)n[nH]2)=O)ccc(F)cc1 12872,c1(C(N2CC(C)C(CNC(=O)C(c3ccnn3C)O)C2)=O)cncc2nc[nH]c12 12873,c1(OCC(=O)NCC(CC)N(C(=O)C(F)C2CCC2)C)ccc(Cl)cc1C 12874,N1(C(CNS(CC)(=O)=O)=O)CCCC2(CCCCC2NC(C2(O)CCOC2)=O)C1 12875,C1(C(=O)NCCN(C(c2cnc(Cl)s2)=O)CC2CC2)CCCC2(CCC2)C1 12876,C1(NC(c2cc(OC)n(C)n2)=O)CCCN(C(=O)CCN2CCCC2)CC1F 12877,CC1C(=O)CCC1CC(=O)N(CC(O)CN(C(=O)CN1CCOCC1)C)C 12878,C(C(C(C)(C)C)NC(=O)CCCn1cccn1)NC(C(C)NC(N)=O)=O 12879,N1(C(C2(C)COCCO2)=O)C2CCC1CN(C(=O)C(c1ccc(F)cc1)CO)C2 12880,Cc1cc2c(cc1C)OC(C(=O)NC1CC(CNC(C3COC(=O)N3C)=O)C1)C2 12881,C1(C(=O)NCC2C3CN(C(COCCCC#C)=O)CC32)CCC(S(N)(=O)=O)CC1 12882,C1(NC(C(C)(CSC)NC(C(C)N(CC)CC)=O)=O)CCOC12CCCC2 12883,N1(C(C(CCCC)NC(=O)CCn2ccnn2)=O)CCC12CCCCC2 12884,C(=O)(C(CC)CCN(CCCCC(C)(C)C)c1cc(N2CCCC2)ncn1)OC 12885,N1(C(c2n(C)cnn2)C(=O)NCC(F)F)CCOC(c2cn(C)cn2)C1 12886,Cc1cc(C(N2CC(NC(=O)CCS(C)(=O)=O)C(C)C2)=O)cc(N)c1 12887,Cc1cc2cc(C(=O)NC(C)CN(C)C(C3OC4CCC3CC4)=O)oc2cc1C 12888,c1(COC)cccc(C#N)c1OC(C1CCC(OC(F)F)CO1)=O 12889,C1(C(N2CCCC(C(=O)Nc3cnn(CCO)c3)C2)=O)CCCC2(CC2)C1 12890,N1(C(Cc2c(C)nsc2)=O)CCC(F)C(NC(c2ccnc(C(F)(F)F)n2)=O)C1 12891,C#CC1CN(C(C2COCCN2C)=O)CCN1C(C1CCCCC1CC)=O 12892,N1(C(=O)C=Cc2cnc[nH]2)CC2CN(C(c3cccc4cncn34)=O)CC2C1 12893,C1(NC(CCC(=O)OC)=O)CC(O)CN(C(=O)C(F)(F)c2cnnn2C)C1 12894,N1(C(c2ccn(CC(F)(F)F)n2)C(=O)NCCSC)CC(CO)C(CO)C1 12895,c1(C(=O)NCC(C2CCCN(C(c3ccc(Cl)cn3)=O)C2)(C)O)cccc(Cl)c1 12896,C1(C(C(=O)NCCCCCC)CC)CCN(c2n[nH]c(=N)s2)CC1 12897,Cn1nc(C(=O)NOCC(N2CC3CC2(CO)C3)=O)cc1O 12898,N1(C(c2cncc(C#C)c2)=O)CCC2CCCC12CNC(=O)C(C)(CO)OC 12899,CCCC(C)(CC)C(=O)NCC1CC(C(=O)Nc2cnn(C(F)F)c2)=NO1 12900,C1(CC)CN(C(=O)CCc2ccncn2)CC1C(=O)NCC(c1cccnc1)O 12901,CCC(CC(=O)NCCCC(=O)N1CC(C)(CCO)C1)C1CCC1 12902,c1(C(N(C2CN(C(C(C(C)C)N3CCC3)=O)C2)C)=O)cc2c([nH]1)CCC2 12903,C1(CCCCCC)CCCC1(c1nnnn1C1CCC1)NC.C1(C)CC1C(F)(F)F 12904,CC12CN(C(=O)C(F)CC3CCCCC3)CC1(C)CN(C(c1cnc[nH]1)=O)C2 12905,c1(C(=O)NC2CCN(C(=O)CC3CC3)CC2)ccc(CN(C(=O)OC)C)cc1 12906,CC(CCCCNC(=O)C(C)Cc1cnc[nH]1)NC(c1cc(Cl)cnn1)=O 12907,c1(NC(CCC)CC)ncccc1S(=O)(=O)N(C)Cc1scnc1C 12908,C(CC(C(C)(C)C)NC(c1ccc(F)c(F)c1)=O)N(C(C1(C)CC(C)C1)=O)C 12909,O=C(C1=CC2CCCCCCC12)N1CCC(CNC(C23CCC(CC2)CO3)=O)C1 12910,C1(NC(CCCSC)=O)CCC2(CC1)CCN(C(=O)C1=NOC3(CCOC3)C1)C2 12911,C(=O)(C(O)CC(N)=O)N1C(C(C)C)(C(N2CC(O)CC2C(N)=O)=O)CCC1 12912,C#Cc1ccc(CC(N2CCCOC(CCNC(=O)OC(C)(C)C)C2)=O)cc1 12913,CC(C)CC(O)C(=O)NCc1ccc(CNC(C2(CF)CC2(F)F)=O)cc1 12914,C(=O)(C(CO)C(C)(C)C)N1CC(C(=O)NC2CCC(C(N)=O)O2)(COC)C1 12915,CC(C)CC(CNC(c1cccc(=O)o1)=O)C(=O)N(C)CC1CC1 12916,C1(CNC(Cc2c(OC)cccc2)=O)CCC(C)N(C(c2cc(C)ncn2)=O)C1 12917,C(C(=O)NCCc1scnc1C)(C(C)(C)C)NC(c1c(CC)ocn1)=O 12918,CC1=C(C(=O)NC2CN(C(c3nn(C)c(Cl)c3Cl)=O)CC2F)SCCO1 12919,C1(CC(=O)N(C)CC2CCN(C(=O)Cc3ncn(C)n3)C2)CCC(=O)C1C 12920,N1(C(CC=CC=C)=O)CCN(C(=O)C(O)C2CCCC2)CC1CC1CC1 12921,CCC(O)C(F)(F)C(=O)N1CCOCC(CNC(=O)C(C)(C)O)C1 12922,N1(C(C=C(C)c2cccs2)=O)CCC2CCC12CNC(c1ccc(O)c(F)c1)=O 12923,c1(C(=O)NCCOCCN(C(CC(C)CF)=O)C)cc2c(s1)CN(C)CC2 12924,C1(NC(CC2N(C(C=C(C)c3ccco3)=O)C3C2CCC3)=O)CCc2n[nH]cc2C1 12925,c1(NC(=O)NCC(O)Cc2ccncc2)cc(Cl)ns1 12926,C1(Br)(C(=O)NCC(CN(C(=O)C2=CC(C)(C)C2)CC)(C)C)C(C)(C)C1(C)C 12927,C(O)(C1CCc2ccccc21)NC(C(CC)NC(c1ccccc1)=O)=O 12928,C1(NC(c2cc(CCC)c(C)s2)=O)CCN(C(C2COCC(C)(C)O2)=O)CC1O 12929,Cn1nc2c(c1C(N1CC(NC(=O)CSC(C)(C)C)C3(CC3)C1)=O)COCC2 12930,C(=O)(CC(C)(C)C(F)F)NC1(CO)CC1.N1(C(C)=O)CCC(O)C1 12931,c1(C(=O)NCCCN(C(=O)C=C2CC2)CC)cc2ccc(F)cc2o1 12932,C1(CNC(C(=Cc2cccs2)C)=O)C2CCC(C2)N1C(=O)CNS(N)(=O)=O 12933,C12(NC(c3coc(Br)n3)=O)CCC(n3cc(-c4ccns4)nn3)(CC1)C2 12934,N1(C(C(C)NC(COC)=O)=O)CCC(CO)(NC(c2cnns2)=O)CC1 12935,n1(CC=C)cc(C(=O)N(CCCNC(c2ocnc2C(C)C)=O)C2CC2)cn1 12936,Cc1[nH]nc(C(N2CCC2(C)CC(N2CC3CCC2C3)=O)=O)c1O 12937,C#CCC(C(=O)NCC(O)CN(C)C)NC(=O)COC(CC)CC 12938,c1(C(=O)NCC(C)(CO)NC(=O)CSC2CC2)cccc(OC(F)F)c1 12939,N1(C(C2(NC(c3ccc(C)n3C)=O)CCCC2)=O)CCOC(C)(C)CC1 12940,Cc1cc(=NCc2cnoc2)[nH]cc1S(=O)(=O)NC(C)CN1CCCC1 12941,c1(C(N2CCN(C(c3ccccc3)=O)C(CC3CC3)C2)=O)cc([N+](=O)[O-])n[nH]1 12942,c1(C(N2C(CNC(CCC(C)C)=O)CCC2)=O)ccc2ocnc2c1 12943,C(C)(CCC(=O)NC(C)C(C)NC(c1cc(=O)n(-c2ccc(C)cc2)[nH]1)=O)OC 12944,c1(C(N2CCN(C(c3c(CC)onc3)=O)C(CC#N)C2)=O)ccc2ccoc2c1 12945,C1(NC(c2c[nH]cc2C(F)(F)F)=O)C(CO)C2CCCCC12 12946,C1(C(=O)NC2CCN(CCC3CC3)CC2)CC2CCCC2C1 12947,c1(C(=O)NC(C=CC(=O)NC2(C)CC(=C)C2)C)cc(C)ccc1O 12948,C1(C(=O)NC(CC(=O)NC)C)CNC(=O)CN1C(C1CC2(CCO1)CC2)=O 12949,Cc1cc(NCCCNC(C2(O)CCCC(C)(C)C2)=O)n2ncc(C)c2n1 12950,C#Cc1c[nH]nc1C(=O)NCCNC(C1CCC(NC(N)=O)CC1)=O 12951,C(CCC#N)(C(N)=O)NC(C(=O)NC1CC(CC(C)C)OCC1)=O 12952,C1(C(N(C)CC2CCCN(C(c3cc(CO)on3)=O)C2)=O)CC2(CCCC2)CO1 12953,C1(CC)CC(CC(=O)NC2(C)CN(C(c3ccncc3C(F)(F)F)=O)C2)CCO1 12954,c1(C(N2CCC2)C)cn(CC2CCCN2C(c2cc(-c3ccns3)on2)=O)nn1 12955,N1(C(C(CCCC)C)=O)CCCC2CN(C(=O)COC(F)F)CC12 12956,c1(NC2C(CC)CN(C(=O)CCC(=O)N(C)C)CC2)ncnc2sc(C)nc12 12957,C=CC1(C(=O)NC(CO)C2CCC2)CCN(C(=O)C(c2ccc(F)cc2)(F)F)C1 12958,c1(C(N2CCC(C)(NC(C(C)=C3CCC3)=O)C2)=O)cn(C)c2c(cnn2C)c1=O 12959,CCCCC(F)(F)C(=O)NC(CN(C(=O)C1=NOC(C)C1C)C)CC 12960,c1(C(=O)NC2CC(C)(C)N(C(C3COC(=O)O3)=O)C2)cccc([N+](=O)[O-])c1 12961,c1(NC(C(C2CCN(C(c3sccc3Cl)=O)C2)C)=O)ccc2c(c1)OCC2 12962,N1(C(C(CCCNC(C2CCC3CC23)=O)O)=O)CC=CC12CCCCC2 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13033,C1(CCNC(CN(C)CC)=O)COCCN1C(=O)CCCc1csc(C)n1 13034,c1(NCCn2c(C)cc(C)n2)ncccc1S(=O)(=O)N1CCn2ncc(Cl)c2C1 13035,c1(C(C(=O)NC(CC)C(=O)c2ccccc2)=O)cn(C)c2ccc(F)cc12 13036,N1(C(C(C)N(C(=O)CC2CCCN2C)C)=O)CC2(CCNC(=O)O2)C1 13037,c1(C(N(C(CO)C2CC2)C)=O)cc(O)nc2c1CN(C(c1cn(C)nn1)=O)CC2 13038,C(CNC(=O)CCOC1CCC1)(C(=O)NCCCn1cccn1)OC 13039,C#Cc1ccc(C(N2CC3CC(C(=O)NC(COC(C)=O)CO)C(C3)C2)=O)c(C)c1 13040,c1(NC(C=CCNC(c2c(CC)nn(C)c2)=O)=O)ccc2occc2c1 13041,c1(C(CNC(CSCCC=C)=O)NC(=O)CC2CNC(=O)C2)ccccc1OC 13042,C(=O)(C(C)(C)CC(F)F)NC1C(OC)CN(C(=O)CN2CCCCC2=O)C1 13043,C(=O)(C1COc2ccc(F)cc21)NCCCC1(N(C)C(N)=O)CC1.C1(=O)CN1 13044,CCCCC(CC)C(=O)NC12COC(C1)C(NC(C1CC1OC(C)(C)C)=O)C2 13045,c1(C(=O)NC2(CNC(C3(C)CCC(=O)NC3)=O)CC2)cccc2c(C#N)c[nH]c12 13046,c1(N(CC#C)C)nnc(Cc2ccncc2)n1CCCn1ccc(Br)n1 13047,CCC(C)CCC(O)CC(=O)N1CC(NC(=O)CS(=O)(=O)C2CCCC2)C(C)C1 13048,C=C(C)C(C)(C)C(=O)NCC(C)N(C)C(C1CCN(C(c2cccs2)=O)CC1)=O 13049,C1(NC(CCC=C)=O)CC12CCN(C(=O)Cc1cnccc1C(F)(F)F)CC2 13050,N1(C(=O)CSc2cccs2)CCCC2CN(c3nc4ccccc4o3)CCC12 13051,c1(C(=O)NC2CN(C(C(CCOC)OC)=O)CC2O)cc2cc(C)ccc2[nH]1 13052,C(C)(CCC(=O)N1CC(C(F)Cn2cc(CC3CCCC3)nn2)C1)OCC 13053,c1(C(N2C(CO)CC(NC(C(CC)SC)=O)C2)=O)n[nH]c2cc(C)ccc12 13054,N1(C(c2cnc(C)[nH]2)=O)CCC(C2CCCN(C(c3nc(C)c(C)s3)=O)C2)C1 13055,N1(C(c2c(C(=O)O)cc(OC)nc2)=O)CCN(Cc2nc(C)cs2)CC12CC2 13056,C(=O)(C(C)(C)CC(F)F)N(C1CCC(NC(c2ccc(F)cc2F)=O)CC1)C 13057,C1(O)(CN(C(=O)COC2CCOC2=O)CC)CCN(C(=O)C(F)(F)CC)CC1 13058,c1(C(=O)NCC2CC(NC(C3CC3F)=O)C2)cccc(Br)c1 13059,N1(C(COCCOCCOC)=O)CCC(O)(CCn2cc(CC(O)CO)nn2)C1 13060,Cc1cc(=NCC2(C)CSC2)[nH]c(N2CC(=O)N(C)C(C)C2)n1 13061,C=C(F)C1(CC(=O)NC(C)(C)C(C)NC(C2CC2(C(C)C)CC)=O)CCC1 13062,C1(N(C(CC)=O)C)CCCCN(C(C23CC(c4ccc(OC)cc4)(C2)C3)=O)C1 13063,c1(CN2CCC(C(C(=O)NC(c3cccs3)C)C)CC2)ccc2c(c1)CCO2 13064,c1(OC)ccc(C(N2CC3CC(NC(C4CCC(=O)CC4C)=O)C3C2)=O)c(C)c1 13065,c1(SC)ccc(OCc2cccn2C(C)C)cc1.N12CC(C(O)C1)NC(C)C2=O 13066,c1(C(C(=O)NCCCN(C2CCCC2)C(=O)CC2CC(F)C2)F)ccccc1 13067,C1(C(C(N2CCC(OC(C)C)C2)=O)NC(=O)OC(C)(C)C)CC(C2CC2)C1 13068,N1(C(C23CC(NC(=O)C=CC(F)F)(C2)C3)=O)CCC2(CCC2)C1 13069,C1(O)(CNC(C(C)(O)C2CCC2)=O)CCCN(C(=O)CCCN2CCCC2)C1 13070,C12(OC)CCC(C(N3CCC(CCNC(=O)CC4C=CCC4)C3)=O)(CC1)C(=O)C2 13071,C1(NC(c2n(C)ccn2)=O)CCCC(NC(c2cn(CCCF)nn2)=O)C1 13072,N1(C(C(C)N(C)C)=O)CCN(C(=O)C(=O)NC2CN(C3CCC3)C2)CC1 13073,C1(C(=O)NC2CCCN(c3ccc(C)cc3)C2=O)CCc2nn(C)c(C)c2C1 13074,C=CC(CC)CC(=O)N1CCC(N(C(=O)C(c2ccccc2F)(C)C)CCC)C1 13075,c1(OC)ccc(CNC(C2OCCC2NC(=O)CCc2ncnn2C)=O)cc1 13076,c1(OC(C)C)ccccc1ON(c1nnc(Cc2nccs2)n1CC=O)C.C(C)=C 13077,C1(C(=O)NC23CCC(CNC(C(CC=CCC)C)=O)(C2)C3)CN2CCN1CC2 13078,C1(C(N(CCCSC)C)=O)C(C)CCN1C(c1cc(C2CC2)n[nH]1)=O 13079,c1(C(=O)NCC(CNC(CC=C=C)=O)(C)O)cc(C(N)=O)cn1C 13080,N1(C(C=C(C)Cl)=O)CCC(C)N(C(C2C(Cl)(Cl)C23CC3)=O)CC1 13081,c1(OC)ccc2c(C(=O)NCC3CC3NC(=O)CCn3ccnc3)cnn2c1 13082,n1(CC)c(=N)[nH]c2cc(C(N3CCC(CNC(C4CCN(C)C4)=O)C3)=O)ccc12 13083,c1(CC)cc(C(=O)NCC(CC(C)C)NC(=O)CNC(=O)NC(C)C)ccc1O 13084,C(=O)(C(CC(C)C)NC(c1cccc(CNC(=O)CCCF)n1)=O)NC 13085,C(=O)(C1CCc2cccc(Cl)c21)N1C(CNC(c2c(C)cc(F)cc2)=O)CC1 13086,c1(NCC2CCCN(C(Cc3cnc(C)s3)=O)C2)ncnc2[nH]c(Cl)cc12 13087,C(=O)(C(F)CC1CN(C(c2cc(C(C)C)on2)=O)C1)N(C(C(=O)OC)C)C1CC1 13088,c1(C(N2C(CCC#C)CCC2)=O)ccc(OC)n2nccc12 13089,C1(C#N)(C(N2CC3C(CNC(CCc4onc(C)n4)=O)C3C2)=O)CC12CCCC2 13090,c1(OC)ccc(C(=O)NC2CCCN(C(C3(C4CC4)CC3)=O)CC2)c2[nH]ncc12 13091,N1(C(C)(C)C)CCCCC1C(C)(C)CNC(=O)NCCS(C)(=O)=O.C1(N)CCOC1 13092,c1(C(N2C3CC(CC(NC(C(C)C(F)F)=O)C3)C2)=O)cc(F)cc2ccncc12 13093,c1(C(N2CCCC(CNC(c3c(C)ncnc3)=O)C2)=O)ccc(F)c(C(F)F)n1 13094,C1(CNC(C(C(C)O)C)=O)CC2(CCN(C(=O)COC3COC3)CC2)CO1 13095,c1(CC(N2CCC3(NC(CN(C(C)=O)C)=O)C(C2)C3)=O)c[nH]c2ccc(Cl)cc12 13096,O=C(C1=CCC2(COC2)OC1)NC(Cc1ccccc1Br)C(=O)O 13097,C1(C(=O)NCC2(C)CC(NC(Cc3c(C)n(C)nc3)=O)C2)CCCCC(=O)N1 13098,C(=O)(CC1=NN(C)C(=O)C1)N(CCCNC(c1cccc2ncsc12)=O)C(C)C 13099,C1(NC(C(C)OCCC#C)=O)(CNC(=O)C(C)Cc2cnn(C)c2)CCCC1 13100,c1(CC(=O)NCC2CC2NC(c2ccc3cccnn23)=O)ccc2ncccc2c1 13101,O(NC(=O)CC(C)(C)C1CC1)C(COCC)COC.C1(N)CC=CCO1 13102,N1(c2cc(NCCc3ccc(C(N(C)C)=O)cc3)ncn2)CCNC(=O)CC1 13103,c1(C(=O)NCC2C(NC(C(c3cnn(C)c3)C)=O)CC2)ccc(C2CC2)nc1 13104,C(CC(=O)NCC(CO)NC(C1CCCN1CC)=O)(OCC)OCC(F)(F)F 13105,C1(C(C(=O)NCC=C)N(C2CC(F)(F)C2)C)CCC(CCC(C)C)CC1 13106,C1(OC)(NC(=O)C(N)CCC2CCC2)CCC(C)(C)C1 13107,CC1CC=C(C(=O)NC2CCC(CNC(c3cnc4n3CCOC4)=O)CC2)CC1 13108,C1(C(N(C2(CNC(C3CC(CC(C)(C)C)C3)=O)CC2)C)=O)CCOC2(CCCC2)C1 13109,CC(C)CC(C(=O)NC1(c2nnnn2-c2ccccc2)CCN(CF)C1)C1CC1 13110,N1(CC)CCN(C(=O)CC2(CNC(c3cnc(O)c(F)c3)=O)CC2)CC1C 13111,c1(C(=O)NCc2ccc(-n3c(C)cc(C)n3)nc2)cc2cccnc2cn1 13112,C1(CCNC(C(C)NS(CCC)(=O)=O)=O)CCCN(C(=O)C(F)(F)COC)C1 13113,n1(CC(=O)N(C2CC3N(C(CCC#C)=O)C(CC3)C2)C)nc2n(c1=O)CCOC2 13114,C#CCC(C(=O)NCCOCCCF)NC(=O)C(C1CCC1)OC 13115,CC1(C)CCC(CC(=O)NC(C)(CO)C(=O)N2CC(N3CCCC3=O)C2)O1 13116,C1(NC(C(CC)F)=O)CCCC2CN(c3ncnc4c3ncn4CC)CC12 13117,c1(CC)ccc2c(c1)OCC2C(=O)NCCCCNC(=O)CC(C)n1cccn1 13118,N(C(=NCCSCc1ccc(F)cc1)NCC(F)F)C1CC(C)SC1 13119,c1(C(N(C2CCCN(C(C(C)(C)CO)=O)C2)CCO)=O)coc2c1COC2 13120,Cn1cc(C=CC(=O)NCc2ccccc2CNC(=O)Cn2nccn2)nn1 13121,N1(C(c2ccc(NC(C)=O)o2)=O)CCC(NC(=O)C(C)S(C)(=O)=O)C2(CCC2)C1 13122,[N-]=[N+]=NCCCCCC(=O)N1CC(C(=O)NCCC2CCC3CC23)CC12CCC2 13123,C(=O)(C1=CCC(C)CC1)NC1CCN(C(CCn2c(C)nc(C)n2)=O)C1C1CC1 13124,C1(n2ccnc2)(CNC(COCC(=C)C)=O)CCN(C(=O)Cc2cc[nH]n2)CC1 13125,CC(=O)CCCC(=O)NC1(C2CCCCN2C(c2ccc(Cl)cc2F)=O)CC1 13126,c1(C(=O)NC2CCCC(N(C(=O)CC3(C#N)CC3)C)C2)ccc2nn[nH]c2n1 13127,C1(NC(c2c(Cl)cn(CC)n2)=O)C(C)CCN(C(c2cnc3sccn23)=O)C1C 13128,c1(C(C(=O)NCC)N(CCF)CCOC)ccc(OCF)cc1 13129,C1(CC)CN(C(=O)C(O)C2CC2)CCC1NC(c1cncn1C)=O 13130,C1(C(=O)NC2(CN(C(=O)CCOCC3CCCO3)C)CC2)(CC2CC2)CCCC1 13131,N1(CC(=O)NC2CC(C)(NC(=O)CC3CC4CC4C3)C2)CCC(=O)NC1=O 13132,N1(C(C(C)Cc2ccco2)=O)CCC(NC(c2ncn(C)n2)=O)C(C(N)=O)C1 13133,N1(C(C(C(C)C)(C)O)=O)CC(NC(c2ccc(F)s2)=O)CC(C)(C)C1 13134,N1(CCNC(=O)COC(c2cnn(C3CC3(F)F)c2)=O)CCc2ccccc21 13135,c1(-c2ccc(C#C)cc2)ccc2c(c1)CN(C(c1ccn(CCOC)n1)=O)CC2 13136,C#CC(CNC(=O)CC1(CNC(C2CCO2)=O)CC1)CC1CC1 13137,N1(C(C2C(CC)C2)=O)CC2(C1)CC1(C)CC(OC)C(C(=O)OC)(C1)C2 13138,NS(=O)(=O)c1ccc(NNC(=O)C(=O)NC2CC2)s1 13139,N1(C(CCCCC#C)=O)CC2(C1)CN(C(C1CC13CCCCC3)=O)CC2CO 13140,C1(N(C(CN(C(=O)C(C)N=[N+]=[N-])CC)=O)C)CCOC(C)(C)C1 13141,CN1CC=C(CC(=O)NCC2CCCC3CN(C(=O)C(C)(C)C(F)F)CC23)CC1 13142,c1(C(N(C(C)CNC(c2ccn(C(F)F)n2)=O)C)=O)ccc(CO)cc1F 13143,N1(C(C2CC(C)(C)OC2)=O)CCC(NC(=O)CNC(N2CCCC2)=O)C1(C)C 13144,Cc1nccc(C(=O)NC2CN(C(C3CC3CC(C)(C)C)=O)CC2C(F)F)c1N 13145,N12C=CC(=NC(=O)C(C)N3CC1C3)N2.c1(C(=O)OC)ccc(F)c(C(=O)OC)c1 13146,N1(C(c2ccn(CC)n2)=O)CC(NC(C2CN3CCC2(C)CC3)=O)CC12CCC2 13147,S(=O)(=O)(c1ccccc1CS(=O)Cc1ccccc1)N1CCOCC(C(C)C)C1 13148,S(=O)(=O)(CC(=O)NCC1CCCC1NC(=O)CCc1ccncc1)NC 13149,c1(OC)ccc(C(=O)NCCCC(C)NC(=O)CN(C)C(=O)C2CC2)c(F)n1 13150,C(=O)(C(CC(N)=O)NC(C1CC(C(C)C)=NO1)=O)NCc1c(C)nn(C)c1 13151,Nc1ccc(CN2CCCC2CNC(=O)CC(O)c2ccccc2)cc1[N+](=O)[O-] 13152,Cn1nc2c(c1C(N1CCC(NC(C3CC3(Cl)Cl)=O)C(F)C1)=O)CCCC2 13153,C1(C(=O)NC23C(CN(C(C4N(C(C)=O)CSC4)=O)C2)C3)CC2CSCC(C1)C2 13154,C1(CC#C)(C(=O)NC2CCC(NC(=O)Cc3cnn(C)c3)C2)CCCCO1 13155,N1(C(C2C(C(N)=O)CCCC2)=O)CC2CC(C1)N(c1cc(F)ncn1)C2 13156,CON(CCC(=O)NOCC(F)F)C(=O)c1ncc[nH]1 13157,C1(CNC(CC2(COC)CC2)=O)CN(C(c2cc[nH]c(=N)c2)=O)C2CC12 13158,c1(OC)cccc(CC(N2CCCC2CNC(C2CN(C)C2)=O)=O)n1 13159,C(=O)(C1CCc2cc(Cl)ccc21)NCCCc1cn(C2(C(=O)OC)CC2)nn1 13160,c1(C(C)NC2(c3nnnn3CCCF)CNC(=O)C2)cnc2n1CCOC2 13161,N(C1c2ccccc2CC1NC(=O)C=C1CCC1)C(C1N(N=O)CCCC1)=O 13162,CC1(C)CC(C(=O)NC2CC(F)(F)C23CCC3)CCN1C(c1ccc[n+]([O-])c1)=O 13163,c1(SCCC)cccc(C(N2CC(COC)C3CC23)=O)c1 13164,n1(C(CC)CC)cc(CN2CCC(C)C2)c(C)n1 13165,Cc1nccc(C(=O)NCc2cncc(C(=O)NC3CC4(CC4)C3)c2)c1N 13166,c1(CNC(c2c(OC)ccs2)=O)ccc(CNC(C2CCC(=O)N2C)=O)c(F)c1 13167,N1(C(c2ccc(OC)nc2)=O)CCN(c2cccc(Cl)n2)C(C)C1 13168,C1(CNC(CC2C(C)(C)OCC2)=O)C2CCC1CN(C(=O)CCCCC(N)=O)C2 13169,N1(C(C(C)C=Cc2ccccc2)=O)CCCC(C)(NC(=O)C#CC(=O)N(C)C)C1 13170,C(CC(C(=O)NCC(C)(C)C(C)O)NC(=O)CC1CCCC(=O)C1)OCC 13171,C1(C(=O)NC(CNC(C(CCSC)O)=O)(C)C)Cc2ccc(Br)cc2C1 13172,C1(COC)CN(C(c2ccc(F)s2)=O)CCN1C(C1CC(=O)N(CC(C)C)C1)=O 13173,C(C(C(=O)N1CCCC1CCNC(=O)C(C)Oc1ccccc1)OC)OC 13174,C1(NC(=O)Nc2ccc(CCSC)cc2)CCC(F)(F)CC1O 13175,N1(C(COCC)=O)CCC2(COC(CNC(C34CC5CC(CC(C5)C3)C4)=O)C2)C1 13176,c1(C(N2CC(C3(NC(CCC4CCC(=O)C4)=O)CC3)C2)=O)cc2cccnn2c1 13177,c1(C(=O)NCC(C)(C2CC2)NC(C2CCC2(F)F)=O)cc2c(nn1)CCOC2 13178,C1(C(N2CCN(C(C3CCC(C)(C)CC3)=O)C3C2C3)=O)CCCN(S(N)(=O)=O)C1 13179,C(CN=c1[nH]nc(C#N)s1)(C1CC1)NC(C1(C)CCNC1=O)=O 13180,CCC(C)(CO)C(=O)N1CC(CNC(c2ccnnc2)=O)C(F)(F)C1 13181,CC1CC(C)(C(=O)NCC2CN(C(=O)CCCOc3ccccc3F)C2)CCO1 13182,c1(CNC(CN(C2CC(C#N)C2)C(C2N(CC)CCC2)=O)=O)ncccc1Cl 13183,CC(CNC(=O)CNC(=O)CN(C)C)C(F)C(=O)NCC1CC1(F)F 13184,C(=O)(C(C)CS(C)(=O)=O)NC1CC(C)(NC(CC2N(C(C)=O)CCC2)=O)C1 13185,c1(OC(CC)C)cccc(NC(c2nccs2)=O)c1 13186,c1(OCC)ncccc1C(=O)NCC1(CNC(c2cn(C)cn2)=O)CC1(F)F 13187,CC1CN(C(c2ccc(C(F)(F)F)cc2Br)=O)CCN1C(c1ccnnc1)=O 13188,c1(C(N(CCC(=O)NC(C(C)SC)C)C2CC2)=O)ccnc(C)n1 13189,N1(C(CN(C)C(N)=O)=O)CC2(C1)C(NC(C1CCC3CCC1O3)=O)CCS2(=O)=O 13190,Cc1cc(C(N2CCC2CNC(c2cc(-c3ccco3)no2)=O)=O)cn1C 13191,c1(C(=O)NCC(c2ccc(OC)cc2)NC(CC=CCC)=O)cc(C)c(F)cn1 13192,c1(C(=O)NC2(CNC(C(CC(C)C)F)=O)CCC2)cc(F)c(C(F)(F)F)cc1F 13193,c1(CN2C(CCC(=O)NCCCCCC)CCC2)ccc([N+](=O)[O-])cc1OC 13194,C1(CC)CN(C(=O)CN2CCNC(=O)C2)CCN1C(=O)CC1CCCCC1O 13195,c1(C(N(C2CCN(C(C3CCCS3)=O)CC2)CC)=O)n[nH]c2c(C)cccc12 13196,c1(C(=O)NCC(C(C(C)C)C)NC(c2nncs2)=O)cc(F)c(F)c(F)c1F 13197,c1(CC(=O)NC2C=CC(CNC(C(C)(F)F)=O)C2)cccc2cnccc12 13198,C(=O)(C1=NOC2(CCC2)C1)NC(CNCC1(C)CCC(=O)N1)CO 13199,C1(C(N2CC(OC(=O)NC)C2)=O)C2CC(O)C1N(C(c1ccnn1C)=O)C2 13200,C(=O)(C(CC)(CC)CC)N1CCC(F)(C(N2CC(C#C)(N(C)C)C2)=O)CC1 13201,C=CCC(C)(C)CC(=O)NC1CC(NC(c2ncccc2Cl)=O)C1 13202,c1(C(=O)NCC(C)NC(=O)CC2CC(CN(C)C)C2)c[nH]nc1-n1cnnn1 13203,C1(C(N2CC(n3cc(CNC(=O)CC4CCC4)nn3)C2)=O)CCCCC1O 13204,C1(NC(C2CC(F)(F)C2)=O)C=CCN(C(=O)CC(c2ccon2)C2CC2)C1 13205,CC1(C)CCC(O)(CNC(=O)CCCC2CN(C(=O)CN3CCOCC3)C2)C1 13206,C(=O)(CCCCCCn1cc(CN(CCO)CCO)nn1)NC(c1ccncc1)C 13207,c1(CN2CCC(N3CCN(c4cc(CC)ncn4)CC3)C2)cccn2ccnc12 13208,CC1CN(C(c2ncn3c2CCCC3)=O)CC(C)C1NC(c1ccc[nH]1)=O 13209,CS(=O)(=O)CC(=O)NCC1(C(=O)Nc2cccc(CCO)c2)CC12CCC2 13210,C1(F)(CNC(C(c2c(C)cccc2)C)=O)COCCN(C(=O)COC(F)(F)F)C1 13211,c1(OCC)cccc(C=CC(N2CC3(NC(=O)C=CC(C)(C)SC)CC2C3)=O)c1 13212,C(CC(=O)NC1CCN(C2CCN(C)C2=O)CC1)(C(F)(F)F)OC 13213,N1(C(c2ccc(C)cc2F)=O)CCC2CN(C(=O)CC3CCCCO3)C2C1 13214,c1(C(C)C)noc(C(=O)NC2CCC(NC(=O)CC3CCC(C4CC4)O3)C2)n1 13215,c1(NC)ccnc(C(N2CCC(CNC(=O)CCC(C)c3ccccc3)C2)=O)c1 13216,C(=O)(CCCC(=O)NCCCC(C)(C)NC(C1CC2CCC1C2)=O)NCC 13217,N1(Cc2cc(C)on2)CCC(N=c2cc(C)nc([N+](=O)[O-])[nH]2)C1 13218,N12CCC(CC1)OCCNC(=O)C2C1C(C)C1.c1(OC2CCCC2)cccs1 13219,c1(CNC(N2CCC(OCC3(CO)CCC3)C2)=O)c(C(F)(F)F)cccc1F 13220,c1(C(N2CC(C(C)NC(c3ncncc3Cl)=O)OCC2)=O)ccnc(C#N)c1 13221,Cc1cccc(CN(CC(C)C#N)Cc2ccc(OCF)cc2)c1C 13222,N1(C(c2ccn(C)c2)=O)CC=C(CC(=O)NCC2(O)CCCCC2)CC1 13223,N1(C(C(N2CCC(=C)C(c3ccccc3)C2)=O)=O)CCCC(C)(C)CC1 13224,C1(CNC(c2nn(CC)nc2C)=O)(NC(C2CC(O)C2)=O)CCCCC1C 13225,c1(C(=O)NC2COCCN(C(C(CCSC)O)=O)C2)cc2ncccc2s1 13226,c1(C(=O)NC(C2CCN(C(C=CCC)=O)C2)C)c(C)cnn1C 13227,c1(CNC(C2CCCN2C(c2ccno2)=O)=O)ccc2ncsc2c1 13228,C(CC(C)C)(C(=O)NC1(CNC(C2CCOC2)=O)CC1)OC 13229,C1(C(=O)OC)CC2CCC(C1)N2S(=O)(=O)CC1(C(=O)NCC(CSC)OC)CC1 13230,C(C(C)C(=O)N(C1CCC1)C)N(C(CCNC(C)=O)=O)C 13231,C1(NC(C(CC=CC)C)=O)C2CCC(C2)C1C(=O)NCCC1CCC(C)C1 13232,c1(C(=O)NCC2C(CNC(C(C=C)(C)O)=O)C2)ccc(C2CC2)c(Br)c1 13233,C1(C(=O)NCC(C)(C)C(F)F)CN(C(=O)CC2CC(C3CC3)C2)C2(CCC2)C1 13234,N1(C(c2cc(CC)n[nH]2)=O)CC(n2cc(C3CC=CCC3)nn2)CC1C(=O)OC 13235,C1(C(C(C)C)NC(C(CC)F)=O)CCN(C(=O)C=Cc2cnccn2)CC1 13236,c1(C(=O)NCCCN(C(c2cnc[nH]c2=N)=O)CC)ccc(F)cc1OC 13237,C1(C(C)OC)CCN(C(=O)C=CC(C)NC(=O)C(C)C2CCCC2)CC1 13238,N1(C(CC(c2ccc(Br)c(F)c2)C)=O)C2CCC1C(NC(=O)C(N)=O)C2 13239,C1(N(C)C(c2cccc(Cl)c2)=O)CN(CC(=O)NCCN2CCC2CO)CC1F 13240,N1(C(CC(CN(C)C)O)=O)CC(C(=O)NCC(C)(C)CCCO)C(F)(F)C1 13241,N1(C(CCC2(C)CN(C(C3CCOC3)=O)C2)=O)CCCN2CCCC2C1 13242,Cc1cccn2c(CC(=O)NCC(CC(C)C)NC(=O)CCC(C)(C)C)cnc12 13243,CN1CCN(C(c2cc(O)n(C)n2)=O)C(C(N2CCCC(OC3CC3)C2)=O)C1 13244,c1(CC)cc(C(=O)NC(C)CCCCNC(=O)CC(C)CF)ccc1Cl 13245,C(=O)(CC(C)(C)C1CC1)N1CCC(C(C)N(C(c2ccc(C(C)=O)o2)=O)CCO)C1 13246,N1(C(C=C(C)Cl)=O)C(CNC(c2cc(C3CCC3)[nH]n2)=O)CC2COCC12 13247,c1(-c2ccc(OC)cc2)n[nH]c(=NC(=O)Nc2ccc(CN(C)C)cc2)s1 13248,C(CCCC(=O)O)n1cc(SCCNC(C(c2ccnn2C)C)=O)nn1 13249,CC(C(CO)NC(c1csnc1-c1ccccc1)=O)NC(c1ncccn1)=O 13250,C(CS(=O)(=O)C1CC1)NC(c1cc(Cl)ccc1C(F)(F)F)=O 13251,C12(C(=O)NCCN(C(C3CC3C(=O)OC)=O)CC)CCC(C1)C2c1ccccc1 13252,CC(C)CC(O)CC(=O)N1CCCCC(NC(=O)C(F)(F)C2(O)CCC2)C1 13253,C#Cc1cc(C(=O)NCC2CCN2C(c2ccoc2C)=O)cc(F)c1 13254,N1(C(CCCC)=O)CCC(NC(c2cnc(-c3ccsc3)s2)=O)C(CC)C1 13255,c1(CC(=O)NC2C(NC(C=CCOC)=O)CC2)nnc(O)c2ccccc12 13256,N1(C(C2CC=CC(NC(C3(CO)CCCCO3)=O)C2)=O)CC2C=CCC(C2)C1 13257,c1(C(=O)N)cn2ccnc2cn1.C1(C2CCCC2)CCCN1C(C1CC1F)=O 13258,C1(C(N(C(C)C(=O)NC2CCOC2)CCC)=O)CCCC(C#N)C1 13259,Nc1ccc(C(N2CC(NC(=O)C(F)C(F)(F)F)C2)=O)nc1C(F)(F)F 13260,C(C(O)CNC(=O)CSC(=N)N)NC(C1C(CCC)C1)=O 13261,C1(C(N(C)CC2N(C(c3c(CC)[nH]cc3)=O)CCC2)=O)(NC)CCCCC1C 13262,C1(C(N2CCC(OCC#C)C2)=O)CN(C(=O)CC2CCCC3CC23)CC1CC 13263,CC1CC(=O)NC1C(N1CCC(CNC(c2ncoc2C(F)(F)F)=O)CC1)=O 13264,c1(OCC)ccc(OCCOC2COC3CC2C3)cc1 13265,c1(NC2(CNC(c3cncc(NC)c3)=O)COC2)ncnc2cc(Br)ccc12 13266,C(=O)(C1CCCc2sccc21)NCC1(NC(C2CCN(C)C2)=O)CC1 13267,Cc1cccc(CNC(=O)C(CCC2CC2)NC(=O)C(C)c2cc[nH]n2)n1 13268,C(c1ccc([N+](=O)[O-])s1)=CC(=O)NC1CCCCN(C(C2CCCN(C)C2)=O)C1 13269,c1(OC)cc2nn[nH]c2cc1C(=O)NCCCCNC(c1cnn(C)n1)=O 13270,C1(CC(=O)NC2(CC(=O)NCC(c3nccs3)C)CC2)CCN(C)CC1 13271,c1(C(N2CC(C(C)NC(C=CC(=O)OCC)=O)C2)=O)ccnn1C(C)CC 13272,c1(CC(=O)NCC2C(NC(C3(C)CC3)=O)CCC2)ccc2nonc2c1 13273,C1(C(=O)NC(C23CCC(CC2)C3)C)(NC(C2CCO2)=O)CCCCC1 13274,c1(C(N2CC3CC3(C(=O)NCc3cncnc3)C2)=O)cc(Cl)c(O)cc1F 13275,C#CC1(C(=O)NCC(C)(C)C2(O)CCC2)CCN(C(=O)CCC2CC2)CC1 13276,CC(C)C(F)(CNC(C1CCCN1C1CC1)=O)C(=O)NCC(C)(C)CN=[N+]=[N-] 13277,n1(CC(N2C(C)CN(C(C3(C(C)(F)F)CC3)=O)CC2)=O)ccc2ccccc12 13278,C1(C(=O)NCC(CCNC(CNC(=O)OC)=O)O)CCS(=O)(=O)N1C 13279,C(=O)(C1CCCn2cnnc21)NCC1(NC(=O)COc2cccnc2)CC1 13280,c1(N2CC(OCCNC(CC3C(C)CCO3)=O)C2)ncnc(N(C)C)c1[N+](=O)[O-] 13281,c1(C(=O)NCCCN(C)C(c2cscc2Cl)=O)nnn(C)c1C(F)(F)F 13282,C1(SCCC(N2CCCC2C2(NC(CC3C(C)C3)=O)CC2)=O)CNC(=O)CO1 13283,C1(C(N2CCN(c3nc(C)cc(C)n3)C3C2C3)=O)CCCC2CCCCC12 13284,Cc1ncccc1NC(c1c[nH]nc1CCCNC(=O)CC1CCCC(C)O1)=O 13285,c1(C(=O)NCC(CC)NC(C2NC(=O)CC2C)=O)ccc(N)cc1O 13286,C1(C(=O)NCC2(C(N)=O)CN(C(c3n(C(C)C)nnc3)=O)C2)CCC12CCC2 13287,c1(OC)cc(F)c(F)cc1CN1CC(C(=O)Nc2cc(Cl)ncc2F)CC(F)C1 13288,N1(C(C2N(C(C3C(C(C)C)CCO3)=O)CCC2)=O)CC2(CCC2)CC1CO 13289,C1(CC#C)(C(=O)NC(CC(N)=O)C2CC2)CCN(C(c2ccnn2C)=O)C1 13290,c1(OCC)cc(C)nc(N2CCC(NC(c3cccc(C4CC4)n3)=O)C(F)C2)n1 13291,O=C1CN(C2(Sc3ccccc3)CC2)CCN1C1CCOC1 13292,N1(C(c2cnc(C)n2C)C(=O)NC(C)C)CC(OCC(F)(F)F)Cc2ccccc21 13293,N1(C(C(CC#C)C)=O)CCOC2CN(C(=O)Cc3cccc(OC)c3Cl)CC12 13294,C1(NC(C2CC(O)(C(F)F)C2)=O)CCC(NC(C2CCOCC2)=O)C1 13295,Cc1ncc(S(N)(=O)=O)cc1C(N1CC2C(CN(C)C(C3CC3C#N)=O)C2C1)=O 13296,O=C(C#CC1CCOCC1)NC12CCCN(C(=O)Cc3cn4ccsc4n3)C1C2 13297,c1(C(=O)NCC(C)N(C(CN(CC)CC)=O)C)coc2cccc(Br)c12 13298,C(CC)(CCCO)Nc1sc(C(=O)OCCCCCC)c(C)c1 13299,c1(OC)ccc2[nH]c(C(N3CC(CNC(=O)CCCC#CC)C3)=O)cc2n1 13300,C(=O)(C(CC(C)C)ONC(C1(O)CCSCC1)=O)NCCCc1nc(C)[nH]n1 13301,c1(C(=O)NC2C(C)CN(C(=O)CCC3(C)CC3)C2)ccc(N)cc1Cl 13302,C(c1cccc([N+](=O)[O-])c1)=CC(=O)NC1CC(C(N)=O)OCC1 13303,Cc1ccc(O)cc1CN1CC(C)CC1C(=O)NC1CCN(S(C)(=O)=O)C1 13304,c1(CC)nn(C)cc1C(=O)NC1CC(CNC(=O)C(C)(C)NS(C)(=O)=O)C1(C)C 13305,CC1(C)C(C(=O)NCC(F)(F)C(F)F)C2CCCN(C(C3C=CCS3)=O)C12 13306,Cc1ccc2ccc(C(=O)NCC(C3CC3)NC(C3C(F)(F)C34CC4)=O)nc2c1 13307,CC1CCN(C(C2CN(S(N)(=O)=O)C2)=O)CCN1C(c1ccn2ccccc12)=O 13308,c1(C(=O)NC(CNC(c2cc(C(C)C)sc2)=O)C(C)(C)C)ccn2ccnc2n1 13309,CC(CO)(C(=O)NC(C1CCCCC1)CO)NC(=O)CCC1CCOCC1 13310,N12CCOC(C1)C2.n1(CCC=C)cc(CC(c2ccccc2)O)nn1 13311,c1(CC)cnc(C(=O)NCCCCNC(c2cc(Cl)n(C)n2)=O)nc1 13312,CC1CN(C(=O)CS(N)(=O)=O)CCC1NC(c1cnc(C(C)(C)C)nc1)=O 13313,C1(CC(=O)N(CC(C)NC(=O)CCCCCn2cnnn2)C)CCS(=O)(=O)CC1 13314,CCC(CC)C(=O)NC(CNC(C1CC(O)(C(F)F)C1)=O)Cc1ccccc1 13315,CC1CC2CN(C(C3CC3(F)Cl)=O)CC2N1C(=O)C(O)CC(N)=O 13316,C1(OCC(N2CC(Oc3cc[nH]n3)C2)=O)CCN(C(C23COCC(C2)C3)=O)CC1 13317,C1(C(=O)NC(c2ccnc(F)c2)C)CCCCCN1C(c1ccc(C(N)=O)o1)=O 13318,CCC(C(=O)N(C)CCN(C(=O)CC1CCCO1)C(C)C)NC(c1ccco1)=O 13319,C1(C(N2CCCC2CNC(C23CC(F)(C2)C3)=O)=O)CCN(CCO)C(=O)C1 13320,C1(NC(C(C)OCC)=O)CN(C(c2c(Cl)csc2Cl)=O)CC1(C)C 13321,N12CCC(CC1)C2=O.S(=O)(=O)(CC1CCOC1)Nc1nccs1 13322,CC(=O)C(C)CC(C)C(=O)N1C(C(N2CCC(C)(C)C2)=O)C2CC(O)C1C2 13323,C1(C(=O)NC2CCC(CNC(=O)CSC3CC3)C2)CC2(CCOC2)C1 13324,C(=O)(CC(C)C(F)F)NCC(CC=C)NC(=O)CN(CCCC)CC 13325,CN(C)S(=O)(=O)N(C)CC(=O)NCCC1CCC(NC(=O)CC2CC(F)C2)C1 13326,c1(OC)cc(-c2cncc(C(N3CCCC(OC)C3CO)=O)n2)c(OC)cn1 13327,c1(C(=O)NCC2(F)CC(NC(C3C(OC)CCC3)=O)C2)oc(CO)nc1C 13328,C1(NC(CC(n2c(C)cc(C)n2)C)=O)C2CC1CN(C(=O)CNS(N)(=O)=O)C2 13329,CC1CCC(CNC(=O)C(O)C(F)(F)F)CN1C(c1cnc[nH]1)=O 13330,CC(C#N)CCC(=O)N1CC(CNC(c2cc(-c3cnn(C)c3)on2)=O)C(C)C1 13331,C1(C)(C(=O)NCc2c(C(N(CCOC)CCOC)=O)nco2)C=CCCC1 13332,C1(N(CC#C)C)CCN(C(C2CC2C(=O)OC)=O)CC1.C1(C=O)CC(=O)N(C2CC2)C1 13333,c1(C(=O)OC)cnc(N2CCC(OCCNC(C3CC=CCO3)=O)C2)s1 13334,C1(C(=O)NCC(C(C)C)O)CN(C(=O)CC2CSCCO2)CC1(C)C 13335,c1(CC)c(C(=O)NCC2CCCN(C(=O)C(C)Cn3cccn3)C2)cnn1C 13336,C(=O)(C(CO)C(C)C)NC1(C)CCN(Cc2cccc(C(C)C)c2)C1 13337,c1(OC)ccc(C(=O)NCCNC(=O)CC2CCCC(C)C2)nc1Br 13338,N1(C(CC(CC)C(C)C)=O)CCCC2(CCN(C(=O)C(C)(C)C(O)CF)CC2)C1 13339,C1(NC(c2c(C)cns2)=O)CCC(CNC(c2csc(Br)n2)=O)CC1 13340,C1(C(=O)N=c2ccnc(-c3ccccc3)[nH]2)CC(c2cccnc2)=NO1 13341,CC(C)C(CNC(=O)CCn1cccc1)C(=O)NC(C)(C)CC1CCCC1 13342,Cc1c(C(=O)NC2CC(C(=O)NCC3COCC3(C)C)C2)ncn1C 13343,N1(C(COCC(C)C)=O)CC2(C1)SCCC2NC(=O)CCCC(N)=O 13344,CC1CN(C(c2cccc(F)c2)=O)CCC1C(=O)NCc1ccc(O)nc1 13345,C1(C(N(CC(CCC)O)C)=O)(CNC(c2c(C)cnn2C)=O)CC12CCC2 13346,C1(C(=O)NCCn2cc(C(=O)NC(C=CC(=O)OCC)C)nn2)CC2(C1)CC21CC1 13347,c1(N(C2CCN(C3CCOCC3)CC2)C)cc(N(C)C)c([N+](=O)[O-])c(F)c1 13348,N1(Cc2ccc(OC)c(OC)c2C)CCC(C2CCN(C)CC2OS(C)(=O)=O)CC1 13349,N1(C(C(CC)NC(N)=O)=O)CC2CCC1C(NC(=O)C(c1cccnc1)SC)C2 13350,C12(C(=O)NCCCC(=O)OC)CC1CN(C(c1cc(C(C)(C)C)no1)=O)C2 13351,C1(CC(N2CCC(NC(CCC#C)=O)CC2C)=O)CSc2ccccc2O1 13352,c1(OC)ccc(F)cc1C(=O)NC1CCC(C(=O)NCC(C)(C)F)CC1 13353,C(C)(CCC(=O)NCCN(C)CCOCCNC(c1cccc(COC)c1)=O)OC 13354,c1(C2(C(=O)NC(C)C(C)(C)c3ccccc3)CC2)cccc(OC(F)(F)F)c1 13355,N1(CC(=O)NC2CCC2NC(C2(CC(F)F)CC2)=O)Cc2ccccc2C1 13356,Cc1nc(O)nc(O)c1CC(=O)NC12CCCC1N(C(=O)C(F)(F)C(C)O)CC2 13357,N1(C(CC(CC)(C)C)=O)CCCN(C(c2ccc(OC3CCC3)cc2)=O)CC1C 13358,CC1CCC(CNC(=O)C(CC23CCC(CC2)C3)NC(C2CC2C#N)=O)N1C 13359,C1(C(=O)NCCN(C(C(c2ccccc2)OCCC(C)C)=O)C)CCCCCC1 13360,c1(CC(=O)NCC(CNC(=O)CSc2ccccc2C)OC)cccnc1C 13361,C12(C(=O)NCCCN(C(=O)CN3CCCS3(=O)=O)CC)CCCCC1C2(F)F 13362,c1(COC)nc(NCCC2(C)CCOC2)cc(=NCc2c[nH]c(=N)s2)[nH]1 13363,N1(C(COCCCC)=O)CCC(C(C)(C)CNC(=O)CC2NC(=O)NC2=O)CC1 13364,CC1CC(NC(=O)CC2CC3(CC3)C2)CCN1C(=O)CCN1CCCCC1=O 13365,CC(C)CC(C)(CNC(C1CC(=O)NC(=O)N1)=O)NC(C1CC(F)(F)C1)=O 13366,C1(C(=O)NCCN(C(=O)CCc2cnoc2)CC)CCC(=O)N1CCC(F)(F)F 13367,C1(OCC(=O)NCC2(CNC(n3ncc(C(C)=O)c3)=O)CC2)CCCCC1C 13368,C1(NC(C2=C(C)CC2)=O)CN(C(c2csc(CO)n2)=O)CC(F)(F)C1 13369,CCC(CC(=O)NCC1(O)CCN(C(=O)COC2(C)CCCC2)C1)CC(C)C 13370,C(=O)(CC(C(=O)NCCN(C(=O)CCCCS)C(C)C)NC(C)=O)OC.C(C)C 13371,N1(C(=O)OC(C)(C)C)CCC(CC(N2CC3CC3(CO)C2)=O)C(C)(C)C1 13372,Cc1cc(C)c(C(=O)NCCC2CN(C(C3CNC(=O)N3C)=O)CCO2)c(C)n1 13373,CCN=c1[nH]c(C)c(C(=O)NCC2(CN(C(=O)Cn3nc(C)oc3=O)C)CC2)s1 13374,c1(CN2CC(CC(=O)NC(C3(C(=O)NC)CCC3)=O)OCC2)ccc(C#N)n1C 13375,c1(C(N2CCC(NC(CC(CC)C)=O)C(F)C2)=O)cc2nc(C)ccc2o1 13376,c1(C(=O)NCC2CC(COC)CN2C(=O)C(C)CF)cc2ccc(F)cc2o1 13377,c1(C(=O)NCCCCCNC(C(C)OCCC#C)=O)ccc(Br)cc1O 13378,C1(CNC(CNC(C)=O)=O)CN(C(c2cc(Cl)ncc2O)=O)CC2(CCC2)O1 13379,N1(C(C(C)NC(C2CN(C)C2)=O)=O)CC(=O)NC(=O)C1C 13380,c1(OCC)ccc(CCC(C)NC(=O)CC2CSCCS2)cc1 13381,CC1(C)OC(=O)NC1C(=O)NC1COCCC1NC(C1CC(F)(CF)C1)=O 13382,c1(SC(C)C)ccccc1C(=O)NCC(C)(C)CN(C)C(c1cc(O)ccn1)=O 13383,c1(C(=O)NCCCN(C)C(c2scnc2C(C)(C)C)=O)ccn(C)c(=O)c1 13384,N1(C(c2cccc(Cl)n2)C(=O)NC(CC)(C)C)CCC2(CC=CCO2)C1 13385,C1(F)(C(N2C(CN(C(=O)C=CC=C(Cl)Cl)C)COCC2)=O)C(C)(C)C1(C)C 13386,C(C(CC(C)C)NC(C1CC(=O)N(CC)C1)=O)NC(c1c(CC)noc1)=O 13387,c1(CC)onc(C(=O)NCC2C=CCN2C(=O)C(O)C(C)C)c1C 13388,c1(C(=O)OCC)ccc(C(=O)NCCNC(C2(C)CCOC2)=O)cc1 13389,C1(CNC(C(C)CC2CCCC2)c2nnnn2C)CCCCS1(=O)=O 13390,c1(CNC(=O)COCCCCCC)cccc(-n2cc(-c3ccncc3)nn2)c1 13391,N1(C(C(c2scc(C)n2)(F)F)=O)CC(NC(c2cc(Cl)ccc2O)=O)CC(O)C1 13392,N1(CC)CCCC(C(=O)NC2CCCC2NC(c2c[nH]c(=S)cn2)=O)C1 13393,N1(C(C(C)CC2CC2)=O)CC(CNC(=O)CCc2ccc(F)nc2)CC1(C)C 13394,C1(Br)(C(=O)NCC(C)N(C(c2cc(CC)on2)=O)C)CC12CCC2 13395,c1(C(=O)NC(C(C)C)CNC(=O)COCC(F)F)cn(C)nc1C(C)(F)F 13396,Cc1ncnc(C)c1NC(c1coc(CNC(=O)CCc2ccncn2)c1)=O 13397,C1(CC(N2CCC(CCNC(CCCC(OC)OC)=O)C2)=O)CCCC2(CC2)C1 13398,c1(N2CC(CNC(=O)C(F)CC3CCCC3)OCCC2)nc2ccc(F)cc2o1 13399,c1(CNc2cccc(C(=O)NCCCN(C)C)c2)ccc(P(C)(C)=O)nc1 13400,C#CCC(C)(C)C(=O)N1CCOC(CCNC(=O)Cn2ccc(C)c2)C1 13401,CC(O)C(C(=O)NCC1CCCCN1C(c1coc(C(F)F)c1)=O)N(C)C 13402,c1(C(N2CCC(C(C)(C)NC(CCC=C(C)C)=O)CC2)=O)cc(S(C)(=O)=O)cs1 13403,N1(C(CCCCSC)=O)C2CC1CN(C(=O)CCP(C)(C)=O)C2 13404,c1(CCC(=O)NCC(C)(C2CC2)NC(C2(F)CCCCC2)=O)nc2ccccc2[nH]1 13405,N1(C(c2cnc(CC)[nH]2)=O)CC2CC2(CNC(=O)CC2CCC(=O)N2C)C1 13406,c1(C2C(=O)NN2C)ccc(OC)nc1C.c1(COCCOCC)cc(Br)cs1.O.O=C.C 13407,Cc1ccc2[nH]c(NC(c3ccc(Cn4cc(CNC(C)C)nn4)o3)=O)cc2c1 13408,Cc1nc(N(C)CCOCCNC(=O)C(C)(C)CNC(N)=O)cc(Cl)n1 13409,C(=O)(CCCCC(F)(F)F)NC1CC(NC(c2cc(C3CCC3)[nH]n2)=O)CC1O 13410,c1(OC)ccc2c(c1)C(C(=O)OCc1cccc(CO)n1)C(C)N2 13411,Cc1cccc(C(N2CCCC(C(=O)Nc3cccc(C(C)F)c3)CC2)=O)c1O 13412,N1(Cc2nnc(C(C)C)o2)CCCOC(CNC(c2occ3c2CCC3)=O)C1 13413,CC1CCN(C(C23CC(C)(C2)C3)=O)CCN1C(=O)C(C)N1CCC1 13414,C1(C(=O)OC)CC(Cc2ccnc(OC3CC3)c2)N(C(c2cn(CCl)cn2)=O)C1 13415,Cc1cc(OCC(C)C)c(-c2ccc(NCc3ncc(Br)cc3Cl)s2)cc1C 13416,C=CCCCCCC(=O)NCC(CCCC)NC(c1cc(=O)cc[nH]1)=O 13417,N1(c2n(CC=C)c(C3CC3CC)nn2)CCCC(n2ccnn2)CC1 13418,C1(CNC(C(C)(F)CC2CCCC2)=O)CCCC2CN(C(=O)CC=C(Cl)Cl)CC12 13419,C#CC1(C(=O)NCc2ccncn2)CCN(C(=O)C(=O)C2CCCC2)C1 13420,Cc1noc(C(C(C)C)NC(=O)CC2CCN(C(=O)C(C)CN(C)C)C2)n1 13421,c1(CC(=O)NCC(C(C)(C)C)NC(=O)CC(C2CC2)C2CC2)c[nH]c(=N)nc1O 13422,C1(N(C(CCOCC#C)=O)C)CCN(C(=O)C=C(CCC)CCC)CC1C 13423,C(=O)(C(CCNC(=O)CCCCC1CC1)OC)N(C1CCN(C)C1)CC 13424,C(=O)(C(C)OCC(C)C)NCC1C(CC(=O)NC(CO)C2(CC)CC2)C1 13425,C1(C(=O)OC)(CNC(=O)C(C2CCCC2)NC(c2coc(O)n2)=O)CCCC1 13426,c1(C2(C(=O)NCCOCCCNC(CC(C)F)=O)CCC2)ccc([N+](=O)[O-])cc1 13427,NS(=O)(=O)CCCC(=O)NCCC1CCCCN1C(=O)CCN1CCCCC1 13428,N1(C(CCN(C)C(C2C3CCCCC23)=O)=O)CCC12CC(CO)C2 13429,C1(NC(=O)OC(C)(C)C)C2CCC(C2)C1NCC1CCCC1C(C)(C)C 13430,C(=O)(C1=CS(=O)CCC1)NCC1CC(NC(CCNS(CC)(=O)=O)=O)C1 13431,c1(C(=O)NCC2(F)CCN(C(CN3C(C)CCC3)=O)C2)nc2ncccn2n1 13432,c1(CNC(c2c(C)cncc2C)=O)nc2c(s1)CN(C(=O)C(C(C)O)N(C)C)C2 13433,C1(CC)CN(C(=O)CCCn2ccnc2)CC1C(=O)NCC1(C)CCN(C)C1 13434,C(C)(C)(CC(=O)NC(C)C(=O)N(C)C)c1cncc(CN)c1.c1(C(C)O)c[nH]nn1 13435,c1(C(=O)NC(C)CN(C(=O)CCCCc2cnc[nH]2)C)cnc2ncccn12 13436,c1(CN(C)CC2CCN(C(=O)CCSC(F)(F)F)C2)cccc(O)n1 13437,C#Cc1cccc(C(=O)NC(CNC(c2ccc(S(C)(=O)=O)o2)=O)C(C)C)c1C 13438,C#CCC(C)(C)C(=O)NC1CCC(CNC(C2CCCOC2)=O)C1 13439,c1(CC(N2CCC(C(=O)Nc3nc(Br)ccc3Cl)C2)=O)ccc2cc[nH]c2c1 13440,c1(C(=O)OC)nn(C)cc1C(=O)N(C)CCNC(C1CC(C)OC1=O)=O 13441,C1(N2CCN(C(C(C)C)=O)CC2)CCN(N2CCC(c3cccc(Cl)c3)C2)CC1 13442,CC(C(C(=O)NC1CCOC1)N(C1CCC1C)C)C(C)(C)C 13443,C1(F)(C(N2CC(OC)C(OC)C2)=O)CCN(C(c2ccc(O)nn2)=O)C1 13444,c1(N2CC3CC(CNC(CSc4n(C)cnn4)=O)C3C2)nc(Cl)nc2ccccc12 13445,C=CCCCC(=O)NCC(C)(C)Cn1cc(-c2ncccn2)nn1 13446,c1(C(N2CCN(C(CS(CC)=O)=O)CC2CF)=O)cc2ccncc2cc1F 13447,c1(CC(=O)NC2CN(C(C3(CCC=C)CC3)=O)CC2C)cc(C)ccc1OCC 13448,C(N=c1[nH]c(=NCc2cc(F)ccc2C2CC2)c2[nH]ccc2[nH]1)c1cc(C)ns1 13449,C(=O)(C(F)(F)C(C)(C)O)NC1CCCC(N(C(c2c(SC)csc2)=O)C)C1 13450,C(=O)(CC(C(F)F)n1ccnc1)N1CC(O)(CC(=O)NCCC2CCCO2)C1 13451,c1(-n2ncc(I)c2)cccc(-n2cc(-c3ccccc3N3CCOCC3)nn2)c1 13452,c1(CNC(N(C(C)CC2CC2)C)=O)nccc(Br)c1O 13453,c1(C(N(CCCCN(C(=O)Cc2ccn(C)c2)C)C)=O)csc(C(C)(C)C)n1 13454,C1(CC)(NC(=O)CCSCCNC(C2CCN(C)C2)=O)CC(C)(C)C1 13455,C(C(CC(C)C)C(=O)NCC(C)CNC(c1nccn2cnnc12)=O)OC 13456,C1(C)(C(=O)NCC2(CN(C(=O)CSC(F)(F)F)C)CC2)CCC2CC2C1 13457,N(C(=NCC1CCCO1)NC1CCC(c2ccc(F)cc2)C1)CC1(C)CCCS1 13458,c1(OC)ccc(C(=O)N(CC(C)CNC(=O)C(=Cc2ccncc2)C)C)c(C)c1 13459,CC(C)C(C#N)C(=O)N1CCC(NC(c2cnc(-c3cnccn3)s2)=O)C12CC2 13460,c1(CCNC(C23CC(NC(C4(F)COC4)=O)(C2)C3)=O)cccc(O)c1 13461,CC#Cc1ccc(C(N2CCN(C3CC3)C(C#N)C2)C(=O)NCC2CCC2)cc1 13462,C(CC1=CCCCC1)N(C(c1cc(Cl)cs1)C(=O)NC(CC)C)C 13463,N1(C(c2cnc(C)c(Cl)c2)=O)CC2CC1CCN2C(C1CC(=O)N(C2CC2)C1)=O 13464,c1(C(=O)NC(CC)CNC(c2conc2C2CC2)=O)ccc(SC(F)(F)F)nc1 13465,N1(C(C(c2cnn(C)c2)C)=O)CCC(C)CC1C(=O)NOCCCCF 13466,O=C(C1=CCCSC1)NCCCCCCNC(C1COCC1C(F)F)=O 13467,C1(C(N(CCNC(C2(C3CCC3)CC2)=O)CC)=O)CCCCN1C(C)=O 13468,c1(C(N(C)CCOCCNC(C2CCC23CCC3)=O)=O)cc2cccnc2cn1 13469,C1(C(=O)NCc2nc(CC)[nH]n2)C=CCN(C(C2CCCC(=O)C2)=O)C1 13470,N1(C(C(C=C)C)=O)CCN2CCN(C(c3cc(Cl)c[nH]3)=O)CC2C1 13471,C(=O)(CC(C)(C)C(F)F)N1CC2C(CNC(C(C)(C)N3CCCCC3)=O)(C2)C1 13472,C1(CCNC(Cc2c(C)n[nH]c2C)=O)CN(C(c2nn(C)cc2Cl)=O)CC(C)O1 13473,C1(N(C)C(C2CC2(C)C)=O)CN(C(=O)Cc2ccc(Cl)cn2)CC1(C)C 13474,c1(C(=O)NC2(CC(N)=O)CCN(C(CC(C)F)=O)CC2)ncnc2c1CCC2 13475,c1(NC(C(=O)N(CCc2c(C)ncs2)C)=O)ccc2nc(Br)sc2c1 13476,c1(CNC(C(C(C)(C)C)O)=O)ccc2c(c1)CN(C(=O)C1=CCCOC1)C2 13477,N1(C(C2N(CC)CCC2)=O)CCC(NC(=O)C(C)NC(=O)NC(C)C)C(C)(C)C1 13478,c1(C(N2CC(NC(CC3(C=C)CC3)=O)C(C)CC2)=O)c(C)cc(C#N)cc1C 13479,CN1CC=C(C(=O)NCC(c2ccccc2)CNC(C2CC3(CSC3)C2)=O)C1 13480,c1(C(N2CC(C(N)=O)(CNC(C(C)n3cncn3)=O)C2)=O)ccnc2[nH]c(O)nc12 13481,c1(OC)ccc(-c2cncc(C(=O)NC3CC3NC(C3CC3C#N)=O)c2)c(C)c1 13482,Cc1[nH]nc(Cl)c1C(=O)NCC1CC(NC(=O)Cc2cn(C)nc2Cl)CC1O 13483,N1(C(C(CC)(CC)CO)=O)CCOC2(CCCN(C(=O)CCC(=O)OC)C2)C1 13484,c1(C(C)C)ccc(C2CCN(C(=O)CN3CCCCC3)CC2)cc1 13485,c1(C(CNC(=O)C(O)COC)NC(CCC=C)=O)ccc(OCC)cc1 13486,Cc1cc([N+](=O)[O-])cc(C(=O)NC2(CO)CCCN(C(=O)COC3CCC3)C2)n1 13487,c1(C(=O)NC2CC(CNC(C3=CCCC3C)=O)C2)n[nH]c2c1CCSC2 13488,C1(C(=O)NCC2(C)CC(NC(C3(OC)CC3)=O)C2)CC(c2ccccc2)=NO1 13489,c1(C(N2C(CNC(COCCCOC)=O)COCC2)=O)cc2ccccc2s1 13490,N1(C(C2CCSCC2)C(=O)NC(C(=O)OC)C)C2CCC1CC(CO)C2 13491,C1(NC(C(N2CCC(C)(CCO)C2)c2ccc(CF)cc2)=O)CCC(F)(F)CC1 13492,CC(C)(O)C(F)C(=O)NCC1CN(C(C2OCCOC2(C)C)=O)C1 13493,C1(C)(N(C)C(C2(CCNC(=O)CCCC3CCCC3)CC2)=O)CCCC1 13494,C(=O)(CC(CC(C)C)NC(c1cc[nH]c1C)=O)NCCC(CC)O 13495,c1(C(N2CCN(C(CCCCC=C)=O)CC2)=O)cc2c(C(=O)OC)cccc2s1 13496,C(=O)(C#Cc1ccccc1)Nc1cc(OC)ncn1.N12CC3C(C3C1)C2=O 13497,C1(CNC(CCN(C(C2(C(C)C)CCCC2)=O)CC)=O)CC(C)CC(C)C1 13498,CC#CCC(C)NC(C1(CCNC(=O)CC(Cl)Cl)CC1)=O 13499,c1(C(=O)NC2CC(CNC(C3C(C)CC(=O)N3)=O)C2)cc(O)ccc1[N+](=O)[O-] 13500,c1(C(N2CC(NC(=O)C(F)C3CCC3)(CO)C2)=O)cncc([N+](=O)[O-])c1 13501,C1(C(F)(F)F)(C(N2CC(NCC(N3CCOCC3)=O)(CO)C2)=O)CC2CC2C1 13502,C1(C(=O)NC2CC(NC(c3c(C)n[nH]c3)=O)CC2O)C(F)(F)C12CCC2 13503,c1(SCC(=O)NCCC2OCCN(C(C3C(C=C)C3)=O)C2)ccc2c(c1)OCO2 13504,C(CC(=O)NCCOCCNC(c1snc(Cl)c1Cl)=O)(C1=CCCC1)OCC 13505,N1(C(C=C(C)C)=O)C2CCC1C(CNC(=O)C(F)F)C2 13506,Cn1ccc(C(N2CC(=C(F)CNC(=O)C(O)C3CCC3)C2)=O)c1C1CCC1 13507,C(C)(C)(CC(=O)N1CC(C(C(=O)NCC(c2ccccn2)O)OC)C1)OC 13508,c1(C(=O)NC2CC(F)(CNC(C(C)C3CCOC3)=O)C2)[nH]nc([N+](=O)[O-])c1Cl 13509,CC1C(NC(=O)CN2C(=O)CCC2=O)CCN1C(=O)Cc1cnn(C(C)(C)C)c1 13510,N1(C(c2n(C(C)C)ncc2)=O)CCSC(C(=O)N(CCO)CCO)C1 13511,C#CC1(NC(C2CN(C(C3CCC3(OC)OC)=O)CCO2)=O)CC2CCCC12 13512,C12(CNC(CCNC(=O)CO)=O)CC1CN(C(c1cc(-n3cccc3)ccn1)=O)C2 13513,C(=O)(C(CC(C)C)n1nnnc1C)NC(CCNC(c1c(C)c[nH]n1)=O)C 13514,N1(C(c2c(C(C)C)n[nH]c2)=O)CC2CC2(CNC(=O)C(O)CC2CCCCC2)C1 13515,n1(CCC)cc(S(=O)(=O)NCC(O)CCC2CC2)c(C)n1 13516,N1(C(Cc2c(C)nc[nH]2)=O)CC2CCCC1C2CNC(c1cn[nH]c1)=O 13517,N1(C(C(CC)O)=O)CCCC(N(C)C(c2ccnc(OC)c2)=O)C1 13518,CCCCCC(C)CC(=O)N(C1CC(NC(C2C=CCS2)=O)C1)C 13519,C(=O)(CC(C)(C)O)N(C(C(N1CC(C(=O)NC)C1)=O)C)C 13520,Cc1cc(CCNC(=O)C(Cn2cncn2)NC(=O)CC2CCSC2)n[nH]1 13521,C(=O)(C(CC(C)C)NC=O)OC.C1(O)(C(C(=O)O)(F)F)CCCCC1 13522,C1(C(N2C(CNC(=O)CN3CCCCC3=O)C=CC2)=O)CCc2cnnn2C1 13523,C(=O)(CC(CC)C(C)C)NCCCCC(=O)NC1(C(NOCC=CC)=O)CC1(C)C 13524,c1(C(N2CCC(O)(CNC(CCC)=O)C2)=O)ccc(Cl)nc1OC(C)C 13525,C(=O)(CCC(=O)N1CCC(C(C)(O)CNC(=O)C(C)SC2CC2)CC1)NC 13526,C1(CNC(C2CSCCS2)=O)CCCN(c2nc(C3CCCC3)ns2)C1 13527,C1(C)(CNC(C2N(CC)CCCC2)=O)CN(C(=O)CCCCC2CC2)C(C)(C)C1 13528,C1(N=c2ccnc(-c3ccccc3)[nH]2)(CNC(C2(O)COC2)=O)CCCC1 13529,CC1CCC(NC(c2nnsc2-c2ccccc2)=O)CN1C(=O)CCCC(F)F 13530,c1(OC)ccc(C(=O)NCC2(C)CCCN2C(c2cnc(S)n2C)=O)c(N)c1 13531,CN1CCN(C(=O)C(CCF)NC(=O)CC2CC3(CCC3)C2)CC1=O 13532,N1(C(CCS(C)=O)=O)C2CCC1CC(NC(=O)CCn1cccn1)C2 13533,c1(-c2ncc(C(=O)NCC(CO)NC(c3cnc(O)s3)=O)s2)ccc(Cl)cc1 13534,c1(C(=O)NC2C(C(=O)NCC3CCC3)CCCC2)cc(Br)cc([N+](=O)[O-])c1Cl 13535,CCC(CC(=O)NCC1(NC(C2CCCSC2C)=O)CCC1)c1ccccc1 13536,c1(C(N2CCC(NC(=O)C=Cc3cocn3)CC2)=O)ccc(Br)cc1[N+](=O)[O-] 13537,C1(C(=O)NC2CC(NC(CC=CC)=O)C(O)C2)CCCCC12CCC2 13538,C(=O)(C1CCCc2ncccc21)N(CCCNC(C1CC2(CC2)C1)=O)C 13539,c1(NC(C2CCN(Cc3cccc(-c4ccncc4)c3)C2)=O)cc(Br)ccc1Br 13540,C1(NC(c2cc(Cl)cnn2)=O)C2CCC1N(C(=O)Cc1cccc(F)c1O)C2 13541,N1(C(C(COCC)C)=O)CCN(C(c2cnn(C)c2C(C)C)=O)CC1CC(F)F 13542,N1(C(CC2(CSC)CC2)=O)CC(NC(=O)C(C)C(C)O)CC12CCCC2 13543,c1(CC)cccc(C(=O)NC2CCC(CC(N3CC4C(CO)C4C3)=O)CC2)n1 13544,C1(NC(C(CCC)C)=O)COC2(CCN(C(c3ccc(CC(N)=O)cc3)=O)C2)C1 13545,N1(C(CN(CCCCN(C)C(=O)Nc2cnn[nH]2)C)=O)CCCC(F)(CO)C1 13546,C1(NC(C(CC)(C)OC)=O)CCCCN(C(c2ccc(C)nc2N)=O)C1 13547,C(C(C)(C)CC(=O)NCC1CCN(C(c2ccnnc2Cl)=O)CC1C)OC 13548,N1(C(C2C(CC)OCC2)=O)CC2CC(NC(=O)C(c3ccc(F)cc3)(F)F)C1C2 13549,N1(C(c2cn(C)nc2)=O)CCC(CNC(c2ccc3n[nH]cc3n2)=O)C12CCC2 13550,N1(C(C(CO)N(C)C)=O)CCn2nc(C(=O)NCC(CO)C3CC3)cc2C1 13551,N1(C(CCC(C)OC)=O)CCC(NC(=O)CSc2ccncc2)C(F)C1 13552,CC(CF)CC(=O)NCC1CC1CNC(c1cc(-c2ccncc2)ccn1)=O 13553,N1(C(Cc2c(C)ncs2)=O)CC2(CCC2NC(=O)CC2COC(C)(C)CO2)C1 13554,c1(C(=O)OCC)cnn2c1C(C)N(C(c1sc3nccn3c1C)=O)CC2 13555,c1(C(N(C2CCCC2)CCCNC(C2C(C)(C)CC2)=O)=O)cc[n+]([O-])cc1 13556,c1(OC(C2CN(C(=O)CC3CCCOCC3)C2)=O)ccc(F)cc1Br 13557,C(N=c1[nH]c2c(c(=NCC3(C4CC4)CC3)[nH]1)COC2)c1cc(Cl)cc(Br)c1 13558,n1(C(C)C)ccc(C(=O)NC(C)(C)C(=O)NC(C2CCC2)C)n1 13559,CC12COCC1CN(C(=O)CN1CCCC1C(O)C(F)F)C2 13560,c1(CC(=O)NCC2N(C(CC(=O)NCC#C)=O)CCC2)cccc(C)c1Br 13561,N1(C(c2n(CC)ncc2Cl)=O)CCN(C(=O)CCc2ccoc2)C(C)CC1C 13562,C1(CC)CCCC(N=c2[nH]c(=NCCc3ocnc3CO)[nH]c3c2CCCC3)C1 13563,c1(C(=O)NC(CC)CN(C(=O)CSCc2cccnc2)C)cn(C)nc1C(C)C 13564,C1(NC(C(C)CC2CCC2)=O)CN(C(=O)CCC=Cc2ccccc2)CCC1C 13565,Cc1nn(C)c(Cl)c1C(=O)NCC1(C)CCCN1C(c1cnc(C#N)s1)=O 13566,Cn1nc(CNC(C2CC(F)(CF)C2)=O)cc1C(=O)NCCC(O)C(F)F 13567,C1(N2CC(C(=O)NCC3C(NC=O)CC3)C2)CCCCC1.C(COCCO)N 13568,N1(C(c2n(COC)ncc2)=O)CCC(C)C(CNC(c2nc(Cl)cs2)=O)C1 13569,N1(C(c2c(C)ccnn2)=O)CC2(CC(NC(C34CC3COC4(C)C)=O)C2)C1 13570,c1(C(N2CCC(C)(NC(c3cc(OC)c(C)cc3)=O)C2)=O)cc2n(n1)CCCN2 13571,c1(NCCC(C)NCC(CC(=O)OCC)C)cc(Cl)ccc1OC 13572,c1(OC)[nH]c(=NC2CCCCCN(C(=O)C(=O)NC(C)C)C2)sc1C 13573,C1(CNC(c2cnc(OCC)s2)=O)CN(C(=O)C(F)C(C)C)CC12CCC2 13574,c12nc(nc3ncn(CC)c13)NCCOC1CCN2C1.C=CCOC 13575,CC(CCCC(=O)NCc1ccc(F)cn1)NC(C1CC1C1CCC1)=O 13576,C1(C)(C(=O)NCC2CC(NC(C3CC(C(=O)OC)C3)=O)C2)CCCNS1(=O)=O 13577,c1(N(C(=O)OC(C)(C)C)CC)cnn(C)c1.C(=O)(CCN)C(COC)=O 13578,c1(CCC)[nH]ccc1C(=O)N(C1(CC(=O)NC2(CC(C)C)CC2)CC1)C 13579,c1(C(N(C=O)C)C2CCC2)ccc(C(F)(F)F)cc1.c1(C=O)cc(I)cs1 13580,Cc1csc(=O)n1CCC(=O)N(C)CCOCCN(C(=O)C=CC(C)C)C 13581,C1(C(=O)NCC2OCCN(Cc3ccc(CCC)s3)C2)Cc2ccccc2O1 13582,N1(C(CC2C(C)(C)CC2)=O)CC2CC(NC(=O)CCN3CCOCC3)C(C2)C1 13583,C1(N(C(C2CSC2)=O)CC)CCCN(C(c2ccc(O)c(F)c2)=O)CC1 13584,c1(CC)ncc(C(=O)NC(CNC(C2CC3C=CC2O3)=O)CCOC)c(O)n1 13585,C1(OCC(N2CCCCC2)=O)CCCN(C(=O)C(=O)OC(C)C)C1 13586,C1(OC(C)=O)CCCN(C(=O)NC(CO)C(C)OC)C1.C(C)(C)(C)O 13587,Cc1cc(C(=O)N(CC2CCN(C(=O)CCC3CC3CC3CC3)CC2)CC)ccn1 13588,C1(N(C(Cc2ccc(C)nc2)=O)C)CCCN(C(=O)CC(O)C(C)C)CC1 13589,C1(OC)CCC12CC(C(=O)NC1CC(CNC(=O)C3=CCCSC3)C1)C2 13590,c1(C(N(C)CC2CCCN2C(c2cc(Br)no2)=O)=O)ccc(C#N)cn1 13591,c1(C(C)C)cncc(C(N2CCC(CNC(C34CC(C3)C(C)O4)=O)CC2)=O)c1 13592,n1(C2CCC(C)C2)nc(-c2ccccc2C2CCC2)nc1C=CC(=O)O 13593,Cc1coc(C)c1CNC(=O)C(C)N(C(=O)C(c1ccccc1)=O)C1CCCC1 13594,N1(C(C)=O)CCCC1C(=O)NC(C1CCCN1C(=O)CC1CCCO1)(C)C 13595,c1(OC)cnc(Br)cc1C(N1CCN(Cc2cnn(C)c2)CC1CC#N)=O 13596,C1(C(N2CC(F)(CNC(c3c(C)cc[nH]3)=O)C2)=O)C2C(=O)OCC12Br 13597,c1(C(N(CCC(=O)Nc2ccc(C3CC3)cc2)CC)=O)cnc(Cl)cc1Cl 13598,Cc1cc(C(=O)NC2CCCC(NC(C3C4CCCOC34)=O)C2)cc2c[nH]nc12 13599,C(c1ccccc1)=C(C)C(N1CC2CC2(C(=O)NC(C)(C)C(F)(F)F)C1)=O 13600,C1(CC(=O)NCC2CCN2C(c2cn(CCl)nn2)=O)CC(=O)c2ccccc2C1 13601,C#Cc1ccc(C(=O)N(CC(CC)NC(=O)CCCC#N)C)nc1 13602,C1(NC(CCCOC(C)C)=O)CCN(C(=O)CN(C)Cc2ccccc2)CC1C 13603,CN1CCC(CCC(=O)NCCC2CCCN2C(c2cc(C3CC3)on2)=O)CC1 13604,N1(C(C2(SC)CN(C(c3c(CC)cccc3)=O)C2)=O)CC2CC(CO)C(C2)C1 13605,C1(NC(CSCCNC(c2cn(CC)nc2)=O)=O)CCCC12CC2 13606,C1(NC(Cn2ncn(C)c2=O)=O)CCN(C(c2cnc(O)s2)=O)CC1O 13607,C(=O)(C(C)(CC)C(N)=O)NC(CC)CNC(=O)COc1cc(F)ccc1F 13608,n1(CCOC)cc(C(=O)NCC(O)CCNC(=O)CSCC(N)=O)c(C)n1 13609,C(=O)(CCC(C)(C)F)NC1C(C)CN(C(c2ccc(N3CCCC3)nc2)=O)C1 13610,C=CC1CN(C(=O)CN(C2CC2)CC)CC1NC(=O)C(F)(F)C1CCOCC1 13611,C1(C(=O)NC(c2ncc(C)o2)C)CCC2(CC2)N1C(c1nn(C)cc1C)=O 13612,N1(C(C(C)CC2CC2)=O)CCCC(C(=O)NC(C)(C)C(F)(F)F)CC1 13613,C1(C)(CCCC)NC(=O)N(CC(=O)Nc2ccc(Cl)cc2Oc2ccncc2)C1=O 13614,c1(C(C)N(C)C)cn(CC(=O)NOCC2CCN(C)C2)nn1 13615,CCC(CC(C)C)C(=O)NCC1CN(C(c2ccc(O)nc2Cl)=O)CCO1 13616,CC1CCC(C(=O)NCc2nnnn2C)N1C(c1ccn(C)n1)=O 13617,N1(C(CCc2n(C)ncn2)=O)CC(NC(=O)CCOC2CCCCC2)C(C)(C)C1 13618,C=CCCCC(C)NC(=O)C(C)CNC(=O)Cn1cc(C(=O)NC)nn1 13619,Cc1ncc(C(=O)NC2CN(C(c3c(C)noc3C3CC3)=O)CC2C)cc1C#N 13620,CCCC(C(=O)N1CC(NC(C2(C3CCCC3)CCOCC2)=O)C1)OCC 13621,c1(OC)c(F)ccc(C(N2CCCC2CC(=O)Nc2cccc3c2OCO3)=O)c1F 13622,N1(C(C2(OCC)CC2)=O)CCCC(O)(CNC(=O)C2=COCCO2)CC1 13623,Cc1cc(C(N2CC(F)CC2CNC(C2CCC(C)C2)=O)=O)c(O)cc1F 13624,c1(CNC(CC2CC(OCC)C2)=O)ccnc(C(=O)Nc2cccnc2C)c1 13625,C12(CNC(C3(CO)CCC3)=O)CC1CN(C(=O)COC1CCC1)C2 13626,N1(C(CCC(C)C)=O)CCCC2C1CCCCN2C(=O)CCc1cccn1C 13627,C(=O)(C(F)C(F)(F)F)NCc1cn(C2CCN(c3cc(SC)ncn3)CC2)nn1 13628,N1(C(c2cccc(C)c2)=O)CCCC2C1CCN2C(c1cc2ccncc2[nH]1)=O 13629,C12(CNC(C=CC(C)(C)C)=O)CCC(CC1)CN2C(C1CC12CCC2)=O 13630,N1(C(c2c(OC)n(C)nc2C)=O)CC(NC(c2cccnc2S)=O)CC12CCC2 13631,C1(CC)C(NC(=O)C(CO)OC)CCN1C(c1ccncc1SC1CC1)=O 13632,c1(NC(C(C2CCN(C(C(C3CC3)OC)=O)C2)F)=O)cncc(CO)c1 13633,CCC(CC(=O)N1CC2CN(C(c3cc(Cl)c(F)cc3F)=O)CC2C1)C(C)C 13634,N1(C(=O)CC2CCC3CC3C2)CC23CCCC2(C1)CN(C(C1CCC=CO1)=O)C3 13635,C1(CNC(Cc2cc(C)sc2)=O)C(C)CCCN1C(c1ccc(C)cc1F)=O 13636,C(C(C)(C(C)C)C(C)C)NC(CC1C(C)CN(C(c2sccc2Cl)=O)C1)=O 13637,c1(C(=O)NC2CN(C(CCc3ccn(C)n3)=O)C3C2C3)ccc2cc[nH]c2n1 13638,c1(OC)cc(C(=O)NC2CCC(NC(=O)Cn3cc(Cl)cn3)CC2)ccc1[N+](=O)[O-] 13639,c1(CCn2cc(CC(C(N)=O)NC(=O)CCF)nn2)cc2c(O)ncnc2cn1 13640,c1(CC)nccnc1C(N1CCC(O)C1C(=O)NCC(C)(CO)OC)=O 13641,C(C(C)(C)C(=O)N1CCC(C(N)=O)CC1)OCC.C12(C)CCCN1C(=O)CO2 13642,c1(C(N(C(CNC(C2CN(C(C)=O)C2)=O)C)C2CC2)=O)ccc(C)c(Br)c1 13643,Cc1ccc(C#N)cc1C(N1CC2CC1CCC2NC(=O)C(F)(F)C(F)F)=O 13644,C1(NC(CC2C(C)CCO2)=O)CCN(C(c2cccc(C(C)(F)F)c2)=O)C(C)C1 13645,Cc1conc1C(=O)NCC1CC1CNC(c1ccc(-c2cccnc2)s1)=O 13646,c1(OCC)cc(Br)cc(CNC(c2ccc(C)cc2-n2cccc2)=O)c1N 13647,c1(C(N(C(C)CCNC(C2SC3C=CC2CC3)=O)C)=O)cc2ccc(Cl)cc2o1 13648,c1(C(C)C)cc(C(=O)NC2CCCCC2NC(=O)C(O)c2ccsc2)cc(O)n1 13649,c1(C(C)=O)ccccc1OC(CCNCC1CCCCN1C(=O)C(C)CCO)=O 13650,c1(SC)cccc(C(=O)NCCN(C(c2cnc(S)[nH]2)=O)C2CC2)c1 13651,c1(CC(C(=O)NCC2(F)CN(C(CNS(NC)(=O)=O)=O)C2)C)ccccc1Cl 13652,C(=O)(C(C)(C)C(N)=O)NCCC1C(C)CN(C(=O)COCc2cccnc2)C1 13653,c1(OC)ccc(C(CF)OC2CCCC(NC(c3nc(C)oc3C)=O)C2)cc1 13654,Cc1cc(C(=O)NC2CCCN(C(C3CCN(C)C3)=O)C2)cc([N+](=O)[O-])c1O 13655,c1(OC)ccc(CC(=O)NC2CC(C)(NC(=O)CCc3ccccn3)C2)cn1 13656,C(=O)(C1=CC2(CCN(C(=O)CCSCC)C2)C1)NCCSCC=C 13657,C1(CC#C)(C(=O)NCCOCCN(C(=O)C(F)CC2CC2)C)CCOC1 13658,C(=O)(C(C)(C)CC1CCOC1)N1C(CN(C)C(C2CCC(=O)C2)=O)CCC1 13659,n1(CC(C)NCCCC(C)(C)CO)cnc2c(cnn2C)c1=O 13660,N1(C(c2c(CC)c[nH]n2)=O)CCC2C(C(=O)NC(c3noc(C)n3)CC)C2C1 13661,CN1C(=O)C(F)CC1C(N1CCCC1(C)CNC(=O)C(C1CC1)N(C)C)=O 13662,CCCCCCCC(=O)N1CC(C)(NC(c2cccc(C3CCCOC3)c2)=O)C1 13663,C(=O)(C(C)CCCC)N1CC(CC(=O)NCC=CC)OCC1 13664,CCCC(O)(CCC)CC(=O)NC1CC(O)(CNC(C2CCC23CCC3)=O)C1 13665,N1(C(Cc2c(C)non2)=O)CC(NC(=O)CCC2CCCC2)CCC1C 13666,C=CC(F)(F)C(=O)NCC(O)CC(=O)NCC1CCOC1C 13667,c1(C(=O)NC(CNC(c2cnn(CC)c2Br)=O)C)ccc2[nH]c(=N)sc2c1 13668,C1(CNC(c2cn(C)cc2C(F)(F)F)=O)COCCN(C(C2(O)CC2(C)C)=O)C1 13669,c1(CN(C2CN(C(COCCC=C)=O)C2)C)ccc(C(=O)OC)cc1Br 13670,C1(CC(=O)N(C2CC2)CC2N(C(C(C)Cn3ccnc3)=O)CCC2)CC2(CCC2)C1 13671,N1(C(c2ncn(CC)c2)=O)CCOCC(NC(=O)CSc2nnnn2C)C1 13672,Cc1nc(C2CC2)oc1C(=O)NCC(O)CCNC(C1(C)CC(F)C1)=O 13673,C1(CC#C)(C(=O)NCC(c2cccc(Br)c2)C)CCCNC1 13674,N1(C(C(C)C2CC2)=O)CC(C(=O)NCc2ccnc(F)c2F)C2(CCC2)C1 13675,N1(CC(=O)NC2CCC=C2Br)CCc2nc(CSCc3cccnc3)cn2CC1 13676,c1(C(=O)NCC2(C(=O)NC(COC)C(C)C)CC(=C)C2)cnc(C)n1C 13677,Cc1cc(C)c(C(N2CCN(C(c3cc(O)ncn3)=O)CC2)=O)cc1N 13678,Cc1cc(C(=O)NCCC23CCC2CN(C(c2sccc2C#N)=O)C3)nc(C)c1 13679,C1(C2CCC2)(C(=O)NC2C(NC(c3ccc(OC)c(F)c3)=O)CCC2)CC1(F)F 13680,C1(CN(C(C(C=C)C)=O)C)CN(C(=O)Cc2csnn2)CC12CC2 13681,O=C1CCC(S(=O)(=O)NC(C2C(NC3CCC(C(=O)OC)CC3)C2)=O)CC1 13682,Cc1nnc2n1CC(CNC(=O)CCn1cncc(Br)c1=O)CC2 13683,C1(CC)CC(C(N2CC(NC(c3cc(C(F)F)cc(F)c3)=O)C2)=O)CC(=O)N1 13684,Cc1cc(C(=O)NCC2(O)CCCN(C(c3cc(C(F)F)cs3)=O)C2)cnc1O 13685,C12(C(=O)NCC(C)CNC(C3CCN(C(=O)OC(C)(C)C)C3)=O)CC(C1)C(C)O2 13686,C(c1nc(C)co1)=CC(=O)NCCC(=C)CNC(C1CC(CC)C1)=O 13687,c1(CC)cccc(F)c1C(N1CC2CC(NC(c3csnc3OC)=O)C2C1)=O 13688,C1(CC(=O)NCC2C(CNC(Cc3nnc(C)s3)=O)C2)CC(O)C1(C)C 13689,N1(C(c2c(Cl)cn(C)n2)=O)CCN(C(=O)CC2CCC(C(N)=O)O2)C2CCCC12 13690,C1(CNC(C2CC(C#C)(O)C2)=O)CN(C)CCN1C(C1CC(C)C1)=O 13691,C(C(CC(=O)NC1CCN(C(=O)Cc2ccn(C(F)F)n2)C1)C(F)(F)F)N(C)C 13692,Cc1cc(Cl)c(F)cc1C(N1CC(F)(C(=O)Nc2ncccc2O)C1)=O 13693,c1(N(C2CCN(C(C3CCC(C)CC3)=O)C2)C)ccnc(-c2nccs2)n1 13694,CCC(CC(=O)NCCCCC1CN(C(=O)C(c2ccccc2)O)C1)CC(C)C 13695,N1(C(C(CC)C#N)=O)CC(CN(C(=O)C(=Cc2cccnc2)F)C)C2(CC2)C1 13696,Cc1cc(C(N2CCC(CCNC(C3(C)CC3Br)=O)CC2)=O)nc(O)c1 13697,N1(C(c2ncc(C)s2)C(=O)NCCCSC)CCC(C(C)(F)F)CC1 13698,N1(C(C(C=C)CC)=O)CC2OCC(NC(=O)C(=O)NCC(F)(F)F)C2C1 13699,N1(C(COCCOC)=O)CCC2(C1)CN(C(=O)Cc1ccnn1CC)CC(C)O2 13700,O=C(CCCC1(NCc2c(Cl)cccc2Cl)CCC1)N=c1ccc2cc[nH]c2[nH]1 13701,c1(CC(N2CC(CC)N(C(=O)CC(C)C(C)C)CC2)=O)coc2cc(O)ccc12 13702,c1(OCC)cc(C(N2CCCN(C(=O)C)CC2)=O)cc(Cl)c1.C1(=O)CN1.C(C)(=O)N 13703,C1(C(=O)OC)CC2CNCC2N1C(=O)CC1CNC2COCC2O1 13704,Cc1cc(=NC(=O)C(=O)N2CC3CC2CCC3NC(c2cccc(F)c2)=O)[nH]o1 13705,CC1(C(N2CCC3(CCC3)C2)=O)CCN(S(=O)(=O)CCCCl)CC1 13706,C(C(C(=O)N(CCCCO)C(C)(C)C)n1cc(C)nn1)OC.n1(CCOC)ccnc1 13707,CN1CC(C(N2CCCCC2CN(C)C(c2cnco2)=O)=O)C(C(F)(F)F)C1 13708,C1(C(=O)NCC2CCN(C(C(C#C)(C)C)=O)C2)CCC(C#N)CC1 13709,CC(F)(F)C(F)C(=O)N1CCC(N(C(C2CCCCC2)=O)CC2CC2)C1 13710,C1(NC(CCCOCCC)=O)CC2CCC1N2C(=O)C(C)(C)OC 13711,CN1CCn2cc(C(N3CCCC4CN(C(C5(C)CC5)=O)CCC34)=O)nc2C1=O 13712,C(=O)(C(C)S(=O)(=O)C(C)C)NC(CCCNC(c1c(C)onc1Br)=O)C 13713,N1(C(C2(C)CC(C#N)C2)=O)CC2CC(NC(c3n[nH]c4c3COCC4)=O)CC2C1 13714,CC1CC(NC(c2ccsc2C(F)F)=O)CN(C(=O)CC2CC3(CC3)C2)C1 13715,N1(C(c2ncn(C)c2)=O)CCCCC(NC(C2OCC3CCCC23)=O)C1 13716,CCCCCCCCOCC(N1CCCC1CN(C(C1CCC(C)C1)=O)CC)=O 13717,C1(NC(c2c(OC)ccs2)=O)CC2CCC1CN(C(=O)CNC(C1CC1C)=O)C2 13718,c1(C(=O)Nc2c(OC(C)C)ccc(C#N)c2)ccc2c(c1)NCCC(=O)N2 13719,C1(C(=O)NC(c2ncc(-c3ccc(Br)cc3)o2)C)(C(C)C)CNC(=O)C1 13720,C(=O)(CCCCOC)NC(C1CCCC1)CNC(c1c(NC)scc1)=O 13721,C1(NC(c2ncc(Cl)cn2)=O)CC12CCN(C(c1ccc3cc[nH]c3c1)=O)CC2 13722,c1(CNC(=O)C(=O)NCC(C)C)ccnc(Oc2ccccc2)c1 13723,C(=O)(C(Cc1cnc[nH]1)NC(C1CCOCC1)=O)NCC(=C)Br 13724,c1(C(=O)Nc2c(F)ccc(NC(CC)=O)c2)c2c(nn1C)CCNC2 13725,c1(C(=O)NCCNC(C2C(C(N)=O)C2)=O)ccnc2ccc(O)cc12 13726,c1(CCNC(=O)NC2C(C(C)(C)C)CC2)ccc2c(c1)NCCC2 13727,C(=O)(C#CC1CCCCO1)NCC(c1ccccc1)CNC(C1(CC=C)CC1)=O 13728,c1(CNC(N2C(N3CCCC3)(CC)CCC2)=O)sccc1S(C)(=O)=O 13729,c1(C(=O)NC2CCN(Cc3ccc(C)[nH]3)CC2F)n[nH]c2c1CS(=O)(=O)C2 13730,N1(C(C(C)C(C)O)=O)CCCC2(CC(NC(=O)COC(F)F)C2)C1 13731,c1(CN(CC(C(CC)C)O)CC)cc(F)ccc1OC 13732,c1(NCC(CC)O)ccc(Br)c(S(=O)(=O)N(CC2CC2)CC2CC2)n1 13733,C(=O)(C#CC1(C)CCCO1)N(CCN(C(C1CC(C)(CC(C)(C)C)C1)=O)CC)CC 13734,C1(NC(C(C)SC)=O)CCCN(C(C2CCC(C)C2)=O)C1C 13735,C1(C(=O)NCC2(C(=O)NCC(CC(=O)OC)OC)CC23CCC3)CC2CCCC2C1 13736,C=CCCCCC(=O)NCC(CC1CC1)C(=O)NC(c1cn(C)nc1C)C 13737,C(C(CNC(C1CCOC1)=O)C(F)(F)F)NC(C1(CC=C)CC1)=O 13738,CCCCCC(C(=O)NC(C)C(=O)Nc1cc(C)cc(O)c1)C(C)C 13739,N1(C(c2n(CC)ncc2)C(=O)Nc2cccc(Cl)c2C)CCOCC12CCOC2 13740,C12(CN3CC(C)(COC)C3)CCC(C)(CC1)OC2(C)C 13741,C(=O)(CC1NC(=O)c2ccccc21)NC1C(C)CN(C(C2CCC(F)CC2)=O)C1 13742,c1(N2C(C3(NC(c4cc(C)n(C)n4)=O)CC3)CCC2)ncnc2c1SCCC2 13743,C1(C(=O)NCNCC2CC2C(CNS(CC)(=O)=O)=O)CCCN(CC(F)(F)F)C1 13744,c1(C(C)C(=O)NCC(C)N(C)C(c2cc(-c3ccco3)no2)=O)cccc(Cl)c1 13745,N1(C(C(CC)CC)=O)CCN(C(c2cnn(C(C)C)c2F)=O)C2CC12 13746,C1(NC(C(=O)NCC(F)F)=O)CCCC(NC(c2c(Cl)cncc2Cl)=O)CC1 13747,C1(C2CCCN(C(=O)C=CCF)C2)(NC(C2OCCN(S(C)(=O)=O)C2)=O)CC1 13748,C1(C(N(CC(CCC)O)C)=O)CCCN1NC(=O)c1c[nH]c2cccnc12 13749,C1(NC(c2cc(OC)c(F)cc2N)=O)CCN(S(=O)(=O)N(C)C)CC1 13750,Cc1cc(C(N2CCC(O)C(NC(c3ccc(C)n3C)=O)C2)=O)c(S(N)(=O)=O)s1 13751,N1(C(CC2CN(C(C)=O)C2)=O)CC(C#C)(C(=O)NCCC(O)CO)C1 13752,C1(CNC(c2cc(C)[nH]n2)=O)(NC(=O)CC2(O)COC(C)(C)C2)CCCCC1C 13753,c1(N2CCCC(CN(C)C)C2)nc2ccccc2nc1NCC1CCC1(F)F 13754,c1(N2CCCC(=C)C2)nc(=NCCC2CCCN2C)[nH]c2c1CC(C)CC2 13755,C=C=CCC(=O)NCC1CCC1NC(=O)Cc1cnn(C(C)C)c1 13756,c1(OC)cc(N2CCC(=C(C)CN(C)C)CC2)ncn1 13757,C1(CN2CCC(N(CCC)C(C3CC4CC4C3)=O)C2)CCCNC1=O 13758,Cc1c(Cl)ccnc1C(=O)NC1CCC(F)(CNC(=O)C=C2CCC2)C1 13759,c1(C(=O)NC2C(C)CN(C(=O)Cc3cnoc3)CC2)c(F)c(F)c(F)c(F)c1F 13760,N1(C(CC)CC)C(=O)NC(CCNC2CCCC(C)C2C)C1=O 13761,N1(C(C2(C)CC2c2ccccc2)=O)C2CCC1C(CNC(C1CCCS1)=O)C2 13762,C1(CNC(Cc2ccc(OC)c(Br)c2)=O)CCc2nccn2C1 13763,N1(C(c2ccc(NS(C)(=O)=O)cc2)=O)CC2CC1CCN2C(=O)CCS(C)=O 13764,C(N=c1nc2sccc2c(NCn2cncc2CC)[nH]1)C1CC(CCC)C1 13765,Cc1noc2nc(C(N3CCCC(O)(CNC(C4CC(CF)C4)=O)C3)=O)ccc12 13766,C=Cc1cc(C(N2CCC(NC(=O)CCSCCCC)C2CC)=O)cc(F)c1 13767,c1(CC(=O)NCC(CN(C)C(C2CCCCC2O)=O)(C)C)cccc(C2CC2)c1 13768,C#CCC(CC(=O)Nn1cnn(C)c1=S)NC(c1cnc(O)o1)=O 13769,c1(NC(C(CC)NC(=O)OC)=O)ccc2nonc2c1 13770,C1(CCNC(C=C(C)C(F)F)=O)(NC(=O)OC(C)(C)C)CC1(C)C 13771,C1(N(C(CCC=CC(C)C)=O)C)CCCC(NC(C2(C(N)=O)CC2)=O)C1 13772,c1(C(=O)NC(=O)CCC(CNC(=O)Cc2nnc(O)s2)OC)ccccc1C 13773,c1(C(=O)OCC(=O)NC(C)CCn2cncn2)ccc(I)cc1Br 13774,Cn1c(C(=O)NC2(C)CC(NC(c3ccc(N)c(CO)c3)=O)C2)cc2sccc12 13775,C1(CC(N2CCC(CNC(Cn3nnc(C)n3)=O)C2)=O)CCS(=O)(=O)C1 13776,C1(NC(C2(C=C)CCC2)=O)CCCC(NC(c2cccc(C(=O)OC)n2)=O)CC1 13777,CC1(CNC(C2CCC(=O)O2)=O)CCN(C(C2CCCN2N=O)=O)C1 13778,C1(C)(NC(CCSCC)=O)CCN(C(C2CCCC2(C)C)=O)CC1 13779,CC1CN(C(=O)Cc2cnns2)CCC1CNC(=O)C(C)SCc1ccccc1 13780,c1(C(C)CNC(C2CCCCC2)C(=O)OCC)ccc(Br)cc1.C(C)(C)(C)O 13781,N1(C(C(C)SC(F)(F)F)=O)CCC(C(C)CNC(c2scnc2C(F)(F)F)=O)C1 13782,C1(CNC(COCc2n(C)ccn2)=O)CN(C(=O)CC2(O)CCC2)CCC1(C)C 13783,Cc1nnc2n1CCC2(C)C(=O)NCC1C=CCN1C(c1ccsc1)=O 13784,C(CCSC)(C(=O)NCC1(C(C)(C)O)CN(C(c2scc(C)c2C)=O)C1)OC 13785,CCC(C)C(O)C(C)C(=O)N1CC(CC(N2CC(N(C)C)C2)=O)C2(CC2)C1 13786,CC1CCC(F)(C(=O)NCC(C)(C)OCC(=O)NCCCCCCC2CC2)CC1 13787,c1(CNc2cncc(CS(C)(=O)=O)c2)cc(F)c(N)c(F)c1 13788,C(=O)(C(CO)C(C)C)NC12CC(CNC(C=C(C)C(C)(C)C)=O)(C1)C2 13789,C(=O)(CCCCc1cnn[nH]1)NCCCC1N(C(C(C)n2ccnn2)=O)CCC1 13790,C(CN=c1[nH]c(=NCCC(C)F)c2sccc2[nH]1)c1c(C)noc1C 13791,CC1C2CCN1CC(NC(c1cnn(CCC(=O)O)c1)=O)C2 13792,N1(C(c2n(C)ncc2)=O)CCC2C(NC(C34CCCC3(C(N)=O)C4)=O)CC12 13793,N1(C(Cc2ccn(C)n2)=O)CC2CC(C(=O)Nc3ccccc3C(C)(F)F)C1C2 13794,N(C1CCCn2ncnc21)C(C(C)NC(C1CN(C2COC2)C1)=O)=O 13795,N1(C(CCN(C(C2C(C)C3CCC2C3)=O)C2CC2)=O)CCCC2CCCCC12 13796,C(CC1=CCN(C(c2nc3cnccc3s2)=O)CC1)NC(CCN(C)CC)=O 13797,Cc1nc(C(=O)NC(c2nccn2C)Cc2ccccc2Br)c(C)n1C 13798,C1(CC(=O)NC2CCCC2NC(=O)C(=O)NCC(F)F)CCCN1c1ncccn1 13799,c1(NC(N(C2CC(C)(C)OC2(C)C)C)=O)nc2ccc(I)cc2s1 13800,CN(CCCC(=O)N1CCOC(CCCNC(C2(C)COCCO2)=O)C1)N=O 13801,n1(C(CC)CC)ncc(C(=O)NC2CN(C(c3cc[nH]n3)=O)CC2F)c1C 13802,C1(CCNC(C2(C(=O)OCC)CC2)=O)CCN(C(=O)Cn2cccn2)C(C)C1 13803,CC(O)C(C)(C)C(=O)NC1CCCC(NC(c2cc(C(F)(F)F)cc(F)c2)=O)C1 13804,c1(C(=O)O)[nH]nnc1C.C(C)(C(=O)OCCOCCOCC)NC(CO)=O 13805,C1(C)CCC(=O)N1.C(CCOCCO)(C(=O)N(CC(F)(F)CO)C)SC 13806,c1(C(N(C2CC(C(N3CC4CCC3CC4)=O)C2)C)=O)cc(I)c(O)c(I)c1 13807,N1(C(CC2(OC)COC2)=O)CCC(C)(NC(=O)Cc2cccc(NS(C)(=O)=O)c2)C1 13808,N1(C(c2c(SC)ccs2)=O)CCC(CNC(c2ccc(=O)n(C)c2)=O)C1(C)C 13809,CCC(O)CC(=O)NCC(C)CNC(c1cncc(NC)n1)=O 13810,C(=O)(CCCCC(=O)NCC1(C(=O)NC2CN(C)CCN(C)C2)CC=CC1)OC 13811,Cc1cccc2cc(C(N3CC(NC(=O)CCF)C3)=O)oc12 13812,C(C(O)CC(F)(F)F)NC(C(C(C)C)NC(c1c(C)cc(C)o1)=O)=O 13813,Cc1[nH]c2ccc(Cl)cc2c1C(N1CCC(NC(=O)C(C)CC2CCCC2)C1)=O 13814,C1(C(N2C(C(C)NC(c3c(C)cc(C)nc3)=O)CCC2)=O)CC(C(C)(C)C)=NO1 13815,N1(CCC)CCCCC1C(=O)NCCC(C(C)C)NC(=O)Cc1cc(C)[nH]n1 13816,C1(C)(C(=O)NCC(CNC(c2c(C)cc(CC)o2)=O)(C)C)CCC(C)=C(C)C1 13817,c1(C(N(C2CCN(C(c3cc(CC)c(C)s3)=O)C2)CC)=O)ncnc2ccsc12 13818,c1(OC)cc(CCO)ccc1NC(c1cccc(CC#N)c1)=O 13819,c1(C(=O)NCC(CO)NC(c2ccn(C)c2)=O)cccc(S(C)(=O)=O)c1 13820,C1(CNC(C(C(C)C)SC)=O)(CNC(=O)C(C)O)CCC(F)(F)CC1 13821,CC1CCN(C(C2CC(O)C2)=O)CC1NC(C12CCOC(C)(C1)C2)=O 13822,CC12CC(C(=O)NCC3CC3NC(c3cc(CO)on3)=O)(CCO1)C2 13823,N1(C(C(C)NS(CC)(=O)=O)=O)CCC2(CCCC2NC(c2cnoc2)=O)CC1 13824,c1(NC(=O)Nc2c(C(C)(C)C)c[nH]c2)cc(Cl)nc(C(F)(F)F)n1 13825,N1(C(COCC(=C)C)=O)CCC(CNC(C2CCS(=O)(=O)C2)=O)C12CC2 13826,N1(C(C2(OC)CCC2)=O)CCC(C2(NC(=O)COc3ccc(Cl)c(F)c3)CC2)C1 13827,c1(CC)nc(C)c(CC(=O)NC2CC3(C2)CC(NC(C2CC2F)=O)C3)c(C)n1 13828,N1(C(C=C(COC)C)=O)CC(NC(=O)C(F)CC2CCCC2)C(C)(C)C1 13829,N1(C(c2cc(C)sn2)=O)CCC(O)(CCNC(C2(CO)CCOC2)=O)C1 13830,N(C(=NCC1CCN(c2ccc(F)cc2)C1)NC1CC1)CC1(S(C)=O)CC1 13831,C1(C(N2CC(C)C(NC(c3cncc(N)n3)=O)C2)=O)CCC2CC(C)CN2C1 13832,c1(CC(=O)NCCN(C(=O)CC2CCNC2=O)C)cc(Cl)sc1Cl 13833,N1(C(CC2CC(CC)C2)=O)CCCC(CCNC(C2CC(OC)C2)=O)CC1 13834,C(=O)(C(C)CS(C)(=O)=O)NCC=CCNC(C(C1CCC(C)CC1)CC)=O 13835,C1(NC(N2CC3C(CC#N)CC(C3)C2)=O)CCCC12CCOCC2 13836,C#Cc1cc(NC(C2CC(=O)C2C(F)(F)F)=O)ccc1C 13837,N1(C(C2C(OC)CCC2)=O)CCC(C)(C(=O)NCC2(C)CC(C)=NO2)C1 13838,C1(NC(c2cccc(OCC)c2)=O)CC(F)CN(C(=O)C=CCOCCOC)C1 13839,CCCCC(C(=O)NCC(C1CCCCC1)NC(=O)C(C)(C)C1CC1)C(C)C 13840,N1(CC(C)N2CCC2)CCCC(C)C1.C(C(=O)O)O 13841,N1(CCC(=O)NC(C2CCCN2C(c2nncs2)=O)(C)C)CCP(C)(=O)CC1 13842,c1(CCOC)nc(CNC(c2nnnn2C2CC2)C(C2CCOCC2)C)cs1 13843,N1(CCS(CC)(=O)=O)CCC(c2ncc(C(=O)O)s2)C1 13844,C1(C2(O)CCN(C)CC2)(C(N(CCCCN(C)C(c2ccoc2)=O)C)=O)CC1 13845,C(C)(C)(C(O)C(F)F)N(C(=O)Nc1c(C)nn(-c2ccc(F)cc2)c1)C1CC1 13846,Cc1nc2[nH][nH]cc-2c(=NC2CCCC3CN(C(C45CCC(C4)OC5)=O)CC23)n1 13847,c1(NC(C2C(Nc3ncc(C)c(C)n3)CCCC2)=O)noc2cc(Cl)ccc12 13848,C123CCC(CC1)(CO2)CNC3=O.C1(CNC(CC(C)OC)=O)CCCC2CC12 13849,Cn1ccc2cc(C(N3CCC(C4CC4)(CNC(=O)C(C)(C)C)C3)=O)cnc12 13850,N1(C(=O)OC(C)(C)C)CCC(F)(NCC2CC3CC2CO3)C1 13851,c1(CCOC)noc(CN(C(=O)C(=O)NC(c2nc(C)no2)C(C)C)C)n1 13852,c1(-c2nc(CCC(C)C)nn2CCn2ccnc2)cncc2c(Cl)cccc12 13853,c1(C(N2CCC(CNC(C(C)=C3CC3)=O)CC2C)=O)cc2cc(C)c(C)cc2o1 13854,N#CC12CCC(CN(C=O)CCc3ncccn3)(CC1)CC2 13855,c1(-n2ccc(C)n2)cccc(C(=O)NCCC2(O)CCCC2)c1 13856,C1(NC(CC(CC)OC)=O)CN(C(c2nccc(C(F)(F)F)n2)=O)C(C)(C)C1 13857,N1(C(c2nncc(C)c2)=O)CCC(C)C(NC(c2ccoc2)=O)C1 13858,CC1C(C(=O)NCc2ccnn2C)CCN1C(=O)CCC1CCCCO1 13859,N1(C(CC2C(NC(C(F)=CCC)=O)CC2O)=O)CCCC2C(O)CC12 13860,Cc1nn(-c2cccc(Cl)c2)c(C)c1CN(C1(CCO)CCCC1)C 13861,c1(C(N(CCNC(C2(COC)CC2)=O)CCOC)=O)c(Cl)ccc(C)c1O 13862,N1(C(c2n(C(CC)C)ncc2)=O)CC(NC(c2cnc(O)c(F)c2)=O)C2(CC2)C1 13863,N1(C(C(C)N(C)C)=O)CCC(C(=O)N(C(C(N)=O)C2CC2)CC)=C(F)C1 13864,c1(OC)cc(C(=O)N(C)CCN(C(=O)C(F)=C2CCC2)C)[nH]n1 13865,c1(C(N2CC3C(C(=O)NCCC#N)(C3)C2)=O)cc2c(F)cc(F)cc2[nH]1 13866,C(=O)(CC1=NN(C)C(=O)C1)NCC(C)N(C(=O)C(F)CC1CCOC1)C 13867,C(=O)(CC(F)(F)C(C)C)N1CCCC(NC(C(CCCOC)C)=O)C1C 13868,N1(C(c2cnc3[nH]nnc3c2)=O)CC(C2CCCN(C(C3CCOC3)=O)C2)C1 13869,Cc1noc2nc(C(=O)NCCCCNC(=O)CCCNC(N)=O)ccc12 13870,C(=O)(C(F)CCC(C)C)N(C(CNC(Cc1c(C)occ1)=O)C)C 13871,c1(C(=O)NCC(C)N(C(=O)CC(C)CF)CC)ccc(CO)c(F)c1 13872,c1(C(=O)NCCN(C(C(C(C)C)SC)=O)C2CC2)ccc2c(c1)OCCC2 13873,N1(c2nccc(OC)n2)CCN(C(c2cncc(-c3cccc(Br)c3)c2)=O)CC1C 13874,C1(NC(C(C#C)(C)C)=O)CN(C(C2CC3(CC3)CO2)=O)CC1C=C 13875,C1(C(=O)NCCSCC)CC2(CC(NC(=O)CCC(=O)NC)C2)C1 13876,c12ccc(cc1)S(=O)(=O)N2.c1(CC)nc(OC)ccc1-c1ccc(N(C)C)nc1 13877,C1(C(=O)NC(CCNC(C(C)(CO)OC)=O)C)CCC2(CC1)CC2(F)F 13878,C(=O)(N=c1cc[nH]cc1P(C)(C)=O)Nc1c2cccc(C)c2c(F)cc1 13879,C(CC1=CCCCC1)NC(c1c(CNC(C2(Cl)C(C(C)=O)C2)=O)ccs1)=O 13880,c1(C(=O)NCC2C(C)CCN2C(=O)CC2OCCCO2)cc(Cl)c(F)cc1Cl 13881,C1(NC(CCc2c(C)nn(C)c2)=O)CCN(C(=O)C(C)(C)n2ccnn2)CC1C 13882,C1(C)(C(=O)NCCCN(C)C(C2(C)CC=CCO2)=O)Oc2ccccc2NC1=O 13883,CC1CCN(C(C2(CNC(c3ccc(F)cc3)=O)CC2)=O)CC1CN(C)C 13884,Cc1ccc(CNC(C2(C(=O)NC(C)CCC3CC3)CCC2)=O)c(O)c1 13885,Cc1sncc1C(=O)NC(C)C(C1CCCCC1)NC(c1csc(Cl)n1)=O 13886,c1(C(=O)NCC(CNC(CCc2cc(C)on2)=O)C)cn(C)nc1C(F)(F)F 13887,C1(C)(NC(c2ccccc2)C(=O)Nc2nccc(C#N)n2)CCN(C(C)C)CC1 13888,C1(C)(C(N(CC(CNC(C2C(OC)CCC2)=O)C)C)=O)CCC(=O)NC1 13889,N1(C(c2c(=N)[nH]cnc2)=O)CC2CCN(C(=O)COCCF)CC12 13890,N1(C(C)=O)CC=CC(C(=O)O)C1.c12ccc(o1)C(=O)NCC2=O 13891,N1(C(C2(COC)N(C(C)=O)CCC2)=O)CCC(C)C(COc2ccccc2)C1 13892,C(=O)(CC1=NN(C)C(=O)C1)N1CCC(n2cc(CC=C)nn2)C(O)C1 13893,c1(C(N2CCC(C)C2CNC(=O)Cc2csc(S)n2)=O)cc(O)ccc1Cl 13894,c1(C2C(C)(C)C(NCC3CCCCC3)C2)ccc(S(=O)(=O)NC)cc1 13895,c1(C(=O)NCC(CC=C)NC(C23CC(COC)(CO2)C3)=O)cnc(OC)cc1C 13896,C12CN(CCO1)C(=O)C(=O)NC2.C(C(O)C(=O)NCCOCCOCCO)SC 13897,C1(CNC(C2CC(SC)C2)=O)C=CCN1C(c1ncn(C)n1)=O 13898,N1(C(C2C(C)C2C)=O)CCCC12CCC(NC(c1n[nH]c3c1CSCC3)=O)CC2 13899,c1(-c2nc(C3CCC(CO)C3)on2)cc(Br)ncc1Br 13900,N(C(=NCC(C)OC)NCC1CCCCC1)Cc1ccc(CC)cc1 13901,c1(C(N(CC(C)NC(C2CC(C#C)(O)C2)=O)CC)=O)cc(Cl)c(C)cc1[N+](=O)[O-] 13902,CC1(C)CC(CC(=O)NCC(C)(CO)NC(c2cccnn2)=O)C1 13903,c1(C(N2C(C(N(CC)CC)=O)CCC2)=O)cc(F)cc2c1CCNC2 13904,C1(C(N(CCCC)CCCC)=O)CCN(C(=O)c2ccc(C(N)=O)o2)O1 13905,Cc1cnc(C=CC(N2CCC(C3CCCCN3C(=O)C(F)=C(C)C)CC2)=O)[nH]1 13906,N1(C(C=CC(=O)NC2CC2)=O)CCCCCC(NC(C2(C3CCC3)CC2)=O)C1 13907,C#CCCCC(C)C(=O)N(C)CCOCCNC(=O)CCc1cocn1 13908,C(c1ccccn1)=C(C(=O)N(CCOC)CCNC(C1CCOC1C)=O)C 13909,Cc1cc(C(N2CCN(C(=O)CC3=CCCC3)C(C)C2)=O)cc(F)c1C 13910,O=C1CC2C(C(=O)NCc3csc(CNC(=O)Cn4nccn4)n3)C2C1 13911,C(=O)(C(C)C(C)(C)C)N1CC(OCC(=O)NC(COC)CO)C1 13912,N1(c2c(C)cc(OC)cc2O)CC2(CCC(NC(=O)CNC(N)=O)CC2)C1 13913,CC1CC(C)(C(=O)NC2CCC2NC(c2cc(F)n(C)n2)=O)CCO1 13914,n1(CC(=O)NC(CC)CNC(c2cc(C(=O)NC)cs2)=O)nc(C)cc1C(F)F 13915,Cc1cc(=NCC2CN(C(c3cc(C(C)(C)C)on3)=O)CC2(C)C)c(C#N)c[nH]1 13916,c1(OCC)cncc(C(=O)N(CCCCCNC(c2cncc(OC)n2)=O)C)c1 13917,CCC(C)CCCC(=O)NC1CCCC1NC(c1c[nH]c(=N)o1)=O 13918,N1(C(CCC#C)=O)CC(NC(=O)CCc2cccnc2C)CC12CCCCC2 13919,C(CC(CC)C(=O)NC1CCCCC1C(=O)NC(C)CCOC)=CC 13920,c1(C(=O)NCC(CN(C(c2ncc(OC)c(C)c2)=O)C)O)cc([N+](=O)[O-])nn1C 13921,C1(NC(C(c2cn(C)nc2)(F)F)=O)CCN(C(=O)CCOCC(F)(F)F)C1(C)C 13922,c1(CC)nc(C)c(C(=O)NCC(C(C)C)NC(=O)CCn2nc(C)cc2C)o1 13923,CN1CCC(C(N2CCC2C(N2CCCC(CCO)C2)=O)=O)CC1=O 13924,CCC(C)C(O)C(C)C(=O)N(CCCO)C1CC1.C1CC(=O)N1CC1CC1 13925,c1(C(=O)NCC2CC(NC(C3CCS(=O)(=O)C3)=O)C2)cc2c(nn1)CCC2 13926,N1(C(C2CCC(N=[N+]=[N-])CC2)=O)CCC2(CC1)CN(C(C1CCCS1)=O)CCO2 13927,Nc1nccn2ncc(C(N3CCC(NC(C4CCC(=O)NC4)=O)C3)=O)c12 13928,C1(C(=O)OCCOCC(C)(F)F)CCCCN1O 13929,CC1(C)CC(C(=O)NCC2CC=CCC2)CCN1C(c1nnc(O)nc1O)=O 13930,CC1CCCCC1(CNC(C1(C(F)F)CCC1)=O)NC(c1cc([N+](=O)[O-])n[nH]1)=O 13931,c1(C(=O)NC2CCC2NC(=O)C(O)c2cnc[nH]2)ccc2c(c1)CCCS2(=O)=O 13932,C1(CNC(c2csc(C)c2C)=O)CN(C(=O)CCC#N)CCC1C 13933,C1(C(N(CCN(C(C)C)C(c2ccc(CCO)cc2)=O)C)=O)C2CC2C2CC12 13934,C1(CNC(c2ccn(CCN(C)C)n2)=O)COC(C)(C)CN1C(c1cn[nH]c1)=O 13935,c1(-c2c(CC)nsc2)nc(-c2ccncc2)nn1-c1cnn(C)c1 13936,C(=O)(C1=C(C(C)=O)N(CCOC)C(=S)NC1c1ccc(OC)o1)OCC 13937,N1(C(Cc2c(C)ccs2)=O)CCC(C)(NC(=O)Cc2nnn(C(C)(C)C)n2)C1 13938,c1(C(N2CCCC(NC(c3ccc(CF)cc3)=O)CC2)=O)cn2ccnc2cn1 13939,c1(CNC(C2CCN(C(CCCCOCCC=C)=O)C2)=O)ccc2cc[nH]c2c1 13940,C#CCCC(C(=O)NCCC1CC=CCC1)NC(=O)CCc1cncs1 13941,CC(=NO)C1CC(C(=O)NCCCC2CCCN2C(=O)CC#N)C1(C)C 13942,c1(C(N(CC)Cc2ncc[nH]2)=O)occc1CNC(=O)CC1CCSC1 13943,C(=O)(C(CSC(=O)NC)N(C)C)NCCN(C(c1cn(C(F)(F)F)cn1)=O)CC 13944,C(N1CCC(c2ccc(F)cc2)CC1)c1cc(=O)n(C)n1CC(=O)CC#N 13945,c1(C(=O)NCC2(C)CCC(NC(C=COCC)=O)C2)ccc(O)nc1Cl 13946,Cn1c(C(=O)NCC(C2CCOC2)NC(c2cnc3n2CCS3)=O)cccc1=O 13947,CCCCC(C)CCC(=O)N1CCC(F)C(NC(c2ncoc2C(C)C)=O)C1 13948,c1(C(=O)NC(c2cnn(C)c2)C(=O)NC(c2ccccc2)C)n[nH]c2c1CCC2 13949,C1(CNC(C=Cc2n(CC)ncc2)=O)CCN(C(=O)C(C)(C)SC)CC1C 13950,Cc1ncncc1C(N1CCC(CCC(=O)NC2CCNC2=O)CC1)=O 13951,C(=O)(CC(C)C(C)(C)NC(C1CNC(=O)N1)=O)N(CC(C(C)C)OC)C 13952,CC(C(=O)NCC(C)(C)CNC(C1(c2ncco2)CC1)=O)C(C)(C)C 13953,c1(C(N2CCCC(CC)(CO)C2)C(=O)Nc2ccc(F)cc2)ccc(OC)cc1Br 13954,c1(N(C)C)ccc(Br)cc1C(N1CCC(C)(CNC(C2CC2(C)C)=O)C1)=O 13955,C1(C(=O)NC2CCN(C(c3cnc(C(C)C)s3)=O)C2)CCC2(CC1)CC2 13956,Cc1cnc(C)c(C(N2CC(N(C(=O)CC(C)C3CC3)C)C3(CC3)C2)=O)c1 13957,N1(C(c2c(C)non2)=O)CCCC(C)(C(=O)Nc2ccnnc2O)C1 13958,CC1(NC(=O)CC23CCC2CN(C(=O)C2=CCCCO2)C3)CCC(O)CC1 13959,CCCC(O)C(=O)NC(C(=O)N1CCCCC1CN(C)C)C(C)C 13960,c1(C(=O)OC)[nH]c(=NCC(C)CNC(=O)C(O)C(C)c2ccccc2F)sc1C 13961,CCCCCCC(C)C(=O)NC1CC(C(=O)NCc2nnn(C)n2)=CC1O 13962,Cc1c[nH]nc1C1(C(=O)NCC(C(C)C)NC(c2cnn(C)c2)=O)CC1 13963,N12CC3CCCC3(C1)C2=O.n1(CC(=O)CCN(C(C)=O)C)nc(C)c(Br)c1C 13964,CC1(C)C(C(=O)NCC(F)CO)CCN1C(=O)CSC1CC1 13965,c1(C(=O)NC2(C(=O)NCC(C)Cn3cccn3)CC2C)cc([N+](=O)[O-])n[nH]1 13966,C1(C(=O)NCC2CCN(CC)C2)CSCCN1C(=O)CSC(C)(C)C 13967,N1(C(C(C)C(C)(C)C)=O)CCC2(CCCCN(C(=O)Cc3ccsc3)C2)C1 13968,c1(N2CCCC(C)(C)CC2)ccc(S(=O)(=O)N2CCOC3(CCSC3)C2)cc1Cl 13969,c1(C(=O)NC2C(O)CCN(C(CCCCC#C)=O)C2)cc(Cl)cc(Cl)c1O 13970,n1(CC)nc(C(C)C)cc1NC(N1CC(c2ccc(C(=O)O)nc2)(O)C1)=O 13971,c1(C(=O)NC2CC(F)(CNC(C(CC)C(C)C)=O)C2)c(F)cc(Cl)cc1F 13972,C1(C(N(C)CC2CCN(C)C2)=O)CC2(CCC2)CN1C(c1ccc(C#N)s1)=O 13973,CCC(C)CCC(=O)NCc1nc(C)c(C(=O)NCC2(CC)CCCC2)o1 13974,C(=O)(C1=NOC2(CCN(c3nccc(Br)n3)C2)C1)Nc1cc(C)c(C)c(C)c1 13975,C1(C(=O)NCC(C(C)C)NC(c2csc(C(F)F)n2)=O)CC(=O)N(C)C1 13976,c1(C(=O)OC)ccc2sccc2c1.N12CCOC(C1)C2C(C)C 13977,N1(C(CCc2ccc(C)o2)=O)CCC(F)CC1C(N1CC(O)(CO)C1)=O 13978,C(CC1=CCCCC1)NC(C1C=CCN(C(c2ccsc2Cl)=O)C1)=O 13979,C(=O)(C(C)(C)CF)N(C1CCN(C(C2CCNC2=O)=O)CC1)C 13980,c1(C(N2CC(C(C)NC(CSc3n(C)nnn3)=O)C2)=O)ccc(N)cc1O 13981,c1(C(N2C(C(N3CC(N(C(CC)=O)C)C3)=O)CCC2)=O)cc(C)c(Cl)cc1F 13982,Cn1c(CNCc2ccc(N3CC=CC3)cc2)nnc1-c1ccccc1 13983,c1(NC2CN(C(C)=O)C2)[nH]c(=NC(C)c2cnc[nH]2)nc2sccc12 13984,N1(C(=O)Cn2cnnc2)CC2CC(N=c3ccnc(CO)[nH]3)CC1C2 13985,C(=O)(CC(C1CCC1)NC(C1CCN(C2CCOCC2)C1)=O)OCC 13986,N1(C(CC(CC)c2ccc(C)cc2)=O)CCC2(CC1)CN(C(=O)CCC(C)=O)C2 13987,C(c1ccc(Cl)cc1Cl)=CC(=O)N(C1CCCN(C(C)=O)C1)C 13988,C(=O)(C(CCC1CC1)NC(=O)C1=CCCC1)NC(c1ccc(O)nc1)C 13989,C1(C2(NC(=O)CCCCN(C(=O)CCC(=O)NC3CC3)C)CC2)(OC)CCC1 13990,C1(C(N2CC(CN(C(C(CC)NC(C)=O)=O)C)C2)=O)CC2(CCC2O)C1 13991,C123CCC(CC1)N2C(=O)N3.N12CCC(CC1)NC(C)C2=O.C(C)(C)(C)OC(C)=O 13992,S(=O)(=O)(CCC(=O)NCC1COCCN1C(c1ncnn1C(C)C)=O)NC 13993,N1(C(CCSCC)=O)CCC(NC(c2ccc3cc(C)cn3c2)=O)C2(CCC2)C1 13994,N1(C(CCCCSC)=O)C2CCC1C(C(=O)NOCC(C)(C)C)C2 13995,c1(C(=O)NCc2c(C(=O)NC3CCC(CO)C3)scc2)cccc2cc[nH]c12 13996,Cc1c(Cl)cc(C(=O)NCC(C)NC(=O)C(N2CCCC(C)C2)=O)cc1Br 13997,c1(C(N2CCN(C(c3nc(CC)oc3)=O)CC2CF)=O)c(C)cc(Br)cc1C 13998,c1(CC)cc(C(=O)NC2CC(C(=O)NC3C=CCC3)C2)ccn1 13999,c1(C(=O)NCC23CC(NC(CN(CCC)C)=O)(C2)C3)ccc2cccnc2c1 14000,C1(C(N(CC(CC)NC(C=C(CCC)C)=O)C)=O)(CC)CCNC1=O 14001,N1(C(Cc2n[nH]c(=NC)s2)=O)CCCC12CCCN(C(c1cnncc1O)=O)C2 14002,c1(C(=O)NCC(CNC(C2C(OC)CC2)=O)(C)C)cccc(SC)c1[N+](=O)[O-] 14003,C(CCCCN(C(=O)CC(C)n1cc(Br)cn1)C)NC(C=C(C)C1CC1)=O 14004,n1(CCC)cc(Cl)c(C(=O)NC(C)CN(C(c2cccc(F)c2)=O)CC)n1 14005,c1(OC)cc(C)c(C(=O)NCC2CCC3(CN(C(=O)CC(C)SC)C3)O2)c(C)c1 14006,C1(C)(NC(CNC(=O)OCC)=O)CCCN(C(c2ccc(N)cc2F)=O)C1 14007,C1(N(C(c2cc(CC)on2)=O)C)CCCC(N(C(=O)CCCN2CCCC2)C)C1 14008,CCC(CC(=O)NCC(C)CN(C(=O)C(c1cccn1C)=O)C)C(C)(C)C 14009,N1(C(CCC(CCCC)C)=O)CC=C(C(C)(C)C(=O)N2CCCC2CCCO)C1 14010,C1=CC(=O)Nc2ccc1cc2.C1(CN)CCC(SC)C1.N(C(=O)N)(CC)CC 14011,c1(CC(=O)N(C(C)CCNC(=O)C(N2CCCCCC2)C)C)cccc(F)c1O 14012,C1(C(=O)NCCOCC(=C)C)CCCC(NC(c2ccc(CC)nc2)=O)C1 14013,N1(C(C(CCC2CC2)NC(c2c(CC=C)cccc2)=O)=O)CC(O)CCC1C 14014,c1(OCC)ccccc1CNC1CCCN1C(c1ccc(C)cn1)=O 14015,N1(C(C(CC=CC)C)=O)C(C(N2CCCC2C(O)CC)=O)CCC12CC2 14016,C1(CNC(C2CC(=C)C2)=O)CC(F)CN(C(=O)C(c2cccn2C)=O)C1 14017,Cc1cccc(C(=O)NCCC23CCC2CN(C(c2nocc2Br)=O)C3)c1O 14018,c1(CC)coc2cc(N)c(-c3cn[nH]c3)cc12.c12cccc(Cl)c1CNC2=O 14019,CC1=C(C(=O)Nc2ccccc2Cl)C(c2sccc2N)NC(=O)N1CC(C)C 14020,c1(C(=O)NC2CC(NC(=O)COCCOCCO)C2)ccc(F)c(O)c1F 14021,C(=O)(CCN=c1cc(NCC2CC(C3CC3)C2)nc[nH]1)N(C)C 14022,c1(SCC(=O)NCC2(F)CC(NC(C3C4CC4C4CC34)=O)C2)cccc[n+]1[O-] 14023,N1(C(C(C=CC)O)=O)CCC2CC12C(=O)NCCCN1CCCC1=O 14024,N1(C(C(c2cccs2)SC)=O)CCN2CCN(C)CC2C1 14025,C1(C(=O)N(CC#CCN(C(C(CC)C)=O)C)CC)(C(N2CCCC2)=O)CCOCC1 14026,N1(CC(=O)NC(CNC(CC=C)=O)C(C)C)C(=O)NC(C)(C2CC2)C1=O 14027,c1(CCCC(=O)NC2C(NCc3cnc(C)[nH]3)CCC2)ccc(Br)cc1 14028,c1(C(=O)NC(C2CCN(C(=O)Cc3cncs3)C2)C)cc2cnn(C)c2s1 14029,c1(OC)ccc(S(=O)(=O)N2CCCC(C)(C(=O)Nc3c[nH]nc3C#N)C2)cc1Br 14030,C(=O)(CCCC(F)(F)F)NCCCN1CCC(NC(C(NOC)=O)=O)C1 14031,C1(NC(CNC(=O)OC)=O)(CNC(c2cnc[nH]2)=O)CCCCCC1 14032,c1(OC)ccc(CN2CCCC(C(=O)N(C)CC3CCCCC3)CC2)c(Cl)n1 14033,C(C(C(=O)NC1CCOCC1)N(C1CCCCC1O)C)(C1CCC1)OC 14034,CCCC(C)(CC)C(=O)NC1CC(CCNC(=O)C(C)(CC)CC)C1 14035,C1(NC(C(CC)N(CC)CC)=O)C2CN(C(c3cccnn3)=O)CC12 14036,N1(C(COCCC#C)=O)CCCC(n2cc(CNC(c3cnn(C)c3)=O)nn2)C1 14037,CC1(NC(=O)CC2(C)CCOC2)CCC2(CC1)CC2.C12CCCCN(C1)C(=O)CC2 14038,Cc1cc(CNC(C23CC(NC(=O)CCc4cccnc4)(C2)C3)=O)n(C)n1 14039,CCCCC(O)C(C)C(=O)NC1(CNC(=O)Cn2ccccc2=O)CCC1 14040,c1(CC(=O)NC(C2(c3cn(C(C)C)nn3)CCC2)=O)cccc(C(F)(F)F)c1F 14041,c1(OC)ccc2c(c1)CCC2C(=O)N1CCC(F)(F)C12COC2 14042,c1(C(=O)NCC(C)NC(=O)C(=O)N(C)C)ccc(NC(=O)Cn2cnnc2O)cc1 14043,c1(C(c2n(CCOCC)nnn2)NCCC2CC=CC2)cc(C)nn1C 14044,c1(C(N2CC(C(C)NC(C3C(OC)CCC3)=O)C2)=O)ccc2nc(O)[nH]c2c1 14045,N1(C(CSCC=C)=O)CC(NC(c2cnoc2-c2ccc(Cl)s2)=O)CC1(C)CC 14046,Cc1c(C(=O)NCC2(C)CCCN2C(=O)C2=COCCC2)nn2c1OCCC2 14047,C1(C(=O)NC(c2ccccc2)CNC(=O)C=C2CCSCC2)CCCC(=O)N1 14048,c1(OC)c(F)ccc(-c2ccc(C(=O)NC(C)(CO)CO)cc2F)c1F 14049,c1(-c2nc(C(C)OC)nn2-c2cccc(C(=O)O)c2)onc2cc(C)ccc12 14050,c1(NC(c2n(CCCC(=O)OCC)nnn2)(C)CCBr)ccc2c(c1)CCCS2 14051,c1(CC(=O)NCC2CN(C(CNC(CC)=O)=O)C2)ccc(OC)cc1C 14052,c1(C(=O)NC2C3CCN(C(c4cnc(COC)s4)=O)C32)ccc(S(C)=O)cc1 14053,C12C3CC4C1C4C3C(=O)N2.C(CCCC(=O)N1CCCC(COCC)C1)OC 14054,Cc1nc(C(=O)NC2CCCC2CNC(c2ncn(C(C)(C)C)n2)=O)c(C)o1 14055,c1(C(N2CC(O)(C(C)SC3CCNC3=O)C2)=O)ccccc1N(C)C.C1C(=O)N1 14056,C(C(C(=O)NC(CNC(C)=O)C1CCC1)C(F)(F)F)OC 14057,c1(OC)ncc(OC(CC(C2CC2)NC(=O)N(C)C)c2nnnn2C2(C)CC2)cn1 14058,C(CC(O)CN=c1[nH]c2c(c(=NCc3c(C)n[nH]c3C)[nH]1)CCCC2)OCC 14059,N1(C(C(C)SC)=O)CC2CCN(C(C3COC4(C)CC3C4)=O)CC2C1 14060,CCCCC(C(=O)NC1CC2(C1)CN(C(c1cc(CC)[nH]n1)=O)C2)NC(N)=O 14061,C(=O)(CCCCCCC=C)NC(CC#C)C(=O)N1CCOC(CO)C1 14062,C1(NC(c2ccc(C#C)o2)=O)(CO)CCCN(C(=O)CCCc2ccccn2)C1 14063,c1(C(=O)NCC2(F)CCCN(C(C3C(C)(C)C3)=O)C2)ccc2c(c1)C(=O)NC2=O 14064,c1(C(N2CC(NC(C3C(C)C3c3ccccc3)=O)C2)=O)nccnc1Cl 14065,C1(CNC(C2(C)CCCS2)=O)CCC(F)(CNC(=O)CN2CCOCC2)C1 14066,N1(C(C(CC=C)OC)=O)CCCC(O)(CCNC(C2(O)CCCCCC2)=O)C1 14067,C(=O)(C(C)(C)C(N)=O)NCCCCCn1cc(-c2c(OC)nccc2)nn1 14068,C1(CC)(NC(c2ccc(Cl)c(OC)c2)=O)CCCN(C(=O)CCc2cn[nH]c2)C1 14069,CC1CN(C(=O)CCCCCN(C)C)C(C)CN1C(c1coc(S(C)(=O)=O)c1)=O 14070,c1(SC)cccc(C(=O)N(CCCNC(C2C3CN(C)CC23)=O)C)c1 14071,c1(C(=O)NC(C2CCCN2C(=O)CN=S(C)(C)=O)(C)C)ncc2c(F)cccn12 14072,CC(C)C(C(=O)NC1CCC1NC(c1cccnc1Cl)=O)c1ccn(C)n1 14073,C1(NC(Cc2c(CC)cccc2)=O)CN(C(=O)CNc2ccccn2)CC12CC2 14074,C12(NC(C34CCCCC3C4)=O)CCC(C(=O)NCc3ccccc3Cl)(CC1)C2 14075,C1(NC(c2c(CC)noc2)=O)CN(C(c2cccc(N)n2)=O)CC(C)(C)C1 14076,C1(C2(O)CN(C(c3cccc(OC)c3)=O)C2)(CNC(C(COCC)C)=O)CC1 14077,C(=O)(CCCCCCNC(=O)C=Cc1cnccn1)N1C(CN(C)C)CCCC1 14078,CCCCC(C)(F)C(=O)N1CC2(CCN(C(c3cocc3Br)=O)C2)C1 14079,c12ccccc1-c1ccc(nc1)N1CCN(CC1)C2.C1(C(N(C)C)=O)CCCS1 14080,C1(C(C)C)CN(C(c2cn(CCC#N)cn2)=O)CCN1C(c1ccc(Cl)nc1)=O 14081,c1(C(=O)NCCC(CNC(c2ccc(Br)s2)=O)OC)cccc(C)n1 14082,N1(C(Cc2scc(C)n2)=O)CCCCC2(CCCCC2)C1 14083,C1(CNC(C2C(CC)C2)=O)CN(C(c2cc(C(=O)C(C)C)c[nH]2)=O)CCC1(F)F 14084,C12(C(=O)NCCCCNC(c3cn(C)nc3Cl)=O)CCC(CC1)C(C)(C)O2 14085,c1(CC(C)C)ccc(C=CC(=O)NCC2(NC(C3C(C)C3C)=O)CCOC2)cc1 14086,CC1CC(NC(=O)C(c2ccccc2)N(C)C)CN(C(=O)CC2(F)CCC2)C1 14087,Cc1c(NCCn2ncc(Br)c2C)nc[nH]c1=NCCc1ncccn1 14088,N1(C(C2CC(C)OC2=O)=O)CCC(C)(NC(=O)CCc2nncn2C)CC1 14089,C(CC(O)C(F)(F)F)NC(C1N(C(c2ccn(C)c2)=O)C(C)C1)=O 14090,c1(C(N2CCC(N)(CC(=O)OC)C2)=O)cc(Br)c(O)nc1C 14091,N1(C(c2cc(CC)c(C)s2)=O)CC(C)CCC1CNC(=O)COC(F)(F)F 14092,c1(OCCNC(=O)CC23CCCC2C3)ccc(C(=O)NC(CC)C(=O)NC)cn1 14093,N1(C(c2n[nH]c(CC)c2C)=O)CCCCC(C(=O)NCC(c2cnn(C)c2)C)C1 14094,c1(CNC(c2c(C)cc(CO)o2)=O)n[nH]c2c1CN(C(=O)CC(=O)N(C)C)CC2 14095,C1(CNC(C(C)(C)F)=O)CCN(C(=O)CC2CCCC(C3CC3)O2)CC1 14096,N1(C(C(C(C)O)(F)F)=O)CC2(C1)CN(C(=O)CC(=O)NC1CC1)CCO2 14097,c1(C(C(=O)NCC(C)N(C)C(c2cnccn2)=O)(C)F)ccccc1F 14098,CS(=O)CCC(O)C(=O)NC1CC(C)(NC(c2cncc(F)c2Cl)=O)C1 14099,C1(C2(O)CN(C(C3CCCC(C(N)=O)C3)=O)C2)(CNC(C(C)(C)CO)=O)CC1 14100,C(=O)(C(C)(C)C(O)C(C)C)NCC1(F)CCN(C(c2n(CC=C)ccc2)=O)C1 14101,CC1CN(C(=O)C=CC2CCCC2)CC(C)N1C(C1CCC(C2CC2)C1)=O 14102,c12ncnc(c1C)NCCCN2C.Cc1cccc(CNC2C=CC(CO)C2)n1 14103,CCCCC(C(=O)N1CCC(NC(c2cc[nH]c2C)=O)C1)N(C)C 14104,Cc1nn(C)cc1C(=O)NC(C)(CNC(=O)CC1CC(C2CC2)C1)C1CC1 14105,C(=O)(C(CC(C)(C)C)OC)NCC(CC(=O)N(CCOCC=C)C)C 14106,C1(CCC)CN(C(c2cn(C3(OCC4CC4)CC3)nn2)=O)CCO1 14107,C1(O)(CNC(c2ccc(-c3cc[nH]n3)s2)=O)CCN(C(c2cnc(S)nc2)=O)C1 14108,C=CCC(CC)C(=O)N(C1CN(C(c2ccnn2C)=O)CC1(C)C)C 14109,C1(C(C(N2CCC(C(C)=O)C2)=O)C)CCN(C(C2(c3ccccc3)CC2)=O)CC1 14110,C1(C(=O)OC)CC12CCC(NC(=O)Nc1ccc(F)cc1Cl)CC2 14111,CC(C)(C)C#CC(=O)NCC1CN(C(=O)C=Cc2ccsc2)CC1(F)F 14112,N1(C(C(c2ccnn2C)NC(Cc2cc(C)[nH]n2)=O)=O)CCC2(COC(=O)N2)C1 14113,N1(C(C(C)NC=O)=O)CC(O)(CCNC(=O)Cc2ccsc2)C1 14114,C1(N(C(=O)CCCC2CCCC2)CC)CCCN(C(C2(C)COC(=O)C2)=O)C1 14115,C(=O)(C(S(C)(=O)=O)C1CC1)NCCCNC(C(Cn1ccc(C)n1)C)=O 14116,C1(C)(C(=O)NC(CC)(C)CNC(=O)CC2(CSC)CC2)CC(C)(C)C1 14117,N1(C(C(C=CC)O)=O)CCC(CC(=O)N(CCCOC)C)CC1 14118,N1(C(c2ncc(C)s2)=O)CCC2(OCCO2)C(C(=O)O)C1 14119,Cc1nsc(CNC(=O)CC(C2CC2)NC(=O)CC2(O)CCC2)n1 14120,N1(c2n(CCc3ccc(OC)cc3)nnn2)CCCC(=O)C1C 14121,c1(OC)cc(NC(C2CC(NC(C3CC(OC)C3)=O)C2)=O)cc(F)c1 14122,c1(C(=O)NC(CC)CNC(C2CCN2C2CCCC2)=O)ccc2ncccc2c1 14123,c1(OCC)cc(C(=O)NC(C)CN(C(=O)Cc2c[nH]ccc2=O)CC)ccn1 14124,c1(C(C)(F)F)ccnc(C(=O)NCCC2CCCN2C(C2CC2Cl)=O)c1 14125,N1(C(CC2C(OC(C)(C)C)C2)=O)CCC(NC(c2ccn(C(F)(F)F)n2)=O)C1 14126,c1(C(=O)NCCOCCC(=O)N(C23CC(C2)C3)C)cnn[nH]1.OC 14127,N1(C(CNC(CC)=O)=O)CC2CC(N(C(=O)C(C)Cn3cccn3)CC)C1C2 14128,C1(S(=O)(=O)C(N2CCSCC2c2ccccc2)=O)(SC)CC1 14129,N12CC3CC(CC1C3)NC(=O)C2=O.Cc1cc(OC(C)C)ccc1-n1cncn1 14130,C#Cc1ccc(C(C2NC(=O)N(c3ccccc3C)C2=O)=O)cc1C 14131,CC(C)C(O)C(=O)NCC1CN(C(c2cc(F)n[nH]2)=O)CC1O 14132,c1(C(c2ccn(C(C)(C)C)n2)c2nc(-c3ccco3)n[nH]2)cccc(S(C)(=O)=O)c1 14133,C1(NC(c2c(OC)ncc(C)c2)=O)CN(C(=O)C(O)c2ccco2)CC1C1CC1 14134,C1(Cc2c(O)ncc(NC(C)=O)c2)CN(c2ncncc2Cl)CC2(CCC2)C1 14135,c1(NC(C)=O)ncc(S(=O)(=O)NC2CCN(C(c3cc(Br)ncc3F)=O)CC2)s1 14136,c1(OCC(CN2C(CNC(c3c(COC)ncs3)=O)CCC2)O)cccc(C)c1 14137,N12CCCN(CC1)C(=O)OCC2.CC(C)(CF)NC(=O)NCCOC(C)(C)C 14138,CC1(C)CC(NC(=O)Cn2cnnc2)CCN(C(=O)CC2CC(OC(C)(C)C)C2)C1 14139,CC(O)C(C(=O)N(C1CC1)CC1CCN(C(c2ncoc2CN)=O)CC1)N(C)C 14140,C1(CC(=O)NC2CCCC(CNC(c3cccc[n+]3[O-])=O)C2)CCS(=O)(=O)CC1 14141,N1(CCCCC(C)Nc2cc(OC(F)F)ncn2)C(=O)c2ccccc2C1=O 14142,N1(C(C2(C)C(C)(C)C2)=O)CCC(CC(=O)NCC2CC3C=CC2O3)CC1 14143,N#CC1(C(=O)NC2CCCC(C(=O)NCc3ccncn3)C2)CC12CCC2 14144,Cc1cccnc1CCNC(=O)Nc1ccc(-n2ccnc2)nc1 14145,c1(C(N2CC(C)(C(N3CCCC(C)(O)C3)=O)C2)=O)ccc2[nH]ccc2n1 14146,Cc1cc(C)c(CCNC(N2CCN(c3ccccc3F)C(=O)C2)=O)c(C)c1 14147,C12CN(CCO1)C(=O)CCCNC2=O.Cc1noc(CCC(=O)NCC2CC2)n1 14148,N1(C(C2(C)CCC2)=O)CCOCC(CNC(=O)Cn2nnc(=N)[nH]2)C1 14149,c1(CC)cc(CC(N2CCCC2CN(C)C(c2cnoc2C(C)C)=O)=O)on1 14150,C1(O)(C(C)CNC(=O)Cc2ccc(F)cn2)CCN(C(c2cc(O)cs2)=O)C1 14151,N1(C(CN(C2CC2)CC)=O)CCC(CNC(c2ccc(O)cc2F)=O)C(CC)C1 14152,Cn1cc(C#N)cc1C(=O)NC1CN(C(c2coc(-c3cccnc3)n2)=O)C1 14153,CCCC(CCCNC(C12CC(CC)(C1)C2)=O)NC(c1cc(CC)cc(C)c1)=O 14154,C1(N(C)C)CCN(C(=O)C(CNC(C)=O)N(C(c2cnn(CCO)c2)=O)C2CC2)C1 14155,C(=O)(C1=CCSC1)N1C(C(C)(C)CNC(C2C(C)(C)C2(F)F)=O)CCC1 14156,C=CCC(F)(F)C(=O)NCC(C1(O)CCN(C(c2coc(C(N)=O)c2)=O)C1)C 14157,CC(CCNC(C1CN(C(c2ccoc2)=O)C(C)(C)C1)=O)CC(C)(C)C 14158,CCCN(CCC)N1Cc2ccc(OC)cc2C1 14159,N1(C(C(C)S(C)(=O)=O)=O)CC(NC(=O)CCC(=O)NCC2CC2)CC2(CC2)C1 14160,N1(C(C2CCC2)C)C2CCC(Nc3ccc(CC(Cl)Cl)cc3)C1CC2 14161,CCCC(C)(O)C(=O)N1CC(C(C)NC(c2ccc(=O)n(O)c2)=O)C1 14162,c1(C(=O)NCC2(O)CN(C(C=COCC)=O)C2)cc(C)c(C)nc1C 14163,C1(NC(COCC=C)=O)CC1C1CCN(C(C2CCc3nn[nH]c3C2)=O)CC1 14164,N1(C(CSCCCC)=O)CC2CCCN(C(=O)C(CC)Oc3cccc(C)c3)C2C1 14165,c1(C(C)NC(=O)C2CC2)coc2ccccc12.C12CCCN(C1)C(=O)C(=O)N2 14166,N1(C(Cc2ccc(C)cc2)=O)CCN(C(c2ccc(C)cc2Cl)=O)C(CC#N)C1 14167,N1(C(C2N(C(c3ccc(C#N)cc3)=O)CCCCC2)=O)CCC2(COC(=O)N2)C1 14168,C1(O)(CC)CCN(C(c2cc(C(N)=O)co2)C(=O)NC(C)CC)C1 14169,c1(CNC(C2CCC3(CN(S(=O)(=O)c4cccs4)C3)O2)=O)c(F)ccc(Br)c1F 14170,c1(C(=O)NCC23CCCCC2C3)ccc(Br)c(F)c1 14171,c1(C(=O)NCC(=C2CN(C(CC3CCC(OC)C3)=O)C2)F)cc(C)ncc1C 14172,N1(C(CC2CCC(C)O2)=O)CC2C(CCC(=O)Nc3ccnn3C3CCC3)C2C1 14173,c1(C(N(CC(C2CCCC2)C)C)=O)cc(C(F)F)nc2ccc(Cl)cc12 14174,c1(C(N2CC(NC(CC3CC(OC)C3(C)C)=O)(CO)C2)=O)ccc(Cl)c(N)c1 14175,N1(C(C)=O)C=Cc2ccccc2C1CC(=O)NCCn1cc(C(C)(O)C(C)C)nn1 14176,c1(CC)ccc(C(N2CCCC(NC(=O)C(=O)C(C)(C)C)C2)=O)c(OC)c1 14177,C1(C2CN(C(c3ccc(O)nc3Cl)=O)C2)(NC(C2CN3CCC2CC3)=O)CC1 14178,CCCC(O)(CCC)CC(=O)NC(C)CN(C)C(C1CCn2nccc2C1)=O 14179,N1(C(CCC=CC)=O)C2CCC1C(F)C(NC(C1(SC)CCN(C)CC1)=O)C2 14180,CC1=NOC2(C1)CC(C(N1CC(NC(c3cc(C)on3)=O)CC(C)C1)=O)C2 14181,C(CNC(C1(O)CCCC1)=O)(CC(C)C)NC(Cc1cnc(C)s1)=O 14182,C1(F)(C(=O)OC)CN(C(c2ccco2)=O)CC1c1cccnc1 14183,c1(C(=O)NC(CC(C)C)CNC(=O)C=CS(C)=O)coc2cccc(O)c12 14184,c1(OC)ccc(C(N2CCC2CNC(=O)Cn2cccnc2=O)=O)c(N)c1F 14185,C1(CC(=O)N(CCNC(COCCCC)=O)C)CCCCC1F 14186,Cc1ccc2sc(NC(=O)C(=O)NCc3cc(O)ccc3C)cc2c1 14187,C1(C(=O)NCCN(C(=O)CC2CC(C)(C)C2)C)CN(S(N)(=O)=O)C1 14188,N1(C(c2ccc(CSC)cc2)=O)CC2CC(C)N(C(C3CCC3CF)=O)C2C1 14189,N1(C(c2ccc(OC)c(Br)c2)=O)CCC2(CCN(Cc3ccc(O)c(O)c3)C2)C1 14190,O=C(C#CC1CC1)NCC=CCC(N1CCCC1c1ccsc1C(F)(F)F)=O 14191,C1(CC(C)NC(c2cc[n+]([O-])cc2)=O)CCN(C(=O)C2=CSCS2)CC1 14192,C(=O)(C#CC1CCCCC1)N(C1C(C)CCN(C(C2(C(=O)OC)CC2)=O)C1)C 14193,c1(C(N(CC(C)N(C(CN(C2CC2)CC)=O)C)C)=O)cnn(C2CC2)c1C 14194,C(=O)(C(C(C)NC(=O)CC1CCC(C)(C)O1)C(C)C)N1CC(CCO)(CC)C1 14195,C(C(C)(C)CN(C)C)N(C(CCN(C(c1cc(C)ns1)=O)CC)=O)C 14196,C#CCCCCCCNC(C1CC(C)CN(C(c2c[nH][nH]c2=N)=O)C1)=O 14197,Cc1cc(C(=O)NCC(C)NC(C2CCC3(CCOCC3)O2)=O)ccc1[N+](=O)[O-] 14198,CON1CCC(C(=O)NC2(C)CC(C(=O)NC3CC(F)(F)C3(C)C)C2)CC1 14199,c1(OCCC)ccc(C(=O)NCC2CC2NC(C2(CF)CCOCC2)=O)cc1 14200,N1(C(C(C)=C2CCCC2)=O)CCC2CC2(C(=O)Nc2cc(C)cc(C)c2O)CC1 14201,c1(SCCC2(c3ccon3)CC2)nocc1C(=O)NC(C1(CC=C)CCC1)=O 14202,C#CCCCCCC(=O)N(CC(C)CNC(c1cc(C)nn1C(C)(C)C)=O)C 14203,N1(C(c2cc(OC)ns2)C(=O)NC2CCN(C(C)=O)CC2)CC2CCCC2C1 14204,CC(C)CC(O)C(=O)NCC1CC(F)CN1C(=O)C1=CCCCC1 14205,C1(C)(OC(CC)(C)NC(=O)C2CC2)CN(C(=O)C(=O)OC(C)(C)C)C1 14206,c1(OC)cccc(CCC(=O)NC2CCCCN(C(=O)C(C)(C)C)C2)c1F 14207,c1(CC2C(C(N(CC(C)N(C(=O)CN3CCCC3=O)C)C)=O)C2)nccn1C 14208,C1(C(=O)NC2C(NC(COCCOCC)=O)COCC2)CC2CCCC2C1 14209,N1(c2ccnc(OC)n2)CCOC2CN(C(c3ccsc3C)=O)CC12 14210,CC1CC=CCC1C(N1CC(C(=O)NCC2(O)CCC(C)C2)C(F)C1)=O 14211,c1(OC)ccc(CCC(=O)N2CCC2CNC(=O)CS(N)(=O)=O)cn1 14212,c1(CC)cc(OC)ccc1N.c12ccc(cc1)N(CC)C(=O)C2N 14213,N1(C(C2CC(OC)C2)=O)CCC2C(NC(=O)CC3CN(C)CC3O)CC12 14214,c1(OC)cscc1C(N1CCC(CCNC(C2CC2F)=O)C1)=O 14215,C1(CNC(CN(C(=O)CC2CC(C)=NO2)CC#C)=O)C=CCCC1 14216,c1(C(C)C)conc1CC(=O)NC(CNC(=O)C(C)CC1CC1)C(C)C 14217,c1(OC)cccc(NC(c2c(C(F)(F)F)ccc(Cl)c2Cl)=O)c1[N+](=O)[O-] 14218,C=CCCCCCCCC(=O)NC1CCCCC1CNC(c1ocnc1CC)=O 14219,C1(CCNC(CCN(C(C)=O)C)=O)(NC(c2nnn(C)c2N)=O)CCOCC1 14220,N1(C(C2(C(C)=O)CC2)=O)CC(C(=O)NC(c2ccc(O)cc2)C)C(F)C1 14221,c1(OC)ccc(C(=O)NC2CCN(C(c3cncn3C)=O)CC2C)cc1N 14222,N1(C(COCCOCC)=O)CCC(NC(=O)COCc2cccc(C)c2)CC1 14223,c1(C(=O)Nc2ccc(-n3cc(-c4cn[nH]c4)nn3)cc2)cc2ccc(O)cc2[nH]1 14224,C=CCC(C)C(=O)NCC1(OC(C)(C)C)CCN(C(c2ccc(Br)nc2)=O)C1 14225,C(=O)(CC(C(F)(F)F)P(C)(C)=O)NCCC1CC(NC(c2c(C)[nH][nH]c2=N)=O)C1 14226,CCCCCCC(CC)NC(=O)C(C1CCCN(C(=O)CC(C)CC)C1)(C)C 14227,C#Cc1ncc(F)cc1NC(=O)NCC(c1ccc(Cl)cc1)CO 14228,c1(NC(CC2CCN(C(c3nc(CC)oc3)=O)C2)=O)cc([N+](=O)[O-])ccc1SC 14229,c1(OC)c(Cl)ccc(C(N2CC=CC2C(=O)NCCN2C(=O)CSC2=S)=O)c1F 14230,C(c1nc2ccccc2o1)=CC(=O)NCC1(F)CCN(C(C(C)OCC)=O)CC1 14231,N1(C(C(CC)c2ccccc2)=O)CC2(CC(NC(c3c(C)ncn3C)=O)CO2)C1 14232,Cc1[nH]nc(Cl)c1C(=O)NC1(C2CCCCN2C(=O)C=C2CCCCC2)CC1 14233,CC1CN(C(=O)Cc2nn(C)cc2Cl)CC1CNC(c1sccc1F)=O 14234,C1(C(c2n(CC(=C)C)nnn2)NCCc2cnoc2)CCCC(C)C1 14235,C(=O)(C1=NNC(=O)CC1)N1CC(C)C(CNC(=O)CC23COC(C)(C2)C3)CC1 14236,c1(CC(=O)NC2C=CCN(C(c3c(C(=O)OC)cco3)=O)C2)cc(F)ccc1Cl 14237,N1(C(c2c(C)occ2)=O)CCC2(CCOC2)C(CNC(C2(C(N)=O)CCC2)=O)C1 14238,c1(CCC(=O)NCCCN(C(=O)C(C)C2=CCCC2)CC)nc2ncccn2n1 14239,c1(NCC23CCC(C(=O)O)(CC2)O3)ncnc2sc3ccccc3c12 14240,N1(CC(C(=C)Br)O)CCN(C2(C(=O)O)CCCC2)CC1 14241,C(C#Cc1nccc(N2CCC(O)C(C3CC3)C2)n1)CCCCN=[N+]=[N-] 14242,C1(CC)CC(CC(N2CC(NC(=O)C(=O)OC(C)(C)C)C2)=O)CCO1 14243,N1(C(CC2C(C(=O)OC)C2(F)F)=O)CCOC(C)(CNC(=O)C(=O)NC2CC2)C1 14244,Cc1cc([N+](=O)[O-])c(F)c(C(=O)NCCc2cnn(C)c2)c1F 14245,c1(OCCCNC(=O)C(=O)Nc2cc(Br)[nH]n2)ccccc1O 14246,N1(C(c2c(C)nn[nH]2)=O)CCC(F)C(NC(c2cc(Br)ncc2Br)=O)C1 14247,c1(C(=O)NCC(c2c(OC)cccc2)C)csc2ccccc12 14248,c1(C(N(C2CCN(Cc3cnn(C)c3)C2)CCC)=O)ncoc1C 14249,c1(C(C(=O)NC2(OC)CC(SC)C2)C(C)C)ccc(C(F)(F)F)cc1 14250,N1(C(c2c(CC)noc2)=O)CCCC(F)(C(N2CCCC2C(C)(C)C)=O)C1 14251,c1(C(=O)NC2CC(NC(C(C(C)C)N(CC)CC)=O)C2)cc(F)cnc1O 14252,C1(NC(C2CCN(C)C2)=O)C2CN(Cc3ncc(Br)s3)CC12 14253,c1(CC(N2CCC(C)(NC(C=Cc3ccc(C)o3)=O)C2)=O)cccc([N+](=O)[O-])c1 14254,c1(NC(C2CCN(C(=O)CCc3ccnn3C)C2)C)ncc([N+](=O)[O-])c(=N)[nH]1 14255,N1(C(Cn2cnc(=N)[nH]2)=O)CCC2CCN(C(=O)CC=C(Cl)Cl)CC2C1 14256,O=C(C1CCCc2c[nH]nc21)NC1CN(C(c2cc(F)c(F)cc2N)=O)CC1F 14257,Cc1cnc(Cl)c(C(=O)NC(C2CCN(C(c3ccco3)=O)C2)C)c1 14258,c1(C(=O)NCC2(CCNC(CC(COC)C)=O)CC2)cnn2ncccc12 14259,C1(OCCC)CCC(CC(=O)NC2CN(C(=O)C=C(C)C)C2)CC1 14260,C1(C(=O)NC2CC(CNC(c3nc(C)oc3C)=O)CC2O)CC2OC1C1CC21 14261,c1(NCC(=O)NCC(c2cccc(Cl)c2)OC)ncc(C#N)cc1F 14262,C1(CCNC(c2csc(Br)n2)=O)CCCCN1C(C1(C2CC2)CC1)=O 14263,n1(CC=C)cc(C(=O)NC2(C(N3CC(C)(OC(C)=O)C3)=O)CCC2)cn1 14264,C1(CN(C2CC(F)(F)C2)C(C)(C)CO)CC(F)(F)C(=O)N1 14265,N1(C(C2N(C(CC(CC)O)=O)CCC=C2)=O)CC2CCCC(O)C2C1 14266,C(=O)(CC(C)CC(C)(C)C)NC(C(C(=O)NCCC(CC)(F)F)C(C)C)C 14267,N1(C(c2ccnc(C)c2N)=O)CCCC(C)(C)C1C(=O)NCCC(C)C(F)F 14268,O(S(=O)(=O)c1cccc2c1OC(C)C2)c1c(C(=O)OC)cc([N+](=O)[O-])c(Br)c1 14269,CC1(C)OCC2CC12C(=O)NCCC1COCCN1C(=O)C=Cc1ccccn1 14270,Cc1n[nH]c(C)c1CC(=O)NC1CCC(CNC(c2cnsn2)=O)C1 14271,CCCC(=O)NCC(=O)NCC(F)CNC(=O)Cn1cccn1 14272,C1(C(=O)Nc2cccc(CC)c2)CN(C(=O)COC2CCC2)CCC1CO 14273,N1(C(C(CCCC)(C)F)=O)CCC2(CCC(NC(C3CCCC3OC)=O)C2)C1 14274,N1(C(COc2cccc(C)c2)=O)CCC2CN(Cc3ccc(C)[nH]3)CC12 14275,c1(OC)cccc(OCC(N2CCC(NC(c3occc3Br)=O)C2)=O)c1[N+](=O)[O-] 14276,C#Cc1cncc(C(N2CC(F)CC2C(=O)Nc2ccc(O)cc2C)=O)c1 14277,N1(C(c2c(C)sc(O)n2)=O)CCC2(CC1)CC(NC(c1ncoc1C1CC1)=O)C2 14278,N1(C(CC=CC=C)=O)CCC(C)(C)C1CNC(c1scc(C)c1Br)=O 14279,C1(NC(C(C(C)C)CO)=O)CCC2(CC1)CCN(C(c1cc(C(N)=O)no1)=O)C2 14280,C1(C(=O)NC(CC)CNC(=O)CN2CCCCC2)CCC2(CCC2)OC1 14281,c1(C(=O)NCC2C(NC(C3(OC)CC(C)C3)=O)C2)cc(S(=O)(=O)CC)ccc1F 14282,CC1CC(CNC(c2ccc(C#N)n2C)=O)CCN1C(=O)C=CC1CCCC1 14283,N1(C(C(C)S)=O)CCN(c2ncc(-c3ccc(CO)cc3)cn2)CC1 14284,Cc1n[nH]c(C)c1C(C)C(=O)N1CC(CNC(c2coc(OCC(F)(F)F)n2)=O)C1 14285,c1(C(N(C)CC2COCCN2C(=O)CC2(C)CCCC2)=O)cccc(S(C)=O)c1 14286,N(C1c2ccccc2CC1NC(=O)C(O)P(C)(C)=O)C(C(CCSC)OC)=O 14287,c1(OC)c(C(=O)NC2CC(C)CN(C(c3cncc(C)c3)=O)C2)cccc1C#N 14288,C1(CNC(CCC2CCN(C(c3c(C)nc(CC)o3)=O)C2)=O)CC12CCCCC2 14289,N1(C(CCC=CC(C)C)=O)CCN(C(C2CCCN2C2CCOCC2)=O)CC1C 14290,N1(C(C(C)CC(F)(F)F)=O)CCC2C(CCN2C(=O)C(c2ccccc2)C)C1 14291,C(S(=O)CC(=O)N1CCC(C(=O)Nc2ncccc2C)CC1)c1cc(OC)no1 14292,C1(C(=O)NCCC(CC)(C)O)CN(C(c2sccc2C)=O)CC(C)C1 14293,Cc1c(C(=O)NC2CC(C)CN(C(C3CCC(C)CC3)=O)C2)cccc1F 14294,C1(NC(c2occ(C(=O)OC)c2)=O)C2CC(CN(C(C3CCC3)=O)C2)C1CO 14295,CCCC(C(=O)NCC(C(C)C)NC(c1cn(CCCOC)nn1)=O)N(C)C 14296,N1(C(CC2OCC(C)(C)OC2)=O)CC2=C(C1)CN(C(=O)CC1CC3CCC1O3)C2 14297,N1(C(c2cc(CCC)[nH]n2)=O)CCN(C(C)CNC(C2CCO2)=O)CC1 14298,Cc1ncc(C#N)cc1NC(=O)CCNC(C1C2CCCC(=O)C12)=O 14299,N1(C(C2C=CCN(C(c3cc(COC)no3)=O)C2)=O)CCC(O)C(C)(C)C1 14300,CC1(C)CC(C(=O)NCCC2CN(CCCS(C)(=O)=O)CCS2(=O)=O)CC(C)(C)O1 14301,C1(C(=O)NCCCN(C(=O)Cc2nn(C)cc2Br)CC)CC2CC(=O)C1C2 14302,C#CC(C(C)OC)NC(=O)C=CC(C)(C)NC(=O)C(C)c1ccco1 14303,Cc1cc(F)c(CC(=O)N(C)CCN(C)C(C2CCCC3CC23)=O)cc1F 14304,C1(C#N)(C(=O)NCC(CNC(c2c(OCC)cccn2)=O)OC)CCCCC1 14305,c1(C(=O)NCC(C)NC(C2CC3CC3C2)=O)ccncc1I 14306,C1(C2CCC2)(NC(c2ccn(C(C)C)n2)=O)CC1.C1CC(=O)NCCS1 14307,c1(CN2CC3N(C(Cc4c(OC)ccc(F)c4)=O)C(C3)C2)cccc(F)c1C#N 14308,C1(C(=O)NCCc2nncs2)CC(F)(F)CN1C(=O)CNC1CCC1 14309,c1(OC(C)C)cccc(-c2ccc(C(=O)Nc3ccsc3CO)nc2C)c1F 14310,N1(C(C(C)=C(CC)C)=O)CC2CC3CC2C1C3NC(=O)Cc1ccoc1 14311,Cc1ccccc1CNC(C1CC1C(N1CCC(NC(=O)Cn2cnnn2)C1)=O)=O 14312,N1(C(C2(C)CC=CC2)=O)CCOCC1CCNC(=O)Cc1cc[nH]n1 14313,C1(CNC(C(COC)O)=O)CC2(CO1)CN(C(=O)CSSC)C2 14314,c1(NC(N2CCN(C(C(CC)N)=O)CC2)=O)cc(C)nc(C)c1 14315,c1(C(N(C2CCN(C(c3cnc4[nH]ncc4c3)=O)C2)C)=O)ccc2ncnn2n1 14316,Cc1nnc2n1CC(C(=O)NC(CNC(c1nccn3cnnc13)=O)C(C)C)C2 14317,C1(C(N(C2CN(C(Cc3c(C)noc3)=O)CC23CC3)C)=O)CC(=O)N(C)C(=O)N1 14318,C#Cc1cccc(C(N2CCOC(C)(CC)C2)C(=O)NC2CCCCC2)c1F 14319,c1(CN)cc2c([N+](=O)[O-])ccc(C(=O)NCc3ccc4ccsc4c3)c2[nH]1 14320,CN1N=C(C(=O)N2CC(O)CC2C(N2CCOCC2CCO)=O)CCC1=O 14321,C1(NC(c2ncc(OC)cn2)=O)CC(N=c2[nH]nc(C3CC3)s2)C12CCC2 14322,C12(CNC(C34CC(CC(C)O3)C4)=O)CN(C(=O)C=C3CCC3)CC1CCO2 14323,C1(OC)CCC(CC(=O)NCC2CC(C)N(C(=O)Cc3cccnc3Cl)C2)CC1 14324,C(=O)(C1=CC2(CCN(C(=O)CC3COC(=O)C3)C2)C1)NC(CC#C)CC#C 14325,C1(C(N2CC(COC)(CNC(=O)Cc3cnoc3)C2)=O)CCC(C)(C)O1 14326,C12(CNC(c3c(C)nsc3)=O)CCCC1CN(C(=O)CCc1ccccc1)C2 14327,c1(CNC(N2CCC(C)C2)=O)nc2cc(Cl)c(Cl)cc2[nH]1 14328,O=C(CCCC1(c2ccccc2)CC1)N(C1CCCCC1)CCO 14329,C(c1cccc(Cl)c1)=CC(=O)NC(c1sc(C(=O)OCC)c(C)n1)C 14330,c1(C(N2CCC(O)(C(C)NC(c3nnc(C)s3)=O)C2)=O)csc2cccnc12 14331,c1(C(N2CCC(N(C(C3CC(O)(C(F)(F)F)C3)=O)CC)C2)=O)cc(F)cc(Cl)c1 14332,CCCC(C(=O)N(C)CCNC(c1ncncc1Cl)=O)S(N)(=O)=O 14333,c1(C(=O)NC2CC3CC(NC(c4c(C)cns4)=O)C2C3)nc2ccccc2[nH]1 14334,c1(C(N2CC(N(C)C)C(C)(C)C2)=O)coc2c1CN(C(C1CCCC(O)C1)=O)C2 14335,C1(C)(CNC(=NCCOC)NCC(C2CCOC2)O)Cc2ccccc2C1 14336,C1(NC(c2ncn(C(C)(C)C)n2)=O)CCNC2(CCOCC2)C1 14337,Cc1cc(C(N2CCC(O)(CNC(=O)C(F)(F)C(C)O)C2)=O)ncc1C#N 14338,CCC(O)C(F)(F)C(=O)NCC1(C)CC(NC(=O)CN2CCCCCC2)C1 14339,C1(NC(c2c(OC)c(F)ncc2)=O)CC2(CCN(C(c3sc(C)nc3C)=O)C2)C1 14340,N1(C(C(C)O)=O)C2CCC1CN(C(C1CCN(CC(F)(F)F)CC1)=O)CC2 14341,N1(C(C=C)=O)CC2CCCC(NC(c3cc(N)cc(OC)c3OC)=O)C2C1 14342,C(N=c1nc(N2CCCC(C3(C)CC3)C2)c2c([nH]1)CCC2)c1ccc(C)cc1Br 14343,C1(NC(CC(C(=C)C)OCC)=O)C2CCCN(C(=O)CC3CCSC3)C2C1(C)C 14344,c1(C(N2C(C)CCC2C(=O)NOCC(O)CO)=O)ccc(Br)c(O)n1 14345,Cn1nnc2cc(-c3nc(Cc4ccnc(Cl)c4O)no3)cnc12 14346,Cc1cc(N)n2ncc(C(N3CCC3CNC(C3(C(=O)N(C)C)CC3)=O)=O)c2n1 14347,CC(C)CC(C)(O)C(=O)NC1CCCC(CC(=O)NCC(O)C(C)(C)O)C1 14348,c1(C(N2C3C(NC(c4ccc(COC)s4)=O)CC(C3)C2)=O)cc(F)cc(N)c1F 14349,C1(NC(c2cc(C)no2)=O)CC(Nc2nccc(CO)n2)C1(C)C 14350,O=C(C(O)C(F)(F)F)N1CCOCCC1C(=O)NOCCCC(F)(F)F 14351,CCC(C#N)C(=O)N(C(C)CNC(=O)Cc1ncc(Br)s1)C 14352,c1(NC2C3CN(C(CCCC(C)CCC=C)=O)C(C3)CC2)cc(=O)n(C)c(=O)n1C 14353,c1(CC(C(=O)NC2C3CCN(C(c4scc(C)c4)=O)C32)O)c(F)cccc1Cl 14354,C(C(CC(C)C)C(=O)N1CC2CCCC1C2)NC(C(CC)CN(C)C)=O 14355,C1(N(C)C(c2cncc(N3CCCC3)n2)=O)CCCN(C(c2csnn2)=O)CC1 14356,c1(NC(=O)NCCc2ccc(C)o2)cccc(N=c2cc[nH]cc2)c1 14357,N1(C(c2c(C)cc(SC)o2)=O)CC2CC(NC(C3CCCC3(C)C)=O)CC1C2 14358,C1(CNC(c2cc(C(C)=O)oc2)=O)CCN(C(=O)C(C)(C)C2CC2)CCC1(F)F 14359,C1(OCC)CCN(C(=O)N(C(C)C)CC2CC2c2ccccc2)CC1 14360,N1(C(CC(C)N(C(C(CCCC)O)=O)C)=O)CC2(CCCCCC2)C1 14361,O=C(C(O)c1ccsc1)NC1(C(=O)NCC(Cl)=CCl)CC1 14362,C1(C(=O)NCCC2N(C(CCN(CCC)C)=O)CCOC2)CCC(C)=C(C)C1 14363,N1(C(c2n(CC(C)C)ncc2)=O)CCCC2(CCC(NC(C3(C)CC3)=O)C2)C1 14364,C(=O)(C1=NOC2C3CCC(C3)C12)NCC(CC)SCC 14365,CC1=CCC(N=c2ccc(Br)c(S(=O)(=O)NC3CCC4(CC3)C3CCC4O3)[nH]2)CC1 14366,C(c1cc(Cl)c2c(c1)OCO2)=CC(=O)NCCCNC(C1(C)CC1F)=O 14367,S(=O)(=O)(c1ccc(Cl)cc1)N(C(CCC)C)C(c1cnn(C2CNC2)c1)=O 14368,c1(OC)cc(C(N2CC(NC(=O)C(C)(F)F)C(c3ccccc3)C2)=O)nn1C 14369,c1(C(=O)NC(C2N(C(C(C(C)C)OC)=O)CCC2)C)cc(Cl)cc2cccnc12 14370,C12(NC(C(F)=C(C)C)=O)CC(CNC(=O)CSC(F)(F)F)(C1)OC21CCOCC1 14371,C(=O)(CC(C(F)(F)F)NC(=O)CCn1ccc(C)n1)NCCC1ON=C(C)C1 14372,Cn1ncc2cccc(C(N3CCC4CN(C(=O)Cn5cccn5)CC34)=O)c12 14373,CC1CCN(C(=O)C(C)Cc2ccccc2)CCN1C(=O)CC1CCCO1 14374,S(=O)(=O)(c1cc(NCCCC(N)=O)ccc1N1CCSC1)N(CC(C(C)C)O)C 14375,c1(C(N2CC(NC(c3cc(CC)cc(N)c3)=O)C2)=O)oc2ccccc2c1Cl 14376,c1(C(C)C)cccc(F)c1C(=O)NC1CC(NC(C2C3CC4C(C3)C24)=O)C1 14377,C#CCCCCC(=O)NC(CC1CC1)C(=O)NC(C)(C)C(N)=O 14378,c1(C(=O)NC(CNC(C(CSC)C)=O)(C)C2CC2)cnc(O)c(C(F)(F)F)c1 14379,Cc1cc(=O)n(CCC(N2CCC(NC(c3cnns3)=O)C2C(C)(C)C)=O)cn1 14380,C=CCC(CO)NC(=O)C(C1CCCCC1)NC(=O)OC1CCC(=O)C1 14381,C1(CN(C)C(C23CSCC2C3)=O)CCN(C(C2CC23CCC3)=O)CC1 14382,C1(C(C)CNC(=O)C(=O)NCC2CC2)CCCN(C(=O)C=CC2CC2)C1 14383,C1(CNC(CCCC#C)=O)COC(C)(C)CN1C(C1CCC(F)(F)C1)=O 14384,C=CC(CCC)CC(=O)NCCC1CCCN(C(C2(C(C)C)CCC2)=O)C1 14385,c1(C(=O)NCCNC(c2c(C)n3c(s2)ncc3)=O)cc2c(s1)CC(C)CC2C 14386,c1(N2C(CNC(c3c(C)cc(C)o3)=O)C(C)CC2)nc2ccccc2s1 14387,n1(CCC)c(CN2CCC(NC(=O)C(c3ccc(C)cc3)=O)C2)nnc1C 14388,N1(CC(C)NC(c2c(C(C)C)c[nH]n2)=O)CCN(C(=O)C(C)(O)C2CCC2)CC1 14389,c1(C(N2CC(NC(CCSCC)=O)C(C)CC2)=O)nn2c(c1C)OCCC2 14390,CCC(CC)(CC)C(=O)N1CCC(N(C(=O)Cc2csc(C3CC3)n2)C)C1 14391,C#Cc1ccc(C(=O)N(C2CCCN(C(c3ccn(C4CCC4)n3)=O)C2)C)nc1 14392,C(CNC(c1c(F)cccc1Cl)=O)(CC(F)(F)F)NC(CC(C=C)C)=O 14393,c1(N(C)C2CC2)nc2c(c(=NCC34CCC3CN(C(c3cccs3)=O)C4)[nH]1)CSC2 14394,c1(OC)ccc(S(=O)(=O)NCC2CCCN2Cc2cccc(O)c2F)cc1Br 14395,C(CCC(N)=O)(C(=O)NCc1cc(C2CC2)n[nH]1)n1cc(CCN(C)CC)nn1 14396,N(C1CCCn2ncnc21)C(C1C2CN(C(=O)C3=C(Cl)CCCC3)CC21)=O 14397,CN1N=CCCC1C(N1CC=CC(C(=O)N(C)CC2(CO)CC2)C1)=O 14398,CC1(C=CC(=O)NCC2CCC(NC(=O)CCn3cccc3)C2)CCOCC1 14399,c1(C(=O)NCC(CCOC)NC(C=COCC)=O)nc(OC)ccc1C 14400,N1(C(CCC(=C)C)=O)CCC(NC(c2ccc(OC)nc2)=O)CC1C1CC1 14401,C(c1ccc(Br)cc1)=CC(=O)NC(C)CCCNC(=O)CP(C)(C)=O 14402,N1(C(COCc2cc(C)no2)=O)CCCC1(C)CNC(c1nccs1)=O 14403,c1(SC)nc(N2CCC(O)(C(N3CCC3(C)C(C)C)=O)C2)c(Br)c(C)n1 14404,C(=O)(C(O)(CN(C)C)C(F)(F)F)NCC1N(C(c2cc(OC)ns2)=O)CCC1 14405,CC1CC(NC(c2cccc(Br)c2)=O)CCN1C(=O)CC1CCCCN1C 14406,C#CC1CCC(C(=O)NCCN(C(=O)C(C)N2CC(C)C2)CCOC)CC1 14407,C12(C(N3CC4C(CC(=O)NCCc5ccc(O)cc5)C4C3)=O)CCCC1OCC2 14408,C1(O)(C(C)NC(CSCCC)=O)CCN(C(C2C=CC=CC=C2)=O)CC1 14409,C(CC(C(=O)NC1CC(C(F)F)C1)NC(C1CC(C(=O)OC)C1)=O)OC 14410,C1(C(=O)NC2C(CCC)C2)CCCN(C(c2ccccc2OCC)=O)CCC1 14411,Cn1[nH]nnc1=NCCCC(C)(C)NC(C1(c2cccc(F)c2)CC1)=O 14412,c1(C(=O)NCCC(C)N(C(=O)C=C2CCCCC2)C)ccc2c(c1N)CCCC2 14413,c1(C(=O)OCC)ncc(C(=O)NCC(CNC(c2cscn2)=O)OC)s1 14414,N1(C(c2ccc(Cl)cc2)C(=O)NCCC#N)CCCN2CCCCC12 14415,c1(C(N2CCC(N(C(CSCC=C)=O)C)C2)=O)cc2c(nn1)CCCC2 14416,Cc1nn(C)c(C(N2CC3C(NC(=O)CC4CCOC4=O)C3C2)=O)c1Br 14417,c1(OC)cc(C)c(C(=O)NC2CC(NC(=O)CN3CCOC3=O)C2)cc1Cl 14418,C(=O)(C(C)(CC)CC)N1CCC(N(CCC)C(c2ccc(CN(C)C)o2)=O)C1 14419,C1(NC(=O)CCNc2ccccn2)CCN(C(c2cncc(C(F)F)c2)=O)CC1 14420,N1(C(=O)NC2C(CC(C)C)C2)CCN(CCN(C)Cc2cc(C)nn2C)CC1 14421,C1(C)(N(NC(C(CC)N(CC)CC)=O)CC)CCCN1c1ncncc1Br 14422,c1(NC(C(=O)NC(CC#C)COC)=O)cc(C)ccc1N 14423,c1(OC)cc(C(=O)NC2CC(N(C)C(c3cn(C)c(O)n3)=O)C2)nc(C)c1 14424,N1(C(C2(NC(=O)CCn3ccnn3)C(C)CCC2)C(=O)OC)CCCCC(CO)C1 14425,O=S(=O)(c1ccc2nc(N3CCC(O)C(F)C3)ccc2c1)N1C2CCC1CC2 14426,c1(CC(=O)NC(C2CCN(C(c3cncnc3)=O)CC2)C)ccccc1S(C)=O 14427,C1(n2c(COC(F)(F)F)nc(-c3ccc(OC(C)C)cc3)n2)C(C)CCCC1C 14428,N1(C(c2c(OC)nc(C)nc2)=O)CCCN(C(c2ccc(F)cc2C)=O)CC1C 14429,c1(NCCCCC2CC(OC)C2)cc(=NCC(C)(c2ccccc2)SC)[nH]cn1 14430,CCCC(CCC)CC(=O)N1CCOCC1CNC(=O)C(C)(CC)CO 14431,CONC(=O)CNC(=O)CCC1CC(NC(c2coc(C(N)=O)c2)=O)C1 14432,C1(CC(=O)NCC(C)=O)C(CCC(C)C)NC1=O 14433,C1(NC(c2cc(C3CC3)cs2)=O)CCN(C(C2CCCCS2(=O)=O)=O)CC(O)C1 14434,N1(C(C2C(CC(C)C)C2)=O)CCN(C(=O)CCCc2ccncc2)C2CC12 14435,C1(C(C)=O)CCN(N2CCN(C3CCCN(C4CCCC4)C3)C(=O)C2CC)CC1 14436,CC(CC#N)N=c1cc[nH]cc1S(=O)(=O)NCC1(OC(F)F)CCCCCC1 14437,N1(C(C2C(CNC(COCCCN=[N+]=[N-])=O)C2)=O)C(CO)CCC12CCC2 14438,c1(C(=O)NC2CCC(CCNC(C3(CCCC)CC3)=O)C2)cc(C)c(O)c(C)c1 14439,c1(C(N(C2CC(NC(c3ccc(C#N)n3C)=O)C2)C)=O)cccn(C)c1=O 14440,c1(C(=O)NCC2C(C)(C)CCN2C(=O)CSCCC#N)cnn2c1OCC(O)C2 14441,C(=O)(C(C)CC(C)C)N1CCC(N(C(C(C(=O)OCC)F)=O)C)CC1 14442,c1(NCCN(C(C)(C)C)C(C2C(NC(=O)OC(C)(C)C)C2)=O)cc(Br)cc(F)n1 14443,N1(CC(n2c(C)ncc2)C)CC2C(C(=O)NC(C)C(C)C)C2C1 14444,c1(CC(=O)NCC2C3CN(C(c4n(CC)ccc4)=O)CC32)nsc2ccccc12 14445,N(C(=S)N1CCC1c1cccc(F)c1)CC.c12cccc(c1)NC2=O 14446,Cn1cc(C(=O)NCC23CC2CN(C(c2ccnn2CC2CCC2)=O)C3)c(Cl)n1 14447,CCC(C)(COC)CNC(=O)CONC(=O)C=CC1(C)COC1 14448,C(C)(C)(CC(=O)NC(C)CC(C)NC(=O)CCCCc1cnc[nH]1)OC 14449,C1(C(N2CCC(CN(C(C(CC)(C)O)=O)C)CC2)=O)CC(c2ccncc2)=NO1 14450,C1(NC(c2cnn[nH]2)=O)CN(Cc2ccn(-c3ccc(C(=O)O)cc3)n2)CC1O 14451,c1(OC)cc(F)c(SCC(C)(C)C(N2CCC(C)C(NC(=O)COC)C2)=O)cc1N 14452,C1(CC)C(C(=O)N(C)Cc2cccc(OC)c2)CCN1C(c1cnn(C)c1Cl)=O 14453,N1(C(CCS(=O)(=O)NC)=O)CCC(NC(=O)C2CCc3c[nH]nc32)CC(C)(C)C1 14454,N1(C(C(C2CCCCC2)C)=O)CCC(C)C(CNC(=O)C(C)(C)CO)C1 14455,CCC(CC)C(=O)N1CCCC1CSC1CN(C(c2ncn(C)c2C)=O)CCO1 14456,c1(C(N2C(C)CC(C(=O)OCCC)C2)=O)cnn2c1CN(C(C)=O)CC2.C(C)(C)(C)O 14457,N1(C(Cc2c(C)non2)=O)CCC2CCN(C(C3CC(C)(C)CN3C)=O)CC12 14458,c1(CN(C(C2C(C(=O)OC)C2)=O)CC=C(C)C)ccccn1 14459,C#Cc1cccc(C(=O)NC2CCN(C(C3CC=CC3)=O)C(C3CC3)C2)c1Cl 14460,c1(N(CC(C)C(C)(C)C)C)nc2c(c(=NC3COC(C)(C)C3)[nH]1)COCC2 14461,C(C(CO)(CO)NC(c1cncnc1)=O)N(C(C1C(OC)C1)=O)C 14462,c1(C(=O)Nc2ccc(OCC(=O)NCC)cc2)c(C#N)cnn1C 14463,C1(NC(C(CC(=O)OC)C)=O)CC2CCC1CC2NC(=O)CC1(CS(C)(=O)=O)CC1 14464,c1(C(=O)NC23C(CN(C(CC4C(C)(C)CC4)=O)C2)C3)cccc2c1OCCO2 14465,C1(C(N2CC(CNC(c3cc(OC)no3)=O)(COC)C2)=O)CCCCN1C(C)C 14466,C(CC(C)(C)C(=O)N1CCCC(NC(c2csc(Br)c2Cl)=O)C1)OC 14467,C1(C(N(CC(C)C#N)C)=O)CCCCCC1NC(C1CCC(F)CC1)=O 14468,N1(C(CCN(C2CCCCC2)C)=O)CCCC(NC(=O)NC2CC3(CC3)C2)C1 14469,N1(C(c2c(C)coc2)=O)CCCN(C(=O)C(CO)N(C)C)CC1c1ccccc1 14470,N=c1cc[nH]cc1C(=O)NC1CC1NC(c1ccn(CC(F)(F)F)n1)=O 14471,C1(O)(CNC(Cc2cncc(C)c2)=O)CCCN(C(c2nn(C)c(C)c2Cl)=O)C1 14472,c1(CC(=O)NCCN2CCN(C(C=C(COC)C)=O)CC2)c(C)nc(O)nc1C 14473,Cc1nc(NC(c2sccc2NC(c2ccnc(OC(F)(F)F)c2)=O)=O)sc1C 14474,Cc1c[nH]cc1C(=O)N(C)CCOCCN(C)C(C1CC1C(C)C)=O 14475,C12(CNC(C=CC)=O)CC(NC(=O)CC(CC)SC)(C1)C(C)(C)O2 14476,C1(N)(N(C)C(c2cccnc2)C)CCCN(C(=O)C(N2CCCC(C)C2)=O)C1.CC 14477,CCCC(CC)CCC(=O)NC12CC(C(N3CC(O)(CO)C3)=O)(C1)C2 14478,CCCCS(=O)(=O)NCC(=O)NC(CNC(c1ccc(COC)nc1)=O)CO 14479,C(=O)(C(CC(N)=O)NC(c1cc(C)n(C)c1)=O)NCCCOCCCC 14480,c1(CCC)nc(C(O)Cc2ccccn2)n(CCO)n1 14481,N1(C(CSCC=C)=O)CCCN(C(C2(C3CC3)CC2)=O)CC1c1ccccc1 14482,N1(C(CN2C(C)CCC2)=O)CC=CC(NC(C2CC2C)=O)C1 14483,N1(C(=O)NC(CCC=C)C2CC2)CCOCC1CC(C)C 14484,C1(NC(Cc2c(SC)cccc2)=O)CCN(C(c2cc(F)c[nH]2)=O)C(C)C1 14485,C1(C2(O)CCOCC2)(C(=O)NC2(C)CN(C(=O)Cc3cccc(N)c3N)C2)CC1 14486,c1(C(N2CC(NC(C3C(CC)OCC3)=O)C(C)(C)C2)=O)cncc(N=[N+]=[N-])c1 14487,c1(OCCCOC)ccc(C(=O)N(CC(O)CNC(=O)C#CC2CC2)C)c(Cl)c1 14488,C1(C(=O)NC2(C)CCN(C(c3oc(CC)c(C)c3)=O)CC2)CCCC1S(C)(=O)=O 14489,c1(C(=O)N(C(=O)CC2CC=CCC2)C2CNC2)cncc2nc[nH]c12 14490,C=Cc1ccccc1NC(=O)CC(=C)C 14491,Cc1c(C(=O)NC2(CCNC(=O)CCF)CC2)cc(-c2ccccc2)n1C 14492,N1(C(CC2(OC)CCC2)=O)CCN(C(c2cccc(F)c2O)=O)C2(CC2)C1 14493,N1(C(c2nc(CC)[nH]n2)C(=O)NC)CCC2CCN(C(C)C(=O)OC)CC12 14494,C1(O)(C(C)NC(COCCNC(c2c(C)scc2)=O)=O)CCCCC1 14495,C1(C(N(CCN(C(=O)CO)C(C)C)C)=O)CCC(C(F)(F)F)O1 14496,CC1CN(C(C2CC3C(C2)C3(F)F)=O)CCC1CNC(c1c[nH]c(C(N)=O)c1)=O 14497,c1(CN2CC3(CC(CC(=O)NC4C(C(C)(C)C)C4)C3)C2)csc2ccccc12 14498,Cc1cc(C(=O)NCC2(C3C(C)(C)C3(C)C)CC2)c(C)[nH]1.C12(C)CC(C1)NC2=O 14499,N1(C(C(C2CC2)SC)=O)CC2(C(=O)N(CC3=CCSC3)C)CC1CO2 14500,N(C1CC2(CN(C(=O)CC3CC3)C2)n2ccnc21)C(C1C(=O)NCC1)=O 14501,C1(C(N(CCNC(c2nc(CCOC)oc2)=O)C)=O)CCc2nnc(O)n2C1 14502,Cc1cccc(NC(=O)C=CCN(C(=O)CCN=[N+]=[N-])C)c1 14503,CCCCC(C(=O)N1CCN(C(c2cc(C(C)(C)C)oc2C)=O)CC1CC)N(C)C 14504,c1(C(NC(=NCCC#C)NCc2noc(C3CC3)n2)C)ccc2ccccc2c1 14505,C(=O)(C(C)S(N)(=O)=O)N1CC(O)(CNC(c2c(C)n(-c3cnn(C)c3)nn2)=O)C1 14506,C(=O)(CC1C(=O)Nc2ccccc21)NCCCCNC(CC(C)(C)CC(F)F)=O 14507,C1(C2CCNCC2)(CNS(=O)(=O)Cc2ccc(Br)c(F)c2F)CCC1 14508,C(=O)(C(C)CC(C)(F)F)NCC(CCNC(CC(C=C)(C)C)=O)O 14509,C1(C(N2CCC(c3cn(C4CCC(F)C4)nn3)C23CC3)=O)CCCN2CCCC12 14510,C(=O)(CCCCC(N)=O)N1CCC(CCNC(CN2CCCC(CC)C2)=O)CC1 14511,CC1OC2(C(=O)NCC=CCNC(=O)C(F)(F)C3CC3)CCC1CC2 14512,c1(CC)nc(N2CCCC2CCCNC(C2(C(C)(F)F)CC2)=O)[nH]c(=N)n1 14513,CCC(C)(C)C(C)CC(=O)NC1CC2CCC1(NC(=O)CN(CC(C)(C)C)C)C2 14514,c1(C(N2CCCC2)=O)cc[n+]([O-])cc1.O=C1CCN1.C12CC1NC(=O)C=CCN2 14515,c1(C(C(F)(F)F)C(=O)NC(c2ccc(C)o2)C(N2CC(F)(F)C2)=O)ccc(O)cc1 14516,C1(NC(C2CC3CCC3C2)=O)CC2(CCN(C(=O)CN3CCCOC3=O)CC2)C1 14517,C1(C(N)=O)CCC(CCC(=O)NCC2CCN2C(c2ccsc2Cl)=O)O1 14518,c1(OC)ccncc1C(=O)N(C)CCN(C(c1ccn(C)n1)=O)C(C)C 14519,c1(C(N2CC3(CCN3C(c3cc(Cl)sc3Cl)=O)C2)=O)cc2n(c1)CCOC2 14520,N1(C(CC=CCC)=O)CCCC(C(N2CCC2CC(=O)OC)=O)C1 14521,c1(C(=O)NCC(C)N(C(=O)CC2C=NN(C)C2=O)C)coc2c(Cl)cccc12 14522,C1(NC(C2(C(=O)NC)CCC2)=O)CCC(Nc2ncncc2I)CC1 14523,c1(CNC(c2c(C)n[nH]c2)=O)ccc(CNC(c2c[nH]c(C(F)(F)F)c2)=O)cc1 14524,C1(C(=O)NCc2c(CNC(c3n[nH]c(C)c3O)=O)cccc2)CC12CCCCC2 14525,C(=O)(C(CCC=C)NC(=O)CCc1cnn(C)c1)NCCC(=C)C 14526,C1(CNC(C(=Cc2cn[nH]c2)C)=O)(NC(C2SCCCS2)=O)CC2CCC1C2 14527,c1(CC)ccc(C(=O)OCC(=O)CC(C)(C)C2CC2)cc1[N+](=O)[O-] 14528,O(N(C(=O)CC1COCCN1C(=O)CCOCC(F)F)C(C)C)CC 14529,CCC(CC)N(CCC(=O)NC(C1CN(C(=O)Cc2cn[nH]c2)C1)C)C 14530,c1(C(N2CC(O)(CN(C(C3(NC(C)=O)CCOC3)=O)C)C2)=O)cc(C)nc(O)c1 14531,C1(NC(c2c(C)ncs2)=O)CCCOC12CCN(C(=O)CC1CC=CCC1)CC2 14532,N1(C(C(CC=C)C)=O)CCN(C(=O)Cc2noc3ccccc23)CC(CO)C1 14533,C1(NC(C(C)=C(CC)C)=O)C=CCCC1C(=O)NCc1cn(CC)nn1 14534,CC1CN(C(=O)CCCC2CC2)CC1n1cc(CCO)nn1.C12(CCC1)CC2 14535,C1(CNC(C(COC)(F)F)=O)CN(C(=O)C(C)NC(C)=O)C2(CCC2)C1 14536,C(=O)(C(C)(C)CC(C)C)N1CCN(C2C(NC(C=NOC)=O)CCC2)CC1 14537,N1(C(CCOC)=O)CCCC1C(C)(C)CNC(C1C(C)C1(F)F)=O 14538,C(=O)(C(C)(C)C(F)F)NC1CC2(C(NC(c3cc(COC)cn3C)=O)C2)C1 14539,c1(NC(C)=O)cccc(NC(=O)CC(c2cn(C)nc2C(F)(F)F)C)c1 14540,C1(NC(c2nc(COC)sc2)=O)CCCC(NC(c2cnc3n2CCC3)=O)CC1 14541,C12(C(=O)NCC3(C)CCCOC3)CCCC1CCN2C(=O)CCS(C)(=O)=O 14542,C1(C(=O)NC2(CO)CCC(C)(C)C2)CN(C(C2CCO2)=O)CC1C1CC1 14543,c1(NC(C(c2ccccc2)NC(C(C)(C)NC(C)=O)=O)=O)cccn2nccc12 14544,C=C(Cl)C(C)(C)C(=O)OCC(=O)OCC(=O)NCc1cc(OC)nnc1OC 14545,Cc1c(C(=O)NCc2ccsc2C(=O)NCC2CCN2C(C)(C)C)cccc1F 14546,c1(C(N(C)CCNC(c2ccc(N)c(Cl)c2)=O)=O)nsc2ccccc12 14547,c1(CN(C(CC(=O)NCC)=O)C(C)C(C)(C)O)cccc(C)n1 14548,O=C(CCC(CF)CF)N1CCC(CO)C(NC(C2(c3ccno3)CC2)=O)C1 14549,C(CCN(C)C(C1CCC1(C)C)=O)(C(C)(C)C)NC(C(C)NC(C)(C)C)=O 14550,N1(C(C=CC(N2CCOCC2)=O)=O)CCCC2C1CCCN2C(=O)C1=CCCCO1 14551,c1(C(=O)NC2COCCN(C(C(CC(=O)OC)C)=O)C2)cnn2ccncc12 14552,c1(C(N2CC(CNC(CSCCOC)=O)C2)=O)nc(N(C)C)nc(=N)[nH]1 14553,C1(NC(CCc2ccc(C)o2)=O)CC(O)CN(C(=O)CSCc2ncc[nH]2)C1 14554,Cc1ccc(C)c(C(N2CCN(C)C(C(N3CCC(OC4CC4)C3)=O)C2)=O)n1 14555,c1(CCC(N2CCC(CNCc3c(C)ncs3)C2)=O)ccc(NC(=O)OC)cc1 14556,c1(OCC(N2CCC(NC(=O)C=CSc3nc[nH]n3)C2)=O)cccc(Cl)c1 14557,CCCN=C(NCCN1CC(C)CC(C)C1)N1CCC(COC)C1 14558,c1(C(=O)NCCN(C(c2cnn(C(C)C)c2Cl)=O)CC)cc(C)n(C)c(=O)c1 14559,C1(C)(CC)CC(C(N2CC(N(C(=O)CCc3cc[nH]n3)C)C2)=O)C1 14560,c1(C(=O)NCCN(C(C2CC(OC)C2)=O)C)cccc(C#CC2CC2)c1 14561,C1(O)(CCNC(C2CCCN(CCC)C2)=O)CCCN(C(=O)COC(C)C)C1 14562,c1(C(=O)NCC(CNC(CCCCC#C)=O)(C)F)ccc2cccnc2n1 14563,CC(C)CC(C)(CNC(C1(CF)CC1(F)F)=O)NC(c1cc(CCO)on1)=O 14564,C1(C(=O)NCC(C#C)CC)(CNC(C2CCCN2C(C)=O)=O)CC2(CC2)C1 14565,N1(C(CCCCC)=O)CC2CCC(C1)N2C(C1(F)CCOCC1)=O 14566,C(=O)(C1SCCc2sccc21)N1C2(C(=O)NCc3nc(C)[nH]n3)CCCC2CC1 14567,N1(C(CCCOCCSC)=O)CCN(C(=O)C(C)OC2COC2)CC1CC1CC1 14568,c1(C(N2C(C(=O)OCC)CCCC2)=O)cc([N+](=O)[O-])c2nsnc2c1 14569,c1(OC)cc(NC(C2CNC(=O)CN2C(=O)CC(C)O)=O)c(Br)nc1Br 14570,CC(C)CCCCCC(=O)NC(C1CC(NC(=O)C(O)CC23CC(C2)C3)C1)C 14571,c1(C(=O)NCCC(C)NC(C2CCC(N=[N+]=[N-])CC2)=O)c[nH]c2cc(O)ccc12 14572,Cc1cc(Br)cnc1C(N1CCCC1CC1CC1)C(=O)NCCC#N 14573,C(=O)(C(F)CCC(C)C)NC(CCC)CNC(=O)C(=O)NC(C)C 14574,c1(SC)ccc(C=CC(=O)NCCC(C(C)C)NC(=O)C(O)CCC)s1 14575,Cc1ccc(F)c(CNC(C2CCC(NC(c3cnc(Cl)c(Cl)c3)=O)C2)=O)c1F 14576,C(=O)(C(F)C(F)(F)F)NC(C1N(C(c2cc(CC)ncc2)=O)CCC1)C 14577,CCC(CCCO)NC(c1sccc1CNC(=O)CC(C)N(C)C)=O 14578,N1(C(COC)=O)CC(C)(C)CCC1CNC(=O)CS(=O)(=O)CC1CCCO1 14579,Cc1cnccc1C(C(=O)NCC(C)C)N(CC(N1CCCCC1)C)C 14580,N1(C(c2cnc(C)s2)=O)CC(NC(c2cc(C)c(Br)o2)=O)CCC(O)C1 14581,c1(OCCCC(=O)N(C2CCCN(C(C(CC)(C)F)=O)C2)C)ccc(F)cc1F 14582,N1(C(C(CN(C)C)(C)C)=O)C(C(=O)NC2CCN3CCC2C3)C2CC(O)C1C2 14583,C1(NC(C(F)=CCC)=O)CCC(NC(=O)CCCC2CCCC2)C1 14584,C#Cc1cccc(C(=O)N(CC(C)O)CCNC(=O)CCC2(C#N)CCC2)c1Cl 14585,C1(CC)CCCN(C(=O)CNC(=O)C=Cc2cnc(C)s2)CC1 14586,N1(C(c2c(OC)cncc2)=O)CC2(CC(NC(=O)CSC(C)C)c3nccn32)C1 14587,C(=O)(CCC(F)(F)F)N1CC(NC(CN2CCC(C)C2)=O)C(CC2CC2)C1 14588,C1(CC(=O)NCC2C(C(=O)NCC3(C(C)(F)F)CC3)COC2)CCCCCC1 14589,CC1CCC2(CN1C(=O)NCCCn1ccccc1=O)OCc1ccccc12 14590,C=CCCN=C(NCCC(CCC)OCC)NC1CCOC(C2CC2)C1 14591,C1(NC(c2c(CC)ncs2)=O)CCN(C(c2cc(Br)n(C)n2)=O)CC1 14592,N1(C(CN(C2CC2)CC)=O)CCN(C(c2cc(O)cs2)=O)CC1COC 14593,CC(C)(C(=O)NCCC(C)(C)NC(C1CCN1S(C)(=O)=O)=O)C1CCCO1 14594,C(=O)(C(CC(F)F)N(C(=O)C=NOC)C)N(CC)CC 14595,c1(CC(N2CC(C)(C(=O)NC(C(=O)NC)C)C2)=O)c[nH]c2cc(OC)ccc12 14596,c1(C(=O)NCCN(C(c2ccc(SC)o2)=O)CC)n[nH]cc1I 14597,C=C1CC2CC1CN2C(=O)CC1CC(C)N(C(c2cnn(C)c2C=C)=O)C1 14598,n1(CCCC)nc(C)c(C=CC(=O)NCc2cccc(C#N)n2)c1C 14599,c1(CN2CCC(O)C(F)C2)ccc2nn[nH]c2c1 14600,C=C(C)C1CCC(C)C(c2nnnn2CCC)(NCc2ccc3c(c2)CCO3)C1 14601,N(C(=NCC(C)C)N1CCCCC(C)(F)C1)CC1(OC(C)C)CCOC1 14602,C1(NC(C2C(N)CCC2)=O)CCCC(F)(F)C1 14603,c1(C(=O)NCC2CCN(C(C(C)SC)=O)C2)sc2ccccc2c1Br 14604,CC(C)CC(C)(C(N)=O)NC(c1ccc(CNC(C2CCC(=O)O2)=O)nc1)=O 14605,Cc1cc(=O)oc(C)c1C(=O)NCCCCCN(C)C(c1c(C)cnnc1O)=O 14606,C1(NC(C2(OC)CC2)=O)CCC2CCN(C(c3c(C(F)F)cccc3N)=O)C1C2 14607,c1(CC)cc(C(=O)NC2CC(CNC(=O)COCc3cc(C)no3)C2)c(C)o1 14608,CC1CCC(NC(C2(C)CC(=O)C2)=O)CN1C(c1ccc(F)c(CO)c1)=O 14609,C1(C#N)(C(N2CC(C(C)NC(c3cc(C4CC4)on3)=O)OCC2)=O)CCOCC1 14610,Cc1ccnc(N2CCC(CNC(c3ccc(F)cc3F)=O)C2)c1[N+](=O)[O-] 14611,Cc1cnc2n1CCN(C(=O)C(C)(C1CC1)N(C(=O)CCc1cn(C)nn1)C)C2 14612,C(=O)(C1=CC2CCCC12)NC(=O)CNc1cc(F)ccc1Cl.CC12CCN(C1)C2 14613,c1(OC)ccc(CCN2CCOC(Cn3ccnn3)C2)cc1 14614,C(c1cncc(O)c1)=CC(=O)NCC(CNC(c1cc(OC)ncn1)=O)O 14615,CCC(CC(=O)N(C)CCC1CCCCN1C(C1CCC(CC#N)CC1)=O)SC 14616,CC(C)C(F)(F)CC(=O)NC(C)(CNC(c1ccc2n[nH]cc2c1)=O)C1CCC1 14617,CC1(C)C(NC(C2CC(F)(F)C2)=O)CC1CC(=O)NCC1CCC(F)(F)C1 14618,Cn1nccc1C(=O)NCC(O)CNC(c1cc(-c2ccncc2)[nH]n1)=O 14619,CC1CC2CC2CC1C(=O)NCC1CN(C(c2cccc(Cl)c2Cl)=O)CCCO1 14620,C=C1CCN(C(C2CC3(CC3)CO2)=O)C(C(=O)NCc2cn(CCO)nn2)C1 14621,N1(C(C2(COC)CC2)=O)CCCC(C2CCN(c3cc(O)nc(=O)n3C)CC2)C1 14622,c12cc(Cl)cnc1NC2=O.C1(C)C(=O)NCCCOCCOCCN1C.CC 14623,c1(C(c2cc(Br)co2)NC(c2nnnn2-c2ccccc2)CF)ccc[n+]([O-])c1 14624,N1(C(C(CC)n2cncn2)=O)CC(NC(=O)CC2CCN(CCF)CC2)C(O)C1 14625,C(=O)(CCC(=O)NC(=O)CN(C)C(=O)C1CC1)NCC(C)CCOc1cc(C)on1 14626,C(C)(C(=O)NCC1(CN(C2(CC(=O)OCC)CC2)CCC)CC1)NCC 14627,c1(C(C(=O)NC2CC(NC(=O)Cc3cnn(C(F)F)c3)C2)O)ccc([N+](=O)[O-])cc1 14628,C1(C(N2CC3C(CN(C(Cc4ccc(C)s4)=O)C)C3C2)=O)CC2OC(=O)OC2C1 14629,C12(C(N3C(CC(NOCC(N)=O)=O)CCC3)=O)CCCC1C2(F)F 14630,Cc1ccc2nc(C(N3CC(O)CC3CNC(C3(C)CC=CCC3)=O)=O)cn2c1 14631,C(=O)(CC(CC)C(C)(C)C)NC(C(CO)NC(C(C=C)O)=O)C 14632,N1(C(c2cn(C(C)C)nn2)=O)CC2=C(C1)CN(C(C1(C3CCCO3)CCC1)=O)C2 14633,C(CNC(C1CC2(CSC2)C1)=O)(CC(F)(F)F)NC(C=NOC)=O 14634,CC(C)(C)C(CO)C(=O)N1CCCC1CCNC(=O)CC1C=CCC1 14635,C12(CNC(CCOCCC)=O)CCCCC1N(C(=O)CCc1cn[nH]c1)CC2 14636,C(C)(C(=O)Nc1scc(C(=O)NCc2ccc(O)cc2C)c1)(C(C)C)OC 14637,C1(CNC(c2ncn(CC)c2)=O)CCCCN1C(=O)CCn1ccnn1 14638,N1(C(c2ccc(C#C)cn2)=O)C2CCC1CN(C(c1ncc(OC)cc1F)=O)C2 14639,C12(COC)CC(CNC(C3C=CCC3)=O)(CN1C(c1ccccc1C(F)F)=O)C2 14640,C1(NC(c2scc(COC)c2)=O)CN(C(=O)CC(C)F)C2(CCCCC2)C1 14641,C1(OC)CCCCC1NC(=O)CC1CCN(C(C2CCNC2=O)=O)CC1 14642,O=S(CC(F)(F)F)N1CCCC(S(=O)(=O)NCc2nnc(-c3cccs3)o2)C1 14643,CN1CCCC(C)(C(=O)N(C)CCN(C(=O)CN2CCCC2)C)C1 14644,C1(CNC(C(C(C)OC)O)=O)CCCN(C(=O)C(F)(F)C2CCOCC2)CC1 14645,N1(CC(=O)NCCOCCNC(C2C(C)CCO2)=O)CCC(O)CC1 14646,c1(C(N2CCN(C(c3c(C)nc(CO)o3)=O)CC2C)=O)cc2cc(Cl)ccc2[nH]1 14647,C#CCCCCCC(=O)N(C(CNC(=O)CC1C(=O)NN=C1C)C1CC1)C 14648,C#Cc1cc(C(N2CCCCC2C2CCN(C(=O)C(O)COC)C2)=O)ccc1Cl 14649,C1(CC(=O)NCCOCC=C)CN(C(c2cn3c(n2)CCC3)=O)CCC1C 14650,C1(C(N2CCCC2C(F)(F)F)=O)CCCN(Cc2ncccc2Br)C1 14651,c1(CC(=O)NC2CN(C(c3c(C)c(N)ccc3)=O)C(C)C2)ccc([N+](=O)[O-])cc1 14652,c1(C(N2CCC(NC(=O)CSCC3CCCO3)C2)=O)c(F)cncc1Br 14653,c1(C(=O)NC(CC)(C)CNC(C2(CCN(C)C)CCC2)=O)cc(C#N)c[nH]1 14654,C#Cc1cccc(C(=O)NC2CC3CCC2(CNC(=O)Cc2cnccn2)C3)c1 14655,c1(SC)ccc(C(N2CC(NC(c3cccc(O)n3)=O)C(SC)C2)=O)c(Cl)c1 14656,CCC(C)(CC(=O)NCCCCCN(C(=O)Cn1cccnc1=O)C)C(=O)OC 14657,S(=O)(=O)(c1cccc(=NCc2c[nH]nc2C2CC2)[nH]1)NC1C(CC=C)CCC1 14658,c1(OC)ccncc1C(=O)NCC1(C(C)NC(c2cc(F)cs2)=O)CC1 14659,C1(OC)CC(C)CN(C(=O)CC(C)CNC(=O)CC2CCOC2(C)C)C1 14660,c1(OC)cc2c(cc1S(=O)(=O)NCC(c1cccc(C)c1)O)C(C)C(C)(C)C2 14661,CC1CN(C(C2(Cl)CC2(C)C)=O)CC1NC(c1ccnnc1O)=O 14662,C#Cc1cnn(C)c1C(N1CC=CC(C(=O)NCC2CCCN2C)C1)=O 14663,C1(C(=O)NCCOCCN(C(CC(CCC)O)=O)C)CCc2nnn(C)c2C1 14664,N1(C(C(C)(C)CO)=O)CC2CC(NC(=O)CCc3cccc([N+](=O)[O-])c3)CC1C2 14665,c1(NC(C)=O)cc(NC(CC(C)C)=O)ccc1Cl.N(C)(S(N)(=O)=O)C(=O)C 14666,c1(CC)ccc(C(c2nnnn2C(C)CC)NCc2nc(C(C)C)nn2C)nc1 14667,C1(C(=O)Nc2cc(-n3cc(C(C)(C)N(C)C)nn3)ncc2)C2C(=O)OCC12Br 14668,N1(C(CNS(NC)(=O)=O)=O)CCCC1(C)CNC(=O)CC1CC(=O)NC1=O 14669,C1(C(N2C(C(=O)Nc3cn(CCOC)nc3)CC2)=O)CC1C1CC1C 14670,c1(C(=O)NCC(C2CC2)NC(=O)C=CBr)cc(Cl)ccc1F 14671,CC(C(=O)NCC1CC(F)CN1C(=O)CC1CN2CCC1CC2)C(C)(C)C 14672,C1(C(=O)NCCC(c2cccc(F)c2)C)CCCCC1NC(C1CCCO1)=O 14673,c1(CC)cccc(C(=O)NC2CC(N(C)C(c3ccc(C(F)F)o3)=O)C2)c1O 14674,c1(N(C2CCCN(C(C)C)C2)S(C)(=O)=O)cc(F)ncc1OCC 14675,c1(C(=O)NCCC2(OC)CN(C(c3c(CC)csc3)=O)C2)cc(C)ncc1C 14676,C12(CNC(C(CC)N(C)C)=O)CCC(CC1)N2C(c1nncn1CC)=O 14677,Cc1sc2ncnc(NC3CCCC(NC(C4CC45CC(O)C5)=O)C3)c2c1C 14678,N1(C(CN(C(=O)OCC)C)=O)CCN(C(c2sc(C)cc2Cl)=O)CC1CCO 14679,c1(C(N(C(CC)CC(=O)NCCc2ncon2)C)=O)ccc([N+](=O)[O-])[nH]1 14680,S(=O)(=O)(c1cnc(NCC(Cl)(Cl)Cl)c(Cl)c1)NC1(COC)CCCC1 14681,C(=O)(C(CC(C)(C)C)NC(c1cscc1C)=O)NCC(CC(=O)OC)O 14682,N1(C(C2C(C)(NC(c3ccnc(OC)n3)=O)CCCC2)=O)CCN(C)C(=O)C1C 14683,CCC(C)CCC(O)CC(=O)NCCC(C)N(C(=O)C(C)(C#N)CC)C 14684,C(C1CCCN1C(=O)Cc1nccn1C)=CC(=O)N(C)CC1CCSC1 14685,N1(C(c2cc(C(=O)OC)cc(O)c2)=O)CCCC2(CC=CCO2)C1 14686,N1(CCC)CCC(N=c2[nH]c(=N)[nH]c(=NCC3CCCN3Cc3cccs3)[nH]2)C1 14687,c1(C(N(CCC(C)NC(C2CC(N(C)C)C2)=O)C)=O)cc(CO)[nH]n1 14688,C1(NC(c2c(C)cc[nH]2)=O)CC2CC(NC(C3CC(=O)N(CC4CC4)C3)=O)CC12 14689,c1(C(N2CCOCC(NC(=O)CC3CCCC4CC34)C2)=O)cnc2occc2c1 14690,C#CCC(CC(=O)NCCc1csnn1)NC(=O)Cc1cnns1 14691,c1(CC(=O)NCCCCCNC(C2CC2C(F)(F)F)=O)cc(O)cc(Br)c1 14692,Cc1nn(C)c(C)c1CC(C)C(N1CCC(C(C)NC(c2cncs2)=O)CC1)=O 14693,C(C1CN(C(C2OCCC2C)=O)CC1C(=O)NCc1cscc1C)=CC 14694,C(C(C(F)(F)F)OC)NC(c1scc(CNC(C(C)OCCCC)=O)c1)=O 14695,C1(C(N(CC(C)N(C(=O)Cc2cncn2C)C2CC2)C)=O)C2C3CCC(C3)C12 14696,C(=O)(C1=CCC(C)(C)CC1)NC1CN(C(c2ccn(C)c2)=O)C(CO)C1 14697,C(=O)(C(C)C(O)C(C)C)NC(CNC(CN(C1CC1)CC)=O)Cc1ccccc1 14698,c1(OC)cc(C(=O)N(CCC(C(C)C)NC(C2CCO2)=O)C)c2c(c1)CCCC2 14699,c1(CCC(=O)NCCOCCN(C(=O)CNc2ncccn2)C)ccc(Cl)cc1 14700,c1(OC)ccc(OCC(=O)N(c2cccnc2)C(c2nccc(Br)n2)C2CC2)cc1 14701,Cc1c(C(N2CCCCC(NC(=O)Cc3ccns3)C2)=O)[nH]c2c1C(=O)CCC2 14702,C1(C)(C(=O)NC(C)CC2CN(C(=O)Cn3cnc(=N)[nH]3)C2)CCC(C)(C)CC1 14703,N1(C(c2cccc(F)c2)=O)CCC2(CCN(C(=O)OCc3ccccc3)CC2)C1 14704,C#CC1(C(=O)N(C(CCO)C(F)F)C)CCN(C(c2cnn(CC)c2)=O)C1 14705,CC1=C(C(=O)NCC(C2CCCC2)NC(C2CCC(C)NC2=O)=O)CCC1 14706,C1(OC)CC(NC(=O)C(CC(C)C)OC)CN(C(C2CCCCC2O)=O)C1 14707,C(c1ccc(C2CC2)cc1)=CC(=O)NC1CCCCC1NC(C1CC1C(F)F)=O 14708,c1(C(=O)NC2C(OC)CN(C(C(F)OC)=O)C2)ccn2cncc2c1 14709,CC1=C(CC(=O)Nc2c(Cl)ccc(Cl)c2Cl)c2ccccc2C1 14710,C(=O)(CCCC(C)(C)C)N1CC(C)(CNC(c2c(C)n(C3CC3)nc2)=O)C(C)C1 14711,CC1(C)CC(NC(c2cccc(C(N)=O)n2)=O)CN1C(c1ccc(Cl)cn1)=O 14712,C(=O)(CC(C)(C)C(=O)NCC1C2CN(C(=O)C(C)OCC(C)C)CC12)OC 14713,N1(C(COC(CC)C)=O)CCOC(C)(CNC(=O)CN2CC(C)(C)C2)C1 14714,C1(NC(c2c(C)noc2N)=O)CC2(C1)CN(C(=O)C(c1cccc(Cl)c1)(C)C)C2 14715,CC(C)(C)CC(O)C(=O)NCCCCCNC(C1CCCCC1C(C)(C)C)=O 14716,c1(OC)nccc(C(=O)N(C)CCNC(C2CCCN2C)=O)c1Br 14717,C(=O)(CCCC#CC)NCC(CC=C)NC(=O)C=CC(c1ccccc1)=O 14718,N1(C(C(CC)OCC)=O)CC(NC(C2(N3CCOCC3)CC2)=O)CC1(CC)CC 14719,Cc1cc(C(N2CCOC(C(C)NC(C3(C#N)CC3C(F)(F)F)=O)C2)=O)nn1C 14720,C(=O)(CC(F)(F)C(C)(F)F)N(C1CCN(C(=O)C(C)(C)C)CC1)CC 14721,N1(C(CC(CC(C)(C)C)O)=O)CCc2sccc2C1CNC(C1CC(F)(F)C1)=O 14722,c1(C(=O)NC(C)CC(C)NC(=O)COc2ccccc2F)cc(N)cc(N)c1 14723,C(CCN=c1[nH]ccc(=NC2CC3(C2)CC(C)(C)C3)[nH]1)c1cnn(C)n1 14724,C(c1ccc(OC)cn1)=CC(=O)NC1(C)CCN(C(C2(COCC)CC2)=O)C1 14725,N1(C(CN2CC(=O)NCC2)=O)CCC(C2CC2)C1CNC(c1ccn(CCF)n1)=O 14726,CC(O)(CC(=O)N1CCCCC1CNC(c1cc(Br)sn1)=O)C(F)(F)F 14727,C1(NC(C2CC(C#C)(O)C2)=O)CCSC12CN(C(C1C(C(=O)OC)C1(C)C)=O)C2 14728,c1(CN2C(CCC(=O)Nc3ncc(Br)cc3I)CCCC2)cc(F)ccc1Br 14729,S(=O)(=O)(c1ccc(C)c(C)c1)NCCC(=O)NCCNC(c1c(SC)cnn1C)=O 14730,c1(NC(N2CCOC(C(F)F)C2)=O)ccc(-c2cnco2)cc1 14731,N1(C(C2C(=O)NCC2)=O)CC2CN(C(=O)C=CC(F)(F)F)CC(C1)O2 14732,c1(C(=O)NC(C(C)NC(c2ccc(F)cn2)=O)(C)C)cn2cc(Cl)cc(Cl)c2n1 14733,Cc1cc(C2CC2)ncc1C(=O)NCC1(C)CC(NC(C2CC2OC(C)(C)C)=O)C1 14734,c1(OC)cncc(CCC(=O)NCc2ncoc2CCNC(=O)C(CC)OC)c1 14735,N1(C(c2c(C)ccs2)=O)CCC2(NC(=O)C(c3ccc(Cl)s3)=O)CC2C1 14736,C1(C(=O)NC2CCCC(CC(=O)N(CCCCCO)C)C2)(CC)CCNC1=O 14737,C#CC1CC2CCC1N(C(C(=O)OC)C(C)CC1CCOCC1)C2 14738,CC(C)(C)C(O)CONC(=O)CC1(NC(C2CC3CCC3C2)=O)CCCCC1 14739,C(=O)(C(O)CCCNC(=O)N(C(C)C)Cc1ccc(Br)cc1)OC 14740,C(CC(=O)NCC1CC1Cl)(C(F)F)NC(C1(Cl)C(C(C)=O)C1)=O 14741,C1(CCC(=O)NC23C(CN(C(C(C=C)(F)F)=O)C2)C3)CCc2ccccc2C1 14742,C1(S(N)(=O)=O)(C(=O)NC(CCCC)CNC(=O)CNC(=O)C2CC2)CCCC1 14743,N1(C(C2C(C)OCCC2)=O)CCOC2(CCN(C(=O)Cc3cnccc3Cl)C2)C1 14744,N1(C(c2c(C)nc(CNC(C3CC(F)C(=O)N3)=O)o2)=O)CCN(C)CC1C1CC1 14745,N1(C(C2C=CC(NC(C(CN(C)C)O)=O)C2)=O)CCC(O)CC1C1CC1 14746,C#CCC(C)(C(=O)Nc1cc(CO)ccc1C)NC(c1ccc(OC)nc1)=O 14747,c1(C(=O)NCC(CC=C)NC(=O)CNC(c2cccs2)=O)cc([N+](=O)[O-])oc1C 14748,c1(OC)ccc2c(C)c(C(=O)NC(c3ccc(-c4ccncc4)cc3)C)oc2c1 14749,O=C(C1CCCn2cnnc21)N1CC2(CNC(=O)C(O)C3CCC3)CCC1CC2 14750,CC(C)(C)C(CNC(c1ccc2nccn2c1)=O)C(=O)NC1(CO)CC(F)(F)C1 14751,CC(CCCC(=O)NCC1(C#N)CCC1)NC(c1ccc(F)c(O)c1)=O 14752,Cc1nccc(C(=O)NC2(C(=O)NCc3ccc(Cl)cc3)CCN(C)C2)n1 14753,C=CCCCC(=O)NC1(CNC(=O)CCN2CCCC(C(N)=O)C2)CCOC1 14754,Cc1ccc(C)c(CC(=O)NC(C)C(C)NC(c2ncccc2C)=O)c1 14755,N1(c2nnc(COC)s2)CCCC(C2CC2NC(c2ncc3ccccn23)=O)C1 14756,Cc1ccc(CN2CCC(O)(CC(=O)NCCC(C)CO)CC2)c(F)c1F 14757,Cc1ccc(S(=O)(=O)NCc2ccnn2CCN2CCOCC2)c2nccnc12 14758,C=CCC(C)(CC)C(=O)N1CCC(COC)(NC(=O)C2=COCC2)C1 14759,c1(NC(c2c(C)nccn2)C)nc(N2CC3CCC3C2)nc2c1ncn2C(C)C 14760,c1(Cc2n(C(COC)C)nc(-c3ccc(Cl)s3)n2)cccc(C#CC2CC2)c1 14761,CC(C(=O)NCC1CC(NC(c2cc(C(C)(C)O)on2)=O)C1)C(C)(C)C 14762,C1(C(N2CC(CC=C)(C(=O)N(CCCOC)C)C2)=O)COC(=O)N1C 14763,CSC1=C(C(=O)NCC2CC3CC3N2C(=O)C(C)(O)CC(C)C)CCCC1 14764,c1(C(=O)NC2C(NC(=O)Cn3cc(C4CC4)cn3)CCCC2)c(O)ncnc1O 14765,c1(C(N2CCC(N(C)C(C3CC3C(N)=O)=O)C2)=O)cccc2nscc12 14766,N1(C(C(C(C)C)SC)=O)CCN(C(=O)CCn2ccnc2)C(CF)C1 14767,N1(C(CNC=O)=O)CCOC2CN(C(c3cccc(C4(F)CC4(F)F)c3)=O)CC12 14768,C(=O)(CCC(=O)NCC1(NC(C2SCC=C2C)=O)CCCCC1)OC 14769,c1(OCC)ccc(NC)cc1.C12CCCN1C2=O.C(=O)(C(F)F)N 14770,CCCCN=C(NCc1nn(CC)cc1Br)NCc1cccnc1OC 14771,c1(C(N(C(C)C)CCNC(=O)CNC=O)=O)cc2n(n1)CCN(C)S2(=O)=O 14772,c1(OC(C)C(=O)NC(CNC(=O)C=Cc2cnc[nH]2)CO)ccc(F)cc1 14773,n1(CC(=O)NC2CCC2NC(=O)CC2(CO)CCCCC2)nc(O)ccc1=O 14774,c1(OC)cn(C)c(C(=O)NC(C)(C)CNC(=O)C(F)CC2CCCCC2)cc1=O 14775,N1(C(c2c(CC)c(C)sc2)=O)CCN(C(=O)C(C)(C)CC)CC1CS(C)(=O)=O 14776,C1(C(=O)NCC2CCN(C(=O)C(c3cccc(C)c3)C)C2)(CC)CCCCC1 14777,N1(C(c2ccc(C)o2)=O)CCCC(O)(CNC(=O)CN2CCCC2=O)CC1 14778,C1(C(=O)NCC2(OC)CN(C(C3(F)CCOC3C)=O)C2)C2CCC1(C)C2(C)C 14779,c1(C(=O)NCCC(C)N(C(CCCC(=O)OC)=O)C)cccc2c1CCO2 14780,CC1=C(C(=O)NCC(CNC(=O)C(C)(C)C2CCOCC2)OC)C(=O)OC1(C)C 14781,C1(C(=O)NCCCNC(CNC(CNC(C2C(C)C2)=O)=O)=O)CCCCN1N=O 14782,C1(C(=O)NCc2cc(C(N(CC(COCC)O)C)=O)ncc2)C2C3CCC(C3)C12 14783,N1(C(C=CCOC)=O)CC(NC(=O)CC(C)C(C)(C)CC)C2(CCOCC2)C1 14784,C1(NC(CCCCC)=O)CC(F)(F)CC1NC(=O)COc1nn(C)cc1Br 14785,C(CC(C)(C)C(=O)NCCC(C(C)C)NC(C12CCC(CC1=O)C2)=O)OC 14786,c1(C(N(C)CCNC(C2CC(=C3CCC3)C2)=O)=O)cc(Br)ncc1F 14787,CCCCCC(=O)N(CC(C)N(C)C(c1ccc(Br)cn1)=O)C 14788,O=C1CC(C(N2CC3CC2(c2cn(CC(F)(F)CO)nn2)C3)=O)C12CCC2 14789,C1(NC(Cn2ncc(C)c2)=O)CCN(C(=O)CCc2cccnc2F)CC1C(N)=O 14790,Cc1ccc(F)cc1C(=O)NC1C2CC3C(C2)C13C(=O)NC1CN2CCC1CC2 14791,C1(CNC(C2N(C(c3c(C(C)C)noc3)=O)C(C)C2)=O)C(C)(C)C1(F)F 14792,N1(C(c2onc(CC)n2)=O)CCC2CN(C(=O)CC3CC4CCC3O4)CC12 14793,N1(C(c2cc(OC)c(Cl)cc2)=O)CCC2(CCN(c3cc(C)ncc3C#N)C2)C1 14794,C1(N(C(CN(C(COCCCC)=O)C(C)C)=O)C)CCCC(C)(C)C1 14795,C(CCN=c1[nH]c2c(c(=NCc3csc(C(C)C)n3)[nH]1)COC2)(C(C)C)OCC 14796,c1(C(=O)NC2CN(C(Cn3c(C)csc3=O)=O)CC2C)cnc2ccc(F)cn12 14797,N1(C(c2ccc(OCCO)cc2)C(=O)NC(CC)(C)C)CCOC2(CCCCC2)C1 14798,N1(C(c2c(C)onc2)=O)CCC(NC(c2cc(C)c(C)nc2C)=O)C12CCCC2 14799,C1(F)(CNC(CN(C)C(c2cccs2)=O)=O)CCN(C(C2(C)CC3CC3C2)=O)CC1 14800,C1(CC(=O)NCC2CCCCCN2C(=O)CN2CCCC2)CS(=O)(=O)CCO1 14801,C12CN(CC1C1CC1)C2=O.C1(NC(C=C2CCN(C)C2)=O)(CO)CC(C)(C)C1 14802,c1(-c2scc(C(=O)NC3CNCCC3(F)F)n2)cc(F)c(F)c(F)c1 14803,C1(S(C)(=O)=O)(C(N2CCCC(CN=c3nc(CC)[nH]s3)C2)=O)CCCC1 14804,C12(C(N3CCC(N(C)C(C4CC=CCC4)=O)C3)=O)CC(C#N)(C1)C2 14805,c1(OCC)ncccc1C(=O)NC12CC1CN(C(c1ccn(C(F)F)n1)=O)C2 14806,C1(C(N2CCCC(NC(c3c(C)cc(Br)o3)=O)C2)=O)CCCC(=O)N1C 14807,CC1CCN(S(=O)(=O)CC(=O)N(CCCN(C(=O)CC2(CO)CC2)C)C)CC1 14808,C(C)(CCN=c1[nH]c(Cl)nc(C(C)C)c1C#N)NC(C(COC)(C)C)=O 14809,c1(NC(CC(C)SC)=O)cccc(C(C)NC(=O)CN(C)C2CC2)c1 14810,N1(C(c2c(CC)csc2)=O)CCC(C)C(N(C)C(c2csc(N(C)C)n2)=O)C1 14811,C(=O)(C(C)CNC(C1CC1(C)C)=O)N1CC(CSC)C1 14812,c1(NC2CCN(C(C(C(C)(C)C)NC(C)=O)=O)CC2)nc(C)c([N+](=O)[O-])cc1Cl 14813,N1(C(C2CN(C)C(=O)N2)=O)CC2CCC(C(=O)NCC(C)(C)CO)(C2)C1 14814,C1(CNC(c2cc3cc(Br)sc3[nH]2)=O)CC2(CCOCC2)CN1C(=O)CO 14815,C(CC(=O)N(C1CN(C)C1)C)(C(F)(F)F)NC(C(CC(C)C)O)=O 14816,C1(CCOC)(NC(c2ccsc2Cl)=O)CCN(C(C2OCCC2C)=O)C1 14817,N1(C(C=C(CC)CC)=O)CCC2(CC1)CN(C(c1cnc3n1CCC3)=O)C2 14818,C1(CNC(c2n(CC)ccc2)=O)CN(C(C2CCCCS2)=O)CC(C)(C)O1 14819,N1(C(CCN(CC)CC)=O)CC(CNC(=O)CCC(C)(C)F)CCC1C 14820,C1(C(=O)NC2CC(c3ccccc3)(NC(C=CC=CC)=O)C2)C2CCCOC12 14821,C(=O)(C1=CC2(CCN(C(=O)CNC(=O)C3CC3)C2)C1)N(C1CCOCC1O)C 14822,c1(CN2CCC(NC(C(C)(C)CC(F)F)=O)CC2)cc(Cl)ccc1[N+](=O)[O-] 14823,C(=O)(C(CCC(N)=O)N(C)C)N(CC(=O)N(CCCCCC(=O)NC)C)C 14824,c1(CC)nn(C)c(CC)c1C(=O)NC1CN(C(=O)CC2CC3CC3C2)CC1C 14825,C1(NC(CC(C=C)C)=O)CN(C(=O)CC23CCCN2CCC3)CCC1F 14826,c1(OC)ccc(C(=O)NC2CCN(C(c3c(C)cnn3C)=O)C2C)c(OC)c1 14827,c1(C(N2CCC(CC#C)(C(=O)NC(C)CF)C2)=O)cccc2c1CCC2 14828,Cc1cc(C(=O)NC(CC2CCOCC2)C(N2C(C)CC2(C)C)=O)sc1C 14829,Cc1c(CC(N2CC(NC(=O)Cn3cncn3)CC2C)=O)sc2ccccc12 14830,c1(OC)ccc(Br)c(C(N2C3CCC2C(C(=O)NC24CC(F)(C2)C4)C3)=O)c1 14831,c1(NC)cnncc1C(=O)NC(C)CNC(c1cncn1-c1ccc(Cl)cc1)=O 14832,C1(C(=O)NC23CC2CN(C(=O)C(C)(C2CCOCC2)OC)C3)(OC)CCCCC1 14833,C(c1cccc(F)c1)=CC(=O)N(CCCNC(C1(C)CC2CC2C1)=O)C 14834,c1(C(=O)NC(C(C)C)CNC(=O)C=CCF)cc2cc(Cl)cnc2[nH]1 14835,CC1CCC(C)(C)N1C(C1CN(C(=O)CSCC(F)F)CC1(F)F)=O 14836,C1(C#N)(C(N(C)CC2CCCC2NC(c2ccc(F)cn2)=O)=O)CC12CCC2 14837,Cc1ncn(C)c1C(=O)NOCc1cn(CC2CC(F)(F)CO2)nn1 14838,N1(C(C(CCC)C)=O)CC(NC(c2cnc(N(C)C)c(Cl)c2)=O)CC2(CCC2)C1 14839,CC1(C)CC=C(c2ccc(NC(C3(O)CC3)=O)cc2F)CC1 14840,CCC(CC)C(C)C(=O)N(CC(=O)N(C1CC(O)C1(C)C)C)C 14841,c1(CC(=O)NC(c2nocc2C(N2CCC(C)C2C)=O)C)ccccc1C 14842,c1(C(=O)NC(C)CCN(C(=O)CCC2CCCCO2)C)ccnc2ccsc12 14843,C=C(C)C1OCCC1C(=O)NCCCN(C(=O)COCCCF)C(C)C 14844,c1(C(=O)NCCCN(C(C2CCCN2C2CC2)=O)CC)cnn(C(C)C)c1C 14845,CC(C)(CCC(=O)N1CC(NC(C2CCC(CN(C)C)O2)=O)C2(CC2)C1)[N+](=O)[O-] 14846,Cc1ccnc(O)c1C(=O)N(C)CC1CCN(C(=O)C(c2cnn(C)c2)C)C1 14847,c1(C(=O)NC2(CC)CCCN(C(C3(O)CCOC3)=O)C2)ccc2c(c1)COCC2 14848,C(=O)(CC1OCCc2sc(Br)cc21)N1C(C)CC(Nc2ncn(CC)n2)CC1C 14849,CC1OCCC1N=c1[nH]c(N2CCC(C)(C)C2)nc2ccccc12 14850,C1(NC(=O)CC2CSCCS2)CCCC(CNC(c2cc(F)c[nH]2)=O)C1 14851,c1(C2N(C(c3cc(C4CC4)no3)C(=O)NCCOC)CCC2)cccc(Cl)c1 14852,c1(C(N2CCC(OCCNC(C3C(OC)C3)=O)C2)=O)ccncc1Cl 14853,Cc1cnc(NC(C(C)C)C2CCC2)c(S(=O)(=O)NCCCCS(C)=O)c1 14854,c1(OC)ccncc1C(N1CC(O)(C(F)C(=O)NCc2nccnc2C)C1)=O 14855,c1(OC)ccc(C(N2CCN(C(=O)C(C(C)C)OC)CC2CCO)=O)nc1Cl 14856,C1(C=O)CC2(CC2)CN1C.N1(C(C(C)NCCC)=O)CCC(C(C)(C)O)C1 14857,c1(NC(C2CC3(CN2)CC3(F)F)=O)cncc2cc(Cl)ccc12 14858,CC1(C(=O)NCC2(O)CN(C(c3ns[nH]c3=O)=O)C2)Cc2ccccc2NC1=O 14859,c1(NC)ccc([N+](=O)[O-])cc1C(=O)NCC1CCCN1C(C1(CF)CC1)=O 14860,O(C1CCCc2ccccc21)CCCC1(C#N)CCOCC1 14861,C1(C(=O)NCC2C(NC(c3c(C)nc(C)o3)=O)CCCC2)CCOC(=O)CC1 14862,CC#CCCC(=O)NCC1CC2CC2N1C(c1cnn(C2CCCC2)c1CC)=O 14863,CCC(C)C(O)C(=O)NCCCCCN(C(=O)C(C)SC(C)C)C 14864,CCC(C)C(=O)C(=O)NCC(C)(F)CNC(=O)CN1CCCCC1C 14865,C1(NC(C2(CC=C)CC=CC2)=O)CC2CC1CN(C(=O)C(C)(C)C(C)(C)C)C2 14866,c1(C(=O)NC(CC(C)C)CNC(=O)C2=CCC2)ncnc2c1c(Br)cn2C 14867,C1(NC(c2c(Cl)cc(C)s2)=O)CCOC12CCN(C(=O)C=Cc1ccsc1)CC2 14868,C1(CNC(C(C)=C2CCC2)=O)CCCCN(C(=O)CC(C)N(C)C)C1 14869,C(=O)(CCCCCC#N)N1CCC(NC(C(C)(O)c2ccccc2)=O)C(O)C1 14870,C1(C(=O)NCC2N(C(c3c(C)n(C)nn3)=O)CCOC2)CC12CCS(=O)(=O)CC2 14871,Cc1cccc(Cn2cc(C3CN(NC(c4cc(F)n(C)n4)=O)C3)nn2)n1 14872,c1(C(=O)NCCC(=O)NC(C#C)CC)c[nH]nc1[N+](=O)[O-] 14873,Cc1ccc(CN2CCC(C)C2CNC(=O)C=CC(C)(C)C)cc1C#N 14874,c1(C(N(C2CCN(Cc3[nH]cnc3C)C2)CCC)=O)cc(Br)ncc1Cl 14875,c1(SC)nc(N2CCOCC2CNC(=O)Cc2cc(C)ccc2C)cc(C)n1 14876,C(N=c1[nH]c(N2CCCN3CCCC3C2)nc2c1SCC2)C1CCC(C)(C)CO1 14877,C1(OC)CC2CN(C(=O)CCCn3ccccc3=O)CCN2C1=O 14878,c1(C2C(C(N3CC(C)(NC(C4(C)CC4F)=O)C3)=O)C2)ccc(Br)nc1 14879,C1(CC(=O)NC2CN(c3cc(C(C)C)ncn3)C(C)C2)CCC(C)(C)CC1 14880,c1(CC(=O)NC(C)(C)COCCCNC(C2CCCS2)=O)cccnc1Cl 14881,C(=O)(CCCC#Cc1ccccc1)NC1C(C)N(C(=O)C2=COCCO2)CCC1 14882,c1(C(N(CC(C)NC(c2c(CC)nn(C)c2)=O)C)=O)ccc(COC)c(F)c1 14883,CC(CC(N)=O)C(=O)NCC1=CCN(C(=O)C(C(C)(C)C)C2CCC2)CC1 14884,C#CC1(NC(=O)C(F)C(C)CNC(c2n[nH]c(=N)[nH]2)=O)CCC(C)CC1 14885,c1(C(C)=O)cc(C(N2CCOCC2CCNC(=O)C=C2CCC(C)C2)=O)oc1C 14886,C(=O)(C(C(C)C)c1cc(C)no1)NCCOCCNC(c1scc(C(=O)OC)c1)=O 14887,C1(N(CCC)C(C2CCC2C)=O)CCN(C(c2ccnn2CCC)=O)C1 14888,Cc1ccc(-c2nc(C(=O)NCC(O)CN(C(=O)Cc3cnsc3)C)cs2)cn1 14889,C(=O)(C(COC)CC(C)C)N1CC2CN(C(CNC(CC)=O)=O)C2C1 14890,C1(NC(c2c(COC)ncs2)=O)CN(C(=O)C=Cc2ccoc2)C2(CCC2)C1 14891,Cc1ccc(C(=O)NCC(O)CNC(=O)CC(C)c2ccco2)c(SC2CC2)c1 14892,N1(C(C=C(C)C2CC2)=O)CC=C(CNC(c2cc(C)cnc2C)=O)CC1 14893,C1(C(=O)NCC23C(CN(C(C4C(C)OCCO4)=O)C2)C3)CC2(C1)CC(O)C2 14894,N1(C(C2(OC)CCOC2)=O)CCC(C(N2CCCC2CF)=O)CC1(C)C 14895,c1(C(=O)NCC2CCN(C(=O)Cc3ccc(F)nc3)C2)ccc2c(c1)C(=O)OC2 14896,S(=O)(=O)(CCC(=O)NC(C1CC2(CCC2)C1)C)NCc1c(OC)ccs1 14897,C(=O)(CC1OCc2ncccc21)NCC1C(C)(C)CCCN1C(=O)C1=CCCC1 14898,N1(C(c2c(C)nn(C)c2)=O)C(C(N2CCOC(C(C)C)C2)=O)CCC12CC2 14899,N1(C(C(CC2CCCC2)NC(C2=NOC(C)C2)=O)=O)CCc2nocc2C1 14900,C1(OC)CC(CNC(=O)CCc2cnc(C)o2)(NC(=O)CCC2CCCCC2)C1 14901,CC1CC(CNC(=O)CCc2cc[nH]n2)CN1C(=O)Cc1cccc(Br)c1 14902,N1(C(c2cc(C)c(N)cc2Cl)=O)C2CCC1C(C)C(NC(=O)C(C)C1CCC1)C2 14903,c1(CC2CCN(c3n(CC)nnn3)C2)cccc2nn(C)cc12 14904,c1(CC(=O)N(C)CC2OCCN(C(C(C=C)(C)O)=O)C2)cc(F)c(C)cc1F 14905,Cc1c(NC(c2cc(I)cs2)=O)cccc1Cl 14906,C1(C(=O)NCC2N(C(C(C(CC)C)O)=O)CC(C)(C)C2)CCOC2(CCC2)C1 14907,C1(C(N2CC(C(C)NC(C3COC3)=O)C2)=O)(OCC)CCCC1 14908,C(=O)(C#CC1CCC1)NC1(C)CC(NC(=O)CCC2CC2(Cl)Cl)C1 14909,C(=O)(C1=C(Cl)CCCC1)NC(C)CCNC(=O)CSc1cnn(C)c1 14910,N1(C(C2CC(OC)C2)=O)CCOC2(CCN(C(=O)Cc3ccccc3Br)C2)C1 14911,c1(C(=O)NC2CCCC(NC(C(CCC)(C)C)=O)C2)ccc2nccc(C)c2c1 14912,c1(C(N(C(C)CNC(C23COCC2C3)=O)CC)=O)cc(F)c(C)cc1O 14913,C(C(F)CC1CC1)NC(=O)COCC(=O)CCOCCCOC1CCC1 14914,C1(C2(O)CN(C(=O)COCCOCCO)C2)(CNC(C(CC)(C)F)=O)CC1 14915,CCCCC(C(=O)N1CC=CCC1C(N1CCC1(C)CCC)=O)N(C)C 14916,c1(C(=O)NCCCOCCCC)ccc2[nH]nc(-c3cnn(C)c3)c2c1 14917,Cc1ccc(=N)[nH]c1C(N1CCCC(CCNC(c2nc(Br)c[nH]2)=O)C1)=O 14918,CC(CS(C)(=O)=O)C(=O)N1CC2(CC(NC(C3SCCS3)=O)C2)C1 14919,N1(C(C(C)(CO)NC(C2CCCSC2)=O)=O)CCC12CCCC2 14920,N1(C(C(C)CBr)=O)CCCn2nc(C(N3CCC(O)C(F)C3)=O)cc2C1 14921,CC(CC(=O)NC1C=CCC(C(=O)NC(C)(CO)C2CCCC2)C1)CC(C)(C)C 14922,C1(NC(c2ccc(COC)s2)=O)CCC(NC(=O)CN(CC(C)(C)C)C)CC1 14923,C1(c2nnnn2C2CCCC2)(NCCC(C=C)(C)C)CCOC(CC(=O)OC)C1 14924,CC1CC(CCNC(=O)C=CC2CCC2)CCN1C(=O)C(=O)NCC(F)(F)F 14925,c1(SC)cc(C(=O)N(C2CCCN(C(C3CCC3(F)F)=O)C2)CCO)c(C)o1 14926,c1(OC(N2CCC(NC(=O)C=Cc3ccco3)C2)=O)cc(C(F)(F)F)c(Cl)cn1 14927,c1(C(N2CC=CC(C(=O)NC(CC)(C)C3CC3)C2)=O)cc(C#N)oc1C 14928,N1(C(c2c(C)cn(C3CCOCC3)n2)=O)CCCC2C1CCN2C(=O)C(O)CF 14929,CC(C)(F)CCC(=O)N1CCC(CCCCCNC(=O)Cc2csc(S)n2)CC1 14930,Cc1ccc(C(C)NC(=O)CN(C(c2csc(C)c2)=O)C(C)C)cc1 14931,S(=O)(=O)(c1cccc(F)c1)NCCNC(c1cc(CC)oc1C)=O 14932,NC(=O)CS(=O)(=O)c1ccc(C(=O)NCCN(CCO)CCO)cc1 14933,C(=O)(C#CC(C)(C)CNC(=O)C(O)C(F)(F)F)NCC1CCN(CC)C1 14934,C1(CNC(CSc2n(C(C)C)cnn2)=O)CN(C(=O)CCCCN(C)C)CC1C 14935,N1(C(c2ccccc2)C(=O)NCCS(C)(=O)=O)CCc2c(F)cccc21 14936,c1(SC)ncc(CNc2nccc(N(C)CC3CCCS3(=O)=O)n2)cn1 14937,N1(C(C2CN(S(CC)(=O)=O)C2)=O)CCCCC(CNC(=O)C(F)OC)C1 14938,C(C(CNC(C1CCCOC1)=O)C(F)(F)F)NC(CCn1c(C)ncc1)=O 14939,N1(C(CCOCC#C)=O)CCCC1(C)CNC(c1ccc(Cl)cn1)=O 14940,c1(CC(N2CCN(CC(C)(C)O)CC2)=O)ccc(O)c(F)c1 14941,C(=O)(C1=CC2CC(C1)CC2O)N1C(=O)CC(COC(=O)C(F)(F)C(F)F)C1 14942,C1(NC(CCc2cncc(OC)c2)=O)CN(C(c2sccc2F)=O)C(C)(C)C1 14943,Cc1ccc([N+](=O)[O-])c(C(N2CC3CC2CN3C(c2cnn(C(F)F)c2)=O)=O)c1 14944,c1(C2CC(C(=O)N(CCO)CCc3ccccc3)C2)ncccn1 14945,C(=O)(C1=CC2CC(C1)CC2O)NCC1N(C(CCSCCC)=O)CC=C1 14946,C1(C(=O)NCCOCCN(C)C)CC2(CCC2)CN1C(c1cn(C)nn1)=O 14947,Cn1ncc(NC(c2conc2C2CCC2)=O)c1-c1cn(C(C)(C)C)nn1 14948,CN1CC2CCN(Cc3cccc4c3COC4)C2C1 14949,c1(CNC(CNS(N)(=O)=O)=O)ccc(CCNC(=O)CCN2CCCC2)cc1 14950,c1(C(=O)NC)cccc(C(=O)N(CCNC(C2CCO2)=O)C(C)C)c1 14951,C1(C(C)=O)CCC(c2nc(-c3ccc(C(F)F)cc3)nn2C2CCSC2)CC1 14952,c1(CNC2CC(C(=O)OCC)OCC2)c(F)ccc(OC(F)(F)F)c1N 14953,c1(N2C(C(=O)NC(CCCC)CO)CC(OC)C2)nc(C)nc2ccccc12 14954,C1(C(=O)NCC(=O)NCCC)CC2(CCC2)CN1C(=O)CNC(C1CC1C)=O 14955,Cc1ccc2ncc(C(=O)NC3CC(NC(c4cnncc4O)=O)C3)c(=O)n2c1 14956,c1(NCC2CCC(C)(CC)O2)cc(=NCc2ccnc(C3CC3)c2)[nH]c(C)n1 14957,CCCCCC(O)C(=O)NCCC(C)(C)NC(=O)CC1(n2cncn2)CC1 14958,C#Cc1ccc(C2CCN(CC(C(C)C)C(=O)NC(=O)O)CC2)cc1.C(C)(C)(C)CCS 14959,C1(C)(OC)CCCN(C(=O)C(C)(C)CCCNC(C2CC(C)(C)CCO2)=O)CC1 14960,C(=O)(CCc1ccco1)N(C(C(C)C(CC)C1CC1)=O)C1CC(n2cccn2)C1 14961,c1(C(N2CCCCC(NC(CCCC(C)C)=O)C2)=O)nccc2c1NCCC2 14962,c1(C(=O)NC2(C)CN(C(C3CC(C)SCC3)=O)C2)cnc2c(ccn2C)c1 14963,C1(CNC(c2ccc(CC)c(CC)c2)=O)CC2(CCC2)CN1C(=O)CC(C)(F)F 14964,CCCC(O)CC(=O)NCC1C2CCC(C2)N1C(c1cnn(CC(F)(F)F)n1)=O 14965,c1(CC)ccccc1-n1nnnc1C(C(C)(C)C1CC1)NC1CCOC1(C)C 14966,c1(C(=O)NC2(C)CCN(C(CCC(C)OC)=O)CC2)cccc2c1OCO2 14967,N1(Cc2ccc(OC)c(Br)c2)CC2CCC1CN2C(c1cocn1)=O 14968,O=C1C=COC2(CCN(C(c3ccc(-c4cn[nH]c4)cc3)=O)CC2)C1 14969,C1(N(C(c2c(CC)n(CC)nn2)=O)C)CCN(C(C2(F)CC=CC2)=O)CC1C 14970,C=CCCCC(=O)N1CC(O)(C2CCCN2C(=O)C=CCCC=C(C)C)C1 14971,c1(OC)ccc(Cl)c(CN2CCCCC2CNC(=O)CC2CCC2)c1 14972,Cc1nc(C)c(C(=O)NC2(CNC(=O)Cn3nnnc3-c3ccsc3)CCC2)s1 14973,N1(C(C(C(C)C)=O)=O)CCC2(CCCN2C(=O)CC2NC(=O)NC2=O)C1 14974,c1(C(=O)NC(CCOC)CNC(=O)C(=O)N(C)C)cccc2c1CCCN2 14975,N1(CC)CCOCC1CC(=O)NCC1(F)CC(NC(c2cccc(CO)n2)=O)C1 14976,CN1CCN(C)CC(C(N2CC(C3CN(C(c4cccc(O)n4)=O)C3)C2)=O)C1 14977,C1(CCN(CCC)C)CCN(C(c2ccc(C(F)(F)F)n2C)=O)CC1 14978,CC1CCCN(C(c2ccc(F)c(F)c2)=O)C1CNC(C1CC(F)(CO)C1)=O 14979,N1(C(CC2C(CNC(C=CC)=O)C2)=O)CC(C2=NOC(C)C2)C1 14980,N1(C(C2(C(C)C)CCN(C(c3cccc(NC)n3)=O)C2)=O)CCC2(CC1)N=N2 14981,C1(C(N(CCC(C)NC(=O)CNC=O)C)=O)OCCC1C(N)=O 14982,c1(N2C(CCCNC(c3cn(CC)nn3)=O)CCC2)cc(C)nc(COC)n1 14983,c1(C(=O)OC)cccc(C(=O)N(CC(O)CN(C(=O)CC2CC(=O)NC2=O)C)C)n1 14984,C1(C(N(CCCNC(=O)CCCN2CCCC2)C)=O)CCc2nncn2C1 14985,C(CCC(N)=O)(C(=O)N(CC)CC1CCC2(CC1)N=N2)n1cc(CC(CC)(C)O)nn1 14986,C1(C(C)C(=O)NCc2ccoc2)CCN(C(c2cocn2)=O)C1 14987,C1(NC(C2C(OCC)C2C)=O)CN(C(c2cnn[nH]2)=O)CC2(CC2)C1 14988,N1(C(c2ccc(C#C)nc2)=O)CC(NC(=O)C(O)CN(C)C)CC2(CC2)C1 14989,c1(N2CCC(Cc3cn(C(C)C(=O)O)nn3)C2)ccnc2ccc(F)cc12 14990,c1(-c2nc(C(F)(F)F)c(Cl)[nH]2)scc2c1OCCO2 14991,N1(C(C(C(CC)C)O)=O)CC2CCCC1C2CNC(=O)C1=CCOCC1 14992,C(CCNC(=O)NC(c1nnnn1C(C)C)CCc1ccccc1)(C(C)C)OC 14993,N1(C(c2cccc(OC)n2)=O)CC(C(=O)NC(c2ccc(F)cc2)C)CC(F)C1 14994,C1(CN(C(=O)C=Cc2cc[nH]n2)C)CCCN(C(C2CCOC(=O)N2)=O)C1 14995,c1(C(=O)NC(CC)CNC(c2ccnnc2O)=O)cc(O)ccc1[N+](=O)[O-] 14996,C12(C(=O)NC3(C)C(C)CCC3)CC(CN(C(c3cccc(O)c3)=O)C1)C2 14997,c1(OC)ccc(F)c(C(N2CC(N(C)C(c3cccc(C#N)c3Cl)=O)C2)=O)c1F 14998,C=CC1(C(=O)N(C)CCC2CCOCC2)CCN(C(c2c[nH]c(=N)o2)=O)C1 14999,c1(-c2n(CO)c(N3CC(O)C(C4CC4)C3)nn2)cncc2c(Cl)cccc12.C1(C)CC1 15000,C#CC(C)CN=C(NCC1CC1)N1CCC(c2ccc(F)cc2)C1 15001,Cc1cnc(-c2noc(C(C3(C)CC3)F)n2)nc1 15002,c1(NCC)ccc(NCc2cc(N3CCOC3=O)ccc2F)cc1F 15003,Cc1nn(C(C)(C)C)c(C)c1C(N1CC=CC(NC(C2(F)CC=CCC2)=O)C1)=O 15004,Cc1cc(F)ccc1NC(=O)C(=O)NCc1cccc(C(N)=O)c1 15005,C1(C(N2CCC(CCc3cn(CCCCCC)nn3)C2)=O)CN(C)CC(C)O1 15006,C(=O)(N=c1ccc(Oc2ccccc2)n[nH]1)Nc1cccc(COC(=N)N)c1 15007,Cc1cccc2cc(C(N3CCC4(C3)CN(C(c3nc(Br)c[nH]3)=O)C4)=O)nn12 15008,C1(CNC(CC(=O)N(C)C)=O)CN(C(=O)C(O)c2ccsc2)CC12CC2 15009,C1(C(=O)NCC2(C)CCN(C(c3ccc(SC)cc3)=O)C2)(COC)CC(F)(F)C1 15010,C1(NC(C2(F)C(C)OCC2)=O)CC2(CCN(C(=O)C=Cc3ccccc3)C2)C1 15011,C1(NC(c2cc(O)cs2)=O)CCC(NC(c2cnncc2O)=O)CC1 15012,C(=O)(C1=CCOC1)NC(C1CCCCC1)CNC(C(C)(O)C1CC1)=O 15013,c1(OC)ccc(CNC(=O)C(c2cc(C)ccn2)N2CCC(F)(CF)C2)cc1 15014,C1(C)(CNC(CCOCCOCC)=O)CCN(C(c2cc3occc3[nH]2)=O)CC1 15015,C=CC1CN(C(=O)CC(C)NC(=O)C(C)OC)CC1O 15016,c1(CCC)n[nH]cc1C(=O)NC1CC(O)C1CC(=O)NCCN1CC=CCC1 15017,N1(C(Cc2n(C)c(S)nn2)=O)CC(NC(C2C3(CC3)C23CC3)=O)C2(CCC2)C1 15018,c1(C(=O)NCCCN(C(=O)C(C)C2CC2)CC)cc(C)ccc1C(C)C 15019,C1(C(N2CCN(CCC#C)CC2)=O)CC2(CCN(C(C3CC3(F)Cl)=O)C2)C1 15020,N1(C(C(CC(=C)C)C)=O)CCC(C2CC2NC(C2(O)CCC(C)(C)CC2)=O)CC1 15021,C1(C)(C(N2CCC3C(NC(CCCC=C)=O)C32)=O)CC(c2ccccc2)=NO1 15022,N1(c2nc(N(C)Cc3ncc(CC)s3)nc(C)c2)CCCc2ccccc2CC1 15023,C1(CC)(NC(C2CCC(=O)C(C)C2)=O)CCN(C(C2CCC(=O)N2CC)=O)CC1 15024,c1(CC)ccccc1OCC(N1CSCC1CNC(=O)Cc1ccnnc1O)=O 15025,c1(C(=O)NC(CN(C(c2cc(=O)n(C)o2)=O)CC)C)csc2ccccc12 15026,c1(C(=O)NC2C3(CCN(C(C=CC)=O)CC3)C2)c[nH]c2ccc(OC)cc12 15027,N1(C(=O)Cn2cnnn2)CCC2CC12C(=O)NC(c1ncc[nH]1)CO 15028,c1(C(=O)NCC(CC=C)NC(c2csc(Br)n2)=O)cc2c[nH]nc2s1 15029,C1(CNC(=O)C=Cc2cccnc2)CC(F)(F)CN1C(c1cc(Cl)cnc1O)=O 15030,c1(CCC)nc(C(=O)NCC(O)C(=O)NCc2ccc(CC)o2)co1 15031,Cc1nn(CC(N2CCC(CO)C(NC(=O)CCNC(=O)CO)C2)=O)c(C)c1Cl 15032,N1(C2CCN(C(C(CC3CC3)OC)=O)C2)CCN(C(=O)CC2CCOCC2)CC1 15033,c1(C(N2C(C)CCC(CNC(c3cnn[nH]3)=O)C2)=O)cc2c(o1)CCCC2 15034,c1(C(N(C(CNC(C(C)NS(C)(=O)=O)=O)C2CC2)C)=O)sc(F)cc1Cl 15035,S(=O)(=O)(CCC(=O)NC(C1CCOC1)CNC(=O)C(F)(F)c1cscn1)NC 15036,CC1(C)CCCC2(CN(C(C3COCCO3)=O)C2)O1 15037,C(=O)(C(C)CC(F)(F)F)NC1CN(C(C(CC#C)C2CC2)=O)CC(F)C1 15038,C(C(C)CN=c1c(C#N)c[nH]c2cccc(I)c12)c1ccc(OC)c([N+](=O)[O-])c1 15039,c1(CC(=O)NCC2CC(NC(CC3CCC(C)CO3)=O)C2)coc2ccccc12 15040,CN1CCCC(CC(c2cccs2)=O)C1=O.c12csc(n1)NC(=O)C2 15041,c1(OC)cc(N)c(C(=O)NC(C2CCCCC2)CNC(=O)COC(F)F)c(F)c1 15042,C(CO)(C(=O)NCC1C=CC(N=O)C1)N.C1(C(=O)C2CC2)CCCN1C(C1CC1)=O 15043,c1(CNC(=O)NC2(c3cccnc3)CCC2)ccc(CN2CCOCC2)cc1 15044,C1(N(C(C2(NC(=O)CC(=O)NC3CC3)C(C)C2)=O)C)CCOC(C)(C)C1 15045,C(=O)(C1CCCn2cnnc21)C(C(C1CCNC1)C)=O.C1(CN)CN2CCC1C2 15046,c1(C(=O)NC2C(C)CCN(C(C3CCS(=O)(=O)C3)=O)C2)cnc2cc[nH]c2c1 15047,C1(CNC(c2ccc3ncccn23)=O)CCCC(F)(F)CC1 15048,CC#CCCC(=O)NC1CN(C(c2cnn(-c3ccncc3)c2)=O)CC1OC 15049,C1(CC)=NC(C)(C(=O)NCCCC(C)(C)NC(C2CCN2C)=O)C(C)=N1 15050,c1(C(=O)NCC(CC(C)C)NC(c2ccc(CO)c(F)c2)=O)ccc(N)c(Cl)n1 15051,C1(C(=O)O)CN(CCC(F)(F)F)C2(CCC2)CO1 15052,C1(C(N2CCN(C(CC(C)(C)O)=O)C(CCO)C2)=O)CC2CCC(C1)S2(=O)=O 15053,c1(C(N2C(CNC(=O)COC(F)(F)F)CCCC2)=O)cnc2sccc2c1 15054,c1(C(=O)NC23CCN(C(c4c(CC)noc4)=O)CC2C3)ccc2c(c1)SCCN2 15055,c1(N(c2ccccn2)C(=O)NCCN2CC3CC3C2)ccccc1 15056,C1(C(N(CCC)CCNC(=O)C(CC)(CC)CO)=O)Cc2cccc(F)c2O1 15057,C(N=c1[nH]c(=NCCn2cncn2)[nH]c2c1SCC2)c1ccccn1 15058,CCCC(C)(C)C(=O)N1CC(CCNC(C2CCC2C(F)(F)F)=O)C(C)C1 15059,N1(C(c2ccnn(C)c2=O)=O)CCN(C(=O)CC(C)(C)C)CC12CC2 15060,C(C)(C)(C(C)(C)CO)NC(=O)OC.N1(C(CN)=O)CCCC(CCC(=O)N)C1 15061,c1(CC)nc2c(C)csc2c(=NCC2CCCN2C(=O)C(C)NS(=O)(=O)CC)[nH]1 15062,CCS(=O)(=O)CC(=O)NC1(C)CCN(c2nnnn2Cc2ccccc2)C1 15063,N1(C(C(CNC(CNC(=O)OC)=O)OC)=O)CCCCCC1OC(C)(C)C 15064,C1(NC(=O)CCCc2cnccn2)CCCCN(C(=O)CC2CCS(=O)(=O)C2)C1 15065,C1(CNC2(CCNC(CCNC(C(C)(C)C)=O)=O)CCC2)C(Cl)(Cl)C12CC2 15066,N1(C(c2cc(CNC(C(CC)NC(N)=O)=O)oc2)=O)CC(F)CC1CO 15067,c1(CN(C)CC)cn(CC2(c3cc(C)on3)CC2)nn1.c1ccco1.C1CC1 15068,CC(CS(C)(=O)=O)C(=O)NCC1(F)CCN(C(c2ccc3ncnn3n2)=O)CC1 15069,C1(NC(CSCC=C)=O)COC2(CCCN(C(c3ccc(N(C)C)cc3)=O)C2)C1 15070,C1(C(=O)NC2CCN(C(C)C)C2)CCN(C(=O)Cc2ccn(C)c2)C1(C)C 15071,S(=O)(=O)(c1c(Cl)cc(Br)cc1Cl)N1C2CN(C(c3c(F)cncc3F)=O)CC21 15072,N=c1[nH]nc(SCC(=O)NCC2CCCN2C(c2ccnn2CCF)=O)s1 15073,C1(CNC(C=CCCC)=O)C=CC(NC(c2ccc(CN3CCCC3)o2)=O)C1 15074,N1(C(CCSCCCC)=O)CCN(CC(C)NC(=O)C(C)C(C)O)CC1 15075,c1(C(=O)NCC(c2ccccc2)NC(C(CSC)OC)=O)ccc(N)c(Cl)c1 15076,N1(C(=O)OC(C)(C)C)CCC(C)(C)C(C(=O)NCc2nc(C3CC3)no2)C1 15077,C(=O)(C1=C(Cl)CCOC1)N1CCC2(C(C(N(C(C(C)C)C)C3CC3)=O)C2)C1 15078,C1(C(=O)NC(CC(=O)NC)C)(NC(C2C(C(=O)OC)C2(C)C)=O)CCCC1C 15079,CC1CCC(NC(=O)COCC(F)F)CN1C(c1cccn(C)c1=O)=O 15080,c1(C(=O)NC2CCCC2NC(C2CCCCC2O)=O)cnc2nccn2c1 15081,C12(OC)CCC(C(=O)NC3(C)CN(C(=O)C(F)(F)C(F)(F)F)C3)(CC1)CC2 15082,N1(C(C2C(C)OCCC2)=O)CC2(CC2)CC1CNC(=O)C1=NNC(C(F)(F)F)C1 15083,c1(C(C(=O)NCCCSC)N(C(CF)CF)C)cncc(Br)c1C 15084,N1(C(c2ccc(C#C)o2)=O)CC2CC(NC(=O)C(C)(C)c3ccc(Cl)s3)CC1C2 15085,N1(C(CCCC(=C)C)=O)CCOC2(C1)CN(C(C1CC(=O)N(CCOC)C1)=O)C2 15086,C1(N(C)C(c2ccc(F)o2)=O)CCCN(C(=O)CC(c2cccc(F)c2)O)C1 15087,N1(C(c2c(C(C)(C)C)noc2)=O)CC2(CNC(C3CC3F)=O)CC(F)(C1)C2 15088,c1(OC)cccc2c(N3CCCC3CNC(C3(CO)CCCCC3)=O)ncnc12 15089,C1(C(N(C(C)CO)Cc2ccccc2)=O)CN(C(C2CCC=CO2)=O)CCO1 15090,N1(C(C(CC)C)=O)C2CCC1CC(F)(CNC(=O)C=C(C)C(C)C)C2 15091,N1(C(C2COCCN(C(C3CN(C(C)C)C3)=O)C2)=O)CCC12CCCOCC2 15092,c1(-c2c(CCC(C)(C)O)scn2)ccc2[nH]c(C(=O)N(C)C)nc2c1 15093,N1(C(=O)NC(c2ccc(NC(=O)OC)cc2)C)CCSC(C)CC1 15094,C1(CC=C)(C(=O)NCc2n[nH]c(C)n2)CCCN1C(=O)CCc1cn[nH]c1 15095,c1(C(C(=O)NCCCOC)N(CC(C)(C)OC)C)cc(NC(C)C)cn1C 15096,N1(C(CC2C(C)C(=O)CC2)=O)C2CC1CN(C(c1ccc(CCF)cc1)=O)C2 15097,c1(C(=O)OCc2nn(C)c(Cl)c2)nc(Cl)c(=O)[nH]c1N 15098,C=C=Cn1ccccc1=O.C(=O)(CCC(C)OCC)OCC 15099,CS(=O)(=O)c1ccccc1-c1ccc2cc(C(=O)NCCCO)[nH]c2c1 15100,N1(C(C(C)OC)=O)CC(F)(F)CC1CCNC(=O)C(C)NC(c1ccccc1)=O 15101,C1(C)(CNC(C2(COC)C=CCN2C(=O)CN(C)C)=O)C(C)(C)C1(C)C 15102,N1(C(C2C(C(C)C)CCC2)=O)C2CCC1C(F)C(NC(c1cc(Cl)cs1)=O)C2 15103,c1(SC)ccccc1C(=O)NC1CC1NC(=O)C(C)(C)CO 15104,C1(NC(=O)CCF)CCN(C(c2ccnn2CC(F)(F)F)=O)CC1CO 15105,c1(C(N2CCC(COCC)CC2)=O)cc2ccc(-c3cccc(F)n3)nc2[nH]1 15106,C(=O)(C(C)(C)CC(C)(C)C)NC1(CC)CN(C(c2cc(OC)c(F)c(F)c2)=O)C1 15107,C1(CNC(c2ccc(C(C)=O)o2)=O)CC2CC2N1C(=O)CCCSC(C)(C)C 15108,c1(C(=O)NCCOCCCN(C)C(c2cnc(O)o2)=O)cc(Cl)ns1 15109,c12ccccc1CNC(=O)C21CCC1.CCS(=O)(=O)Cc1cn(CC2CCC2)nn1.N 15110,Cc1cc(C(N2CC(O)(C(C)NC(c3conc3C(C)C)=O)C2)=O)c(O)c(C)c1 15111,C1(NC(C(C)OCC=C)=O)CCC2(CC1)CN(C(=O)CC13CC(C1)C3)CCO2 15112,c1(C(N2C(COC)(CNC(C3CC3(C)C)=O)CCC2)=O)cncc(N=[N+]=[N-])c1 15113,c1(N2CCC(C)C(F)(F)C2)nc2cc[nH]c2c(=NCC(C)(C)c2ccsc2)[nH]1 15114,C1(C(N2CCC(CNC(c3c(CC)cccn3)=O)C2)=O)CCC2(CCOCC2)C1 15115,c1(N2CC3C(C)C3C2)nc2ccccc2nc1N(C)Cc1ccc(S(C)=O)cc1 15116,C1(C(=O)OCC)CCN(CC(=O)NC2CC(N(C(=O)CC(C)(C)C)C)C2)CC1 15117,C#CCC(C)C(=O)NCC1COCCN1C(c1ccc(N(CCCC)C)cc1)=O 15118,CCC(C(=O)NCCCCC1CN(C(=O)C(C)C2CC2)C1)N1CCCC1=O 15119,CC(O)C(C(=O)NCCCCCCC1CC1)NC(c1ccc(O)cc1)=O 15120,c1(N2CCN(C(CNC(C)=O)=O)CC2)cc(Cl)c2cnn(C)c2n1 15121,c1(C(N(C2(CCCCNC(=O)CC3COCCO3)CC2)C)=O)cnn(C)c1 15122,C1(CC(=O)NCC(C(C)C)C)CC(NC(=O)C=CCN(C)C2CC2)C1(C)C 15123,N1(C(=O)C=CC2CCCC2)CCC(CCCNC(C23CCC(C2)C3)=O)CC1 15124,C1(NC(CC=C)=O)C2CN(C(C3(CO)CC3(F)F)=O)CC12 15125,C1(CCC)CN(C(=O)CCC2CCOC2)CCN1C(=O)Cc1ccon1 15126,CC1(C)CN(C(c2csc(S(N)(=O)=O)c2)=O)C(CNC(=O)C(C)(C)C(F)F)CO1 15127,c1(SCC(=O)NC2CC(NC(C3COCCC3(F)F)=O)C2)ccc(F)c(F)c1 15128,S(=O)(=O)(c1cccnc1N(C)CC1CCCS(=O)(=O)C1)NCCN(C(C)C)C 15129,Cc1ccc(C(N2CCC3CN(C(=O)C=CBr)CCC3C2)=O)c2ccccc12 15130,C(=O)(C(c1ccccc1)=C(C)C)N(CC(C)O)CCNC(C(C=C)(C)O)=O 15131,N1(CC)CCN(CCNC(N2CCCC(COc3cccc(SC)c3)C2)=O)CC1 15132,CC(CCNC(=O)CC1CCSCC1)CCNC(C1(N(C)C)CC1)=O 15133,N1(C(C(CCC)(C)O)=O)CC(C2CCCN(C(c3cnc4cccnn34)=O)C2)C1 15134,C1(NC(C(C2CC2)OCC)=O)CCC(F)(CNC(c2cc(C3CCC3)[nH]n2)=O)C1 15135,C1(F)(CNC(c2ccco2)=O)CCCN(C(C2(F)CCOC2)=O)C1 15136,CCCCC(F)C(=O)NC1(C(N2CCCC2C)=O)CCC1 15137,CC1CN(C(=O)CC2(NC(C3CNC(=O)C3)=O)CCC2)CCS1=O 15138,N1(C(CS(CC)=O)=O)CCCN(C(c2cnc(C)nc2C)=O)CC1C(C)C 15139,c1(C(N(CCOC)CCNC(C2CCC2C)=O)=O)csc(Br)n1 15140,Cc1ccccc1Oc1ccc(NC(=O)C(N2CCOC(CN)C2)=O)cc1 15141,c1(CC)ncc(C(=O)NCc2ocnc2C(=O)N(C)CC2(O)CCOC2)cn1 15142,CC1CN(C(=O)C=Cc2ccco2)CC(CCNC(=O)CCC2CC2)O1 15143,c1(CC)nc(C(N2CC(NC(=O)CC(C)OC)C(C)C2)=O)c2ccccn12 15144,c1(C(=O)NCC2(CC(=O)N(CC(CC)OC)C(C)C)CC2)cncc(OCC)c1 15145,c1(C(C(C)SC)C)ccc(NC2(C)CC(NC(=O)OC(C)(C)C)C2)cc1 15146,c1(NC(C2N(S(C3(COC)CC3)(=O)=O)CC(C)C2)=O)cc(O)c2ccccc2n1 15147,C1(N(C(=O)CCC2CCCCC2)C)CCC(NC(C2CCNC2=O)=O)CC1 15148,Cc1ncc(CNC(=O)C(CN(C)C)NC(=O)Cc2cnnn2C)s1 15149,C(C)(C)(C(CO)C(C)C)C(c1ccc(NC(C(C2CCCC2)OC)=O)cc1)O 15150,C1(NC(C(CCCOC)C)=O)CCCCN(C(=O)Cc2cccc(C)c2)CC1 15151,Cc1cccc(C(N2CCCC(C)C2CNC(c2c[nH]ccc2=O)=O)=O)c1O 15152,c1(NC(c2scc(C(=O)Nc3ccc(I)c(Cl)n3)n2)=O)cccc2[nH]ncc12 15153,N1(C(c2cc(C)ncc2C)=O)CCCC(O)(CNC(=O)CCSCC(N)=O)CC1 15154,N1(C(Cn2c(=O)sc(C)c2C)=O)CC2ON=C(CNC(c3ccn(C)n3)=O)C2C1 15155,N1(C(c2c(C)nc(CC(C)C)o2)=O)CCC2(CC1)CC2NC(=O)CSCC(N)=O 15156,N1(C(c2c(C)cns2)C(=O)NCc2ccco2)CCCC(c2cccnc2)C1 15157,N1(C(C2C(SC)CCC2)=O)CCC(=CCNC(c2sccc2C2CC2)=O)CC1 15158,C1(OC)CN(C(=O)CCN2CCOC2=O)CC1NC(=O)CN1C(=O)CNC1=O 15159,c1(CCCC(=O)NCCN(C)C(c2ccc(F)c(N)c2)=O)c[nH]c2ccccc12 15160,N1(C(=O)Nc2c(C)cc(-c3ccncc3)cc2C)CC2CC(C1)c1ccccc12 15161,Cc1cc(CN2CCCC2CC(=O)Nc2ncc(C(C)(C)O)cn2)c(C)[nH]1 15162,C1(C(N(C2CCN(C(C(C)OC3CCCCCC3)=O)C2)C)=O)CCCCS1(=O)=O 15163,C12(NC(=O)CCCc3cccnc3)CC(C1)N(C(c1csc(Cl)c1)=O)C2 15164,C1(C(=O)NC(C(=O)NCC)CC)CCN(C(c2cc(C)n(C)n2)=O)C1CC 15165,C(C)(C(=O)NNC(=O)C1CCC(C)O1)n1c(C)cc(C)n1 15166,C(CCC(CO)NC(c1coc(C2CC2)n1)=O)NC(=O)CCCF 15167,c1(OC)cc(C(F)(F)F)[nH]c(=NCC2(C)CCN(C(=O)C=C3CCSCC3)C2)n1 15168,Cc1cccc(O)c1C(=O)NC1CC(CCC(=O)NCc2cn(C3CC3)cn2)C1 15169,N1(C(C(CC)OC2CCCC2)=O)CCCC(CC#N)C1 15170,c1(OC)cnc(C(=O)N(C)CCN(C(=O)Cn2ccnc2C)C(C)C)cn1 15171,C1(C(=O)NC(CSC)(C)C(=O)N2CCOC(C(C)C)C2)CC2(CC(=O)C2)C1 15172,C(C(C(=O)NC(c1csc(C)c1)C(=O)O)OC)OC 15173,C1(CNC(CC2(C)CC2(F)Cl)=O)CC2CCC1N(C(c1ccn(CC#N)n1)=O)C2 15174,CCCCCS(=O)(=O)OC(=O)CCS(=O)(=O)c1ccccc1 15175,Cc1c2cnn1C1CC(C1)NC2=O.c1(CNC(=O)CN(C)C)nncs1 15176,N1(C(c2c(CC)ncs2)=O)CCC(CC)C1C(=O)NC(C)C(C)C 15177,N1(C(c2ncn(C)n2)=O)CC2CC2C1CNC(c1cncc(O)c1)=O 15178,c1(NC(NOCCS(C)(=O)=O)=O)ccc(Cl)c(C(=O)NCc2ccco2)c1 15179,N1(c2cccc(-c3nnn(C(C)(C)C)n3)c2)C(=O)C2CC(F)CN2C1=O 15180,CC1(C(=O)NCCN(C(=O)C(c2ccc(F)c(Cl)c2)O)C2CC2)CCCCNC1=O 15181,c1(OC)ccc(Cl)c(C)c1C(N1CCC2(NC(c3cc(C4CC4)[nH]n3)=O)CC2C1)=O 15182,CCCC(O)CC(=O)NCCCCNC(=O)C(c1ccc(Br)cc1)(F)F 15183,c1(C(N2CCC(NC(CC(CC)SC)=O)(CF)C2)=O)ncc(F)c(OC)n1 15184,c1(C(=O)NC(CC)CN(C(C2CCCSS2)=O)CC)ccc2ccccc2c1 15185,c1(C(N2C(C(=O)N(CCO)CC3COCCO3)CC2)=O)c(Br)ccc2cccnc12 15186,Cc1ccc(-c2cc(COC(=O)C(CF)NC(=O)OC(C)(C)C)on2)cc1 15187,c1(C(C(N2CCC(N(C)CC)C2)=O)C)ccc(C#N)cc1.C=CC1(CNCC)CCC1 15188,C(=O)(C=CS(C)=O)NC(C1(O)CN(C(=O)C(F)(F)c2cscn2)C1)C 15189,CC1(C)CCCc2c1n[nH]c2C(=O)Nc1cccc(CNC(c2cccs2)=O)c1 15190,c1(C(=O)NCC(=O)NC2(C)CC(C(N(CC(=O)N(C)C)C)=O)C2)cccc(F)c1 15191,N1(C(C(C)CC2CCC2)=O)CCC(CO)(CNC(c2c[nH]cc2C2CC2)=O)CC1 15192,Nc1cc(C(N2CCCC3(NC(C4CC=CCO4)=O)CC3C2)=O)cc(F)c1O 15193,C1(c2cccnc2)(C(=O)NCC(CNC(C(F)=CCC)=O)O)CCCC1 15194,C1(NC(c2cc(C(C)C)n(C)n2)=O)CCC(C)N(C(c2ccc(Cl)cc2N)=O)C1 15195,c1(CNC(C2CSCCN2C(c2cc(F)c[nH]2)=O)=O)ccccc1F 15196,c1(C(N2CC(COC)(CNC(=O)CC=C(C)C)C2)=O)ccc2cc[nH]c2c1 15197,C1(C(=O)NC(CNC(CC(=O)NCC#C)=O)C(C)C)CC2COCC(C1)C2 15198,C1(CC(=O)NC(C)CCN(C(=O)CN(S(C)(=O)=O)C)C)CCCCCO1 15199,CC(c1cnn(C)c1)=CC(=O)NC1CCC(NC(C2CCN(C)C2C)=O)C1 15200,C#CCCC(O)C(=O)N1CCN(C(=O)CCN(CCC(C)(C)C)C)CC1CCO 15201,c1(C(=O)NC2CC(C)(NC(C(CC)NC(N)=O)=O)C2)cnn(C)c1Br 15202,C1(CC(=O)NCc2sccc2Cl)CCCN(C(C2(C3CCCCO3)CCC2)=O)C1 15203,C1(CNC(C=C(C)Cl)=O)CC2CCC1N2C(=O)Cc1cccc(F)c1 15204,N1(C(C(C)OCC)=O)CC(C2CCCCN(C(c3cc(Cl)ccc3F)=O)C2)C1 15205,N1(C(C(C)(C)N2CCCC2)=O)C(C(=O)NCC=Cc2ccccc2)CC2CC12 15206,N1(C(CC=C=C)=O)CCN(CCNC(=O)CC(F)(F)Cl)C(c2nccn2C)C1 15207,CC1(CNC(C2OCCC2C(F)F)=O)CCN(C(c2csnn2)=O)C1 15208,C(=O)(NNC(=O)C(C)(C)CCCCNC(C1C2CCC3C(C2)C13)=O)C1CC(=C)C1 15209,C(=O)(C(C(C)O)NC(=O)CC1CCCC2CC12)NC1C(OC)COC1 15210,Cn1cccc1C(=O)NC1(CCNC(C2CCN(c3ccncc3)C2)=O)CCC1 15211,C(C(C)(C)C(=O)N1CC(CNC(c2cc(-c3ccncc3)on2)=O)C1)OC 15212,N1(C(c2ccc(CC)cc2)C(=O)NC2COC2)CCC(O)(c2cc[nH]n2)CC1 15213,C1(C)(C(N(C)CC2(O)CCN(C(c3cncs3)=O)C2)=O)CCCCNC1=O 15214,N1(C(COc2cc(C)[nH]n2)=O)CCC(NC(=O)CCCF)CC1 15215,C=CC(C)(C)C(=O)NCCCC1CCN(C(=O)C(C2CC2)COC(C)(C)C)CC1 15216,N1(CC)CCC(CC(=O)NC(CNC(=O)COC2CCCC2)CO)C1 15217,C1(CC)CCOC1C(=O)NCCC1(NC(c2nnn(-c3ccccc3)n2)=O)CC1 15218,C1(NC(C(CC)(C)C)=O)CCC2CCN(C(=O)CCc3ccccc3[N+](=O)[O-])C12 15219,c1(NC(C2CC2CNC(c2nc(Cl)cs2)=O)=O)ncc([N+](=O)[O-])cc1C(F)(F)F 15220,C1(C(c2ccncc2)C(=O)NCC)CCN(C(c2sccc2OC)=O)C1 15221,C(=O)(C(CCCC)C(C)C)N(CCC(C(C)C)NC(c1nccc(C#C)c1)=O)C 15222,C1(NC(CSCCCC)=O)(CC)CCN(C(=O)C(c2cccnc2)C)CC1 15223,c1(C(=O)NC2CC(CNC(C3N(CC)CC3)=O)C2)c(N)cc(F)cc1Cl 15224,C1(C(=O)NC2(CNC(C3CCCC3OC)=O)CCOCC2)Cc2ccccc2N1 15225,C(=O)(C#CC1CCOCC1)N(C)CCNC(=O)COC(C)(C)C(F)(F)F 15226,CC(C)(CCC(=O)N1CC(O)CC1NC(C1CC2CCC1C2)=O)c1nn[nH]n1 15227,c1(SCC(N2CCN(C(C34CCCC3C4)=O)CC2)=O)nc2ccccc2[nH]1 15228,c1(C(=O)NCC2N(C(C(CC(C)C)O)=O)CC=C2)ccc(Br)c2cn[nH]c12 15229,c1(C(=O)NC2CCC(NC(C3N(C(C)=O)CCCC3)=O)CC2)ccc(F)nc1C 15230,N1(C(c2cnn3c2OCC3)=O)CCC2(CCCCN(C(=O)C(O)C3CC3)C2)C1 15231,c1(C(=O)NC2CCC(CNC(CC(=C)Br)=O)C2)nnc(O)cc1O 15232,c1(C(N2CCCC(N(C(c3ccns3)=O)CC)C2)=O)c(OC)cccc1O 15233,CC1CN(C(c2cscc2Cl)=O)CC1C(=O)NCCSCCO 15234,c1(C(N2C3CC(NC(C4(CC(C)C)CC4)=O)C2CC3)=O)cnn2c1CC(F)(F)C2 15235,c1(CC(CC)C)nc(-c2cn(C)cn2)n(-c2cnn(CC)c2)n1 15236,c1(C(N2C(C(C)C)CNCCC2)=O)cc2n(c1)CCCNC2=O 15237,C1(C(=O)NC(CNC(CC(C)C(F)F)=O)CO)CCC2(CC1)NC(=O)NC2=O 15238,CCCC(C)(C)C(=O)NCC1CC(CNC(=O)C(C)O)C1 15239,Cc1cc(C(=O)NC(C)CCN(C)C(c2cc(C(C)C)no2)=O)n(C2CC2)n1 15240,C(=O)(C(O)CC(C)(C)C)NCC1ON=C(C(=O)NCC(C(C)C)(C)C)C1 15241,c1(SC)cccnc1C(=O)NCC(C)N(C)C(c1cc(C)cnn1)=O 15242,N1(C(C2(Cl)C(C(C)=O)C2)=O)Cc2occ(C(=O)NCC34CCCCC3C4)c2C1 15243,C1(O)(CC)CN(C(C2CN(Cc3nc(O)n[nH]3)C2)=O)C1 15244,C(=O)(C1=NOC2(CCC2)C1)NCC(CO)(CO)NC(C(c1ccc(F)cc1)C)=O 15245,N1(C(C2(OCC)CCC2)=O)CC2(CCN(Cc3ccc(C)cc3)CC2)C1 15246,Cc1cnc(C(=O)N(C)CC2CC(F)CN2C(C2CC2F)=O)c(C)c1 15247,Cc1cc(C)c(C=CC(=O)NCCNC(C2CN(C3CCOCC3)C2)=O)c(C)c1 15248,C1(c2cccs2)(C(N2CCC(CN(C(=O)C(F)F)C)C2)=O)CCOCC1 15249,C(=O)(CC(C)CC(C)C)N1CCC(CC)(NC(C2(COC)CC2(F)F)=O)CC1 15250,C(=O)(C#CC1(C)CCCO1)N1CC(CNC(CC2C(C)CCC2)=O)OCCC1 15251,c1(OC(C)C(=O)NCC2(O)CC(NC(C3OCCO3)=O)C2)ccc(F)nc1 15252,c1(C(=O)NCC2N(C(c3scc(COC)c3)=O)CC(F)C2)cccc2c1CCC2 15253,C(=O)(CCCCCN=[N+]=[N-])N(C)CP(C)(C)=O.C(=O)CCNCCNC(=O)CO 15254,C12(NC(C(C)OCC)=O)CCC(CC1NC(C13CCC(C(=O)OC)(CC1)C3)=O)C2 15255,c1(C(=O)NCC(C(C)(C)C)NC(C2CCC(=O)O2)=O)cnc2[nH]ccc2n1 15256,Cc1ccc2oc(C(=O)NC3CC4CC3N(C(c3cnc(C)cn3)=O)C4)cc2n1 15257,c1(OCC)ccc(-c2noc(CN(C)CC3CCCN(C)C3=O)n2)c(OC)c1 15258,C1(NC(c2ccc(C)cc2Cl)=O)CC2CCCC(C1)N2C(=O)CN1CCOC1=O 15259,CC1(C)CN(C(C(=O)NC2CCCCC2)C2CC2c2cncs2)CCS1=O 15260,C(=O)(C1=NOC(C(=O)NC2CCCN(C(=O)CC(C)(C)O)C2)C1)OC(C)(C)C 15261,C1(O)(C(=O)OC(C)(C)C)CN(N2CCC3(C2)CC3(F)F)C1 15262,N1(C(C)CCc2ccco2)C(=O)NC(C2(C)CCC2)C1=O 15263,C1(O)(CCNC(C2C(CC)C2)=O)CCN(C(c2cnn(C)c2)=O)C1 15264,CCC(CN(C)C)CC(=O)NCC(CO)NC(c1csnc1C)=O 15265,N1(C(C(CNC(CC2CCCN(C)C2)=O)N(C)C)=O)CC23CCC2(COC3)C1 15266,C1(NC(C(C)C)=O)CCCCC1CNC(=O)C(O)COCc1ccccc1 15267,CC1(C)CC(NC(=O)Cc2csc(=N)[nH]2)CN(C(C2CC(C)(C)OC2(C)C)=O)C1 15268,c1(C(=O)NCC(CO)NC(c2csc(CO)n2)=O)cc(C(F)F)ccc1Cl 15269,CCCC(CNC(=O)CC1CCC(C)(C)O1)C(=O)NCC1OCCC1(C)C 15270,c1(C(N2CCC(CC(N3CC(C(C)O)C3)=O)CC2)=O)cccc2cncn12 15271,C1(NC(=O)CSCCC(F)(F)F)(CO)CCCN(C(c2csc3nccn23)=O)C1 15272,C1(NC(CS(CC)=O)=O)CC2CC1CN(C(c1c(C)ccc(Cl)c1F)=O)C2 15273,CC1CC2CC(C(=O)NC3CN(C(=O)C=Cc4ccccc4Br)C3)(C2)O1 15274,C1(C(CC(=O)OC)NC(=O)CSc2n[nH]c(C)n2)CCC(F)(F)CC1 15275,c1(C(N(CCCNC(C2(C)CC(C)C2)=O)C2CC2)=O)n[nH]c2cc(Cl)ccc12 15276,C(=O)(CC(C)(O)C(F)(F)F)NC(C1CCCN1C(=O)C=Cc1cccc(O)c1)C 15277,C(=O)(C(S(C)(=O)=O)C1CC1)NC(C1CN(Cc2cn(C3CCC3)nn2)CCO1)C 15278,C1(C2CC2)(CNC(CC2CC(NC(CNS(CC)(=O)=O)=O)C2)=O)CCC1 15279,Cc1noc2nc(C(=O)NC(C)CCCCNC(c3cnc(Cl)s3)=O)ccc12 15280,C1(COC)(NC(C2CC23CC(NC(=O)CCn2ccnn2)C3)=O)CC=CCC1 15281,CC1CN(C(c2ccnc(-n3ccnc3)c2)=O)C(C)CN1C(=O)C=CC=CC1CC1 15282,N(C(=NCc1ccc(C#N)cn1)N1CCC2=C(CCCC2)C1)CC(C)(C)C 15283,C(CCOCCO)(C(=O)NCC1CC12CC2)NC(c1cnc(C)s1)=O 15284,C1(CC)C(NC(c2cn(CCC(C)C)nn2)=O)CCCN1C(C1CC(O)C1)=O 15285,O=C1CN(C(C2CN(C(=O)CC3CCCSC3)CC2F)=O)CCN1 15286,N1(C(CN2CCN(C)CC2)=O)CC2(CC(NC(=O)C(O)CF)CO2)C1 15287,C12(NC(CCC3C(C#N)C3)=O)CC(CNC(C34CSCC3C4)=O)(C1)C2 15288,C1(C(N2CC(C)C=C(C)C2)=O)CN(C(c2ncn(C)n2)=O)CCN1C 15289,c1(OC)ccc(C#N)nn1.c1(C(=O)O)cccc(I)c1 15290,c1(C(=O)Nc2nn[nH]n2)ccc2nc(-c3cnn(C4CCOC4)c3)cn2c1 15291,c1(C(=O)NCCC(C(C)C)NC(c2c(CC)nn[nH]2)=O)cncc(Cl)c1C 15292,c1(C(N2CCCC(C)(C(N3CCC(CC)C3)=O)C2)=O)cnc2cc(Cl)ccn12 15293,CCC(C(=O)N1CC(O)CC1CNC(C1(c2ccccc2)CCC1)=O)C(C)C 15294,c1(OC)c(Br)ccc(C(=O)NCC2CN(Cc3c(C)cc(Cl)nc3Cl)C2)c1F 15295,C(=O)(C(C(C)CC(C)(C)C)N(c1noc(-c2cccs2)n1)C)NCC 15296,N1(C(C=CC=CC)=O)CC23CCCC2(C1)CN(c1nc2cccc(F)c2s1)C3 15297,c1(CC)c(C(N2CCOC(CC(=O)NC3CCC=CCC3)C2)=O)cnn1C 15298,c1(CC(=O)NCCCC(C)NC(C2OCCOC2(C)C)=O)coc2ccccc12 15299,C1(NC(c2cc(C)[nH]c2C)=O)CC2CCC1C(NC(=O)CSc1ccccc1)C2 15300,CC(CNC(=O)COCCc1cccs1)(CO)NC(c1cnoc1-c1ccoc1)=O 15301,c1(C(=O)NC2C(NC(C(C)OCC=C)=O)CCC2)ccc(CN(C)C)cc1 15302,C(C1=NOC2CN(C(c3csc(C4CC4)n3)=O)CC12)NC(c1cnsc1)=O 15303,c1(C(N2CC(N(C)C(C3CC(=C4CC4)C3)=O)C(C)(C)C2)=O)ccc(Cl)cc1CO 15304,S(=O)(=O)(c1nc(N2CCC(O)C2)ccc1Br)N(C)Cc1cn(C)nc1Br 15305,C1(CNC(c2c(C)nn(C)n2)=O)CN(C(=O)Cc2cc[nH]c2)C2CCN1C2 15306,c1(C(=O)NCCN(C(c2c(CC)cncc2)=O)CC)n[nH]c2c1CC1CC21 15307,N1(C(CCC2(C)CN(C(CN(C)C3CC3)=O)C2)=O)CCCC12CCOC2=O 15308,CC1(CN)CCCN(CCC2CC2(Cl)Cl)C1.c12ccccc1CC(=O)NC2=O 15309,c1(C(N(CC(C)NC(=O)C(C)(C)N2CCCCC2)CC)=O)c[nH]cc(C)c1=O 15310,C(=O)(CS(=O)(=O)C1CC1)N1CCC(C(=O)Nc2c(N(C)C)cccc2)C1 15311,c1(C(N(C2CCN(C(C3(F)CCOC3)=O)C2)CCC)=O)cccc(C2(F)CC2)c1 15312,C1(OC)C(OC)CN(C(c2ccon2)=O)C1CNC(C1(C)CC2CC2C1)=O 15313,c1(N(C(CCNC(c2cc(CCC)[nH]n2)=O)C)C)ccc(S(C)(=O)=O)cn1 15314,c1(C(N2CC3N(C(c4ccc(OC)o4)=O)C(CC3)C2)=O)cn2cccc(Cl)c2n1 15315,c1(C(N(C)CCNC(C2(C)CCC(O)CC2)=O)=O)ccnc2c1cnn2C 15316,C1(O)(c2cn(CCC(=O)NC(c3cc(C)on3)(C)C)nn2)CCC(F)(F)CC1 15317,C1(=O)C(Cl)(Cl)C2=CN=CNC3(CC(=O)NC(CC)CC3)C2N1 15318,C1(OC)CN(C(C2CCCO2)=O)CC1C(F)F.C12C=CC1C(=O)OC2=O 15319,c1(NC(C2(NC(C3CCC(N=[N+]=[N-])C3)=O)CC2)=O)cc[nH]c2nccc1-2 15320,CN1CCN(C(C2CC(C)(C)CCO2)=O)C(CNC(c2ccc(N)cn2)=O)C1 15321,C1(NC(C(c2cnn(C)c2)C)=O)CCSC12CN(C(=O)C(C1CCCCC1)F)C2 15322,C1(C(C)NC(=O)OC(C)(C)C)CCN(C(C2CCC(C(=O)O)C2)=O)C1 15323,c1(OC)cc(O)ncc1C(=O)NCC1CCN(C(=O)C(C)(C)CCOC)CC1O 15324,C1(NC(=O)CCC2CC(NC(C3CCC4(CCC4)O3)=O)C2)CC2CCCCCC12 15325,C1(CCC)CN(C(=O)Cc2cc[nH]n2)CCN1C(c1ccc(F)n1C)=O 15326,c1(SC)ncc(C(=O)NCCC2CCN(C(c3cnn(C)c3N)=O)C2)c(O)n1 15327,Cc1cc(O)nc(C)c1C(N1CC2(CO)CC1(CNC(=O)C#CC(C)(C)C)C2)=O 15328,C1(NC(C(C2CCCC2)NC(C(CC(=C)C)OC)=O)=O)CCn2ncnc2C1 15329,c1(CC)cc(C)ccc1C(=O)NC(C1CCCCC1)CNC(=O)C(C)(O)C(C)C 15330,C1(C(=O)NC2CC(N(C)C(c3cc[nH]c3)=O)C2)Cc2ccccc2O1 15331,N1(C(CC(COC)(C)O)=O)CC2C3CCC(C2C1)N(C(=O)CCS(C)=O)C3 15332,N1(C(C(C)CO)=O)CC(O)CC1CNC(=O)CC(C)(C)C 15333,C1(NC(C(CC)N(C)C)=O)CN(C(C2CCC(OC)CC2)=O)C2(CCCC2)C1 15334,S(=O)(=O)(C1CCCN(C(C2CC2C(c2ccc(C#N)cc2)=O)=O)C1)NC 15335,c1(C(=O)NC(C2CCN(C(C=CC)=O)C2)(C)C)ncn2c1CCCC2 15336,N(C(=NCCC(C)F)NC1CC1F)C(C)C 15337,Cc1ccc(C(=O)NCC23CCC(CC2)N3C(c2cc(F)cnc2O)=O)c(C)n1 15338,C(=O)(C(O)CC(C)(C)C)NCCCC1N(C(c2ccn(CC)c2C)=O)CCCC1 15339,N1(C(CN(CCOC)C)=O)C(CNC(c2nc(Cl)ccc2F)=O)CC2COCC12 15340,c1(C(=O)NCC2C(NC(c3cn(CC=C)nn3)=O)C2)cc(OC)cc(Br)c1 15341,c1(N2CCCC(CC)C2)nc(=Nc2cccnc2C)[nH]c2c1cnn2C 15342,C=C(C(=O)N1CCC(OC(C)(F)F)CC1)C1CCNCC1 15343,N1(C(CSc2nc(C)[nH]n2)=O)CCN(C(=O)CC(C)n2cccc2)C2CCC12 15344,N1(C(C(CSC)OC)=O)CCCCCC1CNC(=O)Cc1ccc(F)c(F)c1 15345,c1(C(=O)NC(C(C)C)CNC(=O)C(F)CC2CC2)cc(N)cc2ccccc12 15346,c1(C(=O)NCCC(C)NC(C2CC23CC(O)C3)=O)cnc(C(F)F)nc1 15347,C#CCCN=C(NCCC(C)F)N1CCC(C2CC2)C1 15348,C#CCCCC(=O)N1CC(NC(C2(CC)CC2(F)F)=O)C(O)C1 15349,N1(C(C2(C)CC=CC2)=O)CCCC(CCNC(c2ncsc2C2CC2)=O)CC1 15350,N1(C(c2ccc(CCCCC)o2)=O)CCC(C(C)NC(=O)COC(C)=O)CC1 15351,c1(C(N2CC(O)(CC(=O)NC(C3(C)CC3)CO)C2)=O)ccncc1O 15352,C(C)(CO)(C(=O)NCC(C)OCF)NC(CCCN(C(C)=O)C)=O 15353,c1(OC)ccc(N(C(=O)Cc2sccc2Cl)C)c(OC)c1 15354,Cc1cccn2c(C(N3CCCC(NC(c4cccn4C)=O)CCC3)=O)cnc12 15355,C(=O)(CC(C)(C)CN(C)C)N(CCN(C(C1CCCC(C)C1)=O)C)C 15356,N1(C(c2c(C)cn(C(C)C)c2)=O)CCN(C)C(CNC(c2n[nH]c(C)c2C)=O)C1 15357,C1(CNC(C(C(C)C)SC)=O)CN(C(=O)CC(C)(C)C)CC1(C)C 15358,C1(C)(CC(=O)NC2C(NC(C(CO)N(C)C)=O)CCCC2)CCCCCC1 15359,c1(OC)ccc(N2CCC(C(c3ccccc3Cl)OC)CC2)nn1 15360,C1(C(=O)NCC2CN(C(c3c(CC)c(CC)c(C)[nH]3)=O)C2)CN(C)C(=O)CCO1 15361,C1(NC(C=CCN(C(=O)CC2CCSCC2)C)=O)C=CCCCC1 15362,C#CCC(C)(C(=O)NCC1CCCSC1)NC(=O)CCc1cncn1C 15363,C1(C)(C(=O)NCC(CNC(C(CC)C2CCC(=O)N2)=O)O)CC(C)(C)C1 15364,C(CCC(C)(C)C(=O)N1CCCC1C(N1CC(O)(CCO)C1)=O)OC 15365,N1(C(c2n(C(C)C)ccn2)=O)CC2C(CNC(=O)Cc3cn[nH]c3)C2C1 15366,c1(CC)ccccc1N(CC(=O)OC)C(=O)NCC1CCC1C 15367,c1(C(=O)NCCCCCNC(C2C(OC(C)=O)C2)=O)ccc(Cl)c(Cl)c1 15368,C1(CC)CN(C(=O)CC(C)(F)F)CCC1NC(c1cccc(C2CC2(F)F)c1)=O 15369,c1(C(=O)NC2C(C)CN(C(=O)CSc3ncccn3)C2)nc(Cl)ccc1F 15370,c1(C(N2CCC(N(C(=O)C(CCSC)OC)CC#C)CC2)=O)cccc2ncsc12 15371,c1(C(=O)NC2CCN(C(c3c(CC)nccn3)=O)C2)c(Br)sc(C)c1C 15372,n1(CC)ccc(C(=O)NCC2(NC(=O)C(C(C)C)NC=O)CCCCC2)c1C 15373,c1(N2CC(NC(C3CC4(CCC4)CO3)=O)CC(C)(C)C2)nc2cccc(F)c2s1 15374,C1(CNC(C(CNC(c2ccnc(O)c2)=O)OC)=O)CC2(CC2)C(=O)O1 15375,Cc1ccc2c(C(=O)NCC3(NC(C4CCC4C(N)=O)=O)CCCC3)c[nH]c2c1 15376,N1(C(C2CC=C(C)CC2)=O)CC2CC1CCC2NC(=O)CCc1cn(C)nn1 15377,Cc1nn(C)c2ncc(S(=O)(=O)NCC3(c4cccs4)CCOCC3)cc12 15378,n1(C(CC)(C)C)nnnc1C(C(C)(C)OCC)NCCCC(C)CCC1CC1 15379,C1(C(=O)NCc2cc(OC)no2)CCC2(CN(Cc3ccc(C#N)cc3Cl)C2)O1 15380,N1(C(CCOCCC)=O)CCN(C(C2COCCC2(F)F)=O)C(C)C1 15381,N1(C(CNC(CCC)=O)=O)CCCC2CN(C(=O)CCCN3CCCC3)CCC12 15382,c1(CNC(C(=Cc2cn[nH]c2)C)=O)nnn(C)c1C(N1CCC(O)(CO)C1)=O 15383,C=CC1(C(=O)N(C2CCCC2O)C)CCN(C(=O)C(CCC)N(C)C)C1 15384,N1(C(C)C(=O)NC(C)(C)C)CCN(C(=O)CCCCC2CC2)CC1 15385,C1(NC(C2CS(=O)(=O)C2)=O)C2CC3CN(C(=O)COc4ccc(O)cc4)C1C3C2 15386,CC1(CNC(=O)C2=CCC(NC(=O)Cc3ccoc3)C2)CCCCCC1 15387,C1(CCC(=O)NCC(CC)NC(C2(C(=O)NC)CC=CCC2)=O)CCC(=O)NC1 15388,C12(C(=O)NCC(CNC(C(C)Cc3ccco3)=O)F)CC(C1)C(C(F)(F)F)O2 15389,c1(C(=O)Nc2ccnc(C(C)(C)C)n2)cn(CCO)c(=O)nc1O 15390,C1(C)(OC)CCN(C(C2CC3C=CC2CC3)=O)CC1 15391,C1(C#N)(C(N(C2CN(C(CC(C)SC)=O)C2)C)=O)CC1(C)C 15392,C#CCC(C)(CNC(=O)CC1(NC(=O)CC2CCSC2)CCC1)CO 15393,N1(C(CC2CC(NC(C(C(C)C)F)=O)C2)=O)CCC(C)C2(CCC2)C1 15394,N1(C(C(CC)=CC)=O)CCC(C)C1C(=O)NCC(F)Cl 15395,C(C(=O)NC1CC(C)(NC(c2ccon2)=O)C1)(C(C)C)n1ncc(C)c1 15396,C1(C(N(CCCC)CC)=O)CCOC1CNC(=O)CCN(C)C(C)=O.OC 15397,O=C(NN1C(=O)NC2(CCC2)C1=O)c1c[nH]c2c(F)cc(Cl)cc12 15398,C1(CNC(C(C)OCC2CC2)=O)CC(F)(F)CN1C(=O)CC12COCC(C1)C2 15399,c1(CC(=O)N(CCNC(=O)CC2CCC(=O)N2)CC)cn2cccc(C)c2n1 15400,C(=O)(C(C(C)C)NC(=O)C(C)C)N(CCN(C(C(C)OCC)=O)C)CC 15401,c1(OC)ccnc(N(C(C)=O)Cc2ccnc(CNc3cccc(C)c3)c2)n1 15402,Nc1c(C(=O)NCCOCC(=O)NCC2CC2c2cnns2)cccc1Cl 15403,Cc1cncc(C(=O)NCCC(C)CCNC(c2coc(C3CCC3)n2)=O)n1 15404,c1(CNC(CC2(N(C(C(C3CC3)SC)=O)C)CC2)=O)ccc(Cl)o1 15405,Cn1nc(C(=O)NC2CCOCC2C(=O)NCC=CC2CC2)cc1F 15406,N1(C(C)=O)CCOC2(CCN(C(=O)C(c3cccc(Br)c3)O)C2)C1 15407,c1(C(C)C)nc(C(=O)NC2(CC(=O)NCCCC3(C)CC3)CC2)co1 15408,N1(C(CCOC(N(C)C)=O)=O)CCn2c(cnc2C2CCC2)C1 15409,C(CC(C)C)(C(=O)N1CCCC(N(C)C(c2[nH]ccc2C)=O)CC1)NC(=O)OC 15410,c1(C(=O)NCC(C(=O)N2CC(N3CC=CC3)C2)N(C)C)c[nH]ccc1=O 15411,c1(CN(CCN(C(C2(CC(C)C)COC2)=O)C(C)C)C)ccccc1F 15412,c1(NC(c2c(-c3c(C)csc3)cncn2)c2ccccc2)ccc2cc[nH]c2n1 15413,CC(C)(C)C(CCO)NC(C1(CNC(=O)C2=COCCC2)CC=CC1)=O 15414,Cc1ccc(CCCCC(=O)N(C)CCNC(C2CCSC2)=O)cc1 15415,C1(CNC(CCCOCC)=O)CC2CCC1N(C(C1(C)CCCS1(=O)=O)=O)C2 15416,C1(NC(c2c(C)ocn2)=O)CN(C(c2cc(Cl)cn2C)=O)CC1C 15417,c1(C(=O)NC2CN(C(C3N(C)CCOC3)=O)CC2F)cccc2nn[nH]c12 15418,C(=O)(CC(C)(C)N(C(=O)CN(C1CCC1)C)C)N(CC(C)C)C 15419,c1(OC)cccc(OC)c1NC(C1CSCCN1Cc1cccc(O)n1)=O 15420,c1(C(=O)NCC(C)NC(CCCCCC)=O)cn(CCCOC)c2ccccc12 15421,C1(CC(=O)NC2CCN(C(CCCC)=O)C2c2ccccc2)NC(=O)CN(C)C1=O 15422,CC(C)CC(CNC(c1cnn2ccccc12)=O)C(=O)NC1COCCC1(F)F 15423,c1(C(N(CC(C)NC(=O)CC2CCCSC2)C)=O)ccc2c(c1)CNC2=O 15424,C12(C(=O)NC3CC(NC(=O)CCNc4cncnc4)C3)CC=CCN1CCC2 15425,N1(C(c2nc(CC)oc2C)=O)CCC(C)(C)C(NC(c2cc(C)nc(O)n2)=O)C1 15426,C1(NC(C2(c3ccno3)CC2)=O)C2CN(C(=O)CCc3cccc(O)c3)CC12 15427,c1(C(=O)NC(CC)CNC(C2CCCC2(C)C)=O)cccc2c[nH]nc12 15428,c1(C=O)cccc(C)c1N.CCCCN(CC(C)NC(C1CC1CC)=O)C 15429,N1(C(C2C(C)C2c2ccccc2)=O)CC(NC(C2(O)CCCC2)=O)CC(C)(C)C1 15430,CCC(CCCC(=O)NCC1CC(O)C(O)C1)NC(c1cnc(C)n1C)=O 15431,N1(C(CSCC)=O)CCC(CNC(C2CCC23CCC3)=O)C12CCC2 15432,C1(CC)(CC)SCCNC1C(=O)NCc1ccc(N2CCCCC2)cc1C 15433,Cc1nc(C(N2CCC(C3CCCCN3C(c3cnc(O)[nH]3)=O)C2)=O)c(C)s1 15434,C12(CNC(CC3C(C)(C)CCCC3)=O)CCCC1N(C(C1CC1(Cl)Cl)=O)CCC2 15435,O=C1CC(CC2C3CC4C(C3)C24)C2(CCC2)C1.c12cn(nn1)C1(CC1)C(=O)OC2 15436,CCCCC(C(=O)N1C2CCC(C2)C1C(=O)NCc1cc(F)ccc1C)C(C)C 15437,Cc1cc2cc(C(=O)NC(C)(CNC(=O)CN3CCCC3)C3CC3)c(Cl)cc2[nH]1 15438,n1(CC(=O)NC2CC(C)(NC(C(C3CC3)OC)=O)C2)nc2ccccn2c1=O 15439,c1(CC(CC)C)nc(-c2n[nH]cc2F)n(-c2cccc(SC)c2)n1 15440,Cc1cc(OC(F)F)c(C(=O)NCC(C)NC(c2sccc2N)=O)s1.OC(F)F 15441,C1(NC(C(C)(O)C2CCC2)=O)CN(C(c2cnc(C(F)(F)F)nc2)=O)CCC1F 15442,c1(CC)nc(C)ccc1NC(=O)CC1CCCN1Cc1cccc(F)n1 15443,CC1(C)CN(c2nc(N3CCC(OCCF)C3)c3c(n2)CCC3)Cc2ccccc21 15444,CN1CC(N(C2CCOCC2)C(C2CCC2)=O)N(C(=O)OC(C)(C)C)CC1=O 15445,C(=O)(CCCC(=O)NCC1CC1CNC(c1c(C)nn(C)c1C(F)(F)F)=O)OC 15446,C1(C(=O)NC2C(NC(c3occ(C)c3)=O)COC2)CC2CCCC(C1)C2 15447,N1(C(=O)C(Cl)(Cl)Cl)CCC2(CC1)CN(S(=O)(=O)Cc1ccccc1Br)C2 15448,C1(F)(CNC(CC2N(CC)CCOC2)=O)CCN(C(=O)CN(C)S(N)(=O)=O)CC1 15449,c1(C(=O)NCC(C(C)C)NC(=O)C(c2ccc(Cl)s2)=O)ccnc(O)c1 15450,C(=O)(C(CC)CC(C)C)NCC(CN(C(C(CCCC)C)=O)C)(C)C 15451,Cc1ccc(C(=O)NC2CN(C(C3C4CCC(F)(F)C34)=O)C(C)(C)C2)c(N)c1F 15452,c1(C(=O)NC(COC)C(=O)Nc2cccc(F)c2O)ccc2[nH]ccc2n1 15453,C(=O)(C1CCC(=O)c2cccn21)NC1CCN(C(CC(C)P(C)(C)=O)=O)CC1 15454,c1(C(=O)NCC2CN(C(C(c3ccccc3C(F)(F)F)C)=O)C2)ccc(Cl)nc1 15455,c1(OC)ccc(C(=O)Nc2ccc(-c3ccc(N(C)C)nc3)cn2)cc1Cl 15456,N1(C(c2cn(CCC)nn2)=O)CC(NC(=O)C=Cc2cc[nH]n2)C(CO)C1 15457,c1(OCC(C)C)ccccc1C(=O)N(C)CC1(NC(C2CCOCC2)=O)CC1 15458,C1(CNC(C2CCC(OC)C2)=O)CCC2(CCC2)CN1C(=O)CCc1cccs1 15459,c1(C(=O)NC(C2CN(C(=O)C(C)(F)C(F)(F)F)CCO2)C)cc2n(c1)CCCC2 15460,N1(C(c2c(C)onc2)=O)CCC2CCN(C(c3cnc(=O)n(C)c3F)=O)C2C1 15461,N1(C(CC(C)C2CC2)=O)C(CNC(=O)Cc2nccn2C)CC2COCC12 15462,C1(O)(CC)CN(C(C2(CCNC(=O)C(C)CC3CCCC3)CCC2)=O)C1 15463,c1(NCC2(OCC)CCOC2)ccnc(O)c1 15464,C1(C(N(CC(CC)NC(=O)CCSC)CC)=O)CCc2nc(C)ncc2C1 15465,Cc1nnc(NC2CC(F)(CNC(=O)Cn3ccc(O)nc3=O)C2)nc1C 15466,c1(SC)ccc(O)c(C(=O)NCC2(O)CCCN(C(C3CC3C)=O)C2)c1 15467,C(CCN=C(NCC1CCSC1)N1CCN(c2cccs2)CC1)OC 15468,N1(C(C(CN(C(C2CCC(CC)C2)=O)C)C)=O)CCC(C#N)CC12CC2 15469,CN=c1[nH]cc(C(N2CC(OCC(=O)N(C3CCSC3)C)C2)=O)o1 15470,CCCCCCCCCCCCC(=O)NCC(C)NC(=O)CC(C)n1ccnc1 15471,CN1CCC(O)(CCNC(=O)NC2CCCCCC2CO)CC1 15472,Cc1cc(C(N2CCN(C(=O)CSC(C)C)CC2C(C)C)=O)n2nccc2n1 15473,c1(OC)ccccc1C(O)C(=O)NCC(CNC(c1c[nH]nc1OC)=O)OC 15474,CCCC(C(=O)NCCCN(C(c1ccn2cccc2c1)=O)CC)C(C)C 15475,c1(C(=O)OC)cc(CN(C)C(C2CCN(c3cnn(C)c3)C2=O)=O)oc1C 15476,CC1CN(C(=O)C=CC(C)(C)C)CC1(C)CNC(c1csc(C(C)(C)C)c1)=O 15477,Cc1cnc(C)c(C(=O)N(C)CC2CCCN2C(=O)C(C2CCCCCC2)O)c1 15478,c1(SC)cc(C)c(C(=O)NC(C)CNC(c2cnoc2C2CC2)=O)s1 15479,C(=O)(C(CN=[N+]=[N-])NC(=O)C(O)C1CCC1)N(C)Cc1ccccc1 15480,C(CCOCCO)(C(=O)NCC1(Cl)CC1(F)F)NC(C(N1CCNC1=O)C)=O 15481,N12CC(C3CN(C3)C1)C2.c1(C(c2cc(C(C)C)no2)C)ccc(C2CC2)cc1 15482,N1(C(c2ccc(CCC)[nH]2)=O)CCC(C(C)NC(c2ccccc2C)=O)CC1 15483,Cc1c(F)ccc(NC(=O)C(=O)NC2CCN(C(=O)CN3CCCCC3)C2)c1F 15484,C(=O)(C(O)CC(F)(F)F)N(C)CC1CCCN1C(c1cc2n(n1)CCO2)=O 15485,c1(C(=O)NCC2(COC)CN(C(=O)C(O)C(F)(F)F)C2)ccc2oc(C)nc2c1 15486,N1(C(C2C(NC(c3cn(C(C)C)nc3)=O)CCC2)=O)CCC(O)C(F)C1 15487,c1(C(=O)NC(C(=O)NC(CCC=C)C)COC)cc(O)nc(O)n1 15488,C#CC12CCC(C(N3C4CCCC3CN(C(=O)C(C)SCC)C4)=O)(CC1)CC2 15489,c1(OC)ccc(C)cc1C(=O)N(CCCNC(c1nnn2c1CCC2)=O)C 15490,C1(NC(CCOc2c(CC)cccc2)=O)CC(F)CN(C(=O)C(F)C2CCC2)C1 15491,S(=O)(=O)(c1ccncc1)NC1CCC(CC(=O)NC2CCC(F)(F)C2)CC1 15492,c1(CC)sc(C(=O)NCC#CCNC(=O)Cc2ccc(Cl)cn2)cc1C 15493,N1(C(CCCC(=O)NCCC)=O)CC2CC3CC2C1C3NC(c1coc(C)c1)=O 15494,c1(C(=O)NCC#CC(N2CCC(C)(N(C)C)C2)=O)ccn2ccccc12 15495,C(CC(C)(C)NC(c1cc(CNC(=O)C(C2CCC2)OC)cs1)=O)OC 15496,c1(N2C3CN(C(=O)OC(C)(C)C)C(C3)C2)ncnc2c1ncn2CCCC1CC1 15497,Cn1nc(C(=O)NCC2COCC2NC(C2CC=CCO2)=O)c2c1CCOC2 15498,c1(C(=O)NC(C2CCN(C(C3(COC)COC3)=O)CC2)C)ccccc1CC#N 15499,C12(CCOCC1)C(C1CCC(C)O1)N2.c1(NC(C2CC2)C2CC2)nnnn1C 15500,N1(C(C(CC)C)=O)CCN(C(c2cnn(C)c2F)=O)C(c2cccc(F)c2)C1 15501,C1N=C2NC(=NCC(C)(C)C13CC3)NC1=C2COC1.C=CCCN(C)C 15502,c1(C(N2C(CC)(CC)CC(OC)C2)=O)cc2scc(Cl)c2[nH]1 15503,N1(C(C=C)=O)CC2(CC2)CC1CNC(c1cc(COC)ccc1F)=O 15504,CC(CNC(=O)CC(C)(C)O)C(F)C(=O)NCc1cccnc1F 15505,C1(C(=O)NCC(CCNC(c2ccc(CO)o2)=O)O)CN2CCCN1CC2 15506,C1(C(N2CCC(CNC(C3CC(O)(c4cccnc4)C3)=O)C2)=O)CC2CC1C2 15507,c1(C(N(CC(CN(C(=O)CCn2ncn(C)c2=O)C)O)C)=O)ccccc1CO 15508,N1(CCOC)CCOc2ccc(-c3cccc(-c4nn[nH]n4)c3)cc21 15509,c1(C(=O)NC(CC)CNC(=O)CC2(O)CCCC2)ccc(Cl)cc1O 15510,C12(NC(C34CC(NC(C5CCN(C(C)C)C5)=O)(C3)C4)=O)CCC(CC1)CC2 15511,Cc1oc(C)c(C(=O)NC2CCC2NC(=O)Cc2cccc(F)c2)c1Br 15512,C(=O)(C1CCc2cccc(Cl)c21)N1CCC(NC(c2ccccc2F)=O)C(F)C1 15513,C1(C(F)(F)F)(C(N(CC(C)CNC(C2(C)CC3CC3C2)=O)C)=O)CCCCO1 15514,N1(C(C(=O)NC2CCCCN(CC(=O)O)C2=O)=O)CC2COCC(C1)C(=O)N2 15515,C1(C)(C(N2C(C(=O)NCC(C)S(N)(=O)=O)CC2)=O)CCC(=O)NC1 15516,N1(C(Cc2cc(C)on2)=O)CC=CC(NC(=O)C(C)(C)CN2CCN(C)CC2)C1 15517,C1(NC(=O)CC2C=CCC2)CC(F)(CNC(c2cc(C(F)(F)F)cs2)=O)C1 15518,C(=O)(C1=CCC2(COC2)OC1)NC(CC)CNC(c1nc(Cl)cs1)=O 15519,C(=O)(CCS(C)(=O)=O)NCC1C(NC(C(C)OC2COC2)=O)CCCC1 15520,CC(C)CCCC(=O)NCCC1(NC(c2ccn(C(F)(F)F)n2)=O)CC1 15521,C(c1ccccc1Cl)=CC(=O)NCCC1CCCN(C(C(C)(C)OC(C)=O)=O)C1 15522,c1(C(=O)NCC2(O)CN(C(CC3CCCC(OC)C3)=O)C2)ccc2nsnc2c1 15523,CC1(C)CCC(C(N2CCCC(CNC(=O)Cc3cc(C4CC4)on3)C2)=O)C1 15524,C1(NC(C(=O)NC(CC=CC)Cc2ccccc2)=O)CC2CCC(C1)N2C 15525,CC1CCC=C1C(=O)NCC=CCC(=O)NCCOCC1CC1 15526,C(=O)(CCC(=O)N(C)C(C)C)NC(C)CN(C(=O)CCCn1ccnn1)C 15527,N1(C(C2N(C)CCN(C(c3ccc(C#C)cn3)=O)C2)=O)CCC2(CC(CO)C2)C1 15528,C(c1ccncn1)=CC(=O)NCc1cc(C(=O)NC(C)CO)on1 15529,C(C(=O)NC1CCN(C(C2(F)CC=CC2)=O)C1)(C(C)C)OC 15530,c1(CC(=O)NC(C)CCN(S(C)(=O)=O)C)ccc2oc(O)nc2c1 15531,C(=O)(C(C)(O)C(C)(O)C(=O)O)N1C2CN(C(C(C)CN)=O)C(CC2)C1 15532,c1(CC(=O)NCC#Cc2cn(Cc3c(C)n[nH]c3)nn2)nc2ccc(Br)cc2o1 15533,Cc1ccc(C(=O)NC2(C(=O)NC3(C)CCSCC3)CCSC2)nc1O 15534,n1(CC(=O)NC2CC(C(N(CC(C(C)C)C)C)=O)C2)cnc(C#N)n1 15535,C#CCC(CC(=O)NC(C)C(C)(C)CO)NC(C1(CCC=C)CC1)=O 15536,C(CCN(C(=O)C(C)n1ccnc1)C)(C(C)(C)C)NC(CCOC(C)C)=O 15537,C(=O)(C(F)(F)CN(C)C(C1CC(CNC(=O)CCN(C)CCO)C1)=O)OC 15538,N1(C(C2(CNC(c3ccc(O)nn3)=O)CC(=C)C2)=O)CCCN(C)CC1 15539,c1(C(N2CC(OCCOC)C2)=O)cc(COC)no1.c1(C(=O)N)sccc1 15540,c1(C(=O)NC2C(CNC(=O)CSC(F)(F)F)CCCC2)ccc2nccn2n1 15541,CC1(NC(c2ccnc(C3CC3)n2)=O)CCC(NC(=O)C(C)(C)C2CCC2)CC1 15542,C12C(CC1O)NC(=O)C2.C(=O)(C(C)(C)n1ccnn1)NC(c1cn[nH]c1)C 15543,N1(C(c2cnc(C)s2)C(=O)NCCC)CCCC(c2ccc(Cl)nc2)C1 15544,CC1(O)CCCN(C(C2CCCC(NC(c3cncc(O)c3)=O)C2)=O)C1 15545,C#Cc1ccc(CNC(=O)NC(CO)(C(F)(F)F)c2ccc(Cl)cc2)cc1Br 15546,c1(CCNC(N2CC(C(=O)OC)CC(CC)C2)=O)cc(Br)c(OC)cc1C 15547,c1(-c2cccc(-c3c(C)cccc3)c2)ccncc1S(=O)(=O)NC(CO)C(C)C 15548,N1(C(C(C=CCCC)O)=O)CCN(CCN(C(=O)C(C#N)CC)C)CC1 15549,c1(C(=O)NCCOCCNC(=O)CCCC2CCCOC2)ccc(C2CC2)cn1 15550,C1(NC(c2ccnc(C(C)C)n2)c2nnnn2CCCF)CCC2(CCC2)CC1 15551,CC1(C)CCN(C(=O)C2=CCCSC2)C1CC(N1CCOCC(CO)C1)=O 15552,C12(C(C)C)COC(C(=O)NC(CNC(=O)CCc3cccc(Cl)c3)C(C)C)(C1)C2 15553,C1(NC(C2(OCC)CCCC2)=O)CN(C(=O)CCc2cnn(C)c2)C2CC12 15554,CCCC(C(O)C(=O)N1CCCC(C(C)(C)C)C1)NC(C1CCOC1C1CC1)=O 15555,N1(C(C2CC(NC(=O)Cn3ccnn3)C23CCC3)=O)CCC(F)(F)C(F)C1 15556,c1(N2CC(N(CC)CC)C2)ccc(S(=O)(=O)NC(c2nc(C)oc2C)C)cc1Br 15557,O=C(C1=CCCOC1)NC(C1CC12CCC2)=O.n12ccc(c1)C(=O)N1CC2C1 15558,CCC(C)CC(CO)NC(=O)C(N1CCN(C)CC1)=O 15559,C(=O)(C(COC)C(F)(F)F)NCCN(CCC)C(c1ccn(C2CC2)n1)=O 15560,CC(N)CCCC(=O)N1CCC(CC(=O)NCc2ccc(F)cc2F)CC1 15561,Cc1cc(-c2cn(CC(=O)NCC3CC4(CNC(C)C4)C3)nn2)c(C)cc1Cl 15562,c1(NC(C(N2C(CNC(C(CCC)F)=O)CC2)=O)=O)c(C)cccc1C 15563,N1(C(c2cn(CCC)nc2)=O)CC2CN(C(c3ccnc(C)n3)=O)CC12 15564,CC(C)C(C#N)C(=O)NC1(c2ccccc2)CN(C(C2CSCCS2)=O)C1 15565,C1(NC(C2CCN(CCC#C)CC2)=O)CC2CCC(C1)N2C(c1n[nH]c(C)n1)=O 15566,c1(C(=O)NCCCCNC(CSCCOC)=O)ccc(F)c(Cl)c1 15567,N1(C(CCCCC=C)=O)CCC2C(C1)CN2C(=O)CC1CCN(CC(F)(F)F)C1 15568,Cn1nc(C(=O)NCC2CCCC(NC(C3CC(O)C3)=O)C2)cc1Br 15569,Cc1cnc(C(=O)NCC2CN(C(c3ccc(Br)cc3)C#N)CCCO2)cc1C 15570,C1(C(=O)NCc2cccc(C)n2)(COC)C=CCN1C(c1sccc1CO)=O 15571,c1(N2CCC(CCNC(=O)C(c3ccc(F)cc3)F)C2)ncnc(O)c1Br 15572,C12(C(=O)NCCOCCOCCNC(c3c(C)noc3C)=O)CCCC(F)(C1)C2 15573,CC1OC(=O)NC1C(=O)NCC(C)(C)CCNC(=O)Cn1ncnn1 15574,C=CC(C)C(C)C(=O)N(CC(C)(C)CNC(c1cnc(-c2cccs2)s1)=O)C 15575,C=C(F)C1(CC(=O)NC2CCCC(NC(C3(CO)CCCO3)=O)C2)CCC1 15576,N1(C(C2CCCC(C)C2)=O)CC2(CNC(c3coc(N(C)C)n3)=O)CCC1CC2 15577,c1(CC(=O)NCC2(F)CCC(NC(C(C)(C)C3CC3)=O)C2)ccc(O)c(Cl)c1 15578,c1(OC)ccc(CCC(=O)NC2(CNC(=O)COc3ccsn3)CCC2)cc1 15579,O(N1C(=O)c2ccccc2C1=O)CC(=O)N(C(C1CCOC(C)C1)C(=O)O)C.CO 15580,N1(C(C(C2CC2)OC)=O)CC(F)(F)CC1C(=O)NCCN1CCCCC1 15581,c1(C(=O)NC(CC(C)NC(CCOC)=O)C)ccc(C(C)=O)c(F)c1 15582,C#Cc1cncc(NC(C2C(CC)CCN2C(=O)C(C)CC2CCC2)=O)c1 15583,C1(CNC(C(COC)OC)=O)CCC2(CN(C(c3cc(N)c(N)c(O)c3)=O)C2)O1 15584,S(=O)(=O)(c1ccc(N2CCSCC(C)C2)c(C#N)c1)NC1C(CCC)C1 15585,c1(NC(C2CCCC(NCc3cccc(OC)c3O)C2)=O)c(O)cccc1C#N 15586,C1(C)(C(=O)NCCCN(C(=O)Cc2n[nH]cc2Br)CC)CCC(C)C1 15587,C1(CC(=O)NCC23CC(NC(C(c4cscn4)N(C)C)=O)(C2)C3)CC(O)C12CCC2 15588,c1(C(=O)NCC)scc2c1OCCO2.C(C(=O)NCC)(C1CCCC1)N(CCC)CC 15589,C1(C(N(C)CC2COCCO2)=O)CN(C(=O)CN2CCC(F)CC2)CCN1C 15590,c1(C(N2C(C)(CC)CC(NC(c3csc(SC)n3)=O)C2)=O)noc2c1CCCC2 15591,N1(C(c2c(N)csn2)=O)CCCC(C2CC2NC(C2C3CCCC23)=O)C1 15592,CCC(C)(C)C(O)C(=O)NC1CC(C)CN(C(=O)C(F)(F)CN(C)C)C1 15593,c1(C(=O)NC23C(NC(C4(C(C)=O)CC4)=O)CC(CC2)C3)ccc2nc(C)[nH]c2c1 15594,c1(CC(=O)N(C)CC2(NC(C3CNC(=O)N3)=O)CC2)ccc(CSC)cc1 15595,N1(C(c2c(C)ocn2)=O)CCCC(NC(c2cc(=O)c(Br)c[nH]2)=O)CC1 15596,C1(CC#C)(C(=O)NCc2cc(C(=O)NC3CCSC3C)on2)CCCO1 15597,CCCC(C)(C)NC(=O)NC(C(=O)N(C)C)c1ccco1 15598,C#CCCCC(=O)NCC1C=CC(NC(c2ncsc2-c2ccccn2)=O)C1 15599,CCCC(F)C(=O)NCc1cccc(CNC(=O)C(F)CC)c1 15600,c1(CC(N2CC(Nc3ncnc(CC)c3F)C(C)C2)=O)noc2ccccc12 15601,CC1CCCC(O)(C(=O)NCCCCN(C(=O)COc2cnc(Cl)cn2)C)CC1 15602,CCCCC(O)C(C)C(=O)NC1CCOC(C(=O)NCc2occc2C)C1 15603,C(=O)(CCCCC(C)(C)OC)N1CCC(NC(CCCCC=CC)=O)(CC)CC1 15604,Cc1cc(C(=O)NCCC(C)(C)NC(=O)C(=O)N(C)C)nn1CC(F)(F)F 15605,CC1CCCCC1N1CCCC(CN2CCSCC2)C1 15606,c1(NC2CN(Cc3c(OCC)nccc3)CC2(F)F)ccnc2cc(Br)nn12 15607,CCCC(CCCNC(=O)CCCOC)NC(c1cc(F)ccc1N)=O 15608,c1(C(=O)NC(CC)(C)CNC(c2cc(Cl)c[nH]2)=O)n[nH]c2c1CC(C)CC2 15609,C1(CC(=O)NCCCC(C)NC(c2c(C)nsc2C)=O)CCCNC(=O)C1 15610,C1(C(N2C(CN(C(=O)Cc3ccc(O)nc3)C)CCC2)=O)CC2(CCC2)CCO1 15611,O=S(=O)(c1c[nH]ccc1=NC1CCC(CO)CC1)NCCCC(F)F 15612,C=C(C)CCC(C)(c1nnnn1Cc1ccco1)NC(CCC)CCCC 15613,N1(C(CCS(C)=O)=O)CC2CCC1C(CNC(c1cnc(CC3CC3)s1)=O)C2 15614,Cn1cc(C#N)cc1C(N1CCC(F)CC1C(=O)NC1CN(CCO)CC1(C)C)=O 15615,C1(NC(C2(C)CN(C(c3c(C)cn(C)c3)=O)C2)=O)CCC(N=[N+]=[N-])CC1 15616,N1(C(CC(C=C)C)=O)CCc2sc(CNC(=O)CCn3cc(C)cn3)nc2C1 15617,C1(NC(CC2N(C(CC(CC)C)=O)CCC2)=O)CNCC(F)C1 15618,CC1CCCCCC1Nc1cc(N2CCN(C(=O)N(C)C)CC2)ncn1 15619,c1(OC)cc(C(=O)NC2CCN(C(c3cc(F)cnc3Cl)=O)CC2O)cc(Br)c1 15620,CC1CN(C(=O)CC2CCCSC2)CC(C)N(C(c2cc(O)nc(O)n2)=O)C1 15621,C1(CC=C)(NC(=O)CN2CCCCC2C)CCN(C(c2cnn(CCF)c2)=O)C1 15622,C=C1CCN(C(c2ccco2)=O)C(C(=O)NOCCOCCF)C1 15623,N1(C(CN(CCOC)C)=O)CCC2(C)CN(C(=O)CN(C(=O)C(C)C)C)CC12 15624,CCCCC(C(=O)NCC(C)(C)C#CC(=O)NC1CC(CCF)C1)C(C)C 15625,C1(CC(=O)N(C(C)C(N2CCCC2CC(C)(C)C)=O)CC)COCCO1 15626,C1(NC(COC(C)=O)=O)CCCC2CN(C(c3ccc4cccnc4n3)=O)CC12 15627,C(=O)(C(O)CCC(F)(F)F)N1CCN(C(c2c(CC)nns2)=O)C2C1C2 15628,CC(C)C(C(=O)NCC1(C(=O)NC2CCOC2(C)C)CCCO1)NC=O 15629,c1(OC)cc(C(=O)NC(C)CCCCNC(C2CCCC23CC3)=O)cc(OC)n1 15630,C#CCC(C(=O)N(C(CO)CC(C)C)C)NC(c1cnc(CC)nc1)=O 15631,c1(CN(C2CCCN(C(=O)C(c3ccccc3)F)C2)C)nccc(C(F)F)c1F 15632,C#Cc1ccc(C(=O)NCC(CC)NC(c2ccc(C3CCOC3)cc2)=O)o1 15633,C=C(F)C1(CC(=O)N(CC(C)NC(=O)CCCC(=O)OCC)C)CCOCC1 15634,n1(CC(N2CCC(F)C(NC(C3CC(O)C3)=O)C2)=O)ccc2ccccc12 15635,C=CCC(CC(=O)NCC(N1CCC=CC1)=O)NC(=O)Cn1nc(C)oc1=O 15636,C1(CNC(C(C)(C)OC(C)=O)=O)CN(C(=O)CN2CCS(=O)(=O)CC2)CCCO1 15637,c1(C(N2C(C(=O)Nc3ccc(F)cc3Cl)CC3(CC3)C2)=O)c(Cl)cc(F)cc1Cl 15638,c1(CN2C(C(=O)NC(CCC)CCO)CC3(CC3)C2)c(F)cc(Br)cc1Br 15639,C1(C)(C(N(CC(CC)NC(c2cc(CC)c(C)s2)=O)CC)=O)CCC(=O)N(C)C1 15640,CC(C)C(CCO)N=c1ccnc(NC2CNC(=O)C2)[nH]1 15641,C1(CC(=O)NCC2(C(=O)OC)CCC2)CCN(C(=O)C(C)O)CC1 15642,C(=O)(C1CCc2c[nH]nc21)N1CCC2CN(C(=O)CC3CCSCC3)CC21 15643,C1(C(=O)NCC(C)(C)OCCNC(CCC(=O)OCC)=O)CC12CCCOC2 15644,N1(C(c2c(CC)c[nH]c2)=O)CC(NC(=O)Cc2cc(=O)n(CC(C)C)[nH]2)C(O)C1 15645,c1(OC)cc(=NC(=O)C(C)(C2CCC2)OC(=O)CC2C=CCC2)[nH]n1C 15646,N1(C(C(CC)COC)=O)CCCC12CCN(C(c1cnc(O)n(C)c1=O)=O)C2 15647,c1(C(N)=O)ccc(NCC2CCN(C(C3CCOCC3(C)C)=O)C2)c([N+](=O)[O-])c1 15648,CC(=O)CCN=C1NCC(C)N1.c1(C(C2(C)COCCO2)S(C)(=O)=O)ccc(F)cc1 15649,C(=O)(C(CCCCCN)C(F)(F)F)NC1CC2(CC(C(=O)OC)C2)OCC1 15650,C1(C(=O)NCC(CC)(C)O)CC(OC)CN1C(c1cc(Cl)n[nH]1)=O 15651,N1(C(C2C3(CCC3)C23CCC3)C(=O)NCSc2ccccc2)CCC(F)(F)C(O)C1 15652,c1(C(=O)NCCC(C)NC(c2c(C)scc2)=O)cc2cnccc2[nH]1 15653,C(=O)(CCC1=NNC(=O)CC1)NCC(CNC(C1(C)C=CCCC1)=O)C(F)(F)F 15654,C(CC(F)F)(C(=O)NC1C(O)CC1O)N(C)C(C1CCC1)=O 15655,CCC(CNC(C1CC(=O)CN1C(=O)CSCCC(C)C)=O)(CC)CO 15656,C1(C)(C(=O)NCC(CN(C(C(C=C)O)=O)C)(C)C)CCC2CC2C1 15657,C12(C(N3CC4C(NC(c5c(CC)scc5)=O)C4C3)=O)CCC(CC1)C(C)O2 15658,Cc1cc(=NCc2csc(C)c2C)[nH]c(=NCc2ccnc(O)c2)[nH]1 15659,Cc1ccc(C(=O)NC2COCC2NC(c2snnc2C(C)C)=O)c(Cl)c1 15660,c1(C(=O)NCC(CNC(c2cc(C(C)C)on2)=O)O)cccc2c[nH]nc12 15661,Cc1ncsc1C=CC(=O)N(CCC(C)NC(=O)CS(=O)(=O)NC1CC1)C 15662,C1(CNC(C(CC)N(CC)CC)=O)CCN(C(c2cncc(OC)c2)C)CC1 15663,c1(C(=O)NC2C(OC)CN(C(c3cnn(C(F)F)c3)=O)C2)ccc2cc[nH]c2n1 15664,C1(C(N2CC(NC(=O)Cc3ncc(Cl)s3)C(F)C2)=O)(COC)CCC(=O)N1 15665,C1(c2ccc(CC(=O)OC)o2)COCCN1C(c1ccc(CN(C)C)o1)=O 15666,c1(C(=O)NC2CC(CNC(c3c(COC)scc3)=O)C2)c(F)ccc(F)c1N 15667,C1(NC(C2(OC)CC2)=O)C2CN(C(C3CCCN3Cc3ccccc3)=O)CC12 15668,c1(OC)c[nH]c(C(=O)NC(C)CCCCNC(=O)C(F)n2cccn2)cc1=O 15669,N1(C(C2CC(NC(C3CCCC4CCCCC34)=O)C2)=O)CCOc2ccccc21 15670,N1(C(Cc2nc(C)sc2)=O)CC(NC(c2ccsc2)=O)C2CC2C1 15671,C1(CC(=O)NCC(C23CCC(CC2)C3)NC(C2CC(F)C2)=O)CC2C=CC1CC2 15672,C1(NC(=O)CCc2ccc[nH]2)CCC(NC(C2(C(F)(F)F)CCC2)=O)C1 15673,N1(C(C=C(C)C)=O)CC2CC(NC(c3ccc4ncoc4c3)=O)CC2C1 15674,Cc1ccc2ncc(C(N3CCC4CCN(C(C5(CF)CCC5)=O)CC34)=O)cc2c1 15675,c1(C(N2CC(C)(NC(c3cncc(CC)c3)=O)C2)=O)c(C)cc(F)cc1Br 15676,CC1CN(Cc2ccnn2C)CCC1OC(C1CCCN(C(C)(C)C)C1)=O 15677,N1(C(C(C2CN(C(c3cccnc3O)=O)C2)O)=O)CC2C(C1)C2(F)F 15678,N1(C(C2(C)CC(F)C2)=O)CC(C)CN(C(c2ccc(C3CC3)cn2)=O)C(C)C1 15679,N1(C(C2CC(CNC(CC#N)=O)OC2)=O)C(CO)CCC1C1CC1 15680,C#CCC(O)C(=O)NC(C(=O)NC1CC(CC(N)=O)C1)C1CCOC1 15681,C1(NC(Cc2c(C)nc[nH]2)=O)CC2CCC1CN(C(c1cccc(O)c1C)=O)C2 15682,c1(C(=O)NC2C(C)(CNC(C3C(=C)C3)=O)CCC2)c(S(C)(=O)=O)cnn1C 15683,CS(=O)(=O)CCC(=O)N1CCCC(O)(CNC(=O)CC2(C#N)CCC2)C1 15684,CC(CC(C)(C)C#N)n1ccnc1C(=O)CC(C)(C)C 15685,c1(C(C)(C)C)cnn(CC(=O)OC2CCC2NS(C)(=O)=O)c1.C12CN(C1)C2=O 15686,Cc1cnccc1CNCC(=O)NC(C(=O)N(C)C)C.c1cccs1 15687,Cc1cnccc1C(C)C(=O)NCC(C)(C)CN(C)C(c1[nH]cnc1C)=O 15688,C1(NC(C2COCCO2)=O)CN(C(c2ccc(-n3ccnn3)cc2)=O)CC1(F)F 15689,N1(C(=O)OCC)CC(NC(=NC)NCc2cccc(Cl)c2)C(C)(C)C1 15690,CN1CC=C(CC(=O)NC2(CF)CN(C(c3cnc(S)[nH]3)=O)C2)CC1 15691,C(=O)(CCCCC(=O)OC)NCC1CCC(N(C(C(CCOC)OC)=O)C)CC1 15692,CCCCC(COC)NC(=O)CCN(CCO)C(C1(O)CCOC1)=O 15693,C1(C(=O)NCc2cn(CC#C)nc2)COCCN(C(=O)Cc2scnc2C)C1 15694,c1(C(=O)NCC2N(C(=O)C3=CCCSC3)CCC(C)C2)cnc2ccoc2c1 15695,C1(NC(=O)COC2CCOC2)CCCC1CNC(C1CCOC1C(C)C)=O.O 15696,N1(C(=O)CCCc2cnn[nH]2)CCN(C(C2CC3(CCC3)C2)=O)C(CO)C1 15697,N1(C(C2(OC)CCCOC2)=O)CCC=C(CNC(=O)C(C)C(C)C)C1 15698,C1(CN(C(c2cc(CNC(CCCC)=O)on2)=O)C)CCCCCC1 15699,C1(CNC(c2c(OC)nccc2)=O)CN(C(=O)C(C)(C)OC)CCC1C(F)(F)F 15700,Cc1nnc2n1CCCC2C(=O)NC1CN(C(=O)C(c2ccnn2C)C)C1 15701,c1(C(=O)NCC(CNC(C2=CCC(C)CC2)=O)F)ccc2c(c1)CCCS2(=O)=O 15702,c1(CC(=O)NC2CCN(C(C(C)SC)=O)CC2)cnn2ccccc12 15703,C(=O)(C(C)(C)C)N.n1(C(C)CNC(=O)COCC)cc(C2CCCC2O)nn1 15704,Cc1cc(NC(N)=O)cnc1C.C12CN(CC13CC3)C2=O.C1(=O)CCCCN1C 15705,Cc1nn(C)c(C(=O)NC2CCCN(Cc3ncccc3C(=O)O)C2)c1F 15706,C(=O)(CCC(CF)CF)N1CC2C(NC(C3C(C(C)=O)C3(C)C)=O)(CC2)C1 15707,c1(CCC)nc(C)c(C(=O)NCCNc2ncc(C(=O)OC)cn2)s1 15708,c1(CC(=O)NC2C(CC(C)(C)C)CN(C(C3CCC3)=O)C2)ccc(Cl)cc1F 15709,c1(C2(NC(=O)NCCOC3CN(C(C(C)CO)=O)C3)CC2)cccc(C#N)c1 15710,C(CCN=c1[nH]c(=NCC(C)NS(C)(=O)=O)[nH]c2c(F)cccc12)NC(=O)OC 15711,C(CCC(C(=O)NC(=O)C(=O)OCCCOCCOC)OC(C)(C)C)OCC 15712,c1(N(C)C)ccncc1C(=O)NC1CCN(C(c2coc(O)n2)=O)C1 15713,c1(CN(C(CCC(C)SC)=O)C)cnc(C)c(C)c1.C12CCC(CC1)NC2=O 15714,N1(C(C2CCC(C)(C)C2)=O)CC2CCCC2(CNC(c2ccc(C#N)o2)=O)C1 15715,c1(CC(N2CC(N(C(=O)C=Cc3cnc[nH]3)C)C2)=O)ccc([N+](=O)[O-])cc1 15716,C12(C(=O)NC(c3ccncc3F)C)CCCC1CCN2C(C1CCCCC1O)=O 15717,C1(C(=O)NCC(C)N(C(c2cn[nH]c2)=O)CC)COCCC1(F)F 15718,c1(C(=O)NCc2c(CNC(C(C)CC3CCC3)=O)cccc2)ccc([N+](=O)[O-])s1 15719,C(=O)(C(O)C(F)F)N1CCC(N(C(COCCOCC)=O)CC)C1 15720,c1(C(N2CC(CNC(c3ccn(CC)n3)=O)C2)=O)cc(Cl)cc2c1NCCC2 15721,N1(C(=O)CO)CC(F)(F)CCC1(C)C.C1(CNC(=O)OC(C)(C)C)(C)C=CCC1 15722,N1(C(c2ccc(C(=O)OC)s2)=O)CCC2(CCCN(C(=O)C(O)P(C)(C)=O)C2)C1 15723,N1(C(c2c(C)cco2)=O)CC2(CC(NC(=O)C(F)C3CCC3)CO2)C1 15724,C1(CC)CN(C(c2cc(OC)ccc2Br)C(=O)NC2(C)CC2)C(C)CO1 15725,c1(C(=O)NC(C(CC)CC)C)n[nH]c2c1CN(C(C1(F)CC=CCC1)=O)C2 15726,N1(C(c2cnc(CNC(C3(C)CCCC3)=O)nc2)=O)CC2CCCC(O)C2C1 15727,Cc1cnc(Br)cc1NC(C1(F)CCN(C(=O)CCc2cccc(C#N)c2)C1)=O 15728,N1(C(C2(SCC)CC2)=O)CC(NC(=O)C=C(C)c2ccsc2)C(O)C1 15729,c1(OC)ccc(C)cc1C(N1CC2(C1)CN(C(c1c(Cl)cccc1Cl)=O)C2)=O 15730,C1(NC(c2cc(COC)no2)=O)CC2CCC(C1C)N2C(=O)CCCCCC#N 15731,C1(O)(CCNC(c2nn(C)c(F)c2)=O)CCN(C(c2cnsn2)=O)CC1 15732,N1(C(CCC(=C)Cl)=O)CC(NC(c2cnn(C3CCCC3)c2C)=O)CCC1C 15733,c1(NC(CCSC)C)[nH]c(=NCC2OCCc3ccccc32)nc2c1cnn2C 15734,c1(OC)cccnc1C(=O)NCC1CCC1NC(=O)C(C)C(F)F 15735,N1(S(C2CC(OC)C2)(=O)=O)c2ccccc2C(C)(C)C1C 15736,C(C(C)(C)NC(=O)CCNC(=O)CO)N(C(=O)CN(C)C(=O)C1CC1)C 15737,N1(C(c2n(C)nnc2)=O)CCOC(C(=O)NC2COC3(CCC3)C2)CC1 15738,N1(C(C2C(CCC)C2)=O)CCC2(C(=O)NCC(N3CCOCC3)C)CCCC12 15739,c1(C(=O)NC2CC(CNC(CN(C)C(N)=O)=O)C2)cncc2ccc(F)cc12 15740,c1(C(=O)NCC2N(C(C3CC(C)(C(=O)OC)C3)=O)C3C(C2)C3)cccc(Cl)c1C 15741,CC1CCCC1(C(=O)Nc1ccccc1)NC(=O)CCc1cn(C)nn1 15742,CCC(CC)(CCNC(C1CCC1C)=O)NC(=O)Cc1ccc(C)c(Cl)c1 15743,C1(C(N(C(C)C)C)=O)COCCN1C(C1CC1C(C)(C)C)=O 15744,Cc1[nH]nc2c1CCC(C(N1CCC(C)(CNC(c3c(Cl)n[nH]c3C)=O)C1)=O)C2 15745,Cc1cc(F)c(F)cc1C(=O)NC1CN(C(c2ccc(F)c(F)c2)=O)CC1F 15746,Cc1cc[nH]c1C(=O)NCC1CC(NC(C2CC2c2ccn(C)n2)=O)C1 15747,C1(C(N2CCCC(OCCC)C2)=O)CCN(C(=O)CCC2CCC(=O)C2)C(C)C1 15748,CCCCCCCCC(=O)NCC(C)(CC(C)C)NC(=O)CC1CC1(Cl)Cl 15749,N1(C(CCCC=C)=O)CC2CCC2(CCNC(=O)COc2c(C)cccc2F)C1 15750,c1(C(=O)NCCCCNC(=O)C(C2CCCO2)C2CC2)ccc2c[nH]nc2c1 15751,C12CCN(S(=O)(=O)NCC(=O)N1)CC2.C1(OC)CCSC1 15752,c1(C(N2CCCCC(NC(c3ncn(C)n3)=O)C2)=O)ccc(Br)cc1C#N 15753,c1(C(N2CC(CC=C)(NC(C3(F)CCOC3)=O)C2)=O)ccc(C)c(C)n1 15754,c1(C(=O)NCC2(NC(c3c(C#C)c[nH]n3)=O)CCCCC2)cc(C)ccc1O 15755,CCC(CC(=O)NC(C)(C)CNC(=O)CCCNC(c1ccccc1)=O)C(F)F 15756,Nc1cnc(C(F)(F)F)cc1C(N1CCC(F)(CNC(C2CC(F)C2)=O)C1)=O 15757,S(=O)(=O)(c1cncc(Br)c1)N(CC)Cc1cccc(C2CC2)c1F 15758,C1(O)(CCNC(c2c(C)nc[nH]2)=O)CCN(C(C2(C)CC2(Cl)Cl)=O)C1 15759,C1(C(N2CC(CC)OCCC2)=O)CC(N=[N+]=[N-])CN1C(=O)CC1CCC(C)(C)O1 15760,c1(C(=O)NC(CO)C(O)C2CCCCC2)cnn2ncccc12 15761,c1(OC)cc(CCC(=O)NC23CC(NC(=O)CC4CCCO4)(C2)C3)ccc1O 15762,c1(OCC)cccc(C(=O)NC2CCC(CCNC(C3(OC)CC3)=O)C2)c1 15763,CC(C)C(C)C(C)CC(=O)NCCC1CC(NC(=O)COc2ccccc2F)C1 15764,C12(C(N3CCC(C(=O)NC(c4ccccc4)CC)C3)=O)CC1CN(CC)C2 15765,C1(C(c2nnnn2C(C)C(=O)OC)(C)NCc2ccn(CC)n2)CCCCCC1 15766,C1(C(C(=O)NC2CC2)N(C2CCCOC2)C)CCC2CC2C1 15767,C(=O)(C1CCCc2ncnn21)N1CC(C)(NC(c2ccc(S(N)(=O)=O)cc2)=O)C1 15768,N1(CCC)CC(C(=O)NCCC2(C)CCN(C(c3cncnc3C)=O)C2)CC1=O 15769,CC(C)CC(C)(O)C(=O)NCC12CCC(CC1)N(C(C1CCSCC1)=O)C2 15770,C(CC(F)=C(F)F)NC(C12CC(CNC(=O)C=Cc3cc[nH]c3)(C1)C2)=O 15771,c1(CC2CCC(C)(C#N)CC2)cccc2c1CN(C1CCS(=O)(=O)C1)C2=O 15772,c1(OC)cc(C)c(Cc2ccccc2Nc2cc(Br)c(N(C)C)cn2)c(C)c1 15773,C1(CC=C)(NC(c2cnccc2C)=O)CCCN(C(C2CC(OC)C2)=O)C1 15774,N1(C(c2cccc(CC)n2)=O)CC2CN(C(=O)Cc3cc(O)nnc3O)CCC12 15775,N1(C(C(C)NC=O)=O)CCCCC1C1(C(=O)NCC2(F)CCOCC2)CC1 15776,c1(C(N2CC(c3n(C)ncc3)OCC2)=O)cc2c(n1C)CCOC2 15777,Cc1ccc(C)n1CC(=O)NCCC(C)N(C)C(C1CC(CCO)C1)=O 15778,C1(C(N2C(C(=O)Nc3c(C)nn(C)c3)CC2)=O)CCCC2(CC2)C1 15779,C1(C(=O)NCC2(NC(C3CC(CC)C3)=O)CCOC2)CC2CC1CC2O 15780,c1(C(=O)NCC2C3CN(C(c4nc(C)sc4)=O)C2C3)c[nH]c2cc(F)c(F)cc12 15781,c1(CNC(=O)C=Cc2cn[nH]c2)ccc(C(=O)NC(C2CCOC2)CO)nc1 15782,c1(C(=O)NCC(C)CNC(c2ccccc2Cl)=O)ncc(C(F)(F)F)cc1O 15783,c1(NC(=O)NCC2CCC(C)CC2)ccc([N+](=O)[O-])cc1I 15784,c1(NC(C2C3CN(C(c4n(C)cnc4)=O)C2C3)=O)cc(Cl)nnc1Cl 15785,C1(CC(=O)NCC(C(C)C)(C)NC(C2C(F)(F)C23CC3)=O)CCCCCCC1 15786,C(=O)(C1=CNS(=O)(=O)N=C1C)NC12CCCN(C(C3CCC(CC)O3)=O)CC1C2 15787,c1(NCC2C(C(C)C)C2)ccc(S(=O)(=O)NCCC2OCCC2C)cc1Cl 15788,N1(C(C2OCC(C)C2)=O)CCOCC(CNC(=O)CC2NC(=O)NC2=O)C1 15789,C(CC(F)F)(C(=O)N1CCC(CN(C)C)C1)N(C(CCc1onc(C)n1)=O)C 15790,C1(NC(C(C)Oc2ccc(C#N)cc2)=O)CC2CN(C(=O)C(Cl)=CCl)CC2C1 15791,CC(c1ccccc1)=CC(=O)NCC1CN(C(C2(C(F)(F)F)CC2)=O)CCN1C 15792,CC(C)CC(C(=O)NCC(C)(C)CCNC(=O)CC1CCCN1C)C(C)C 15793,C1(CC(=O)NCC=CCNC(C2CC3OC(=O)OC3C2)=O)CCc2sccc2C1=O 15794,C(CCS(=O)(=O)c1ccccc1)N(C)S(=O)(=O)N.CCCC 15795,c1(C(N(C2CC(NC(CN(CC)CC)=O)C2)C)=O)cnn2c1CCCC2 15796,N1(C(C(C)=CC)=O)CCC(NC(=O)CC(O)c2ccccc2)C1(C)C 15797,c1(C(=O)NCC(C)NC(c2cc(-n3ccnc3)ccc2Cl)=O)cc([N+](=O)[O-])n[nH]1 15798,N1(C(=O)CC2(C3CC3)CC2)CC2ON=C(CNC(C3(CO)CC(F)(F)C3)=O)C2C1 15799,c1(NC(CC)C(c2ccccc2F)O)ncnc(NCC2COCC2(C)C)c1C 15800,n1(CC)nc(C2CC2)cc1C(=O)NC1CN(C(C2CN(C(=O)C3CC3)CCO2)=O)C1 15801,C1(S(N)(=O)=O)(C(=O)NCCNC(C(c2ccc(Cl)cc2)(C)N(C)C)=O)CCCC1 15802,C1(C(=O)NC2CN(C(c3n[nH]c(C)c3O)=O)CC23CC3)CCc2cn(C)nc2C1 15803,CC1(NC(C2CC(NC(c3n[nH]cc3Cl)=O)CCO2)=O)CCC(O)CC1 15804,C=CCC(C(=O)NCCCOC1CCCCCC1)C(C)C 15805,c1(C(=O)NC2CC(C)(NC(c3cnc[nH]3)=O)C2)ccc(-c2ccon2)cc1 15806,C(=O)(C1COc2ccc(F)cc21)N1CCC(NC(C2(C(F)(F)F)CC(=C)C2)=O)C1 15807,c1(C(N(C2CCCN(C(=O)Cn3nccc3C)C2)CC)=O)cnn2c1OCCC2 15808,c1(SC)c(C(=O)NC2CCCCC2NC(c2nc(C3CC3)oc2C)=O)cnn1C 15809,c1(SCCC)ccc(C(=O)NCC2CC(NC(=O)C(F)CC)C2)cc1 15810,c1(C(N2CC3CC2CO3)=O)cc2n(n1)CCCN(Cc1cc(F)c(Cl)c(F)c1)C2 15811,N1(C(C2(C=C)CC2)=O)CCC(C2(CNC(C3CCC(=O)N3)=O)CCOCC2)CC1 15812,c1(CNC(C2CC(O)CN2C(=O)CCN2CCOCC2)=O)cc(F)c(O)cc1F 15813,C=C(C)C1OCCC1CNC(=O)NCc1cc(OC(F)F)ccc1F 15814,c1(OC)ccc(Br)c(NC(C2CC2NC(c2ccc(C)cc2O)=O)=O)n1 15815,c1(OC)cccc(C(=O)NCC2CC(C)CCN2C(=O)C(C2CC2)OC)c1OC 15816,CC(C)C(CNC(c1cn(CC2CC(CF)C2)nn1)=O)NC(C1CC12CCC2)=O 15817,c1(C(N2C(CN(C)C(C3CCCN3N=O)=O)CCCC2)=O)ccc2ncsc2c1 15818,C1(CN(C(c2ccc(N)c(F)c2)C(=O)Nc2c(C)cccc2)C)CCS(=O)(=O)N1C 15819,N(C(=NCCSC)N1CCC(c2nncs2)C1)NC(N1CCC(CC)C1)=O 15820,N1(CCNC(c2c(OC)nsc2)=O)CCC(NC(=O)C#CC(=O)N(C)C)CC1 15821,C1(NC(C=CC)=O)CCN(C(=O)CCOc2ccccc2C(N)=O)C(C)C1 15822,c1(C(N2CCC(C(CNC(C(=O)NCC)=O)F)CC2)=O)c[nH]c(=N)cc1C 15823,C(c1nc(C)co1)=CC(=O)NCC(c1ccccc1F)NC(CC1CC(=C)C1)=O 15824,C12(CNC(c3n(C)ccc3)=O)CCCC1CCN2C(c1csc(CO)n1)=O 15825,CC(CN=c1nc(N2CCc3ncncc3C2)c2c([nH]1)COC2)c1nccs1 15826,c1(OC)cc(C)cnc1C(N1CC(CNC(c2cc(C)co2)=O)C(C)(C)C1)=O 15827,C1(NC(C(COC)O)=O)C2CCN(C(=O)CCSc3nnnn3C)C12 15828,CCC(C(=O)N1CCCC1CC(=O)NC(C1CC1)C1CC1)NC(N)=O 15829,N1(C(CSCC(C)C)=O)CC2CC1CCC2NC(c1c[nH]c(C(N)=O)c1)=O 15830,Cc1cccc(OCCC(N2CC(NC(=O)Cc3occc3C)C(C)C2)=O)c1C 15831,c1(C(=O)NC2C(NC(C(CC)N(C)C)=O)CCOC2)cccc2[nH]cc(C#N)c12 15832,C1(C(N(CCNC(C)=O)C)=O)CC2CC1CC2NC(c1cncc(O)c1)=O 15833,Cc1cc(C(=O)NCC2CCN2Cc2ccsc2Cl)ccc1[N+](=O)[O-] 15834,N1(C(C2CNC(=O)O2)=O)CCCCC1CNC(C1CCC(O)CC1)=O 15835,c1(C(=O)NC(CC(C)C)C(=O)N2CCC(N3CC=CC3)C2)ccn2ccccc12 15836,C#CCCCC(C)C(=O)N1C(CNC(=O)Cn2ccccc2=O)CC2CCCC12 15837,C(=O)(C(C)CN(C)C(C1CCSCC1)=O)NCC(c1ncco1)C 15838,C1(N(CCCN2CCN(C)CC2)C(c2nn(CC)c(C)c2)=O)CCNCCC1C 15839,C=CCC(C)(C)C(=O)N1CCN(C(C2CC23CC(OCC)C3)=O)C(CCC)C1 15840,N1(C(Cn2ncc(CC)c2)=O)CC(CN(C(=O)CCCC#N)CC)CCC1C 15841,N1(Cc2ccc(C#N)cc2)CCC2CN(C(c3csc(Br)c3)=O)CC2C1 15842,c1(N(CCCC(N2C(CNC(C(CC)C)=O)CC(O)C2)=O)C)ccc(C)c(C)c1 15843,N1(c2nccc(C)n2)CCC2(CCC(NC(c3cc4c(s3)CCC4)=O)CC2)C1 15844,O=C1NCCCCC1C(=O)OCCCNC(c1ccccc1Br)=O 15845,C=C(C)CN=c1[nH]c2c(c(=NCCCC3CCCC3)[nH]1)CC(C)CC2 15846,N1(C(C(n2cc(C(C)NC(C)(C)NC(N)=O)nn2)C)=O)CCCC2CN(C)CCC12 15847,c1(CC(=O)NC2CCCC(NC(CCS(N)(=O)=O)=O)C2)cnc2c(=O)[nH]ccn12 15848,CCCCCCC(=O)N1CCCC(CN(C)C(C2CCCNC2=O)=O)C1 15849,Cc1ccc(C)c(C(=O)NCc2cc(C(N3CCC4CC34C)=O)on2)n1 15850,N1(C(CC(CC)OC)=O)CCc2nc[nH]c2C12CCN(C(=O)C=CI)C2 15851,c1(C(=O)NC2C(CNC(COC)=O)C2)cc2ccccc2nc1C(F)F 15852,N1(C(=O)NCC(c2cnn(C)c2)Oc2ccc(C)cc2)CCC2(CCCC2)CC1 15853,c1(C(N2CC3C(C(N(C(C)C(N)=O)C)=O)(C3)C2)=O)c(O)cccc1F 15854,C1(CC(=O)NCCC2C=CCC2)(NC(C2C(CC)OCC2)=O)CCOCC1 15855,C1(C(N(C2C(C)C(C)CCC2)C)=O)CCC(C)(C)N(C(=O)C=CCN2CCC2)C1 15856,C12CCN(CC1)C2=O.C1(C)(CN(CC(=O)Nc2ccccc2)C)C=CCCC1 15857,C1(NC(C2CN(C(C=C(CCN(C)C)Cl)=O)CC2CO)=O)CC2CCCCN2C1 15858,N(C(=NCCOC1CCC1)NCC1CCNC(=O)C1)C1C(C)C1 15859,c1(OCC)cc(C(=O)NC(C)CSC2CN(C(C)=O)C2)[nH]n1 15860,C(=O)(CC(O)CCCCC)NCCCOCCC(N1CC(C#C)N(C)CC1)=O 15861,N1(C(CCC2CCN(C(CC(COC)C)=O)CC2)=O)CC2(C1)CN(C)C2 15862,c1(OC)ccccc1C1(OCC(N2CC(n3c(O)nnc3O)C2)=O)CCC1 15863,C1(C(N2CCC(CNC(CCN(c3ccncc3)C)=O)C2)=O)CCC2(CC2)C1 15864,CC(C)CC(CNC(C1(C)CCCCO1)=O)C(=O)NCc1cccnn1 15865,C(C1CC1)(C1CC1)=CC(=O)NC1CC(NC(C2CSCC2c2ccccc2)=O)C1 15866,C(=O)(CS(=O)(=O)C(C)(C)C)N1CCC(OC)(CNC(C2CCC(CO)CC2)=O)C1 15867,N1(C(c2cccc(SC)c2)=O)CC2CCC1CN2C(=O)C(C)(C)F 15868,c1(N2C(CN(C(C(C(COC)C)C)=O)C)CCC2)ncc2c(Br)cccc2n1 15869,C(=O)(C(C)C(F)(F)F)N(C(C)C)CCN(C(=O)C(O)Cc1ccc(Cl)cc1)C 15870,C(=O)(C(F)(CNC(=O)CCc1cnco1)C(C)C)NC(c1cccs1)CC 15871,c1(C(=O)NCCC2CCN(C(C(C)OCCOC)=O)CC2)nccc2n[nH]cc12 15872,C(CCCC(=O)NCC1CCC(NC(=O)CC2CCCN2C)CC1)OC(C)C 15873,C1(CN(C)C(=O)OC(C)(C)C)(CO)CCCN(C(=O)Cc2c(F)cccc2Cl)C1 15874,C(c1cccc(O)c1)=CC(=O)NCC1CN(C(c2cccc(C)n2)=O)CC1C 15875,C1(NC(c2c(C)[nH]cc2)=O)CCC12CN(C(C1CCN1S(C)(=O)=O)=O)C2 15876,O=C1CCC(CC(N2CCC(O)(C(=O)O)C2)=O)CN1 15877,N1(C(Cc2c(C)nc(C)s2)=O)CC(C)CN(C(c2cn(C(C)C)cn2)=O)C(C)C1 15878,C1(C(=O)NCC2(NC(=O)Cc3ccccc3Cl)CCC2)CCC(F)(F)CC1 15879,c1(C(N2CCC(CNC(CNS(NC)(=O)=O)=O)C23CC3)=O)cc2ccncc2[nH]1 15880,N1(C(CCOC)=O)CC(=O)NCC1C(=O)NC1(CN(C)C)CC1 15881,C1(C(=O)OC(CC(=O)OCC)CC#N)CC2(CCCCC2)C1 15882,C#CCC(C)(CC)C(=O)NC1CC12CCN(C(c1cc(COC)oc1C)=O)CC2 15883,C(CCCCC(=O)NC1(C2CCCCN2C(=O)C(C)n2cccn2)CC1)OCC 15884,Cc1cnccc1CN(C)C(c1cc(C2CC2)nn1C(C)(C)C)=O 15885,C1(NC(=O)C=Cc2ncc[nH]2)CC2CC1N(C(C1(c3ccc(F)cc3)CC1)=O)C2 15886,C1(CN(C(=O)Cc2conc2C)CC)CCCN1C(c1coc(Cl)c1)=O 15887,N1(c2n(CC=C)c(C(c3ccc(F)cc3)CC)nn2)CCCc2ccccc2C1 15888,C1(C2(O)CN(C(C3(Cl)CC3(F)F)=O)C2)(CNC(CC=CCC)=O)CC1 15889,c1(OC(C)=O)cccc(C(N2CCN(C(c3cnc(O)cc3C)=O)CC2)=O)c1C 15890,C(C)(CCCCN=c1nc2c(cnn2C)c(NCC(C(C)C)C(C)C)[nH]1)SC 15891,Cc1csc2ncnc(N3CCCCC(CNC(=O)CCc4cc[nH]n4)C3)c12 15892,c1(CCOC)n[nH]c(=NCCCN(C)C(C2CCCC2OC)=O)s1.c1cccc(F)c1 15893,c1(-c2ccc(C(=O)OC)cc2)ccc2c(c1)CCN(c1cc3ncnn3cn1)C2 15894,c1(N2CC(O)(CCNC(c3c(C)noc3C)=O)C2)ncnc(Cl)c1C 15895,O=C(C1=NOC(C2(O)COC2)C1)NC1(C(N2C(Cc3ccc[nH]3)CCC2)=O)CC1 15896,c1(CC(N2CC(CCNC(C)=O)C2)=O)c(N)nc(C)nc1O 15897,C(C(C)CC(F)(F)F)OCCOCC.c12cccc(c1)N2 15898,Cc1csc2ncc(C(N3CC4CC4(NC(C4CC5(CCC5O)C4)=O)C3)=O)n12 15899,N1(C(c2cc(O)cs2)=O)CC2CC(C1)N(C(=O)CC1CCCC3(CCC3)O1)C2 15900,C1(n2cc(CCCOC)nn2)CCCC=C1Br.C1CC(C)N1 15901,C1(N(C(=O)Nc2ccccc2)C(C)C2CC2)CCN(C(c2ccoc2)=O)C(C2CC2)C1 15902,c1(C(N(CCNC(C=Cc2cc(C)no2)=O)C2CC2)=O)ccccc1S(C)(=O)=O 15903,C1(NC(c2n(CC)ncc2)=O)CC2CCC(C1)N2C(c1nonc1N)=O 15904,Cc1cc(=NC(=O)C=C2CC3C2CCN3CCCF)[nH]o1.C1(=O)C(C(C)(C)C)N1 15905,N1(C(c2n(CC)ccc2)=O)CCC(CC(C)NC(C2(OC)CCOC2)=O)CC1 15906,Cc1cc(NC(C2CN(Cc3cccc(C#N)c3)CCO2)=O)cnc1F 15907,Cc1cc(C(=O)N(C(C(=O)NCC2(C)NC(=O)NC2=O)C2CC2)C)nc(O)n1 15908,C1(C2CCN(C(C=C(C)C3CC3)=O)C2)CCCCN1C(=O)CC1CCCOC1 15909,CC1CC(C)N(C(=O)CC(C)(C)C)CCN1C(c1nc2cc(Cl)ccc2s1)=O 15910,c1(NCc2cc(C)cc(F)c2)ccc2c(c1)CCC2NC(=O)OCC(C)(C)C 15911,c1(C(N2CC3CCN(C(CN(CCC#C)C)=O)C3C2)=O)cnc2c(c1)CCCO2 15912,C1(NC(c2c(CC)cno2)=O)CN(C(=O)Cc2cscn2)CCC1O 15913,C12(C(N3C(CNC(c4nccc(C(C)(F)F)c4)=O)CCC3)=O)CCC(CC1)OC2 15914,C1(NC(=O)CC2CCSCC2)CC2CC1N(C(=O)C1=CSCS1)C2 15915,n1(CCC)nc(CC2CCC2)nc1-c1nc(-c2ccncc2)ns1 15916,C1(NC(c2c(CC)nc(=N)[nH]c2)=O)CCN(C(=O)CC2COCC2O)CC1(C)C 15917,Cc1csnc1C(=O)NC(Cc1ccoc1)C(=O)NC(C)CCC1CC1 15918,c1(C2NCCN(C(c3cccc(F)c3COCCN)=O)C2)ccc2ccoc2c1 15919,C(=O)(C(F)CCCC)NC(C1CCN(C(CCC=CC)=O)CC1)CO 15920,C1(NC(c2cc(CC)n(CCO)n2)=O)CN(C(c2nocc2C)=O)CCC1O 15921,c1(OCC)ccc(OC(c2nnn(C)c2Cc2ccccc2)=O)cc1C(F)(F)F 15922,Cn1ncc2c1CCN(C(=O)CC1(C)CCN(C(=O)C(O)CC3CCCC3)C1)C2 15923,c1(C(N(C2COCC2C(N)=O)CCNC(C2(CC#C)CCC2)=O)=O)cc(C)c[nH]1 15924,C1(CNC(=O)NCc2cnc(Br)s2)CC(O)CN1C(=O)C(Cl)(Cl)Cl 15925,C(N=c1[nH]c(N(CCCN2CCCC2=O)C)nc2c1SCC2)C(C)(C)N(C)C 15926,c1(NC(C2(C)CCCN2C(=O)Nc2cccc(Cl)c2)=O)nc(Cl)c(Br)cc1I 15927,N1(C(CCC#N)=O)CCC(O)(CNC(C2CC23CCOCC3)=O)CC1 15928,N1(C(C(c2n(C)ccn2)O)=O)CCCC2(CC(NC(=O)C(C)(C)CF)C2)C1 15929,c1(OC)ccc(CN2CCC(Cc3ccc(SC)c(C#N)c3)CC2)cc1[N+](=O)[O-] 15930,C(C(O)CC(=O)NC1CC(CNC(=O)C(N2CCOCC2)C2CC2)C1)N(C)C 15931,Cc1ccc(C2(NC(=O)NCC3CCC(S)CC3)CCC2)cc1.c1nn[nH]n1 15932,C12(NC(C3C(CNC(c4c[nH]c(=S)cn4)=O)OCC3)=O)CC1COC21CCC1 15933,N1(C(c2c(CCC)occ2)=O)CCC(C2CCN(C(=O)CCCCO)C2)C1 15934,C(=O)(C(CCC)S(N)(=O)=O)NC(CCC)CCCNC(=O)Cn1nc(C)nc1C 15935,C1(F)(C(=O)NCC(CNC(C2(CC3CCC3)CC2)=O)CO)CCCOC1 15936,c1(C(=O)NC2(CF)CCN(C(=O)CC3(C(F)(F)F)CC3)C2)cccc2nc[nH]c12 15937,Cc1nc(C(N2CC(NC(=O)COc3cccc(F)c3F)CC2C)=O)cc(O)n1 15938,C=CCC(C)(C(=O)N1CC(O)(C(C)NC(=O)CCc2cnn(C)c2)C1)N(C)C 15939,N1(C(C(CC)Sc2cccc(C)c2)=O)CCC2(CC1)CN(CC1CNC1)CCO2 15940,C1(NC(=O)C(=O)c2ccco2)COC2(C1)CN(C(c1nc(Cl)ccc1F)=O)C2 15941,c1(NC(C(C2CCCC2)OC)=O)ccc(NC(=O)C(C)=CC(C)(C)C)c(C)c1 15942,N1(CC(=O)NC(C)CCNC(=O)CCc2nc[nH]n2)CCCOC1=O 15943,c1(C(N2CCCC(Nc3nc(COC)nc(O)c3)C2)=O)ccc(F)c(C#N)c1 15944,Cc1cc(C(=O)NC2CC(NC(C3CCCN(CC(C)C)C3)=O)C2)ncc1C#N 15945,C1(C2(O)CN(C(C3C(C)C3C)=O)C2)(CNC(C2(C)N(C)CC(OC)C2)=O)CC1 15946,c1(C(=O)NC(CC)CNC(C2(CF)CC2)=O)ccc2c(n1)NC(=O)CO2 15947,c1(C(=O)NC2CN(C(C3CCC(F)(F)C3)=O)C2)cnc2cccnc2c1 15948,c1(N2CCC(CNC(CC(CC)OC)=O)C(C)C2)ncnc2n[nH]c(C)c12 15949,C#CCC(C)(C(=O)NCc1nc(C)ccc1C)NC(=O)CC1CC(SC)C1 15950,N1(C(C2(C)CCCS2)=O)CCC(OC(C)=O)CC1.C(=O)(C(F)(F)C1CCOCC1)NC 15951,C1(NC(CCCCN(C)C)=O)CCCC12CN(C(C1CN3CCCC1C3)=O)C2 15952,CON1CCC(C(=O)N(CCNC(C2CCCC(F)C2)=O)C2CC2)CC1 15953,c1(NC(=O)NCCc2nc(C(F)(F)F)cs2)cccc(Oc2ccc(F)cc2)c1 15954,C1(C(=O)NC(c2ccco2)COC)CN(C(=O)Cn2nc(C)nc2C)CC1C 15955,C1(N(C)C(c2ccc(-n3cccc3)cc2)=O)CN(C(=O)C(C)(F)F)CCC1O 15956,c1(C(=O)NCC(CC)NC(C2CCC(C)(C)CC2)=O)csc2cncn12 15957,CCCCCCC(C(=O)N1CC(CNC(=O)C(CCC)C(C)C)C1)N1CCOCC1 15958,CC(CC(=O)NC1(C)CCN(c2cc(C3CC3)ncn2)C1)C(F)(F)F 15959,CC1(F)CN(C(=O)CSC(F)F)CCN(C(=O)CN2CCC(F)CC2)C1 15960,CN1CCCCC1C(=O)NC1CCN(C(=O)NS(C)(=O)=O)C1.c12ccnc(c1)N2 15961,C1(C(=O)NC2(CF)CCN(C(C3C(OC)(OC)CC3)=O)C2)CC2(CCCC2)CO1 15962,N1(C(C2C(CC(C)C)C2)=O)CC(NC(=O)C(=O)N(C)C)C2(CCOCC2)C1 15963,Cc1cc2c(C(N3CC4CC(NC(C5CCC(C)CC5)=O)C3C4)=O)nccn2n1 15964,C(CC1=CCCCC1)N(C)Cc1cc(-c2ccc(Cl)cc2O)on1 15965,O=C1C=C(C(=O)NNC(=O)C(O)C2CCC2)S1 15966,C1(C)(NC(=O)NCC2CCC(C(=O)OC)O2)CCCC(C)(C)C1 15967,C1(C(N(C2CCCC(NC(=O)COCCCF)C2)C)=O)Cc2cccnc2C1 15968,C12(C(=O)NCC(C(=O)OCC)Cc3ccccc3)CCCC(C1)C(=O)NC2 15969,C1(C(N(CC2CN(CC)C(=O)O2)Cc2ccccc2)=O)CCOCC1(C)C 15970,Cc1nc2cc(F)ccc2cc1C(=O)NC(C)CNC(c1ccnn1C)=O 15971,S(=O)(=O)(c1ccc(NCCCC2CC2(Cl)Cl)cc1Br)NCc1cncc(OC)n1 15972,c1(-c2cccc(NC(N3C(C(=O)O)CCOCC3)=O)c2)c[nH]c2ccc(Cl)cc12 15973,C1(CC(N2CCC(Nc3cc(SC)ncn3)C2)=O)CCC(=O)NC1=O 15974,CC1(C)CC(C(N2CC(OC(=N)O)C2)=O)CN(C(c2cnc(S)nc2)=O)C1 15975,C1(NC(CCOCCOC)=O)C(C)(C)C(NC(c2cc(F)n[nH]2)=O)C1(C)C 15976,N1(C(C2N(C)C(=O)NC2)=O)CC2(CC2)CC1CNC(=O)CCC(F)(F)F 15977,C(C#CC(F)(F)F)NC(C1CCCN1C(=O)CNC(=O)NC1CCCC1)=O 15978,N1(C(CC2(C)CC2(F)F)=O)CCC2(CCN(C(=O)CC3(O)CCOCC3)CC2)C1 15979,C1(C(=O)OCC)CC(NC(=O)NCc2ccnn2CC(F)F)CCO1 15980,C(CCCCC(=O)N1CC(N(C)C(c2c(C)cnn2C)=O)C1)OC 15981,Cc1cc(F)cc2[nH]c(C(=O)NCC34CC3CN(C(=O)C3=CCOC3)C4)cc12 15982,C(=O)(C1=CCN(C(C2CC(=O)N(OC)C2)=O)C1)NC(CC)CCCO 15983,c1(C(=O)NC(C(=O)NC(C#C)Cc2ccco2)C2CC2)cc([N+](=O)[O-])c[nH]1 15984,C1(CNC(CCCN(C(=O)C(F)C(C)(F)F)C)=O)CCC2(CC1)CC2 15985,c1(CCC(=O)NCCOCCN(C(C(c2cncnc2)C)=O)C)n[nH]cc1Br 15986,c1(C(=O)NCCC2CC(NC(CC=C)=O)C2)cn(-c2ccn(C)n2)cn1 15987,S(=O)(=O)(c1ccccc1[N+](=O)[O-])OCCOCC.C=CC1CN2CC1OCC2=O 15988,C1(C(=O)NC(CNC(Cc2nc(C)sc2)=O)C(C)C)C2CCC3C(C2)CC13 15989,C(=O)(C(CC(C)C)N(C)C(C1CNC(=O)O1)=O)N(C(CC)C1CC1)C 15990,N1(C(C(C=C)(C)O)=O)CC2CCC(C1)C(NC(c1ccccc1OC)=O)C2 15991,C1(O)(C(c2n(CCC)nnn2)NCC2COC2)CCCN(C(=O)OC(C)(C)C)C1 15992,N=c1nc2c(c[nH]1)CCN(N1CCC(c3nc4ccccc4s3)CC1)C2 15993,N1(C(C2N(C)CCCC2)=O)CCCCCC(NC(=O)Cc2ccc(F)cc2F)C1 15994,C1(C)(CNC(c2ccc(C(C)(C)C#N)o2)=O)CCOC2(CCC2)C1 15995,CC(O)C(C)C(=O)NCCC1CCCN1C(=O)Cc1csnn1 15996,C1(NC(C(C)Cc2cnco2)=O)CCNCC1c1cccc(F)c1 15997,C(=O)(CC(C)(O)C(F)(F)F)NCC(C)NC(CCC(=C)Cl)=O 15998,C1(NC(C(C)OCCCC)=O)CC(C)(C(=O)N(CCO)CCO)C1 15999,C1(NC(C(C=C)C)=O)CCN(C(=O)C(CC2CC2)OC)CC1(C)C 16000,N1(C(c2cc(C)nc(C)n2)C(=O)NC(CC)C)CCc2ccc(F)c(Br)c2C1 16001,c1(C(C)OC)noc(CC(N2CC(c3nc(C(F)(F)F)cs3)C2)=O)n1 16002,N1(C(c2cnc(C(C)=O)s2)=O)CCCC(C)(NC(C2C(F)(F)C23CCC3)=O)C1 16003,c1(C(N(c2c(C)cccc2Cl)C)=O)ccc(S(=O)(=O)Cc2nn[nH]n2)cc1 16004,c1(C(N(CCCC(=O)NC2(CN(C)C)CC2)C)=O)cc(C(N)=O)[nH]n1 16005,N1(C(CC2N(C(C)=O)CCC2)=O)CCCCC(N(C(=O)CCC(=O)N(C)C)C)C1 16006,c1(C(N2CCC(C)(NC(c3cnn(C)c3F)=O)C2)=O)ccc2ncncc2c1 16007,n1(C2CCCN(C)C2)ccc(=NC(=O)C(=O)N2CCC(N(C)C)CC2)[nH]1 16008,N=c1cc[nH]cc1CNc1ccccc1C(=O)Nc1cncc(C(N)=O)c1 16009,c1(OCC(=O)NCCN(C(C(CCCC)C)=O)C)ccc2c(c1)CCCC2 16010,C(CC(C(=O)NCC1CCCC1(C)C)NC(c1cncc(C)n1)=O)=CC 16011,CCCC(C)(O)C(=O)NCC1CCCC1C(=O)NC1CN(C)CCC1O 16012,c1(C(=O)NCC2(COC)CCCN2C(c2scnc2Cl)=O)cc2ccccn2n1 16013,S(=O)(=O)(c1cccc(NC(N2CCC(c3nncs3)C2)=O)c1)N1C(C)CCCC1 16014,C(=O)(CS(N)(=O)=O)N(CCCCCNC(C1(C)CC1Br)=O)C 16015,c1(C(N2CC(C)CC(NC(CC3(OC)CC3)=O)C2)=O)cc2n(n1)CCCO2 16016,C1(OC)CCC(C(F)(F)F)(NC2CCCN(Cc3nccn3C)C2)C1 16017,C1(C(=O)N(C)CCNC(c2ccn(C(C)C)n2)=O)(CC)CCOC1 16018,CN1CC(C(=O)NC2CC(F)(CNC(=O)Cn3cnnc3)C2)C(C(F)(F)F)C1 16019,C12(CNC(C(=O)N(C3CC(OC)C3(C)C)C)=O)CCC(O)C1CC2 16020,C1(CN(C(=O)CC2CCOC2)C)CN(C(=O)CCc2cccs2)CC12CC2 16021,CC1CCC(NC(=O)CCCCN(C)C)C(=O)N1 16022,C(c1cccc(F)c1)=CC(=O)NCC(C)(F)CNC(C1CC(F)(CF)C1)=O 16023,C1(c2cccc(OC)c2)CCN(Cc2nnnn2CC(F)(F)F)C1(C)C 16024,CC(C)(C)C(O)C(=O)NCC1(c2cccc(C(F)(F)F)c2)CCCC1 16025,N1(C(CC(CC)OC)=O)CC(C)(C)C(NC(c2cnc(Cl)s2)=O)C(C)(C)C1 16026,Cc1cccc(C(=O)NCCCCCNC(C2(C3CCCCO3)CC2)=O)c1O 16027,N(C(=NCC1CCN(c2ncccc2F)C1)NCC1CCCO1)CC(C)(C)C 16028,C1(NC(=O)Oc2ccc(Br)cc2Cl)CCCN(CCO)C1=O 16029,C1(CC)CCCN1C(=O)C(=O)NC1CCC1NC(C1(CC2CC2)CCCC1)=O 16030,C(=O)(C(C)CC(F)F)N(C1CCN(C(c2ccc(C(C)C)s2)=O)CC1)CC#C 16031,N1(C(CCc2n(C)ccn2)=O)CCC2(CC2C(=O)NCC2CC3C=CC2O3)C1 16032,Cc1cc(C(=O)NCC2CC(C(=O)NCC3C4CCCCC34)CO2)sc1C 16033,CC1CC(NC(=O)C(C)C(=O)OC(C)(C)C)CCN1C(=O)CN1CCS(=O)CC1 16034,c1(C(=O)NC2(C)CN(C(C(COCC)C)=O)C2)cc(S(=O)(=O)NC)ccc1C 16035,N1(C(C(C)N(C(=O)C(CC(C)C)C(C)C)CC)=O)CC2(CCN(C)CC2)C1 16036,C(CCC(=O)N(CCC(C)NC(=O)C(=O)NCC(F)F)C)=CC 16037,C1(NC(C(C)(C)n2cc(Cn3cncn3)nn2)=O)CC2CCCN2C1 16038,CC(C)C(C(=O)NC(C)CCN(C)C)NC(C1(CO)CC(C)(C)C1)=O 16039,CC1C(NC(c2c[nH]cc2C(F)(F)F)=O)CCCN1C(=O)Cc1cnccc1Cl 16040,c1(C(=O)NC(C2CCN(C(C3CCC(=O)O3)=O)CC2)C)cccc2ncccc12 16041,C1(CNC(C2CN(C)C2)=O)CN(C(c2ccc(Br)nc2O)=O)CC1(F)F 16042,[N-]=[N+]=NC1CN(C(C2C3CC4C(C3)C24)=O)CC1NC(C1(C(=O)NC2CC2)CC1)=O 16043,N1(c2ncc(C(c3nnnn3C(C)C)OC)cn2)CCC(S(=O)(=O)N(C)C)C1 16044,C1(CNC(CS(CC)(=O)=O)=O)CN(C(=O)CC2(CSC)CC2)C2COCC2O1 16045,Cn1c(CCNC(c2ccnc3[nH]nc(N)c23)=O)nc2cc(F)ccc12 16046,c1(OC)ccc(CC(N2CC(CNC(=O)Cc3cnc(C)nc3O)C2)=O)c(Cl)c1 16047,N1(C(CCS(C)(=O)=O)=O)CCC2(CC1)CC(NC(=O)C(F)(F)Cl)CO2 16048,c1(CC)nc(C(C(=O)NCC(C)C)N(C)Cc2csc(C(F)(F)F)n2)cs1 16049,CN1CCN(C(=O)C2=CCN(C(=O)CCc3cccs3)CC2)CCC1=O 16050,C(=O)(C1CCc2ccccc21)NCC(C)N(C)C(c1ccc(CO)cn1)=O 16051,CN1CCCC1C(=O)NCC(C)(C)CNC(c1ncoc1C1CC1)=O 16052,CC1(C)CCC(CC(=O)Nc2ccc(F)cn2)CC1.C12CC(C1)CNC2=O 16053,C=C=CC(C)C(=O)NCC(C)(C)CN(C(c1cnc(OC(C)C)cn1)=O)CC 16054,Cc1cc(CC(N2CC(C(=O)NCC=CCO)C2)=O)c(C)s1.C1(=O)CCCN1 16055,c1(CNC(C2C3CN(Cc4ccc(OCCC)cc4)C2C3)=O)cc(C)cc(C)c1 16056,c1(C(=O)NCC(CNC(c2c(C)n(CCO)nc2)=O)C)cc(S(N)(=O)=O)cn1C 16057,c1(C(N(C2CCC(NC(C=CC=CCC)=O)C2)C)=O)c(F)cc(OC)cc1Cl 16058,C1(NC(CCN(CCC)C)=O)CC(O)CN(C(c2cnc(CC)s2)=O)C1 16059,C(=O)(C1CCc2c(Cl)cccc21)N1C(C(N2CCC(NC(C(C=C)O)=O)CC2)=O)CC1 16060,C(=O)(CC(=O)NC1CCC1NC(c1nnc(C(C)(C)C)s1)=O)N(C)C 16061,c1(C(N2CCC(NC(C(N3CCSCC3)C)=O)CC2C)=O)ncn2ccccc12 16062,C1(NC(CC(=O)N(C)C)=O)CC2CCC(C1)N2C(=O)Cc1cccc(F)c1Cl 16063,C1(NC(C2CC(CSC)C2)=O)CN(C(=O)C(C)(C)OC(C)=O)CC1F 16064,C12(C(=O)NCC3CCCC(C)C3)CC(CCO1)N(C(C1CCC1C#N)=O)C2 16065,CC(CC(N)=O)C(=O)N1CC(CNC(c2ccnn2C(C)(C)C)=O)C2(CC2)C1 16066,c1(CNC(C2(CC)CCCC2)=O)cccc(NC(=O)CC2CC(C)OC2C)c1 16067,c1(C(=O)NC(C(=O)NCC(O)CC2CCCC2)C2CCCO2)ncoc1C1CC1 16068,Cc1cccc(F)c1CC(=O)NC1CC(NC(C2C3CCC(F)(F)C23)=O)CC1O 16069,Cn1cc(C(=O)NC2COCC2CNC(=O)CC(=O)NC2CC2)c(C2CCC2)n1 16070,CC1=C(C(=O)NC2CCN(C(=O)C=C(C3CC3)C3CC3)C(C3CC3)C2)CCC1 16071,C1(F)(CNC(C2C(=O)NCC2)=O)CCN(C(c2cccc(OC(F)(F)F)c2)=O)C1 16072,C1(NC(Cc2nnc(C)s2)=O)CCN(C(c2cc(N(C)C)nc(Cl)c2)=O)CC1C 16073,c1(NC(C)=O)cccc(-n2nc(C3CC34CC4)nc2-c2coc(C)n2)c1 16074,CCCCS(=O)(=O)NC(C)C(=O)NC1CC(CNC(=O)C(C)(C)NC(C)=O)C1 16075,CC1=C(C(=O)NCC2CC2CNC(=O)CCc2cncc(Br)c2)CCC1 16076,N1(C(C)=O)CCC2(CCC2)C(NCNC(c2cnc(C)nc2C)=O)C1 16077,CC1(C(N2CCCOC(CNC(C3CCOCC3)=O)C2)=O)CCC(=O)NC1 16078,C(CN=c1[nH]cnc2c1COC2)(CC(C)C)NC(C(c1c(C)n[nH]c1C)C)=O 16079,O=C(CCCc1cccs1)NCC(O)CCNC(C1(F)CCC1)=O 16080,c1(CC(N2C(CNC(=O)C=CCF)CCC(C)C2)=O)csc2ccccc12 16081,C1(NC(C2CCC(C)C2)=O)CCOC2(CCN(C(C3(O)CCSC3)=O)CC2)C1 16082,O(C1CCCc2ccccc21)CC(=O)NCCCCNC(C1(C)CC2CC2C1)=O 16083,C1(NC(c2cc(F)cc3c2CCC3)=O)CN(C(=O)C=CC2CC2)C2CCCCC12 16084,C1(CC(=O)NCc2c(C)scc2)CC2(C1)CN(C(=O)C(C)Cn1ccnc1)C2 16085,Cc1cc(N2CCC(CNC(c3nc4ccccn4n3)=O)C2)n2nc(C)cc2n1 16086,C(=O)(C(F)(F)C(C)O)NC(C1CCCCC1)CNC(C(CCC)O)=O 16087,C1(NC(c2cc(C)c(C)[nH]2)=O)CN(C(c2ccc(O)cn2)=O)C2CCCC12 16088,C(CCCCC(=O)NCCOCCCF)N(C(CN(C(=O)OC)C)=O)C 16089,CCCCCC(O)CC(=O)NC(c1cn(C)nn1)CNC(c1cc(Cl)c[nH]1)=O 16090,c1(CNC(CCCCOC)=O)ccc2c(c1)CCC2NC(C1CCC1C(F)F)=O 16091,C1(C(N2C(Cn3cc(-c4n[nH]c(C)c4C)nn3)CC=CC2)=O)CCOC(=O)CC1 16092,C(=O)(CCN=C1NS(=O)(=O)c2ccccc21)N1CC(CC)OC(CC)C1 16093,C(=O)(C(CCOC)OC)N1CCC(NC(c2nc(CC)sc2)=O)C1 16094,N1(C(=O)OC(C)(C)C)CCC(O)(C(N2CCC(N(C(=O)CC(F)(F)Cl)C3CC3)C2)=O)C1 16095,N1(C(COCCCOC)=O)CC2CC(O)C1C2NC(C1CCCCNC1=O)=O 16096,C(=O)(C1=NNC(=O)CC1)NCC1CC(NC(C(C(C)(C)C)OC)=O)CC1O 16097,c1(C(=O)NCC2(C(=O)NCc3ncc(C)o3)CC2)cccc(O)c1C 16098,CC(C)CCC(=O)C(=O)N1CCC(C(=O)NCCC2CCOC2)CC1(C)C 16099,c1(C(N2CC(NC(COCCC#C)=O)C(C)(C)CC2)=O)cc(S(N)(=O)=O)c(C)s1 16100,C1(NC(c2nc(COC)[nH]n2)=O)CCN(C(C2CCC3CC3C2)=O)C(C)C1 16101,Cc1ccc(C(F)(F)C(=O)NC2CCCN(C(=O)CSCCN(C)C)C2)cc1 16102,c1(C(=O)NC(C(C)NC(C(COC)NC(C)=O)=O)(C)C)cc(N)c(Cl)c(O)n1 16103,CCC(CC)CCC(=O)NCC1CC2CC2N1C(=O)CS(=O)C(F)(F)F 16104,C1(C(=O)NC2CN(C(C=CCOC)=O)C2)(OC)CCCC(C)C1 16105,C1(CNC(C(CC)N(C)C)=O)CN(C)CCN1C(C1C(c2ccccc2)C1C)=O 16106,C1(C(NOCC(C)C)=O)CCN(C(c2cc[nH]n2)=O)CC1O 16107,CCCCCCCCNC(=O)C(=O)NC(C)CNC(=O)CC1CC(SC)C1 16108,c1(CN(C=O)Cc2n(C)cnn2)nc2c(o1)CCSC2 16109,C1(C(N2CC(N(C(=O)Cc3cc[nH]n3)C)C(O)C2)=O)CCn2ccnc2C1 16110,c1(C(C(=O)NCc2ccnn2C)N(C)C)ccccc1F 16111,C1(NC(C(C(C)C)SCC)=O)CC2CCC(C1)N2C(c1ccc(C(C)(C)C)[nH]1)=O 16112,N1(C(C(C=C)OC)=O)CCC(C)CC1C(=O)NC(COC)CCCC 16113,C(C1CC(C)(C)Oc2ccccc21)NC(CC(C)OC)c1nnnn1CC(F)F 16114,c1(C(=O)NC2C(CNC(C=CCCC)=O)C2)cn(C)nc1-c1ccnn1C 16115,Cc1ccc(C(=O)NC(C)C(CO)NC(C2CC(S(C)(=O)=O)C2)=O)cc1C 16116,C1(CN(C(=O)CCN2CCCC2)C)CCCN1C(=O)CCc1nccs1 16117,c1(C(C(=O)NC2CCCC2)N(C2CCCC2)CC(=O)OCC)ccc(C)c(C)c1 16118,Cn1ccc2c(C(N3CCN(C(c4ccnc(O)c4)=O)C(C#N)C3)=O)cccc12 16119,C1(CC)CN(C(C2(F)CCOC2=O)=O)CCN1C(=O)CCCCc1ccc(Cl)cc1 16120,n1(CC)cc(CNC(=NCCSC2CC2)NCCSC(C)C)ccc1=O 16121,C1(NC(=O)CC2(CO)CC2)CN(C(C2CC(=O)N(C3CC3)C2)=O)CC1F 16122,C12(C(=O)NCCCCN(C(=O)CN3CCSCC3)C)CC(C1)C(C)(C)O2 16123,N1(C(CCn2c(C)ccc2C)=O)CCOCC(CNC(=O)C2CC2)C1 16124,c1(OC)cc(C(N2CC(NC(=O)CC3CC(F)C3)C(C)(C)C2)=O)nnc1C1CC1 16125,C(=O)(C(C)(C)C(F)F)NCCN(C(c1c(C)occ1)=O)C 16126,C(c1ccc(F)c2ccccc12)=CC(=O)NCC1CC(NC(C2(O)CCC2)=O)C1 16127,C12(CC(=O)NCCNC(C(C)(C)N(S(C)(=O)=O)C)=O)CCCN1CCC2 16128,C(CC(C(C)C)NC(=O)C(F)CC1CCCCC1)NC(COCC=C)=O 16129,c1(C(=O)NC(C2CCN(C(Cc3ncc(CC)[nH]3)=O)C2)C)cc(F)cc(F)c1N 16130,CS(=O)CCC(=O)N.c1(CC(=O)N(CCCC)CC2CC2)ccc(C(F)(F)F)nc1 16131,CC(C)CCCC(C)C(=O)N1CC2(CC(C(=O)NC3(C)CCCC3(F)F)CO2)C1 16132,C(=O)(CCS(N)(=O)=O)N1CC(=C(CNC(c2ncc(CC)nc2)=O)F)C1 16133,c1(NC(C(c2cnn(C)c2)NC(c2nc(CC)oc2)=O)=O)ccc(C)c(C)c1 16134,c1(C(N(CCC(C)NC(c2cn(C)nn2)=O)C)=O)cccc(-c2nc(=O)o[nH]2)c1 16135,C1(CC#C)(C(N2CCC(NC(=O)CC3CCCN3C(=O)OC)C2)=O)CCCCC1 16136,CC1CC(C(=O)N(CC(O)CNC(c2cnnc(O)c2)=O)C)=NO1 16137,CC(C)(C)C#CC(=O)NCCC1COCCN1C(=O)CCC1CC1(F)F 16138,c1(CC(N2C(CN(C(c3cnc(C)s3)=O)C)CCC2)=O)ccc2[nH]ccc2c1 16139,CC1CCCN1CC(=O)NCC1(O)CC(C(N2CCC(C(C)(C)O)C2)=O)C1 16140,n1(CC(=O)NCC(CNC(CC(n2ccc(C)n2)C)=O)O)cc2ccccc2n1 16141,C#CCCC(O)C(=O)NCc1cccc(NC(=O)Cc2ccc(F)cc2)c1 16142,n1(CCC)nc(C)cc1C(=O)NC(CN(C(=O)C(C)CC)C)CC 16143,N1(C(CSCC)=O)CCC2(CCN(C(c3ccc(OC)nc3)=O)C2)C1 16144,Cn1cc(CC(=O)NC2CCCCC2NC(=O)CCC2(C)CC2)c2ccccc12 16145,c1(SC)ccc(C(=O)NCC2(C(C)NC(=O)CC3COC(=O)N3)CC2)cc1 16146,c1(C(N2CCCC(N(C)C(C3CCS(=O)(=O)N3)=O)CC2)=O)ccc2nc[nH]c2n1 16147,CC1(C)CN(C(=O)CC2OCCC2(C)C)CC1NC(=O)CNc1ccc(O)cc1 16148,C1(NC(c2c(C)nc(C3CC3)s2)=O)CCCC12CN(C(C1CN(C(N)=O)C1)=O)C2 16149,C#CCC(C(=O)N1CCCC1(C(N1CC(F)C(F)C1)=O)CC)C1CC1 16150,c1(C(=O)NC(CC)CNC(C2CC(O)C2)=O)ccncc1C(F)(F)F 16151,C1(CC(=O)NCCN(C(c2c(C)cc(F)cn2)=O)C(C)C)CCC2(CCC2)CO1 16152,CC(C)CC(C(=O)NCc1ccc(F)cc1F)n1ccnc1C1CCC12CCCO2 16153,c1(N2CC(CNC(C(C)CN(C)C)=O)OCC2)ncnc2cccc([N+](=O)[O-])c12 16154,CC(C(=O)NC(CC1CC1)CC(=O)N1CC(c2cccnc2)C1)C(C)(C)C 16155,C(CC(F)(F)CO)NC(C1(n2cccc2)CCOCC1)=O 16156,C1(C(N(CCNC(CCOC(CC(C)C)C)=O)CC2CC2)=O)CCCCCC1 16157,c1(C(=O)NC(CNC(=O)CC2(O)CCOC2)C2CCC2)cccn2ccnc12 16158,N1(CC)CCCCC1C(N1CC(C(=O)NC(C2CSC2)C)C(C(C)C)C1)=O 16159,CC(O)C(=O)N1CC(C(=O)NCC2CC2CO)C1 16160,c1(C(N2CCCC(C(N(C)Cc3c(C)occ3)=O)C2)=O)cc2ncccc2[nH]1 16161,n1(CCCOC)nnnc1C(c1nncn1C1CC1)NC1CC(OCCSC)C1 16162,C(=O)(CC(C)C(=O)N(CC(=O)NCC1CC(C)C1)C1CC1)OC 16163,c1(C(C(N2CC(O)(CCNC(C(C)N(C)C)=O)C2)=O)O)ccc(Cl)cc1Cl 16164,N(C(=NCCC(C)C)N1CCc2ocnc2C1)CC(c1c(C)noc1C)C 16165,C1(C)(C(=O)NC(CCCNC(c2c(CCC)n(C)nn2)=O)C)CC2(C1)CC2(F)F 16166,c1(CNC(c2c(OC)ccs2)=O)ccc(NC(=O)C(C)OCC2CCCO2)cc1 16167,c1(C(=O)NC2CC(CNC(CC3(OC)CC3)=O)C2(C)C)cc([N+](=O)[O-])cc(C)c1Cl 16168,C(=O)(CC1OCCc2ccccc21)NC12CCCN(c3c(OC)cncn3)CC1C2 16169,N1(C(CN(C)C(C2CCC(C3CC3)C2)=O)=O)CCCCCCCC1 16170,C1(C(=O)NCCCN(C(C(C)NC(COC)=O)=O)C)COCC(C)(C)O1 16171,C1(NC(C2CC3(CC3)C2)=O)CN(C(=O)CCC2CCCC2)C2(CCCC2)C1 16172,C(=O)(C#CC1CCCOC1)N1CCOCC(C)(CNC(C=C(CC)CC)=O)C1 16173,N1(C(C(C)(C)NC(C(CCC)CC)=O)=O)CC2C3CCC(O3)C2C1 16174,N1(C(C(C(CC)C)NC(C)=O)=O)CCC2(CCC2)C(NC(C2CCC(=O)N2)=O)C1 16175,C1(NC(C2(NC)CC2)=O)COCCC1NC(c1scc(C)c1C(=O)OC)=O 16176,n1(CC)nc(C(=O)NCC(=C2CN(C(c3cccc(C(N)=O)n3)=O)C2)F)cc1C 16177,C(=O)(C1=C(C)N(C)c2ncnn2C1C)NCCN(C(C(C)OC)=O)C(C)C 16178,N1(C(C(C)OCCCC)=O)CC2(NC(=O)CCn3c(C)csc3=O)CCC1C2 16179,C(=O)(C1=CCCCC1)NCC(CC1CN(C(C(CCC)=CCC)=O)C1)(C)C 16180,N1(C(c2c(SC)ccs2)=O)CC2CCC2(CNC(=O)CCC=C(C)C)C1 16181,c1(CNC2C(C)CCOC2)cccc2nc(C(F)F)sc12 16182,c1(C(CC(=O)N2CC(NC(C3C(CCC)C3)=O)C2)C)ccc(F)c(F)c1 16183,C1(C2CCCN(C(c3c(C4CCC4)cnn3C)=O)C2)(NC(CC(C)C)=O)CC1 16184,N1(c2c(C(=O)OCC)nsc2N)CCC(=O)N(C)CC1 16185,Cc1noc(C)c1CC(C)C(N1CCN(CCNC(C2(CCO)CC2)=O)CC1)=O 16186,N1(C(C2C(C)(C)OC(=O)N2)=O)CC2(C1)CN(C(=O)CCCC1CCCO1)CCO2 16187,O=c1nc(O)c(CNCCNc2nc3ccccc3s2)cn1-c1ccccc1 16188,CC1CCN(C(c2cc(C3CC3)ccn2)=O)C1CNC(=O)C=Cc1cc[nH]c1 16189,CCC(CC)CCC(=O)N1CCN(C(=O)CC(O)CC(C)C)CCC1C 16190,C1(N(C(c2ccc(C)cc2)C(=O)NCCC#N)CCC)CCN(C)C1(C)C 16191,C(=O)(C1CCc2nccn21)NC(C(=O)NC1(CC)CCCC1)CC1CC1 16192,C(C)(C(=O)NOCCO)N(C(CC1CCC(C)C1)=O)CC(C)N 16193,N1(C(C(CCC)O)=O)CCN(C(c2c[nH]c(Br)c2)=O)CC1c1ccc(F)cc1 16194,Cc1cnc(C(=O)NC2CCC(N(C)C(c3c(Br)cnn3C)=O)CC2)c(C)c1 16195,C1(NC(c2cn(C)nn2)=O)CCN(C(=O)CC2CC(C(F)F)C2)C12CC2 16196,N1(C(C(N)=O)=O)CCCOC(CNC(=O)CC(O)C2CCCC2)C1 16197,C1(C(N(C)CC2CC(=C)C2)=O)CCN(C(=O)CCCCOCC)C1CC 16198,C=CCC(C)(C)C(=O)NC1CCN(C(=O)CCCCCNC(C)=O)C(C)C1 16199,N1(C(C=C(CC)C)=O)CC2C(N(C)C(c3cc(-c4cccc(Cl)c4)ns3)=O)C2C1 16200,C1(CN(C(C(c2ccc(CC)s2)=O)=O)C)CCCCN1C(=O)CCSC 16201,C1(C(N2C(CC)CC(C)C2)=O)CCC2(CC2)N1C(c1c[nH]c(C)c1)=O 16202,c1(C(=O)NC2CCC(C)(CNC(c3c(CC)scn3)=O)C2)ccc(OC)c(O)c1 16203,C(=O)(C1=CCCOCC1)NC(c1cnn(C)c1)C(N1CCN(CC#C)C(=O)C1)=O 16204,C1(C)(CNC(C=C=C(C)C)=O)CN(C(=O)CC2CCC(C)(C)O2)CCO1 16205,N1(C(C(C=C)O)=O)CC(NC(=O)CC2CCCCCC2)CC2(CCC2)C1 16206,c1(OC)c(C(N2CC(CNC(=O)C=Cc3ccoc3)C2)=O)cccc1F 16207,N1(C(C(CN(C)C)O)=O)CCC2C(CCCN2C(C2CCCCN2C)=O)C1 16208,C1(CC)CCC(NC(=O)CC2(N(C)C(C3CCCN3C3CC3)=O)CC2)C1 16209,N1(C(CC2(C)CCOC2)=O)CCC2(CC1)CC2C(N1CC2CC2C2CC12)=O 16210,C12(CNC(C3C(C)(C)C3)=O)CCC(C1)N(C(=O)CCCN1CCCC1)C2 16211,Cc1ncc(C(=O)N(C2CCC(C(=O)NCC(C)(C)C3(C)CC3)C2)C)cc1C#N 16212,c1(OC)cccc(N2CCN(C(c3cccnc3O)=O)CC(C)(F)C2)c1[N+](=O)[O-] 16213,N1(CC(=O)NCC(CO)NC(Cn2c(=N)scc2)=O)CCN(S(C)(=O)=O)CC1 16214,c1(NC(C(=O)N(CC(C)CNC(=O)C=C2CCC2)C)=O)ccccc1 16215,C1(NC(C#CC(C)C)=O)CN(C(=O)C(C2CCOCC2)F)CC12CCOCC2 16216,C(CC(C)C(=O)N1CC(C)(NC(=O)C(C)NC(C2(CC3CCCC3)CC2)=O)C1)OC 16217,C=CC1(C(=O)NC(c2ccccc2F)C)CCN(C(c2ccsn2)=O)C1 16218,N(C1CCCc2occc21)C(C1CC(C)(C)N(C(C2CCCC2O)=O)C1)=O 16219,c1(OC)cc(CC(=O)NCCCNC(=O)CC(C)OC)ccc1F 16220,Cc1cc(C)n(C(C)C(=O)NC2CC(NC(C3CCC(F)(F)C3)=O)C2)n1 16221,c1(C(N2CCN(C(c3n(CC)ccn3)=O)CC2CF)=O)cc(F)cc(N)c1F 16222,N1(C(c2cc(C)no2)=O)CCN(C(=O)CN2CC(=O)NC2=O)C(C(F)F)C1 16223,Cc1ccc(C)c(C(N2CC(CNC(=O)C(F)(F)CO)OC(C(F)(F)F)C2)=O)n1 16224,Cc1cc(Oc2ccncc2)ccc1C(=O)Nc1cc(O)ccc1Cl 16225,c1(C(=O)NC2C(C)CN(C(c3ccnc(S)c3)=O)CC2)cc2c(F)cccc2[nH]1 16226,c1(OCC)cc(O)c(C(=O)NCC(C)N(C)C(C2CC(OC)C2)=O)cc1OC 16227,N1(C(C(C2CCN(C(C(C)OC)=O)C2)F)=O)CCC(C)(C)C(CO)C1 16228,c1(OCC(=O)NCC=C(C(=O)NCCOCC)C)ccc(F)nc1 16229,C12(NC(c3cc(C)ns3)=O)CCCC1N(C(=O)CCCCC(F)F)CCC2 16230,c1(SC)cccc(C(N2CC(C(C)NC(c3cn(C4CC4)nn3)=O)C2)=O)c1 16231,C1(C)(COC)CCN(C(C2C=CCN2C(=O)C(C)CN(C)C)=O)C1 16232,CC1CCN(C(c2cn(C)nc2-c2ccoc2)=O)CCN1C(C1CNC(=O)N1)=O 16233,CC1CC(CNC(c2cn(C3CC3)nn2)=O)CN1C(c1cn(C)c(O)n1)=O 16234,Cc1nn(C)cc1CCC(=O)NC(C1CCCN1C(c1ccccc1)=O)C 16235,N1(C(C2(C)CCOCC2)=O)CCC(F)(C(=O)NCc2ccc(Cl)c(F)c2)CC1 16236,c1(C(=O)NC2CCN(C(C3N(C(=O)OC(C)C)CSC3)=O)C2)c[nH]nc1[N+](=O)[O-] 16237,c1(C(N(CCC(C)NC(C2CC(OC)C(OC)C2)=O)C)=O)c(F)cc(F)cc1F 16238,C1(NC(C(C)n2cccn2)=O)CN(Cc2ccccc2CCBr)CC1C#N 16239,c1(C(=O)NCC2(C)C(C)CN(C(C(CC)CC)=O)C2)cnc2cc[nH]c2c1 16240,N1(C(c2ccc3c(c2)COC3)C(=O)NC(C)(C)C)CCc2cc(Br)cc(F)c2C1 16241,C1(NC(C(C)OCCCC)=O)CCN(C(=O)CSc2ccc(OC)cc2)C1C 16242,C#Cc1ccc(C(=O)NCC2CCN2C(c2nocc2Br)=O)o1 16243,c1(C(=O)NC(CCOC)CNC(=O)COc2ccccc2Cl)cc(O)cc(=O)o1 16244,C1(C(=O)NCCN(C(=O)CC(C)(C)c2ccccc2)CCC)CC(O)C1(C)C 16245,CC1(C)CCN(C(=O)COCCF)C1CC(N1CC(O)C(O)C1)=O 16246,CCC(F)(C(=O)OC)C(=O)N1CCCC1c1ccc(C2CC2)cc1C 16247,N1(C(C2(OCC)CNC2)=O)CCC(=O)N(C)c2cc(F)ccc21 16248,C(C(CC(C)C)C(=O)N1CC2=C(C1)CN(C(=O)CC1CC13CC3)C2)OC 16249,c1(C(=O)NCCOC)cc(=NC(=O)C2CC2c2nccc(I)n2)[nH][nH]1 16250,c1(C(=O)NC23CC(CNC(CCOC)=O)(C2)OC3C)snc2ccccc12 16251,C1(NC(c2c(C)ncnc2)=O)CC2CC1N(C(c1ccc(F)cc1Br)=O)C2 16252,c1(C(=O)NCC2C(NC(c3cc(CCOC)on3)=O)C2)cccc(F)c1C 16253,C=Cc1cccc(Nc2ccccc2NC(=O)CSCCOC)c1 16254,C1(CC)CN(C(c2ncccc2O)=O)CC1NC(C1COCC1(C)C)=O 16255,c1(N2CCC(N(C)C(C3(c4ccc(F)cn4)CC3)=O)C2)nc(CO)nc(Cl)c1C 16256,C1(C(N2CC(CNC(C3CCCN(CC)C3)=O)C2)=O)CCCC1C1CC1 16257,C(=O)(C(C)CC(F)(F)F)N(C1CN(C(c2cc(C)cc(N)c2)=O)CC1(C)C)C 16258,CCS(=O)CC(=O)N1CC(CNC(c2ccnn2C2CCCCC2)=O)C(C)C1 16259,N(C)(C1CS(=O)(=O)c2ccccc21)C(=O)NCC1N(C(=O)OC(C)(C)C)CC(C)C1 16260,N1(C(CCOCCC)=O)CCC2CCN(C(=O)CCNS(C)(=O)=O)CC12 16261,c1(NC(CC)=O)ccc(Cl)cc1C.N12C(CC1C)C(=O)NC(C)C2=O 16262,c1(C(=O)NCCC2N(C(CCCCOC)=O)CCCC2)cnc(N)c(Cl)c1 16263,C1(C(=O)NCC2CC(NC(c3cnn(C)c3C3CC3)=O)C2)CCC2C1C2(F)F 16264,C(CCC(=O)NNC(=O)c1ccc(F)cc1Br)OC 16265,c1(C(=O)NC(CNC(CC2CC(SC)C2)=O)(C)C)cnc(OC)cc1OC 16266,c1(N(c2ncccn2)C(C2(F)CCNCC2)=O)ncnc2sccc12 16267,Cn1nncc1CC(=O)NC1(C)CC(NC(=O)C=CCSC(C)(C)C)C1 16268,N1(C(C(CSC)O)=O)CC=CC(C(=O)N(C)CCOCCO)C1 16269,c1(OC)cccc2[nH]cc(CC(=O)NC(C3CN(C(C4CCC(=O)O4)=O)C3)C)c12 16270,C1(C(N(CC(C)NC(C=Cc2c(C)nccc2)=O)C)=O)CCc2ncncc2C1 16271,C1(NC(C(C=C)O)=O)CN(C(c2csc(C)c2)=O)CC1S(C)(=O)=O 16272,C1(CNC(C2(COC)CCOC2)=O)CCC(c2ccccc2)=NO1 16273,C1(C2CN(C(C3CC3Cl)=O)C2)(NC(c2ccc(CN(C(C)C)C)cc2)=O)CC1 16274,c1(C(=O)NCC(CNC(=O)Cc2cnccc2Cl)F)cc(Cl)c([N+](=O)[O-])[nH]1 16275,N1(C(C2N(C)CCC2)=O)CCN(C(c2nn(C)cc2Cl)=O)C(C2CC2)C1 16276,C1(C(=O)NC(CNC(C(C)OCC=C)=O)C2CC2)CCC(C)(C)O1 16277,CC(=Cn1ccnn1)C(=O)N(C1CCCC(NC(c2ncsc2C(C)C)=O)C1)C 16278,N1(CC(=O)N(C)CCNC(=O)C(C2CC2)C2CC2)CCNC(=O)C1 16279,C1(C(N2C(CNC(c3ccoc3)=O)CC(O)C2)=O)CC12CCOc1ccccc12 16280,N1(C(c2c(CC)c(C)sc2)=O)CCC2(CC1)CC2NC(C1COCCO1)=O 16281,c1(C(N2C(CNC(CCCN(CCC)CCC)=O)CCC2)=O)nc(C)oc1C 16282,C(C(C)CN=c1ccnc(NCCS(=O)C(C)(C)C)[nH]1)OCC 16283,c1(CC)cc(N)ccc1C(=O)NCC(C)CN(C(=O)CC1CC(CC)C1)CC 16284,Cc1cnc(C(N2CCC(CCNC(c3cnc(N)c(Cl)c3)=O)C2)=O)cc1Cl 16285,C1(C2CC2)(NC(CCCC)=O)CCN(C(c2ccc(-n3ccnc3C)cc2)=O)C1 16286,c1(C(=O)NCC2(F)CCN(C(c3c(C)c[nH]n3)=O)C2)cnc2[nH]nc(O)c2c1 16287,N1(C(c2c(OC)cncc2)=O)CC2=C(C1)CN(C(=O)C(c1cnccn1)C)C2 16288,O=C(CC(F)(F)C(F)(F)F)NC1CCC2(CC1)CN(C(c1ccccc1O)=O)C2 16289,C1(CC(=O)NCC)CC(F)CN1C(=O)Cc1csnn1.C1CC=CC1 16290,C(=O)(CC(F)(F)Br)N(CCCNC(CN(C)CC)=O)CCO 16291,c1(C(N2C(CCC(=O)NCC(CNC(N)=O)O)CCC2)=O)ccc2c(c1)CC2 16292,C1(C(N2CC(C(=O)Oc3ccon3)OC2=O)=O)CCCN(OC)C1C 16293,C1(CNC(C2(CC#C)CCCO2)=O)CC(C)CN(C(=O)CS(N)(=O)=O)C1 16294,CC1=C(C(=O)NC2CCCC(NC(c3c(N)sc(C)c3C)=O)CC2)CCCC1 16295,C1(CC(=O)N(C)CC2N(C(Cc3c(C)n[nH]c3)=O)CCC2)Cc2ccccc2N1 16296,C1(C(N(CCCNC(c2ccc(CO)nc2)=O)CCC)=O)CC2(C1)CC1(CC1)C2 16297,C1(CNC(C2CCCC(O)C2)=O)CCCCN(C(=O)CNc2cccnc2)C1 16298,c1(C(N2C3(CNC(C=CC)=O)CCC2CC3)=O)cccc2scnc12 16299,c1(OCCC(=O)N(CCCCN(C(C(CC)C#N)=O)C)C)ccc(F)cc1F 16300,C(=O)(CCCc1ccsc1)NC(C1CCCN1C(=O)C(C1CCCCC1)=O)C 16301,C1(C)(CNC(C2C(C)C2)=O)CN(C(c2ccc(CO)c(Cl)c2)=O)C(C)(C)C1 16302,C1(C(N(C(CC)CC)C)=O)CC2(CCN(C(=O)CCC3CCCCO3)C2)C1 16303,C(C)(CNC(C1CCS(=O)(=O)C1)=O)(C(C)C)NC(CC(=C)Br)=O 16304,C(=O)(C(F)C(C)(F)F)N1CC(C(=O)NC2CCC3(CC3)C2)(SC)C1 16305,c1(OC)ccc(C)c(C(N2CCCCC2Cc2cn(CCC(F)(F)Cl)nn2)=O)n1 16306,Cc1[nH]nc(Br)c1C(=O)NC(C)CC(C)NC(=O)C(C1CC1)N(C)C 16307,CC(=O)CCCCC(=O)N1CCC(NC(=O)CCCN2CCCC2)CC(O)C1 16308,N1(C(C=C2C(C)(C)CCCC2)=O)CCC2CC1CN(C(=O)C(O)c1ccsc1)C2 16309,S(=O)(=O)(c1cccc(C(N2CC(=O)N(C(C)CC)C2)=O)c1)NCC#C 16310,c1(C(=O)NC2CN(C(C3CC34CC4)=O)CCC2F)cc2ccnc(Cl)c2s1 16311,c1ccc(C2=CCN(N(C)CP(C)(C)=O)CC2)cc1.C(=O)CC1CCC1 16312,c1(OCCOCC)ccccc1C=CC(=O)OC(C)Cc1ccccn1 16313,C1(CNC(C(C)(C)C)=O)Cc2ccccc2CN1C(C1CC(S(C)(=O)=O)C1)=O 16314,C1(C(=O)NCC(CNC(COC(CC)(C)C)=O)(C)OC)OC(C)(C)OC1(C)C 16315,N1(c2nccc(C)n2)CCC(C(=O)Nc2cnn(-c3ccccc3Br)c2)C(O)C1 16316,Cc1cc2ccc(C(=O)NCC(F)CNC(c3cocc3C)=O)cn2c1 16317,C=C=C(C)CC(=O)NC1(CN(C)C(C2CCN2C2CCCC2)=O)CC1 16318,N1(C(CC2C(C)C2)=O)CC2=C(C1)CN(C(=O)CSc1c[nH]nc1Br)C2 16319,C(=O)(C(F)(F)C(O)C(C)C)N1CC2(C(NC(c3cccc(C)c3F)=O)CCC2)C1 16320,C1(C(=O)NC2(C(N3CC(N(CC)CC)C3)=O)CCCC2C)CC(=O)CC12CCC2 16321,c1(C(N2CCN(C(C)C(=O)NCC(F)(F)F)CC2)=O)nccn2nccc12 16322,c1(NC(C(C)(C)C)=O)cccc(C(=O)NCCCCNC(C23CC(C)(CO2)C3)=O)c1 16323,Cc1c(Cl)ccc(C(N2CCOC(C)(CNC(=O)C(C)OCC(C)C)C2)=O)c1O 16324,c1(C(=O)NC2CC3CN(C(=O)C#CC4CCCO4)CC23)cccc2c1OCCC2 16325,N1(CCCCCCC)CCC2C(CCCN2C(=O)CC2(C(F)(F)F)CC2)C1 16326,C1(OC)CCCCC1(c1nnnn1C1COC1)N(c1nccs1)C1COC1 16327,C1(C(=O)Nc2ccns2)CC2(CCN(Cc3cc(O)cc(Cl)c3)CC2)C1 16328,C1(O)(C(C)NC(Cc2ccc(OC)cc2)=O)CCN(C(=O)Cc2cnns2)CC1 16329,c1(OCC)ccnc(N2C3CCC2CC3)n1.C1(=O)CN(C)C(=O)CO1 16330,N1(CC(=O)N(C2CN(C(Cc3nc(C)[nH]n3)=O)C2)C)CCCCS1(=O)=O 16331,N1(C(c2nccc(CC)c2)=O)CC2CCC(C1)C(NC(=O)C(C)C(C)COC)C2 16332,C(=O)(NN1CCCC(C(=O)OC(C)(C)C)C1)C1(C(=O)OC)CC(N)C1 16333,n1(CC(=O)NC(C)CCCNC(c2cnnn2C)=O)cc(Cl)c(O)nc1=O 16334,C1(C(N2C3(CNC(C4CC(OC)C4)=O)CC(C2)C3)=O)CC12CCC(=O)CC2 16335,C1(C(C)C(=O)N(C2(C)CC2)C)CCN(C(C2CC(=O)C2)=O)C1 16336,C(CCCCS(=O)(=O)CC)OC(C(c1ccc(OC)nc1)(F)F)=O.C12CCN1C2 16337,N1(C(C(C)OC)=O)CC2(C1)OC1(C)CC2(NC(=O)C(=Cc2cccc(Cl)c2)C)C1 16338,N1(C(c2cnn(CC)c2C)=O)CCC(NC(=O)CCn2ccccc2=O)C(C)C1 16339,N1(C(=O)CCC2CC2)CC2(CCN(C(c3cc(C4CCOC4)[nH]n3)=O)C2)C1 16340,C1(C(=O)NC(CC(=O)OCC)C)CCN(C(c2c(C)cnn2C)=O)CC1(C)C 16341,Cc1cc(Cl)ncc1NC(C1CC(F)CN1C(=O)CSc1c(F)cccc1F)=O 16342,C=C(C)CC(C)C(=O)N1CC2CC2(CNC(=O)CCC=Cc2ccccc2)C1 16343,c1(C(N2C(CN(C(c3nc(Cl)oc3C)=O)CC)CCC2)=O)cnn2ccsc12 16344,N1(C(CC2N(C)CCCC2)=O)CCN(C(=O)CCCF)C(Cc2ccccc2)C1 16345,c1(OC)ccc2cc(C(=O)NC3CC3NC(=O)C(C)S(C)(=O)=O)n(C)c2c1 16346,N1(C(C2(F)C(C)C2)=O)CCC(NC(=O)COc2cccnc2Cl)CC1 16347,Clc1ccc2ccc(=NCCc3cnn(-c4ccccc4)c3)[nH]c2n1 16348,C1(NC(C2CC3CCCCC23)=O)CCCNC12CC2 16349,c1(Nc2c(-c3c(C(=O)OC)ncnc3)ccc(OC)n2)cc(Cl)nc2ncnn12 16350,c1(NCC(CCC)OCC)ccc(S(=O)(=O)NCC(CO)C(C)(C)C)cc1Cl 16351,c1(-c2cn(CC(C)NC(C3C(CC)OCC3)=O)nn2)ccc(Cl)cc1Cl 16352,N1(C(C(CCC)NC(N)=O)=O)C2CCC1CC(CC(n1cc(C3CCC3)nn1)C)C2 16353,N1(C(Cc2cc(OC)cc(OC)c2)=O)CCC(C)C(NC(=O)COCC(F)F)C1 16354,c1(C(C)C)ncc(C(=O)NC2CC(CNC(c3cn(CCO)nn3)=O)C2)s1 16355,C1(CNC(=O)OC(C)(C)C)CN(C(=O)Cc2cn[nH]c2)CC1O 16356,C1(NC(C2(SC)CC(O)C2)=O)CN(C(=O)CSc2cccc(Cl)c2)CC1(C)C 16357,C(N=c1[nH]cnc2c(Br)nn(C)c12)C1CN(C(C=NOC)=O)C(C)C1 16358,c1(C(C)C)cc(C(=O)NCC2CCC2NC(C2(C#N)CCC=CC2)=O)cc(F)c1 16359,N1(C(C2CC(OC)C2)=O)CC(CNC(c2cc(CO)[nH]n2)=O)C(C)C1 16360,CCCCCCCCC(F)C(=O)N1CCCCC1c1nnc2n1CCOC2 16361,c1(C(N2CC3C(NC)C3C2)=O)ccc(Oc2ccccc2)c(F)c1 16362,C12(CCNC(C=CSC)=O)CCC(CC1)N(C(=O)Cc1cc[nH]n1)C2 16363,c1(C(=O)NC2(CF)CCN(C(C(CCC)OCC)=O)C2)cncc2ccsc12 16364,c1(C(=O)NCC(CC=C)NC(=O)CCc2cncs2)n[nH]c2c1CC(C)OC2C 16365,c1(C(=O)NC(CN(C(C(c2cccc(C)c2)=O)=O)C)C)cccc(C)c1O 16366,C(=O)(CC(C)CNC(c1ccccc1CC#N)=O)NCC(=C)Cl 16367,c1(C(N(CCN(C(=O)CCCn2cccc2)C(C)C)C)=O)cc2ccccc2o1 16368,c1(NC(c2nc(NC(C3N(C(C)=O)CC(O)C3)=O)sc2)=O)c(C)ccnc1C#N 16369,c1(C(=O)NCC(C)NC(c2ccnc(F)c2)=O)cn2cnnc2cn1 16370,C1(NC(=O)CN2CC(C(F)(F)F)CC2=O)CCCCN(C(c2ccoc2)=O)CC1 16371,C1(CNC(c2ncc(NC)nc2)=O)C2CCC(C2)N1C(C1(C#N)CC2CC2C1)=O 16372,N1(C(C2CCN(C)C2=O)=O)CC(NC(c2cn(C)c(C(F)F)n2)=O)CC1(C)C 16373,c1(N2C(C)CCN(C(c3cccc(F)c3Cl)=O)CC2)nc2c(cc1Cl)C(=O)OC2 16374,c1(OC)ccnc(OC)c1C(=O)NCc1ncoc1CCNC(C1(C)COC1)=O 16375,Cc1ccc(F)cc1NC(C1C2CN(C(=O)CCc3cncnc3)CC12)=O 16376,C1(N(C(=O)CC2CCCCC2)C)CC2CC1N(C(c1c[nH]cc1C(F)(F)F)=O)C2 16377,C1(CC#C)(C(=O)NC(C)CN(C(=O)Cc2ccnn2C(C)C)C)CCCCO1 16378,N1(C(CNC(CN(C)C)=O)=O)CC(NC(C23CCCC2C3(F)F)=O)C(C)(C)C1 16379,c1(C(=O)NC2(CF)CCN(C(=O)CSC(F)(F)F)C2)ccc(C2CC2)c(Cl)c1 16380,C(N=c1[nH]c(=NCCC(F)(F)Cl)[nH]c2c1SCC2)c1cc(CO)ncc1 16381,c1(SC)ncc(C(=O)NCCC2(O)CN(C(c3csc(F)c3)=O)C2)n1C 16382,c1(C(N2CCC(NC(CC(CCC)O)=O)CC(O)C2)=O)cnc2c(cnn2C)c1 16383,C#CCCCCCCCC(=O)N(CCCCCNC(=O)C(C)OCC1CC1)C 16384,N1(C(c2n(CC)nc(C)c2)=O)CCCCC(CCC(=O)NCC2CC(CF)C2)C1 16385,N1(C(c2cc(N3CCOCC3)ncn2)=O)CCC(C2CC2(F)F)C1 16386,CCC(F)(F)C(=O)NCc1ccccc1N1CCN(C(C2(C#N)CC2C)=O)CC1 16387,c1(C(=O)NCC(O)CCNC(C2CCCCCCC2)=O)cncc2c1CCCC2 16388,C1(N(C(C=C(C)C(F)F)=O)C)CCC2CN(C(=O)Cc3ccsc3C)CC12 16389,N1(C(CCCC(C)(C)NC(C2CC2(F)Cl)=O)=O)CCCC2(CCOC2)C1 16390,C1(C(=O)NC(CCOC)C(=O)NCc2ncn(C)n2)CC2C(C1)C2(F)F 16391,N#Cc1ncn(CC(=O)NC2(CC=CC(=O)NCC3C=CCOC3)CCC2)n1 16392,C(CNC(c1nscc1C)=O)(CC(=O)NCCN1CC2CCC1C2)OC 16393,c1(-c2ccccc2)ncc(OCCn2cc(C3CCCO3)nn2)cn1 16394,N1(C(CC2(NC(C)=O)CC2)=O)CCCN(C(C2CCS(=O)(=O)N2)=O)C(CO)C1 16395,C(C(C(=O)O)NC(=O)Nc1cn(C2CCOC2)cn1)OCC=C 16396,c1(C(N2C(C)CCC(NC(c3c(CC)cno3)=O)C2)=O)ccc2cnncc2c1 16397,c1(C(=O)NC2CC(CCNC(c3cncc(C#C)c3)=O)C2)cc(S(C)(=O)=O)cs1 16398,N1(C(Cc2cn(CC)nn2)=O)CCC2(CCC2)C(CNC(c2cn[nH]c2)=O)C1 16399,C(=O)(C#CC(C)(C)CNC(C1CCCN(CCC)C1)=O)Nc1ncccc1NC 16400,C(=O)(C(C)CC(C)C(C)=O)N1C(CCN(C(c2n(CC)ncc2)=O)C)CCCC1 16401,Cc1cc(C(=O)NCC2CCC(CNC(C3CC(N(C)C)C3)=O)CC2)ccc1F 16402,C1(C(N2CCC(N(C(=O)CCSCC)CCC)C2)=O)CC(F)CN1C 16403,C(=O)(CCCC(C)(F)F)N1CCN(C(CC(C)(C)C#N)=O)CC1CF 16404,C1(CNC(c2c(C)onc2Cl)=O)CN(C(C2CCC(=O)C2)=O)CCC1(F)F 16405,C1(CCC(=O)NCC2CC(NC(C(C)C3CCC3)=O)C2)CCCCO1 16406,c1(C(=O)NC(C)CCCCNC(=O)C(C)(O)C2CCC2)cn(C)c(=O)nc1O 16407,Cc1cc(F)c(C(N2CCN(C(=O)CC(C)(C)C)CC2c2cn[nH]c2)=O)cc1F 16408,N1(C(CC2CC(C)(C)OC2)=O)CCC2CN(C(c3ccncc3)=O)CC2C1 16409,n1(CC(=O)NC2CN(C(c3scc(C)c3)=O)CC2F)nc(C)ccc1=O 16410,N1(CC(=O)NCC2CCCN2C(c2cnc(C3CC3)o2)=O)Cc2ccccc2C1 16411,Cc1cc(CC(=O)NC2(CF)CCN(C(C3CCS(=O)(=O)CC3)=O)C2)cc(F)c1 16412,c1(SC)ccc(C(=O)NCC2CC2CNC(c2nn(C)cc2Cl)=O)cc1 16413,Cc1cc(C)c(CC(=O)N(C(C(=O)NCc2cncc(O)c2)C2CC2)C)s1 16414,C(C(=O)NOC(CC(C)C)C(=O)O)C(C)O.Cc1nccn1CCCC(C)C 16415,CC(=O)C(C)CC(C)C(=O)NCC1CC1CNC(c1c(C)cc(C)oc1=O)=O 16416,C1(C)(CNC(CCc2c(C)ncs2)=O)COCCN(C(=O)C(C)C(F)F)C1 16417,N1(C(CC2(C)CC2)=O)CC2CCC2(NC(=O)CCc2ccc[nH]2)C1 16418,C1(O)(CCNC(CC(C)CN(C)C)=O)CCCN(C(=O)C(C)(C)N2CCCC2)C1 16419,c1(NC2C(NC(CSC(=N)N)=O)CS(=O)(=O)C2)nc(N(C)C)cc(C(F)(F)F)n1 16420,Cc1ncc(C(N2CC3(CCN(C(=O)C(C)(C)C)C3)C2)=O)c(Br)c1Cl 16421,C(=O)(C#CC1(C)COC1)NCCCCCN(C(c1c(C)ccnn1)=O)C 16422,c1(CC(=O)NCC2CN(C(C3(C(F)F)CC3)=O)CCCO2)cn2ccsc2n1 16423,C1(NC(CCCC2(NC(C3CCN(CC)C3)=O)CCC2)=O)C(C)CCC1C 16424,Cc1ccc2nc(C(N3CCOC(CN(C(=O)C4=CCOC4)C)C3)=O)c(N)n2c1 16425,C1(OC)CCCC(C(=O)NCC23CC2CN(C(=O)C(CCSC)OC)C3)C1 16426,CC1CN(C(c2cc(F)cs2)=O)CC(C)N(C(c2cc(Cl)c(F)cc2O)=O)C1 16427,c1(CC(=O)NCC2C(NC(C(C)OC)=O)C2)cc(C)nn1C 16428,C#CCC(O)C(=O)N(C)CCC1CCN(C(C2C(Cl)(Cl)C23CC3)=O)CC1 16429,N1(C(c2c(N(C)C)cccn2)=O)CC2CC(NC(=O)CNC(=O)C(C)(C)C)C2C1 16430,C(=O)(NNc1cc(F)ccc1C(F)(F)F)c1ccc(OC(C)C)cc1Cl 16431,C1(NC(c2cc(C(N)=O)ncc2)=O)CN(C(=O)C(F)(F)Cl)CC1(F)F 16432,c1(OCC=C)ccc(S(N)(=O)=O)cc1C(N1CCC1CNC(=O)C(O)C1CC1)=O 16433,c1(CN(C(=O)C(C)OC(C)C)CCNC(C(CSC)O)=O)cccc(Cl)c1 16434,C(=O)(CC(C)(CN(C)C)C(F)(F)F)N(C)CC1CCCN(C(C(F)=CC)=O)C1 16435,c1(CC)ccc(-c2ccc(C3(NC(=O)ON4CCN(C)CC4)CCC3)cn2)cc1 16436,Cc1ccc(C(O)CNC(C2(CN)CCCO2)c2nn[nH]n2)cc1 16437,C(Cc1ccccc1)(C(=O)N1CC(O)(CNC(=O)Cc2nc(=N)[nH][nH]2)C1)N(C)C 16438,c1(C(=O)NC2C3CN(C(c4n(CC)ccc4)=O)C2CC3)nc(C)c(N)cc1C 16439,C(CC(C(=O)N1CCC(C)(CN(C)C)C1)NC(=O)COC)=CC 16440,C1(C(=O)NCc2ccc(C)cc2O)CC2CN(C(=O)CC3CCCCC3)CC2C1 16441,C1(CNC(COC(CC)CC)=O)CCCN(C(c2nnsc2C)=O)CC1 16442,N1(C(C)C)CCC(C(=O)NCC2CCCN2C(C2CCCC3CC23)=O)CC1 16443,Cc1ccc(O)c(C(N2CC3(CC3C(=O)NCC(F)(F)F)C2)=O)c1 16444,N1(C(=O)C2=CCCO2)CCCC2(C1)CN(C(C1C3C4CCC(C4)C13)=O)CCO2 16445,c1(C(=O)NC(C(=O)NC(CCSC)C)C2CCCO2)cnn2cccc2c1 16446,Cn1c(C(=O)NCCCCCNC(c2n[nH]cc2Cl)=O)c2n(c1=O)CCCC2 16447,CCCC(C)CC(C(=O)NCC(C)C)N(CC1CC1)CC1CC1 16448,C12(NC(CCCCC(N)=O)=O)CN(C(=O)CCN3CCCC3)CC1CS(=O)(=O)C2 16449,CC(CC(=O)NC1CCCN(C(c2ccc(C3CC3)cn2)=O)CC1)C(F)F 16450,CC1CCN2CC1C(=O)N1CCC(CC1)C2=O.C(C)(C)(C)NC(C1(C)CC1)=O 16451,CCCC(CC)CC(=O)N1CC(CNC(=O)COCc2nc(C)no2)(OC)C1 16452,N1(C(c2[nH]nc(OC)c2Cl)=O)CCC2(NC(=O)Cc3cscn3)CCCCCC12 16453,c1(C(=O)NC2C=CCCC2)cc2c(OC(F)F)cccc2[nH]1 16454,C(=O)(C(C)P(C)(C)=O)NC1C(N(C(c2cncc(C(=O)OC)c2)=O)C)CCCC1 16455,Cc1cc(Cl)c(C(=O)N(CC(C)(C)NC(c2onc(C)c2C)=O)C)s1 16456,CCCC(CNC(=O)C(C)CC(F)F)CCO 16457,S(=O)(=O)(c1cc(NC(c2ccc3c(c2)CCO3)=O)ccc1F)NCC#N 16458,c1(OC)ccc(C(N2CCCC(C)(CNC(C3(N(C)C)CCC3)=O)C2)=O)cc1Cl 16459,CC1CC(C(N2CCCC2CN(C)C(c2cncs2)=O)=O)CC(C)C1 16460,c1(CNC(C2CC2Cl)=O)cccc2c1CN(C(c1ccn3nnnc3c1)=O)C2 16461,c1(C(N2CCC(NC(C3(OC)CCCC3)=O)C(F)C2)=O)ccc2nc(O)[nH]c2c1 16462,N1(C(Cc2scc(C)c2)=O)CCCC(C(C)NC(=O)C(C)(C)n2cccn2)C1 16463,c1(C(N(C(CC2(NC(C)=O)CC2)=O)C)=O)nc(CNC(=O)C=CC(C)(C)C)cs1.C 16464,CC(CC(C)(C)C)NC(=O)C(c1cccs1)NC(=O)CC1NC(=O)NC1=O 16465,C(=O)(CCCCC(C)CC)N1CCC(C)(CCNC(c2c(CC)noc2C)=O)C1 16466,c1(OCC)ccnc(N(CC(C)(C)CNC(C2CC2c2ccco2)=O)C)n1 16467,N1(C(CNS(CC)(=O)=O)=O)CCN(C(=O)Cn2cnnc2O)C2CCCCC12 16468,C=C1CCN(C(=O)CSCCCOC)C(C(=O)NC(C)Cn2ccnn2)C1 16469,C1(CC(N2C(CNC(=O)C(C3CCCCC3)O)COCC2)=O)CCC(F)(F)CC1 16470,N1(C(C(C(C)C)C)=O)CC(CNC(c2cc3ccccc3o2)=O)OC(C)(C)C1 16471,N1(C(CC(C=C)C)=O)CCC2(CCC2CNC(c2oc(CO)nc2C)=O)CC1 16472,C1(C(N(CCNC(CCCOCCOCCOC)=O)C)=O)Cc2ccncc2C1 16473,c1(C(C(=O)OC)C)cn(CCCC(=O)N(C)C)nn1 16474,C1(NC(CCN(CC)CC)=O)CC2(C1)CC2NC(c1scnc1Cl)=O 16475,CC(CC1CC1)C(=O)NCC(C)(C)NC(=O)C(C)n1ccnc1 16476,C1(C(=O)N2CCC(COC)C2)(CCC)CCOc2ccccc21 16477,CS(C)(=O)=NC(=O)C(=O)NC1CC(c2ccccc2)(NC(=O)COC(F)(F)F)C1 16478,C1(CNC(C(COC)OC)=O)CN(C(=O)CC2CN(C(C)=O)C2)CCN1C 16479,O=C1NCC2(CCN(C(C3CCOCC3NC(=O)C(O)CC3CCCC3)=O)C2)N1 16480,C(=O)(CC(C)NC(=O)CC1(C)OCCO1)NC(CC#C)C 16481,N1(C(CS(C(C)C)(=O)=O)=O)Cc2nccn2CC(NC(=O)C=C2CCC(C)C2)C1 16482,C(c1cccc(CO)c1)=CC(=O)NC1CCN(Cc2nccc(C)c2)C1 16483,c1(OC)ccc(C(CO)NCC(O)COC(C2CC2C(C)(F)F)=O)cc1 16484,Cc1cc(C(=O)NC(C)(C)CC=CC(=O)NC(C)C(C)F)n[nH]1 16485,CCC(CC(=O)N1CCC1CNC(c1ccc(CNC(C)=O)o1)=O)c1ccccc1 16486,N1(C(c2c(C)oc(C(C)C)c2)=O)CC2(C1)SCCC2NC(c1ccnn1C)=O 16487,CC(CN(C)C(c1cccc(OC(F)F)c1)=O)N=c1ccnc[nH]1 16488,c1(OC)cc(Br)cnc1C(=O)NCC(C)NC(c1cnn2c1OCC2)=O 16489,c1(C(=O)NCC(C)N(C(=O)C=Cc2cc[nH]c2)C)cc2cc(Cl)cc(Cl)c2[nH]1 16490,c1(CC(=O)NCCNC(c2ccn(CC)c2C)=O)ccc(C)cc1C 16491,C1(NC(C2CC(C(=O)Nc3ccc(CO)s3)C2)=O)CCOC12CCOC2 16492,N1(C(C=CC(C)C)=O)CC(NC(c2ccc(-n3ccnc3)nn2)=O)CC2(CC2)C1 16493,CC(=O)CCCC(=O)NC(C)(CNC(c1nccc(Cl)c1Cl)=O)C1CC1 16494,n1(CCNC(C(C)C2(O)CCC2)=O)ccc(C(=O)NC2(C(C)(F)F)CC2)c1 16495,CC1CN(C(=O)C=CCF)CC1NC(C1(c2cccc(Cl)c2)CCCCC1)=O 16496,CCCCCC(C1CC1)NC(=O)CC1CC(C(=O)NC2CCOC2C)C1 16497,C(=O)(CCCCCCNC(c1cccnc1)=O)N1CC(CC(C#C)C)C1 16498,C(C)(C)(CCN=c1[nH]cnc(C)c1Br)NC(COc1c(C)occc1=O)=O 16499,CC(C)(C(=O)NCC(CC1CC1)C(=O)NCCCP(C)(C)=O)C(F)(F)F 16500,C#CCN(OC)C(=O)C1(CF)CCN(C(c2cn(C)c(C)n2)=O)C1 16501,CC(CCC(F)(F)F)NC(=O)CC(C)(C)NC(=O)Cc1ccsn1 16502,C(=O)(C1=CC2(CCN(C(=O)C(C)(C)C(O)C(C)C)C2)C1)NCCC(CC)(C)O 16503,c1(COC(C)C(=O)NC(C2(O)CN(C(c3cc(Cl)no3)=O)C2)C)ccc(F)cc1 16504,Cn1cc(C(=O)N(CCCNC(c2cn(C)cn2)=O)CC2CCCC2)c(Cl)n1 16505,Clc1ccc(C(c2nnnn2Cc2ccccc2)NCCOCC2CC2)cc1I 16506,c1(SC)nc(C)c(CCC(=O)NCC23CCCC2CCN3C(=O)C(C)C)c(O)n1 16507,C(CC(=O)NNc1ccccc1)c1cn(C(C)C)nc1.C(C)(C)SC 16508,C1(NC(CS(C)(=O)=O)=O)CC(NC(=O)CCCn2cnc(C#N)n2)C12CCC2 16509,C(=O)(CC1=CCCCC1)N1CC2C(COc3ccc(OC)c(O)c3)(CC2)C1 16510,c1(C(N2C3C(NC(=O)C=CC(F)(F)F)C(CC3)C2)=O)sc2ccccc2c1CO 16511,Nc1nc(C(N2CCC3(NC(=O)CCSC(F)(F)F)CC3C2)=O)ccc1O 16512,C1(CCCC)CCC(C(N2CC(NC(c3cncc(F)c3)=O)C(C)C2)=O)CC1 16513,c1(C(N2CCC(N(C(C=CC=CCC)=O)CC)C2)=O)csc(=NC2CC2)[nH]1 16514,N1(C(c2cn(CC)nn2)=O)CCC(NC(=O)CCc2cccc(C)c2)C(CO)C1 16515,C(C1=CCN(C(c2coc(CC)n2)=O)C1)NC(C(=O)NCC)=O 16516,CCC(C)(C)C(=O)N1CCC(N(CCO)C(C2CCC(C)(C)O2)=O)C1 16517,c1(C(=O)NCC23N(C(COCC)=O)CCC2CC3)cc(Cl)c(OC)c(Cl)c1 16518,C1(C2CCCN(C(=O)CN3CC4CC4C3)C2)(NC(C2(OC)CCOCC2)=O)CC1 16519,CN1CCCC2(CCN(C(C(=O)NCCCF)C3=NOC4CC34)C2)C1 16520,N1(C(Cc2c(OC)nccc2)=O)CCN(C(C2CC2CF)=O)C(CCO)C1 16521,N1(C(=O)NC2CC3(C2)CC2CCCC32)CCn2ncc(-c3nn[nH]n3)c2C1 16522,N1(C(c2onc(CC)n2)=O)CCC(C)C(CNC(=O)CCCCF)C1 16523,c1(C(=O)NC(C2CCN(C(C3CC(=O)NC3(C)C)=O)CC2)C)cccc(O)c1Cl 16524,N1(C(C2C(OCC)C2C)=O)CCOC(CNC(=O)CN2CC(=O)NC2=O)C1 16525,Cc1ccc(C(N2CCC(F)(C(=O)NCCCC(C)(C)O)CC2)=O)nc1C 16526,C1(CCC)CN(C(C2OCCC2C)=O)CC1C(=O)NCCc1ccn(CC)n1 16527,CCC(C)(CNC(=O)COC1CC(NC(C2CCCCO2)=O)C1)CC 16528,C1(O)(C(=O)NCCN(C(=O)Cn2ccc(C3CC3)n2)CC)CCCC(C)(C)CC1 16529,Cc1ocnc1CC(N1CSCC1C(=O)NOC(c1ccccc1)C)=O 16530,N1(C(C)=O)CCCC1C(N1CC(O)(C(C)NC(=O)C(C)(C)c2ccnn2C)C1)=O 16531,C(=O)(C1=CCC(NC(c2cnn[nH]2)=O)C1)N(C)Cc1ccccc1O 16532,CN1CC(N=c2nc3c(ncn3C)c(NCc3c[nH]ccc3=N)[nH]2)C1 16533,c1(N2C(C)CC(NC(C34CCC(N=[N+]=[N-])(CC3)C4)=O)C2)nc2ccc(F)cc2s1 16534,CCC(C#N)(CC)C(=O)NC1CCCC(NC(=O)CCNC(=O)CC(C)C)C1 16535,CC(C)(CC(F)C(=O)NCCC1CCSC1)NC(C1CC12CC2)=O 16536,c1(NC(C2(C)CCN2C(c2ccc3c(c2)OCO3)=O)=O)ccc2ncnc(O)c2c1 16537,c1(C(N(C(C)CCNC(C2CCCC(F)C2)=O)C)=O)cn2c(n1)CCC2 16538,C(=O)(CCCN=[N+]=[N-])NCCOCCCNC(C1(OC)CCCC1)=O 16539,C1(CNC(c2coc3c2CSC3)=O)CN(C(=O)C=CBr)C2CCN1C2 16540,c1(C(=O)NC2(CCn3ccnc3)CCOC2)ccc(OC(F)F)c(F)c1 16541,c1(C(=O)NCCOCC(=O)OCC2C(OC(C)=O)COC2)ccnc(O)c1 16542,C1(C(=O)NCC2(F)CC(NC(C3(CC(C)C)CC3)=O)C2)CCC2C(C1)C2(F)F 16543,C1(NC(c2c(C)cc(CO)o2)=O)CN(C(C2(C)CCCCO2)=O)CC1(C)C 16544,C1(NC(C2(C(=O)NC)CC2)=O)CC2CCC1CC2NCc1cc(Cl)ncc1OC 16545,N12CCC3CC(C3C1)C2=O.N1(c2n(C)ccn2)CCC(F)(CO)CC1 16546,C(C)(C)(C(C)CC(=O)NC1CCCC1CCC(C)C)OC 16547,N1(C(C=CC(C)(C)C)=O)CC2(C1)SCCC2NC(=O)COCC1(F)CC1 16548,C1(N(C(C=CC(CC)=CC)=O)C)CN(C(=O)Cn2ncc(Cl)c2C)CC1(C)C 16549,Cc1nnccc1NC(=O)C(=O)Nc1ccc(CC(=O)NC2CC2)cc1 16550,N1(C(C=CC(C)=O)=O)CCC2CN(C(=O)CCCc3ccsc3)CC12 16551,C1(C(=O)NCC(C)NC(=O)C(c2ccc(C)cc2)(F)F)(CC)CCCCC1 16552,Cc1nn(C)c(N)c1C(N1CCOC(CC(N2CC(C)C2(C)C)=O)C1)=O 16553,CC1(C)C(C(=O)NCC2CN(C(=O)Cc3ccno3)CCO2)C1(C)C 16554,NC(CC(=O)N1CCCCC1CCc1ccccc1F)C(=O)O 16555,c1(OC)c(Br)cc(C(=O)O)cc1S(=O)(=O)NCCSC.C(C)(=O)N 16556,Cc1cnc2n1CCC(NC1CCS(=O)(=O)CC1)C2 16557,c1(OC)ccc(C(=O)NCC(C(C)(C)C)NC(=O)Cc2cc[nH]n2)c(F)n1 16558,S(=O)(=O)(c1cccs1)NCCC(=O)NCCN(C(C(C)(C)SC)=O)C(C)C 16559,N1(c2snc(C)c2C#N)CC2CCC1C1CN(C(=O)CSc3nc[nH]n3)CC21 16560,C(C(C)(O)CC(=O)N(C1CCCN(C(c2nc(C)n(C)c2C)=O)C1)CCO)OC 16561,c1(CC)[nH]nc(C(=O)NC(CNC(c2ccnc(C(C)C)n2)=O)C(C)(C)C)c1C 16562,c1(C(=O)NC2CC(NC(c3c(C)ccc(F)c3)=O)C(O)C2)cccc2c1NCC2 16563,O=C1CN(C(c2cocn2)=O)C2CCN(C(=O)CSC(F)(F)F)CC2N1 16564,C(=O)(CCC(C)NC(C1CC(O)C(F)C1)=O)NC1(C(=O)OC)CC(C)C1 16565,c1(C(=O)NCC2CC(C)N(C(=O)CN=S(C)(C)=O)C2)cc2c(F)ccc(F)c2[nH]1 16566,c1(C(=O)NCC(CC(C)C)NC(c2cnc(S)[nH]2)=O)cc(O)ccc1Br 16567,C1(C(N2C(C(=O)NC3(COCC)CC3)CC(O)C2)=O)CCCCN1N=O 16568,N1(C(C2C(CC)C2)=O)CC2CN(C(=O)CC3(OC(C)=O)CCCC3)CC2C1 16569,C(=O)(C(CC(C)C)C(C)C)N(CCC(O)CCc1cn(CC(C)(C)CO)nn1)C.CO 16570,N1(C(C2(CC=C)CCOC2)=O)CC(NC(c2cccc(F)c2C)=O)C(C)(C)C1 16571,C(=O)(C1=NOC(C)C1)N(CCCC(=O)NC(CCOC)COC)C 16572,NS(=O)(=O)c1cccc(C(N2CCOCC2Cc2cn(CCCF)nn2)=O)c1 16573,C(=O)(C1=CCC2CCC1N2C(=O)C(C#N)C(C)(C)C)N(CC=CC)CC 16574,C1(OCC)CC2(C1)CC2C(=O)NCCN(C(=O)CC1CC2C=CC1C2)C(C)C 16575,C1(C(N2CC(CNC(COCc3ncc(C)o3)=O)C2)=O)CC2(CCC2O)C1 16576,N1(C(COCC=C)=O)CCc2ccc(C(N3CC(C)CC(C)C3)=O)nc2C1 16577,CN=c1[nH]c(C(N2CC(C(C)NC(C3CCN(CC(F)F)CC3)=O)C2)=O)cs1 16578,c1(OC)ccc(C(C(=O)O)NC(C2CCCCC2(F)F)=O)cc1Cl 16579,C(=O)(C(CNC(c1cc(C(N)=O)[nH]n1)=O)OC)NCC(=C)Cl 16580,C1(O)(CN(C(C2C(C#C)C2)=O)C)CCN(C(=O)Cc2sccc2Cl)C1 16581,N1(C(C#CC(C)(C)C)=O)CCCC(NC(=O)C=C2CCCCC2(C)C)C(F)C1 16582,Cc1ncccc1CC(=O)N(C1CCCCC1)CCNC(=O)CC1CC2(COC2)C1 16583,C(=O)(C(C)CCCOC)N1CCC(CC(C)NC(COCC(C)C)=O)CC1 16584,c1(C(=O)NC2(CC=C)CN(C(=O)C(C)S(N)(=O)=O)C2)c(OC)cccc1OC 16585,c1(C(N2CC(NC(C3CN(OC)C(=O)C3)=O)C(C)C2)=O)nccn2cc(C)nc12 16586,C1(C(=O)N(CCO)CC2CCCO2)CC(F)CN(C(=O)Cc2cc(F)cc(F)c2)C1 16587,N1(C(CC2CCC(C)CO2)=O)CCC2CN(C(c3ccc([N+](=O)[O-])[nH]3)=O)CC12 16588,S(=O)(=O)(c1ccc(C#N)c(N2Cc3ccc(C)nc3C2)c1)NC1CC(=C)C1 16589,C(=O)(C(O)CC[S+](C)C)N1CCC(NC(c2c(C#C)cnn2C)=O)CC1C 16590,N1(C(c2c(C#N)cn[nH]2)=O)CCCCC(CNC(c2nc(Br)c[nH]2)=O)C1 16591,c1(C(=O)NC2C3CN(C(c4ccc(NC)c(F)c4)=O)C2C3)cc2n(n1)CCCO2 16592,N1(CC(COC)O)CCC(N(C(=O)CC2CCN(c3ccccc3)C2)C)CC1 16593,C1(C(=O)OC(C)(C)C)CCOC(=O)CC1.C12(C(=O)Cc3cccnc3)CCN(C1)C2 16594,C#CC1CCN(C(=O)C(CCCOC)NC(=O)C(C)N(C)C(C)=O)CC1 16595,c1(C(N2C(CC)C(NC(C3CC(=O)C3C)=O)CCC2)=O)cc2nc[nH]c2cn1 16596,N1(C(C(C2CCN(C(=O)CCCC3CC3)C2)C)=O)CCCC2(CCC2)C1 16597,C1(CC)C(C(=O)NCCNC(C)=O)CCN1C(=O)CC(=O)NC 16598,CC1(C)CC(NC(c2ccc(C3CC3)cn2)=O)CN(C(c2cccnc2S)=O)C1 16599,N1(C(C(CC=C)CNC(C2C3(CC3)C23CC3)=O)=O)CCc2ccc(F)cc21 16600,N1(C(CC(C(N)=O)NC(C)=O)=O)CC(CCO)OCC1(C)C 16601,c1(C(N2CC(COC)(CNC(C3CC3C)=O)C2)=O)noc2ccc(Cl)cc12 16602,N1(C(c2c(C)oc(CNC(=O)CCc3ccncc3)n2)=O)CCc2nc(O)[nH]c2C1 16603,S(=O)(=O)(c1cc(Cl)sc1Cl)CNC(C(=O)OC)C(C)C1CC1 16604,c1(-n2c(CCCSC)nc(-c3ccccc3C)n2)cc(C)cc(C)c1 16605,CC1CN(C(c2cccc(C#N)n2)=O)CCC1NC(c1ccoc1Br)=O 16606,C1(OC)CCC2(C(=O)NCCC(C)(C)NC(c3cccc(OC)n3)=O)CCC12 16607,C(C(CC(=O)NCC(O)COC)OC)NC(CC=CC=C)=O 16608,c1(NC(C2(CC(C)C)CCCC2)=O)cccc(CNC(c2ccoc2Br)=O)c1 16609,C1(NC(CSCCC)=O)CCCN(C(c2c[nH]cc2C(C)(C)C)=O)CC1 16610,C1(C2(O)CCN(C(C3CC3[N+](=O)[O-])=O)CC2)(NC(C=C(C)c2ccco2)=O)CC1 16611,C1(C)(CNC(c2cnc(CC)o2)=O)CN(C(C23CC(F)(C2)C3)=O)C(C)(C)C1 16612,CCC(C(=O)NCCC1CCCN1C(=O)C(C)ONC(=O)OC(C)(C)C)N(C)C 16613,n1(C(C)(C)C)cc(Cl)c(=NC(=O)NCC(F)(F)F)[nH]1 16614,N1(C(c2c(OC)ccnc2O)=O)CCOCC(C)(CNC(c2cn(C)nn2)=O)C1 16615,Cc1c(C(=O)NCC(C2CCC2)NC(c2cc(-c3ccco3)no2)=O)nnn1C 16616,N1(CC)CC(C(N2CC=C(CNC(=O)CCc3ccnn3C)CC2)=O)CCC1=O 16617,c1(C(=O)OC)cccc2c1CCC2NC(C1CCC(C(F)(F)F)N1)=O 16618,C1(C(=O)NC2CC2C(N(CC(CC)OC)C)=O)(OCC)CCCCC1 16619,C1(NC(C2N(C)CCCC2)=O)C2CC3C(C2)C13C(N1CC(OCC(N)=O)C1)=O 16620,c1(C(N2C3CC(C(=O)NC(CC#C)C(=O)NC)C2CC3)=O)ccn2ccccc12 16621,C1(NC(C2ON=C(C)C2)=O)CCOCC1NC(c1nocc1C1CC1)=O 16622,c1(CC(=O)NCC(C2CC2)NC(C(C2CCC2)OCC)=O)sc(O)nc1O 16623,C1(N(C(CC2(C=C)CCC2)=O)CC)CCN(C(=O)CNC(C2CCCC2)=O)CC1 16624,N1(C(C2COCCN(C(=O)NC(C)C(C)(C)CO)C2)=O)CCCc2ccccc21 16625,C1(CC)CCCN(CC(=O)NCCN(C(=O)Cc2ccc(CC(C)C)cc2)C)C1 16626,CCCCN=C(NCCc1ncc(C)cn1)NCC1CC1CC 16627,CC1OCCOC1C(=O)NC(C)(C)CC(=O)N1CCC(C(N)=O)C1 16628,c1(C(=O)NCC2CCN(C(=O)Cc3cn[nH]c3)C2)cc2n(n1)CCO2 16629,C1(NC(c2c(CCC)nco2)=O)CCN(C(=O)C(C)c2ccco2)C1C(C)C 16630,C1(C(N2CCOCC(CNC(CC(C)C)=O)C2)=O)CCCN2CCCCC12 16631,CCCCCC(C(=O)NC1CN(C(=O)CN2CSCC2=O)CC2(CC2)C1)C(C)C 16632,C1(C(=O)NCC2(NC(C(CC)F)=O)CCCC2)CCCCN1S(C)(=O)=O 16633,N1(C(C2C(CNC(Cc3c(C#C)cccc3)=O)CC2)=O)CCC(C2CCC2)CC1 16634,CC(C)(F)CC(=O)NCC1COC(CNC(c2ncsc2Br)=O)C1 16635,C(=O)(C1=NN(CCO)C(=O)CC1)N1C(CC)CN(C(c2cnc[nH]2)=O)CC1 16636,CSC=CC(=O)N1CCCC1CNC(=O)COC1CCC1 16637,CCCCCC(O)C(C)C(=O)NC1CCCN(C(=O)CNC(C)=O)CC1 16638,c1(CC(C)NC(=O)C(Cn2cncn2)NC(c2cncs2)=O)ccccn1 16639,C=CC1CN(C(C2(N(C)C)CCCC2)=O)CC1NC(=O)CC(C)C1CCCCC1 16640,N1(C(C2CC(C(C)C)C2)=O)CCCC(CO)(CNC(=O)C(C2CCCCC2)F)C1 16641,c1(NCCC2CCSCC2)nccc(=NC2CC(NC3CCCC3)C2)[nH]1 16642,C1(NC(C(CNC(=O)C(C)n2cncn2)OC)=O)CCC(C2CC2)C1 16643,C1(CC)CCCCC1C(=O)NCC(O)CN(C(=O)Cc1sc(O)nc1O)C 16644,Cc1oc(C)c(C(=O)NCc2ocnc2C(=O)NC2CCCC(O)CC2)c1C 16645,C1(C(N2C(C)(CNC(=O)C=CBr)CCC2)=O)CCCC12CCC2 16646,C1(CNC(CC(C=C)c2ccccc2)=O)CN(C(=O)C(F)(F)CC)CCCO1 16647,N1(ONC(C2C(C)OCCC2)=O)CCSCCC1c1ccccc1.CC(=O)O 16648,C1(C(=O)NC(C(N2CC(C(N)=O)OCC2)=O)c2ccco2)CC2CCCC2C1 16649,Cc1cc(=NC(C)CCNC(C2(F)CCC2)=O)c([N+](=O)[O-])c(C)[nH]1 16650,c1(CC(CO)N(C2CCCC2)C(c2[nH]cc(C(=O)O)c2)=O)ccccc1 16651,C#CCC(C)(CNC(C1C=CCN(C(=O)CC(C)n2cccc2)C1)=O)CO 16652,N1(C(CC(C)SC)=O)CCCC(C)(C(=O)Nc2cccc(F)c2)C1 16653,c1(OC)ncc(CN2CC(NC(C3CCC3)=O)C(C#N)C2)c(OC)n1 16654,Cc1c(C(=O)NC(C2CCOC2)CNC(=O)C2=CCCCO2)nc2sccn12 16655,C1(CC(=O)NC2C(C(=O)OCC)CC2)CN(C(C2(SC)CCC2)=O)CCC1C 16656,C=CCC(C(=O)N1CCCC1CCNC(C1CN(C(N)=O)C1)=O)C(C)(C)C 16657,c1(CN2CC(C)(CNC(c3cc(Cl)c(F)cc3F)=O)C2)cn2ccccc2n1 16658,CCCC(C(=O)N1CC(O)CC1CC(N1CC2(CC(N(C)C)C2)C1)=O)C(C)C 16659,CC1CN(C(c2cc(=O)cc[nH]2)=O)CC1CNC(=O)CC1(O)CC1 16660,C1(NC(C2CC(OC)C2)=O)CS(=O)(=O)CC1NC(c1sccc1-n1ccnn1)=O 16661,S(=O)(=O)(c1ccc(Cl)cc1)NCCC(=O)NC(CNC(CCC(=C)Cl)=O)C(C)C 16662,CCCC(CCCNC(=O)C(c1ccc(C(F)(F)F)nc1)C)NC(C12CC1C2)=O 16663,C1(CNC(C(C(CC)C)O)=O)C(C2CC2)CCN1C(c1ccsc1C)=O 16664,c1(NC(C23CC(C(=O)Nc4cncc(Br)n4)(C2)C3)=O)cc(O)cc(O)c1 16665,C1(C(N2CC(N(C(c3c(CC)ncs3)=O)C)C(F)C2)=O)CCC2(CCC2)CC1 16666,C1(C(=O)NC(c2ccncc2)CC)CN(S(=O)(=O)Cc2cccnc2)CCN1 16667,CC(C)(C)C#CC(=O)NCC1CCCN(C(C2CCC(=O)N2C(C)=O)=O)C1 16668,c1(C(=O)NCC2OCCC(NC(CC3C(C)CCO3)=O)C2)cn2cccnc2n1 16669,N1(CC(=O)NCC(CC)NC(c2ccc(CNc3nccs3)o2)=O)CC(C)(C)C1 16670,Cc1ccccc1C1CC1C(=O)NC1CC(NC(c2ccnc(S)c2)=O)C1 16671,c1(NCCNC(=O)NC2C(C)CN(c3ccc(F)cn3)C2)cccc(F)c1[N+](=O)[O-] 16672,C1(N(C(C(CSC)OC)=O)C)CCC(NC(=O)C(C2(O)CCCCC2)(F)F)CC1 16673,C(=O)(C1CCCc2nn[nH]c21)NC1CN(C(C(C)OCOC)=O)CC(F)C1 16674,CC1CCCN1CC(=O)N(CC(=O)NC(c1cnn(C)c1)CO)CC(C)O 16675,C1(CNC(c2n(CC)cnn2)=O)CC2CC2N1C(c1ccncc1Br)=O 16676,N1(C(CCC(C)NC(c2c(C)c[nH]c2)=O)=O)CCC(O)CC(C)(C)C1 16677,c1(CNCC2N(C(c3cnc(OC)nc3C)=O)CCOC2)cnc2[nH]ccc2c1 16678,Cc1nc(C)c2c(n1)OC(CNC(=O)N(C)CCc1ccc(Cl)cc1)C2 16679,CC(C)C(C)(F)CNC(C1CC(C)N1C(=O)C(=O)NCC1CC1)=O 16680,c1(C(=O)NCC(C)N(C(C(C)OCC#C)=O)C)ccc(-c2cccs2)cc1F 16681,C(=O)(CCC(C)NC(=O)CC1(NC(C)=O)CC1)NC1(CC=C)CCCC1 16682,C12(CC(N3CC(SC)C3)=O)CCC1CN(C(C1CCC=CCC1)=O)C2 16683,c1(CCC(=O)NC(CCCC)CNC(c2c[nH]nc2F)=O)n[nH]c2c1CCCC2 16684,C1(F)(CNC(c2c(CC)cco2)=O)CCN(C(c2c(C)nsc2N)=O)CC1 16685,c1(NCC2N(S(C)(=O)=O)CCOC2)cccc(F)c1CNC1CCCC1 16686,N1(C(N=c2n(CC(C)C)[nH]cn2)=O)CCCC2CN(C)CC12 16687,Cc1cc(F)c(I)cc1C(N1CC2CN(C(c3cnnn3C)=O)C2C1)=O 16688,CCCC(C(F)(F)F)c1nc(-c2cc(OC(C)C)ccn2)nn1CCN(C)C 16689,c1(C(N(CCCNC(C(c2scc(C)n2)C)=O)C)=O)ccc(O)c(F)c1 16690,C1(NC(C(=O)NC(C)C)=O)CCS(=O)(=O)C2(C1)CC(CNC(=O)CC(C)C)C2 16691,Fc1ccc(C(=O)CN2CCC(COc3ccccn3)C2)c(F)c1Cl 16692,C1(C)(NC(CC(=O)NCC)=O)CCCN(C(C23CCC(CC2)C3)=O)C1 16693,c1(C(N2CC(CCCCNC(C(C)CC(F)F)=O)C2)=O)c(O)cc(Cl)cc1F 16694,N1(C(C(Cc2ccc(C)cc2)C)=O)CCC(NC(=O)COCCO)C12CCCC2 16695,C1(CNC(C(=O)NC(c2cccc(Cl)c2Cl)C)=O)CC1C1CCOCC1 16696,c1(NC(c2c(C(N(CCC)CCC)=O)[nH]nn2)=O)cccc(F)c1C(=O)OC 16697,C(=O)(C1=CCCOCC1)NC(C1CCN(C(c2n[nH]c3c2CCSC3)=O)C1)C 16698,c1(OC)cc(Cl)c(CN2CCC3CN(C(=O)C=CC(C)C)CC23)cc1OC 16699,C1(C(=O)OCC2C3(CC)CC3CC2)(NC(=O)OC(C)(C)C)CCS(=O)(=O)C1 16700,c1(OC)nc(Cl)ccc1C(N1CCC(CNC(c2ccc(Cl)[nH]2)=O)(OC)C1)=O 16701,c1(C(=O)NC2C(NC(C3OCCN(CC)C3)=O)CCC2)cc(=O)c(C)c[nH]1 16702,C(=O)(CCC(=O)NN(C)C)NC(CCNC(C(CCC)OC)=O)Cc1ccccc1 16703,S(=O)(=O)(c1cccc(Br)c1F)N1CCN(C(c2ccc(OC)cc2Br)=O)C(C)C1 16704,C1(O)(C(N2CCCC(CN(C)C(c3ccnnc3Cl)=O)C2)=O)CCCC(C)CC1 16705,C(C(=O)NCCSC)(C1=CCSC1(C)C)N(CCCN(C)C)CC.C(=O)OC 16706,CCC(CC)CCNCC1(C)CCOCC1 16707,c1(NC(=O)NC2CCCC2Cc2c[nH]c(Br)c2)ccc(N2CCCC2=O)cc1 16708,C1(CCOC)CN(C(C2CC3C=CC2O3)=O)CCN1C(c1cn(C(C)C)nn1)=O 16709,c1(C(=O)NC2CCN(C(C(C)OC)=O)CC2F)n[nH]c2c1CCC2C 16710,C(=O)(C(CCF)NC(c1ncccc1C)=O)NC(CCC=C)C 16711,C(CCC(=O)N(C)CCNC(C1CCCC1CC)=O)N(CCC)CCC 16712,N1(C(c2ccsc2)=O)CCCC(C(=O)NCCNC(=O)CN2CCCC2=O)C1 16713,C1(NC(C(CCN(C)C)NC(c2ncccc2O)=O)=O)CCC(C2CC2)CC1 16714,c1(C(C)OC(C2C(C)(C)C2(C)C)=O)ccc(Cl)cc1F 16715,CC1(C)CCC(=CC(N2CCCCC2CNC(c2n[nH]cc2[N+](=O)[O-])=O)=O)CC1 16716,c1(CCOC)n[nH]c(=NCCC2CCN(C(=O)CNC(c3ccc(C)s3)=O)C2)s1 16717,C12(C(=O)NCC(CN(C(Cc3cc(C)ns3)=O)C)O)CC(C)(C1)OC2(C)C 16718,c1(OC)cc(C(=O)NC(Cc2cnn(C)c2O)C(=O)N2CC(C(C)O)C2)n(C)n1 16719,C1(OC)C2CC3CN(C(c4sncc4C)C(=O)NC4CCOC4)C1C3C2 16720,C1(N(C(CC(=O)N(C)C)=O)C)CN(C(=O)C=Cc2ccccc2)CC1O 16721,c1(CNC(=NCCc2ccncc2)NCCc2cccs2)csc2ccccc12 16722,C(=O)(C(CCC)NC(=O)C(C)(C)O)NCc1cn(CC=C)nn1 16723,Cc1cc(F)cc(C(=O)N(CC(C)NC(c2nc(C)n(C)c2C)=O)C)c1N 16724,CC(C)(C#N)CCCC(=O)NC1CC(NC(C2(C)CC2F)=O)C1 16725,n1(CC(=C)C)nnnc1C(c1nc(C(F)(F)F)cs1)NCC1(C)CCCC1 16726,CCC(C)CCC(=O)N(CCC(C)NC(c1cnn(CCN(C)C)c1)=O)C 16727,c1(NC)ccc(C(N2CC3CC(NC(c4cc(C)c(C)o4)=O)C2C3)=O)cc1F 16728,N1(C(C(C)SCCCC)=O)CCN(C(=O)C=C(CC)CC)CC(CO)C1 16729,c1(CNC(C2CCC3(CCC3)CC2)=O)nc2cccnc2[nH]1 16730,C12(C(=O)NCCOCCNC(C3CCS(=O)(=O)N3)=O)CCN(CC1)CC2 16731,c1(C(N(C(C)C)CCNC(C23CC4CC2C3C4)=O)=O)nccn2nccc12 16732,c1(NC(C(CCSC)OC)=O)ccc(NC(C)C(=O)NC)cc1F 16733,C1(CNC(=O)Cc2cc[nH]n2)CCCC12CCN(C(c1cccnc1Cl)=O)CC2 16734,c1(C(N2CC3C(C(=O)NC4CCCCC4(F)F)C3C2)=O)cc(F)cc(F)c1F 16735,Cc1cnc(C(N2CC(C(=O)NC3(C)CCSC3)C(C(C)C)C2)=O)cn1 16736,C1(C(N2CCCC(NC(CCC(C)C)=O)C2C)=O)CCC2(CCC2)CO1 16737,N1(C(CC2(N(C(C(CSC)OC)=O)C)CC2)=O)CCC(O)C1C 16738,N1(C(C2C(C(=O)Nc3cc(C)[nH]n3)C2)=O)CCSCC1(C)C 16739,c1(C(N2CCC(NC(C(COC)N(C)C)=O)C2(C)C)=O)cnc2n1CCCCC2 16740,CCCCC(O)CC(=O)N1CCC(C(=O)N(C)Cc2cccc(C)n2)C(C)C1 16741,c1(CCC(=O)NC(CC=C)CNC(c2coc(C)c2)=O)ccc(O)nc1 16742,c1(C(=O)NCC2C(NC(C3CC(C)(C)C3)=O)CCC2)c[nH]c(=O)cn1 16743,C1(NC(CCCCCOC)=O)CN(C(=O)CCC2CC2(C)C)CC2CCCC12 16744,c1(C(N(CCCOCCNC(C2C(C=C)C2)=O)C)=O)ccc(C)nc1N 16745,c1(CC)nc(C(=O)NC(C)C(C(C)C)NC(c2ccnn2CC(F)F)=O)c(C)o1 16746,C1(NC(c2c(SCC)nccn2)=O)COC2CN(C(c3cscc3OC)=O)CC12 16747,C(=O)(CC(C)C(C)(C)NC(=O)CSc1cn[nH]c1)N(CC(COCC)O)C 16748,C(C1CCCN1C(c1cscc1OC)=O)=CC(N1C(C#C)CC1)=O 16749,c1(C(=O)NC2CC2C(=O)Nc2ncncc2Cl)cc(O)nc2ccccc12 16750,C(C1=NOC2CN(C(C3(C)CCCC3)=O)CC12)NC(C1(COC)CC1)=O 16751,c1(C(=O)NCC2(F)CCCN(Cc3c(C)ccc(C)c3)C2)c(Br)ccc(C)c1F 16752,C1(NC(c2c(C)ccn2C)=O)COC2(CNC(=O)C(=O)NC(C)C)CC1C2 16753,C1(C(=O)NCCCNC(=O)CC2C=CCCC2)C(Cl)(Cl)C12CC2 16754,c1(OC)cncc(NC(C2(O)CCN(C(=O)C(C)(C)N3CCCC3)C2)=O)c1 16755,N1(C(CCC(=O)N(C)C)=O)CCCC12CCN(C(=O)CCC(F)(F)C(F)F)C2 16756,S(=O)(=O)(c1cnn(CCl)c1)N1CCN(CC(=O)NC)C(C)C1 16757,C1(NC(C(C=C)(C)CC)=O)CC2(CCN(C(C3(C#N)CCCC3)=O)CC2)C1 16758,C(CC1=CCN(CC(=O)Nc2ccccc2Cl)CC1)NC(c1c(Cl)cn(C)n1)=O 16759,CC1=C(Br)CN(C(CCC2CC2)C(=O)NCSc2ccccc2Cl)CC1 16760,CN1CCC(C(=O)NCC2(C(=O)Nc3ccccc3O)CCC2)CC1=O 16761,n1(C(C)C)cc(C(=O)NCCNC(c2cc(N)c(Cl)cn2)=O)c(O)nc1=O 16762,c1(CC(=O)NC(C)(C)CCNC(C2CCCC2(C)C)=O)cc(Cl)cc2c1OCC2 16763,CC1CC2(CC(CN(C(c3sc(Br)cc3Cl)C(=O)NCC(F)F)C)C2)C1 16764,C1(NC(c2cc(C(C)(C)C)n[nH]2)=O)COCCC1NC(=O)C(C1CC1)C1CC1 16765,Cc1nc2cccc(C(N3CC(CNC(c4ccc(=N)[nH]c4)=O)CC3C)=O)c2[nH]1 16766,N1(C(c2nc(Br)cs2)=O)CCN(Cc2ccc(Br)c(F)c2)C2CC12 16767,N1(C(c2snnc2C)C(=O)NCCOCC)CCC(CCN(C)C)CC1 16768,c1(C(=O)NCCC2(CNC(COCC=C)=O)CC2)ncn2c1CCC2 16769,C1(CCC(=O)NC2CCCC2NC(=O)C(F)(F)c2cnccn2)CCCCO1 16770,c1(NC(C2CC3N(c4cc(C)nc(C)n4)C(CC3)C2)=O)cccc(Br)c1[N+](=O)[O-] 16771,C1(C(=O)NC2(C3N(C(Cn4c(C)ccc4C)=O)CCC3)CC2)CCC2CCCCN12 16772,C1(N(C(C2C(C)C2)=O)Cc2ccccc2)CCN(C(=O)C(O)CCN(C)C)CC1 16773,N1(C(C(N2CCC(O)CC2)C)=O)CCCCC(NC(c2cncn2C)=O)C1 16774,c1(CC(N2CC(C)C(CNC(C3C4CC5C(C4=O)C35)=O)C2)=O)ccc(F)cc1Cl 16775,N1(c2c(C)cncn2)CCCC2(CN(C(c3[nH]nc([N+](=O)[O-])c3Cl)=O)CCO2)C1 16776,N1(C(C(C)OCCc2ccccc2)=O)CC2CC(C1)N(c1ncnc(O)c1Br)C2 16777,N1(Cc2nnc(C(C)C)o2)CCC2(CCN(C(c3c(F)cccc3Cl)=O)C2)C1 16778,N1(C(CC2(NC(=O)Cc3nncs3)CCC2)=O)CCC(C2CC2)C1 16779,C(=O)(C(CO)C(C)(C)C)NC(C(=O)NCC(C(=O)OC)C)C 16780,N1(C(c2c(CC)oc(C)c2)=O)CCCC(C)(C)C1CNC(=O)COCC(F)F 16781,C=CC(C)(C)CC(=O)NCC1(C)CCC(NC(=O)CCC2CCCO2)CC1 16782,C(CNC(C1(S(C)(=O)=O)CCC1)=O)(C(C)C(C)C)NC(c1nc(CC)oc1)=O 16783,c1(SCC(CN(C)C(c2cc(F)cs2)=O)O)nnc(CCOC(C)(C)C)s1 16784,C1(Nc2c(OCCOC)cc(C(=O)O)cc2)CCc2nnc(C(F)F)n2C1 16785,c1(C(N2CC(C(C)NC(C=C(C)C(C)(C)C)=O)OCC2)=O)cncc(N=[N+]=[N-])c1 16786,C1(NC(C2C(OC)CCC2)=O)CCN(Cc2ncc(C)o2)CC(C)(C)C1 16787,N1(C(=O)C(O)Nc2ccccc2)CC2CN(C(c3c(Br)ccnc3Br)CCOCO)C2C1 16788,C1(C(=O)NC2(CNC(c3c(C)[nH]cc3)=O)CCOCC2)CC12CCOCC2 16789,c1(OC)cc(C(=O)N(CCCNC(=O)COC2CC2)C2CC2)cc(Cl)n1 16790,c1(CC)ccc(C(=O)N(C)CCNC(c2ccccc2CS(C)(=O)=O)=O)cn1 16791,c1(C(c2n(CCCOC)nnn2)NC2CC(CCSC)C2)cc(Br)cc(F)c1O 16792,c1(C(=O)NC2CC(O)CN(C(=O)Cc3ccnc(Cl)c3)C2)cnc2nccn2c1 16793,c1(C(=O)NC2C(C)CN(C(c3ccc[nH]3)=O)C2)ccc2c(c1)C(C)(C)C(=O)N2 16794,C1(NC(C(=Cc2cccs2)C)=O)CC2(CCN(C(=O)Cc3ccsc3Cl)C2)C1 16795,C1(NC(c2cnn[nH]2)=O)CCN(C(c2nnc(O)cc2O)=O)C(C2CC2)C1 16796,C1(C(N(CC(C)C)CCNC(CCOC)=O)=O)CCCCN(C)C1=O 16797,c1(C(N2CCN(C(c3c(SC)ccs3)=O)C(CO)C2)=O)cccn2nncc12 16798,C(CCCCC(=O)NCC(CC)N1CCCC1)N(C(c1cn(CC=C)nc1)=O)C 16799,O=C(C1Cc2ccc(Cl)cc21)N1CCCC2(CCCN2C(=O)C2=CCCCC2)C1 16800,C(=O)(C1=NOC2(CCNC2)C1)N1C(CCNC(CN(C)C(N)=O)=O)CCCC1 16801,C1(C(=O)NCCn2c(CC)ncc2)CC(CC)CCN1C(=O)CCC(CC)OC 16802,N1(C(c2nn(CC)c(C)c2)=O)CC2CN(Cc3ccc(C)cc3C)C2C1 16803,N1(C(C(CC#C)C)=O)CCN(C(=O)C=C(Cl)Cl)C(c2cc(F)ccc2F)C1 16804,C1(CC(NOCCCC)=O)CCN(C(c2ncoc2C2CC2)=O)CC1 16805,C(=O)(CC(F)(F)Cl)NCCOC1CCN(C(C2CC(CC(C)(C)C)C2)=O)C1 16806,CC1CC(CSc2nc(C3CCCCC3(F)F)no2)CC(C)C1 16807,CC(CC(=O)NC1C(C)(C)CN(C(=O)C2=CCCSC2)CC1(C)C)CC(C)(C)C 16808,Cc1ccc(SCC2(C(F)(F)F)CCCCO2)cc1C1CC1 16809,CN1CCOC(C(=O)NCC(C2CCCC2)NC(c2cnc(N(C)C)s2)=O)C1 16810,C#CC1(C(N2CC(CO)C2(C)C)=O)CN(C(=O)COCC2CCOC2)C1 16811,C(=O)(CCC(C(C)C)SC)NC(C(=O)Nc1cn(CCOC)nc1)(C)CO 16812,c1(-c2cn(CC(C)NC(C3(C)C(C)(C(=O)OC)CC3)=O)nn2)c(C)sc(C)c1C 16813,N1(C(CCC(C)OCC)=O)CCN(C(c2ccc(OC)cc2Cl)=O)CCC1C 16814,N1(C(=O)CC2CCC2)CCC(C2CCCN(C(c3cc(Cl)nnc3O)=O)C2)C1 16815,N1(C(c2ccc(CO)nc2)=O)CC2CC(C1)CN(C(=O)C(F)C(F)(F)F)C2 16816,c1(OCC(=O)OC)ccc(OC(=O)COC(=O)C(C(C)C)NC(C)=O)cc1 16817,C=Cc1ccc(C(N2CC(NC(=O)CCc3ccsc3Cl)CC(O)C2)=O)cc1 16818,c1(C(N2CC(O)(C(C)NC(=O)CC3(C(F)F)CC3)C2)=O)cc2n(n1)CC(F)C2 16819,CC1CCN(C(=O)Cn2cncn2)CCN1C(=O)CC1CC2(CC2)CO1 16820,CC(C)(C(=O)NCC1CCN1C(=O)COc1cncnc1)C1=CCS(=O)(=O)CC1 16821,c1(C(=O)NC(CNC(C2C(c3cccc(C)c3)C2)=O)C(C)C)ncc(Cl)cc1F 16822,c1(C(N2C(CC(N3CCC(NC(C)=O)C3)=O)CCC2)=O)nccc(Cl)c1F 16823,C1(NC(C2(NC(C)=O)CCC2)=O)CCN(C(C2CCS(=O)(=O)C2)=O)CC1 16824,N(C1c2ccccc2C2CC12)C(N1CCC12CCOCC2)=O 16825,C(=O)(C1=CS(=O)CCC1)NCCN(C(c1cn(C(F)F)c(C)n1)=O)CC 16826,c1(C(N(CC(CC)NC(=O)Cn2nnc(C)n2)CC)=O)cccc(O)n1 16827,N1(C(c2nccc(C)n2)=O)CC(N(C)C(c2oc(C)cc2C)=O)C2(CC2)C1 16828,c1(OC)cc(NC(=O)C(=O)NC(CC)C(C)O)c(CNC(C)=O)cc1OC 16829,Cc1ccc(N)c(C(N2CCC(C(C)NC(C3C(C)C3C)=O)C2)=O)c1 16830,c1(NC(N2CCN(CCc3cccs3)CC2)=O)cn2ccc(Cl)cc2n1 16831,N1(C(=O)Nc2ccc(OC(F)F)cc2)CCc2cc(C(F)(F)F)ccc2C1 16832,C1(C)(CC)C=C(C(=O)N2CC(C(=O)NC3CN(C(C)C)CC3C)(CC)C2)C1 16833,C1(C(N(CC(C)O)CCNC(C(CC(C)C)N(C)C)=O)=O)CCC2C(C1)C2(F)F 16834,c1(NC(CCC)c2ccco2)cc(C(N2CCCC2CS(C)(=O)=O)=O)ncn1 16835,Cc1cc(C(F)F)ccc1S(=O)(=O)NCC1CCc2cccnc21 16836,N1(C(C(C)C#N)=O)CCCC1(C)CNC(=O)CCNC(C1CCCC1)=O 16837,C1(COC)(NC(=O)CCNC(C)=O)CCN(C(=O)CC2CCNC2=O)C1 16838,C(=O)(C1CCCc2cncn21)N(C)CCNC(c1cccn1-c1cnccn1)=O 16839,c1(C(N2CC(NC(c3cnc(Br)s3)=O)C(F)C2)=O)c(F)cc(C2CC2)cc1F 16840,C1(C(=O)NCc2cnc[nH]2)CC2CC2N1CC(c1ccc(F)cc1)NS(C)(=O)=O 16841,c1(C(C(=O)NCC(F)F)N(C)Cc2nc(CC)sc2)cc2c(s1)CCOC2 16842,C(=O)(C(F)CC(C)(C)NC(=O)OC(C)(C)C)N1C(CC)C(c2ccccc2)CC1 16843,c1(CCC(=O)NC2CN(C(C(COC)O)=O)CC2C(F)F)ccc2c(c1)CCO2 16844,N1(C(C(C)NC(N)=O)=O)CC2CCN(C(c3cnc(-c4cccnc4)s3)=O)C2C1 16845,O(NC(=O)C(C)(C1CC1)N(C)C(c1ccc(C2CC2)o1)=O)CC(C)C#N 16846,c1(COC)nc(N2CC=CC(NC(=O)CC(O)CN(C)C)C2)cc(Cl)n1 16847,N1(C(C(C2CC2)OCC)=O)CCN(C(c2c([N+](=O)[O-])cnn2C)=O)CC(C)(F)C1 16848,CC1CC(O)CCN(C(C2CC(CNC(=O)C(O)CC(F)(F)F)C2)=O)C1 16849,c1(NC(CC2(C)CCN(C(C(CC#C)C3CC3)=O)C2)=O)ccc(O)c(CO)c1 16850,C(=O)(CCCN(C(=O)C1=CCC1)C)NC(C1CCCCC1)C#C 16851,S(=O)(=O)(c1ccc(N2CCC(CC(C)O)CC2)c(C#N)c1)NC(C=C)(C)CC 16852,c1(OCC)ccc(C(N2CC(CO)(NC(c3ccc(F)o3)=O)C2)=O)c(F)c1F 16853,N1(C(c2n(CC)cnn2)=O)CC(NC(c2nc(Cl)cs2)=O)CC(C)C1 16854,C(=O)(CCCCCO)NC12CC(C(N3CCCC3c3ccc(Br)cc3)=O)(C1)C2 16855,C1(N(C)C)CCCN(C(C2CC23CC(NC(c2ccc(Cl)cn2)=O)C3)=O)C1 16856,C(=O)(C(O)C(C)(C)C)N1C(CC(=O)N(C)CC2CC2(C)C)CCC1 16857,CC1CCC(O)C(C2CCCN2CCC2CC23CC3)C1 16858,CC1CCc2nc(C(=O)NC3CCCC3NC(=O)CC3CC=CC3)cn2C1 16859,CC1(C)C(C(N2CCCC(NC(C3CCCC(=O)O3)=O)C2)=O)C1(C)C 16860,c1(CN(c2c(C#N)scc2)C=O)ccc(F)c2c1CCC2 16861,c1(C(=O)NCC(CC)NC(=O)C(c2cn(C)nc2C)C)cncc(NC)c1 16862,c1(C2C(CNC(=O)CCc3cscc3Br)C2)cccc(F)c1 16863,CCC(CCCC(=O)N1CCOCC(F)(F)C1)NC(c1cnn(C)c1N)=O 16864,c1(CC)ccc(OCCC(=O)NC(C)C(C)NC(C2CCCCC2)=O)cc1 16865,c1(C(=O)NCCCCCC(=O)NC2CCCCC2)cccc2occc12 16866,C1(C(N2CC(SC)C2)=O)CCN(C(C2C3CCCC23)=O)C(C)C1 16867,c1(C(N2C(CNC(=O)C(c3ccccc3)O)CCCC2)=O)cc(F)nc(F)c1 16868,c1(CNC(C(Cc2cnn(C)c2O)N)=O)c(Cl)ccnc1Br 16869,C1(C(=O)NCCC=C=C)CN(C(=O)Cc2ccccn2)CCN1C 16870,C(=O)(C(CC(C)C)OC)NC(C(N1C(CC)(CC)CC1)=O)CC1CC1 16871,c1(-c2nc(C(c3ccc(Cl)cc3)CC)n(CC)n2)ccc(F)c(C)c1 16872,C1(OC)CN2CCCC2(C(=O)NCC2CCCN2C(C2CC23CC3)=O)C1 16873,c1(C(=O)NC2CCC(N(C)C(c3ccc(Cl)s3)=O)C2)cc2ccc(F)cc2o1 16874,Cc1[nH]nc2c(C(N3CC4(CNC(c5conc5C)=O)CCC3C4)=O)cccc12 16875,c1(-c2occ(CNC(c3nn(C)nc3Br)C)n2)cc(F)cc(F)c1 16876,n1(CC(=O)NC(C2CCCC2)CNC(=O)C2=CCC2)nc2n(c1=O)CCCCC2 16877,C(C)(C(C)(C)C(=O)NC1COC(C(C)C)C1)NC(c1cccc(CC)n1)=O 16878,N1(C(CCC=CCC=C)=O)CC2CC(C)N(Cc3ncc[nH]c3=O)C2C1 16879,c1(OC)ccccc1C(=O)NCC(CNC(=O)Cc1sc(C)nc1C)OC 16880,C#CC1(OCC(=O)NCC(=O)NCCc2noc(CC)n2)COC1 16881,n1(C2CN(C(=O)OCC)C2)cc(C(ONC(=O)OC2CC(OC)C2)C)nn1 16882,CCC(C)CCC(=O)N1CC(C(=O)NCC(=O)OC(C)C)CC1(C)C 16883,N1(C(C(N2CCC(NC(c3c(C)con3)=O)C2)=O)C)CCCCCC1 16884,N1(C(C)=O)CCC2(CC1)CN(C(C1NC(=O)CC1c1cccc(Cl)c1)=O)CCO2 16885,C#CCC(CC(F)F)C(=O)NC(C)CCNC(=O)C=CCN(CC)CC 16886,c1(NCC2(C)CCN(C(=O)CC3(C)CC3(Cl)Cl)C2)cc(O)nc(O)n1 16887,c1(OC)cccnc1C(N1CCC(O)(CCNC(=O)C(F)(F)C2CC2)C1)=O 16888,C(=O)(C(C)C(O)CC(C)C)N1C2(C(=O)NCC)CC(C1)C2 16889,C1(CC(=O)NCC(C)N(C(C(=O)N(CC)CC)=O)CC)CC=CCC1 16890,c1(CCCC(=O)OC2COCCC2=O)ccc2nc(O)[nH]c2c1 16891,C1(C(=O)NCC2CN(C(C(C)(C)c3nccs3)=O)C2)CCCC2C1C2(F)F 16892,C(=O)(CCC(=O)N1CCN(C2CCC2)CC1)NCC(CC)CC 16893,N1(C(c2c(C)nn[nH]2)=O)CCC(C(=O)NC2C(O)CC2O)=C(F)C1 16894,c1(C(N(CC(C)CNC(C2CC3CC3C2)=O)C)=O)cccc(SCC(F)(F)F)c1 16895,C=CCC(C)(C)CC(C(=O)NCC1CC1)N1CCC(n2ccnc2)CC1 16896,c1(C(C(=O)N(CCOCCNC(C(CCC)C#N)=O)C)O)cccc2c1OCC2 16897,c1(C(N2CC(CN(C(CN(C3CC3)CC)=O)C)C2)=O)cnn(C(C)C)n1 16898,CC1(C)CCC(C)(C(=O)NC2CC(O)CN(C(=O)Cn3cnccc3=O)C2)CC1 16899,C1(C)(OCC(=O)NC(C2CCN(C(=O)CC3CCOC3)C2)C)CCOCC1 16900,C1(OC)CCCC(C(=O)NC2CC2CNC(=O)C(C)=C2CCC2)C1 16901,N1(C(c2c(CC)nco2)=O)CCCC(CNC(=O)CCC2CC(OC)C2)C1 16902,C1(NC(CC2CCCC(C)(C)C2)=O)CCC2(CCN(C(=O)C=C3CCC3)CC2)C1 16903,C1(OC)CN2CCCC2(C(=O)NCC(C(C)C)NC(=O)Cc2nc(C)sc2C)C1 16904,C12(C(=O)NC(CC)CN(C)C(C3CC(C)(C)C3)=O)CC1COC2(C)C 16905,C1(CNC(CCn2c(C(C)C)ncc2)=O)CC2CCCCC2N1C(=O)CC(C)O 16906,C1(F)(C(N2CCN(C3CN(C(C4C(C)C4C)=O)C3)CC2)=O)CC2(CCC2)C1 16907,C1(CNc2nc(C)nc(Cl)c2)CCC2(CCC2)C1NC(c1cc(O)nc(O)n1)=O 16908,c1(OC)ccc(C#N)c(Cl)c1.c12noc(C)c1C(=O)O2 16909,c1(OC)cccc(C2=NOC(C(=O)NC3CCCC(C4CC4)C3)C2)c1 16910,c1(NC(CCN(C(CCCOCC)=O)C)C(C)C)ncc(C)c(S(C)(=O)=O)n1 16911,C(=O)(NNc1cc(Br)ccn1)Nc1c(C)cc(C(=O)NCC2CC2)cc1 16912,C1(C(=O)NC2(CCNC(=O)C(=O)N(C)C)CC2)(CSC)CCC1 16913,CC1(CNC(=O)CCOC2CCCOC2)CCN(C(C2(C)CC=CCC2)=O)C1 16914,CC(O)CC(C)(C)CNC(c1cc(C2CC2)on1)c1nnnn1CCCF 16915,CC(C(=O)NCC1CCC(NC(C2CC(F)(CF)C2)=O)CC1)C(F)F 16916,N1(C(C(C(C)C)SC)=O)CC2CCCC(NC(c3cn(C)c(O)n3)=O)(C2)C1 16917,C(=O)(CC=C(Cl)Cl)N(C1CCN(C(=O)C(=Cc2ccccc2)NC(C)=O)C1)CC 16918,c1(C(=O)NCCN(C(CC2CCCC(C)C2)=O)C)c([N+](=O)[O-])cnn1C 16919,C12(NC(c3c(C)cn(C)c3)=O)CCOCC1CN(C(c1ccc(Cl)c(N)c1)=O)C2 16920,N1(C(CN(CC(C)(C)C)C)=O)CCN(C(C2CC3C=CC2O3)=O)C(C2CC2)C1 16921,N1(C(c2ccn(C)n2)=O)CCC2(NC(c3cnnn3C)=O)CCCCCC12 16922,Cc1cc(C(N2CCCC(CC(N3CC(CO)CC3CO)=O)CC2)=O)nc(O)c1 16923,C1(CNC(=O)CCc2cncnc2)CC(F)CN1C(C1OCCCO1)=O 16924,c1(OC(c2n(CCOC)ncc2C)=O)ccc2c(c1)OC(C)(C)CC2=O 16925,c1(CC)onc(C)c1CNC(=O)CCN(CCO)C(C12CCCCC1C2)=O 16926,C1(OC(C)(C)C)CC(NC(c2sc(Br)cc2I)=O)C1(C)C 16927,N1(C(c2sc(CC)c(C)c2)=O)CCCC(C2(NC(c3cnsn3)=O)CC2)C1 16928,C(CC(C)CCNC(=O)C(N)=O)NC(C1CN(C(=O)NC)C1)=O 16929,c1(SC)ccc(NC(=O)CN(CCCNCC(C)C)CCCO)cc1 16930,C(=O)(C1=NN2CCCN=C2N1)N1CCN(C(C=CC)=O)CC1CC(F)(F)F 16931,c1(C(N(CC(C)N(C(C2C(OCC)C2)=O)C)C)=O)cc(=O)n(-c2ccccc2)[nH]1 16932,c1(C(=O)OC)ccccc1-c1cn(C2CC(C(=O)NC3CCN(C)C3C)C2)nn1 16933,C(=O)(C(F)CCC(C)C)NC(C(C(=O)NCC1CC(CC)C1)(C)C)C 16934,C1(NC(C(CCC)(C)C)=O)CCC2CC1CN2C(c1ccc(F)cc1OC)=O 16935,c1(OCCCC)cc(CNC2COC(C)(C)C2O)ccc1OC 16936,c1(C(=O)NCCCN(C(CC2ON=C(C)C2)=O)CCO)cccc(C)c1O 16937,O=C(CC(C(F)F)n1ccnc1)NCCCNC(=O)C=Cc1cccnc1Cl 16938,c1(CC)cc(C(=O)NC(C)(C)CNC(=O)C=CCO)ccc1Cl 16939,c1(C(=O)NCC2C(NC(c3c(CC)nccc3)=O)C2)cc2nc[nH]c2cn1 16940,c1(C(=O)NC2CCN(C(CC(COC)C)=O)CC2F)nc2ccccn2c1F 16941,CS(=O)(=O)c1ccc(Cl)cc1NC(=O)C(=O)NCC(F)C1CCC1 16942,C1(NC(CC2(C)CCCO2)=O)CCC2CN(C(C3CC4CCC3C4)=O)CC2C1 16943,C1(C)(C(N(C2(C(=O)NCC(C(C)O)O)CCC2)C2CC2)=O)CCN(C)CC1 16944,C(=O)(C1CCCc2nc[nH]c21)N(C(C)CNC(C1(CN(C)C)CC1)=O)CC 16945,C1(C(=O)NCCC2COCCN2C(C2CCSCC2)=O)Cc2ccccc2O1 16946,Cc1c(C(=O)N(C2CCN(C(C34CC(C(C)C)(CO3)C4)=O)C2)C)cccc1Cl 16947,N1(C(c2n(CC)nc(C3CC3)c2)=O)CC2CCC(Nc3ncncc3I)CC2C1 16948,c1(C(=O)NC(CC)CN(C(=O)CCOCC(C)C)C)cc(C)nn1C1CCC1 16949,c1(C(=O)NC2C(NC(C3C(OC)C3)=O)CCC2)c(C)cc[nH]c1=N 16950,c1(C(N2CCC(C(CNC(C(C)SC)=O)C)CC2)=O)ncc(Cl)cc1F 16951,C1(C(=O)NC(CCSC)C)(SC)CN(C(=O)CC(C)C2CCCO2)C1 16952,c1(C(=O)NC2C(N(C(CC(C)C3CC3)=O)C)CCCC2)ncc2cc(Cl)ccn12 16953,N#Cc1ccc(O)c(NC(C2CC23CCN(Cc2c(F)cc(F)cc2F)C3)=O)c1 16954,C(=O)(C#CC(C)(C)CNC(=O)Cc1cn(C)cn1)NC(C(=O)OC)CCF 16955,c1(C(N2CC(NC(C3CC(OC)C3)=O)C2)=O)cnoc1C1CC1 16956,C(=O)(C(C)(C)C(C)NC(=O)OC(C)(C)C)N(CCOCC)CC 16957,c1(C(=O)NC2C(NC(CC3N(C(C)C)CCC3)=O)C2)ccccc1Cl 16958,N1(C(c2cc(OC)cc(C)c2)=O)CCn2cccc2C12CCNC2 16959,C(N=c1[nH]c(-c2ccoc2)ccc1OC)c1scc(-c2c(OC)cccc2)c1 16960,C1(CN(C)C(c2csc(O)n2)=O)COCCN1C(c1cc(C2CCCC2)[nH]n1)=O 16961,N1(CCOC)C(=O)CCC1C(=O)NCC1(NC(c2ccn(C(F)F)n2)=O)CCC1 16962,C1(NC(=O)Cc2ccc(Cl)cc2Cl)CC2CC(C1)N(C(=O)C(O)C1CC1)C2 16963,c1(C(=O)NCC2N(C(C(COC)C)=O)C3CCC2C3)cc2c(F)cc(Cl)cc2[nH]1 16964,C1(CNC(C2C(C)CC(=O)N2)=O)CCN(C(c2cc3sccc3s2)=O)CC1C 16965,c1(-n2cc(CNC(c3cc(Cl)cnc3Br)=O)nn2)ccc(F)c([N+](=O)[O-])c1 16966,C#CCCCCCC(=O)NCCCCC(C)(C)NC(C1CC12CC2)=O 16967,c1(NC)ccc(F)cc1C(N1CC(C(F)(F)F)OCC1CNC(=O)C(C)(C)C)=O 16968,c1(C(N(C)CC2CCCC(NC(CN(C(C)C)C)=O)C2)=O)ccc(CO)c(F)c1 16969,N1(C(c2c(C)[nH]nc2CO)=O)CC2(C1)CN(C(C1COCCN1C=O)=O)C2 16970,c1(C(N2CCN(C(=O)CCc3cnc(O)[nH]3)C3CC23)=O)cccc2oc(O)nc12 16971,C1(CC(=O)NCCN(C(c2n[nH]cc2Cl)=O)CC)CCC2(CCOCC2)CO1 16972,c1(OC)ccc(NCC(C)=CC(=O)NCCNC(C23CCCC2C3)=O)cc1 16973,C1(C(=O)NC2CC3CNCC23)CC2(CCCCC2)CN1 16974,c1(N2C(C)CCC(NC(=O)CCOCC3CCCO3)C2)ncc2c(n1)CCOC2 16975,c1(C(N2C(C)CC(CNC(c3ccsn3)=O)C2)=O)sc2nccnc2c1N 16976,CC(C)(C)C(C)(C)C(=O)N1CCOC(C(N2CCC(O)C23CCC3)=O)CC1 16977,N1(C(Cc2cn(CC)nn2)=O)CC(C)CCC1CNC(c1[nH]cnc1C#N)=O 16978,C1(N(C(c2cc(C)c(O)cc2)=O)C)CC2CCC(C1)N2C(=O)CCc1cnn[nH]1 16979,C(CC1CC1)(C(=O)NC1COCC1NC(=O)C=CSC)OC 16980,c1(C(=O)NC2CC(C)N(C(=O)CC#N)C2)cc2c(Br)cccc2c(=O)o1 16981,c1(NC(C(C)(C2CCC2)NC(=O)C(C2CCOCC2)F)=O)ccc(F)cc1 16982,C1(NC(=O)C=CC2CC2)CCC1C(=O)NCC(c1cnc[nH]1)O 16983,c1(OC(C)C(=O)NCC2COCCN2C(c2cccc(F)n2)=O)cccc(F)c1 16984,Cc1ccc(S(=O)(=O)N(C2CCNC2=O)C2(C(N)=O)CC2)cc1[N+](=O)[O-] 16985,c1(CCC(=O)NC)ccc(OC(C2CC2)(CC)OC)cc1.C1COC1.C1CO1.C1CC1 16986,C1(CNC(c2ccc(F)cn2)=O)CCCC2(CN(C(=O)CCC(F)(F)F)C2)O1 16987,C1(C(=O)NC(C2CN(C(CC3CC(C)C3)=O)C2)C)NC(=O)OC1C 16988,C(=O)(CC(C)CC(C)(C)C)NC1C(CC(=O)N(C(CCC(C)C)C)C)CCC1 16989,C(=O)(C(CCC1CCC1)NC(=O)NCCc1cnsc1)OC 16990,Cc1ncccc1CC(N1CCC(NC(=O)CN(CC(C)(C)C)C)CC1)=O 16991,c1(C(C)NC(C(C2CCC(C)C2)N(C2CCCC2)C)=O)ccc(F)cc1 16992,C1(C)(NC(COC(CNC(CC2CC(=C)C2)=O)(C)C)=O)CCOCC1 16993,C12(C(=O)OC)CCCC1(C(=O)NCC=CCNC(=O)COc1ccsn1)C2 16994,C12(C(N3CC(CNC(C4CC(CF)C4)=O)C3)=O)CC1CNC2=O 16995,Cc1coc(C2CN(C(=O)Oc3cn(C(=O)OC(C)(C)C)nn3)C2)c1C(C)(C)C 16996,c1(C(N2C(CNC(CS(C)(=O)=O)=O)CCCC2)=O)c(Cl)ccc(F)c1F 16997,C1(CCNC(CSCC(C)C)=O)CC(NC(c2ccsc2)=O)C1 16998,c1(CNC(c2nnc(CF)o2)CC)cn(-c2ccccc2)nc1-c1ccccc1 16999,C1(NC(COCCN(C)C)=O)CCCC12CCN(C(c1ccc([N+](=O)[O-])o1)=O)C2 17000,C1(NC(c2ccccc2SCC)c2n(CCCC)nnn2)(CC)CCOCC1 17001,C1(OC)CN(C(c2ccc(C3CC3)o2)=O)C(C)(CNC(c2cnn[nH]2)=O)C1 17002,CC(C)C(N=[N+]=[N-])C(=O)NCc1nocc1C(=O)NCC1(CC2CC2)CC1 17003,C(=O)(C#CC1(C)COC1)NCC1(O)CCCN(C(CC(C=C)CC)=O)C1 17004,c1(CC(N2C(C(C)(C)NC(=O)CC3CCS(=O)(=O)C3)CCC2)=O)cncc(C#N)c1 17005,C1(CNC(CSC)=O)CN(C(c2cc(C(C)(C)C)n(C)n2)=O)CC1C 17006,CCCC(O)CC(=O)NCC(CNC(c1ccc(CCC(C)C)cc1)=O)CO 17007,Cc1nc(=N)[nH]cc1C(N1CCOCC(CNC(=O)Cc2ccc(F)cc2)C1)=O 17008,C#CCC(CC(=O)NOCCC(F)(F)F)NC(=O)C=Cc1nc(C)cs1 17009,N1(C(=O)C=Cc2ccsc2)CC2CN(c3ncncc3F)CC2C1 17010,c1(OC)cccc(C)c1NC(=O)CCCCCNC(=O)CC1NC(=O)NC1=O 17011,N1(C(CCCn2ncc(C)c2)=O)CCN(C(c2cc(C)ccc2O)=O)C2CCC12 17012,N1(C(c2c(C)ocn2)=O)CCC2(CC1)COC(CNC(C1(O)CCSC1)=O)C2 17013,c1(OCC(N2CCC(C(C)(C)NC(CC(C)C)=O)C2)=O)cncc(Br)c1 17014,CC1N(C(C2(C)CCN(C(C3CC(C)(C)CO3)=O)CC2)=O)CCC1(C)C 17015,N1(C(c2ccncc2Cl)=O)CCN(C(C2CCCC2F)=O)C2CC12 17016,C1(CC(=O)N(C2CC(C#N)C2)CC(=O)NCC(C)CO)CCCC(O)C1 17017,N1(C(c2cccc(CC)c2)=O)CC(C)CCC1C(N1CCCC(CCO)CC1)=O 17018,C1(=O)CCCSCC(=O)N1CCOCCO.C(C)(C)(CC)OCC(=O)NCC(C)=O 17019,C12(C(N(CCCNC(CCC=C(C)C)=O)C)=O)CC3CC1C2C3(F)F 17020,N1(C(C(=O)Nc2c(OC)ncc(Br)c2)=O)CCC2OCCCC2C1 17021,c1(C(N(C(C)CNC(c2n[nH]c(=N)[nH]2)=O)C)=O)cncc2ccccc12 17022,c1(OC)cc(C(=O)NCCN(C)C(C2(C)CC=CC2)=O)on1 17023,C1(CC)CCN(C(C2CC(NC(C34CCC(CC3F)C4)=O)C2)=O)CCO1 17024,N1(C(Cn2c(C)ncc2)=O)CCC(NC(C23CC2CNC3=O)=O)CC1C 17025,c1(OC)cc(C)c(C(=O)NCC2CC(O)CN2C(=O)CCC(N)=O)cc1Br 17026,c1(C(N2CC(O)(CC#N)C2)=O)nc2nc(C(F)(F)F)ccn2n1 17027,C(=O)(C(C)(C)C(=O)NCC1(F)CCCN(C(=O)CC2CC(C)(C)CCO2)C1)NC 17028,c1(C(N2C(C)CC(CNC(c3cncc(F)c3)=O)CC2)=O)nn(C)c2c1CCC2 17029,C1(C(=O)NCCC(O)CNC(c2cnccc2C)=O)(COC)CCCCC1 17030,N1(C(c2cc(CCC)oc2C)=O)CCN(C)CC1CNC(=O)CCC(C)O 17031,C(c1ccc(Cl)c(Cl)c1)=CC(N1CC2C(NC(=O)CC3CCCC3(F)F)(C2)C1)=O 17032,C1(C(=O)NCCCOCCCNC(c2c(C)cco2)=O)CC(C)CCO1 17033,C=CC(C)CC(=O)NCCn1cc(CNC(c2cncs2)=O)nn1 17034,C1(C(=O)NC2CC(CCNC(c3cccc(C(F)F)c3)=O)C2)CC2CCCC2C1 17035,c1(C(N2C(C)CN(C(C=C(C)Cl)=O)C(C)C2)=O)cc(Cl)cc2c1NCCC2 17036,N1(C(CCC#CC)=O)CCCC(C(=O)NCC2CCCCS2)C1C 17037,N1(CC)CC(N=c2nc3scnc3c(NC(c3nn[nH]n3)C)[nH]2)C1 17038,CC(O)C(C(=O)NCCCC(C)NC(C12CC(C(=O)NC(C)(C)C)(C1)C2)=O)N(C)C 17039,CC(C(=O)NC(C)(C)C(C)NC(c1sccc1Br)=O)C(=O)N1CCOCC1 17040,c1(C(=O)NCC(C)C(=O)NC2CC2)cc(=O)n(C)cn1 17041,c1(C(=O)NC(CNC(CCC(=C)C)=O)(C)CC)cc(S(C)(=O)=O)ccc1Cl 17042,C1(CC)CCCC(C(=O)OC)C1.N12CCC1C(=O)N1CC(C1)C2=O 17043,C(=O)(C(C(C)(C)C)NC(=O)CCc1ccc(C)nc1)NCc1cn(CC=C)nn1 17044,C(=O)(C(C)CC(C)(C)C)N1CCC(Cn2cc(C3C(C)OCC3)nn2)C1 17045,N1(C(C(CC)CC)=O)CCN(C(=O)CSc2ccncc2)C(CO)C1 17046,C1(CNC(COC(CNC(C2(C(=O)OC)CC2)=O)(C)C)=O)CCCSC1 17047,C(=O)(C(O)CC(F)F)N(CCN(C(CCn1c(C)csc1=O)=O)C)C 17048,N1(C(C(CCC)F)=O)CCN(C(c2cc(Cl)nn2C)=O)C(CCO)C1 17049,c1(C(=O)NC2(C)CN(C(=O)CCN3CCOCC3)C2)ccnc(C(C)(C)O)c1 17050,C1(N)(C(=O)NCC(c2cccc(OC)c2)N)CC2CCC1CC2 17051,c1(N2CC(CCCCNC(C3(C)C(CC)CCC3)=O)C2)ccc(C#N)nn1 17052,c1(C(=O)NCCC(CCNC(C2CC(=C)C2)=O)C)cc(Br)ccc1OC(C)C 17053,N1(C(c2cc(CC)no2)=O)CCN(C(=O)CCC2CCCC2)CC1c1cn[nH]c1 17054,c1(-c2cn(CC3N(C(c4ccc(C(=O)O)nc4)=O)CC3)nn2)c(F)cccc1Cl 17055,c1(CCCNC(=NC)NCC2COC(=O)N2)cc(Cl)ccc1Cl 17056,C#CCC(O)C(=O)NCC1(CNC(c2cnn(CCO)c2C(C)C)=O)CC1 17057,Cn1nc2c(c1C(N1CCC(NC(C3CCCOCC3)=O)C(F)C1)=O)COCC2 17058,C1(NC(c2c(OC)cc(C)cn2)=O)CCC2(CCN(C(=O)CC3(SC)CC3)C2)C1 17059,S(=O)(=O)(c1cnc(NC2CC3CCCC3C2)c(Cl)c1)NC(CCCC)CC 17060,C1(C(=O)NCC(C)NC(=O)C(C)(C)n2cc(Cl)cn2)(OC)CCCCC1 17061,N1(C(Cc2c(C)nc[nH]2)=O)CC2CC(O)C1C2NC(=O)C(C(C)C)C(C)C 17062,C(=O)(N=c1cc(Cl)nc(C)[nH]1)c1c(CC)nc(-c2ccc(C)o2)cc1 17063,N1(C(c2c(O)nc(CC)c(C)c2)=O)CCC2(CCCN(c3nnnn3C)C2)C1 17064,C1(CC(=O)NCC(C)COC)(NC(COCCCC#C)=O)CCCC1 17065,c1(N2CC(CC)N(C(C3C=C3C)=O)CC2)ncc2c(ccn2CC)n1 17066,N1(C(CCN(C)CCO)=O)CC(CC(=O)N(C2CC2C2CC2)C)C2(CC2)C1 17067,C1(NC(C2CCC2(F)F)=O)CC2CC1CN(C(c1cccn3nccc13)=O)C2 17068,Cc1nc(NC2CCCN(C(=O)Cn3nnnc3C(C)C)C2)cc(Cl)n1 17069,c1(C(=O)NCC(CCOC)NC(c2c[nH]c(C#N)c2)=O)ccc2c(c1)COC2 17070,c1(CN2CC(CNC(c3cc(C)c(C)s3)=O)C2)ccc(F)cc1F 17071,C(=O)(C1=C(Cl)CCCC1)NC1C(C)CCN(C(C2CCC2(C)C)=O)C1 17072,CC(C)C(CCc1ccccc1)C(=O)N1CC2(CCCC2NC(=O)C=CCO)C1 17073,c1(N(c2cc(SC)ncn2)CC2(O)CNC2)ncnc2ncn(C)c12 17074,C(=O)(CC(F)(F)F)NC(C(=O)N1CC(CC(C)NC(c2c(OC)c[nH]n2)=O)C1)C 17075,CC1=C(C(=O)N2CCC(F)C(NC(c3cnc(C)[nH]c3=N)=O)C2)S(=O)(=O)CCO1 17076,N1(C(C2C(CC)CCC2)=O)CCN(C(C)CNC(=O)Cn2cccn2)CC1 17077,C1(CC)CCN(C(C2CC(=O)N(C)C2)=O)C(C(=O)NCc2ccc(OC)cn2)C1 17078,Cc1cc(F)ccc1NC(=O)C(c1cn(C)nc1I)N1CC2CC1CO2 17079,C=CCC(CC(=O)NC(c1nc[nH]n1)C1CC1)NC(C1CC2CC2C1)=O 17080,c1(C(=O)NCC(C)N(C(C(CC)F)=O)CC)cncc(OC(F)F)c1 17081,Cn1cnc(C=CC(=O)NCCCC2CCCN2C(=O)CCCc2cc[nH]n2)c1 17082,N1(C(c2ccc(C)c(C#N)c2)=O)CC2(CCN(C(c3ccc(Cl)nc3)=O)CC2)C1 17083,Cc1ccc(O)cc1NC(c1csc(C(=O)NC(c2c(C)n[nH]c2C)C)n1)=O 17084,c1(C(=O)NCCN(C(C2(CC)CCNC2=O)=O)C2CC2)nccc2ccncc12 17085,N1(C(c2scc(CC)c2)C(=O)NCC2CCCO2)CCN(C)C(=O)C1C 17086,c1(C(N2CC(CNC(CN(C(COC)=O)C)=O)C(OC)C2)=O)ncc(F)cc1F 17087,C1(CNC(C(C2CCOCC2)C)=O)CCN(C(C2CC3(CCC3)C2)=O)CC1O 17088,C(=O)(CC(CN(C)C)CC(C)C)NC(C1(O)CN(c2cc(OCC)ncn2)C1)C 17089,C1(NC(C#C)CC2CCOC2)CCNCC12CCC2 17090,C1(CNC(=O)Cc2cccs2)CCC1C(N1CCC1C(N)=O)=O 17091,C1(COC)CN(C(=O)Cc2ccnc(O)c2)CCN1C(=O)CC1C=CCC1 17092,c1(C(N2CCCC(NC(C3C(C)C3)=O)C2)=O)cc(S(N)(=O)=O)cc(Cl)c1Cl 17093,C1(C(N2CCC(OC3CC3)C2)=O)COCCN(C(C2(O)CCCCCC2)=O)C1 17094,N1(C(C(C)CN(C)C(C2(CO)CCCC2)=O)=O)CCC(N=[N+]=[N-])C1 17095,C(=O)(CCN(C1CCCC1)CCC)NCC(=O)N(CC#CC)CC#C 17096,c1(CC(N2CCC(COC)(NC(=O)CCC(C)SC)C2)=O)ccc(C)c(F)c1F 17097,c1(Cn2cc(C3(C)N(C(c4[nH]c(=NC)sc4)=O)CCC3)nn2)ccc(F)cc1Cl 17098,CC(C)(C)CC(C(=O)NCc1cccnn1)NC(=O)CCCC#N 17099,CCCC(C(=O)NC(c1nc[nH]n1)C)NC(=O)C(CCC)NC(N)=O 17100,Cc1oc2ccccc2c1C(N1CCCC(CCNC(C2CCCOC2)=O)C1)=O 17101,N1(C(C(n2ccnn2)C)=O)CCC(C)(C)C1C(=O)N(CCCCCO)C 17102,c1(OC)ccc(NC(=O)C=C2CCN(C(c3ccc(Br)c(C#N)c3)=O)CC2)c(C)c1C 17103,c1(NC(=O)CC2(NC(=O)C(F)CC3CCCC3)CC2)ccc(F)c(CO)c1 17104,C(c1cccc(F)c1F)=CC(=O)N(C(C)CN(C)C(C1COCC(C)(C)O1)=O)C 17105,c1(C(CC)CNCc2cn(C3CC3)nn2)ccc(Cl)cc1 17106,N1(CC(=O)N(CCC(C)NC(=O)CSc2ccccc2F)C)CCS(=O)CC1 17107,C1(CC(=O)NC(C2CN(C(c3nc(COC)sc3)=O)C2)C)CCCCC1C 17108,c1(CN(CC(=O)NCC2C=CCN2C(=O)CCc2cnoc2)C)ccccc1Cl 17109,c1(CNC(C(C)NC(C23CC(CCO2)C3)=O)=O)ccc(O)cc1F 17110,CCCCCCC(C)C(=O)N1CCC(O)(CCNC(c2csc3nccn23)=O)C1 17111,c1(NCCc2c(C)ncs2)cc(N(C)Cc2cccc(F)c2)ncn1 17112,c12cccc(c1)CCNC2=O.C=CC1(C(=O)N(CCCSCC)CCO)CC1 17113,N1(C(C(N2CC(C)C2)C)=O)CC=C(CC(=O)NCC(C)C(C)(C)CN(C)C)CC1 17114,C1(CNC(C2CN(C)C(=O)C2)=O)CN(C(c2cnn(C3CC3)c2)=O)CCCO1 17115,c1(C(=O)NCC(C)(CO)NC(CCCCCC=C)=O)ccc2oc(O)nc2n1 17116,N1(C(C(C)CC(F)(F)F)=O)CC(CNC(=O)CS(C)(=O)=O)CC12CCOCC2 17117,CC1(C)CC(NC(C2CCCN2CC(F)(F)F)=O)CN1C(c1cncs1)=O 17118,C1(C(=O)NCc2nc(C)on2)CCC=CC1NC(c1csnn1)=O 17119,C=C(C)CCCC(=O)NCCC(O)C(=O)N(CCCN(C)C)CCC 17120,Cc1ccc(C(F)(F)C(=O)NC2CCC(NC(C3CCNC3=O)=O)C2)cc1 17121,c1(CNC(=O)NCC)cccnc1NC1CC(NC(c2n[nH]c(=N)[nH]2)=O)C1(C)C 17122,CC(CCS(=O)(=O)c1ccc(Cl)cc1)NC(c1cc(O)nc2c1CCCC2)=O 17123,CC1CN(c2nnco2)CC1NC(=O)Cc1cccc(C(N)=O)c1 17124,c1(-c2nc(N3CCCC(CC(=O)NC)C3)n(C)n2)ccc(Cl)c(Cl)c1 17125,c1(SCC(=O)NCC2N(C(C(C)C(C)(C)C)=O)CC2)nn(C)c(=O)n(C)c1=O 17126,C#Cc1ccc(C(=O)N(C(CNC(c2cnn(C(C)C)n2)=O)CC)C)c(C)c1 17127,C1(NC(=O)CCC2CC2(F)F)CCN(C(C2(n3ccnn3)CC2)=O)CCC1(F)F 17128,CC1CCN(C(=O)CNC(C2CCC2(F)F)=O)C1CO 17129,C1(CNC(CS(CC)=O)=O)CCC2(CN(C(=O)Cc3ncc(C)o3)C2)O1 17130,C1(SC)CCc2cc(N)ccc2O1.CCC1Cc2ccccc2OC(=O)OC1=O 17131,Cc1sc(C(=O)NC2CC(CNC(C3CC4CCC4C3)=O)C2)cc1[N+](=O)[O-] 17132,C1(NC(CC(C)(C)N(C(CCCC=C)=O)C)=O)CCOC12CCOC2 17133,c1(N2C(N(C(C(CC)Oc3ccccc3F)=O)C)CCC2)cc(O)nc(C)n1 17134,C1(C(=O)OC)COCC2(CCN(C(C34CC(Br)C3C4)=O)C2)O1 17135,c1(C(=O)NCCC(C)(C)NC(c2cc(C3CC3)ccn2)=O)cc(Cl)cnc1O 17136,c1(OC)cccc(Cl)c1C(N1CC(NC(C2CC23CCC3)=O)CC(F)C1)=O 17137,c1(OC)nc(N2CCC(F)(C(=O)Nc3cccc(-c4nnco4)c3)C2)ncc1Br 17138,C1(NC(C2(C(=O)OCC)CC2)=O)CN(C(=O)C(C)(OC)OC)CCC1CO 17139,CCC(C(=O)N1CCC(CN(C)C(C2(CN(C)C)CCCCC2)=O)C1)C(C)(F)F 17140,CC1CC(NC(c2cc(CO)on2)=O)CN1C(c1cnc(-c2ccccc2)s1)=O 17141,CC(C)(C)C(CNC(=O)CC(=O)C(C)(C)C)C(=O)NCC(C)(O)CO 17142,C1(NC(=O)Cn2cc(Cl)cn2)CN(C(C2CC(CF)C2)=O)CC2(CC2)C1 17143,N1(C(C(Cc2cn[nH]c2)NC(C(C(C)C)=O)=O)=O)CCCC(C)C1CO 17144,C(c1c(C)noc1C)=CC(N1C(C)(CNC(C=C(C)c2cccs2)=O)CCC1)=O 17145,c1(NCC)cc(N2CCC(CF)(OC(=O)CC(=O)N(C)C)C2)ccc1[N+](=O)[O-] 17146,CCCCCC(O)CC(=O)N1CCN(C)C(CNC(=O)C(c2cnn(C)c2)C)C1 17147,CC(C)CC(C(=O)NCC(C)(CO)NC(c1csc(Br)n1)=O)N(C)C 17148,c1(C(N2CC(NC(C(C)=C(C)C)=O)C3(C2)CC3)=O)nc2cccnn2c1Br 17149,N1(C2CCC(NC(CNS(CC)(=O)=O)=O)C2)CCN(C(=O)C(COC)COC)CC1 17150,c1(C(=O)NCC2CCCC(NC(C(CSC)C)=O)C2)c(C)ccc(N)c1C 17151,C1(COC)CN(C(c2cc(NC(C(COC)N(C)C)=O)ccn2)=O)CC1(C)C 17152,C1(NC(c2ccc(Cl)nc2)=O)CN(C(C2CC(C3CC3)=NO2)=O)C2CCCC12 17153,C1(F)(CNC(COCCC)=O)CC(NC(c2occc2C(C)C)=O)C1 17154,C(=O)(CC(CC)CC)NC(CSCC)C(=O)N(C)Cc1cnnn1C 17155,CCC(CC)CC(F)C(=O)NC1(C(N2CCOCC2CO)=O)CC1C 17156,c1(C(N2C(C(=O)NC(c3cn[nH]c3)C3CC3)C=CC2)=O)ccncc1F 17157,C1(NC(c2cn(CC(C)(C)CNC(C3CCSCC3)=O)nn2)=O)CC(F)C(=O)N1 17158,N1(C2CN(C(C(C)OC)=O)C2)CCC(NC(c2sccc2-n2cnnn2)=O)CC1 17159,c1(NC(=O)NC2C(C)COCC2)c(Cl)cc(Cl)cc1Cl 17160,C#CCCCCCCC(=O)NCc1ccc(C(=O)NC2(C3CC3)CCOC2)n1C 17161,N1(C(CN(C2CCSC2)C)=O)CC2CCCC(NC(=O)C=C(Cl)Cl)(C2)C1 17162,c1(C(N(CC(CN(C(=O)CCC(N)=O)C)O)C)=O)cccc2occc12 17163,c1(C(=O)NC(C)(C)CNC(=O)CC2CCOCC2)coc(S(N)(=O)=O)c1 17164,C1(NC(=O)C2=CCSC2)CC2CC1CN(C(=O)CCOC1CCCOC1)C2 17165,C(=O)(C(F)C(F)(F)C(F)(F)F)NC1CCC(NC(C2OCC(C)(C)C2)=O)CC1 17166,C(c1cn(CC(=O)Nc2ccccc2)cn1)=CC(=O)OC(C)C(=O)N(C)C 17167,S(=O)(=O)(c1cccnc1N1CC2(CC(C)CO2)C1)NCC(c1ccsc1)OC 17168,C1(C(N2C(C)CN(C(=O)CC#N)C(C)C2)=O)=CC=CC=CC=C2N(C=C1)C2=O 17169,N1(C(CSSC)=O)CC2CCCC(CNC(C3CC34CCCCC4)=O)C2C1 17170,CN1CCN(C(c2cc(C(F)F)cs2)=O)C(CNC(c2cc(C(N)=O)c[nH]2)=O)C1 17171,c1(NC(C2C3CN(C(CCCN(C)C)=O)CC32)=O)ccc2ncnn2c1 17172,c1(C(=O)NCC(C)(O)CNC(=O)CC2CC2)ccccc1O 17173,c1(C(C(=O)NC(C)C)N(C)Cc2nc(CO)n[nH]2)cc(C#N)cs1 17174,N1(C(c2ccc(OC)nc2C)C(=O)NCCC2(C)CC2)CCC(C2CC2)CC1 17175,c1(OC)ccccc1C(O)C(=O)NC1CCC1CNC(=O)Cc1ccc(Cl)cn1 17176,C12(C(N(C(CNC(c3cc(OC)nc(OC)c3)=O)C)C)=O)CC=CCN1CCC2 17177,c1(C(=O)NC2C(C(=O)NC(CC=C)CO)CCCC2)cc2ccoc2cc1C 17178,N1(C(C2(COC)CCCO2)=O)CCCC(NC(=O)CCNC(=O)OC)C1 17179,N1(C(CN(c2cnn(C)c2)C)=O)CC2=C(C1)CN(C(=O)C1=CCCCO1)C2 17180,C(C)(C)(CC(=O)NCc1ncccc1C(N1CC(C)(CO)C1)=O)OC 17181,c1(C(=O)NC(C)CC(C)NC(=O)C=CS(C)=O)cccc2nc(C(F)(F)F)[nH]c12 17182,n1(CC)cnc(C(=O)NCCC2CCCN2C(=O)C(F)=CC2CC2)n1 17183,C(=O)(CCCC(F)(F)CO)NCC1(NC(C(CCCC)N(C)C)=O)CC1 17184,C1(NC(c2c(OC)scc2)=O)CCN(C(=O)CCn2cc(Cl)cn2)CC1F 17185,S(=O)(=O)(c1cccc(F)c1)N(CC(c1ccccc1)C)CCCC1CCC1 17186,N1(C(=O)NCCCCOC)CCCC(NCc2ccnc(OC)c2)C1 17187,n1(CCOC)ncc(C(=O)N(CC(C)(C)CNC(C2C3CCN2CC3)=O)C)c1C 17188,C1(COC)CN(C(=O)CC2(C)CC(F)(F)C2)CCN1C(C1CC(C)(C)CO1)=O 17189,S(=O)(=O)(c1ccc(F)c(F)c1)N1C2CCN(C(c3cc(Cl)ncn3)=O)C2CC1 17190,N1(C(C2CC(C3CC3)=NO2)=O)CCC2C(CCCN2C(C2CCCC2)=O)C1 17191,c1(C(N2CCC(NCc3cccc(NC(C)=O)c3)CC2)=O)cnc(F)c(C)c1 17192,c1(NC(C)=O)cccc(C(=O)NC2CCCN(C(=O)C(C)(C)C3CC3)C2)c1C 17193,C1(C(N2CCC(COCC)C2)=O)CCC(CNC(c2ncn(C)c2C)=O)CC1 17194,c1(SC)ccccc1CNC1CC(CC(=O)NC2CC2)C1 17195,Cn1nc(O)cc1C(N1CCOCC1CNC(c1ccoc1C(F)(F)F)=O)=O 17196,C(N=c1nc(C)[nH]s1)C1C2CN(C(C3CCC(C(=O)OCC)CC3)=O)CC21 17197,c1(C(=O)NC(CC(C)NC(COCC#C)=O)C)c(N)cc(OC)cc1F 17198,CC(C)CC(O)C(C)C(=O)N1C(C(=O)N(C)CC2(C)CCCO2)CC2CC12 17199,N1(C(C(C(C)(C)C)=O)=O)CCC=C(C(=O)Nc2cnn3cccnc23)C1 17200,Cc1c(Cl)ccnc1C(N1CCCCCC1CNC(C1(F)CC2CCC1O2)=O)=O 17201,C(C)(N=c1[nH]c2c(c(=NCCOc3ccncc3)[nH]1)COCC2)c1c(C)ncs1 17202,CCCC(C)(C)CC(=O)N1CCCC(C)(C)C1C(=O)NC1CN2CCCC1C2 17203,N1(C(c2nc(C)c(C)[nH]2)=O)CCC(C2CCNC2)C1 17204,C1(C(N(CC(O)CNC(=O)C2=CCSC2)C)=O)CCCC2(CCC2)C1 17205,N1(C(CCCOCC=C)=O)CC=CC(C(=O)NC(c2scnc2C)C)C1 17206,CC1CC(NC(=O)C(c2ccccn2)O)CN1C(c1cc(C(N)=O)cs1)=O 17207,c1(C2CN(C(c3cc(C(=O)OC)on3)=O)C2)ccc(-c2nn[nH]n2)cc1 17208,C1(CCC)CN(C(=O)C(C)(CC)OC)CCN1C(=O)C(c1cccc(C)c1)=O 17209,C(=O)(Nn1c(C)nc2ccccc2c1=O)C1(c2cccc(OC)c2)CCCC1 17210,c1(N(CCC(N)=O)C)nc(N2CCC(CC(F)(F)F)C2)c2c(n1)CCS2 17211,Cc1ncccc1CC(=O)N(C(C(=O)NOCCN1CCOC1=O)C1CC1)C 17212,N1(C(c2cnc(C)nn2)=O)CC2CCN(C(=O)COc3ccc(F)nc3)CC2C1 17213,C(C(=O)NCC(C)(O)CO)(C(C)C)NC(COC)=O 17214,c1(OC)ccc(S(C)(=O)=O)cc1C(N1CCC(NC(C2CN(C(C)C)C2)=O)C1)=O 17215,CC(C(=O)NCC(=O)C=O)N(C)C(C1CC1)C1CC1.c1(CCCNC2CC2)cn[nH]c1 17216,CCCC(C)(CC)C(=O)N1CCC(NC(c2cc(Cl)c([N+](=O)[O-])[nH]2)=O)C(C)(C)C1 17217,c1(C(N2CC3C(C(=O)OC(C)(C)C)C3C2)C(=O)NC)ccc(C#N)cn1 17218,c1(C(=O)NCCN(C)C(c2cnn(C)c2Br)=O)cc(Cl)c(N)c(Cl)c1 17219,CC(C)(O)C(C(=O)NCc1ccsc1)NC(=O)COCCCF 17220,C(CCS(C)(=O)=O)(C(=O)NC1CCN(C(C2CC(=O)OC2(C)C)=O)CC1O)OC 17221,c1(C(=O)NCC(C#C)C(C)C)ccc2c(c1)C(=O)N(C)C2=O 17222,N1(CCOCC=C)CCN(C2CCN(C(C3CC34CC4)=O)C2)CC1 17223,N1(C(C(C)OCCC(C)C)=O)CC2CCN(C(c3cc4ncccc4s3)=O)C2C1 17224,c1(SC)ccc(F)c(C(N2CCC(NC(c3ccnc(Br)c3F)=O)C(O)C2)=O)c1 17225,C1(COC)(CNC(=O)C(O)CC2CCCC2)CCN(C(=O)C(C)(O)C2CCC2)C1 17226,C(C)(C(C(=O)NCC1CC(C)C1)C(C)C)NC(C(C)=CC=C)=O 17227,C(=O)(C(F)(CNC(=O)C=C=C(C)C)C(C)C)NC(CCOCC)C 17228,c1(C(=O)NC2C(CC)CN(C(=O)Cc3ccsc3C)C2)ccc(C)c2c1CCC2 17229,N=c1cc(C(N2CCC(CF)(NC(=O)CCC3CCOC3)C2)=O)cc(N)[nH]1 17230,Nc1cc(C(=O)NCC2(CNC(=O)CC3CCOCC3)CCC2)ccc1Cl 17231,C1(C)(CNC(CC(CC)C)=O)CCC(NC(=O)CCNC(c2ccco2)=O)CC1 17232,c1(CNC(C(CCCC)NC(=O)CN)=O)n[nH]c2c1COCC2 17233,C(=O)(CCS(C)(=O)=O)N1CC(OCC)C(CNC(c2cc(N)ccn2)=O)C1 17234,c1(CC)nc(N2CC(NC(c3cc(=O)c(OC)c[nH]3)=O)C(C)(C)C2)cc(C#N)n1 17235,c1(C(=O)OCC(CC)F)cnc2sc(C)nc2c1 17236,C=CCCCC(C(=O)NCC(C)Cc1ccc(OC)cc1)N(C1CC(F)(F)C1)C 17237,N1(C(C2C(NC(c3ccns3)=O)C2)=O)CCc2c(cccc2[N+](=O)[O-])C1 17238,c1(OC)[nH]nc(C(=O)NCC(Cc2ccccc2)N(C)C)c1Br 17239,C(CC(F)F)(C(=O)N1CCC(n2ccnc2)C1)N(C(C(CCC)O)=O)C 17240,C1(c2nc(CNC(=O)CC3(O)CC3)[nH]n2)CCCN(C(=O)CC2CCOC2)C1 17241,C#Cc1ccnc(C(N2CCC(N(C)C(c3cccc(N)c3F)=O)C2)=O)c1 17242,N1(C(C2(NC(=O)CC3CCCSC3)CCCC2)=O)CCc2cncnc2C1 17243,C(=O)(C(C)CCCC(C)C)N1C(C(=O)NC(CCC)C2CC2)(COC)C=CC1 17244,CN1CC=CCC1c1nnc(O)n1Cn1cc(C2CCOC2)nn1.N12CCC1C2 17245,C(=O)(CC(CC(N)=O)CC(C)C)NC(CN(C(c1c(C)nco1)=O)C)(C)C 17246,C(=O)(CCCCCC(C)C)NC(CCCCNC(C(C)=CC)=O)C 17247,N1(C(C(=C(C)C2CC2)F)=O)CC(CNC(=O)CN2CCS(=O)CC2)C(C)(C)C1 17248,C(=O)(C1=C(c2ccccc2)SCCO1)NC1CN(C(CC(C)(C)C#N)=O)C2C1C2 17249,c1(CC(N2CC(CNC(C(C)SC)=O)C(C)CC2)=O)cn2cccc(C)c2n1 17250,CC1CC(C(=O)N2CCN(C(=O)Cc3cccnc3CC3CC3)C(CF)C2)=NO1 17251,c1(CNC(=O)NC2C(F)(F)C23CC3)ccc(F)c(N2CCCC(CO)C2)c1 17252,N(C(=NCC(C(C)C)C(C)C)NCC1CCC1(F)F)C(CC)CC 17253,C1(O)(CCNC(C(CC)SC)=O)CCN(C(=O)C(c2ccc(C)cc2)O)CC1 17254,Cc1ccc(C)c(C(=O)NCC2CC(NC(c3cnc(S)nc3)=O)C23CCC3)n1 17255,c1(OCCN(C)C)ccc(CNC(C2CCC(NC(=O)CCC(C)=O)C2)=O)cc1 17256,C(=O)(C(C(C)C1CCCCC1)NC(=O)CN1CC(O)CC1C(=O)N(C)C)OC 17257,Cc1nc(C2CC2)nc(C)c1C(=O)NCC1(C(N)=O)CN(C(c2ccoc2)=O)C1 17258,CCCCCC(C)(CC)C(=O)NCC(C)(C)CC1CN(C(=O)C(F)=C(C)C)C1 17259,C12(C(N(CCCCNC(C3CC(=O)CS3)=O)C)=O)CC3CC(CC1C3)C2 17260,C(=O)(C1=CC2C=CC1C2)N1C(C(=O)NCCc2ccccc2O)CC(C)(C)C1 17261,Cn1c(O)nc2ccc(C(=O)NCC3CCC(NC(=O)CNC=O)C3)cc12 17262,C=Cc1cnn(C)c1C(=O)NCC(CCCC)NC(c1scnc1CC)=O 17263,c1(CC)cnn2ccc(C(=O)NC(C)CCCNC(=O)CN(C)CC)nc12 17264,C1(C(=O)NCCN(C(=O)CCC2CCCCC2)C(C)C)(OC)CC(CF)C1 17265,C1(NC(CCCCC)=O)C(CNC(=O)C(C2CC2)C2CC2)CCC12CCC2 17266,CN1Cc2ccccc2CC1C(=O)NCC1CCC(F)C1.N12CCC(F)(C1)C2=O 17267,c1(C(N2CC(C)(NC(c3c(C)c[nH]n3)=O)C2)=O)cc(S(=O)(=O)CC#N)ccc1F 17268,CC1=C(Br)CCN(CCC2CCC(c3ccccc3)CC2)C1 17269,CC(C)(CCC(=O)N1CC2CC1CS2=O)NC(c1cc[nH]c(=N)n1)=O 17270,C1(=CNC(C(N2CCC(C)C2)=O)=O)CN2CCC1CC2 17271,Cc1sc(=O)n(CCC(N2CC(NC(=O)CCCCCF)C(C(F)F)C2)=O)c1C 17272,c1(C(N(CC)Cc2nncs2)=O)ccc(CNC(c2oc(C)cc2C)=O)nc1 17273,N1(C(C2CC(C)OC2)=O)CCC(NC(=O)CCc2ccn(C)n2)C12CCCC2 17274,c1(NC(CNC(=O)OC(C)(C)C)CF)nc2ccccc2n1-c1ccc(Cl)c(Cl)c1 17275,CCC(CC)CC(F)C(=O)N1CCCC1C(C)NC(c1n[nH]cc1C)=O 17276,CC(C)C(C(=O)N(CCNC(=O)C(c1ccccc1)F)C1CC1)NC(N)=O 17277,c1(SCc2ncc(C)o2)nc(-c2cncs2)nn1CCc1csc(Cl)c1 17278,CCC(C)C(C(=O)NCC1(CNC(=O)CC2CSC2)CC12CCC2)N(C)C 17279,N1(C(Cc2cccc(OC)c2)=O)CC2CCC(C1)N2C(=O)CC1CN(C)CC1O 17280,C1(CNC(C(CC)(C)CO)=O)N(C(c2nc(C)ccc2F)=O)CCCC1(C)C 17281,CC(F)(F)C(C)(C)CC(=O)N1CCCCCC(S(C)(=O)=O)C1.c12nc(cs1)C2=O 17282,C=C1CC(C)(C(=O)NC(C)C=CC(=O)NC2(CO)CC(F)C2)C1 17283,C1(C)(C(=O)NCc2cccc(NC(CCCCCOC)=O)c2)CC(C)OC(C)C1 17284,CC(C)C(O)C(=O)N1CC=CC1(C)C(=O)N(C)CCC1CN(C)C1 17285,C(=O)(C(C#N)C(C)(C)C)N1CC(OCCC(=O)NCc2ccc(C)cc2F)C1 17286,C12(CCNC(C(CC)(F)F)=O)CCC1CN(C(c1cncc(C)n1)=O)C2 17287,C1(C2CC2)(CNC(=O)CCc2cnoc2)CCN(C(c2cccnn2)=O)C1 17288,c1(CCC)cnnc(C(=O)N(C2CCC(NC(C3CC3COC)=O)CC2)C)c1 17289,CC(C)(C)CCCC(=O)NCC1CN(C(=O)CCOc2cc(F)cc(F)c2)C1 17290,CCC(CNC(=O)C(c1cc(Br)ccc1F)(C)C)(CCOC)C(=O)O 17291,c1(C(C)NC(c2c(CNC(CCCOCC=C)=O)noc2)=O)cccnc1F 17292,C(=O)(C(CCOC)NC(=O)C=C1CCC(C)CC1)NCCN1CCC(OCC)C1 17293,c1(NCCN(C(CCC(=O)NCC)=O)CC2CC2)ccc(O)nc1Cl.C(SC)CC 17294,C1(CNC(=O)CC2(O)CCOCC2)CCC2(CN(C(=O)C(F)CC3CC3)C2)O1 17295,C1(CNC(CN(C)CC)=O)CCC(NC(=O)CCc2ccccn2)CC1 17296,c1(NCC(CC)CCO)cc(=NCCOC2CCCC2)[nH]cn1 17297,c1(CN(C(=O)C(=O)NCc2snnc2C)CCC#C)ccc(F)c(F)c1F 17298,C(=O)(C1=NN(C)C(=O)CC1)NCC(CCOC)NC(c1c(C)cccc1Cl)=O 17299,c1(N(CC(CN(C)C(C2(F)CCCCC2)=O)O)C)nc2c(cc1C#N)CCOC2 17300,Cc1cc(C(N2CC(NC(c3c[nH]c(=N)o3)=O)C3(CC3)C2)=O)cc(Br)c1C 17301,n1(C(C)C)ncc(C(=O)NC(CNC(=O)Cn2cccn2)C(C)C)c1F 17302,C1(C(N2CC(C)(CC=C)C2)=O)(C(C)C)CCN(C(C2CCC2C)=O)C1 17303,C(=O)(C1=CC2CCC(C1)C2)N1CC2C(CCNC(c3c(CC)[nH]cc3)=O)(CC2)C1 17304,N1(C(C2CC(OC)CN2C(=O)CC2CCN(C)CC2)=O)CCC2(CNC(=O)O2)C1 17305,c1(C(=O)NCC(=C)CCNC(=O)CN(C)C)cnc(OC)cc1C 17306,C1(CCC)CCC(C(=O)NC2CCC(NC(=O)C(F)C(C)C)C2)CC1 17307,c1(CC(N2CCC(N(C(=O)C=CCO)CCC)C2)=O)cnccc1Cl 17308,c1(C(N(C)CC2N(C(C3C(C(=O)OC)CCC3)=O)CCC2)=O)cc(OC)n(C)n1 17309,c1(C(CC(=O)NCC)NC(C2(C(=O)OC)CCC2)=O)ccc(C(F)(F)F)cc1 17310,N1(C(C(C)Cc2cccnc2)=O)CCCN(C(=O)COCC2CCOCC2)CC1 17311,C=Cc1cncc(C(N2CCC3CC23C(=O)NCCc2cc(C)no2)=O)c1 17312,C1(C(=O)NC2(C(C)NC(C(CC)N(C)C)=O)CC2)CCN(CC2CC2)CC1 17313,C(=O)(CC(C)(C)COC)NC1(CC=C)CCN(C(c2cc(Br)nn2C)=O)C1 17314,c1(C(N2CCCC(NC(C3(C)CC3(Cl)Cl)=O)CC2)=O)ccc2c(n1)COCC2 17315,C1(C(N2CCC(=O)NC2=O)=O)CC(OC)CCN1C(C1CCCN(C)C1)=O.CO 17316,C1(NC(c2scc(OC)c2)=O)CCN(CC2CCS(=O)(=O)CC2)C(C)C1 17317,c1(C(N2C(CCNC(CC3C(C)C3)=O)CSCC2)=O)cc2c(cc1N)OCO2 17318,C1(NC(C(COC)(C)C)=O)CN(C(c2cc(Cl)c(Br)[nH]2)=O)CCC1C 17319,C1(CC(=O)NC(C=C)(C)CC)CCN(C(C)=O)C1(C)C 17320,N1(C(C2(OCC)CCC2)=O)CCC(CN(C(=O)CN(C)C(C)C)C)CC1 17321,C(=O)(C(F)CC1CN(C(=O)CCc2nc(O)n[nH]2)C1)NCCCOC=C 17322,N1(C(C2C(C=C)C2)=O)CC(NC(c2ccc(Br)cn2)=O)C2(CCC2)C1 17323,c1(C(=O)NCCN(CCC)C(c2ocnc2C2CCC2)=O)c(Cl)cccc1Cl 17324,N1(C(Cn2nc(C)oc2=O)=O)CCC(NC(C2(CO)CCCO2)=O)C(C)(C)C1 17325,c1(N(C)Cc2n(CC)ncc2)ccc(S(=O)(=O)NC2CC(C)OC(C)C2)cn1 17326,CC(C)(C)CC(C)(C)C(=O)NCC(F)CNC(c1nccnc1N)=O 17327,c1(C(=O)NC(CNC(c2nc(C)[nH]n2)=O)C)coc(=O)c2ccccc12 17328,c1(C(=O)NC2CCC(CNC(C3CC(N4CCCC4)C3)=O)C2)sc(F)cc1Cl 17329,c1(SC)cc(C(=O)NCC2CC2NC(=O)CS(=O)(=O)NC(C)(C)C)c(C)o1 17330,c1(NC(C2(C)CCN(C(C3CCS(=O)(=O)CC3)=O)C2)=O)cc(Br)ccc1C(N)=O 17331,C1(NS(=O)(=O)Cc2cc(F)ccc2F)CC2CCC(C1)S2(=O)=O 17332,n1(CC=C)cc(C(=O)NC2(C)CC(C(N3CCC3(C)C(=O)NC)=O)C2)cn1 17333,N1(C(c2cccc(-c3cn[nH]c3)c2)C(=O)NCC=C)CCC(C)C(C)(C)C1 17334,c1(C(N2CC(N(C(=O)C3=NOCC3)C)C(F)C2)=O)ccc(O)nc1Cl 17335,C1(CNC(C(C)C2CCC2)=O)CN(C(c2cc(C3CC3)cc(F)c2)=O)CCCO1 17336,C1(NC(c2nc(CC)oc2)=O)(CF)CCN(C(C2(C(N3CCCC3)=O)CC2)=O)C1 17337,CCCCCCCC(=O)N1CC(NC(c2cc(F)ccc2C)=O)C(O)C1 17338,c1(SC)cccnc1C(=O)NC(CO)C(C)NC(C1CCCS1)=O 17339,c1(CNC(C2(C(N(C)C)=O)CC2)=O)cnn2c1CN(C(c1cnns1)=O)CC2 17340,Cc1sc(Cl)c(C(=O)NCCOCCCNC(=O)CCC2CCN(C)CC2)c1C 17341,CC#CCCCC(=O)N1CCCC1CCCNC(=O)COc1cccc(C)c1 17342,N1(C(C(COCC)C)=O)CCC2C1CCCN2C(c1cccc2ncnn12)=O 17343,C1(NC(C(C2CN(C(=O)Cc3ccsc3C)C2)OC)=O)COCCC1(F)F 17344,C1(C(N2CCN(C(=O)OC)CC2)=O)CC12CCN(Cc1ccc(I)c(O)c1)C2 17345,C1(C(N(C)Cc2c(C)cco2)=O)CC(NC(=O)Cc2cncn2C)C1(C)C 17346,N1(C(=O)NCc2cc(OC(CC(C)C)C)ncc2)CCc2ccc(Cl)nc21 17347,c1(OC)ccc(-c2cn(C3CN(C(C4C5CC6C(C5)C46)=O)CC3O)nn2)cc1OC 17348,CC1CCCC(C(=O)NCCCNC(=O)Cc2csc(C(C)(C)C)n2)CC1.C(C=O)=C 17349,N1(c2ncc(COC)cn2)CCN(C(=O)C(O)CC(C)C)C2CC12 17350,C1(NC(CCn2ncn(C)c2=O)=O)CC(NC(C2(S(C)(=O)=O)CC2)=O)C12CCC2 17351,N1(C(C(C(C)NC(C2CN(C(C)=O)C2)=O)C)=O)CCC2=C(CCCC2)C1 17352,C#CCCCCC(=O)NCc1ncoc1C1CN(C(=O)C(C)Cc2cnc[nH]2)C1 17353,c1(CC)ccc(O)c(C(=O)NCC(CC(C)C)NC(c2n[nH]c(C)c2F)=O)c1 17354,C1(C(=O)NC(C(C)NC(c2cc3occc3s2)=O)(C)C)CCc2nnnn2C1 17355,c1(C(=O)NC2CCC(CNC(C3C(OCC)C3C)=O)CC2)cc(O)ccc1N 17356,C=CCC(C)(C)CC(=O)NC1CN(C(c2cnc(CC)s2)=O)CCC1CO 17357,c1(C(N2CCC(NC(c3c(CC)ocn3)=O)C2C2CC2)=O)c(F)cc(F)cc1Cl 17358,N(C1CCc2c(Br)cccc21)C(C(CC)CC)c1nnnn1Cc1ccccc1 17359,CCCC(CCC)C(=O)NCCC(C)NC(C1CCS1(=O)=O)=O 17360,C1(C(N2CCC(OCCNC(c3ccc(SC)cc3)=O)C2)=O)CCCCN1N=O 17361,c1(C(C)=O)cc(C(=O)NCCC2CO2)co1.c1(N(CC(=O)NC(C)C)C)nccs1 17362,C=C(C)CCC(=O)N1CCCC(CCNC(=O)Cc2ccccc2OC)C1 17363,O=C(C1=C(F)CN(C(C2(F)CCOC2)=O)CC1)NCc1cn[nH]c1 17364,c1(C(=O)OC)nn(C)cc1C.C12CCN(C1)C(=O)C(C1CN(C(C)=O)C1)O2 17365,N1(C(c2n(CCC)ncc2)=O)CCOCC1CN(C)C(C1CCOC(=O)N1)=O 17366,O=C1COc2ccc(C(=O)NC34CC3CN(C(c3cnc(Cl)[nH]3)=O)C4)cc2N1 17367,c1(C(=O)NCC(C)(CO)NC(c2ccc3c(c2)CCC3)=O)cc(Cl)c([N+](=O)[O-])[nH]1 17368,N1(C(CCS(C)=O)=O)CCC(NC(=O)Cc2ccc(F)c(Cl)c2)C12CC2 17369,c1(C(N(CC(CNC(Cc2scc(C)n2)=O)C)C)=O)cccc(C2CC2)n1 17370,CCCC(O)(CCC)CC(=O)N1CCCC(C2(NC(C3(CCO)CC3)=O)CC2)C1 17371,C(c1cnn(C)c1C)=CC(N1CC(NC(c2cc(CC)ncn2)=O)C(OC)C1)=O 17372,c1(C(N2CC(N(C)C)C2)=O)cnnc2ccccc12.C12(CC13CCC3)C(=O)NC2 17373,c1(C(C2CC2)CNC(c2cnn(C)n2)=O)cccc(F)c1.N12CC=CC1C2=O 17374,C(=O)(C1CCCc2cccnc21)NC(C1CN(C(C2(C#N)CCSCC2)=O)C1)C 17375,S(=O)(=O)(c1ccc(C(N2CCC(C)(CNC(c3ccoc3)=O)C2)=O)cc1)NCC 17376,c1(C(=O)NC(CC)C(=O)NCc2nn(C)cc2CO)cnc(C)n1C 17377,N1(C(c2cc(CCC)on2)=O)CCCC(CC(=O)NC2CC3CCC2O3)C1 17378,CC1CN(C(=O)C(N)=O)CC2(CCN(C(c3ccc(S(N)(=O)=O)[nH]3)=O)C2)O1 17379,c1(CSC)c(C(=O)NC(C2CN(C(c3csc(=N)[nH]3)=O)C2)C)oc2ccccc12 17380,C1(NC(C(C)(C)OC)=O)C2CN(C(C3CCCC3C(C)C)=O)CC12 17381,C1(C)(NC(c2ncn(C(C)C)c2)=O)CCN(C(c2cc3n(n2)CCO3)=O)CC1 17382,c1(C(=O)NCC23OCC(NC(C(C)O)=O)(C2)C3)cc2c(F)ccc(Br)c2[nH]1 17383,N1(C(c2c(C)csc2C)=O)CCCN(C(=O)C=CCCc2ccccc2)CC1 17384,S(=O)(=O)(c1csc(C(N2CC(CNC(=O)C(C)(C)F)C3CC23)=O)c1)NC 17385,c1(C(=O)NCC(CO)NC(c2c(CC)con2)=O)cn(C)nc1-c1ccccc1 17386,c1(CNC(c2ccc(C)nn2)=O)ccc2c(c1)CCCC2NC(=O)CCCCO 17387,CC(O)CC(=O)NC(Cc1cc[nH]n1)C(=O)N1CC(O)(c2cc[nH]n2)C1 17388,CN1C(=O)CCC1C(=O)N(C1CCN(CCNC(=O)C(F)C2CC2)CC1)CCO 17389,N#Cc1cc(N2CCC(NC(=O)CSc3n[nH]c(O)n3)C2)nc(C2CC2)n1 17390,C1(NC(c2c(CC)occ2C)=O)CN(C(c2oncc2C)=O)CCC1F 17391,CC1CCCN(C(c2cnsc2)=O)C1CNC(C1OCCN(C)C1=O)=O 17392,C1(C(=O)NCC(C2CCC2)OC)CN(C(c2cn(C)cc2C)=O)CC1(F)F 17393,c1(N(CCCNC(CC2C(OC)COCC2)=O)C2CC2)ncn(C)c(=O)c1Br 17394,c1(C(=O)NCCCCCN(C(C)C)C(C2C=CCC2)=O)ccc(O)c(F)c1F 17395,N(C(=NCCC(=O)Nc1ccc(CC)s1)N1CCC(C2CCCC2)CC1)CC 17396,c1(C(C2CC2)NC(=O)NC(CC)CCCO)cc(Cl)ccc1Cl 17397,CC1(C)CC(NC(C2CC2c2ccc(Cl)cc2)=O)CN1C(c1ccc(F)cn1)=O 17398,C(CCCC(=O)NC(C)(C)C(=O)N1CCC1CN=[N+]=[N-])N(C)C 17399,C1(C(=O)NCCC(=O)NC2CCCCC2)CC2CCC1C1C(=O)NC(=O)C21 17400,C1(C(=O)NCCC(=C)CNC(c2ncsc2C)=O)CCc2nnc(O)c(C)c2C1 17401,c1(C(N2CCN(C(C3CC3c3ccccc3)=O)C3C2C3)=O)cn2ncccc2n1 17402,N(C1CC(F)(F)c2ccccc21)C(=O)C(N1CCc2ccc(F)cc21)=O 17403,Cc1nc2cc(C(=O)NCC3(F)CCN(C(c4cnc[nH]c4=N)=O)C3)[nH]c2s1 17404,CCC(CCCC(=O)NCCOC(C)C)NC(c1[nH]ccc1COC)=O 17405,C1(CC(N2CCC(COC)(NC(=O)C3=COCC3)CC2)=O)CC(C)CC(C)(C)C1 17406,c1(CC)cc(CN(C(C2CCC2C#N)=O)C(C)C)no1 17407,c1(C(=O)NC2CC(C(N(CCCC(C)O)C)=O)C23CCC3)cccc2[nH]ncc12 17408,Cc1c(NC(=O)C(=O)N(C)CCC2CCCN2C)cnn1-c1ccncc1 17409,CCC(CC)C(C)C(=O)NC1(C(N2CC(O)C(O)C2)=O)CC1(C)C 17410,c1(C(=O)NCC(C)CNC(=O)CCN(C)CCO)ncnc(O)c1Cl 17411,CC1CCC(CCC(=O)N(C(Cc2cccs2)CO)CC(F)F)O1 17412,c1(C(N2CCCC(C(=O)Nc3cccnc3)C2)=O)cccc2ncccc12 17413,C(=O)(CCCC(C)(C)C(=O)OC)NC(CN(C(C(C(C)OC)N(C)C)=O)C)C 17414,Cc1ccc(C(=O)NCC2CN(CC3CC3)CCO2)cc1N1CCOCC1 17415,N1(C(CSCC(C)C)=O)CC2(C1)CN(C(=O)C=CC1CCCC1)CCO2 17416,c1(C(N(C2CCCCCC2)CCNC(c2c(C)csc2)=O)=O)nnn2c1CCCC2 17417,c1(C(N2CC(NC(CS(=O)(=O)N(C)C)=O)C(F)CC2)=O)ccc2c(c1)OCCCO2 17418,N1(c2ncc(C#C)cn2)CCN(C(c2cc(F)c(Cl)cc2F)=O)C(C#N)C1 17419,Cc1cc(C(=O)NCCC(C(C)C)NC(=O)C(C)(C)C2CC2)c([N+](=O)[O-])c(O)n1 17420,C1(NC(C2(CCCC)CC2)=O)CC2(C(=O)NCC3CC(=O)N(C)C3)COC1C2 17421,c1(C(N(C2CN(C(=O)CN3CCNC(=O)C3)CC2O)C)=O)cc2occc2n1C 17422,C(C(=O)N(CCCCN(C(=O)C(O)C(F)F)C)C)(C(C)C)NC(CC(C)C)=O 17423,N1(C(C=CC(CC)=CC)=O)CC2CCN(C(c3scc(C)c3Cl)=O)C2C1 17424,Cn1cnc2c(C(N3CCOC(CNC(=O)CC4(C)CCCO4)C3)=O)ccnc12 17425,Cc1cc(C(N2CC(C)C(C)(CNC(=O)CN(C3CCC3)C)C2)=O)nnc1C 17426,CCCCCC(CC)C(=O)NC1CCC1CNC(c1cnnc(C)c1)=O 17427,N(C(=NCCOc1ccc(Br)cc1)NC1CC12CC2)C(CC)C 17428,c1(CC)nn(C)cc1C(=O)NC(C)(C)C(C)NC(=O)CCc1cn(C)nc1C 17429,Cc1cc(C)c(S(=O)(=O)N2CCC(O)(C(=O)NCC(O)C(C)(C)C)CC2)c(C)c1 17430,O=C1COc2c(C(N3CCC(C(=O)Nc4cc(Br)cc(I)c4)C3)=O)cccc2N1 17431,N1(C(c2cc(CC)ncc2)=O)CCCC(O)(CNC(C2(C)CC3CC3C2)=O)C1 17432,C1(C)(C(N2C(C(C)(C)CNC(c3sccc3Cl)=O)CCC2)=O)CCCOC1 17433,C1(C(=O)NCC(=O)NCC(NOCCC(=C)C)=O)CC12CCCC2 17434,C(=O)(C(C)(C)CC(F)F)NC(C)CC(C)NC(C1CCN1C(C)(C)C)=O 17435,CCC(C(=O)NCC12CC1CN(C(=O)Cn1nc(C(F)F)cc1C)C2)C(C)(F)F 17436,Cc1sc(O)nc1C(N1CC(C(N)=O)(CNC(=O)Cn2cnnc2)C1)=O 17437,CC1OCC2(CCN(C(=O)CC3CCCN3C(c3nccnc3Cl)=O)CC2)C1N 17438,CC1C(C)CCN1C(=NCC1(CC#N)CCC1)NC1CC(c2cccc(Cl)c2)C1 17439,N1(C(c2c(C)nc(CNC(C(C)(C3CCC3)OC)=O)o2)=O)CCN(C)C(=O)C1 17440,c1(OC)cc(C(=O)NC(C)C(C(C)C)NC(=O)CCC(F)F)ccc1S(N)(=O)=O 17441,C(CCNC(C1CCCN1C(C)=O)=O)(C(=O)NCC(O)(COC)CO)OC 17442,CC1CN(C(C2CS(=O)C2)=O)CCC1NC(=O)CC(C)(O)C1CC1 17443,CC(C)(C)CCCCC(=O)NC1CN(C(c2ccn(CC#N)n2)=O)CC(C)(C)C1 17444,C(C)(CCC(=O)NCC1CCCC1C(=O)NC1(CCF)CC1)OC 17445,c1(-c2ccc(NC(c3ccc4c(n3)CCC4)=O)cc2)cc(Cl)c(Cl)cc1Cl 17446,C1(NC(c2sc(CC)c(C)c2)=O)CN(C(C2(CCOC)CCC2)=O)CC1(C)C 17447,CC1CC(N(C(=O)CC(F)(F)F)C(=O)CC2CC3CCC2O3)CN1CCC 17448,c1(CC)ccc(C(=O)NCC(Cc2ccccc2)CC(=O)OC)cc1CC 17449,C1(NCCC2N(C(CCC(=O)NC3(C)CC3)=O)CCSC2)CCCC(F)(F)CC1 17450,N1(C(C=CCC)=O)CCC(NC(c2cc(C(C)=O)c[nH]2)=O)CC1 17451,C12(C(=O)NC3C(NC(c4[nH]cc(C)c4)=O)COC3)CCCC(C)(C1)OC2 17452,C1(CNC(c2cc(C)ns2)=O)CC(F)(F)CN1C(c1ccc(N)c(Cl)n1)=O 17453,N1(C(c2n(CC=C)ccc2)=O)CC(NC(c2cc(C3CC3)on2)=O)C(C)C1 17454,CCCCN=C(NCC(c1ccc(F)cc1)OC)NC1CC(=O)N(CC(C)C)C1 17455,N1(C(Cn2c(C)ccc2C)=O)CCC2C(NC(C3C(C4CC4)C3(F)F)=O)CC12 17456,c1(NC(CCC(C)NC(=O)C=CC2CCOC2)=O)cccn2ncnc12 17457,CC1(C)CCC=C1C(=O)NCC1CC(O)(CNC(c2cn(CCC3CC3)nn2)=O)C1 17458,CN=c1cc(C(=O)NCC(c2cn(C(C)C(=O)O)nn2)(C)C)c(Br)c[nH]1 17459,C1(CNC(C(C)SC(F)(F)F)=O)CN(C(=O)COCc2ccnn2C)CCN1C 17460,C(c1ccc([N+](=O)[O-])cc1)=CC(=O)NCCNC(c1cc(F)c(OC)c(F)c1)=O 17461,c1(CN2CCC(N(C(c3cccc(CC)n3)=O)C)C2)ccc2c(c1)OCCO2 17462,C1(CNC(C2(NC(=O)NC)CCCC2)=O)CCC(NC(C2CC2CF)=O)CC1 17463,C=CCCC(O)CN(C)C(C1CC(F)CN1C(=O)C=C1CCCCC1)=O 17464,C1(NC(Cn2c(C)cnc2)=O)CC2CC1N(C(C1(NC(N)=O)CC1)=O)C2 17465,c1(CC)ncc(Br)cc1C(N1CC2CC2(NC(C2(CO)CCCO2)=O)C1)=O 17466,c12c(sc3c1CCC3)NC2=O.c1(SC)ccc(NC(=O)CS(C)(=O)=O)cn1 17467,c1(-n2cc(CSCCNC(C3(C)CCC(C)C3)=O)nn2)cccc([N+](=O)[O-])c1 17468,c1(C(N2C(CN(C(=O)CCn3cccc3)C)CCC2)=O)cn2c(n1)COCC2 17469,CC1(C(=O)NCC(C)(C2CC2)NC(=O)Cc2ccc(Cl)cn2)CS(=O)(=O)C1 17470,Cc1ccc(CC(=O)NC(C)(C)CC=CC(=O)NCCCC2CCOC2)o1 17471,C12(C(N3CCN(C(C(C)O)=O)C(C)C3)=O)COCC(c3ccc(F)cc3)(C1)C2 17472,CC1CCC(CNC(c2cccc(F)c2O)=O)N(C(=O)CCc2cnn[nH]2)C1 17473,c1(C(N2CC(CC)N(C(c3cccc(=O)o3)=O)CC2)=O)ccc2c(c1)COCC2 17474,N1(C(c2c(COC)onc2)=O)CCOC2CN(Cc3cc(Cl)cnc3Br)CC12 17475,C12(NC(CC(C)C3CC3)=O)CCCN(C(=O)COc3ccccc3O)CC1C2 17476,N1(C(C(C)OC)=O)CCCC(CNC(C2CC3CC3CC2C)=O)CC1 17477,C1(NC(C(CCC)NC(N)=O)=O)CCN(C(=O)CS(=O)(=O)CC)CCC1CO 17478,C(=O)(C1=CS(=O)CCC1)N1C(C(N2CCC(c3ccccc3)C2)=O)C2CCC1C2 17479,c1(C(=O)NC(CCC)CNC(c2ccncn2)=O)cc(F)c(C)cc1F 17480,c1(C(=O)NCCCCCNC(C2(C)CC2(Cl)Cl)=O)cc2c(nn1)CCC2 17481,Cc1cc(F)c(C(=O)NCC(C)(C2CC2)NC(C2CC(=C3CC3)C2)=O)c(Cl)c1 17482,C(=O)(C(C)(C)S(C)(=O)=O)NCC(C)(C)CCNC(C1CCCCCC1)=O 17483,c1(OC)ccc(-c2noc(C3CCCC3N)n2)c(Cl)c1 17484,N1(C(C2C(=O)NCC2)=O)CCC2CC1CN(C(c1ccc3c[nH]nc3c1)=O)C2 17485,c1(C(N(CCC2N(C(C3(SC)CCC3)=O)CCCC2)C)=O)noc2ncccc12 17486,Cn1cc(C(Cc2cn(CCO)nn2)NC(=O)CC2COC(=O)C2)cn1 17487,N1(C(C(ONC(C(C)c2cc(C)[nH]n2)=O)(C)C)=O)CC2CCCC(O)C2C1 17488,CC1(CC(=O)NCCNC(=O)C(F)=CC2CC2)CC1(F)Cl 17489,N1(C(CCc2nnc(C(C)C)o2)=O)CCN(C(=O)C=CCF)CC12CCC2 17490,c1(C(N2CC3C(C(=O)Nc4cncc(N(C)C)c4)C3C2)=O)ccnc([N+](=O)[O-])c1 17491,N1(C(C(C)C2(O)CCC2)=O)C(C(=O)NCCOC2CC2)CCC1C 17492,c1(OC)cccc(NC(=O)CSC2CCN(c3cc(C(C)=O)ncn3)C2)c1.CN 17493,CC1(C(N2CC(NC(=O)CCN3CCC3)C2)=O)CCC(=O)N1 17494,c1(CC=CC(=O)NCC2N(C(C(C)O)=O)CC2)cccc(C#N)c1.C1(N)CCCCC1 17495,C#CCC(CC(F)F)C(=O)N1CC(O)CC1CC(=O)NCCC(C)C(F)F 17496,c1(C(=O)Nc2cc(C(N3CCCC(C)(O)C3)=O)n(C)c2)ccc([N+](=O)[O-])cc1Br 17497,c1(NC(C(CSC)C)=O)cccc(NC(=O)CCc2nncn2C)c1 17498,C1(NC(c2c(CCC)n(C)nc2)=O)CN(C(=O)C(C2CC2)N(C)C)CC(C)(C)C1 17499,N1(C(CCCOCCOC)=O)CC2(CC(NC(=O)CC3(OC)CC3)CO2)C1 17500,N1(C(c2cc(CC)on2)=O)CC2CCN(C(C3(c4cc[nH]n4)CC3)=O)C2C1 17501,C12(NC(c3cc(C(F)F)ccn3)=O)CCC1CN(C(=O)CC1CCCCC1O)C2 17502,c1(N(CCNC(=O)CSCC(=O)NC2CCC2F)CC2CC2)ccccc1Cl 17503,CC(C(=O)NCC(C)(C)C(=O)N1CCC(OC(=O)C(C)(C)C)CC1)C(F)F 17504,c1(OC)cc(OC)c2ccnc(NCc3cccnc3C)c2c1 17505,c1(C(C)C)ccc(C(=O)NCCn2cc(-c3cccs3)nn2)cc1F 17506,c1(SCC(=O)N(CC)CC)nccn1C(C)(C)C.C1(=O)C(=O)NC(C)CN1 17507,c1(C(=O)NCC2(NC(C3CCC4(CCC4)C3)=O)CC2)ccnc2cc[nH]c12 17508,c1(C(=O)OCC)ccc(C(=O)NC(C)(C)CNC(=O)C(c2ccccc2)O)nc1 17509,C1(C(N(C(C)C(=O)NCC(C(C)(C)C)OC)CC)=O)CCN(C)C(=O)C1 17510,c1(N2CC(OC)C2)ccnc(NC(=O)NCC(c2occc2Br)(F)F)n1 17511,C(CCCCCNC(c1nocc1Br)=O)N(C(=O)COC1CC(F)(F)C1)C 17512,C12(CNC(c3c(C)nc(N(C)C)s3)=O)CCC(CC1)N2C(c1cocn1)=O 17513,N1(C(C(CC=CCC)C)=O)CC(C(=O)N(CC(F)Cl)C)CC12CCC2 17514,C1(C)(C(=O)NCC(=C2CN(C(CC(C)C3CC3)=O)C2)F)CCNC1=O 17515,C1(C(N2CCCC(CC(=O)NC3(C)CC3(F)F)C2)=O)CC2CCCC2C1 17516,C1(NC(C(C(CC)O)C)=O)CCN(C(=O)C(C)(O)c2ccccn2)CC12CCC2 17517,c1(C(C(=O)NC2CC(NC(c3c(CC)occ3)=O)C2)(F)F)ccc(Br)cn1 17518,c1(C(N2CC3CN(Cc4nc5ccccc5o4)C3C2)=O)ccc(Br)c2cc[nH]c12 17519,C(=O)(C(C)(C)C(=O)N(CC(C)NC(c1cc(Cl)ncc1NC)=O)C1CC1)OC 17520,CC1(C)CCCC(C(=O)NC2CN(C(c3cccnn3)=O)CC2(C)C)C1 17521,N(C(=NCCc1ncccc1C)NCc1nn(C)cc1Br)C(COC)C 17522,N1(C(C(C)OCC(F)(F)F)=O)CCN2CCN(C(C3(C)CC3C)=O)CC2C1 17523,N1(C(C(C)=CC2CC2)=O)C2CCCC1CN(C(C1CC3CCC1O3)=O)C2 17524,c1(OC)ccc(C(N2CCC(C)(CC(=O)Nc3ncccc3C#N)C2)=O)cc1C 17525,c1(CC)occc1C(=O)NCC(C1CC1)NC(=O)CC#N 17526,c1(C(N(CCC(N2CC(CC)C(NC(N)=O)CC2)=O)C)=O)cc(C)cc(C)c1N 17527,c1(C(C)C)ncncc1C(=O)NCC1(C(F)F)CCN(C(=O)C(C)C(F)F)C1 17528,CC1CCCN(C(c2cnn(C(F)(F)F)c2)=O)C1CNC(c1ccsn1)=O 17529,c1(NC(CC)CN(C)C)ncccc1S(=O)(=O)NCc1cccc(C)c1 17530,C1(CNC(=O)C=Cc2cnc[nH]2)CC2CCC(C1)N2C(=O)CSCC1CCCO1 17531,c1(C(=O)NCC(C2CCN(C(CC(C)SC)=O)CC2)(C)O)c(O)cccc1F 17532,CCCCC(F)C(=O)NC1CC(OCC(N2CCC(CC(C)(C)C)C2)=O)C1 17533,c1(CNC(C)=O)cccc(N(C)C(C2CCC(NC(C3(OC)CCC3)=O)C2)=O)n1 17534,CCC(CC(=O)N(C(CC)C(=O)NCCn1nc(C)cc1C)C1CC1)CC(C)C 17535,C1(F)(CNC(C=CCCC)=O)CCN(C(=O)CN(C)CCOC)C1 17536,C(=O)(C(O)CC(C)(C)C)NCC1(F)CCN(C(C(CC)C#N)=O)CC1 17537,C(=O)(C1=C(Cl)CCC(C)C1)NCC(C1CCN(C(CCC#CC)=O)CC1)F 17538,C1(Nc2n(C)c(=O)nc(O)c2)CC2(CCCCN2C(=O)CCN2CCC(F)C2)C1 17539,N1(C(CCC)=O)CCCC(CCNC(=O)C(c2cc(Cl)cc(Cl)c2)(C)C)CC1 17540,Cc1ccc(C(CNC(=O)CSCC(=O)OC(C)(C)C)NC(=O)C(C)C(C)O)cc1 17541,c1(CN(C(c2ccncc2)C)C)cc(Cc2ccccc2)on1 17542,CN1CCOCC1CC(=O)NC1CCC1NC(C1CC(n2ccnn2)C1)=O 17543,c1(C(N2C(CNC(C(C=C)(C)CC)=O)CC(F)C2)=O)cc(S(=O)(=O)NC)oc1C 17544,C(C(=O)NOCC(F)F)(C1CC1)NC(C1CC(C(C)C)C1)=O 17545,C=CCC(C(=O)NC1(CCSC)CN(C(=O)CC2CC(F)(F)C2)C1)NC(C)=O 17546,N1(C(C2CN(C(C)=O)C2)=O)CC(N(C)C)C(CCNC(=O)Cc2csc(C)n2)C1 17547,N1(C(c2nn(CC)c(C)c2)=O)CCC2(CCCN2C(=O)C(O)C2CC2)CC1 17548,Cc1nn2cc[nH]c(=O)c2c1C(=O)NCCC(O)CNC(=O)C(C)C(C)(C)C 17549,C1(C#N)(C(=O)NC2C(OC)CN(C(=O)CC3(OC)CCCC3)C2)CC12CCC2 17550,c1(NC2C(SC)CCC2)ccc(S(=O)(=O)N(C)Cc2ccc(F)cc2C)cc1F 17551,N1(C(=O)NCC(=O)OCC)CC(OC)CC(NCc2ccc(O)nc2Cl)C1 17552,CC(C)CC(C)(C)CNC(C1CCN(C(=O)C2C=CCC2)O1)=O 17553,C1(C(N(C(CC)CNC(=O)CC(O)C2CCCC2)C)=O)CCC2CC2CC1 17554,C1(NC(CCOCC)=O)CN(C(C2Cc3nccnc3C2)=O)C2(CCOCC2)C1 17555,c1(NC(C2COCCN2C(C2CC(O)C2)=O)=O)c(F)c(F)nc(F)c1F 17556,c1(C(=O)NC)cc(C)[nH]c(=NCC2CCCC2NC(c2nn(C)cc2Cl)=O)n1 17557,C1(C)(CCC(=O)NCCCCc2cn(CCCC)nn2)CCC(=O)N1 17558,CC1(C)C(NC(c2ccnc(NC3CCC3)c2)=O)CCN1C(=O)Cn1cncn1 17559,c1(C(=O)NC2CCN(C(c3c(C)c(F)ccc3N)=O)C2)c(F)cccc1[N+](=O)[O-] 17560,CS(C)(=O)=NCC(=O)NC1CCOCC1NC(=O)C=Cc1ccccn1 17561,C#CCC(CC(F)F)C(=O)N(CC(C)(C)C(=O)NC1CC2(C1)CC(C#N)C2)C 17562,C12(NC(C=CS(C)=O)=O)CCOCC1CN(C(=O)Cc1ncnc3sccc13)C2 17563,C1(NC(c2cc(OC)n(C)n2)c2n(CCCC)nnn2)CC2(CCOC2)C1 17564,c1(C(=O)Nc2c(OCC)ncnc2)ccc2[nH]nc(-c3c(C)nn(C)c3C)c2c1 17565,N1(C(CCN2C(=O)OCC2)=O)CCC(CCO)(CNC(C2(CF)CCC2)=O)C1 17566,c1(C(=O)NC2C(CNC(c3c(CC)[nH]cc3)=O)CCCC2)nn(C)c(N)c1C 17567,Cc1nc(SCC(=O)NC(CNC(=O)C(C)N2CCCC2)C2CCC2)n[nH]1 17568,Cc1ccc(-c2ccnn2C)cc1C(=O)NC(C)Cc1ncc(Br)cn1 17569,N1(C(C(=O)NCC)=O)CC2CCC2(CC(=O)NCCN2CCCCC2C)C1 17570,C1(NC(c2cnc(CCCC)s2)=O)CCCN(C(c2cscc2F)=O)C1 17571,N1(C(CC2(NC(C)=O)CC2)=O)CCC12CN(C(C1CCCS1(=O)=O)=O)C2 17572,c1(C(N(C(CNC(=O)C2=CCCC2(C)C)C2CC2)C)=O)cc(F)cc(N)c1F 17573,C(=O)(CCS(C)(=O)=O)NCC(CC)(CC)NC(C1CC2C=CC1O2)=O 17574,Cc1cc(Cl)ccc1C(N1CC(CN(C(=O)Cn2cnnn2)C2CC2)C1)=O 17575,C1(NC(c2n(C)nc(O)c2)=O)CC2CC1CN(C(C1CNC(=O)CC1(C)C)=O)C2 17576,C1(OC)CN(C(c2cocn2)=O)CCC1NC(c1cc(Cl)cnc1Br)=O 17577,Cn1cc2c(n1)CCC(C(=O)NC1CC1NC(=O)C=Cc1ccc(Cl)cc1F)C2 17578,Nc1ncc(F)cc1C(=O)NCCNC(c1c[nH]nc1C1CCOC1)=O 17579,C1(C(=O)N(CCCNC(C2CC2CF)=O)C)(NC(C)C)CC1 17580,N1(C(C(CC#C)O)=O)CCCCCC1C(=O)Nc1cc(CC)ccc1C 17581,CC1CN(C(c2coc(C3CC3)n2)=O)CCN1C(=O)Cc1cc(Cl)cs1 17582,c1(NC2CN(C(Cc3cc(C)cc(C)c3)=O)CC(F)C2)ncnc2occc12 17583,CC(C)C(C)CC(=O)NC(CC1CCC1)C(=O)N1CC(c2cnsc2)C1 17584,CC(C)(C)C(CNC(C1CC2(CCC2=O)C1)=O)C(=O)NCCC(F)=C(F)F 17585,C1(CNC(c2ccc(C=C)cc2)=O)CN(C(=O)CO)C2(CCC2)C1 17586,C(=O)(C1=CCC(C)CC1)NCC(CC)(CC)NC(=O)Cn1ncnn1 17587,C1(C(N2C(CNC(c3c(CC)noc3)=O)CCCC2)=O)Cc2cccc(C)c2O1 17588,N1(C(CCCCCC)=O)CC(C)CN(C(=O)CCC=CC(C)C)CC1C 17589,c1(C(=O)NC(CNC(C2N(C(C)C)CCCC2)=O)C)ccc(N)c(O)c1 17590,c1(C(N(CC(C)N(C)C(C2CCC(=O)N2)=O)C)=O)coc2c(F)c(Cl)ccc12 17591,CC1CCOC(C(=O)NCCCNC(=O)CSc2cccs2)C1 17592,c1(C(=O)NC2C(CNC(C3C(CC)CCO3)=O)CCC2)ccc(C2CC2)cc1C 17593,CC1(C)C(C)(C(=O)NC2CN(C(c3sccc3C(F)F)=O)CCC2CO)C1(C)C 17594,c1(CCC=C)ccc(OC(=O)Cc2nccn2-c2ccc(F)cc2)cc1 17595,C1(C(N2CCC2CNC(C23CCN(CC2)C3)=O)=O)CC12CCCOC2 17596,N1(C(=O)Nc2c(CC)cccc2)CC2CC1CN2C(=O)OC(C)(C)C 17597,C1(C(N2CCC(CCNC(c3ccccc3Cl)=O)C2)=O)CCC2(CC1)CC2(F)F 17598,N1(C(Cc2cc(OC)no2)=O)CC(CNC(=O)C(=O)N=S(C)(C)=O)CC(C)(C)C1 17599,N1(C(CCCC#N)=O)CC2CC(C1)C2NC(=O)C(Cc1ccccc1)OC1CC1 17600,CC1CCN(C(C2C3C4CCC(C4)C23)=O)CC1NC(=O)CN(C)CCN(C)C 17601,N1(C(=O)CCc2ccsc2)CCC(CNC(C2(F)CCOC2)=O)C1 17602,C1(NC(C2CC(n3cnnc3)C2)=O)(CF)CCN(C(=O)CC2CSC2)C1 17603,C1(C(=O)NC2(C)CC(NC(c3ccc(C(=O)OC)cc3)=O)C2)CC2(CCO1)CC2 17604,C1(N(C)C(C2CCC(O)CC2)=O)CCCN(C(=O)CN2CSCC2=O)CC1 17605,c1(CC)nc(C)oc1C(=O)NC(CO)C(=O)NCC1CCCSC1 17606,C(=O)(C1=CC2CCCC12)NCCCCC1CN(C(C(OC)OC)=O)C1 17607,N1(C(CCCCCSC)=O)CCC2C(C1)CN2C(C1CCCN(CC(F)F)C1)=O 17608,N1(C(N2CCC(N(C)C)CC2)=O)CCc2c1ccc(F)c2F 17609,C1(CNC(C(c2cn(C)nc2)O)=O)CN(C(=O)Cn2nccn2)CC12CC2 17610,c1(C(NOC(c2ccccc2)C)=O)cc(O)c(F)cn1 17611,C1(CNC(c2n(CC)ncc2Br)=O)CC2CCC1N(C(=O)C=CCOC)C2 17612,C=CCCCCCCCC(=O)N1CC2(C1)CN(C(c1cnccc1Cl)=O)CCO2 17613,C(CS(=O)(=O)CC(=O)NCc1ccc(C(=O)NC(CO)C2(O)CC2)o1)OC 17614,C(=O)(C#CC1CCCCO1)NC(C1CN(C(c2cc3ncccc3s2)=O)C1)C 17615,C(CC(C)(CC)NC(=O)Cn1ncn(C)c1=O)NC(COCCCOC)=O 17616,C1(C2CCCN(C(C3CC3(C)Br)=O)C2)(NC(C(C2CCC2)OC)=O)CC1 17617,c1(Sc2scc(C)n2)ccc(NC(=O)C(=O)NCC2(C)COCCO2)cc1 17618,c1(C(=O)NCC(C2CCC2)NC(CC2C(C(C)=O)C2(C)C)=O)n[nH]cc1[N+](=O)[O-] 17619,C1(CCC(=O)N(C(CC)C)CC)CCC(NC(c2nccn2CC)=O)C1 17620,c1(C(N(C)CCNC(C2CC3C(C2)C3(F)F)=O)=O)cc(=O)c2ccncc2o1 17621,c1(OC)cc(C(=O)NCc2nccnc2Cl)c(NC(c2cnc(Br)s2)=O)cn1 17622,C(C)(CO)(C(=O)NCCCN(C(c1cnc(N)cn1)=O)C1CC1)OC 17623,C(C)(CCC(=O)NC(C)CC(C)NC(=O)CCC1CCCC1)SC 17624,N1(Cc2ccc(C(=O)NCC)cc2)CCC(C#N)(Nc2ccc(SC)cc2)C1 17625,C(CC(=O)NC1CCCC1NC(c1c(C)nn(C)c1Cl)=O)(C1=CCCC1)OCC 17626,Cc1nc2ccc(C(N3CC(N(C)C(C4CC4(C)C)=O)C4(CC4)C3)=O)cc2s1 17627,c1(CC)cc(C(N2CCC(C(=O)N(C(C)C(=O)NC)CC)C2)=O)n(C)n1 17628,C(=O)(C(C)C(O)C(C)C)N1CCC2C(C(=O)NCC(CSC)OC)C2C1 17629,N1(C(CNS(N)(=O)=O)=O)CC2CCCN(C(c3cc4n(n3)CC(F)C4)=O)C2C1 17630,Cc1ccc(O)c(NC(c2cc(CNC(C3(CN(C)C)CC3(C)C)=O)cs2)=O)c1 17631,C1(C(=O)O)CN(C(c2cc[nH]n2)=O)CC12CN(C(c1cnc(Cl)cc1I)=O)C2 17632,N1(C(CCOCCN(C)C(C2CC(C)(C)CO2)=O)=O)CCC2(CCCCC2)C1 17633,CC1(F)CCC(C(=O)NC2CCC(NC(=O)CC3CC(=O)NC3=O)CC2)CC1 17634,Cc1cc(CNC(=O)CC2CC(NC(C3CCOC3C(C)C)=O)C2)nn1C 17635,CC(C)P1(=O)CCN(C2CC(C)(C)S(=O)(=O)C2)CC1 17636,c1(SCC(N2CCC(CNc3n(C(C)C)ncn3)C2)=O)cccc[n+]1[O-] 17637,c1(C(=O)NC(c2ccc(Br)c(F)c2)C(=O)OC)ccnc(OC)c1OC 17638,c1(C(N2CC(C(C(=O)NCC(O)C=C)OC)C2)=O)ccc(O)cc1 17639,Cc1cc(C)n(C2CCN(C(c3cccc(OC(F)(F)F)c3)C)CC2)n1 17640,Cc1cc(=O)oc(C)c1C(=O)NC1CCN(C(=O)C(C)Cc2ccc(O)cc2)C1 17641,N1(C(c2cnn(CCC)c2C)=O)CCCCC(CNC(C2(F)CCOCC2)=O)C1 17642,c1(CC)ccccc1C(=O)NC1CCC1NC(c1cn(CCO)nc1C)=O 17643,CN=C(NCCc1csc(-c2ccccc2)n1)N1CCC(C)C1C 17644,n1(CC(=O)NC(C(C)C)C)cc(C2CCCCC2)nn1 17645,C=Cc1cc(C(=O)NCC2(O)CCN(C(=O)CC3CCCN(C)C3)C2)cc(F)c1 17646,C12(C(N(C3CCN(C(=O)CN4CCCC4C)CC3)CC)=O)CCC(F)(CC1)C2 17647,CCC(CC(=O)NCc1cc(C)cs1)NC(=O)COCCCN=[N+]=[N-] 17648,C(CCN(C)C(C1CCS(=O)(=O)N1)=O)(C(C)(C)C)NC(c1c(C)csc1)=O 17649,N1(C(c2c(C)cc(Cl)cc2)=O)CC2CN(C(C34CCCC3C4(F)F)=O)CC2C1 17650,N1(C(CCC(C)(C)OC)=O)CCCC2(NC(=O)CN3CC(=O)NC3=O)CCCC12 17651,c1(SCC(=O)NCCOCCCNC(c2n[nH]cc2F)=O)cccc(F)c1 17652,CC12CC(NC(=O)CCC3CC3)(C1)C1(CN(C(c3cncc(N)n3)=O)C1)O2 17653,c1(COc2c(Br)cc(C(=O)NC)nc2)ccc(F)c2[nH]ncc12 17654,O=C1CC(N=c2[nH]c3c(c(=NCCn4ccnc4)[nH]2)CCCC3)CN1CCO 17655,C(C1c2ccsc2CCN1C(=O)CC(C)CC)NC(COCCC#C)=O 17656,c1(OC)cncc(C(N2CC(NC(=O)COC3(C)CCCC3)CC2C)=O)n1 17657,N(C1c2ccccc2CC1NC(C1CCCOC1)=O)C(=O)CC1CCOC1 17658,N1(C(C(C)C)=O)CCC(C2CC2)(CNC(c2coc(O)n2)=O)C1 17659,c1(C(c2n(CC=C)nnn2)Nc2ccccc2C)cccn(C)c1=O 17660,c1(C(N2CCC(O)(CN(C(=O)CNS(N)(=O)=O)C)C2)=O)cc2c(cn1)OCCO2 17661,Cc1ccc(O)c(CC(=O)NCc2cc(C(=O)NOCc3c(C)noc3C)n[nH]2)c1 17662,C12(C(=O)NCC(CC)NC(=O)C(C)OC3CCCCC3)CCC(C1)C(C)(C)O2 17663,N1(CC(=O)NCC)CCCC(C(=O)N(C2CC(O)(C(=O)OC)C2)C)C1 17664,c1(C(=O)NCC2(F)CCC(NC(CCC=CC)=O)C2)c(Cl)ccc(OC)c1N 17665,C=CC1(C(=O)NCCOCCN(C)C)CCN(C(=O)CC2CCCN2C)C1 17666,c1(C(N2CC(COC)(NC(=O)C(C)(C)F)C2)=O)cc(C)c(OC)c(C)c1 17667,C1(C(N2CC(C(C(N3CCC(C(=O)OC)C3C)=O)OC)C2)=O)CCC(=O)N(C)C1 17668,c1(C(=O)NCCCC(C)NC(=O)C(F)C2CC2)ccc(C(F)F)c(F)c1 17669,C1(CC(=O)N(CCC(=O)NCCS(N)(=O)=O)CC)CCN(C)CC1 17670,N1(C(c2c(C(C)C)c[nH]c2)=O)CCC(F)(F)C(NC(=O)C2CC2)C1 17671,C1(OC)CCC2(C(N3CC(NC(c4ccc(CO)s4)=O)C(C)C3)=O)CC12 17672,C(=O)(C(C)(C)CCS(C)(=O)=O)N(C(C)CNC(c1c(O)cccc1Cl)=O)C 17673,c1(C(=O)NCC(C(C)C)(C)NC(C2CC3C(C2)C3(F)F)=O)ccc2ncnn2c1 17674,Cc1coc(C)c1C=CC(=O)N(C(C)CCNC(=O)CC(C)(C)CN(C)C)C 17675,C1(CC(=O)NC2CCC2NC(C2CCCC2)=O)CCCCC1(F)F 17676,C1(NC(CC2(C)CC2)=O)CC2COCC(C1)C2NC(c1cnn(CCF)c1)=O 17677,C(=O)(C1=CC2CCC=CCCC12)N1CCC(NC(CS(=O)(=O)NC)=O)C(C)C1 17678,C(c1ccccc1F)=CCC(=O)NCC(CC)(C)NC(c1cnc(O)n1C)=O 17679,CC(C(=O)N1CC(O)CC1CNC(c1ccc(CO)cn1)=O)S(C)(=O)=O 17680,C1(NC(CC(=O)NCC#C)=O)CC2CCC(C1)N2C(C12CCC(F)(CC1)CC2)=O 17681,c1(C(N2CCN(C(Cn3ncc(C)c3)=O)C(CO)C2)=O)c(C)[nH]c2ccccc12 17682,C(c1ccc(C(F)(F)F)cc1)=CC(=O)NC1(C)CCN(C(c2ccsn2)=O)C1 17683,c1(C2CC(C(N(CC(C)N(C)C(c3c[nH]c(=O)cn3)=O)C)=O)C2)ccc(Cl)cc1 17684,c1(CC)ccc(C)cc1COC1CC(NC(=O)OCCCOC(C)(C)C)C1 17685,C12(Nc3scc(C(C)(C)C)n3)CCC1CN(C(=O)C=CC1CCOCC1)C2 17686,CC1=C(C(=O)N(C2CCN(C(=O)CC3CC3C(F)(F)F)C2)CC2CC2)CCO1 17687,C(=O)(C(F)(F)CCC1CC1)N(CCCn1cc(C(CC)OC)nn1)C 17688,C(c1ccc(O)cc1)=CC(=O)Nc1c(CC)cc(-c2cccnc2F)cc1 17689,CC1(C)CN(C(=O)CC2(O)CCC2)CCC1C(=O)NCCC(O)C(F)(F)F 17690,C1(CCC)CN(C(c2cnc(OC)nc2C(F)F)=O)CCN1C(C1CC12CC2)=O 17691,C1(O)(CNC(C2CC23CCCC3)=O)CCN(C(c2cscc2C(F)(F)F)=O)C1 17692,C1(CCCNC(c2c(C)nsc2)=O)CCCCN1C(=O)COCCCC(C)C 17693,C(=O)(CCCC(C)(C)C#N)N1CC(NC(C2(CC)CCCC2)=O)C(C)C1 17694,c1(CC)nc(C)c(C(N2CCOC(CCOCCC(=O)NC3(CF)CC3)C2)=O)s1 17695,c1(C(=O)NC2CN(C(CCOCC#C)=O)C3C2C3)ncnc2c(C)csc12 17696,c1(CC)c(NC(=O)C#CC2(CC)CC2)nc(C)nc1Cl.C12CCCCC1CN2 17697,c1(-c2onc(-c3c(C)cc(F)cc3)n2)c[nH]c2c(Cl)cccc12 17698,Cc1cn(C)cc1C(=O)N(CCC(=O)NC1C=CC(C(=O)OC(C)C)C1)C(C)C 17699,C1(c2ccccc2)CN(C(=O)OC(C)(C)C)CC1SCC1CN(C2COC2)C1 17700,CC(C)(C)CC(=O)NCC1CC(F)(CNC(=O)CSc2ccc(F)cc2)C1 17701,N1(C(COCC=C)=O)CC2(CCC2CNC(=O)C(=O)NOC)C1 17702,c1(C(N(C(c2ccccn2)C)C)=O)c[nH]n(C)c1=O 17703,CC(C(C)(C)NC(=O)COC1CC1)NC(=O)CC1CN(C)C1 17704,Cc1nc(N2CC(CNC(C3(N(C)C)CCCOC3)=O)CC2C)c2cnn(C)c2n1 17705,Cc1nc(Cl)ccc1NC(=O)CC=CCNC(=O)C(C)(C)C 17706,N1(C(c2[nH]nc(OC)c2Cl)=O)CCC2CN(C(C3CCN(C)C3)=O)CC12 17707,c1(CCC(=O)OCC)cc(=NC(C)CC(C)NC(=O)CCSC)[nH]c(C)n1 17708,C1(C)(C(N(CC(C)(C)CNC(c2ccoc2)=O)C)=O)Cc2ccccc2C(=O)O1 17709,N(C1COc2ccccc21)C(C1N(Cc2cc(OCC)c(O)c(Br)c2)CCC1)=O 17710,N1(C(C2(CC(=O)OC)CC2)=O)CC2C(CNC(=O)C(c3ccc(F)cc3)O)C2C1 17711,C1(CC(=O)NCc2ccccc2F)C2CN(C(=O)CC3CCOC3)CC12 17712,C1(C(=O)NCc2cc(C)ns2)CN(C(=O)CCc2ccoc2)CCO1 17713,C(=O)(C(C)(C)C(=O)N(C)CC1CCCN1C(=O)CCc1csc(C)n1)NC 17714,C(=O)(C(F)(CNC(=O)C1=CCN(C)C1)C(C)C)N(C)Cc1cccc(C)n1 17715,N1(C(C2CC(=O)NCC2)=O)CC(NC(=O)CCc2cnc[nH]2)C(F)(F)C1 17716,CCCC(C)(C)C(=O)NC1CCCC1C(=O)NCC(=O)N1CCCO1 17717,c1(C(=O)NCC(CNC(=O)COCC2CCC2)CO)cc2c(s1)COCC2 17718,C(=O)(C1=C(Cl)CCCC1)NC1C(N2CCN(C(C(C(C)C)C)=O)CC2)COC1 17719,CC(CC1CCCCC1)CN=c1[nH]c2c(c(=NCc3ccncn3)[nH]1)SCC2 17720,C12(C(N(C3CCN(C(=O)C(O)c4ccsc4)CC3)C)=O)CCCC1CC(=O)CC2 17721,C1(CNC(c2ccc(C(=O)OC)[nH]2)=O)C2CCC(C2)N1C(C1COCC1CF)=O 17722,N1(C(C2C(C)C2(F)F)=O)CCN(C(c2cscc2C(F)F)=O)CC(C)(C)C1 17723,C1(C(=O)NCC(C)(O)CCNC(C2CC(OC(F)F)C2)=O)CCCC2(CC2)C1 17724,CC1CC(C)C1C(=O)N(C)CCN(C)C(C1(C(N)=O)CC1)=O 17725,Cc1ccc(C(=O)NCC2CCN(C(C3CCOC3=O)=O)C2)c2ncccc12 17726,N1(C(CC2CC(C(=O)OC)C2)=O)CCC2CC12C(=O)N(CC(O)CO)C 17727,N1(C(CCCCCCC)=O)CCc2sc(CNC(=O)Cc3cncnc3)nc2C1 17728,CC1CN(C(C2CCCC(CF)C2)=O)C(C)CN1C(=O)CC1CSCCO1 17729,C1(CNC(C(=Cc2ccccn2)C)=O)CCN(C(=O)C(C)(C)C(F)F)CC1C 17730,C(CCCC(C)(F)F)NC(CNC(C(c1ccnn1C)C)=O)=O 17731,CCCCC(C)C(=O)N1CC(CNC(=O)CCOCC)C(O)C1 17732,Cc1c[nH]c(C#N)nc1=NCCNC(C1COc2ccc(F)cc2C1)=O 17733,C1(NC(C(C)NC(N)=O)=O)CCN(C(=O)CCCc2csc(=N)[nH]2)C12CC2 17734,c1(OC)ccc(Cl)cc1-c1cccc(NC(c2cc(F)ccc2Br)=O)c1 17735,N#CC1CN(C(c2ccc(S)cc2)=O)CC1NC(c1ccc(Br)cc1)=O 17736,c1(C(N(CCCCCC)CCNC(=O)Cc2ccco2)=O)ccc(OC)cc1C 17737,CC(C)C(O)CC(=O)N(C1CCN(C(C23CSCC2C3)=O)CC1)C 17738,C1(CNC(c2nc[nH]c3ncnc2-3)=O)CN(C(=O)C(F)(F)C2CC2)CC12CCC2 17739,c1(C(c2n(CC)nnn2)NC(C2CCC2)C2CC2)ccc(OC)cc1[N+](=O)[O-] 17740,C1(NC(C=C(C)C(C)C)=O)CCCCC1CNC(c1ccns1)=O 17741,C1(C(=O)NC(CNC(c2ccc(Br)s2)=O)C2CCC2)CCCCS1 17742,n1(CC)nnc2c1CCC(C(=O)NCC1CCN(C(C3COC(=O)N3)=O)CC1)C2 17743,c1(C(=O)NC2(CCNC(C3C(C(=O)OC)C3)=O)CC2)cccc2c1NC(=O)CO2 17744,C(=O)(C(CC=C)CC(C)C)N1CCC(N(C(=O)C=C2C3CC4C(C3)C24)CC#C)C1 17745,c1(C(N2C(C(=O)NCC(C)CC3CC3)C=CC2)=O)cc(F)ccc1O 17746,C1(NC(c2ccc3occc3c2)=O)CN(C(C2CC2CF)=O)CC2(CCC2)C1 17747,n1(CCOC)cc(-c2ccc(C(=O)NCc3cc(C#N)cs3)nc2C)ccc1=O 17748,c1(C(N2CCC(NC(C3(OC)CCCC3)=O)C(O)C2)=O)ccc(P(C)(C)=O)cn1 17749,c1(C(=O)NCCCOCCC(=O)NCC2(SCC)CC2)ccc(C)cc1C 17750,C(=O)(CCS(=O)(=O)N(C)C)N1CCC(C)(CNC(c2c(C)nccc2)=O)C1 17751,O(NC(=O)C(C)(C)N(C)C(=O)Nc1ccccn1)CCOCC#C 17752,C1(NC(C=Cc2nc(C)sc2)=O)CC(CNC(=O)CC2(O)CCOCC2)C12CCC2 17753,c1(OC)cnc(C(N2CCCC2CCNC(=O)C=C(C)C(C)C)=O)nc1 17754,N1(C(c2cn(CCC)nn2)C(=O)NC2CC2)C2CCC1CN(C)CC2 17755,C1(CC(=O)Nc2ccc(Br)nc2)COCCN1Cc1ccc(-c2ccncc2)o1 17756,CCCCC(C)(F)C(=O)N1CC(NC(C23CC(C)(C2)OC3(C)C)=O)C(O)C1 17757,C(=O)(C(CNC(=O)C1=CC2(CCOC2)C1)CC(C)C)Nc1c(COC)cccc1 17758,c1(C2(N(C(=O)Cn3cc(C(F)(F)F)cn3)C(C)C)CC2)ccnc2ccccc12 17759,C12(NC(c3c(OC)c(F)ccc3)=O)CCCCC1CN(C(=O)CC1CC13CC3)C2 17760,N1(C(Cc2ccn(CC)n2)=O)CC2(C1)CN(C(C1(C#N)CCSCC1)=O)C2 17761,N1(C(CSCC)=O)Cc2ccccc2CC1CNC(c1cc(Cl)ccc1OC)=O 17762,NC(=O)CCCC(=O)N1CCC(C2CCCCN2C(c2ccns2)=O)CC1 17763,CC1CCN(C(c2cccnc2N(C)C)=O)CC1NC(C1OCCC1(C)C)=O 17764,CCC(C)CCCCC(=O)NC(C)CNC(c1ccc(S(C)=O)cc1)=O 17765,CN1CCN(c2ccc(C(N3CC(NS(=O)(=O)CC4CC4)C(O)C3)=O)cc2)CC1 17766,c1(C(=O)NC(C)(CNC(c2ccco2)=O)CO)[nH]c(=N)sc1-c1ccccc1 17767,c1(N2C(=O)NC(CC(=O)C3CC3)C2)ccc(-c2noc(C3CCC3)n2)cc1F 17768,N1(C(c2c(C)c[nH]n2)=O)CCCC(NC(=O)Cc2ccsc2Cl)C1C 17769,c1(C(=O)OC)cc(S(=O)(=O)N2CCCC(S(N)=O)C2)ccc1OCC(F)(F)F 17770,CN1CCC(NCCOCCN(C(=O)C(c2ccc(Br)cc2)(C)O)C)CC1 17771,C1(C(=O)NCCOCCCC#C)CCN(C(C2CC(C)CCO2)=O)C1(C)C 17772,C1(C(N(CCN(C(C(C(C)C)(C)C)=O)C)C)=O)CCC2(C1)CC2(F)F 17773,C1(C2CC2)(CNC(c2c(CCC)n[nH]c2)=O)CCN(C(=O)CC(C)(F)F)C1 17774,C(=O)(CCCC(=O)NCC1(OC)CCN(C(C2CNC(=O)C2)=O)C1)OC 17775,C1(F)(C(=O)NCCC2(CNC(c3c(CC)nccn3)=O)CC2)CC2(CCC2)C1 17776,c1(C(=O)NCC(CNC(Cc2c(C)ocn2)=O)(C)C)cccc(OC2CCC2)c1 17777,c1(NC(CN2CCCC(C)C2)=O)ccc2nn[nH]c2c1 17778,C(=O)(C(CC)CCOC)N(CCC(=O)NC(c1ncc[nH]1)C)CC#C 17779,C12(F)CC3CCC(C1)N3C(=O)CN2.C1(CC(=O)NS(=O)(=O)C2CC2)CS(=O)(=O)C1 17780,Cn1cnc(NC2CC(NC(C3CCCC(n4ccnc4)C3)=O)C2)cc1=O 17781,c1(C(=O)NC2C(CNC(C(COC)(F)F)=O)CCCC2)cnc2c(n1)CCCC2 17782,c1(C(=O)NC2CCC(CC(C)C)C2)cccnc1CNC(=O)C1=CCCC1 17783,C1(C)(CCC(=O)NC2CC(CCNC(c3c(Cl)cc(C)s3)=O)C2)NC(=O)NC1=O 17784,S(=O)(=O)(c1cnc(C(C)C)[nH]1)N1CCC2(C(CC)C2)C1 17785,NS(=O)(=O)c1cc(C(=O)NCCCCNC(c2cncc(Cl)c2)=O)ccc1Cl 17786,c1(CC(N2CCC(C(C)C(=O)NC3CC(F)C3)CC2)=O)ccc2c(c1)CCCO2 17787,c1(C(N2CCC(N3CCN(C(CCSC)=O)CC3)C2)=O)c(C)cc(O)nc1C 17788,N1(C(CCC(C)N(C)C)=O)CCC=C(C(=O)N2CCC(C)(C#N)CC2)C1 17789,Cc1ccc(C2CC2C(=O)NCCCN(C(C2CC(Cl)(Cl)C2)=O)C2CC2)o1 17790,c1(OCC)ccc(SCC(N2CC(NC(=O)CCc3cn(C)cn3)C2)=O)cc1 17791,C1(N(C)C)(C(=O)NCC(CNC(=O)Cc2nc(C3CC3)cs2)CO)CCCSC1 17792,c1(C(N2CC(CCOC)N(C(C3CCCS3)=O)CC2)=O)ccc2cc[nH]c2n1 17793,C1(NC(CC2(C(=O)OC)CC2)=O)CCCCN(C(C2CC(F)C2)=O)C1 17794,N1(C(CC(C)OC)=O)CCCC(CC(=O)Nc2cccc(-n3cncn3)c2)C1 17795,c1(C(=O)NCCC2(O)CN(C(C3(Cl)C(C)(C)C3)=O)C2)oc2ccccc2c1Cl 17796,C1(C(=O)NCC2CC2NC(C2CS(=O)(=O)C2)=O)CCCC1C(F)(F)F 17797,C1(C)(C(N(C2CN(C(=O)CCc3cocn3)C2)C)=O)CCCCNC1=O 17798,CC(C#N)C(=O)Nc1ccccc1.C1C(C)CNC(=O)COCC(=O)O1 17799,C1(C(C)(C)C)(CNC(CC(C)SC)=O)CCN(C(c2coc(C(C)=O)c2)=O)C1 17800,C#CCCCC(C)C(=O)NCc1cc(C(N2CCCC(C)(C)C2)=O)cs1 17801,N1(C(C(CC)(C)C)=O)CCN(C(C2CCCC23CCC3)=O)C(C)C1 17802,c1(C(=O)NC2(C)CC(NC(C3N(C(C)=O)CC(O)C3)=O)C2)cc(O)cc(C#N)c1 17803,Cn1cnc(C=CC(=O)NC2CCCC2CNC(=O)CCc2cc[nH]n2)c1 17804,n1(CC)cc2ccc(C(N3CC4CCOC4(CNC(=O)CSC)C3)=O)cc2n1 17805,c1(C(=O)NC2CCCC(NC(=O)CCc3ccc(Cl)cc3)C2)c[nH]cc(F)c1=O 17806,c1(CCN(C)CC2(O)CCCNC2)nc2ccccc2n1C 17807,Clc1ccc(-c2cc(-c3nc(C4CCCC4)nn3C34CC(C3)C4)n[nH]2)cc1Cl 17808,c1(CNC(C2CC(C)(C)C2)=O)cccc(NC(=O)CCc2ccsc2Cl)c1 17809,C1(C)(C(=O)NCCNC(C(C)OC)=O)CC=C(C)CC1 17810,C1(C(=O)NC2(CO)CCN(C(C34CC(C)C3C4)=O)CC2)CN(CP(C)(C)=O)C1 17811,C1(c2cn(CCOCC)nn2)CN(C(=O)Cc2csc(C)c2C)CC1C 17812,c1(C(=O)NCC2CC(NC(CCn3c(C)ncc3)=O)C(O)C2)cc(F)ccc1C 17813,N1(C(c2ccc(OCCC)cc2)=O)CCN(C(C2CC(CCC)C2)=O)C(CC)C1 17814,c1(OC)cc(C(N2CCC(NC(=O)C=CC(C)(C)C)C(C(C)C)C2)=O)ccc1C 17815,c1(C(N2C(C)CN(C(=O)CN3CCOCC3=O)CC2)=O)cn2cnnc2cn1 17816,N1(C(C(C)C(F)F)=O)CCC(F)(C(N2CCC(C(C)(C)C)CC2)=O)CC1 17817,C(c1cccs1)=CC(=O)N(CC(CC)NC(=O)CC1CCOC1)C 17818,c1(C(=O)NCC2N(C(CC(CC)SC)=O)CCN(C)C2)cc(C)c(C#N)c(C)c1 17819,C=CCC(C(=O)NC(C=C)CO)NC(=O)C=CC1CCCN1C 17820,C1(CNC(CSCC=C)=O)CN(C(C2COCOC2)=O)CCC1C 17821,CN1CCCC12CCN(C(=O)COc1ccc(Br)cc1F)CC2 17822,C=C(C)C(C)(C)C(=O)NC1CCCC1NC(C1CCC(C#N)C1)=O 17823,CC1CC(NC(=O)Nc2nccc(-n3cccn3)n2)CCN1C 17824,c1(C(C)=O)c(C)[nH]c(C(=O)NCC2(O)CN(C(=O)C(C)N=[N+]=[N-])C2)c1C 17825,N1(C(COCCCCC)=O)CCC(CC)C1CNC(=O)Cn1cnc(C#N)n1 17826,C1(C(=O)NC2CC(CNC(C(Cc3ncn(C)c3)O)=O)C2)Cc2nccn2C1 17827,c1(NC(=O)C(C)(CO)CO)ccc(C(F)(F)F)cc1O.C12(CC=C)CN(C1)C2=O 17828,C1(COC)CN(C(=O)C(C)C#N)CCN1C(=O)CCc1cnc(O)[nH]1 17829,c1(NC(CSCC(=O)N(C)CCc2ccccn2)=O)ccc(Cl)cc1 17830,C(=O)(C1CCc2c[nH]nc21)NC1CCC(C(N(c2cccc(O)c2)C)=O)CC1 17831,C1(C(=O)NCC2CCN2C(=O)C(F)(F)CC2CC2)CCC([N+](=O)[O-])CC1 17832,CCC(CCOC)NC(C1CC(N(C(=O)C(C)OC)C)C1)=O 17833,Cc1nc(Br)oc1C(=O)NC(C)CNC(c1cc(C(C)(F)F)n[nH]1)=O 17834,c1(C2C(CC(=O)NCC(C3CC3)NC(C(C)=CCC)=O)C2)ccccn1 17835,C1(C(N(C(CCNC(c2ccc(OC)cc2)=O)C)C)=O)OCCOC12CCC2 17836,N1(C(c2n(C(C)C)ccn2)=O)C2CCCC1CN(C(C1CCCSS1)=O)C2 17837,CC1C(NC(c2ccc(N(C)C)s2)=O)CCN1C(=O)CC(F)(F)F 17838,N1(C(CC(CC)OC)=O)CCC(C2(O)CN(C(C3(CO)CCC3)=O)C2)CC1 17839,N1(C(c2ccc(C)nc2C)=O)CCC2C(CCN2Cc2cc(Br)cc(Cl)c2O)C1 17840,CCC(C)CC(=O)C(=O)N1CCOC(C(=O)NCC2(C)C=CCCC2)C1 17841,N1(C(C(=O)N(C)C)=O)CCCC2(C1)CN(C(c1c(F)cccc1F)=O)CCO2 17842,Cc1csc(C(=O)NCC(C2CCCC2)NC(=O)C(F)F)c1Cl 17843,c1(C(=O)NC(CC=C)CNC(=O)Cc2csc(=N)[nH]2)nn(C)c(Cl)c1Cl 17844,C1(C(=O)NC(COCCOC)C)C=CCN(C(=O)C(C)(O)C2CC2)C1 17845,C1(C)(CCNC(CC(C)OC)=O)CCN(C(c2ccc(SC)s2)=O)C1 17846,C1(NC(C=CSC)=O)CCN(C(=O)Cc2nccs2)CC1F 17847,O=C1NCCCCC1C(=O)NC1CC(CCC(=O)NCCn2cncn2)C1 17848,S(=O)(=O)(c1ccc(O)c(NC(=O)C(C(C)CC)N(C)C)c1)N(CC)CC 17849,N1(C(c2c(CC)nc(C)[nH]2)=O)CCC(CNC(C2(C#N)CC3CC3C2)=O)C(C)C1 17850,C1(C)(CNC(=O)COc2ccc(C(=O)NC3C(OC)C3)o2)CN(C(C)=O)C1 17851,c1(C(N2CCCC(c3ncc[nH]3)C2)=O)cccc(-n2cnnn2)c1 17852,c1(C(=O)NC2C(OC)CN(C(=O)C(O)C(F)(F)F)C2)cnc2[nH]ncc2c1 17853,c1(C(N(C2CN(C(C=CC(C)(C)SC)=O)CC23CC3)C)=O)ccn2ccnc2n1 17854,c1(OC)ccc2c(c1)CCC2C(=O)NC(c1ccccc1C)CF 17855,C#Cc1ccc(F)cc1C(=O)NCC(C)(C1CC1)NC(c1cccc(CC)n1)=O 17856,N1(C(CC)=O)CCCC(C(=O)NC(CNC(c2ocnc2C(F)F)=O)C2CC2)C1 17857,N(C1CC2(CC2)Oc2ccccc21)C(C1(F)CCS(=O)(=O)C1)=O 17858,C12(CNC(CC3(C#N)CC3)=O)CC1CN(C(=O)C=CCO)C2 17859,c1(CNC(CSC(C)C)=O)cccc(C(=O)Nc2ccc(C(N)=O)nc2)c1 17860,Cc1cc(C)c(C(N2CCC(N(C)C(c3cn(C(C)(C)C)nc3C)=O)C2)=O)cn1 17861,CCCCCC(=O)N(CCCNC(c1ccc(-c2nc(C)no2)cc1)=O)C1CC1 17862,N1(c2ccnc(C(C)C)n2)CCCC(C(N2CCC(C)(O)CC2)=O)CC1 17863,C1(NC(C2(CC(C)C)CCC2)=O)CN(C(c2sc(C)nc2C)=O)CC1C.CC 17864,CC#CCCCC(=O)NCC1(F)CC(NC(=O)Cc2noc(C)c2C#N)C1 17865,N1(C(C=NOC)=O)CCC(C2CC2)(CNC(c2cccc(NS(C)(=O)=O)c2)=O)C1 17866,C1(NC(C2(CC)CCN(C(c3ccc[nH]3)=O)C2)=O)CCC(C)(C)CC1COC 17867,C1(CC(=O)NC)CN(C(c2cc(C(C)=O)[nH]n2)=O)CCN1C(=O)C(C)C(C)O 17868,N1(C(CC(CC#C)NC(C2CC(=O)C23CCC3)=O)=O)CC2(C1)OC(=O)NC2C 17869,C1(CC)CCCN(C(C2CCN2C)=O)C1C(=O)N(C1COCC1O)C 17870,Cc1cc(C(N2CCC3(C2)CN(C(=O)C(C)C(F)(F)F)C3)=O)c(Br)c(C)c1 17871,c1(NC(C2N(C(CCc3ccc(C)cn3)=O)CC2)=O)ncc([N+](=O)[O-])cc1I 17872,c1(C(=O)NC(C(C)NC(C2CCOCC2(C)C)=O)CO)cc2cc(Cl)cnc2[nH]1 17873,c1(Cn2cc(COC)nn2)cc2cc(C)cc(C)c2[nH]1 17874,CC1CN(C)C(C)CN1C(=O)CC1CC2CCC1C2.C1(N)CC2CNC1C2 17875,c1(C(N2CCC(C)(CNC(CC3C=NN(C)C3=O)=O)C2)=O)cc2ccncc2o1 17876,Cc1ccc(NC(C2(Nc3ccc(-c4ccc(Br)cc4)cc3)CCC2)=O)c(O)c1 17877,N1(C(C2CCCC(C3CC3)O2)=O)CCC2(CCCN2C(=O)CC2OCCO2)CC1 17878,c1(C(=O)NC2C(C(N(C3CCC(CO)CC3)C)=O)COCC2)ncnc(O)c1F 17879,C1(C(=O)NCC2CC(NC(C(Cn3ccc(C)n3)C)=O)C2)CCC(=O)NC1 17880,C1(CC(=O)NCC2C(NC(COCC(C)C)=O)C2)CC(OC(C)(C)C)C1 17881,c1(C(N2C(CC)CCC2)=O)ccc(OCC(C)NC(=O)C(=O)NCC(C)C)cc1 17882,c1(C(=O)NC(C(C)NC(C(CC#C)C2CC2)=O)(C)C)[nH]cc2c1CCCC2 17883,c1(C(N(C)CCC2CCCCN2C(=O)CC2CCOC2)=O)cc2sccc2[nH]1 17884,N1(CC(=O)N(C(c2ccc(F)cc2)C)CC)CCC(C)(O)C(O)C1 17885,C1(C)(C(=O)NCC2CN(C(C(c3ccc(Cl)s3)C)=O)C2)CC2CC2C1 17886,CCCC(C(=O)OC)N1CC2C(C1)N2C(=O)C(Cc1cnc[nH]1)NC(C)=O 17887,c1(NC(C2C(CCC)CN(C(=O)C(C)(O)C3CCC3)C2)=O)ccc2c(c1)OCO2 17888,N1(C(CCSC)=O)CCN(C(C2(CO)CCC2)=O)CC1c1ccccc1Cl 17889,c1(OC)nc(Cl)ccc1C(=O)NC(C)CC1CN(C(=O)C(c2ccc(Cl)s2)C)C1 17890,c1(NCC=CC)[nH]c(=NC(CCO)CC(C)(C)C)nc2c1ncn2C 17891,C1(O)(C(C(=O)N(CC=C)C)N(C(=O)CC2(N(C)C)CCC2)C2CC2)CCCCC1 17892,C#CCC(CC(F)F)C(=O)N1CCC1CC(=O)NCCN(C)CCO 17893,c1(N(C(CNC(C(C(C)C)OC)=O)C)C)cc2nnc(-c3ccccc3)n2cn1 17894,C(=O)(C1Cc2c(Cl)cccc21)NCCC1(C)CCN(C(CCCOCC=C)=O)C1 17895,c1(NC(C=CC2N(C(CN3CCC(OC)C3)=O)CCC2)=O)ccc(Cl)nc1C 17896,N1(C(C(C=C)(C)C)=O)CC(NC(c2cc(CC(C)C)on2)=O)CC2(CCC2)C1 17897,N1(C(c2n(CC)ncc2)=O)CCOC(C)(CNC(c2nn(C)nc2Br)=O)C1 17898,C1(CNC(=O)NC(C)COC(F)(F)F)Cc2ccc(F)cc2C1 17899,C12(C(N3CCC4(NC(=O)C=Cc5ccco5)C(C3)C4)=O)CCC(F)(CC1)CC2 17900,Cc1ccc(CO)cc1NC(C1COCCC1NC(=O)C(C)C)=O 17901,N1(C(C2N(N=O)CCC2)=O)CC(F)(F)CC1CCNC(c1ccccc1CO)=O 17902,C1(C(N2CCC(C)C2)=O)C2C3CCC(C3)C12.C1(=O)CCC2(CCC2)N1 17903,Cc1ccc(Cl)c(C(=O)NCC2CCCCN2C(=O)Cc2cc(C)ccc2C)c1 17904,c1(C(C)C)ccc(C(=O)NCC2C3CCC(C3)N2C(C2(C)CCOC2)=O)c(F)c1 17905,c1(C(=O)NCC2C3CN(C(CC(C)NC(N)=O)=O)C2C3)cc2cccnc2o1 17906,c1(-c2ccc(SC)cc2)c[nH]c(=NCc2ccc(C(=O)O)cc2F)s1 17907,N1(C(C(CC)NC(N)=O)=O)C(C(N2CCC(CO)C2(C)C)=O)CCC12CC2 17908,Cc1ccncc1-c1cn(C2CCCN(C(C3CCC(C(=O)O)O3)=O)C2)nn1.C 17909,Cn1c(C(N2CCCC3C(=O)NCC23)=O)c(Cl)c2ccccc12 17910,N1(C(c2cccnc2)C)CC2CC(C1)N(C(=O)Cn1nc(C)cc1C(F)(F)F)C2 17911,N1(C(COCCSC)=O)CC(C)(NC(=O)Cc2csc(S)n2)C1 17912,c1(C(=O)NCCCCCNC(c2cncc(N)n2)=O)ccc(S(N)(=O)=O)cc1Cl 17913,c1(CC)cc(C(=O)NCCNC(=O)COCc2cccc(C)c2)nn1C 17914,C1(C(=O)NC(c2cnc(C)s2)C)CCC(C)(C)N(C(=O)CC2=CCCCC2)C1 17915,c1(OC)ccc(OCCOC(C2CCCOC2)=O)cc1 17916,N1(C(C=Cc2nc(C)sc2)=O)CCCCC1C1CCCN1C(=O)C(O)C1CCC1 17917,C(=O)(C(C)(C)C(=O)c1ccccc1)NCC(CC=C)NC(=O)CSCCN(C)C 17918,c1(C(=O)NCCNC(c2n(CC=C)ccc2)=O)cc(Cl)ccc1F 17919,C1(O)(CNC(C2C(COC)CC2)=O)CCN(C(C2C=CCS2)=O)CC1 17920,c1(C(=O)NCC(C)NC(c2cn(C3CCOC3)nn2)=O)cc2ccsc2s1 17921,C1(C#N)(C(=O)OC)CC2CCC1CC2NC1CCCC1c1ccccc1 17922,C1(C(=O)NC2(C(COC)O)CC2)CC2CC1CN(C(=O)Cn1ccnc1C)C2 17923,CC(C(=O)NCC1CCN(C(=O)Cc2cncs2)CC1CO)C(F)(F)C(F)F 17924,c1(C(=O)NCC(CO)NC(c2cnc(O)c(F)c2)=O)cc2cn[nH]c2cn1 17925,C1(NC(C2N(CC#C)CCC2)=O)CC2(CCCN(C(=O)C(F)C(C)(C)O)C2)C1 17926,C=C1CCN(C(c2ccnc(OC)c2)=O)C(C(=O)NCCOCCF)C1 17927,c1(C(N2CCC(OCC(=O)NCCCCN=[N+]=[N-])C2)=O)ccc(O)cc1F 17928,CNS(=O)(=O)NCC(=O)NC1CC(CNC(c2coc(C(F)(F)F)c2)=O)C1 17929,C1(CC(C)C)CCCN(c2cccc(C(F)(F)F)n2)C1.N1CCCC1 17930,N1(C(C2CN(C(C)=O)C2)=O)CC(O)CC1(C)C(=O)NCCCC(C)(F)F 17931,Cn1cccc(-c2ncc(Cl)cc2C(N2CCCC(O)C2C)=O)c1=O 17932,C1(O)(C(C)NC(C2C(CC)CCC2)=O)CCN(C(C2CN(C)C(=O)N2)=O)CC1 17933,n1(CCNC(c2nnnn2CCCF)CCc2cn(C)nc2)cc(Br)ccc1=O 17934,C(c1ccc(F)cc1)=C(C)C(N1CCC(C)(NC(=O)CN2CCCCS2(=O)=O)C1)=O 17935,c1(C(=O)O)ccc(OC(F)F)cc1Cl.n12cc(nn1)CNC1CC2C1 17936,C(=O)(C(C)CC(F)F)N1CC(OC)C(NC(=O)C=C2CCCC2)C1 17937,N(C(=NCCCN1CC(C)OC(C)C1)N1CCN(C2CC2)C(=O)C1)CC(=C)C 17938,c1(OC2CCCC2)ccc(C(=O)COCCn2cc(C(CC)(C)O)nn2)cc1 17939,C=CC(C)(C)CC(=O)NC(C1CCN(C(=O)C(Cc2cccc(Cl)c2)=NO)C1)C 17940,Cc1ccn(C)c1C(N1CC(C(C)NC(=O)CCc2ccnc(Cl)c2)C1)=O 17941,C(=O)(C1=CCC2CCC1N2C(=O)C(Cl)Cl)NC(C)Cc1ccco1 17942,c1(OC)cc(Br)ccc1-n1cc(CN(C)CC2CC2)nn1 17943,c1(OC)cc(CC(=O)NC2CCC(NC(=O)CSS(C)(=O)=O)C2)c(F)cc1O 17944,C1(NC(CCCC#C)=O)CCCC12CN(C(c1cccnc1OCCOC)=O)C2 17945,C1(NC(CN(CC)CC)=O)CC2(C1)CC2NC(c1cnn(-c2ccccn2)c1)=O 17946,C1(CNC2CC(CNC(C3(OC)CCC3)=O)C2)CCCC1C 17947,c1(C(=O)NCC2C(NC(CC(C=C)C)=O)CC2)ccc(CC)c(N)c1 17948,C1(NC(C2(C)CC2(F)F)=O)CN(C(=O)CCc2cccc(O)c2)CC1F 17949,c1(-c2scc(C)n2)ccc(C(=O)N(C2CN(C(C3(C)CCCN3C)=O)C2)C)cc1 17950,c1(C(=O)NC2(CNC(CCC(CC)C)=O)CCOC2)cnc2ccccn12 17951,N1(CC(=O)N(c2nc3ccccc3s2)CC)CCC(C2CC(F)(F)C2)C1 17952,c1(CNC(=O)NC2CC(C(C)C)OCC2)cnc2n1CCC(CO)C2 17953,CC1CN(C(c2cn(CCNC(=O)C(C)(Cl)Cl)cn2)=O)CC1(C)CO 17954,C(=O)(CCCC(F)(F)CO)NC1C(SC)CN(C(c2c[nH]nc2[N+](=O)[O-])=O)C1 17955,N1(C(c2ccc(Br)cn2)=O)CCC(F)C(NCc2cc(O)cc(F)c2)C1 17956,N1(C(C2C(C)CCO2)=O)CCC(F)(C(N2CC(CC3CC3)C2)=O)C1 17957,N1(C(=O)Nc2cn(CCC#C)nc2)CCC(O)C(O)CC1 17958,CC1CC(C(=O)N(C(C)CNC(=O)C=Cc2ccc(=O)oc2)C)CC(=O)N1 17959,N1(C(CC2CC(=C)C2)=O)CC(NC(c2cncc(C3CCCCC3)c2)=O)C(C)C1 17960,C1(C(C)NC(=O)Cc2cnc[nH]2)CCCCN1C(c1ccc(C2CCC2)cc1)=O 17961,c1(OC)ccccc1Cn1cc(C2(O)CN(CC(C3CC4CC4C3)=O)C2)nn1 17962,CC1(C)C(CC(=O)NCC2(C#N)CC2)CCN1C(c1nc(C2CC2)cs1)=O 17963,C1(CCNC(Cc2ccc(C)o2)=O)CCCN(C(=O)C=C2CCC2)C1 17964,C1(C(N2CC(C#N)C2)=O)CC(OC)CCN1C(C1CC2CCC(C1)C2)=O 17965,c1(CN(N2CCC(F)(CNC(C)(C)C=O)C2)C)ccc(Cl)c([N+](=O)[O-])c1.CC 17966,N1(C(CC2CC(CC)C2)=O)CC(C)N(C(=O)CN2CSCCSC2)CC1C 17967,c1(CC(=O)NCC(C)NC)ccc(NC(=O)NC)c(C)c1 17968,C(=O)(C1(C)CCn2c(C)nnc21)N1CCC(N(C(C(CNC(C)=O)(C)C)=O)C)C1 17969,c1(C(=O)NC2CCCC3CN(C(CCSC)=O)CC32)cccc(S(N)(=O)=O)c1C 17970,N1(C(C2(C(C)C)CC2)=O)CC(NC(c2sncc2Br)=O)C2(CCC2)C1 17971,c1(NC(C2(C)CCN(C(C(C)(C)F)=O)CC2)=O)c(F)cccc1C#N 17972,Cc1cccc(C(O)C(=O)NC(C)CN(C)C(C2CC3C=CC2CC3)=O)c1F 17973,C1(NC(c2cc(CCC)[nH]n2)=O)CC2CC1CN(C(=O)C(C)(CC)OC)C2 17974,C1(CC(N2C(CNC(=O)C(F)C3CC3)COCC2)=O)CC(=O)NC(=O)C1 17975,c1(C(N2C(CNC(c3ccn(C)n3)=O)CCCCC2)=O)c[nH]c2cc(O)ccc12 17976,N1(C(C(Cc2ccccc2)OC)=O)CCC2(C1)CN(C(=O)C(O)C(C)C)C2 17977,N1(C(c2cc(CC)oc2C)=O)CC(C)N(C(c2cn(C)c(C)cc2=O)=O)CC1C 17978,CCC1=NOC(C(=O)NCCC2(NC(c3cnc(CC(C)(C)C)s3)=O)CC2)C1 17979,c1(CNC(CCC(C)NC(C2CCCCCN2C)=O)=O)cccc(C#N)n1 17980,C(=O)(CC1c2ccccc2CCN1S(C)(=O)=O)NCC1N(C(CC=C)=O)CC1 17981,N1(C(C2CCC(CC)CC2)=O)C(CNC(c2cc(Cl)cnn2)=O)CC2COCC12 17982,N1(C(c2ccc(C)cc2)=O)CC2(CC(NC(c3cnc(N)c(N)c3)=O)C2)C1 17983,C1(Cn2cc(-c3c(CC)cccc3)nn2)CCN(C(=O)C(F)(F)Cl)CC1(F)F 17984,N1(C(C(CC#C)CC#C)=O)CCC2(CC1)CN(C(C13CC1CCC3(F)F)=O)C2 17985,N1(C(C(COC)C)=O)CCOC2(CCN(C(C3CC(=O)C3)=O)C2)C1 17986,c1(C(=O)NCC(C)N(C)C(c2cc(C3CC3)ncn2)=O)cccc(C2(F)COC2)c1 17987,CCCC(CCC)CC(=O)NCC1CN(C(c2cnn(CC)c2)=O)CCC1C 17988,n1(C(CC)C)cc(CN(C)CC2CN(C(=O)OC(C)(C)C)C2)c(C)n1 17989,N1(C(c2c(OC)cccc2F)=O)CC(NC(C2(F)CCOC2)=O)CC2(CCC2)C1 17990,CC1CCCn2cc(C(=O)NCC3CN(C(C4CN(S(N)(=O)=O)C4)=O)C3)nc21 17991,CCC(O)(C(=O)NCCCCC(C)NC(c1nc(C)cs1)=O)c1ccccc1 17992,c1(NC2CCCC(CO)C2)nccc(=NCc2ccc(Cl)c(C(F)(F)F)c2)[nH]1 17993,CN1CC(NC(C2CC23CC(NC(=O)CC2CCC(=O)NC2)C3)=O)C(C)(C)C1 17994,C1(C(N2CCCC(CN(C(=O)CC(C)(C)C)CC)C2)=O)CC12CCOCC2 17995,Cc1cc(Cl)cc(C(=O)NC(c2ccc(Br)cc2)CC2CCCC2)c1N 17996,N1(C(C(C)NC2CC2)=O)CCCN(C(=O)C(C2CCCCC2)N(C)C)CC1 17997,c1(C(=O)NCCCN(C(c2c(C)ccnc2)=O)C)c(C)nc(O)nc1S 17998,n1(CC)nc(C(=O)NC2(C3CCCN3C(=O)CCCCNC(C)=O)CC2)c(Br)n1 17999,c1(CC(N2C(CNC(C3(C#N)CCCO3)=O)CC2)=O)cc(F)ccc1Cl 18000,CC(C)CC(O)CNC(C1CCC(C2CC2)N1C(c1cnns1)=O)=O 18001,N1(CC)CCN(C(=O)CCC(=O)C(C)(C)C)C(=O)C12CCCCC2 18002,N1(C(CC(C=C)CC)=O)CC2(CNC(=O)CCc3cncnc3)CC1CCO2 18003,c1(CC(=O)NCCC2(O)CN(C(c3c(C)coc3C)=O)C2)cccc(Cl)c1Cl 18004,C1(C(N(CCNC(C(c2ccc(OC)cc2)CC)=O)C(C)C)=O)CSCC(=O)N1 18005,C1(NC(c2conc2C2CCCO2)=O)CCCN(C(C2CC=CCC2)=O)C1 18006,c1(C(N2CC=CC(NC(C3CC(CC)OCC3)=O)C2)=O)cc2nc[nH]c2cn1 18007,C(c1ccc(C)c(C)c1)=CC(=O)NC(CCOC)CNC(=O)C(C)C1CC1 18008,c1(C(=O)NCC(C)N(C(C(CCC)CC)=O)C)ccc2c(c1)CN(C)CC2 18009,C=CCC(C(=O)NCC1(CN(C)C(C2CCC3CC3CC2)=O)CC1)C(C)C 18010,C(=O)(C(C)(F)C(C)(C)F)NCCC(CNC(CCCCOCCC=C)=O)O 18011,Cc1cc(Cl)cc(C(=O)NC2CC3CCCCN3C2)c1O 18012,C(C(CC(=O)NC1CCN(C(C2CCCS2)=O)CC1)C(F)F)N(C)C 18013,C1(NC(CCOc2c(CC)cccc2)=O)CCCCN(C(c2cnns2)=O)C1 18014,C=C(Cl)CC(C(=O)N1CCC1CO)NC(c1nnn(C)c1C)=O 18015,C(=O)(C(C)(C)C(=O)NC1CCCN(C(c2cc(Cl)sc2Cl)=O)CC1)NC 18016,C1(NC(c2c(CC)oc(C)c2)=O)CN(C(c2cocn2)=O)CC12CC2 18017,C(=O)(C1=CCSC1)NCC(C1CCCCC1)NC(CC(C)OC)=O 18018,N1(C(c2c(SC)cccc2)=O)CCC2CC1CN2C(=O)C(O)Cn1cncn1 18019,C1(CNC(c2c(C)nco2)=O)C(C2CC2)CCN1C(=O)CC1CC12CC2 18020,N1(C(C2=CCCC2C)=O)CCC2CCCCC2C1.N1(C(=O)OC(C)(C)C)CCCCC1 18021,C1(C(=O)NCCC(C)NC(=O)CCN2CCC(F)C2)CCN(C(=O)C2CC2)CC1 18022,C1(NC(CCC#CC)=O)CCSC12CN(C(=O)CCOc1cccc(C)c1)C2 18023,C=CC1(C(N2CC(C3C(C(=O)OC)C3)C2)=O)CCN(C(=O)C(C)CC(N)=O)CC1 18024,CC1(C)CC(SC(=O)NOCC(C2CCOC2)O)C1 18025,C1(CNC(C(c2cn(C)nn2)NC(=O)CCc2cnoc2)=O)C2CCC(F)C12 18026,N1(Cc2nc(N(C(C)=O)C(C3CCCC3)=O)sc2)CCCCC12CCCCCC2 18027,C12(NC(c3n(C)ccc3)=O)CN(C(C3CCOCC3)=O)CC1CS(=O)(=O)C2 18028,C1(NC(C(C2CN(C(C3(CC)CCCO3)=O)C2)O)=O)CCCCCC1C 18029,Cn1ncc(C(=O)NCCOCCOCCCNC(=O)CCc2ccccn2)n1 18030,CCCCCCCC(=O)NCC(C)(O)CNC(C1CNC(=O)CC1(C)C)=O 18031,c1(NC(C2(NC(C(C)N=[N+]=[N-])=O)CC2(C)C)=O)ccc(O)c(F)c1 18032,c1(C(N2CC(NC(=O)CCC3CCCC(O)C3)(CO)C2)=O)cccc2ncoc12 18033,Cc1oc2ccccc2c1C(N1CC(NC(C2CCCCN2C)=O)CC1(C)C)=O 18034,c1(CCC(=O)NCC2C(NC(C(C)OC(C(C)C)=O)=O)C2)ccc(Br)nc1 18035,C1(C(=O)Nc2cccc(C(F)F)n2)CC(O)CCN1C(c1cccc(Cl)c1Cl)=O 18036,Cc1ccc(OCC(=O)NCCOCCNC(C2CNC(=O)CC2C)=O)c(C)c1 18037,CC1CN(C(=O)C(F)CC2CC2)CC2(CCN(C(c3cc(O)nc(O)c3)=O)C2)O1 18038,C(=O)(CC(C)C(F)F)N1CCC(CNC(CNC(c2c(C)occ2)=O)=O)C1 18039,Cc1ccc(Cc2nc(-c3ccc(Br)cn3)nn2CC(N)=O)c(C)c1 18040,C1(NC(CC(=C)I)=O)CC(C)CN(C(c2ccc(C)nc2)=O)C1 18041,c1(-c2cn(C3CCN(C(C4CCCO4)=O)C3)nn2)ccc(Cl)c(Cl)c1 18042,CC(C)(C)CCC(F)C(=O)N1CCC(N(C(=O)CSCC(N)=O)CCO)C1 18043,c1(NC(C2CC(NCc3c(Br)cc(F)cc3Br)C2)=O)cnc2ccccc2n1 18044,C1(CC(=O)N(CCCO)CC#C)CN(C(=O)C(C)c2cc[nH]n2)CC12CC2 18045,CCC(C)(CO)C(=O)NCC(F)CNC(=O)CN1CCOC1=O 18046,C1(C)(CC(=O)N(CC(=O)N(CCOC)C(C)C2CC2)CCC)CC1(F)F 18047,C1(C(=O)NC(c2cc3cnccc3[nH]2)C)CCC2(CCCC2)C1 18048,C1(O)(C(=O)NC2CCC(NC(C3=NOC(C)C3)=O)CC2)CCCC(C)(C)CC1 18049,Cc1cc(C)c(C(=O)NCC(CC(C)C)NC(=O)CSc2ccccn2)c(Cl)n1 18050,C1(CNC(C2(CC#C)CC=CCC2)=O)N(C(=O)Cc2cnsc2)CCC1(C)C 18051,C1(NC(C2(Cl)C(C)(C)C2)=O)CCCN(C(c2nc(=N)cc[nH]2)=O)C1 18052,c1(C(=O)NC2CCC(C)(NC(C=CCCC)=O)CC2)cc2c(C)ccc(C)c2[nH]1 18053,c1(C(C)=O)csc(C(=O)NCC2(O)CN(C(C3CC3(C)C)=O)C2)c1 18054,N1(C(C(COC)OC)=O)CC(NC(=O)CC2CCN(C)CC2)CC1(C)C 18055,N1(C(C(=O)NC(C)C)=O)CC(NC(=O)Cc2ccccc2Cl)CC12CCC2 18056,C1(NC(C(C)n2ccnc2)=O)CC(F)(F)CC1NC(c1ccc(C2CC2)o1)=O 18057,c1(OC)cc(C(=O)NCCCC(C)(C)NC(=O)CC(C)O)ccc1C 18058,c1(C(=O)NC2C(CNC(=O)CCC3CCCCO3)CCC2)cc(Cl)cnn1 18059,C1(NC(Cn2c(C)cnc2)=O)CN(C(=O)CCCSc2ccccc2)CC1C 18060,S(=O)(=O)(c1ccc(F)cc1)N(c1ccccc1)CCC(=O)OCC 18061,c1(NC(C2C(CC)N(C(c3cc(O)nc(O)n3)=O)CC2)=O)cc(C)cnc1C 18062,c1(C(=O)Nc2cccc(NC(CC(C=C)CC)=O)c2)cc2cccnc2o1 18063,C1(NC(=O)Cc2cnnc(O)c2)CC2CC1N(C(=O)COCCN1CCCC1)C2 18064,c1(NC(C23CC(NC(c4ncc(C(C)(C)C)cn4)=O)(C2)C3)=O)cccc(Br)c1Cl 18065,C(=O)(C(C)(C)C(C)(C)O)NC(CNC(C1CCN(CC)C1)=O)C(C)C(C)C 18066,C(=O)(CC(C(F)F)NC(=O)CC1CCSC1)NCCCCC 18067,C(=O)(C1=CCCCO1)N1CC(NC(Cc2c(C)oc(-c3ccco3)n2)=O)C2C1C2 18068,CC1(C)CC(CCNC(N2CC(Cc3cccs3)C2)=O)C1 18069,C1(C(=O)NCCCC(C)NC(C2(COC)CC2)=O)CN(C(C)C)CCO1 18070,Cc1nc2c(Cl)cccc2cc1C(=O)NCCN(C)C(C1CNC(=O)N1)=O 18071,c1(C(N2CC(O)(CCNC(c3c(CC)ocn3)=O)C2)=O)c(C)cc(Cl)nc1N 18072,C1(N(C(c2nccc(CNC(C3CCC(C)O3)=O)c2)=O)C)CCCCC1(C)O 18073,C1(NC(C2CCCC2)=O)CCOC12CCN(C(C1COC3COCC13)=O)CC2 18074,c1(C(=O)NCC(CNC(C(C=C)(C)C)=O)CO)ccc2c(c1)OCCC2 18075,C1(CNC(C2CCN(c3ncccn3)C2)=O)CC2(CC2)CN1C(=O)C1=NOCC1 18076,N1(C(C2CC(=O)NC2)=O)CCOCC(F)(CNC(=O)Cc2cnn(C(F)F)c2)C1 18077,c1(C(=O)NC(C(C)NC(CCN(C(CCC)C)C)=O)C)cc(C)nc(O)n1 18078,c1(OCC)ccc(C(=O)N(CC(C)NC(=O)Cc2nncn2C(C)C)CC)cn1 18079,N1(c2n(CCc3onc(C)n3)nnn2)CCC2(CCOC2=O)C1 18080,CCCCC(CCCC)C(=O)NC(C)CNC(C1CCC(F)(F)C1O)=O 18081,N1(C(c2ncc(C(C)(C)C)s2)C(=O)NCCCC)CC(OC)CC(O)C1 18082,C(=O)(C1CCCn2cc(C)nc21)N1CCC(NC(c2cc(OC)no2)=O)C1 18083,N1(C(C(=O)N(CCOC)C(C)C)=O)CCCCCC(NC(C2CC23CC3)=O)C1 18084,N(C(=NCCCP(C)(C)=O)NCC(c1ccccn1)C)Cc1ccc(OC)cc1 18085,C1(CNC(C2(OC)CCSCC2)=O)C2CCCC1N(C(c1nc(=O)n(C)[nH]1)=O)C2 18086,CN1CCC(C2(C(=O)OCC(C)(C)CCl)CC2)CC1 18087,CC1CCC(C(=O)NCCCN(C)C(c2ccc(Br)c(O)n2)=O)C(=O)N1 18088,N1(C(C(CC2CCC2)NC(C2CN(C)C(=O)C2)=O)=O)CCN(C)C2(CCC2)C1 18089,c1(C(=O)NC2(CF)CN(C(C3OCC(C)C3)=O)C2)ccc(C#N)c(O)c1 18090,CCC(C(C)C)NC(c1[nH]ccc1CNC(C1COC(=O)N1)=O)=O 18091,c1(N(C)CC2CCN(c3ncncc3I)C2)ccc(Cl)c(F)c1 18092,C(=O)(C(O)P(C)(C)=O)N1CCCC(N(C(CS(N2CCC(C)CC2)(=O)=O)=O)C)C1 18093,c1(OC)c(C(=O)NC(C)CCCCNC(c2c(C)ncn2C)=O)cc(F)cc1F 18094,CC1(C)CC(NC(C2CC3(CSC3)C2)=O)Cc2ccc(Br)cc21 18095,C1(CCNC(C(CC)N(C)C)=O)CCCN(CC(=O)N(c2cnccn2)C)C1 18096,N1(C(=O)CSCc2ncc[nH]2)CCCC(NC(=O)CC2CC3(CC3)CO2)CC1 18097,c1(C(=O)NC2CC(NC(c3cc(OC)ncc3F)=O)C2)cccc(C=C(F)F)c1 18098,c1(C(N2CC(NC(c3c(NC)nccc3)=O)C2)=O)ccc(-n2ccnc2)cc1C 18099,N1(C(Cc2nc(C)sc2)=O)CC2(CNC(C3CCSC3)=O)CC1CO2 18100,O=C(C1=Cc2ccccc2OC1)N1CCC(CNc2ccccn2)C1 18101,CC(C)C(C(=O)NC(C1(C)CN(C(=O)C(=O)NCC2CC2)C(C)(C)C1)C)C(C)C 18102,C1(C(=O)NCCCOCCCNC(C2C(C(C)(C)C)C2)=O)CCS(=O)(=O)CC1 18103,C(=O)(C(C)CC(F)F)N1CCC(N(C(=O)C=Cc2ccccc2)CC#C)C1 18104,C1(C(=O)NCCCCN(C)C(C2CCCCC(=O)N2)=O)C2CCC3C(C2)CC13 18105,N1(C(CC(C)SC)=O)CCC2(CCCN(C(c3scc(Cl)c3Cl)=O)C2)C1 18106,C(C(C)(O)C(=O)N1CCC(N(C)C(c2c(C)noc2N)=O)CC1)OC 18107,Cc1ncsc1C(=O)NCC(O)CN(C(=O)C(c1ccccc1)C1CC1)C1CC1 18108,C1(C(C)N)CCN(C(=O)C(=O)NCC(c2ccccc2)CC2CCOCC2)C1 18109,c1(C(=O)NC(CCNC(CCC=C)=O)(C)C)nnn(Cc2ccccc2)c1N 18110,c1(C(=O)NC(CC(C)NC(CNC(=O)NC)=O)C)cc(C(C)C)ccc1F 18111,CN1C2CCCC1CN(C(=O)C(C1CCN(C(C3CC3C(N)=O)=O)C1)F)C2 18112,N1(C(COCC(=C)C)=O)CC=CCC1C(=O)NC1CC(C)OC1=O 18113,C(=O)(CC(O)C(C)CC)NC1(CC=C)CCN(C(=O)CC2OCCCO2)CC1 18114,C(=O)(CC(COC)N(C(=O)COCCCC(C)C)C)N(C(C=C)C1CC1)C 18115,n1(CC2(CC)CC2)nncc1C(N1CCC(C(=O)NOCC(O)C(C)C)C1)=O 18116,c1(OC)c(C(N2CCC(NC(=O)COC3CCCOC3)C(O)C2)=O)ccnc1F 18117,C1(S(C)(=O)=O)(C(=O)Nc2c(CN3C4CN(CC)C(C4)C3)cc(Br)cc2)CCCC1 18118,OCCCCCN=C(NCC1CCCCO1)N1CCC(c2ccncn2)CC1 18119,N1C(=NCCC)NCc2ccc1cc2C(F)(F)F.C#CCCC1(CCOC)N=N1 18120,c1(COC)ccc(NC(=O)Cn2cnc(Br)n2)nc1 18121,c1(CC)nc(C(=O)N(CC(N2C(CO)CC2C)=O)CC2CC2)co1 18122,N1(C(c2c(COC)cco2)=O)CC2CC1CN2C(c1cc(C(C)C)on1)=O 18123,CC1CN(C(=O)CC2CC(O)CN2C(=O)CCCn2cncn2)CCS1 18124,Cc1nc(Cl)ccc1CC(N1CC(OC2CCN(C(=O)C(C)C3CC3)CC2)C1)=O 18125,c1(C(=O)NCC(CN(C(C2CN(C)C(=O)N2)=O)CC)(C)C)cc2[nH]ccc2s1 18126,C1(CNC(c2c(C)coc2C)=O)CC(C)(C)CCC1NC(=O)CC1CCOCC1 18127,c1(NC(CN2CCCC(c3nc(C)no3)(OC)C2)=O)cccc([N+](=O)[O-])c1O 18128,C1(NC(C(CC)(C)C)=O)CC2CN(C(=O)C=Cc3ccn(C)c3)CC2C1 18129,C1(NC(c2ccc(CN(C)C)[nH]2)=O)CCCC(CNC(=O)Cn2nccn2)C1 18130,N1(C(COCCOC)=O)CC=C(C(=O)NC2(CCO)CCOC2)C1 18131,C(C(C)(C)CNC(c1ccc(CNC(=O)CSCCC(F)(F)F)o1)=O)N(C)C 18132,C1(C(=O)NC2CC(N(C(c3ncn(CC)c3)=O)C)C2)CC(C(C)C)=NO1 18133,c1(OC)cc(F)c2c(C(=O)NCCCn3c(C)cccc3=O)n[nH]c2c1 18134,O=S(=O)(c1[nH]c(=NCC(O)c2ccncc2)ccc1Br)NC1CCCC1C1CC1 18135,N1(C(C(C(C)C)(C)C)=O)CC2CCOCC2(NC(=O)COc2ccc(Cl)cc2)C1 18136,C(=O)(CCCC(C)(C)C)N(C1CCN(CCC2CCCCO2)CC1)CCC 18137,C1(NC(c2ccc(OCCCOC)cc2)C)CCCC(C)(C)C1 18138,c1(C(=O)NC(CCC)CNC(c2cnc(COC)s2)=O)cncc(Cl)c1 18139,C1(NC(C=C2CCC(C)CC2)=O)CCC(C)(CNC(=O)Cc2[nH]cnc2C)CC1 18140,N1(C(c2c(OC)nccc2)=O)CCCCC2(CCN(C(c3cc(N)ccn3)=O)C2)C1 18141,c1(C(N2CCC(NC(COCCCCCC)=O)(CF)C2)=O)nnn2c1CCCC2 18142,CCC(C)(CCC(C)C)C(=O)N1CC(NC(=O)CCc2cnn(C)n2)C2(CC2)C1 18143,c1(C(=O)NC(C(C)C)C(C)NC(=O)OC(C)(C)C)cnc(O)nc1O 18144,C1(CNC(=O)C(C2CCN(C(=O)CC3COCCO3)C2)F)CCC2(CC2)C1 18145,N1(C(C(=O)NC(c2cccs2)C)=O)CCCC2CCCC12 18146,CC1(C)CC(C(=O)N2CCC2CNC(c2cnc(O)c(F)c2)=O)=NO1 18147,c1(C(=O)OCC)c(C)nc(N2CC(CN3CCCCC3CCO)C2)n1C 18148,c1(OC)ccc(CC(N2CCC(NC(C3(O)CCSCC3)=O)C(O)C2)=O)cc1Cl 18149,N1(C(c2cc(CNC(COCCCCC)=O)[nH]n2)=O)CCCC(C)C1CO 18150,O=C(NOC)C(CC1CC1)n1ccnn1.C1(C(CO)C(=O)O)CCOCC1 18151,CCCC(CC)CCC(=O)N(C)CC1(O)CCN(C(c2cc(F)cc(Cl)c2)=O)C1 18152,CN1CC2CCC(C1)N(C(C1CC3(C1)CN(C(C1CCC(=O)N1)=O)C3)=O)C2 18153,C1(NC(=O)C(=Cc2c[nH]cn2)F)CCCN(C(C2CC3(C2)CC3F)=O)C1 18154,c1(CC(=O)OC)ccnc(S(=O)(=O)NNC(=O)C2COCCC2(F)F)c1 18155,Cc1cc(C(=O)OCc2cnoc2C2CC2)nnc1C 18156,C1(c2ccccc2)(C(=O)NCCCCC)CCN(C(C2CCCO2)=O)CC1 18157,N1(C(CC2(C=C)CCOCC2)=O)CCC(NC(=O)CN(C2CC2)CC)C12CCC2 18158,N1(C(c2cc(F)cc(Br)c2F)=O)CCN(Cc2csc([N+](=O)[O-])c2)CC12CC2 18159,C1(C(C(=O)CC(=C2CCCCC2)F)F)CCCCC12CC2.O=C(CCN)O 18160,N1(C(C(CC)(C)C)=O)CC(NC(=O)CCc2nnc(C3CC3)o2)CCC(O)C1 18161,CCC(CCCC(=O)NOCc1ccccc1)NC(C1CC2(CC2)C1)=O 18162,Cc1csc2ncc(C(=O)NCC3CCCN(C(C4CNC(=O)C4)=O)C3)c(=O)n12 18163,C1(N(C(C)=O)C)CCCCC12CCCN(C(=O)C1CC1)C2 18164,c1(CCC(N2CC3(CN(Cc4cncc(C)n4)C3)C2)=O)c[nH]c2ccc(F)cc12 18165,C(CC(=O)NC1(C)CCCC1(C)C)(C(C)OC)NC(CC=CCCCCC)=O 18166,c1(CC)oc(C)cc1C(=O)OCc1ccnn1C(F)(F)F 18167,N1(C(CN(S(CC)(=O)=O)C)=O)CCC2(CC1)CC2CNC(=O)CC(C)CN(C)C 18168,CC1C(C(=O)N(C(C)(C)CC(=O)NC(c2cccnc2)C)C)CCN1C 18169,N1(C(CN2C(C)CCCC2)=O)CCC(NC(=O)CC2CCC(=O)NC2)C(C)(C)C1 18170,N#CC1(C(N2CC(CNC(=O)C(O)C(F)F)C3(CCC3)C2)=O)CCS(=O)(=O)CC1 18171,C=C(Cl)CCC(=O)NCCOCCNC(=O)CCCOC1CCCCC1 18172,c1(C(N2CC(C)N(C(=O)CC3CCC4CC4C3)CC2)=O)cc2ncccc2[nH]1 18173,C1(C(=O)NCC(C)(C)NC(Cc2c(C)noc2)=O)CCS(=O)(=O)C1 18174,C1(NC(C(=O)NCCOCC)=O)CCC(CCC(=O)NC(N2CCCC2)=O)C1 18175,N(C(=NCCCCF)NC1CCOCC1)CCNC1CCCN(C(C)=O)C1 18176,N1(C(C(C(C)(C)C)=O)=O)CC2(CCC(CNC(=O)CC3CCC4CC4C3)O2)C1 18177,C12(CC)CCN(CC1)N1C(CC1)CC(=O)N2.C(=O)CN(S(C)(=O)=O)C.C(C)(=O)N 18178,c1(CC(N2CCC(CN(C3CC3)C3CC3)C2)=O)cc(F)ccc1C(F)(F)F 18179,N1(C(Cc2c(C)cc(O)cc2)=O)CCN(C(=O)CCCC(C)C)CCC1C 18180,C(=O)(NNC(=O)C(C)(C)CCCCNC(c1cccnc1)=O)c1c(C)ccs1 18181,n1(CCNC(C(C)C2CCCC2)=O)cc(C(=O)NC2(C)CSC2)cn1 18182,CC1(C)C(C)(C)C1(F)CNC(=O)CNc1cnc(Cl)c(Cl)c1 18183,C1(NC(CC(C)(C)C2CC2)=O)CCN(C(=O)CCCC#N)CC1O 18184,N1(c2ncnc(C)c2Br)CCC(F)(F)C(C(=O)NC2CCCC(O)C2)C1 18185,c1(OC)ccccc1C(=O)C(=O)NC1CC(C)N(C(=O)CCc2cnc[nH]2)C1 18186,C1(C(N(CCCNC(=O)CC(F)(F)Cl)C)=O)CCCC1S(C)(=O)=O 18187,c1(C(CC)N(S(CC)(=O)=O)C2(CO)CC2)ccc(O)nc1 18188,c1(NC(C2N(C(c3c(C)cnnc3)=O)CC=C2)=O)ncc(Br)c(C)c1[N+](=O)[O-] 18189,N1(C(=O)NCc2c(Cl)cnc(Cl)c2F)CCC2(CC(=O)NC2=O)C1 18190,c1(CC(=O)NC2C=CCN(C(C(C)Oc3ccccn3)=O)C2)c(Cl)cccc1Cl 18191,N1(C(c2cnc3sccn23)=O)CCN(C(c2cncnc2)=O)C2CCCCC2C1 18192,C1(C(=O)NCC2C(CNC(Cc3c(C)ncs3)=O)C2)CC2CC(=O)C1C2 18193,C1(NC(CCOC(C)C)=O)Cc2ccccc2C1NC(C1CCC(F)C1)=O 18194,N1(C(COC)=O)CCC(C(=O)N2CCn3ncnc3C2)=C(F)C1 18195,C1(CC)CCN(C(=O)CC2CN(C(c3cc(C)[nH]n3)=O)C2)C1CNC(C)=O 18196,c1(CC(=O)NC(CC)CNC(C2(C)C=CCC2)=O)ccc(OC)cc1Br 18197,C1(=O)CC(C)C(=O)N(CC(=O)N(C)C)CC(=O)N1.C(C)(C)(C)O.CCO 18198,Cc1cc(Br)cnc1NC(=O)CC1CCCN1Cc1ccn(CCF)n1 18199,CCC(CN(C)C(c1cnsn1)=O)NC(C1CCCO1)=O 18200,S(=O)(=O)(CC(=O)NC1COCCN1C(=O)C(F)F)NCCOCCOCC 18201,Cc1ncc(C=CC(=O)NC(C2CCN(C(C3(Br)CC3)=O)C2)(C)C)c(O)n1 18202,c1(C(=O)NCC(C2CCOC2)NC(Cc2nc(C)[nH]n2)=O)nc(O)c(C)s1 18203,N1(C(c2cn(C3CCN(C)C3)nn2)=O)CCCC(CN(C(=O)CC(F)F)C)C1 18204,N1(C(C(N2C(=O)CCC2=O)C)=O)CCC2(CC1)CC(NC(=O)CC(C)(C)C1CC1)C2 18205,c1(C(C)C)ncc(Br)c(C(=O)NC2CCC2NC(c2cc(O)cc(F)c2)=O)n1 18206,Cc1cccc2c(C(N3CC(NC(=O)CC(C)O)CCC3C)=O)nccc12 18207,C=CC1(C(=O)NC2(c3noc(C)n3)CC2)CCN(C(C2CC=CC(O)C2)=O)CC1 18208,C=CCC(CO)NC(C1CC(c2nnnn2C)(NC(=O)OC(C)(C)C)C1)=O 18209,C1(CNC(C(c2cccc(F)c2)C)=O)CC(C)N(C(c2cccnc2F)=O)C1 18210,c1(NC(N2C(C#N)(c3ccccc3)COCC2)=O)ccc2c(Br)cccc2n1 18211,c1(SC)cccc(C(N2CC(NC(=O)CCc3ccccc3O)C(C)C2)=O)c1 18212,c1(OCC)cc(C(N2CCC(CNC(=O)C3=CCC(C)CC3)C2)=O)cc(Cl)c1O 18213,C1(NC(c2cc(C)c(O)nc2)=O)CC2CCC(C1)N2C(C1(C)CC1(C)C)=O 18214,CCCCCC(CC)C(=O)N1CCC(CNC(=O)CCC2CC2)(COC)CC1 18215,N1(C(CCc2cncc(C)c2)=O)CC2CN(C(c3ccc(C)nn3)=O)CCC12 18216,C(=O)(CC(C(C)OC)NC(c1ccc(O)nc1C)=O)NCC(CC)(C)Cl 18217,c1(CNC(C2C3CN(C(c4ccc(F)cn4)=O)CC23)=O)cccc(O)c1F 18218,C1(C(=O)NCCC(CNC(c2cn(C)c(=O)cc2)=O)O)CCC(=O)CC1(C)C 18219,N1(C(C2CC2C2C(C)OCC2)=O)CCC(CC(=O)O)C12CCC2 18220,c1(C(=O)NC(C)C(C)NC(C2(C)CS(=O)(=O)C2)=O)cc2c(cc1O)CCCC2 18221,c1(OCC)ncc(C(=O)NC2CC(CNC(c3ncn(C)n3)=O)C(O)C2)cn1 18222,Cc1cc(C(C)C(=O)NC2CCCN(C(C3(C)COC3)=O)C2)cc(F)c1 18223,C(=O)(C(C)P(C)(C)=O)N(CCOC)CCNC(=O)Cc1c[nH]ccc1=O 18224,CC1CCN(C(c2scnc2C2CC2)=O)CC1CNC(=O)C=Cc1ccsc1 18225,C(CCCCCN=[N+]=[N-])OCCSC.c1ncccn1 18226,C(=O)(CCC(F)(F)C(F)F)NC1C(NC(C2OCCN(CC)C2)=O)CC1 18227,Cc1ncc(C(N2CCC23CN(C(c2cn4ccnc4s2)=O)C3)=O)c(C)n1 18228,C1(CC(=O)N(C)CC2CCCN(C(c3c(C)nc(O)[nH]3)=O)C2)CCCCC12CC2 18229,N1(C(=O)Cc2ncsc2Cl)CCOC2(CCN(C(=O)C=Cc3cc[nH]n3)C2)C1 18230,c1(C(=O)NCCN(C(CC(C)OC)=O)CCCN(C)C)csc(C)c1C 18231,c1(C(=O)OC)cc(F)ccc1CNC(c1cc(Br)ccc1C)CO 18232,c1(C(CC)=O)cc(C(N2CCC(CCNC(C3CC4CC3C4)=O)C2)=O)ccc1F 18233,c1(OCC(C)O)ccccc1NC(=O)NCC1CCCC(C(F)(F)F)C1 18234,n1(CC2(CC)COC2)cc(C(=O)NC(C)CNC(c2cc(C(N)=O)c[nH]2)=O)nn1 18235,C1(O)(CCC)CCCN(C(c2ccc(CNC(=O)CC3CC3(C)C)o2)=O)C1 18236,C1(C(=O)NCC2C(NC(CO)=O)C2)CCN(C)CC1.CCC(C)N(CC)CC 18237,C1(NC(=O)CCOC2CC2)COC2(CCN(C(=O)CCN3CCOCC3=O)C2)C1 18238,Cc1ccc(C(=O)NC2CC3CN(C(C4CC4(C)C)=O)CC23)c(C2CC2)n1 18239,C(=O)(CCCCCC#N)N1C(C(N2CCC3C(C(N)=O)C3C2)=O)CC(C)(C)C1 18240,c1(C(=O)NCCCCC2CN(c3c(C)cnc(C)n3)C2)cc(C)c(C)cc1Cl 18241,c1(C(N2C(CCNC(C3CCC(=C)CC3)=O)CCC2)=O)ccc2nc(S)oc2c1 18242,N1(C(c2ccccc2Oc2cccnc2)=O)CCN(C(C2CC2F)=O)C(CF)C1 18243,c1(C(=O)NC(C(C)NC(C2(CC)COC2)=O)C)cccc(P(C)(C)=O)c1 18244,C1(C(=O)NC(CC=C)CO)CN(Cc2ccccc2C(=O)O)CCS1 18245,c1(C(=O)NCCSCC(=O)NCC2C(C)(C(F)F)C2)cc2ccncc2s1 18246,N1(C(CCOc2cn(C)nc2)=O)CCN(C(c2cnn(C)c2)=O)CC12CCC2 18247,N1(C(C2(CC)CC2(F)F)=O)CCC(C2(NC(C3CCCCCC3)=O)CC2)C1 18248,c1(C(=O)NC2CCC(CCNC(=O)Cc3cn[nH]c3)C2)ccc2c(c1)C(=O)NC2 18249,N1(C(=O)OC(C)(C)C)CC2(CC2)CC1C#CC(=O)NC1CC2C=CC1C2 18250,C1(C(N2CC(C(=O)NC)OCC2)=O)CN(c2ccncc2)CCO1 18251,N1(C2CN(C(Cc3cc(C)no3)=O)C2)CC(NC(c2ccoc2Cl)=O)CC1=O 18252,c1(C(=O)NCCC2(C=C)CN(C(=O)C(CC)(CC)OC)C2)cncc(F)c1C 18253,C1(CNC(c2c(OC)csc2)=O)COCCN1C(=O)CCCc1cc[nH]n1 18254,N1(C(CC2C3CN(C(C(C)(CO)OC)=O)CC32)=O)CCCC(C)(C#N)C1 18255,S(=O)(=O)(c1cccc(Br)c1)N1CC2(CCN(C(C(CC)c3ccccc3)=O)C2)C1 18256,c1(OC)cc(NC(=O)CCCC(C)NC(=O)C(C)NC(C)=O)cc(F)c1 18257,CCC(O)C(C)(C)C(=O)NOCC(N1CC2CCC2C1)=O.C1(O)CC1 18258,C1(CC)CNC(=O)CN1C(=O)CN(CC(C)(C)C)C(C1CC=CC1)=O 18259,N1(C(C2C(C)OC(C)C2)=O)CC2CN(C(=O)CNc3ccc(Cl)cc3)CC2C1 18260,c1(C(N2CCC(C)C(CNC(=O)C=Cc3ncc[nH]3)C2)=O)ccn2ncccc12 18261,CCC(C)(C)C(O)C(=O)NCCCN(C)C(C1CC1c1ccoc1C)=O 18262,c1(C(C)C)nocc1C(=O)NC(C)CN(C(=O)C(C)CC1CCCC1)C 18263,C(=O)(C(CCCCSC)N(C)CCOCc1ccccc1C)NC 18264,C1(O)(C(N(C(=O)CCC2(C(=O)OC(C)(C)C)CCCC2)C)=O)CCNCC1 18265,C1(C(c2ncn(C(C)C)c2)N(C)C)CCC(C)N1C(=O)OC(C)(C)C 18266,Cc1nn(C)c(Cl)c1C=CC(N1CC(CNC(=O)Cn2ccc(O)nc2=O)C1)=O 18267,N1(C(CC2(NC(c3n[nH]c(O)n3)=O)CCC2)=O)CC2(C1)NC(=O)NC2=O 18268,c1(OC)cccc(CC2CCCN2C(C2CC(Cl)(Cl)C2)=O)c1.C1(=O)CCN1C 18269,C1(CNC(CCCOCC=C)=O)CCCC(NC(=O)CCC=CBr)C1 18270,CC(CC(F)F)C(=O)NC1CN(C(c2ccsc2)=O)CC12CC2 18271,Cc1cc2ncn(CC(=O)NC3CCCN(C(=O)CC4CCCO4)C3)c2cc1C 18272,c1(C(=O)NCC(CO)NC(C2(COC)CCOC2)=O)ccc2nc(C)sc2c1 18273,C1(C(=O)NC2CC(CC(=O)NCC(C)OCC=C)C2)CCCC(=O)N1 18274,C1(NC(c2c(CC)ncs2)=O)CCC2CN(C(c3nccnc3N)=O)CC2C1 18275,c1(CCC(N2C(CCNC(C(C=C)(C)C)=O)CCCC2)=O)ccc2ncsc2c1 18276,CC(C)CC(CC(C)C)C(=O)NC1CC1NC(C1(Cl)CC1)=O 18277,N#Cc1cc(F)cc(-c2cn(CC(=O)NCC(N)=O)nn2)c1N 18278,CC1C(C)N(C)CCN1C(=O)CC1COCCN1C(c1c[nH]nc1Cl)=O 18279,c1(C(=O)NCc2ccc(CNC(CC(C=C)CC)=O)cc2)c(F)ccc(F)c1N 18280,N1(C(C(C(C)C)c2cccnc2)=O)CCN(C(c2cn(C)cn2)=O)C(C)C1 18281,C(=O)(CC(O)CC(C)(C)C)N1CC2C(NC(c3nc(OCC)c(Cl)cn3)=O)C2C1 18282,N1(C(C)=O)CCC(O)C(NC(=O)CNC2(C(=O)NC(CCSC)C)CC2)C1 18283,c1(C(=O)NC2CC(C)(NC(=O)CC3CC34CC4)C2)csc2c1CCCC2 18284,Cc1nc(N2CC3CC3C2)cc(N2CCCC(N3CCCC3)CC2)n1 18285,c1(OC)nc(C)ccc1C(=O)NC1CCCN(C(=O)C2=CCCCO2)C1C(C)C 18286,C(CCC(C)(C)C(=O)NCC(C)(C(=O)OC)OC)NC(c1ncc(CC)cn1)=O 18287,c1(C(N(C2CCCN(C(=O)Cc3cnns3)C2)C)=O)cnc2c(c1)NCC2 18288,C(C1CN(C(C2CC2c2ccco2)=O)CC1C(=O)NC1CC(C)C1)=CC 18289,N1(C(Cc2c(C)ocn2)=O)CC(C)(C)CC1CNC(c1nn(C(F)F)cc1Cl)=O 18290,N1(C(c2c(C)nco2)=O)CC(C)(C)OCC1CNC(C1(C)CC2CCC1O2)=O 18291,C1(C)(CC)CCCN1C(=O)CCCN(C)C(c1nnn(CC)c1C)=O 18292,CC1CN(C(=O)COCCF)CC1NC(=O)CCc1cn(C)nn1 18293,CC(CO)C(C)N=c1[nH]c2cc(Cl)c(S(=O)(=O)N3CC=CC3)cc2s1 18294,C1(C(C2CCCC2)NC(CSS(C)(=O)=O)=O)CCCN1C(=O)CC1CC=CC1 18295,C(=O)(CC(Cn1cc(CCCCCCC)nn1)CC(C)C)N1CCNCC1.CCO 18296,c1(CC(=O)NCCN(C(c2sccc2C#N)=O)CC)cc(F)ccc1OC 18297,C(=O)(C#CC1(C)COC1)N(CCCNC(c1c(C)cnn1C(C)C)=O)C1CC1 18298,CC1(C(=O)NC(CNC(c2cc(O)ncn2)=O)C2CC2)CCC(F)(F)CC1 18299,N1(CC)CCCC(C(=O)NC2CC(NC(c3cn(C)cc3C)=O)C(O)C2)C1 18300,N1(C(C(CSC)O)=O)CCOC(CNC(c2cc(C)co2)=O)C1 18301,C(=O)(CS(=O)(=O)CC(C)C)NCCCCC1CN(C(Cc2cnc(C)[nH]2)=O)C1 18302,CC(C)(CC(=O)NC1CCN(C(c2nccc3c[nH]nc23)=O)CC1)CC(F)(F)F 18303,CCC(C(=O)NC12CC(CNC(c3c(C)cc[nH]c3=N)=O)(C1)C2)C(C)(F)F 18304,CC(CCNC(=O)CC1CCCO1)NC(=O)C=C1CC1 18305,CCC(CC)(CO)C(=O)N1CCC(O)C(N(C(=O)C=CC2CCC2)C)C1 18306,CC(C)CC(O)C(C)C(=O)N1CC(C(=O)NCC2(C)CC=CCC2)C(C=CC)C1 18307,N1(CCCNC(CC(C=C)C)=O)CCN(C(=O)CC2CCC(=O)N2)CC12CCC2 18308,Cc1ccc2oc(-c3nc(C4CCCCN4)no3)nc2c1.c1(Sc2ccccc2)ccncc1Cl 18309,CC(C)(C)CC(C)(C)C(=O)NCc1csc(C(=O)NC2CCCC3(CC2)CC3)c1 18310,CN1CCOC(C(N2CCCC2CN(C(=O)C#CC(=O)N(C)C)C)=O)C1 18311,c1(C2(C)CC2C(N2CC(O)(CCNC(c3csnn3)=O)C2)=O)ccc(F)c(F)c1 18312,c1(N2CCN(C)CC2)ccccc1C#N.C1(CC(=O)OC(C)(C)C)(O)COC1 18313,c1(CNC(C2(F)CCN(C(C=Cc3cn(C)nc3)=O)C2)=O)nnc2n1CCC2 18314,C=CCC(C)(C)CC(=O)NCCOCCn1cc(Cc2cc(Br)ccc2C)nn1 18315,c1(C(=O)NC(C2(O)CN(C(C3(n4nccn4)CC3)=O)C2)C)cnc2nccn2c1 18316,N1(C(C=CCN(C)C)=O)CCN(C2CN(C(=O)CC3CCCS3(=O)=O)C2)CC1 18317,C(CCN=c1cc[nH]cc1S(=O)(=O)NC1CC1)N(CC(CC)CC(F)(F)F)C 18318,c1(C(N2CCCN(C(c3coc(Cl)n3)=O)CC2)=O)cc(=O)c2cc(Cl)ccc2[nH]1 18319,c1(C(=O)NCC2N(C(CNS(C)(=O)=O)=O)CC(F)C2)c(OC(F)F)cccc1F 18320,c1(C(=O)OC)cc(C(=O)NCC23CN(C(=O)OC(C)(C)C)C(C)(C2)C3)ccc1O 18321,c1(C(=O)NCC(C)NC(c2snc(O)c2Cl)=O)ccc(C2COC2)cc1 18322,C1(NC(CSC)=O)CCCC1(C)CNC(=O)CCCF 18323,n1(CC)ccc(C(=O)NC(CNC(=O)C(C)n2cnnn2)CO)n1 18324,C1(CNC(C2(SC)CCC2)=O)CN(C(=O)CC2CCCCC2)C2(CCOCC2)C1 18325,c1(OC)cccc2cc(CNC(=O)NCc3ccc(C#N)c(OC)c3)oc12 18326,c1(C(N2C(C(CN(C3CCCC4CC34)C(C)=O)(C)C)CCC2)=O)cc2n(n1)CCC2 18327,CCCCCC(F)C(=O)N(C(C(=O)NCC1(CN=[N+]=[N-])CC1)C(C)CC)C 18328,C(=O)(CC(C)CC(C)(C)C)N1CCC(COC)(NC(=O)Cc2ccoc2)C1 18329,Cc1cc(C(=O)NC2CCC2NC(=O)C(C)(C)C2CCCO2)ccc1N(C)C 18330,c1(C(c2cnc(COC)o2)NS(=O)(=O)CC2CCC2)cccc(C(F)(F)F)c1 18331,CCC(C)(C)C(O)C(=O)N1CC(F)CC1CN(C(=O)CC1CC1)C 18332,CC1CN(C(C2CC(O)CN2C(c2ccc(C(N)=O)[nH]2)=O)=O)CCC1N(C)C 18333,CC1CCCN(C(=NCC(O)c2ccccc2N(C)C)NC(C)C2CCC2)CC1 18334,N1(C(COc2c(OC)cccc2)=O)CCC(C)(C(=O)N(C)CCOC)C1 18335,c1(C(=O)NCC(C)N(C)C(c2cc(F)ccc2F)=O)ccc2[nH]ccc(=O)c2c1 18336,c1(C(=O)NCC23C(CN(C(Cn4c(C)csc4=O)=O)C2)C3)cccn2cncc12 18337,C(=O)(CCCCCNC(=O)Cn1nc(C)cc1C)N(CCC(=O)OC)CC=C 18338,Cc1cncc(CC(=O)NC23COC(CNC(c4cc(CO)c(C)o4)=O)(C2)C3)c1 18339,Cn1ncc2c(N3CC4CCN(Cc5c[nH]c6ncccc56)CC4C3)ncnc12 18340,C1(NC(C2(C)CNC(=O)C2)=O)CCCCN(C(C2CC2(C)Br)=O)C1 18341,c1(C(=O)NCCN(C(c2cn(C(C)(C)C)nc2C)=O)CC)ccccc1NCC 18342,C1(N(C(CC)=O)CC)CCN(C(=O)CCC2CC(F)(F)C2)C1 18343,C1(NC(C(C2CCC2)OCC)=O)CC2CC1N(C(=O)Cc1ccns1)C2 18344,Cc1cc(CCCNC(=O)C(C)Sc2ccccn2)oc1C(=O)O 18345,c1(C(N(CCN(C(CC(CC)OC)=O)C)C)=O)[nH]cc2c1CCS2(=O)=O 18346,Cc1cccc(C(=O)NCCC2(O)CN(C(=O)CCOc3cccnc3)C2)c1 18347,C1(NC(C2CCC(C)(C)O2)=O)CN(C(=O)C=Cc2cc[nH]n2)Cc2nccn2C1 18348,C=CCCC(C(=O)OC)NC(=O)CCCCN(C(=O)C=C=C(C)C)C 18349,C(CC(=O)N(CC(C)CC)C)(C(F)(F)F)NC(C(CC#C)C1CC1)=O 18350,c1(OCCOCCOCCOC(C(=O)CCNC(CC)=O)C)cccc(C#N)c1 18351,c1(OC)c(F)c(C(N2CCN(C(c3ccc(Cl)cc3)=O)C3CC23)=O)cc(F)c1F 18352,c1(CCC(N2C(CNC(CCNC(N)=O)=O)CC(O)C2)=O)cc(F)ccc1Br 18353,CC1CC(c2nnnn2C)(NS(=O)(=O)CC2=CCCC2)CC(C)O1 18354,C(c1ccncc1C)=CC(=O)NCCc1c(CNC(CC=C(C)C)=O)nco1 18355,CC1(C)C2COC1(C(=O)NCC(C)(C1CC1)NC(c1cc(Cl)c(Cl)s1)=O)C2 18356,C1(CC(=O)Nc2cn(CCC#C)nc2)C2CN(C(c3csc(Cl)n3)=O)CC12 18357,C12(CNC(c3cnc(C4CCCCC4)s3)=O)CC(CO1)N(C(=O)C1CC1)C2 18358,C1(CNC(CC2N(C)CC=CC2)=O)CC(C(N)=O)=NO1.C1(C)(C)C(=O)N1 18359,c1(C(=O)NCC2(OC)CCN(C(C(C(C=C)C)C)=O)CC2)ccc([N+](=O)[O-])cc1 18360,CC(C)(CNC(C1CC(O)CCN1C(C1CCCO1)=O)=O)CN=[N+]=[N-] 18361,c1(C(=O)NC2CC(F)CN(C(c3ccnn3CCF)=O)C2)cccc2sccc12 18362,CC(C)C(F)C(=O)NCC(C1CC1)N(C(=O)CNc1occc1Br)C 18363,c1(C(=O)NCCNC(C(F)OC)=O)nc2ccccc2c(Cl)c1Br 18364,c1(-c2nc(C3N(C)CCNC3)on2)ccnc2[nH]ccc12 18365,c1(C(=O)NCCCCCNC(CCCC(=O)NC(C)C)=O)ccnc2c1CCO2 18366,C(=O)(C(C)(C)C(F)F)N(CC(O)(C(F)(F)F)c1ccc(Cl)cc1)C.n12cc(nn1)C2 18367,C1(NC(CCC2CC(C)C2)=O)CCCC1NC(c1ccc(Cl)s1)=O 18368,O=C(C1=NOC2COCC12)NC(c1ccccc1)Cc1cccc2ccccc12 18369,C1(C#N)(C(=O)NC2CC(C(=O)NC(C(=O)NCC(C)C)C)C2)CC1(C)C 18370,N1(C(C(C)SC)=O)CCOC2(C1)CN(C(c1cc3c(C)nn(C)c3s1)=O)C2 18371,C1(CC)CCc2nc(O)c(C(=O)NC3CC4(C3)CC(C(=O)O)C4)cc2C1 18372,CP(C)(=O)c1cccc(C(=O)NCCC(O)CNC(C2CC3CCC3C2)=O)c1 18373,c1(NC(=O)Cc2cccnc2O)cc(-n2ccnn2)ccc1F 18374,Cc1nc2nccc(C(N3CC(C)(NC(=O)CC4CC(F)(F)C4(F)F)C3)=O)n2n1 18375,C1(C(=O)NCC(CN(C(C=CCC)=O)C)O)CN2CCN1CC2C 18376,N1(C(C=C(CCC)C)=O)CC(C2CC2)(C(=O)NCCC(O)C2CCCC2)C1 18377,c1(C(=O)NC(CCN(C(C=C(C)Cl)=O)C)C(C)(C)C)sc2cncn2c1C 18378,C=CC1(CC(=O)NCC2CCOC(C)C2)CN(C(c2cncnc2C)=O)C1 18379,S(=O)(=O)(c1c2ccccc2nn1C)NCCC1CC1.CN=c1[nH]cc(C(N2CCCC2)=O)s1 18380,C12(C(N3CC(C)(NC(CC(CC)C4CC4)=O)C3)=O)CCCC(C1)OC2 18381,C1(O)(CN(C(C2CC(=C)C2)=O)C)CN(C(c2cnc(Br)s2)=O)C1 18382,c1(C(N2CCN(C(C(C)OC)=O)CC2CCO)=O)cc(C)cc2c1OCC2 18383,N1(C(CC2(C)CN(C(c3ccc4n[nH]cc4c3)=O)C2)=O)CCCCC(C)(F)C1 18384,N1(C(C(C(=C)C)(C)C)=O)CC(CNC(=O)CC(O)CC(C)(C)C)OC2(CCC2)C1 18385,c1(C2(C(N3CC(C(C)NC(C(=O)NCC)=O)C3)=O)CCC2)c(OC)cccc1Cl 18386,C1(C(N2CC(CCOC)C2)=O)(CNC(c2cscn2)=O)CC12CCC2 18387,N#Cc1cnc(C(=O)NCC2C=CC(NC(=O)CC3(O)CCCCC3)C2)c(Cl)c1 18388,CC(O)C(C)C(=O)N1CCN(C(=O)C(CSC(C)=O)Sc2ccccc2)CC1 18389,C1(NC(=O)CCn2cncn2)CCC(CNC(c2cc(-c3cccs3)[nH]n2)=O)C1 18390,N1(C(CC(C)C(F)(F)F)=O)C(C)CC2CN(C(c3c(Cl)cnn3C)=O)CC12 18391,n1(CC)cnc2c(NCCOC)[nH]c(=NCc3cc(OC)cc(OCC)c3)nc12 18392,c1(C(N2CC(C)C(NC(=O)C=CC3(C)CCOCC3)C2)=O)cc2cnn(C)c2s1 18393,C(CC(C(=O)N1CCOC(C2(C)CC2)C1)NC(C1CC=CCC1)=O)N(C)C 18394,c1(C(N2C(CNC(C3CC4C=CC3O4)=O)COCC2)=O)cc(Cl)ccc1Cl 18395,c1(C(N2CC(NC(CN(c3ccccc3)C)=O)C(O)C2)=O)cc2occc2s1 18396,C12(C(=O)NCC(N3CCN(C(c4cncc(Cl)c4)=O)CC3)C)CCCN(CC1)C2 18397,c1(C(=O)NC2CCC(NC(C(CC)(C)C#N)=O)C2)cnn2c(Br)cccc12 18398,C1(CC)C(C)CCN1C(=O)COC(C)(C)CNC(c1cccc(NC)n1)=O 18399,c1(C(C)(C)C)nc(=N)[nH]cc1C(N1CC2CC1CN2C(=O)C(=Cc1cnc[nH]1)F)=O 18400,c1(N2CCC(C)(NC(C(CCC)NC(N)=O)=O)C2)ncc2c(ncn2C)n1 18401,C(C1=NOC2CC12)(c1nnnn1C1CC(F)(F)C1)NCC(C(C)C)(C)C 18402,C(=O)(CCCCCCc1ccccc1)N1CCC(NC(C(C=C)(C)CC)=O)C1 18403,c1(C(=O)NC2C(CNC(c3cccs3)=O)COC2)nc2n(c1Cl)CCCC2 18404,C(c1nc2ccccc2o1)=CC(=O)NCC(C)CNC(=O)Cc1ccnc(O)c1 18405,CCC(CCCC(=O)N1CCCOCC1C)NC(C1CC(C)CCO1)=O 18406,c1(CC(=O)NC2CC(F)(CNC(=O)Cc3ccccc3O)C2)cc(F)ccc1Cl 18407,N(C1CCc2cc(Br)ccc21)CC(c1c(OC)ccc(C)c1)=O 18408,N1(C(C(N2CCC(C)(CCC)C2)=O)=O)CCCN(C(=O)OC(C)(C)C)CC1 18409,c1(C(C(=O)NCC2N(C(COC3CN(CC(C)C)C3)=O)CC2)O)cnccc1C 18410,c1(NC(c2ccc(-c3c(OCC)cc(OC)cc3)cn2)=O)nc(C)ccc1C#N 18411,N1(C(C(C)OCC2CC2)=O)CCCC(C)(CNC(c2ncccc2F)=O)C1 18412,Cc1coc(C=CC(=O)NCC(CC(C)C)NC(c2coc(Br)c2)=O)n1 18413,C(c1ccc(F)cc1)=CC(=O)NCCC1CCCN(C(=O)Cc2ccccn2)C1 18414,Cc1nccn1CCC(=O)NC1CC(NC(c2ncoc2-c2ccco2)=O)C1 18415,c1(NC(C(CC)N(C)C(C2CC2(F)Cl)=O)=O)cc(C)cc(O)c1 18416,CN1CCCC1C=CC(N1CCC(C)(CNC(c2ccsc2Cl)=O)C1)=O 18417,C1(OC)CCCC(CNC(=O)C=CCC(C)(C)NC(c2cc(O)nn2C)=O)C1 18418,C(=O)(C(CC1CCCO1)C(F)(F)F)N(C)CC1(NC(CCCCC=C)=O)CC1 18419,Cc1cc(=NCCN2CCCn3nccc32)[nH]c(NC2CCC(F)(F)C2)n1 18420,CCC(C)CC(C)C(=O)NCCCCNC(=O)CNC(=O)Nc1ccc(C)cc1 18421,C(=O)(CCCC(O)c1ccccc1)NC(C1CCCN1C(C1CCCO1)=O)C 18422,N1(C(C=Cc2n(CC)ccn2)=O)CCCCC12CC(NC(=O)CCC1CC1C)C2 18423,N1(C(c2cn(C)c(=O)cn2)=O)CCN(C(C2(F)CC2(Cl)Cl)=O)CC12CCC2 18424,C1(NC(c2c(C)nn(C)c2)=O)CCCCC12CCN(C(=O)COC1CCOC1)C2 18425,C=C(C)CC(C(=O)NC(CNC(=O)Cc1cccnc1O)C1CCC1)OC 18426,C1(C(=O)NC2C(C#C)CCC2)CNC(=O)CN1C(=O)COC1CCC1 18427,C(=O)(CC(C)C(F)(F)F)N1CCCC(F)(C(N(CCCC(=O)NC)C)=O)C1 18428,NC1CCCc2c(F)cccc21.C=CC1(CCN=c2[nH]ccs2)CCOCC1 18429,C#CC1CN(C(c2cnc3ccoc3c2)=O)CCN1C(=O)C(C)OC1CCOC1 18430,C1(CC)CC(C(=O)NC2(CNC(c3ccc(Cl)nc3C)=O)CC2)CCC1=O 18431,c1(C(=O)NCC(CC=C)NC(=O)C(c2cnn(C)c2)O)nc(Cl)sc1C(C)C 18432,C1(NC(C=C2CCC(C)CC2)=O)CCN(C(c2cc(Cl)n(C)n2)=O)C12CC2 18433,c1(C(N(C2CC(C(=O)OCC)C2)CC=C)=O)ccoc1I 18434,N1(C(C(C(C)(C)C)=O)=O)CC(CNC(C2CC(F)(CO)C2)=O)CC12CCC2 18435,N1(C(c2cc(OC)ncc2)=O)C2CCC1CN(C(C1CC1c1ccnn1C)=O)C2 18436,c1(CC)nccc(=NCCOCCN(C(=O)CCc2cc(C)cc(C)c2)CC)[nH]1 18437,CC(C)C(C(=O)NCC1CN(C(=O)CCCn2cccc2)CCO1)C1CCC1 18438,N1(C(C(C)=C2CC2)=O)CCC2(C1)CN(C(c1ccc(F)c(O)c1F)=O)C2 18439,C1(CNC(C2C(C)=C2)=O)CCC2CN(C(c3ccc4ncnn4c3)=O)CCC2C1 18440,n1(CC)nc(CN2CC3CC2(C)C3)c2c1CCOC2 18441,C1(NC(C2(CCOC)CC2)=O)CN(C(c2cncn(C)c2=O)=O)C2CCCCC12 18442,C#CC(C)(C)C(=O)NC1CCC(C(=O)NCC2CC2Cl)CC1 18443,Cc1nn(C)cc1C(C)NC(c1conc1C(C)NC(=O)CC1C=CCC1)=O 18444,c1(C(N2CC(N(C(c3c(C)cn(C)c3)=O)C)C(F)C2)=O)ccc2nonc2c1 18445,c1(CCC(=O)NC2CC(CNC(C(CC)(C)OC)=O)C2)ccc2c(n1)NCCC2 18446,C1(C)(C(=O)NCCOCCCNC(C(C2CCOC2)OC)=O)CC2(CCC2)C1 18447,C(=O)(C1=CC2CCC1C2)N(CCN(CC)C(c1cnn(-c2ccccn2)c1C)=O)CC 18448,C1(CNC(C(C)(C)SC(F)(F)F)=O)CN(C(c2cnns2)=O)CCO1 18449,C1(NC(=O)NCC2CN(C3CCCCC3)C2)CCC(c2ccccc2)C1 18450,N1(Cc2ncc(CC)o2)CCC(NC(c2cc(C3CC3)on2)=O)C(C)C1 18451,N1(C(c2c(CC)onc2)=O)CC(C(=O)NCC2CC(C)(C)C2)C2(CC2)C1 18452,N(C1c2ccccc2CC1NC(=O)C1CCCc2ccnn21)C(CCC(C)C)=O 18453,c1(C(=O)Nc2ccc(C3(C(=O)OC)CCOCC3)cc2)cnc(F)cc1C 18454,C(CCN=C(NCCc1cncc(O)c1)NC1CCOC(C)C1)OCC 18455,C#Cc1ccc(C(N2CCCC2CN(C(=O)C(F)CC)C2CC2)=O)c(OC)c1 18456,C(=O)(CCC(=O)NCC(C)(C1CC1)NC(=O)C(n1ccnc1C)C)NC 18457,N1(C(CCCN(C)C)=O)CCCC2CCN(C(=O)C(F)(F)CN3CCCC3)CC12 18458,Cc1cc(C#N)cnc1C(=O)NCCc1n[nH]cc1C(=O)NOC(C)(C)CO 18459,c1(C(N2C(CCNC(C(CCOC)C)=O)CCCC2)=O)ccc(C#N)c(Cl)c1 18460,C1(C(=O)NC(CCCNC(C2(CC(C)C)CCC2)=O)C)CC2(C1)CC(C#N)C2 18461,c1(NCCC)ccc(C(=O)N(c2ccc(Cl)cn2)C)cc1 18462,c1(OC)cccc(C(N2CCC(N(C)C(C3C(C)(C)C3(F)F)=O)C2)=O)c1[N+](=O)[O-] 18463,C(=O)(N(OC)C(C)C)c1cn(CCN(C(CC(C=C)C)=O)CC)nc1 18464,N1(C(c2cc(COC)sc2)=O)CC(CNC(c2cscc2COC)=O)C(C)C1 18465,C(C1CCCCCC1)=CC(=O)NC1(CCNC(C2(C)CCCOC2)=O)CCCC1 18466,C1(CC)CCN(C(=O)CCc2ccoc2)C(C(=O)NCc2cc[nH]n2)C1 18467,c1(NCC2(CC)CCCC2)[nH]c(=NCCC2CCCO2)nc2c1ncn2C(C)C 18468,N1(C(C)C(=O)Nc2ccccc2)CCN(c2ccc(F)cn2)CC1C 18469,C(=O)(C(C)C1=CCCC1)NC(CCCNC(CCC#C)=O)CCC 18470,C1(NC(C(OC)OC)=O)CCC(NC(c2cn(CC3CCOC3)nn2)=O)CC1 18471,c1(COC)cc(C(=O)NC2CCC2NC(=O)CC23CCC(CC2)C3)n(C)c1 18472,N1(C(C(CCCC)C)=O)Cc2n[nH]cc2C1C(=O)NCCc1nnc(C)s1 18473,CN1CCC(C)(C(=O)NCC(O)CCNC(=O)C(CN(C)C)N(C)C)CC1 18474,c1(C(N2CC(NC(Cn3nnc(C)n3)=O)CC(C)(C)C2)=O)ccc2c(c1)OCCO2 18475,N1(C(CCC=C=C)=O)CCOC2CN(C(c3[nH]c(=N)ccc3C)=O)CC12 18476,N1(C(C2(CC#C)CC2)=O)CCc2nc(O)cc(C(=O)NC3CCN(C)C3C)c2C1 18477,C12(C(=O)NC(C(N3CC(C(N)=O)C3)=O)C3CCCO3)CC(F)(C1)C2 18478,c1(COC(C23CCC(OC)C2C3)=O)ccc(F)cc1C#N 18479,c1(OCC)cccc(C=CC(=O)NC2CCCN(C(C3(C)CNC(=O)C3)=O)C2)c1 18480,CC1(C)CCN(C(=O)C=Cc2cccnc2)CC1CNC(=O)Cc1cc(Cl)cs1 18481,CC1CCCN(C(=O)CC(F)(F)c2ccccc2)C1CNC(=O)CC1OCCO1 18482,S(=O)(=O)(c1c[nH]ccc1=NCC1CCCOCC1)NCc1c(Cl)cn(C)n1 18483,N1(C(C2N(Cc3cc(OC)cc(F)c3)CCNC2)=O)Cc2ccc(Br)cc2C1 18484,c1(OCCC(=O)NCC=CCNC(C2CCCCCC2)=O)ccc(F)cc1Cl 18485,C1(C(N2CCC(c3ccon3)C2)=O)COC2(C1)CN(C(c1cccnc1O)=O)C2 18486,C#Cc1ccnc(C(=O)NCC(C2CC2)N(C(=O)C(CSCC)SC)C)c1 18487,C(CC(=O)N1CC(C)(CCO)C1)(C(C)OC)NC(C(C)OCCOC)=O 18488,C1(NC(c2cc[nH]n2)=O)CN(C(c2cscn2)=O)C2(CCC2)C1 18489,C1(C(=O)NCC2OCCN(C(C3(n4cccn4)CC3)=O)C2)CCCCNC1=O 18490,c1(OC)cc(C(N2CC=CC(NC(=O)Cc3ccsc3)C2)=O)cc(N)c1O 18491,C(=O)(N=c1[nH]nc(-c2c(F)cccc2Cl)s1)Nc1c(C)nc(CO)s1 18492,N1(C(C2C(NC(C(C)NC(CC)=O)=O)CC=CC2)=O)CCOC(C)C1C 18493,C1(C(=O)NC(C)C=CC(=O)NCCN2CCC2)OCCCC1(C)C 18494,S(=O)(=O)(c1ccc(S(=O)(=O)N2CCCC2)cc1)N1CCC(C#CC)C1 18495,C1(CCC)(NC(=O)CC(C)C(C)C)CCCN(C(=O)C(Br)=C(C)C)C1 18496,C(C(C(=O)N(CC(C)(C)C#N)C)NC(=O)Cn1cnnc1O)OCC 18497,c1(C(=O)NC2C(C=C)CN(C(C3(COC)CC3)=O)C2)cc(Cl)cc2c1CCC2 18498,Cc1cc2c(cc(C(N3CC4CCN(C(=O)CO)C4C3)=O)n2CC2CC2)s1 18499,C1(NC(c2c(C#C)c[nH]n2)=O)CCN(C(=O)CSCCN(C)CCO)CC1(C)C 18500,C12(C(N3CC(C)N(C(c4cnc(=N)[nH]c4)=O)CC3)=O)CCC(C1)C(C)(C)O2 18501,c1(C(=O)NC2CC(F)(CNC(Cc3n(C)ccn3)=O)C2)cc2cccc(F)c2o1 18502,CCC(F)(F)CC(=O)N1CC(O)(C(C)NC(C2CCC(C)O2)=O)C1 18503,C1(O)(C(=O)NCC(C)N(C(=O)CC2CCCCC2C)C)CN2CCC1CC2 18504,c1(SC)cc(C(N2CCC2CNC(=O)C2CC2)=O)nn1C 18505,C(=O)(CCC(C)(C)C#N)N1C(C(C(N2CC(CC)(CC)C2)=O)(C)C)CCC1 18506,C1(NC(CC=C=C)=O)(CNC(=O)C(C2(OC)CCOCC2)(F)F)CCOCC1 18507,C1(CC(=O)OC)CN(C(=O)Cc2cccc(CC(F)(F)F)c2)CC(C)(C)O1 18508,c1(CC(=O)N(C(C)CCNC(c2c[nH]c(=N)s2)=O)C)cccc2ncccc12 18509,Cc1cccc(C(=O)NCC2CCN(c3ccccc3C(N)=O)CC2)c1N 18510,Cc1ncn(C)c1C(N1CC(n2cc(CNC(c3csc(S)n3)=O)nn2)C1)=O 18511,c1(C(N2CCC(C)C2C(=O)NCC2CCC(C)(C)CC2)=O)cc2occc2[nH]1 18512,C1(NC(Cc2c(C)csc2)=O)CCCCCN(C(c2ccc3cnnn3c2)=O)C1 18513,N1(C(C=C(C)C(C)(C)C)=O)CCCCCCC1C(N1CC2CCOC2C1)=O 18514,CC(C(=O)N(C1CCN(C(=O)C(c2cc(F)ccc2F)=O)C1)C)C1=CCCC1 18515,Cc1oc(S(C)(=O)=O)cc1C(=O)NCC1CC(O)CN1C(=O)CCOCC(F)F 18516,N1(C(C2(C)CCN(C)C2)=O)CCC(NC(c2ccc3ccsc3c2)=O)C(C)(C)C1 18517,N1(c2nnc(CC)o2)CCC2(CC1)CN(C(=O)C(F)C1CCOC1)CC(C)O2 18518,c1(N2CCN(C(CN(C)Cc3ccc(F)cc3)=O)CC2)ncc([N+](=O)[O-])cc1F 18519,N1(C(c2ccco2)=O)CC2CC(C1)N(C(c1ccc(-n3ccnn3)cc1)=O)C2 18520,N1(C(C2CC(C)S(=O)(=O)CC2)=O)CCC2(C1)CN(C(=O)Cc1ccsc1)CCO2 18521,n1(CC)cc(C(N2CC(C(O)C(=O)NC3CC(C(C)C)C3)C2)=O)nn1 18522,C1(NC(c2ccc(C)nn2)=O)CN(C(=O)CCC2CCCOC2)CCC12CCC2 18523,N1(C(C(C(C)C)n2cnnn2)=O)CC2(CCC2CNC(=O)C(=O)N(C)C)C1 18524,N1(C(c2c(CNC(C3CC(C)N(C)C3)=O)noc2)=O)CC(C2CC2(F)F)C1 18525,c1(C(=O)NCCCCNC(C(C)OCOC)=O)cnn(CCCN2CCCC2)c1 18526,C1(NC(C=Cc2ccc(CC)o2)=O)CCCCC12CCN(C(=O)C(C)CO)CC2 18527,C1(CCC(=O)NC2C(CNC(CNS(CC)(=O)=O)=O)CC2)CCCN1C 18528,N#Cc1ccc(C(N2CC3CC3(NC(=O)CCC3CCCCCC3)C2)=O)[nH]1 18529,c1(CC)ccc(CC(=O)NC2CCCCC2CNC(C2CCS(=O)CC2)=O)cc1 18530,c1(C(=O)NC2CC(N(C(C(CC)C)=O)C)C2)cccnc1-n1ccnc1C 18531,c1(NC(C2(F)CCN(C(c3cncs3)=O)C2)=O)ccc2c(c1)OCCO2 18532,CONC(=O)C(=O)N1CCC(O)(CC)C1.N1(C(=O)NCC)CCCCC1 18533,c1(C(=O)NCCC(C)CCNC(=O)CS(C)(=O)=O)cc(C(F)F)cc(F)c1 18534,C1(NC(CCC(C)OC)=O)C(C)CCN(C(=O)COCCN(C)C)C1C 18535,C1(NC(CC2CCN(C)C2)=O)CCCC(C(N2CCN(C(=O)C(C)(F)F)CC2)=O)C1 18536,C(=O)(C1=CCS(=O)(=O)C1)N1CCC(O)(C(C)CNC(c2cc(O)nc(Cl)c2)=O)C1 18537,CS(=O)C=CC(=O)N1CCC(C(O)CNC(=O)C(C)(F)c2ccon2)CC1 18538,c1(CC(=O)N(CC(C)CNC(C2CC(C)OC2C)=O)C)coc2ccc(F)cc12 18539,Cn1c(C(N2CC(O)(CNC(=O)Cn3ccnn3)C2)=O)cc2c1CCOC2 18540,N1(C(C(C)OCOC)=O)CCC2(CCC(NC(c3ccc4n[nH]cc4c3)=O)C2)C1 18541,C1(CNC(C(N2CCC(C#C)(O)CC2)C)=O)CC2(CO1)CC(F)(F)C2 18542,c1(C(N2CCC(NC(C3CCN(CCC)CC3)=O)C2)=O)cc(C)c(CO)cn1 18543,c1(CC(=O)NC23CC(CNC(c4c(C)occ4)=O)(C2)C3)cn(C)nc1C 18544,c1(CNC(CNC(=O)OCC)=O)ncc(C(=O)NCCCC2C=NNC2=O)o1 18545,CC1CC(C(=O)NC2CCCC2CN(C)C)N1C(C1CSC1)=O 18546,c1(C(N(CCCCCNC(C2(C)CS(=O)(=O)C2)=O)C)=O)n[nH]c2c1COC2 18547,C1(CNC(NNC(=O)C2CC(OC)C2)=O)CCn2ccnc2C1 18548,N1(C(CN2CCN(C)CC2)=O)CCN(Cc2ccc3nonc3c2)CC12CC2 18549,c1(C(=O)NCCN(C(C2CC(CCC)C2)=O)C)occ(C)c1C 18550,N1(C(=O)OC(C)(C)C)CC(O)(C(=O)NC2(C(F)F)CC(Nc3cc(O)no3)C2)C1 18551,N1(C(CC(CC2CC2)NC(c2c(C)ocn2)=O)=O)CCc2ccc(C#N)cc21 18552,c1(C(=O)NCC2CCN(C(C3(CCCC)CC3)=O)CC2O)cccc2c1CCN2 18553,c1(C(N2CCC(C)(NC(C(C)OCC)=O)C2)=O)cnc2cc[nH]c2c1 18554,c1(CC(=O)NC2C(NC(C3(C#N)CCCC3)=O)COCC2)ccc2c(c1)CCO2 18555,N1(C(c2c(C)cc(C)[nH]2)=O)CCC(CNC(c2c[nH]nc2C2CC2)=O)C(C)C1 18556,C(c1ccc(Cl)c([N+](=O)[O-])c1)=CC(=O)NCC1N(C(c2nc(C)sc2)=O)CC1 18557,N1(C(CCOCC)=O)CC(NC(=O)Cn2ncc(C#N)c2N)CC1(CC)CC 18558,C1(NC(CSC(C)C)=O)CN(C(c2cc(C3CC3)on2)=O)CC1C(F)F 18559,C(=O)(C1=CCOCC1)NCC1CCC(CNC(C2N(C(=O)NC)CCC2)=O)CC1 18560,N1(C(C(C2CCCC2)OCC)=O)CC2CCC1C(CN=c1ccnc(Cl)[nH]1)C2 18561,c1(CSC)nn(C)cc1C(N1CCCC1(C)CNC(=O)Cn1cc(CO)nn1)=O 18562,N1(Cc2c(N3CCCC3)ccc(C)c2)CCN(CCCOC(C)C)C(C)(C)C1 18563,N1(C(C)=O)CCN(C(=O)CC2(NC(=O)C(C3CCC(=O)N3)C)CCC2)CC1 18564,c1(C(C)(C)C(=O)NC2(C)CC2(Cl)Cl)ccnc(P(C)(C)=O)c1 18565,C1(NC(c2cc(OC)no2)=O)CC2CCC1CC2NC(C1CCCC1(C)C)=O 18566,C(C(C)C(=O)NC(c1cccnc1)C(=O)NCC1(CO)CCC1)SC 18567,Cc1ccc(Br)c(N)c1NC(=O)Cn1cc(CN2CCCCC=C(Br)CC2)nn1 18568,CCC(C)C(C(=O)NCC1CC2(CC2)CO1)NC(=O)Cn1cnnc1O 18569,N1(C(CN(CCOC)C)=O)C2CCC1CC(NC(C1(C)CCC(O)CC1)=O)C2 18570,Cc1cc(CC(N2CCC(N(CCO)Cc3cnc(S)[nH]3)C2)=O)n(C)n1 18571,CC1CC(CCNC(c2c[nH]nc2C(F)F)=O)CCN1C(=O)Cc1cnns1 18572,c1(C(=O)NCC(CC=C)NC(C2COCCN2C(C)=O)=O)ccc2nccn2n1 18573,C1(C(=O)NC(C)CCCNC(c2cc(C(C)(C)C)ccn2)=O)COC2(CCC2)C1 18574,CC1CCC(NC(C2CCC(C)(C)CC2)=O)CN1C(C1CN2CCC1CC2)=O 18575,c1(CC)ccc(C)cc1C(N1CCCC1C(C)NC(c1[nH]cnc1C)=O)=O 18576,C1(C(=O)NCC2(C(N(CCN(C)CCO)C)=O)CC(C)(C)C2)CC(=O)NC(=O)C1 18577,C1(C(C)(O)CNC(=O)CCc2cn(CC(F)(F)CO)nn2)CCOC1=O.C1CNN1 18578,C1(NC(c2ccc(CF)cc2)=O)CCCN(C=O)C1.C1(N2CCCC2)(C)CCC1 18579,c1(N2CC3C(NC(=O)OC(C)(C)C)C(C3)C2)ncc2cccc(Br)c2n1 18580,Cc1cc(C(=O)NC(C2(CNC(c3sc(F)cc3C)=O)CC2)C)c(C)[nH]1 18581,c1(C(N2CC(C(=O)NCc3nn[nH]c3C(F)(F)F)C2)C)ccccc1F 18582,C1(N(CC#C)C(=O)Nc2ccc(C)c(C(F)(F)F)n2)CCC(F)(F)CC1 18583,c1(NC(C2CC2C(=O)Nc2cnccc2Cl)=O)cc(F)ccc1Br 18584,C1(F)(C(=O)NCCC2(CNC(C3CC=CCC3)=O)CC2)CC1(Cl)Cl 18585,C(=O)(C1CCCc2ncnn21)N1CC2CC(Nc3nc(C)nc4c3ccs4)C2C1 18586,C(=O)(CC(C)O)NCC(C)=CC(=O)N(CC(c1nn[nH]n1)C)C 18587,c1(C(N2CCN(C(Cc3ccc(OC)c(C)c3)=O)CC2)=O)c(C)nc(C)nc1C 18588,Cc1nccc(C(=O)NCC2(CNC(c3cscc3F)=O)CCCCC2)c1N 18589,c1(C(=O)NCC2C(NC(C(C)C#N)=O)CC2)c(F)ccc(F)c1Cl 18590,c1(C(N2CCC(N(C(C3CCC4CC34)=O)CC)C2)C)ccc(Br)cc1 18591,N1(C(CN(C(C)=O)C)=O)CC2CN(C(=O)Cc3nccs3)CCC2(CO)C1 18592,c1(C(N(C(C)CNC(c2ccoc2C)=O)CC)=O)cc(Cl)n(C)n1 18593,N1(C(c2c(OC)csc2)=O)CCOCC1C(=O)Nc1cncc(CO)c1 18594,C1(CC(N2C(CNC(C(C)n3cccc3)=O)CCC2)=O)SC(=N)NC1=O 18595,C(CCC(C(=O)NCc1cccc(Br)c1)N1CCC1CC(C)(C)CCC)OC 18596,C1(CC=C)(NC(=O)Cc2nc(C)sc2C)CCN(C(C2(C)CC2(F)F)=O)C1 18597,c1(CC)cc(NC(=O)C(CC2CCC2)NC(=O)C(C)(O)C2CC2)cc(F)c1 18598,C(CC(F)(F)F)CC(=O)NCc1cn(C2CCN(C(=O)CC3CC(F)C3)C2)nn1 18599,c1(C(=O)NCC23CC(NC(C(c4ccccc4)OCC)=O)(C2)C3)cnn(C)c1F 18600,C1(NC(=NCCN(C(C)=O)C)NC2CCN(CC)CC2)CCCC12CCOCC2 18601,C1(C(N2CCC(C(=O)NC)C2C)=O)CCCCCN1C(=O)CC1CCCC2CC12 18602,C1(CNC(c2cc(C)[nH]n2)=O)CC2CC2N1C(=O)CC(F)(F)Cl 18603,C(CC(=O)NCc1c(C)cccc1O)(C(F)(F)F)NC(C=CC=CC)=O 18604,N1(C(c2c(CC)nns2)=O)CC2CCCC(C1)N2C(=O)C(C)(O)COC 18605,c1(C(N2C(C(C)NC(C(CC)=CCCC)=O)CCC2)=O)nc(O)sc1C 18606,C(=O)(C(C(C)O)NC(=O)COCCSC)NC(CC)CO 18607,C1(C(=O)NC2CCN(CC)C2)(CC)CN(C(=O)Nc2ccccc2)CC1CN 18608,NS(=O)(=O)c1sccc1C(=O)NCCN(C(C1COCCO1)=O)C1CC1 18609,c1(C(=O)NCC2C=CC(NC(CC(CCC)O)=O)C2)cc(F)cc2nc[nH]c12 18610,C1(CCNC(c2c(CC)ocn2)=O)CSCCN1C(C1CCCC1C)=O 18611,c1(C(=O)NC2(C)CN(C(CC(CCOC)(C)C)=O)C2)ccc2c(n1)NCCO2 18612,c1(C(N2CCC23CN(C(C2C4CCCC24)=O)C3)=O)ccc(C(F)F)c(F)c1 18613,c1(NCc2cccc(CN(C)C)n2)cc(=NCc2csc(O)n2)[nH]cn1 18614,c1(C(C(=O)OCCC(C=C)C)NC(=O)CCc2ncc[nH]2)ccccc1C 18615,N1(C(Cc2cn(C(C)C)nc2)=O)CCOC2(C1)CN(C(=O)CCN1CCC1)C2 18616,C1(CCCNC(C(C=CC)O)=O)CN(C(=O)CC=CCCCCC)CCO1 18617,c1(C(=O)NC2CCN(C(c3cn(CCC)nc3)=O)C(C)C2)ccc(C)c(C)c1N 18618,CC1CCC(CNC(=O)OCc2cc(C(N3CCC3C)=O)sc2)N1C.C(C)(C)(C)O 18619,C1(CNC(C(C)(C)OCC)=O)CCC(CNC(=O)CCc2cn[nH]c2)CC1 18620,c1(C(N2C(C(C)(C)NC(CCCNC(C)=O)=O)CCC2)=O)cc(C)nc(C)c1O 18621,N1(C(C(C)=CC2CC2)=O)CCCCC1CCNC(=O)C(n1ccc(C)n1)C 18622,N1(C(c2cc(OC)nn2C)=O)CC(C)N(C(c2cc(C)n(C)c2)=O)CC1C 18623,Cn1nc(Cl)cc1C(=O)N(C1CCCCC1)CCNC(=O)C(F)=C1CCC1 18624,N1(C(c2c(OC(F)(F)F)cccc2Cl)C)CC2CCC(C1)C2N1CCC(C)(O)C1 18625,c1(C(N(CC(C)(C)O)CCOC)=O)cc(C(C)C)ncc1F 18626,C1(NC(CCCCC#C)=O)CC(C2CCN(C(c3c(N)sc(C)c3C)=O)C2)C1 18627,c1(NC(C2(F)CN(C(c3cc(Br)ccc3Cl)=O)C2)=O)cnc2ccc(F)cn12 18628,c1(C2C(n3ccc(C(c4n(CC)nnn4)NCCOC(=N)O)n3)C2)cccc(Br)c1 18629,N1(Cc2c(-c3ccc(CC)cc3)nc(C)s2)CC2(CC=CC2)C1c1ccccc1 18630,N1(CCN(CCC)C(=O)NCC2CC2(F)Cl)CCCCS1(=O)=O 18631,N1(C(C(C2CCC(=O)N2)C)=O)CC2CCC(C1)N2C(c1sc(F)cc1Cl)=O 18632,C(=O)(C(F)(CNC(=O)CCc1ccoc1)C(C)C)NCCC(=C)C 18633,C1(C#N)(CC)CCCN(C(=O)CNC(=O)CNC(C2CCC(C)C2)=O)C1 18634,C1(NC(C2CC(C#C)(O)C2)=O)CCN(C(c2cnnc(C)c2)=O)CC1F 18635,C(=O)(CCCC(=O)N1CCCN(C(=O)CNC(=O)CCCCO)CC1)NCC 18636,c1(C(=O)Nc2nnc(C3CC3)o2)cc2c(s1)CCN(Cc1ncccc1O)C2 18637,CC(O)C(C)(C)C(=O)NCC#CCNC(C1CC(O)CN1C(=O)OC(C)(C)C)=O 18638,C1(C(=O)Nc2cnc(-c3ccccc3)nc2)CCN(C(=O)CCF)CCC1CO 18639,N1(C(c2ccc(C(C)=O)cn2)=O)CC(CNC(=O)Cc2ccccc2)CC(C)C1 18640,C1(C(=O)NCC2CN(C(=O)CO)CCC2(F)F)Cc2cncn2C(=O)N1 18641,c1(OC)cccc(NC(C2(C)CCN2C(c2cccnc2O)=O)=O)c1 18642,C1(NC(CCC#C)=O)COC2(CNC(c3cc(Cl)sc3Cl)=O)CC1C2 18643,C1(NC(C2CN(S(CC)(=O)=O)C2)=O)CC(F)CN(C(c2csc(C(F)F)n2)=O)C1 18644,Cc1ccc(Cl)c(C(=O)NCCCN(C(=O)CN2CCC2C)C2CC2)c1 18645,C1(SC)CCN(C(=O)CCNC(=O)CC2(O)CCCCC2)CC1 18646,c1(OC)ccc(N)c(C(N2CCC(NC(C3(CC(C)C)CCC3)=O)C2C)=O)c1 18647,c1(CS(N2C(CC(=O)O)CCC(C)(C)C2)(=O)=O)cc(Br)cc2cccnc12 18648,c1(C(=O)NCC(C)(C)NC(c2cnn[nH]2)=O)ccc(F)c(F)c1N 18649,CN1CC(F)CC1C(=O)NCC1CCC(C(=O)NCC2(O)CCCC2)O1 18650,CC1(C)OCCCC1C(=O)NCC1CN(Cc2ccccc2)CCCO1 18651,N1(C(CSC)=O)CC(NC(=O)Cn2nc(C)c3cccnc23)C2CCCCC12 18652,c1(C(N(CCC(=O)N(C2CCCC(O)C2)C)C(C)C)=O)cccc(C#N)c1 18653,C1(CNC(c2ccccc2)c2nc[nH]n2)CC(C2CC2)=NO1 18654,C12(C(N(CC(C)O)CCNC(=O)CC(C)(C)C)=O)CC3CC1C2C3O 18655,c1(CNC(C(C2CCC2)OCC)=O)ccc(CNC(=O)CC2CCCO2)nc1 18656,CN1CC(C)(C(N2CC(NC(c3cc(C4CC4)n(C)n3)=O)C3(CC3)C2)=O)CC1=O 18657,C(=O)(C(CC(C)(C)C)NC(=O)OC(C)(C)C)Nc1ccc(C(C)O)cc1 18658,C(C(C)C(=O)NC(C)CNC(c1cnc(-c2ccoc2)s1)=O)OC 18659,c1(CC)cccc(C)c1C(N1CCCC(O)(CCNC(=O)CC2CC2(Cl)Cl)C1)=O 18660,CC(CC(=O)NCC(C1CCCC1)NC(C1(C(F)(F)F)CC=CC1)=O)C1CCCO1 18661,C1(N(C)C(c2cn(-c3cnn(C)n3)nn2)=O)CCCN(Cc2ccc(Cl)nc2)CC1 18662,Cc1cc(C#N)nc(N2CCC(NC(c3ccc(-c4cccs4)[nH]3)=O)C(C)C2)n1 18663,c1(C(=O)NCC(c2ccccc2Cl)N(CC)CC)ccc2c(c1)CC(=O)N2 18664,c1(CC)cc(C(=O)NCC2CCN2C(C2(F)CCCC2)=O)cn(C)c1=O 18665,c1(C(N2C(CC(=O)Nc3ccc(C)c(F)c3)COCC2)=O)c(O)cc(O)cc1O 18666,Cc1cc(-c2cn(C3CC(NC(c4c[nH]nc4Br)=O)C3)nn2)ccc1F 18667,N1(C(Cc2c(C)cccc2)=O)C2CCCC1CN(C(C1CCN(C)C1)=O)C2 18668,n1(CC)cc(Cl)cc1C(N1CC(CCNC(c2ccc(C#N)[nH]2)=O)C1)=O 18669,N1(C(=O)CCc2nnc(C3CC3)o2)CC2(CCN(C(C34CCCC3C4)=O)C2)C1 18670,C1(C(=O)NCCc2c(C)n[nH]c2)CCN(C(c2cc(C(N)=O)co2)=O)CC1O 18671,C1(C)(C(=O)NCC2(NC(C3CCCN(C)C3)=O)CC2)Cc2ccccc2C(=O)O1 18672,c1(C(=O)NCC(CC)N(C(=O)C=Cc2ccc(C)s2)C)ccc(=N)[nH]c1 18673,C1(=CCNC(C2CCC(OC)C2)=O)CCN(C(=O)CCC2(C)CC2)CC1 18674,C(=O)(NNc1ccc(F)c(Br)c1)NCC1=NOC(C)C1 18675,N1(CC)CCC(NC(=O)OC(C)(C)C)CC(C)(C)C1.C(=O)(C)N(CC(C)C)C(C)C 18676,C1(NC(CSCC=C)=O)CC2(CCN(C(=O)C=Cc3cncc(C)c3)C2)C1 18677,CCC(C)(CCNC(=O)CCCC1CCCO1)NC(=O)CC1(C)CC1 18678,c1(C(=O)NCC(C)CNC(C2(C(F)F)CCCO2)=O)ncccc1Cl 18679,c1(OC)ccc(F)c(F)c1-c1cncc(C(N2CCN(C3CCCC3)CC2)=O)n1 18680,C1(CNC(C(C2CCOCC2)C)=O)CC2CCC(C1)N2C(C1CCS(=O)(=O)N1)=O 18681,C1(OC)CN(C)C(C)(C(N2CCCCC(CNC(C3(O)CCCCC3)=O)C2)=O)C1 18682,C1(CNC(c2c(C)n(C3CC3)cc2)=O)CN(C(=O)C(C)SC(F)(F)F)CCCO1 18683,N1(C(C(COC)OC)=O)CC(NC(c2ccc(OC)c(Br)c2)=O)CC1(C)C 18684,Cc1cnccc1CNC(=O)C(CCF)NC(c1cnccc1C)=O 18685,C#CCC(C)(C)C(=O)N1CCC(C)C(NC(c2cncc(C(C)C)c2)=O)C1 18686,c1(Nc2scc(CC(=O)NC(C3CCC3)C)n2)cccc2c1OC(F)(F)O2 18687,c1(OC)ccnc(C2CCN(C(C)C(=O)NC(C)Cn3cc(C)cn3)CC2)c1 18688,Clc1scnc1C(c1nc(C2CC2)no1)NCc1nnnn1CC1CC1 18689,OC1COc2c(NCc3cc(Cl)sc3Cl)cnn2C1 18690,C(C(C(=O)N(C)CC1(O)CCOC1)C(C)C)NC(C(COCC)C)=O 18691,c1(C(N(CCCNC(C2CCN(CC(C)C)C2)=O)C)=O)cc(Cl)cc2c1OCC2 18692,C#Cc1cccc(CC(=O)NC2CCOC2C(N2CCNC(=O)C2CCC)=O)c1 18693,C1(CNC(C2N(C)CC(O)C2)=O)CC2(CCC2)CN1C(=O)CC1C=CCC1 18694,Cc1ccnc(C(=O)NCC2(NC(=O)C=CS(C)=O)CCC2)n1 18695,C(C(F)(F)C(=O)NCCC(CNC(=O)Cc1ccon1)OC)OC 18696,c1(C(N(CC(=O)NC2(CC(=O)OC)CC2)CC2CC2)=O)nnnn1C 18697,C=CCCCC(C)(C)C(=O)N1CCC(NC(c2ccc(C)c(Br)c2C)=O)C1 18698,C=CCN=C(NCCc1ccc(N2CCCC2)nc1)NC(C)C 18699,N1(CC2(NC(CCOC)=O)CC2)CCN(C(C2OCCOC2C)=O)CC1 18700,c1(N(CC(CN(C)C)(C)C)C)nc(N2CCC(C)(C)C2)nc2c1SCC2 18701,C(=O)(C(C)(C)CC(=O)OC)NCC(CC=C)C(=O)Nc1ccc(Cl)cc1 18702,n1(C(CCO)C(N)=O)cnc2c(N3CC(N(C4CC4)C(=O)C4CC4)C3)ncnc12 18703,c1(C(N2C(CNC(C(C)NS(C)(=O)=O)=O)CC2)=O)ccc(C2CC2)cc1F 18704,CC#CC1CCN(C(=O)C(C(C)C)n2cnc(C(F)(F)F)c2)C1 18705,C#Cc1ccc(C(=O)NC23CC(NC(=O)CC4(C)CC4(Cl)Cl)(C2)C3)cc1Cl 18706,c1(C(=O)NCCOCCNC(C(C)SCC)=O)ccc2cn(C)nc2c1 18707,C(=O)(C1CCCn2cnnc21)NC1C(CNC(c2cccc(C(C)C)c2)=O)C1 18708,CC(C)CC(C)CC(C)C(=O)N1CCN(C(c2c[nH]c3nccc(Cl)c23)=O)CC1 18709,C(=O)(N(CCC(=O)OC)OC)C1CC2CN(C(c3c(NC)cccc3)=O)CC1C2 18710,c1(C(N(CCCN(C)C(C2(O)CCOC2)=O)C)=O)cccc(O)c1F 18711,Cc1ccc2oc(C(=O)NC3CC(CNC(c4cc[n+]([O-])cc4)=O)C3)cc2n1 18712,c1(C(N2CCC(NC(CCCOCCC)=O)C(C)C2)=O)cnc([N+](=O)[O-])n1C 18713,C(C(CNC(C1(c2cc(C)no2)CC1)=O)C(F)(F)F)NC(C(COC)(F)F)=O 18714,C(=O)(C#CC1(C)CCCO1)N(C(C)CNC(=O)Cc1cnn(C)n1)C 18715,CC1=NOC(C)(C(=O)NCC2(C(N)=O)CN(C(=O)CSC(F)(F)F)C2)C1 18716,C1(O)(CNC(c2c(CC)occ2C)=O)CCN(C(=O)C=CCOC(C)(C)C)CC1 18717,N1(C(C(N2CC(CNC(CC3CCN(CC(C)C)C3)=O)C2)=O)C)CCN(C)CC1 18718,CC(C(=O)N1CCC1CNC(C1CSCN1C(c1ccco1)=O)=O)C(C)(C)C 18719,N1(C(C(=O)Nc2ccc(Br)cn2)=O)CCCC(O)(C(c2ccccc2)O)C1 18720,C1(CC(=O)NC2CCN(C(c3cnc(S)nc3)=O)CC2O)CC2CCC1CC2 18721,N1(C(c2c(COC)ccs2)=O)CCCCC2(CCN(C(c3cnc[nH]3)=O)C2)C1 18722,N1(C(c2ncc(OC)cn2)=O)CCC(NC(c2cc(C)c[nH]2)=O)C(C)(C)C1 18723,c1(CC(=O)N(CCCNC(C2CCN(CC(F)(F)F)C2)=O)C)cc(F)ccc1F 18724,C1(C(C)C)CNC(=O)CN1C(C1CC12CC(NC(c1nccn1C)=O)C2)=O 18725,C1(OC)CC2(C1)CN(C(=O)C(CNC(c1ncccn1)=O)C(C)C)C2 18726,C1(NC(NC2OCCC(OC)C2)=NCC2CCCCC2)Cc2nccnc2C1 18727,C1(CC(=O)N(CCn2cnc(C)c2C)CC)CC(NC(=O)OC(C)(C)C)C1(C)C 18728,N1(C(c2ncn(C)c2)=O)CC(NC(=O)CSc2nc[nH]n2)C2(CC2)C1 18729,O=C(C#CC1CCCC1)NC1(CNC(c2cc(NC3CC3)ncc2Cl)=O)CC1 18730,C(=O)(C1=CCC(C)(C)CC1)NC1CC2CN(C(CC(C(C)C)O)=O)CC21 18731,Nc1c(C(N2CCC(CNC(=O)Cc3ccon3)C2)=O)cccc1Cl 18732,C1(NC(CCC)=O)CCC12CN(C(=O)CCC(c1ccccc1)N(C)C)C2 18733,Cc1ncc(NC(C2CC3CC3N2Cc2cccc3nonc23)=O)c(C)c1Br 18734,N1(C(C(F)=C(C)C)=O)CCOCC(C(=O)NCc2cc(F)ccc2F)C1 18735,Nc1c(C(N2CC3CC3(c3cccc(OC(F)(F)F)c3)C2)=O)ccnc1Br 18736,CC1=CCC(C(=O)NCC2CC2NC(c2ccc(NC3CC3)nc2)=O)CC1 18737,c1(CNC(=O)COCCNC(C2C3CCCC23)=O)ccnnc1 18738,C(C(C)(C)C(=O)N1CCC(c2ncc[nH]2)C1)N(C(C(C)c1cccs1)=O)C 18739,C1(CNC(C(CC=C)NC(C)=O)=O)CN(C(c2c(Cl)n[nH]c2C)=O)CCN1C 18740,Cc1cc(C#N)ccc1C(N1CCC2(CC2NC(C2CC3(CCC3)CO2)=O)C1)=O 18741,CCCCCCCCC(C)CC(=O)NCc1ccc(OC)cc1 18742,C#CC1CCCC(CNC(=O)C(C(C)C)NC(C2C(C#N)C2(C)C)=O)C1 18743,C1(CC)(CO)CCN(C(C2CSCN2C(=O)C(C(=O)OC)OCC)=O)C1 18744,C(=O)(C(C)CCCC(C)=O)N1C(CNC(c2ccn(CC)n2)=O)CCC1 18745,N1(C(C2CCC(n3cc(C(C)O)nn3)C2)=O)CCC(O)(c2ccc(F)cc2)CC1 18746,N#Cc1cc(NC(=O)NCC23CC(CCO2)C3)co1 18747,c1(OC)ncccc1C(c1nnnn1C)NC(C1CCC1)C 18748,c1(C(N2CCC(N(C)C)C2)=O)cccc(F)c1Cl.C1(C#N)(C2(CC(=O)N)CC2)CC1 18749,N1(C(C(c2cccnc2)C)=O)CCC2CC(CNC(=O)CCF)CCC2C1 18750,C1(CC(C)C)CC(C(=O)NCCCNC(c2cc(=O)cc[nH]2)=O)CC(=O)N1 18751,C1(CC=C)(C(=O)NCc2csc(C)n2)CN(C(=O)C(C)N2CC(C)C2)C1 18752,N1(C(c2cc(CC)nn2C)=O)C2CCCC1CC(NC(C1CC1(C)Br)=O)C2 18753,c1(CN2C(C(=O)OC)(CO)CCC2)cc2nccc(Cl)c2s1 18754,N1(C(=O)NCC(c2cccc(C)c2)C)CCCC(O)(c2cnn(C(C)C)c2)C1 18755,C12(NC(=O)CC3CCOCC3)CCCC1N(C(C1CC1(Cl)Cl)=O)CC2 18756,c1(CC)nccnc1C(=O)NCC1CCN1C(=O)C(=CC1CCCC1)C 18757,C(=O)(NNc1cccc(F)c1OC(F)(F)F)Nc1n(C)cc(Br)n1 18758,CC1(C)CCCCC1C(=O)NCC(C)(C)CNC(=O)CC12CC(C1)C2 18759,N1(C(CCCNC(=O)OC)=O)CC2(COC(CNC(=O)C(C)C)C2)C1 18760,S(=O)(=O)(c1ccc(F)cc1)N1CC(NC(C(=O)NC2CC(C)SC2)=O)C1 18761,c1(CN2C(C(=O)NC(CC)C(=O)OC)CC(F)C2)ccc(C#N)cc1[N+](=O)[O-] 18762,C1(NC(C(C)OC2CCCC2)=O)CC2CC1N(C(=O)CC1(O)CCOCC1)C2 18763,C12(NC(CCc3ccnc(C)n3)=O)CCCC1N(C(=O)COCC(F)F)CCC2 18764,Cc1cc(Cl)cc(C(=O)NCC2(NC(C3CCC(=O)N3)=O)CCCC2)c1C 18765,C=CC(CCC)CC(=O)N1CC(C(=O)NCC2CCOC(C)(C)C2)C(F)(F)C1 18766,c1(OCCCC)cc(C)ccc1C(=O)NC1(C(=O)N(C)C)CC1 18767,C1(C(=O)NCC(C)NC(c2ncc(OC)nc2)=O)COCCN(C(C)=O)C1 18768,c1(C(N(C)CCNC(C2CC2C2CCC2)=O)=O)ccc2ccc(Br)cc2c1 18769,c1(C(=O)NCC(CCCC)NC(=O)C(C)CF)ccc2n[nH]c(C)c2c1 18770,N1(C(c2c(C)nc(N(C)C)s2)=O)CCC2C(CCCN2C(c2cscn2)=O)C1 18771,c1(CNC(=O)NC2CCC(N(C)C)CC2)cc(C#N)ccn1 18772,C1(NC(C(C)O)=O)CCN(C(C2Cc3ccncc3N2)=O)CC1(C)C 18773,c1(C(=O)OC)ccc(C(=O)N(C)CC2CN(C(=O)C(C)c3ccco3)C2)c(Cl)c1 18774,C1(C(=O)NCC(C2C(C)C2)C)N(C(c2coc(N(C)C)n2)=O)CC12CCCC2 18775,CCC(CC(=O)NCC1CN(C(C2(C(F)F)CCCC2)=O)CCO1)C(C)C 18776,C(C)(N=c1[nH]c2c(c(=NCCCC3(C)CC3)[nH]1)CCC2)c1nnc(C(C)C)n1C 18777,Cc1nnn(CC(=O)NC(C2CC=CCC2)C(=O)N(C(CF)CF)C)n1 18778,c1(CC)cc(C(=O)NC2CCCN(C(=O)C(C)OC)C2)cc(C(F)(F)F)c1 18779,C1(F)(C(N(C(c2ccccc2)CNC(=O)CC(C)(C)O)C)=O)CCC(F)(F)CC1 18780,C1(CNC(CCSC)=O)CC2(CCN(C(c3cc(C(F)F)ccn3)=O)CC2)CO1 18781,C(=O)(CCCS(C)(=O)=O)N1CCN(C(CNC(CCNC(C)=O)=O)=O)C(C)C1 18782,c1(C(=O)NC(C2CCN(C(=O)CCc3ncc[nH]3)CC2)C)cc(Cl)cnc1O 18783,CCC(CCCC(=O)NCc1cc(C)cc(C)c1)NC(C1(Cl)CC1(F)F)=O 18784,c1(C(=O)OC)cnc(NC2CC(C)(NC(=O)C(c3ccc(F)cc3)F)C2)c(Cl)c1 18785,N1(C(CCSCCCC)=O)CCC(NC(C23CSCC2C3)=O)C1 18786,Cc1cc(CNC(C2CC2C2CC2)=O)oc1C(=O)NC1(C(N)=O)CCOC1 18787,CCC(C)(C)C(=O)N1CCOC(CCNC(=O)CCn2cncn2)C1 18788,N1(C(C2C(CC)CN(C(=O)C(C)(C)CO)C2)=O)CCCC(O)(C(N)=O)C1 18789,N1(C(c2c(OC)nsc2)=O)CCC(NC(c2sccc2Cl)=O)CC1 18790,c1(N(C)CCc2ccccc2F)nc(=NCC2(C)CCCCC2)[nH]c2c1CCC2 18791,n1(C(C)C)cc(C(=O)NCC(C2CCN(C(=O)COC3CCCCC3)C2)F)cn1 18792,c1(CC(=O)NC2CC(C)N(C(c3cccn(O)c3=O)=O)C2)c(F)cccc1F 18793,N1(C(CCCCSC)=O)CC2(C1)CN(C(C1CCN(CC(C)C)C1)=O)C2 18794,O=C(C1=CCCOC1)NCCCCNC(C1CCCCS1)=O 18795,CC1CCC(C)(C(=O)NC2CC2NC(c2ccnc(OC3CCC3)c2)=O)C1 18796,N1(C(C#C)C)CCN(C(=O)C(CCF)NC(c2cnncc2C)=O)CC1 18797,C(=O)(Nn1cccc1)C1C(C(=O)CCC)C1.OC 18798,c12cc([nH]n1)CS2.C1(C(=O)NCC(CO)NC(=O)OC(C)(C)C)CC(C)=NO1 18799,Cc1cccc(C(=O)NC(CC(=O)NC2CCCCC2)C2CC2)c1N 18800,c1(OC)ccc2c(c1)cc(C(=O)N(CCNC(c1cn(C)nn1)=O)C1CC1)n2C 18801,N#CC1(C(=O)NCCCNC(C2CCCN2C2CCOCC2)=O)CC2(CCC2)C1 18802,C1(C(=O)NC(C2CCN(C(C3COC(=O)O3)=O)CC2)C)CCSC(C)C1 18803,C1(F)(CNC(c2ccnc(O)c2)=O)COCCN(C(=O)C(O)c2cnc[nH]2)C1 18804,Cc1cc(C)c(C(=O)NC(Cc2ccoc2)C(=O)NCc2ccc(C#N)s2)s1 18805,C1(C(C)C)N(C(=O)OC(C)(C)C)CC12CCN(C(n1nc(CO)nc1Cl)=O)CC2 18806,N1(C(CCN(C(=O)C(n2ccc(C)n2)C)CC#C)=O)Cc2cccc(F)c2C1 18807,CC(C(=O)NC1(CF)CCN(C(c2cc(=O)n(C)o2)=O)C1)C(F)(F)F 18808,C1(C(=O)NCC2CC(F)CN2C(C2(F)CCCCC2)=O)CCCC1C1CC1 18809,c1(C(=O)OC)ccc(C=CC(=O)NC2CCN(C(=O)C=CCOC)C2C(C)C)o1 18810,C(=O)(C1=CCOCC1)N(C1CCCN(C(c2c(SC)cccn2)=O)C1)OCCF 18811,C(=O)(CC(C(F)F)C(C)(C)C)N1CC(CN(CCC(O)C(=O)OCCCN)C(C)(C)C)C1 18812,Cc1cc(Cl)cc(C(N2CCCC2CCNC(c2ncnn2C)=O)=O)c1O 18813,Cc1cc(NC2CNC3(CCCC3)C2)c(C#N)cc1NC(C)C 18814,C1(C(=O)OCC)CC=CC(NC(=O)C(C(C)C)OC)C1.n12ncnc1C2 18815,C1(NC(CCN(CCC)C)=O)CCCCC12CCN(c1nc(Cl)nc(C)c1Cl)C2 18816,c1(CCC(=O)NC2CN(C(=O)Cc3ccoc3)C2)cccc(F)c1 18817,c1(C(=O)NC2CCC(NC(CNC(C)=O)=O)C2)cnc2cc(C)ccc2c1 18818,c1(C(=O)OC)ccc(CC(C)C)nc1N1CC2CC(NC(=O)CC3(C)CC3)C2C1 18819,c1(C(=O)NCCCCC2CN(C(C3C(C)CC3)=O)C2)cc(Cl)ccn1 18820,N1(C(=O)C2=CCCCC2)CC2CC(C1)N(C(=O)CNc1ccccc1[N+](=O)[O-])C2 18821,c1(OC)ccc(-c2ccnc(C(N3CCC(F)(c4cn(CCO)nn4)C3)=O)n2)cc1 18822,c1(C(=O)OC)sc(C(N2CCC(NC(c3c(C)coc3C(C)C)=O)C2)=O)cc1N 18823,c1(C(=O)NC2(c3cccc(C(=O)OC)c3)CC2)cc(C)cc(C)n1 18824,CC1=NS(=O)(=O)NC=C1C(=O)N1CC(CNC(=O)CSc2ccccn2)C(C)C1 18825,c1(C(=O)NC(C(C)C)CCNC(C2(N(C)C)CC2)=O)nn(C)c(C(F)(F)F)c1Cl 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19143,c1(CC)[nH]c(C(=O)NC2(C)CC(NC(=O)C(C)(O)CC)C2)nc1Cl 19144,Cc1ccc(F)c(C(N2CC3CC2C3NC(=O)C2=CCOC2)=O)c1 19145,C1(C)(NC(CCOC)=O)CCCN(C(C2OCCO2)=O)C1 19146,N1(C(C2CSCCN2C(=O)CN(CCO)CCO)=O)CCc2ccccc2C1 19147,c1(C(N(CCCOCCNC(C(CC)=CC)=O)C)=O)ccc(CC#N)cc1 19148,N1(C(CN(S(CC)(=O)=O)C)=O)CC2OC(=O)N(C3CCN(C(=O)CO)C3)C2C1 19149,Cc1c(NC(C2CC(C)CN2C(C2(C(C)C)CCC2)=O)=O)cc(Cl)cc1Br 19150,c1(SC)nc(=NCC(C)NC(c2ccc3cc[nH]c3c2)=O)s[nH]1 19151,C1(CNC(COCCCC#C)=O)CCC(C(=O)NC2(C(=O)N(C)C)CC2)CC1 19152,c1(C(=O)NCCCN(C(C2(C)CC(=C)C2)=O)C2CC2)ccnc(C2CC2)c1 19153,N1(C(c2ccc(C)n2C)=O)CCN(C(c2n[nH]cc2F)=O)C(CS(C)(=O)=O)C1 19154,C(C#Cc1cn(CCO)nn1)NC(C1CC(=O)N1Cc1cccs1)=O 19155,O=C(N=c1[nH]ccc2cc(Br)ccc12)C1CC(F)CN(Cc2ccc(Cl)cc2)C1 19156,C1(CNC2C(C)CN(C)CC2)CCCCCCC1(C)C 19157,C(=O)(CCCC(F)F)NCC(C1CCCCN1C(=O)C1=NOCC1)(C)C 19158,c1(CC)ccnc(C(=O)NCC#CC(N2CC[Si](C)(C)C2)=O)c1 19159,N1(C(c2c(CC)ncs2)=O)CC2CC(C1)CN(C(=O)C(C)(O)CC)C2 19160,N1(C(C2(CC#C)C=CCC2)=O)CCC2(CCC(NC(=O)Cc3ccsn3)C2)CC1 19161,C1(C(N(C(=O)CN2CCOC(c3cccs3)C2)C)=O)CC2(CCCO2)C1 19162,NS(=O)(=O)N1CC(NC(=O)COC2CCN(C(C3(COC4CC4)CC3)=O)CC2)C1 19163,c1(CC)noc(C(=O)N(C2CN(C(c3cn(C(C)C)nc3C)=O)C2)C)c1C 19164,C(=O)(C(C#N)NC(c1ccccc1)=O)NC(C1CCCO1)CNC(=O)OC(C)(C)C 19165,C1(CNC(C(C)OCC)=O)CN(C(=O)Cc2sc(C)cc2C)CC1O 19166,c1(C(=O)NCC(C2(O)CN(C(C(C)OCC)=O)C2)(C)C)ccc(Cl)c(F)c1 19167,C1(CN(C)CC2CC2(C)C)CCC(=O)N(C(c2ccc(Br)cc2)=O)C1 19168,N1(C(c2ccc(NC(C)=O)c(F)c2)=O)CCC(C)(C)C(c2ccccc2)C1 19169,CC1CC(C)(C)N1C(=O)C=CCC(C)(C)NC(=O)CSC(C)(C)C 19170,c1(C(=O)NCC(C)N(C(Cc2cc(COC)on2)=O)C)ccn2c1CCCC2 19171,C1CCCCC(N2CCCC2COC(C)(C)C)C1=O.C1(CNOC)CCCO1 19172,CC(c1ccccc1)=CC(=O)NCC1CC(NC(c2cc(Cl)nn2C)=O)C1(C)C 19173,C1(C(=O)O)CN(Cc2cnn(C3CCCCO3)n2)C2CCOCC12 19174,C(=O)(C(C(C)C)NC(C)=O)N1CCC(OCCNC(C2(C)CC(=C)C2)=O)C1 19175,N1(C(c2c(CC)oc(C)c2)=O)CCN(C(=O)CC(O)CC)C2COCC12 19176,c1(CCC)ccc(C(=O)NC2CCN(C(=O)CCS(C)=O)C2C)cc1[N+](=O)[O-] 19177,CCC(C)(CC)C(=O)N1CCN(C(c2sc(C)nc2C)=O)C(CC(F)(F)F)C1 19178,N1(C(=O)NC(C)Cc2ccccc2)CCC2(CCC2(C)C)C1 19179,c1(C(=O)NC2CC(CNC(COC)=O)C2)cc(NC(CC)=O)c(O)c(Cl)c1 19180,N1(C(C2C(C(N)=O)C2)=O)CCC(C(=O)NC2CC(CO)C23CCC3)=C(F)C1 19181,c1(C(=O)NC(C)C(C2CCCCC2)NC(N)=O)cn(CC(F)(F)F)nc1C1CC1 19182,N1(C(C2CCC=CCC2)=O)CCN(C(=O)CC2CCC3(CCC3)O2)C(C(F)F)C1 19183,CC1CCC(CN)N1C(=O)NCCC=CBr 19184,C1(N(C)C(c2ccncc2O)=O)CCN(C(c2cnc(-c3ccoc3)s2)=O)CC1 19185,Cc1c(C(N2CC(F)(CNC(=O)COC3CCCCC3C)C2)=O)cnn1CCO 19186,Cc1nc2c(C)cc(C(=O)N(C(CO)CC(C)C)C)cn2n1 19187,c1(C(N(CC(CC)NC(c2c(F)ccc(C)c2Cl)=O)C)=O)cccc(S(C)=O)c1 19188,C1(C(N(C(C)CNC(c2ccc(OCF)cc2)=O)CC)=O)CC(F)(F)C1(C)C 19189,N1(C(c2c(CCC)[nH]cc2)=O)CCC2(CCC2)C(NC(=O)CCS(N)(=O)=O)C1 19190,CCC(CC1CCCC1)C(=O)N1CC(COC)(NC(=O)Cc2nonc2C)C1 19191,c1(C(N2CC(CN(C(C(C(C)OC)O)=O)C)C2)=O)cn2ccccc2n1 19192,CC1CCC(CNC(=O)CC(C)(C)O)N(C(c2csnn2)=O)C1 19193,C(=O)(CCCCCC#N)NCCC1CCCN(C(c2c(C)noc2C(F)F)=O)C1 19194,C(=O)(C1COc2ccccc21)N1CC(CN(C(C(C)OCC2CCCO2)=O)C)C1 19195,C1(CC(=O)NCCC(C)N(CCC)C)CCN(C(c2cscc2C)=O)C1 19196,c1(CNCc2ccc(F)nc2)c(F)cc(Cl)cc1Cl 19197,C1(C(C)(C)C)(CNC(C(C)Cc2cnco2)=O)CCN(C(=O)CNC=O)C1 19198,N1(C(CC)C)CCN(C(=O)C(CCF)NC(C2CCC(C(N)=O)C2)=O)CC1 19199,C(=O)(CC(C)(C)C)NC(C1CCN(C(c2cnc(C(=O)O)[nH]2)=O)CC1)C 19200,[N-]=[N+]=NCCCCCC(=O)NC1CCCC(NC(=O)CC(F)(F)F)CC1 19201,C1(CNC(c2ccc(C(F)(F)F)s2)=O)CC2(CCC2=O)C1 19202,CCC(CC)(CO)NC(c1cncc(CNC(C2CCN(CC)C2)=O)c1)=O 19203,CCCC(O)(CCC)CC(=O)N1CCC(NC(c2ccc3nccn3c2)=O)C1 19204,N12CC(C3(CC3)C1)CC(=O)NCCOCCOCC2=O.C(CC(C)C)OCC 19205,C(=O)(C(CCCOC)N1CC(C(=O)OC)C(C#N)C1)N(CCS(C)(=O)=O)CC.CCN 19206,C#CC1(C(=O)NCC(C)(F)C(C)(C)F)CCN(C(C)=O)C1.C1C(=O)NCCS1 19207,C1(NC(Cn2c(C(C)C)nnn2)=O)CC2CCC(C1)N2C(=O)C(C)(Cl)Cl 19208,C(=O)(C(F)C1=CCCCC1)N1CCC(C(C)NC(=O)COCC2CCCC2)C1 19209,c1(NC(c2cccnc2)CC)nc2ccccc2nc1NCC1CCC(C)CC1 19210,C(=O)(NNc1ccc(S(=O)(=O)N(C)C)cc1)NCCOc1c(OC)cccc1 19211,C(c1ccoc1)=CC(=O)N(C(C)CNC(=O)Cc1[nH]cnc1C)CC 19212,C1(NC(C(c2ccccc2)NC(C2CCC(=C)CC2)=O)=O)CCCC(C)(C)C1 19213,c1(C(=O)NCc2cc(C)ncn2)coc2c1CN(C(=O)C(c1ccccc1)C)C2 19214,C(=O)(CC(CNC(C1C=CCS1)=O)OC)NC1CCN(CC)C1 19215,C(CC1CC1)(C(=O)NCC(C)C1CCC1)NC(CSCC)=O 19216,C(CCCCCn1cc(CCn2cncn2)nn1)N(C)C(C1(C)CCOC1)=O 19217,C(C(C(C)C)NC(c1ocnc1C1CC1)=O)NC(CC1(NC(C)=O)CC1)=O 19218,C(=O)(C(CC)N(C(=O)CC1(COC)CC1)C1CC1)N(CC(CC)OC)C 19219,C=C(Br)CCC(=O)NC(C1CCN(C(C2(c3n[nH]cc3C)CC2)=O)C1)C 19220,c1(C(C)=O)cc(C(=O)NC(CNC(c2cc[nH]c2C)=O)C2CCC2)cs1 19221,C(CCSC)(C(=O)NC(C)(C)C(C)NC(=O)COCCc1cccs1)OC 19222,c1(C(=O)NCC(C)(CO)NC(c2nc(Br)c[nH]2)=O)c(F)cc(F)cc1F 19223,C1(C2CC2)(NC(C2CC(F)(F)C2)=O)CCN(C(C2CCCN2C2CC2)=O)C1 19224,c1(C(C)C)nc(NCCCC2CC2)cc(=NC2CCC3CC2C3(C)C)[nH]1 19225,CN1CC(NC(=O)CC2CN(C(C3CC4(CC4)C3)=O)CCO2)C2(CC2)C1 19226,CC1=C(C(=O)N2CC3=C(C2)CN(C(c2c(C)ncn2C)=O)C3)C(=O)OC1(C)C 19227,N1(C(CCCC(C)=O)=O)CC(C)CN(C(=O)Cc2cc[nH]n2)C(C)C1 19228,c1(C(=O)OC)cccc(CCCOC2CC(SC(C)C)C23CCC3)c1F 19229,C1(CNC(CC2CC(CC)C2)=O)(NC(C2CCCC(=O)C2)=O)CCCCCC1 19230,CC(CC(=O)N1CCCCC(NC(=O)CCCN2C(=O)CCC2=O)C1)C(F)(F)F 19231,C1(NC(C(C)(C)CF)=O)CCN(C(=O)Cn2ccccc2=O)CCC1CO 19232,CC1CC(NC(c2cc(C(C)(C)C)n[nH]2)=O)CCN1C(=O)CC1CCC2CC12 19233,CCC(C(=O)OC)C(=O)N1CCN(C(=O)CCOCC(F)(F)F)C(CO)C1 19234,c1(C(=O)NCC2C(C(=O)NCC(C)(C)OC)CCC2)csc(C#N)c1 19235,N1(C(C(COCC)C)=O)CCC2CN(C(=O)C=CC3CCCN3C)C2C1 19236,c1(C(=O)NC2(COC)CN(C(C3(OC(C)=O)CC3)=O)C2)nccc(C)c1N 19237,CCCC(C)CCNC(=O)CCOCCNC(=O)CC1CCOC1(C)C 19238,Cn1cnc(CCNC(=O)CC2CCN2C(=O)CC2(N(C)C)CCC2)n1 19239,c1(C(n2cc(Cl)cn2)C(=O)OC)ccc(O)cc1.N1(C)CCCC1=O 19240,C1(=O)C(C(C)(C)C)n2cc(nn2)N1.CS(=O)C1CN(Cn2cc(CO)nn2)C1 19241,CCC(C)(CNC(C1(NC(=O)CC2CCCOC2)CC1)=O)CC 19242,c1(NC(Cc2nccc(CC)c2)=O)ccc2c(c1)CCC2N(C)C 19243,C12(NC(C=CCCC)=O)CC(NC(=O)Cc3nnc(O)s3)(C1)C2 19244,C1(C(N(C)CC2(N(C)C)CCC2)=O)CC12CCCCC2.C1(=O)C(C)(C)CN1 19245,Cc1ccc(C(=O)NC2CC(N(C(=O)CC(C)C3CC3)C)C2)c(O)c1C 19246,C(=O)(C1=NOC(CNC(C2CNC(=O)C2)=O)C1)NCCOCCCC 19247,c1(NC)c(C(=O)NC2CC3(NC(=O)C#CC4(C)CC4)COC2C3)cccc1F 19248,c1(NCC(C(CC)CC)CO)[nH]c(=NCCC(C)c2cn[nH]c2)nc2ncn(C)c12 19249,Cc1nc(-c2ccco2)ccc1C(=O)NCC1CN(C(=O)C(C)(C)O)CC1C 19250,C(CCN(C)C)(CN=c1[nH]c(=NCc2cscn2)[nH]c2cc[nH]c12)OCC 19251,N1(C(COC(C)C)=O)CC2CN(C(=O)Cn3nc(Cl)ccc3=O)CC2C1 19252,c1(C(=O)NCCOCCNC(C(C)NS(CC)(=O)=O)=O)ccc(CO)cc1F 19253,C1(c2cn(CC3C(CC(N4CCCOCC4)=O)CCC3)nn2)CCCS(=O)(=O)C1 19254,C1(C(=O)NC2(CO)CN(C(CC3(C)CC3F)=O)C2)CC2(C1)CC1(CCC1)C2 19255,C(=O)(CCC(=O)NN(C)C)N1C(CNC(c2ncn(C(C)C)c2)=O)CC(O)C1 19256,N1(C(C2N(CCC)CCC2)=O)CCOCC(NC(=O)C(CO)N(C)C)C1 19257,C1(C)(C(=O)NC2CCN(CC)C2)C=CCN1C(c1cc(Cl)cs1)=O 19258,c1(C(=O)NC(C(C)C)CCN(C)C(c2coc(Cl)n2)=O)cc(F)ccc1N 19259,c1(CNC(=NCc2ncc(C)c(O)c2)NC2CC2)cccc(Cl)c1[N+](=O)[O-] 19260,C1(c2cn(C)nc2)CN(C(C2C3CCCCC23)=O)CCN1C(C1(CCF)CC1)=O 19261,N1(C(c2c(C)cc(C)cc2O)=O)C2COCC1CC(NC(C1(C)CCOC1)=O)C2 19262,c1(C(=O)NCC2N(C(C(C(C)C)C)=O)CCC2)ccn(C(=O)OC(C)(C)C)n1 19263,C1(OC)CCC2(C(=O)NCC#CCNC(C3CCCCN3C)=O)CCC12 19264,Cc1ccc(Cl)c(C(=O)NC2CC(CNC(=O)Cc3nccn3C)C2)c1N 19265,C1(C(=O)NCC23CC(CN2C(c2sccc2Cl)=O)C3)(OC)CCS(=O)(=O)C1 19266,CC1CCc2sc(C(N3CC4CCCC3C4CNC(=O)C(C)C)=O)cc2C1 19267,C12(C(=O)NCCC(C)N(C(=O)C(C)OCC3CCCO3)C)C=CC(CC1)C2 19268,N1(C(C=CC(C)(C)NC(c2c(C)n(C)nn2)=O)=O)CCC(C)C2(CCC2)C1 19269,C1(CC(N2CCCC(CN(C(=O)COC3COC3)C)C2)=O)CCCNC(=O)C1 19270,c1(C(N(C2CCCCC2)CCNC(C(C2CCOC2)OC)=O)=O)c(C)ccn1C 19271,C1(NC(C2CCC=CCCC2)=O)CCC2CN(Cc3ccncc3Cl)CC2C1 19272,C(CN=c1nc(C2CC2)[nH]s1)NC(CCN(CC)CC)=O 19273,c1(C(N(CCN(C(=O)Cc2ccc(F)cc2F)C)C)=O)ccc(F)c2[nH]ccc12 19274,N(C(=NCC#CC1CCCCO1)NC1CC1)C(C(CC)CC)COC 19275,C1(C(C)=O)CCC(NCC2(C(F)(F)F)CCC(N)C2)CC1 19276,c1(OC)ccc2cc(C(=O)NCC3CN(C(=O)C(C)S(C)(=O)=O)CCO3)[nH]c2n1 19277,C1(NC(c2c(SC)nn(C)c2)=O)CC2CCC1CC2NC(C1(C)CNC(=O)C1)=O 19278,c1(NCC2CC(C)C2)cc(N2CCOC(NC(C)=O)C2)ncn1 19279,CC(C)C(C(C)NC(c1sccc1C1CC1)=O)NC(=O)CCc1ccc[nH]1 19280,C=CC1COCC1NC(=O)CNC(=O)C(C)(C)CC 19281,c1(NC(C(C2CCC2N(C2CC2)CC2CCOC2)OC)=O)n[nH]cc1C(C)C 19282,N1(C(C2CCC(CC)CC2)=O)CCCC2(CCC2NC(=O)Cc2cnn(C)c2)C1 19283,CCCCCCCCC(=O)N(CC(O)CNC(=O)CNC(c1ccoc1C)=O)C 19284,c1(C(=O)Nc2scc(C)n2)cccnc1CNC(c1ccncc1)=O 19285,N1(C(C(C)OCC)=O)CC(NC(=O)C=C(C)C(C)C)CC(F)C1 19286,c1(NCC(=O)NC(CNC(C(CC(=C)C)OC)=O)C)cccc([N+](=O)[O-])c1 19287,C1(NC(c2c(C)scc2)=O)CCCC(N(C(=O)C=CCN(C(C)(C)C)C(C)=O)C)C1 19288,c1(C(=O)NC2CC2CNC(C2OCCO2)=O)ccc(C2CC2)cc1F 19289,c1(CCC)cc(C(=O)N(CCC(=O)NC2CC(CC)C2)CC2CC2)no1 19290,N1(C(C(CC)F)=O)CCC(C)C(NC(c2ccn(C3CCC3)n2)=O)C1 19291,C1(NC(c2cc(C)c(C)o2)=O)CCC2CC1CN2c1nnc(C(N)=O)s1 19292,C1(O)(CNC(C(C)N(CC)CC)=O)CCCN(C(c2ncccc2N)=O)CC1 19293,C(=O)(C(F)C(F)(F)F)NC(c1c(CC)cccc1)CNC(=O)CC(=O)NC 19294,C(=O)(NNc1cc(F)c(F)c(F)c1)c1n(CCN)ncn1 19295,CC1CCN(C(=O)CC2(N(C(=O)C3=CCC(C)CC3)C)CC2)CC1(C)C 19296,C12(C(N3CC(CC)C3)=O)CC(C)(CN1C(=O)CC1NC(=O)NC1=O)C2 19297,N1(C(C2C(C(=O)NCC#C)C2)=O)CCN(C(=O)CC2CC3(CCC3)C2)CC1CF 19298,S(=O)(=O)(c1cccc(=NCC2(C3CCCO3)CCC2)[nH]1)NC(CC)CN(C)C 19299,CCC(CC)C(=O)N1CC(NC(C2(Cc3cccc(F)c3)CC2)=O)C(C)C1 19300,C(=O)(CCC(CC)CC)NC1C(CC)N(C(c2nnn(C)c2C)=O)CCC1 19301,C(=O)(C(C)C(C)(F)F)N(CC(C)O)CCNC(c1n[nH]c(C(C)C)c1Br)=O 19302,Cc1cc(C)c(C(=O)NCCOCCN(C(=O)C(C)C(C)(F)F)C)c(Cl)n1.C(C)(=O)OCC 19303,CN1CCN(C(=O)CCc2cccnc2)CC1C(=O)NC1(CO)CCOC1 19304,N1(C(C(C(C)C)n2ncc(N)n2)=O)CC2CCC1C(CNC(C1CSC1)=O)C2 19305,Cc1ccccc1C(=O)NCC(=O)N(C(C)C)C1CC1.C12CCCN1C2=O 19306,c1(C(=O)NCC2C3(CC(NC(C4(CC)CNC(=O)C4)=O)C3)C2)ncc2ccccn12 19307,Cc1noc(C2CC(N(C(=O)CCn3cccc3)C)C2)n1 19308,C1(CNC(c2cn(CC3CCCO3)nn2)=O)CCN(c2ncc(Cl)cn2)CC1 19309,CS(=O)(=O)CCC(=O)N1CCC(C2CCCN2C(c2ccoc2Cl)=O)CC1 19310,C1(NC(C(c2c(OC)cccc2)OC)=O)CN(C(C2(CF)COC2)=O)CCC1F 19311,C(=O)(C(C)CNC(=O)C(Cn1ccnn1)NC(=O)CCn1cncn1)NC 19312,C(=O)(C1=C(C)OCCS1)NC1CC2CN(C(c3nn(C(CC)C)c(C)c3)=O)C1C2 19313,C(=O)(C(F)CCC(C)C)NC12C(NC(C3N(C(CC)=O)CSC3)=O)CC(CC1)C2 19314,C12(C(=O)NC(CC)COCC3CC3)CC1CCN2C(=O)CC1CN(C)C1 19315,C1(C(=O)NCC2(NC(c3c(OC)scc3)=O)CC2)CCCC(C(N)=O)C1 19316,N1(C(C2(C)CC=CC2)=O)CC(NC(=O)CC2CCCN2C(C)C)CC(F)(F)C1 19317,C(=O)(C1=CC(O)C(NC(c2cccc(CC)n2)=O)C1)NCC 19318,CCCC(CCCNC(=O)C(C)Oc1cccc(C(C)=O)c1)NC(=O)C(C)(C)C 19319,CS(=O)c1cccc(C(N2CCN(C(=O)CCc3cnc[nH]3)C3CCC23)=O)c1 19320,C(CC(C)(C)C)(C(=O)NCCOCCCNC(=O)CCCN(C)C)OC 19321,c1(C(=O)NCC(C)CNC(=O)CCc2cncs2)ccc2c(n1)NCC2 19322,C1(C(=O)NCCc2cn[nH]c2)CCCN(C(c2ccc(C3COC3)cc2)=O)CC1 19323,c1(CC)ncc(S(=O)(=O)Nc2c(C)[nH]c(C(=O)CN(C)C)c2C)n1CCC#N 19324,c1(C(N(CCCNC(C(C2CCCC2)OCC)=O)C)=O)c(C)nn2ncccc12 19325,C1(NC(c2c(CCC)nns2)=O)CN(C(=O)C(C)S(N)(=O)=O)CC12CCC2 19326,N1(C(c2c(C)[nH]cc2)=O)CCC2(CC(NC(=O)C(=O)NC(C)C)CO2)C1 19327,C1(CNC(Cn2nnc(C)n2)=O)CCC2(CN(C(=O)C=Cc3ccnn3C)C2)O1 19328,c1(CC)nc(C)cc(=NC(=O)c2ccn3ncc(I)c3n2)[nH]1 19329,Cc1cc(C)c(CNC(C2CC(n3cc(-c4c[nH]nc4C4CC4)nn3)C2)=O)s1 19330,c1(C(=O)NCC2=CCN(C(C3CC34CCCC4)=O)CC2)ccc2nn[nH]c2c1 19331,C#CC(CNC(=O)C(C1CCOC1)NC(c1ccc(C2CC2)o1)=O)CC1CC1 19332,c1(OC)cccc(C)c1CNC(C1CC1C(=O)Nc1cc(OC)ccc1F)=O 19333,C#Cc1cn(C)nc1C(=O)N(C(C)CC(=O)N(CC(C)(C)O)C1CC1)C 19334,c1(C(=O)Nc2c(C)cc(NC(c3coc(C#N)c3)=O)cc2)ccc(F)c(Cl)c1F 19335,N1(C(Cc2nc(C)oc2)=O)CC2CC(NC(c3cc(C4CC4)no3)=O)CC2C1 19336,Cc1nc2ccc(C(=O)NCC3CCCC3NC(=O)CC3CC3(Cl)Cl)cc2n1C 19337,N1(C(c2cnc(CC)o2)=O)CCCC(CN(CC(C)C)C)C1.C1(C)C(=O)N1 19338,N1(C(CC(C)C(C)(C)C)=O)CCC2CCN(C(c3cc(C(F)F)cs3)=O)CC12 19339,C1(CCC(N2CCN(CC=C)CC2)=O)CC12CCN(c1ncc(Br)c(C)n1)CC2 19340,CC(C)(C)CC(O)CC(=O)NC1CCN(C(c2c(N)cccc2[N+](=O)[O-])=O)CC1 19341,C1(NC(=O)CCC2CC2(Cl)Cl)(CO)CCCN(C(C2CCCNS2(=O)=O)=O)C1 19342,C1(CC=C)(C(=O)NC2CC3C=CC2C3)CCCN1C(C1CSCC(=O)N1)=O 19343,N1(C(C2CC(CNC(=O)OC(C)(C)C)C2)=O)CC(O)CC1c1nc[nH]n1 19344,C1(NC(CC2ON=C(C)C2)=O)CCN(C(c2cnccn2)=O)CC1CO 19345,N(C(C)S(=O)(=O)c1ccccc1)c1c2cnn(C(C)C)c2ccc1.C(=O)O 19346,c1(OC)ccc(C)c(C(N2CC(NC(=O)C(C)CSC)C(C)(C)C2)=O)c1 19347,C1(NC(C(C)C2CC2)=O)CN(C(=O)CCc2cccc(Cl)c2)CCC12CCC2 19348,Cc1cc(N)cnc1-c1cn(CC2N(C(=O)Cc3[nH]cnc3C)CC2(C)C)nn1 19349,C(=O)(C1=NOC(C)C1C)N1CCC(NC(c2cc(C(C)C)on2)=O)(CO)C1 19350,Cc1cnc(C(N2CCC(NC(c3cc(F)c[nH]3)=O)C(CO)C2)=O)c(C)c1 19351,CC(CC(C)(C)C)C(=O)NCc1cc(C(=O)NCCCC2CC2C)n[nH]1 19352,CC1CCN(C(C2C=CCC2)=O)CC1CNC(c1cnccc1Cl)=O 19353,C(=O)(C(C)(C)C(C)C)N(CC(CNC(Cc1ncc(C)s1)=O)O)C 19354,C(CCCCCNC(C1CCCN1C)=O)NC(C=CCCC=C(C)C)=O 19355,C(=O)(CCCCC(=O)N1CCC(C)N(C(C2CCC(F)C2)=O)CC1)OC(C)(C)C 19356,CC1CC(=O)NC(C(=O)NCC2(CNC(c3nocc3C3CC3)=O)CC2)C1 19357,N1(C(C(C)NC=O)=O)CCC2CN(C(c3cnc(O)nc3O)=O)CCC12 19358,N1(C(C(C(C)C)OC)=O)CC(CNC(c2cccc3nn[nH]c23)=O)CC12CCC2 19359,C12(C(N3CCC(CNC(C(C(C)C)O)=O)C3)=O)CC3CC(CC1C3)C2 19360,c1(CSC)nc(C)ncc1Cl.C1C(=O)N(C(C)C)CCNC1=O 19361,N1(C(c2c(C)noc2N)=O)CCCC(NC(=O)CC(O)C2CCCC2)CC1 19362,C12(C(=O)NC3CCN(CC)C3=O)CC(CCO1)N(C(=O)Cc1cc(C)cs1)C2 19363,C(=O)(CC(=O)NC(C)CNC(=O)C(C)C1CC1)NCC 19364,N1(C(C(C)NC(c2ccco2)=O)=O)CC2CCCC(NC(=O)C(C)(C)F)C2C1 19365,CC(C)CC(C)CC(=O)NC1CCC(CN(C(=O)CC2=NNC(=O)C2)C)CC1 19366,CC1CCCC(CC(N2CCN(C(=O)C3=CCCSC3)CC2C2CC2)=O)C1C 19367,CC1CN(C(c2ncc[nH]c2=O)=O)CC(CCNC(c2cn(C)nn2)=O)O1 19368,C(=O)(CC(F)(F)C(F)F)NCC(C1CCCCC1)NC(C(C)NC(CC)=O)=O 19369,C12(C(N(CCCNC(C3CC3C(F)F)=O)CC)=O)CC3CC1C2C3O 19370,N1(C(c2nnc(C)o2)C)CCCC(C(C)NC(c2cn(C3COC3)nn2)=O)C1 19371,C(=O)(CCC(=O)NN(C)C)N1CC(C2CC2)(C(=O)NC(C2CCCC2)C#C)C1 19372,Cc1cc(NC(C2CC(O)CN2C(c2cnn(C)c2)=O)=O)cc([N+](=O)[O-])c1 19373,C1(CC(=O)NC(CNC(c2ccc(COC)[nH]2)=O)CO)(NC(C)=O)CCOCC1 19374,c1(C(N2CCCC(CNC(CSC(C)(C)C)=O)C2)=O)cccc2nonc12 19375,N1(Cc2cccc(CCC=C)c2)CCS(=O)(=O)CCC1c1ccccc1 19376,N1(C(C(C)(N(C(CCc2onc(C)n2)=O)C)C2CC2)=O)CC=C(CO)CC1 19377,C(=O)(C(CO)NC=O)OCC(=O)N(C(c1ccccc1)COC(=O)C(F)(F)F)C 19378,C1(CN(C(C2(CNC(c3cc(C)on3)=O)CC(=C)C2)=O)C)CCCCCC1 19379,c1(C(=O)NCC2CCCC(NC(C(C)c3cccs3)=O)C2)ccc2nccn2n1 19380,C=CCC(C(=O)NCC1CC2CCC(C1)N2C(=O)C=NOC)C(C)(C)C 19381,C12(C(N3C4CN(C(CC5(C)CCC5)=O)C(C4)C3)=O)CCCCN1CCC2 19382,C(C)(CNC(=O)C(c1ccc(-c2nnnn2C2CC2)cc1)=O)(C(C)C)NC(C)=O 19383,C#CCCC(O)C(=O)NCCCCNC(c1cccc(OC2CC2)c1)=O 19384,CC(C)(C(=O)NC(CNC(=O)C(C)(O)C1CCC1)CC(F)(F)F)C(F)(F)F 19385,CC1(C(=O)NCC2COCC2NC(C2(F)CCOC2)=O)CCC2(CC1)OCCO2 19386,N1(C(c2c(F)ccc(C)c2)=O)CCC2(CCCN2C(C2CSCCS2)=O)C1 19387,N1(C(CC2(C#N)CC2)=O)CCC2(CCCC2NC(C2C=CC=CC=C2)=O)CC1 19388,CC(C)C(CC(=O)NCCCc1ccsc1)NC(c1c[nH]nc1C(F)F)=O 19389,C(C(C)(C)C(=O)NC1C2CN(C(C3CCCN3C(C)=O)=O)CC12)NC(C)=O 19390,c1(-c2cn(C3C(NC(=O)COC(F)F)CCC3)nn2)cc(F)c(F)c(F)c1 19391,C(C(=O)NCc1ccoc1C(=O)NC(C(C)(C)O)C1CC1)(C(C)(C)C)OC 19392,CCCC(C)C(=O)NC(C)(CNC(=O)Cc1nccc(OCC)n1)C1CC1 19393,C12COCCN(C1)C2=O.C(=O)(CC(F)(F)F)NCc1c(C(=O)O)scc1 19394,N1(C(C(CC=C)NC(=O)OC(C)(C)C)C)CC(SC)CC1(C)C 19395,C(=O)(C(F)CC(C)(C)NC(=O)CC(C)(C)CC)N1CCCC(C=C)C1 19396,C1(N(CCC)C(c2[nH]cnc2C)=O)CCN(c2nnc(CCOC)o2)CC1 19397,c1(NC(C2C(NC(c3c(C)cccc3O)=O)CCCC2)=O)ncc(C#N)cc1I 19398,c1(C(N(CCN(C)C(c2c(F)ccc(F)c2O)=O)C)=O)c(F)ccc2nc[nH]c12 19399,C1(NCCCn2c(C)ncc2)CN(C(=O)CC2(c3ccccc3)CC2)CC12CC2 19400,c1(-c2nnc(CNS(CC(C3CC3)OC)(=O)=O)o2)cccc([N+](=O)[O-])c1 19401,C(CCCCC(=O)NCC1CC(C(=O)N(C)CC2COC(=O)N2)C1)=CC 19402,C1(C)(CNC(C(C2CCN(C(c3coc(C4CC4)n3)=O)C2)C)=O)CCCOC1 19403,Cc1cc(CC(N2CCC(F)C(NC(c3ccoc3Cl)=O)C2)=O)ccc1CO 19404,N1(C(c2c(C)ccs2)=O)CC2CCC(NC(c3ccc4n[nH]cc4c3)=O)(C2)C1 19405,C(=O)(CCCCCc1ccccc1)N1CCC(CN(CCCSC)C)C1 19406,CC(C(=O)NCc1cn(C2CN(C(c3ncccc3Cl)=O)C2)nn1)C(C)(F)F 19407,C1(N(CC(=O)NCC)C)CCN(C(C2(C3CCCO3)CCCC2)=O)C1 19408,C(=O)(C(C#N)C(C)(C)C)NC(c1cnn(C)c1)C(N1CC(C(C)C)NC(=O)C1)=O 19409,C1(CNC(C=CCCC)=O)CCN(C(=O)C(C)CSC)CC1C1CC1 19410,CN1CC2CCN(C(=O)C=CCN(C)C(C3CS(=O)C3)=O)CC2C1 19411,c1(CC(=O)NC2CC(C)N(C(c3ocnc3C3CC3)=O)C2)ccc2c(c1)CCC2 19412,C(=O)(CS(=O)C(F)(F)F)NCC1CCCCN(C(CN(C)CCO)=O)C1 19413,CCCCCC(C(=O)N(CC(CC)NC(=O)CC(F)(F)F)C)C(C)C 19414,N1(C(C2N(C(C)(C)C)CC2)=O)CCCC2CN(C(C3CC3F)=O)CC12 19415,N1(C(c2c(CC)cccc2)=O)CCCCC(NC(C2C(C(=O)OC)C2(C)C)=O)C1 19416,C=CCC(CC(F)F)C(=O)N1CCC(CNC(c2cccc3ncnn23)=O)C1 19417,C1(CNC(C2CC(C)OCC2)=O)COCCN(C(C2(CCN(C)C)CC2)=O)C1 19418,c1(CCNC(=O)NC(CC)CC2CCCO2)cccc(F)c1Br 19419,c1(OC)n[nH]c(C(=O)N(CC(C)(C)NC(=O)CC2CC(C(C)(C)C)C2)C)c1Cl 19420,CCC(C(=O)NCCCCCNC(=O)CCSc1ccccc1C)C(C)O 19421,CCC(CC(=O)N1CCC(F)CC1C(N1CCC(C)(CN(C)C)C1)=O)C(C)(C)C 19422,Cn1nc(C(N2CCCCC2CCC(=O)NCC(C)(F)C(C)(C)F)=O)ccc1=O 19423,c1(OCC)nccc(C(=O)NCCCN(C(=O)CS(=O)(=O)NC)CC2CC2)c1N 19424,C12(CNC(c3c(C(C)C)cccc3)=O)CCCC1CN(C(=O)C(C)N(C)C)C2 19425,c1(N(C)C)ncc(C(=O)NCC2CC(O)CN2C(c2ccc(O)cc2)=O)cc1Cl 19426,c1(NC(C(=O)N(C2CCC(c3ccc(F)cc3)C2)C2(C)COC2)=O)csc(C#N)c1 19427,N1(C(C(c2ccccc2)C)=O)CCN(C(=O)Cc2ccc(Br)cn2)C(CO)C1 19428,C(=O)(C1=COCCO1)NCC(C)(C1CCC1)NC(c1cc(CN(C)C)on1)=O 19429,C(=O)(C1CCCc2ccccc21)NC(C1CCCN1C(c1ccoc1)=O)C 19430,Cc1nc(C)n(O)c1C(=O)NC1CCCN(C(=O)C(C)(C)C(N)=O)C1 19431,N1(C(CC(C)n2ccnc2)=O)CCCC(CC(=O)NC2CCN(C3CC3)C2)C1 19432,C1(C(N2CCC(C(C)NC(=O)C(C)(C)F)CC2)=O)CC2(CCO1)CC2 19433,c1(OC)cc(C(=O)OC(C)C2CC2)cnc1-c1cnn(-c2ccc(C)cc2Cl)c1 19434,N1(C(C=CCN(C)C(c2ccc([N+](=O)[O-])o2)=O)=O)CCC2CCCCC2C1 19435,C1(NC(C2(OC)CCCC2)=O)CC(NC(C2(C#N)CC2)=O)CC1O 19436,Cc1ccc(C)c(NC(=O)CCC(C)NC(=O)CCc2nncn2C)c1 19437,Cc1cc(C(N)=O)cc(C(=O)NCCN(C(C2CCCCC2(C)C)=O)C2CC2)c1 19438,N1(C(CNC(C2CC=CC2)=O)=O)CCC2(CC1)CN(C(c1n[nH]cc1C1CC1)=O)C2 19439,C=CCC(C)(C)C(=O)NC1CCC1NC(c1cccc(C(C)=O)c1)=O 19440,O=S(=O)(c1ccc(N2CCC3(C2)CC(F)(F)C3)c(Br)c1)NCC1=CCCCC1 19441,C=CCC(C)(CC)C(=O)N1CCC(C)(CC(=O)NCCc2cc[nH]n2)C1 19442,N1(C(c2cocn2)=O)CCC(F)(C(=O)NCCN2CCCC2=O)C1 19443,CC(O)(CNC(=O)C(C1CCC1)NC(c1cc(O)ccc1F)=O)C(F)(F)F 19444,N1(C(=O)CC2OCCCO2)CCC2CCCN(C(=O)Cc3ccoc3)C2C1 19445,C1(C(N(CCOC)CCNC(C2CCCO2)=O)=O)CCC(O)C1 19446,c1(OCC)ncc(Cl)c(N2CCCC(NC(=O)C=CCN3CCCCC3)C2)n1 19447,N1(C(C(C)N(C)C(c2[nH]ccc2C2CC2)=O)=O)CC=CC(O)C1 19448,N1(C(c2c(C)nsc2)=O)CCC(C(C)NC(=O)CC2CCCO2)CC1 19449,Cn1nc(C(=O)NCC2CC3(C2)CC(F)(F)C3)c2c1CCCC2 19450,c1(C(N2CCC(OC)(CNC(=O)Cn3cccn3)C2)=O)c(F)ccc(F)c1Cl 19451,C1(C(=O)NCCc2c(C(=O)NCCC(=O)NC)c[nH]n2)OCCOC1C 19452,O=C(CC1CCN(C(=O)COCCOC2CC2)C1)NOCCNC=O 19453,C(C(C)(C)C(=O)NCC1CCCN1CC)NC(C=C(CCC)C)=O 19454,O=S(=O)(c1cnc(N2CCCC(F)C2)c(Cl)c1)NC1CCC1n1cccn1 19455,C1(CC=C)(NC(=O)CC(C)F)CCCN(C(c2cc(C(F)F)ccc2Cl)=O)C1 19456,CC(C(=O)NCC1(O)CCCN(C(c2ccn3c2CSCC3)=O)C1)C1=CCCC1 19457,CC(C(=O)N(CCC(N1CCC(C)(F)CC1)=O)CCO)S(N)(=O)=O 19458,CC(=O)CC(C)(C)C(=O)NCC1(CNC(c2c[nH]cc2C2CC2)=O)CC1(F)F 19459,N1(C(CSCC#C)=O)CCC(NC(=O)C(C(C)C)n2cnnn2)C1C1CC1 19460,C(=O)(CC(C)CNC(C1CCNC(=O)C1)=O)NCC(COC)OC 19461,c1(C(N(CC(C)NC(C2(C)CC2C(F)(F)F)=O)CC)=O)ccc(C)cc1C 19462,c1(CNC(c2cn(C)cc2C(F)(F)F)C)nc2c(s1)CCC(C)C2 19463,N1(C(C(C)S(C)(=O)=O)=O)CC(N=[N+]=[N-])CC1C(=O)NCc1ncc(CO)[nH]1 19464,N1(C(=O)CCc2cccs2)CCCN(C(C2CC3CC2CC3O)=O)CC1 19465,N1(C(C2(F)CCC(C)CC2)=O)CCOC2(C1)CN(C(=O)CCC1CC1(C)C)C2 19466,c1(C(=O)NC(CCOC)C(=O)N2CC=CC2)ccc2c(c1)CCC2 19467,C1(N(C(c2n(CC)ncn2)=O)C)CCCCN(C(=O)C=Cc2ccc(C)cn2)C1 19468,N1(C(C(c2cn(C)nn2)NC(c2c(OC)ccnc2)=O)=O)CCNC(=O)C1C 19469,N1(C(CC=CC=C)=O)CCC(CNC(=O)CC(C(F)(F)F)OC)C(F)(F)C1 19470,CC1(NC(=O)CNC(N)=O)CCN(C(C2CCCC(F)(F)C2)=O)CC1 19471,C1(C(=O)NC(C(=O)NCCC(=O)NCC)Cc2cn[nH]c2)CCCCCCC1 19472,n1(CC(=O)NCCC(CC)=O)ccc2ccc(F)cc12 19473,N1(C(CC2CCC(NC(CN=[N+]=[N-])=O)C2)=O)CC=CC(O)C1 19474,c1(COC)onc(OC)c1C.C12CN(CC1C)C2.c1(NC)ccc(-c2ccco2)cc1 19475,C(C(O)C(=O)N(CC(C)N(C(=O)C(CN(C)C)N(C)C)C)C)=CCCC 19476,c1(NC(C2CCC(NC(=O)CSCC3CCCO3)CC2)=O)nnc(O)cc1O 19477,c1(C(C)OC)nc(C)c(C(=O)N(C)CCNC(=O)C(=Cc2cccs2)C)s1 19478,CCC(CC)(C(N)=O)NC(=O)C(C)=CCNC(C1CC(=O)CC(=O)C1)=O 19479,C(C)(CC(C)CC(C)C)(c1n(CC=C)nnn1)NCc1ccc(COC)o1 19480,c1(OC)cc(C(=O)NCCC2CCN(C(c3ccc(Cl)cn3)=O)CC2)nc(C)c1 19481,C1(N(C(Cc2nc(C)sc2)=O)CCO)CCN(C(=O)CC2(O)CCOC2)CC1 19482,Cc1nc(N2CCSCC2CCNC(C23CCCC(CO2)C3)=O)c(Cl)cc1C#N 19483,C1(CN(CC)CC)CC2(CCN(C(c3cc(SCC(=O)OC)n(C)n3)=O)CC2)C1 19484,N1(c2ncc(OCC)cn2)CC2CCC(C1)N(C(c1nc(C3CC3)cs1)=O)C2 19485,c1(CC)nc(C(=O)NC2CN(C(c3cc(OC)no3)=O)C(C)C2)c(N)s1 19486,c1(C(=O)NC2CCC(N(C(COc3cn(C)nc3)=O)C)C2)csc(S(N)(=O)=O)c1 19487,c1(C)ncc(CNC(C2(C(=O)O)CC2C(F)(F)F)=O)s1.C(F)(F)F 19488,C1(C(=O)NC(C)CNC(=O)CC2COC(=O)N2)CCC12CCC2 19489,N1(C(C(C)C2CCCO2)=O)CCC2CCN(C(c3ccc(O)nn3)=O)CC2C1 19490,c1(CC)nnc(C=CC(=O)NC2CCCCC2NC(=O)CC(C)n2cccn2)o1 19491,Cc1cccc(C)c1NC(=O)C(N1CCOC2CC12)c1ccc(C(N)=O)s1 19492,C(c1cc(Cl)ccc1Cl)=CC(N1CC(CNC(C2(COC)CCC2)=O)C2C1C2)=O 19493,c1(OC)ccc(C(N2CC(NC(=O)CC(C)OC)C(F)C2)=O)c(F)c1 19494,C(C)(CC(=O)N1C2CCC1CC(NC(C1(CF)CC1)=O)C2)(C(F)(F)F)N(C)C 19495,C(=O)(C(F)C(C)CC(C)(C)C)NC(C1CCN(C(c2n(CC)ncc2C)=O)C1)C 19496,C(C(C(=O)NCC(CC)NC(=O)C(c1cncn1C)O)c1ccccc1)OCC 19497,S(=O)(=O)(c1cnn(C)c1)N1C2C(C(N3CCC(NS(C)(=O)=O)CC3)=O)C(C2)C1 19498,S(=O)(=O)(CCC(=O)N1CCC(C)C(NC(c2cc(C3(C)CC3)on2)=O)C1)NC 19499,c1(OC)ncc(C)cc1C(=O)NC1CC(CNC(C2CCC(C)S2)=O)C1 19500,N1(C(CCC#CC)=O)CCc2nc(CNC(c3cc4c(s3)COCC4)=O)sc2C1 19501,C1(n2cc(CCC(=O)Nc3c(CC)con3)nn2)CCCN(C(=O)CC(C)F)C1 19502,C1(C(C)OC(=O)CC(c2cccnc2)NC(=O)OC(C)(C)C)CC2(C1)CC(O)C2 19503,c1(SC)ccnc(C(=O)NCCCCC2CCCN(C(=O)Cc3cncs3)C2)n1 19504,N1(C(Cc2n(C)cnc2)=O)CCN(CC(=O)NC(CC2CC2)C2CC2)CC1 19505,c1(C(=O)NC(c2ccccc2)C(C)NC(C=CSC)=O)cccc2c1OCCN2 19506,C1(C2CCCN(C(=O)C3=CCCC3)C2)(NC(c2cc3cnccc3o2)=O)CC1 19507,c1(CC)nn(C)c(Cl)c1C(N1CCC(O)(CN(C)C(C2CC23CCC3)=O)CC1)=O 19508,c1(OC)ccn2ncc(NC(=O)NCCOCC(F)(F)C(F)F)c2c1 19509,C(C(=O)N(C)CC1(O)CN(C(c2ccnc(O)c2)=O)C1)(C(C)C)NC(C)=O 19510,C12(NC(COC(C)C)=O)CCC(NC(c3cc(Cl)ncn3)=O)(CC1)C2 19511,CCC(CC(=O)N1CCC(c2n[nH]cc2CNC(c2ncc[nH]c2=O)=O)C1)C1CC1 19512,c1(C(=O)NCC2CCCCN(C(C(C=C)O)=O)CC2)c(C)nn2c(C)cccc12 19513,N1(CC(=O)Nc2c(C#C)nccn2)Cc2ccccc2C1C(=O)NC 19514,C(C)(C)(CCCC(=O)N1C2CCCC1COC2)NC(C(CC)COC)=O 19515,S(=O)(=O)(c1ccc2ccccc2c1)NC(CC(N1C2COCC1CC(F)C2)=O)=O 19516,N1(CCC=C)CCCCC1CNC(C1CC(=O)N(C2CCOCC2)C1)=O 19517,C12(CC(=O)NCCCCCN(C(C3CC(SC)C3)=O)C)COCC(C1)C2 19518,C1(CNC(CC(CNC(=O)C(N2CCOC2=O)C)OC)=O)CCCCC1(C)C 19519,c1(C(N(C(CNC(C2(C)C(C(=O)OC)C2)=O)C)C)=O)cc(-c2ccncc2)on1 19520,C(=O)(C(C)CC(C)(F)F)NCC1(C(C)(C)O)CN(C(C=CSC)=O)C1 19521,C1(C(=O)NCCC(N)=O)C=CCN1C(=O)CC1COC(=O)C1 19522,Cc1cc(C(=O)NC2CCC2NC(=O)C=CBr)cc(Cl)c1Br 19523,c12ccc(C)c(c1)C(=O)N2.C1(CC(=O)NC2CC(NC(COC)=O)C2)COCC1O 19524,C12(C(=O)NCC3(NC(C4C(C)CC4C)=O)CC3)CC3CC1C2C3 19525,C1(C(=O)Nc2n[nH]c(-c3ccc(Cl)c(Cl)c3)n2)CCn2c(O)nnc2C1 19526,C1(C(=O)NCC2(F)CN(C(C(CSC)OC)=O)C2)CCCCN(C)C1=O 19527,C(=O)(C(CC(C)C)C(N)=O)N1CCCC(O)(c2cn(Cc3c(C)sc(Br)n3)nn2)C1 19528,C(=O)(C(F)(F)CO)N1CC(F)(N)C1.c1(CCC(=O)C(=O)CO)cnccn1 19529,N1(C(C2CN(C(C3SCCS3)=O)CC2(F)F)=O)CCOC2C(O)CC12 19530,N1(C(c2cc(CC)ncc2)=O)CC(C)(C)CC1CNC(C1CCCSC1)=O 19531,c1(CN(C(CNC(c2ccc(C)o2)CC)=O)C)ccc(S(N)(=O)=O)cc1 19532,N1(C(CS(=O)(=O)NCC)=O)CC2CC1CCC2NC(=O)COCC1CCC1 19533,C1(C(C(=O)NC)N(C2CC(n3cncn3)C2)C)CC2CCC1C2 19534,C(=O)(C1SCCc2ccccc21)N1CC(CNC(C(=O)NCC)=O)C(C)C1 19535,c1(C(N2CCC(O)(C(N3CCN(S(C)(=O)=O)CC3)=O)C2)=O)cccc(F)c1Br 19536,Cc1ccoc1C(=O)Nc1cnn(C2CCOCC2)c1 19537,C1(C)(CNC(C=C(C)C(C)(C)C)=O)CCN(C(C2(C#N)CC(=O)C2)=O)CC1 19538,N1(C(CC(CC)C)=O)CCCCC2(CCN(C(C3CCC3)=O)C2)C1 19539,c1(C(=O)NCC2CN(C(c3c(C)ncnc3)=O)C(C)(C)C2)cc(Cl)cc(Cl)c1O 19540,Cc1ccc(C(=O)NCC(=O)NCC2CN(C(C3CC3F)=O)CC2O)cc1C 19541,C1(NC(C2=NNC(=O)C2)=O)CCCC2CN(C(C3C=CC=CC=C3)=O)CC12 19542,CC(C)CC(O)C(=O)NC(Cc1ccco1)C(=O)N(C)CC1(O)CCC1 19543,O=C(C1=CCCOC1)NC12CC(NC(c3cnn4c3SCC4)=O)(C1)C2 19544,C12(C(=O)NCCCCC)CCCC1CCN2C(c1ccc(CC)cn1)=O 19545,c1(C(N2CCC(NC(c3c(CC)nn(C)c3)=O)C2C)=O)ccc(C(C)C)nc1C 19546,C(=O)(CCC(CC)OC)NC1CCN(C(C(CC)c2ccccc2)=O)C1C(C)C 19547,CCC(CC(F)F)C(=O)N1CCCC1CNC(c1c(F)ccc(C)c1N)=O 19548,C1(CC)CN(c2ncc(C3CC3)cn2)CCN1C(c1ccccc1CO)=O 19549,Cc1cc(C(=O)N(CCNC(C2(OC(C)C)CCC2)=O)C2CC2)c2ncccc2c1 19550,C(CC(C(C)(C)C)NC(=O)C(O)c1ccsc1)N(C)C(c1cc2n(n1)CCO2)=O 19551,C1(CCCN(C(=O)CCC)CC)CCN(C(=O)C(O)c2ccsc2)CC1 19552,C(=O)(C(F)(F)C(O)C(C)C)N1CCCCC(NC2CN(C(CS(=O)(=O)NC)=O)C2)C1 19553,C1(C(=O)NC2(C(=O)OC)CC2)CCOC1CNC(=O)Cc1ccco1 19554,N1(C(=O)NC(c2nc(=O)[nH][nH]2)C)CCCC2(C=CCO2)CC1 19555,N1(C(=O)C(c2ccc(Cl)cc2)O)CCN(C(C2CC2(F)F)=O)CC(O)C1 19556,c1(C(=O)OC)ccc(F)c(C(=O)NCC2CC(NC(=O)C(F)(F)C(C)O)C2)c1C 19557,C1(C(=O)NCC(C)(C)C(=O)N2CCCC(CCO)C2)CCCC(C#N)C1 19558,C1(CC(=O)OC)CCC2CN(C(=O)NC3CC(c4ccncc4)C3)CC12 19559,CC(C)C(Cc1ccccc1)C(=O)NCCC(C)N(C)C(c1cc(C#N)c[nH]1)=O 19560,c1(N2CCN(C(N(C3CC3c3ccncc3)C)=O)CC2)cc(C#N)ccc1F 19561,C1(N(C)C(c2cnn(C(F)F)c2)=O)CN(C(=O)CC2C(C)(C)C2(C)C)CCC1O 19562,CC1(CNC(=O)NC2CCN(C(=O)OC(C)(C)C)CC2)OCCc2sccc21 19563,N1(CC)CC(C(N2CC3CC2C3NC(c2nccnc2N)=O)=O)CCC1=O 19564,C1(C(=O)NCCC2(O)CN(C(C(C(CC)O)(C)C)=O)C2)CCOC2(CCCC2)C1 19565,c1(C(=O)OCC)ccc(N(C2CCCN(C(c3cc(C(F)F)[nH]n3)=O)C2)C)nc1 19566,C1(C(=O)NC(C)CC(=O)O)CCCCC1C(N)=O 19567,C(=O)(CN1C(=O)CSc2ccccc21)N1CC(C)(NC(C2C(C)CCC2)=O)C1 19568,c1(SCCCNC(C2CC(NCC)C2)=O)cccc(OC(C)C)c1 19569,N1(C(C2(CC)CCC2)=O)CCC(C(F)C(=O)NCC2(C)CC2)C1 19570,O=C1CCC(C(N2CCN(C(c3cn(C4CCC4)nn3)=O)C(CF)C2)=O)CCO1 19571,c1(C(C)C)cc(C#N)nc(N2CC(NC(c3cnccc3Br)=O)C2)n1 19572,C1(C(=O)OC(c2ccc(C(F)(F)F)cc2)CC)(COC)CCOCC1 19573,c1(C(=O)NCCCN(C(C2CCCNC2=O)=O)CC)ccc(-n2ccnc2)nn1 19574,C#CC12CCC(C(N3CCC4(CC3)CC4CNC(=O)C=CBr)=O)(CC1)CC2 19575,C1(CCC(=O)OCC)CCCN(C(=O)NCc2cc(C)[nH]c2C)C1 19576,c1(NC(C(C)NC(C(C)OC)=O)=O)cnc(F)nc1 19577,C1(CNC(CC(C)C)=O)C(O)C(O)CN1C(=O)CCC#N 19578,C1(N(C)C(c2cc(-c3cccnc3)no2)=O)CCC(NC(C2CC2F)=O)CC1 19579,N#Cc1ccc(C=CC(=O)NC2CC2CNC(=O)Cc2cn3ccsc3n2)cc1 19580,c1(C(N2CC(c3cn(C4C(C)(O)CCC4)nn3)(O)C2)=O)ccc(C2CC2)c(F)c1 19581,CC1(F)CCN(C(=O)C(CCC2CC2)NC(C2CCS(=O)CC2)=O)CC1 19582,c1(C(=O)NC(CC=C)CNC(=O)C=C(CCC)CCC)cc2ccc(O)nc2s1 19583,N1(C(c2cc(C)sc2)=O)CCC(CNC(=O)CCOCC(C)C)CC1C 19584,N1(C(c2scc(C)c2C)=O)CCC2(CC2NC(C2CC(C(C)C)=NO2)=O)C1 19585,C1(NC(CCCCCSC)=O)CCN(C(=O)CC2C=CS(=O)(=O)C2)CCC1(F)F 19586,C1(CCNC(C23CC(C)(C2)C3)=O)CCCCN1C(=O)C(C1(O)CCCC1)F 19587,CN1C(=O)CC(C(=O)Sc2ccccc2)C1SCCF 19588,Cc1c(Br)cc(C(N2CC3CC3(CNC(C3CC3C)=O)C2)=O)cc1Br 19589,C(=O)(C(O)CC(N)=O)N1CC(NC(c2ccc(CNC(C)=O)s2)=O)C(O)C1 19590,c1(N2CC(NC(c3c(Cl)nc(OC)s3)=O)C(F)CC2)ncnc2c(Br)cccc12 19591,N1(CC(N2CC(CC(=O)OC)OC(C)C2)=O)C(=O)C(=O)N(C)C1=O 19592,C1(NC(C2C(CCC)CCC2)=O)CC12CCC(NC(c1ccc(Cl)cn1)=O)CC2 19593,N#Cc1ccccc1-n1ccc(C(N2CCC(NC(=O)C=C(Cl)Cl)C2)=O)n1 19594,N1(C(c2cnc(CC(C)C)s2)=O)CCN(C)C(CNC(=O)C(C)CN(C)C)C1 19595,CC1CN(C(C2(C)CCCN2C)=O)CCC1C(N1CCCC(C(N)=O)C1)=O 19596,CCCCC(O)CC(=O)N1CC(CO)(NC(=O)CSC2CCS(=O)(=O)C2)C1 19597,C1(C(N2C(C)CCC2)=O)CCCCCCN1C(=O)C=CC1CCCC1 19598,c1(NC(C2CCC(NCc3c(F)ccc(C(N)=O)c3)CO2)=O)cccc(F)c1O 19599,C1(c2cn(C(C)NC(C3CC(F)CN3)=O)nn2)COCCN1Cc1ccccc1 19600,C(=O)(C(CC(N)=O)OC(=O)NC(C(C(=O)OC(C)(C)C)C)C)OC 19601,c1(C(N(C2CCN(C(=O)C=Cc3cccs3)C2)C)=O)cc(C(F)(F)F)ccn1 19602,N1(C(CC(=O)NCC2CC2)=O)CC2CCC1CN2C(=O)Cc1cc[nH]n1 19603,C1(C)(CNC(c2n(C)ncc2)=O)CCCN1C(=O)CCc1ccc(CO)cc1 19604,Cc1ccnc(SCC(=O)NC2(C)CCN(c3nnnn3C)C2)n1 19605,c1(OC)sc(C(=O)NCC2(F)CN(C(=O)C(C)(Cl)Cl)C2)cc1Br 19606,C1(C(N(CC(CNC(C(C)=C(CC)C)=O)(C)C)C)=O)CCCCC(F)(F)C1 19607,CC1C(NC(c2ccc(F)c(F)c2)=O)CCCN1C(c1coc(C(F)F)c1)=O 19608,c1(OC)cccc(F)c1C(=O)N(C1CCN(C(C2CCC(F)CC2)=O)C1)C 19609,N1(C(C(c2cn(C)nc2)=O)=O)CCCC2(NC(=O)COC3CCCC3)CCCC12 19610,Cc1c(C(=O)NC23CC(NCc4cc(O)ccc4F)(C2)C3)cncc1Br 19611,C(CC(c1nnnn1CCSC)C1CCCC1)(C(C)C)(c1cc(C)no1)NC(N)=O 19612,c1(N2C3CC(CNC(C4(C(=O)NC)CCC4)=O)C2CC3)ncc2scc(Br)c2n1 19613,CC1CC(C(N2CCCC(CF)C2)=O)CCN1C(=O)CCc1cnccn1 19614,c1(CCC)ncc(C(=O)NCC2CCN(C(=O)C(C)c3ccsc3)C2)s1 19615,N1(c2nnc(C)c(C)n2)CC(C)(C)CCC1CNC(=O)C(C)C(C)C 19616,C1(C(N(CCOC)CCF)=O)CC(O)CCN1C(c1ccns1)=O 19617,C#CCC(CC(=O)N1CCC=CC1COC)NC(C1CC(F)(F)C1(C)C)=O 19618,C1(C(C(=O)NCCOCCNC(C2(COC)CCC2)=O)C)CCCCC1 19619,c1(C(=O)NC2C3(CC(NC(C(CC=C)(F)F)=O)C3)C2)ccc2cnc(C)n2c1 19620,N1(C(C2CC(C(F)(F)F)(OC)C2)=O)CCOC(CNC(C2CCO2)=O)C1 19621,c1(C(CC)C)nc(C)cc(=NCC2(O)CN(C(=O)C(C(C)C)SC)C2)[nH]1 19622,c1(C(N2CCC(OCc3ccccn3)CC2)=O)cnccc1Cl 19623,c1(C(N2CC=C(COC)CC2)=O)ccc2[nH]ccc2c1.C1(OC)CC2CC1NC2=O 19624,CC(C)(C)C(O)C(=O)Nc1ccoc1CC(=O)NC(=O)COc1cnc(Cl)cn1 19625,C1CC(C(=O)O)Sc2cn1nn2.n1(C(C(=O)N(CC=C)CCC)C)ccc(C)n1 19626,c1(OCCCC(=O)NC(C2CCN(C(C(CC)=CC)=O)C2)C)ccccc1F 19627,C1(NC(c2c(C)c[nH]n2)=O)CC2C1CCN2C(=O)C=C1CCCCC1(C)C 19628,N1(C(CC(C)F)=O)CCSCC1C(=O)NC(c1cscn1)CO 19629,c1(C2(C(=O)NC(C3(O)CN(C(=O)COc4ccon4)C3)C)CC2)ncccc1F 19630,C1(COCC)(COC(c2ccc(N3CCCC3)nc2)=O)CC2(CC(O)C(O)CO2)C1 19631,Cc1cc(C(N2CC(O)(CNC(=O)CC3(O)CCCN(C)C3)C2)=O)cc(C)c1F 19632,c1(-c2c(CC(=O)N(CC=C)Cc3ccccc3)scc2)ccc(C)c(C)c1F 19633,CCC(CCCC(=O)NCC(O)CC(C)C)NC(=O)C(=O)C(C)C 19634,c1(OC)ccc2cc1CNCCSCCC2.C(C)(COC)N(C)C(C)C 19635,C1(CC)CCC(C(=O)N(CC(O)CN(C)C(c2csc(C(C)(C)OC)n2)=O)C)O1 19636,C1(C(=O)NCC(C)(C)F)C2CC(O)C(C2)N1C(c1cccc2[nH]ncc12)=O 19637,C1(C)(NC(C(C)OCC(C)C)=O)CCCCC1C(=O)N(C)CC1CCN(C)CC1 19638,CC1(CCNC(C2(C)C=CCC2)=O)CCN(C(c2csc(Br)n2)=O)C1 19639,C(=O)(C1=CCOCC1)NC1CCC(NC(C2C(C#C)C2(C)C)=O)CC1 19640,CN1CC(C(=O)NCC2(NC(C3CC3c3cccs3)=O)CC2)NC1=O 19641,N1(C(c2c(CCC)nco2)=O)CCN(C(=O)Cc2cnns2)C(CC(C)(C)C)C1 19642,C=CC(C)(C)CC(=O)NCC1(C)CCCN1C(=O)C=Cc1scnc1C 19643,CN(CCCC(=O)N1CCN(C)CC1CNC(=O)CC1CC(O)C1(C)C)N=O 19644,c1(C(=O)NC2(C)CCN(C(C3(CCF)CC3)=O)C2)ccc(Br)cc1[N+](=O)[O-] 19645,c1(CC(=O)NCC(CO)NC(C(C)OCCOC)=O)cc(Cl)c2c(c1)OCO2 19646,c1(C(=O)NCCCCCN(C(CNC(CC)=O)=O)C)ccc(N(C)C)cn1 19647,N1(C(CCCC#CC)=O)CC(CNC(=O)C(O)CC(C)C)CC(C)(C)C1 19648,N1(C(C2C(=O)OCC2)=O)CCC2(C1)CN(C(c1c(Cl)nsc1Cl)=O)C2 19649,N1(C(CC2C(C(=O)OC)C2(C)C)=O)CCC(NC(c2nn(C)cc2C)=O)C(C)C1 19650,c1(C(=O)NC2(CNC(C3C(OCC)CC3)=O)CCC2)csc2nccn12 19651,c1(C(=O)NCC(C)NC(c2n(CC)nc(C)c2)=O)ccc(F)c(C)c1C#N 19652,N1(C(c2occ(C)c2)=O)CC(C)(C)CC1C(=O)NCc1ccc(Cl)o1 19653,CC1=NOC(C)(C(=O)NCC(CO)NC(=O)CC2CCN(C)C2=O)C1 19654,c1(C(N2CC(CC(C)NC(C3(C#C)CC3)=O)C2)=O)noc2c1CCCCC2 19655,C=CCC(C(=O)N(CC(C)O)CCNC(C12CCC(OC)(CC1)C2)=O)C(C)(C)C 19656,CCC(CC(=O)NCC1(CNC(c2cc(Cl)nn2C)=O)CCC1)C(C)C 19657,N1(C(C(C(C)C)OC)=O)CC2C(NC(=O)CC(C)(C)C(C)(F)F)CS(=O)(=O)C2C1 19658,C1(NC(c2ccc(CNC(C(COC)COC)=O)cn2)=O)CN2CCC1(F)CC2 19659,Cn1nc(C(N2CCC(N(CCO)C(C3CCNC3=O)=O)C2)=O)cc1F 19660,C(=O)(C(F)C1=CCCCC1)NC1(CCOC)CCN(C(=O)COC(C)=O)CC1 19661,C(=O)(CCC(F)(F)F)N1CCCC(C(=O)Nc2c(CC)nn(C)c2)C1 19662,c1(C(N2CCCC2CC)C(=O)NCC=C)ccc(SC2CCC2)o1.C(C)(=O)OCC 19663,c1(C(=O)NC(C)(CNC(C2COCOC2)=O)C2CC2)c[nH]c2nccc-2c1 19664,N1(C(CC(C)(C)C)=O)CC2(CCCN(C(c3cccc4nscc34)=O)C2)C1 19665,C(=O)(C1=CNC2=NCCCN12)N1C(CCNC(CCC2C(C)(C)C2)=O)COCC1 19666,c1(C(=O)NCC(CNC(c2cn(C(C)(C)C)nc2)=O)CO)cc2ccccn2n1 19667,c1(C(N2CC(C(C)NC(=O)C(C)C(F)F)C2)=O)ccc(N)c(F)c1F 19668,c1(C(N(C2CCCCN(C(C=CC(=O)N(C)C)=O)C2)C)=O)ccnc2c1CCC2 19669,c1(C(=O)NCCCCC(=O)N(C2C(C)CN(C)CC2)C)nccc2[nH]ccc12 19670,C1(NC(CC(=O)OCC)=O)CN(C(c2ccnn2CC)=O)CC12CCC2 19671,N1(C(C(c2cccnc2)OC)=O)CCCC(C2CCCN(C(=O)CSC)C2)C1 19672,n1(CC)ccc(C(=O)N(CC(C)(C)NC(c2cc(C)c(Cl)s2)=O)C)cc1=O 19673,N1(C(c2scc(C)c2C)=O)CCN(C(C2CC(OC(F)(F)F)C2)=O)C(CCO)C1 19674,N1(C(C(C)NC(N)=O)=O)Cc2nccnc2CC1C(=O)NCCC1CCOCC1 19675,C1(NC(COC(c2cn(CCC)nc2)=O)=O)CN(C(=O)NC(C)(C)C)CC1C 19676,CC(N=c1ccc(C#N)n[nH]1)C1CCN(C(C2CCc3nn[nH]c3C2)=O)C1 19677,c1(C(N(C)Cc2cnc(CC)s2)=O)ccc(=N)[nH]c1 19678,Cc1cccc(CC(=O)N(C2CCCN(C(=O)CC(C)O)C2)CC2CC2)c1 19679,c1(C(=O)NC2C(NC(C(C(C)C)OCC)=O)CCC2)nc(C)c(C)nc1C 19680,CCC(CC(C)C)C(=O)NCC(C)C(=O)N1CC(OC(F)F)C1 19681,c1(C(=O)NCCCCNC(C2CC3CCC2C3)CC)cc2ccccc2o1 19682,N1(C(c2ccc(C)nc2C)=O)CC(C(N2C(CO)CC2C)=O)C(C2CC2)C1 19683,C1(C)(C(=O)NCC(CNC(c2occ3c2CCC3)=O)OC)CCCNC1=O 19684,N1(C(=O)Cn2cc(C(F)(F)F)cn2)CC(C(=O)Nc2ncc(F)s2)CC(F)(F)C1 19685,C(CCCCC(=O)NC(C)CCN(C(=O)Cc1cc(C2CC2)no1)C)OCC 19686,N1(C(C2C(OCC)C2)=O)CCC(NC(=O)C(N2CCCCCC2)(C)C)C(C)C1 19687,C#Cc1cc(OCC(N2CCC2CC(=O)NC2(C)CC2(C)C)=O)cc(F)c1 19688,c1(CNC(=O)NC2CCCC2Cc2ccccn2)ccncc1F 19689,N1(C(C(C)N(C(CSC(C)C)=O)C)=O)CCCC(C)(O)C1 19690,C12(CNC(C3C(=O)NCC3)=O)CN(C(C3CCS(=O)CC3)=O)CC1CCO2 19691,c1(C(=O)NC(CCNC(c2nc(C)nn2C)=O)(C)C)nccc(N)c1Cl 19692,CC1CC(CNC(=O)C(=O)NCCOCc2cccs2)CC(C)C1 19693,c1(OC)cc(Br)c(C(=O)NCCN(C)C(c2nccc(C)c2F)=O)cc1OC 19694,N1(c2nnc(C)o2)CCC(C(F)(F)F)C(NC(c2nccc(C(F)(F)F)n2)=O)C1 19695,c1(C(=O)NCC(CN(C(c2nc(C(C)=O)sc2)=O)C)C)nnc(C)cc1O 19696,Cc1noc(C)c1S(=O)(=O)N1CC2CN(Cc3cc(Cl)cnc3Br)C2C1 19697,c1(OC)cc(C(=O)NC(C2CN(C(C3(OC)CC3)=O)C2)C)cc2cn(C)nc12 19698,c1(-c2snc(OC)c2N)c(C)ccc(F)c1OC 19699,C(=O)(N=c1ccn(C2CC2)[nH]1)C1(C(C)NC(C2C(COC)N(C)CC2)=O)CC1 19700,c1(C(=O)NCCC2(O)CCCN(C(C3(N=[N+]=[N-])CC3)=O)C2)cccn2nccc12 19701,N1(CC(COCC(C)C)O)CCS(=O)(=O)C(CCNC(C2NC(=O)NC2=O)=O)C1 19702,CCS(=O)(=O)CCCNC(N1CC(C(=O)OC)OCC1C)=O 19703,N1(C(C2C(CC)C2)=O)CC(C)CN(C(c2cccc(N)c2N)=O)C(C)C1 19704,N1(C(C(C=C)C)=O)CC(O)(C2(CNC(=O)COCc3cccc(C)c3)CC2)C1 19705,c1(C(=O)OCC)nc(=NC(C)CSCc2cccs2)c2sccc2[nH]1 19706,N1(C(c2c(CC)cno2)=O)CCC2C(C(=O)NCCCCC3CC3)C2C1 19707,c1(C(=O)NCC2CCN(C(C3ON=C(C)C3)=O)C23CC3)coc2ccc(C)cc12 19708,C1(N(C)C)CN(C(=O)C(O)C2CC2)CC1CNC(c1csc(C#N)c1)=O 19709,c1(C(=O)NC2CCN(C(=O)CC3CCOC3)C2)cnnc2ccccc12 19710,c1(NC(C)=O)ccccc1SCC(N1CC(C)(NC(=O)CC2CCC(O)C2)C1)=O 19711,N=c1[nH]c(=NCC2CC23CCOCC3)[nH]c(=NCCCCCC(=O)NC2CC2)[nH]1 19712,c1(C(N2C(C(=O)OC)(COC)CCC2)=O)ncn2c1CCNCC2 19713,CCC(CN(C)C)CC(=O)NCC1(O)CN(C(=O)CCC(C)N(C)C)C1 19714,c12ccc(c([N+](=O)[O-])c1)CN2C.C1(C(C)=O)CC(C(F)(F)F)CCN1C 19715,N1(C(C(CC)(C)OC)=O)CCN(C)C(CNC(C2CN3CCC2CC3)=O)C1 19716,C12(C(N3C(CN(C(CCCC(C)C)=O)C)CCC3)=O)CC=CCN1CCC2 19717,C1(NC(c2c(C)csc2)=O)COCCN(C(c2cn(C(C)C)cc2C)=O)C1 19718,Cc1cc(CO)oc1C(=O)NCC1(F)CC(CNC(=O)CC2CC3CC3C2)C1 19719,C(C1CN(C(=O)COCC2CC2)CC1C(N1CCOCCC1C)=O)=CC 19720,C1(NC(C2CCN(C)C2=O)=O)CC2(C1)CC(NC(=O)C(c1cccn1C)=O)C2 19721,C1(C(N2CCN(C(c3c(CC)ncs3)=O)CC2COC)=O)CCc2nn[nH]c2C1 19722,C(C)(C(=O)N=c1cc(CC)n(C)[nH]1)(N(C)C(n1ncc2ccccc12)=O)C1CC1 19723,c1(C(=O)OCC)nccnc1NC(C1CC1NC(c1cccc(C)c1)=O)=O 19724,C1(CNC(c2nnnn2C)CCc2c(F)ccc(OC)c2)CCOC2(CCC2)C1 19725,Cc1cc(F)cc(C(=O)NC2CCCN(C(C3CCCN3C(N)=O)=O)CC2)c1N 19726,n12c(C)cc(c1C)C=CC(=O)NC1CC1NC(=O)C2.C(=O)(C(C)CC)N.CCC 19727,N1(C(c2c(C)nn[nH]2)=O)CCCCCCC1C(N1CCC(C)(CO)C1)=O 19728,Cc1cn(C)nc1C(=O)NC1(C)CN(C(C2CC(F)(F)C2)=O)C1 19729,C(=O)(C1=CCN(C(=O)CC(C)C2CC2)C1)N(C(CC(CC)C)C)C 19730,N1(C(=O)Nc2cc(F)ccn2)CCn2cc(-c3cccnc3OCCO)nc2C1 19731,C1(C(=O)NC23CN(C(c4c(C)n(C)nn4)=O)C(CC2)C3)CNC(=O)CC12CCC2 19732,C#CCC(C)(CNC(=O)C(CCSC)NC(=O)C(C)C(C)(C)C)CO 19733,C(=O)(C1CCCc2nncn21)NCCNC(c1c(C(F)F)ccc(C)c1)=O 19734,N1(C(C2C(CCC)CCC2)=O)CC2CC1CCC2NC(C1(COC(C)C)CC1)=O 19735,c1(C(=O)NC2CC(C)(NC(C(CC)CN(C)C)=O)C2)cc(O)cc(F)c1 19736,N1(CC(c2c(C)ccnc2)=O)CCC(C#N)(C2CCO2)CC1 19737,C1(CNC(C=CC=CC)=O)CN(C(c2n[nH]cc2C2CCC2)=O)CCC12CCC2 19738,C1(OC)CCC2(C(N3CCC(C)C3CNC(C3C=C(C)CS3)=O)=O)CC12 19739,N#CC1(C(=O)NC2CC(CNC(C3(S(N)(=O)=O)CCC3)=O)C2)CC2CC2C1 19740,C=CC(C)(O)CC(=O)NC(CCN(C(=O)CNC(C1CCC1)=O)C)C(C)C 19741,CCC(CC1CCCCC1)C(=O)NC1CCCCC1CNC(c1[nH]ccc1C)=O 19742,N1(C(C2(CC)CC2)=O)CCCC(C)(CNC(=O)CS(=O)(=O)NC2CC2)C1 19743,CC(C)C(C)(C)C(=O)NCc1nc(C(=O)NC2CNC(=O)C2)co1 19744,C1(C(=O)OC)Cc2ccccc2C1NC(=O)CC1C(=O)ON=C1C 19745,C1(F)(CNC(c2cc(C)nn2C)=O)CCN(C(=O)C(C)(Cl)Cl)CC1 19746,C12(NC(c3nnc(-c4cccs4)o3)=O)CC(c3ccccc3)(C1)C2 19747,Cc1cccc(C(=O)N(CC(C)N(C(=O)CCSc2ccccc2)C)C)c1C 19748,Cn1c(CN(C=O)Cc2ccco2)ccc1C=O 19749,c1(C(N2C3C(NC(c4coc(O)n4)=O)C(C3)C2)=O)ccc2c(c1)CCCC2=O 19750,C1(CC)CN(C(C23CC(F)(C2)C3)=O)CCC1NC(c1conc1C)=O 19751,C1(C(N(CC(C)CNC(=O)CCC2CCOCC2)C)=O)OCCC1(C)C 19752,C(CCCCC(=O)N(C1CCN(C(c2cc(C)cs2)=O)C1)C)OCC 19753,c1(C(N(CC(=O)Nc2ccc(SC)nc2)CC#C)=O)[nH]ccc(=O)c1C 19754,C1(CN(C(c2ccc(OC)nn2)=O)C)CC2CCC1CC2 19755,C(=O)(CC(C)(C)C(F)F)NCCCCC(C)NC(C1CCS(=O)(=O)C1(C)C)=O 19756,c1(NC(C2(C(=O)ON(CC)Cc3ccccc3)CC2)C2CC2)cccc(Br)c1F 19757,c1(NCC)ncc(C(N2CCC2CC(C)C)=O)cc1-c1cccc(C(F)(F)F)c1 19758,C1(C(NOCCC#C)=O)CCC(C)(C)N(C(=O)C=CC2CCCN2C)C1 19759,C(=O)(CC(C)(C)NC(=O)C=CC1CCOC1)NC1C(CN(C)C)C1 19760,C1(C)(CNC(c2ccc(C(C)C)o2)=O)CN(C(=O)COC2(C)CCC2)CCO1 19761,n1(CCC(=O)N(C2CCN(C(CC(=O)OCC)C)C2)CC)ncn(C)c1=O 19762,N1(C(C2(CCC)CCC2)=O)CC2(CCC(CNC(=O)C(C)CC(C)(F)F)O2)C1 19763,Cc1cc(-n2cc(C(C(C)C)NC(=O)C(CO)NC(N)=O)nn2)cc(C)c1 19764,c1(OCC)nccc(C(=O)N(CC(O)CN(C)C(C2(CC)CC2)=O)C)c1F 19765,C1(CNC(c2nnc(CC)s2)=O)CC2COCC2N1C(c1sncc1C)=O 19766,N1(C(c2ncn(CC)n2)=O)CCC(NC(c2c(C(F)F)nn(C)c2C)=O)C(C)C1 19767,C1(NC(CN2CCC(C)C2)=O)CCCCN(C(c2cccc(OC(F)F)c2)=O)C1 19768,C(C)(C(C)(C)C(=O)NCC12CCCC1CCO2)NC(C(C)OCOC)=O 19769,C1(C(N2CCC(C3CC3)CC2)=O)CCCN(CC2CCCCC2)C1 19770,N1(C(CC(=C=C)C)=O)CC(CNC(=O)Cc2cnc[nH]2)CC(C)C1 19771,C1(NC(c2ccncc2Cl)=O)CC2CN(C(C3CCCSC3)=O)CC12 19772,C1(NC(c2coc3c2COC3)=O)CCCC2CN(C(=O)CC3CC34CC4)CC12 19773,c1(C(N2CC3C(CNC(C4(CCOC)CC4)=O)C3C2)=O)cc(=O)cc(Cl)[nH]1 19774,N1(C(c2cc(Br)ncc2Br)=O)CCC2CN(c3ncc(F)cn3)CC2C1 19775,c1(C(=O)NC(C(=O)NCCNC(=O)NC)CCOC)cccc2ccoc12 19776,C1(NC(c2cc[nH]n2)=O)CCOC2(CCN(C(C34CCCC3CCC4)=O)CC2)C1 19777,C1(N(C(=O)C(C)n2ccnc2)CCC2(COC)CC2)CCCC12CCNCC2 19778,c1(C(=O)NC(COC)CC(F)(F)F)ccc2n1CCNC2 19779,N1(C(c2nc(CNC(C3N(C)CCOC3)=O)oc2)=O)CCC(O)C(O)C1 19780,C1(C(=O)NCC(C)(CNC(C23CCC(CC2)CC3)=O)OC)CCC(=O)CC1(C)C 19781,Cc1cccc(F)c1CNC(c1nc(CC2CC2)cs1)c1nnnn1C(C)C 19782,c1(CNC(C2CCN(C(CC(C)C)=O)C2)=O)ccc2ccc(O)nc2c1 19783,CC1CCCN(C(c2cccnn2)=O)C1CCNC(c1cc(F)ccc1Br)=O 19784,N1(C(C(C)OCCCC)=O)CCCC(C)(CNC(C2(C)CCCO2)=O)C1 19785,N(C(=NCC=Cc1ccc(Br)cc1)NCC1CCOC1)C(C)CF 19786,c1(CC)nc(O)c(C(=O)NC2CCCCC2CNC(C2(CF)CC2)=O)cc1C 19787,N1(C(c2c(CC)ncnc2)=O)CCC(NC(=O)CSCCC(C)C)C(O)C1 19788,C1(C(=O)NC2(C(C)O)CC2)CCCC(NC(C2COCC2(C)C)=O)C1 19789,N1(C(c2cc(I)c(F)cc2F)=O)CCC2C(CCN2Cc2cccc(Br)c2F)C1 19790,N1(C(Cn2c(C(C)C)nnn2)=O)CCC2CCC(C1)N2Cc1cc(C2CC2)no1 19791,C(C(C)C(F)C(=O)NCC(C1CCCCC1)C)NC(c1scc(CC)c1)=O 19792,CC1C(C(=O)NC23CC(NC(C4OC(C)(C)OC4(C)C)=O)(C2)C3)C(O)C(=O)N1C 19793,c1(NC(C2CCCCN2C(c2ccnnc2O)=O)=O)cc(Cl)ccc1CO 19794,CCC1=C(C(=O)NCC(C2CC2)NC(c2cn(C)nc2C(F)(F)F)=O)SCCO1 19795,c1(CC)ncnc(N2CCCC23CC(C(=O)N(C(C)(C)C)CC)C3)c1F 19796,C1(C(=O)NCc2cn(CCNC(CCc3n(C)ncc3)=O)nn2)C2CC2C2CC12 19797,C1(CC(=O)NC2C(OC)CCCC2)C2CCCC2N1C(c1nscc1C)=O 19798,N1(C(C2N(C(c3n(C=C)ncc3)=O)CCC(C)C2)=O)CCC2(C=CCO2)C1 19799,N1(C(c2ncc(C)cc2F)=O)CCC2C(CCCN2C(=O)CC(C)(F)F)C1 19800,C1(C(=O)NCCN(CCC)C(c2ccnn2CC(C)C)=O)CCCC1S(C)(=O)=O 19801,CCS(=O)CC(=O)NCC(c1ccc(F)cc1)NC(C1(OC)CC1)=O 19802,Cn1nc(C2CC2)cc1C(=O)NCCCCCCNC(=O)CC1CNC(=O)C1 19803,C(=O)(CC(C)N(C)CC)NCC(CC)NC(=O)CCc1sccc1Br 19804,N1(C(C(C(CC)C)O)=O)CCCC2(C1)CN(C(=O)CN1CCP(C)(=O)CC1)C2 19805,CC1(C)CCOC(CC(=O)NC2CN(C(C3CN4CCN3CC4)=O)C2)C1 19806,c1(C(N(C)CC=CC(=O)NCCCS(N)(=O)=O)=O)cc(N(C)C)ccn1 19807,c1(CC(CC2(C)CC2)(C)C)nc(C2Cc3ccccc32)nn1C1CCCCCC1 19808,c1(NC(CNC(c2ccc(OC)nc2)=O)CC(C)C)c(Cl)cccc1[N+](=O)[O-] 19809,N#CC1(C(=O)NCC2CCN2C(=O)CCCCCNC(N)=O)CC2CCC1CC2 19810,C(=O)(C(CC(N)=O)NC(=O)CCOC1COC1)NC(CCC=C)CO 19811,C=CCCCC(=O)NCCC1(C(=O)NC2(C3CCC3)CC2)CCC1 19812,CC(C(C)(C)CO)NC(=O)C(C)(C1CC1)N(C(=O)COc1ccn(C)n1)C 19813,c1(C(=O)NCC2(CO)CCN(C(C(CC)OCC)=O)C2)c(Cl)ccc(C)c1O 19814,N1(C(C2CCC(C)CC2)=O)CCC(NC(c2cnn(C3CC3)c2)=O)CC(C)(C)C1 19815,c1(NCC(c2ccc(Cl)cc2)C)cc(S(=O)(=O)N)ccc1C#N.N1(CCF)CCCC1 19816,N1(C(C(C)C)=O)CCN(C2CCC(NC(C3(C)CCC(C)C3)=O)CC2)CC1 19817,C1(NC(c2cn(C)nc2C2CC2)=O)CCCCN(C(=O)CO)CC1 19818,N1(C(C(CC)OCC)=O)CCc2nc(CNC(c3cn(C)nc3C)=O)sc2C1 19819,C(N=c1[nH]cnc2c1COC2)C1(CNC(C2CC3(CCOCC3)C2)=O)CC1 19820,C1(=O)C(CC)NC(=O)OC(CC)CN1.C1(NC(N)=O)CCCN1C(C)=O 19821,C(CCCCCC(=O)NCCC1CCC(=O)N1)NC(C(=Cc1cn[nH]c1)C)=O 19822,C12(CNC(c3c(C)coc3C3CC3)=O)CCCC1CCN2C(c1ccncc1)=O 19823,N1(C(Cc2cc(C)sc2)=O)CC2(CO)CC1(C(=O)NC1CC(O)CC1O)C2 19824,C(=O)(C(C(C)CC)NC(=O)CSCC1CC1)N(CCCO)CCC 19825,C1(NC(c2ccnc(CC(C)C)n2)=O)CN(C(=O)CC2OCCCO2)CC1C1CC1 19826,c1(CNC(C2N(C(C)C)CCC2)=O)ccc(CNC(C2CC2(C)C)=O)cc1F 19827,N1(C(C2N(C)C(=O)CC2)=O)CCC(O)(C2CCN(C(=O)C3=CCC3)CC2)CC1 19828,N1(C(C2(C)CC2(F)Cl)=O)CCC2(CC1)CCN(CC1CC(F)(F)C1)C2 19829,N1(C(C2(C#C)CN(C(=O)CS(=O)(=O)CC)C2)=O)CC(OC)C(C2CC2)C1 19830,c1(CN(CCNC(C)=O)C(=O)OCC(C)(C)C)ccccc1C1(C)CC1 19831,c1(C(=O)NCCNC(c2nocc2Cl)=O)c[nH]c2ccc(Cl)cc2c1=O 19832,c1(C(=O)OC)ccc(N2CC(CCNC(=O)Cn3ccnc3C)(OC)C2)nc1 19833,c1(NC(C2CCCC2NC(c2cn(-c3ccccc3)nn2)=O)=O)c[nH]nc1Br 19834,c1(C(=O)NC(CCC)CCCNC(=O)CCS(C)(=O)=O)ccncc1N=[N+]=[N-] 19835,Cc1cc(C(=O)NCC2C(C3CC3)CCN2c2cc(O)ncn2)cc2nc[nH]c12 19836,c1(C(=O)NC2C=CC(C(N3CC(C(CC)CC)C3)=O)C2)ccnc(C)c1C 19837,Cc1cccc(C)c1C(=O)NCC12CC1CN(C(c1cn[nH]c1)=O)C2 19838,CCCC(O)CC(=O)N(CCNC(=O)CCNC(=O)C(C)(C)C)CC1CC1 19839,CC(C)(C)C1=NOC(C(N2CC3CC3(NC(c3ccns3)=O)C2)=O)C1 19840,C1(NC(C(=O)NCC)=O)C2CCCN(Cc3cc(C)ns3)C2C1(C)C 19841,c1(C(N2CC(O)(CCNC(C3C(C)(C(F)F)C3)=O)C2)=O)cccc([N+](=O)[O-])c1N 19842,Cc1cc(C(=O)N(C(C)CCNC(c2[nH]nnc2C)=O)C2CC2)cs1 19843,C1(CC)CN(C(c2cncn2C)=O)CCC1CNC(c1ccnn1C)=O 19844,C1(C(=O)NC(c2ccccc2)C#N)CC(F)CN(C(c2cc(O)n[nH]2)=O)C1 19845,N1(C(C(CC(C)C)(F)F)=O)CCCC2(C1)CN(C(c1ccnn(C)c1=O)=O)C2 19846,C(=O)(CS(=O)(=O)NC1CC1)NCC(C)CNC(=O)C(N1CCCC1)C1CC1 19847,c1(C(N2C(C)CN(C(C3(C)CC=CCC3)=O)CC2)=O)cccn2ccnc12 19848,N1(CC)CC(C(=O)NC2CN(C(C3(C)CC=CC3)=O)CC2C)CC1=O 19849,c1(C(=O)NCC2CC(NC(=O)C(F)(F)c3nccs3)C2)cc2c(Cl)cncc2s1 19850,c1(C(N(CCCNC(C(CCC)NC(C)=O)=O)CC)=O)c(Cl)ccc(Cl)c1O 19851,C12(CNC(C(C)(C)SC)=O)CCC(CN(C(C34CCC(C)(C3)OC4)=O)C1)C2 19852,CC1CC(O)CN(C(C2CCN(C(=O)Cc3ccsn3)C2)=O)C1 19853,C1(CNC(COCCCC#C)=O)C(C2CC2)CCN1C(=O)C#CC1(C)CC1 19854,Cc1cccc(Cl)c1N1CC(C(=O)NNC(=O)c2cc[nH]c2)CC1=O 19855,c1(C(=O)NC2CCC(C)N(C(C3C4CC5C(C4)C35)=O)C2)ccc2nn[nH]c2c1O 19856,CC(C)CC(C(=O)N(CCC(=O)NC1CC12CC2)C)C(C)C 19857,N1(C(C(=O)NCC=C)c2cccs2)CCc2ncncc2C1 19858,C1(C(C)(F)F)(C(=O)NC(CN(C(C2C(C)(C)C2(F)F)=O)CC)C)CCOCC1 19859,c1(OC)ccc(NC(=O)NC2CCCN(C(=O)CCCCC#N)C2)cc1C 19860,c1(C(=O)OC)ccc(COC(c2occc2Br)=O)c(OC)c1 19861,C(=O)(C(CC(C)C)N(C(=O)Cc1ccccc1C)C)N1CC(OC)(CO)C1 19862,c1(C(C)=O)ccc(C(=O)NCC2CC(C)N(C(=O)OC(C)(C)C)C2)cc1Cl 19863,c1(N2CC(CNC(c3cccc(COC)c3)=O)OCC2)ncc([N+](=O)[O-])cn1 19864,C12(NC(n3cc(C4CCC(C(F)F)CC4)nn3)CCC)C3CCC(CC13)C2(F)F 19865,Cc1sc(O)nc1C(=O)N(C)CC1CCN(C(=O)COCC(F)F)C1 19866,c1(C(N2CCC(C)(NC(CCCCCC)=O)C2)=O)c(F)cc(OC)c(F)c1F 19867,C1(C(N2CCC(OCCNC(c3cc(F)c[nH]3)=O)CC2)=O)CCCC(C2CC2)O1 19868,C1(OC)CCN(CC(=O)NC(C)(C)CNC(=O)CN(CCOC)C)C1 19869,c1(CC(N2CC(O)(C(C)NC(C=C(C)C3CC3)=O)C2)=O)cc(F)ccc1F 19870,C1(CNC(c2ccc(F)cc2)=O)CCC2(CN(C(C3(CO)CCC3)=O)C2)O1 19871,C1(SC)CN(C(=O)CC(F)(F)F)CC1C(=O)NC1CC(N(C)C)C1 19872,O=C(CN=c1nc2sccc2c(N2CCC(C3CC3)C2)[nH]1)NCC1CC1 19873,c1(C(=O)NC(CNC(C2N(CC)CCC2)=O)C(C)C)ccn(CC)c(=O)c1 19874,c1(C(=O)NC2C(NC(c3n(CC#C)ccc3)=O)CC2)cc2n(c1)CCC2 19875,c1(C(N2CCC(C)(NC(=O)CC3CCCC(=O)C3)C2)=O)onc2c1CCCC2 19876,N1(C(Cc2n(C)c(S)nn2)=O)CCCC(F)(CNC(=O)CC2CNC(=O)O2)C1 19877,Cc1ccn(CC(=O)NC2CC(N(C)C(c3coc(C4CCC4)n3)=O)C2)c(=O)c1 19878,c1(C(N2C3C(NC(c4ccc(C)nn4)=O)C(C3)C2)=O)n[nH]cc1[N+](=O)[O-] 19879,C1(CNC(COC(CC)(C)C)=O)CC(O)CN1C(=O)C(CC1CCCCC1)OC 19880,N1(C(c2c(C)cc(N)c(Br)c2)=O)CCCC2(CCCCC2NC(=O)C2CC2)C1 19881,CCC(CCOC)C(=O)NCC1CC(OC)CN1C(c1ccccc1CC#N)=O 19882,S(=O)(=O)(CCCCCl)NC1CCC(CN2CCC(C(N3CCOCC3)=O)CC2)C1 19883,C=CCCCCC(=O)NC(CO)C(C)NC(c1ccnc(OCCOC)c1)=O 19884,N1(C(C2CCC2)=O)CC2C3CCC(C2C1)N(C(c1c(F)cc(F)cc1Cl)=O)C3 19885,CON1CCC(CN(C)Cc2ccc(O)cc2)CC1 19886,N1(C(C=C(C)C(F)F)=O)CCC(NC(C23CCC(C2)C3)=O)C(C(C)C)C1 19887,c1(C(N2CC(NC(=O)C=C(Cl)Cl)C(CO)CC2)=O)ccn2nccc2n1 19888,c1(C(=O)N(c2ccc(OC)c(F)c2F)C)cccc2sc(CN)nc12 19889,c1(C(=O)NCC(CNC(CC2(C)CC2(F)F)=O)CO)ccc2c(c1)NC(=O)CN2 19890,c1(C(=O)NCC2CC(OC)CN2C(=O)C(C)NC(C)(C)C)ccc2ccsc2c1 19891,CC1CCN(C(=O)COCCN(C)C(C2CC23CC3)=O)C1 19892,c1(CC)ccoc1C(=O)NCCCCNC(c1ccc(-c2ccco2)[nH]1)=O 19893,S(=O)(=O)(C=Cc1ccccc1)N(C1C(F)(F)CCN(C(c2ccc[nH]2)=O)C1)CCO 19894,N1(C(C(CSC)C)=O)CC(O)CC1CNC(c1nc(C2CC2)cs1)=O 19895,C12(C(=O)NCC3C(NC(CSCCOC)=O)CCCC3)CCN(CC1)S(=O)(=O)C2 19896,CCC(C)(CNC(=O)C=Cc1ccncc1)C(=O)N(C)CC1(C)CCCC1 19897,N1(C(C(CCC)C)=O)CC2(CCC2)CC1CNC(C1(NC(C)=O)CCCC1)=O 19898,c1(C(=O)NCC(CNC(CC2(OC)CCCCC2)=O)F)c(C)cc(F)cc1C 19899,N1(C(Cn2c(=O)ccc(C)n2)=O)CCC2CCN(C(c3oncc3C)=O)CC12 19900,C1(NC(C2C(CC)OCC2)=O)CC=C(C(=O)N(C(CC)C(=O)OC)C)C1 19901,CC(C(=O)NC1CC2(C1)CC(NC(=O)CSc1ccncc1)C2)C(C)(F)F 19902,C1(C(=O)Nc2ccc(CCO)cc2)(CC)CCCN1C(C1CC2CC2C1)=O 19903,O=C(CCCCC(F)F)NCC(C1CCOC1)NC(=O)CC1(CO)CCCC1 19904,C(=O)(CCC(N)=O)N(C)CC1CC1.C1(O)CCN(C(=O)CCOCC(F)F)C1 19905,C1(C(=O)NC2C=CC(CNC(C3(C(F)F)CCCC3)=O)C2)(OC)CCSC1 19906,c1(OC)ccc(C(=O)N(C)Cc2cc(Cl)ccc2C)c(Br)c1 19907,c1(OC2CCCC(C(CNC(CC(=C=C)C)=O)NC=O)C2)ccccc1C#N.OC 19908,C(C1CCCC1)=CC(=O)NC1CCC1CNC(C1CCC(C(F)(F)F)O1)=O 19909,C(=O)(C1=CCCCCC1)NC(C(=O)NCC1CC[Si](C)(C)C1)C1CCCC1 19910,c1(NC(COC(C(CCOC)C)=O)=O)ccc2c(c1)CCC2 19911,Cc1cc(C)n(C(C)CC(=O)NC(C2CCCN2C(=O)CCC(=O)C2CC2)C)n1 19912,C(=O)(C(C)CC(=O)c1ccccc1F)NCC(C)NC(C(N1CCNC1=O)C)=O 19913,C1(CC(C)C)CCN(C(=O)CC2CCCC(NC(c3cc(C#N)cs3)=O)C2)CC1 19914,c1(OC)cc(C(=O)NCCCN(C(=O)C(C)C(F)F)Cc2ccccc2)ncn1 19915,c1(C(N2CC(CNC(C3CC(OC(F)F)C3)=O)C3(CC3)C2)=O)cccc(F)c1Cl 19916,c1(C(=O)NC2CCN(c3c(OC)c(Cl)ncn3)C2)cc2nc(=O)ccn2[nH]1 19917,Cc1sc(C(=O)NC(C(=O)OC(C)(C)C)C2CC2)c(C#N)c1C 19918,C1(NC(c2c(C)cn(C)n2)=O)C2COCC1CN(C(=O)C=Cc1scnc1C)C2 19919,C(C)(C)(C(=O)NC(Cc1ccco1)C(=O)OC)N(CC)CC 19920,N1(C(C2C(=C)CC2)=O)CCN(c2ncc(C(F)F)cn2)C(C)C1 19921,O=C(C1=CC2(CCN(C(=O)C(F)n3ccnc3)C2)C1)NCC1(CC2CC2)CC1 19922,N1(C(=O)CC(F)F)CCN(C(c2ccc(C(F)(F)F)cn2)=O)C(CF)C1 19923,C(=O)(C(C)(C)C1=CCN(C(=O)CC=CCCCCC)C1)NCCCC=C 19924,N1(C(CC=CC)=O)CCCC(F)(C(=O)Nc2ccc(F)c(CO)c2)C1 19925,c1(C(=O)NCC(CC(C)C)NC(C(COC)(C)C)=O)cnn2cc(C)cnc12 19926,N1(C(c2scc(C(C)=O)c2)=O)CCCC(C)(NC(=O)CCN2CCCC2=O)C1 19927,CC(CC(F)(F)F)C(=O)NCC(C)(C)CCNC(c1cccc(NCCO)c1)=O 19928,c1(C(N(CCCCCNC(=O)CNC=O)C)=O)ccc2ocnc2n1 19929,C1(Oc2c(NC(N3CC(OC)C3)=O)cccc2)CCc2c[nH]nc2C1 19930,N1(C(Cc2c(C)ncs2)=O)CC2CC(N(C(=O)COCCOCCO)C)C1C2 19931,N1(C(C(F)=C(C)C)=O)CCN(C(C2CC2(Cl)Cl)=O)C(C(C)C)C1 19932,N1(C(Cn2c(C(C)C)ncc2)=O)CCCC2CN(C(=O)C=CC=C(Cl)Cl)CC12 19933,Cc1nc(NC2CCSC2)cc(N2CCC(c3nnn(C)n3)CC2)n1 19934,C1(N(C)C(c2cncnc2)=O)CCCC2CN(C(=O)CC3(O)CCC3)CC12 19935,c1(C(N2CC(CCOC)N(C(=O)CCNC(C)=O)CC2)=O)cc2oc(C)cc2[nH]1 19936,C(c1c(C)nn(C)c1Cl)=CC(N1CC(OC)(CNC(c2cnc(=N)[nH]c2)=O)C1)=O 19937,c1(C(=O)OC)ccc(CC(=O)NC2CC(CNC(=O)CN3CCC(C)C3)C2)cc1 19938,N1(C(CCOC)=O)CC(c2cccc(F)c2)C(CNC(c2cn(C)nc2Cl)=O)C1 19939,Cn1cc[nH]c(=NNC(=O)C2CCc3ccccc3C2=O)c1=O 19940,C12(C(=O)NC3CCN(C(=O)Cc4ccsc4)CC3)CCCCC1C2Br 19941,O=C1CCOCCN1Cc1cn(CCC(=O)NCc2cc(Br)ccc2F)nn1 19942,C(CC(C)C(=O)NC(CO)C(=O)NCc1ccncc1Cl)=CCC 19943,C1(CCOC)(NC(c2ccc(Br)o2)=O)CCN(C(=O)Cc2ccco2)C1 19944,c1(C(=O)NCC(CO)NC(C2(OCC)CCOC2)=O)cccc2nc(O)ccc12 19945,n1(CC)cncc1CN1CCCC1CCC(N1CCOCC1)=O 19946,CC1(C)CC(NC(=O)Cc2ccc(Br)cn2)CN(C(C2COCCO2)=O)C1 19947,Cc1noc(C)c1CC(C)C(=O)N1CCC(NC(=O)Cn2nnc(=N)[nH]2)C1 19948,N12CC(C(=O)NOCC3CCCNC3=O)C(=CC1=O)C2.N(CCO)(CC)CC 19949,C(=O)(CC1=CCN(C)CC1)NCC1(C(N2CC(C)C(F)C2)=O)CC(=C)C1 19950,c1(C(C)=O)cc(C)n(CC(=O)NC2CC(NC(=O)C(=O)N(CC(F)F)C3CC3)C2)n1 19951,c1(C(=O)NC2CN(C(c3nc(C)oc3)=O)CC2(C)C)ccc2cccnc2n1 19952,O=C(CCC(F)(F)F)NCC1CC1NC(c1cnn[nH]1)=O 19953,c1(CNC(CC(C)CF)=O)nc(CNC(=O)C(CO)c2ccccc2)cc(O)n1 19954,C1(N(c2ccc(CO)o2)C)CCC2CN(C(c3ccc4occc4c3)=O)CC12 19955,C1(C(=O)NCC(C)(CNC(c2cc(C3CCOC3)[nH]n2)=O)OC)CC2(CCC2)C1 19956,N1(C(CSCCNC(=O)C=CC(F)(F)F)=O)CCC(F)(CO)CC1 19957,c1(C(N2CCC3(NC(=O)Cc4cscn4)C(C2)C3)=O)cc2c(O)ncnc2cn1 19958,C(=O)(C(F)CCC(C)(C)C)N1CCC(CC#C)(C(=O)NCC2CC2(Cl)Cl)C1 19959,C1(C(N2CC(O)(CCNC(c3n(C)c(Cl)nc3)=O)C2)=O)CC1C1CCCC1 19960,C#CCC(CC(F)F)C(=O)NC1(C)CCCN(C(C2CCC=CCCC2)=O)C1 19961,CCCC(CCCO)C(=O)NC1CCN(C(c2cccc(O)c2C)=O)CC1(C)C 19962,C(=O)(CN1C(=O)COc2ccc(Cl)cc21)NCCC(N1CCC(N(C)C)CC1)=O 19963,C(c1cccc(F)c1)=C(C(=O)NCC1N(C(C(N2CCCC(O)C2)C)=O)CC1)F 19964,C1(CNC(C(=Cc2cn[nH]c2)C)=O)CN(C(=O)C(F)C(C)(F)F)CC1(C)C 19965,N1(C(C(C(C)C)C)=O)CCC2(CC2NC(c2ncccc2F)=O)C1 19966,C1(CC(=O)NCC(C)N(C(C)=O)C)C(=O)NN=C1C.C1(C2C(=O)N2)CCCCC1 19967,C1(C(N(CCN(C)C)CCO)=O)CC2CCC1N2C(=O)CCCOC(C)(C)C 19968,C1(NC(C=CS(C)(=O)=O)=O)CC2(CCCN(C(C3CC4CCC3C43CC3)=O)C2)C1 19969,N1(C(C(C)(C)CCF)=O)CCC2CN(C(C3CC(=O)OC3(C)C)=O)C2C1 19970,C1(NC(c2cn(CCC)nc2C)=O)CCC2CN(C(C34CC(C3)C4)=O)CC2C1 19971,C(C(N=[N+]=[N-])C(=O)N(CCC(=O)Nc1cscc1C)CC1CC1)OCC 19972,CC1(C)C(C)(C)C1(F)C(N1CCC(CC(=O)NCc2cccc(N)n2)C1)=O 19973,C(=O)(CC(C)(C)COC)NC(c1nc(NC(COC)=O)sc1)C1CC1 19974,c1(N(C(=O)COCCCN=[N+]=[N-])C)ccccc1C1CCC1 19975,c1(C(=O)NCC2N(C(C3C(=C)C3C(=O)OC)=O)CC(O)C2)cccc2c1CNC2=O 19976,CC1(CNC(=O)CCn2ccnn2)CN(C(c2ccsc2C(F)F)=O)CCO1 19977,CN=c1[nH]c(=NCCCCCCNC)[nH]c(=NC(C)CC(N)=O)[nH]1 19978,CC1(NC(=O)CC2(O)CCC2)CCC(NC(C2C=CCC2)=O)CC1 19979,c1(NCCN2C(CC(=O)OCC)CCCC2)ccc(C#N)cc1C(F)(F)F 19980,C1(NC(C(N)=O)=O)CC(C2CCN(C(c3n[nH]c4c3CCOC4)=O)CC2)C1 19981,C1(n2cc(SC(C(OC)OC)C)nn2)CN(C(c2conc2C)=O)CC1C 19982,c1(C(N2CC(CC(C)NC(=O)CCS(C)(=O)=O)C2)=O)ccc2c(c1)OCO2 19983,N1(C(c2cc(CCC)[nH]n2)=O)CCC(O)C(NC(c2ncoc2CC)=O)C1 19984,c1(NC(C)=O)ccc(C(=O)NCCCN(C)C(c2ccc(CO)cn2)=O)cc1F 19985,C1(C(N2CCC(CO)C(O)CC2)=O)CC12CCN(C(C1(CO)CC1)=O)CC2 19986,c1(N(C)C)ccc(C=CC(=O)NC2CCCC2NC(=O)CCn2ccnc2)cc1 19987,O=C(C1=COCCO1)NCC1(NC(C2CC3C=CC2C3)=O)CCCCC1 19988,CC(=O)C(C)CC(C)C(=O)NC(C(=O)NCCSCCCO)C1(O)CCC1 19989,c1(C(N(CCCNC(c2c[nH]ccc2=O)=O)CC)=O)cc(OC)cc(C)c1 19990,C1(N(C(=O)CC(F)(F)F)CCO)CC2(C1)CN(C(=O)CNCC(F)(F)F)C2 19991,c1(C(N(CC(C)NC(=O)COCC2(C)CNC(=O)C2)CC)=O)ccncc1OC 19992,c1(C(N(C2CCN(C(C(C(C)C)OC)=O)C2)C)=O)cc2nccn2c(O)n1 19993,C1(CN(C(=O)CC2CC(SC)C2)CC)CCN(C(=O)C(c2ccccc2)C)CC1 19994,N1(C(c2ccc(OC(CC)C)cc2)=O)CC2(CC([SH](C)C(=O)OC)=NC2=O)C1 19995,c1(C=O)cc2nc(C)sc2[nH]1.C(=O)(C(C)(COC)OC)N(CCOC)CCOC 19996,N1(C(C2(C#N)CCC2)C(=O)NCC(F)F)CCN(Cc2ccc(F)cc2)CC1 19997,C(CCN=c1[nH]c(=NC2CC(n3ccnc3)C2)c2c(F)cccc2[nH]1)=CCCC 19998,C(O)(C(=O)O)(C(F)(F)F)c1cnc(NC(c2c(C)oc(C(C)C)n2)=O)s1 19999,N1(C(c2c(CC)ccs2)=O)CC2CCC2(CNC(=O)CC2CCCC(C)(C)C2)C1 20000,C1(C)(C(=O)OCC)CN(C(=O)CCCCCF)C(C)(C)C1.C1C(CO)C(=O)N1 20001,C(=O)(C1SCCc2sccc21)N1CC(CCCNC(C(C)(C)c2cc[nH]n2)=O)C1 20002,c1(C(N2CC(CNC(C=CCCC(C)C)=O)N(C)CC2)=O)cnc2occc2c1 20003,C1(NC(c2cc(SC)oc2C)=O)CN(C(C2(C)CCCCO2)=O)CCC1O 20004,N1(CC)CCCN(C(C2OCCC2NC(=O)C(C2CCCCC2)O)=O)CC1 20005,N1(C(c2cnc(OC)s2)=O)CCCC1C1CCCN1C(=O)C=Cc1nc(C)co1 20006,C(CCC(C)(C)NC(c1sc(C(C)C)nc1C)=O)NC(C(COC)OC)=O 20007,C1(C(N2CC(OCC(=O)NC)C2)=O)CCC(O)CN1C(C12CC(C#N)(C1)C2)=O 20008,n1(CC(=O)NC2C(n3cc(C(C)OC)nn3)COC2)cnnc1O 20009,C(=O)(CC(C(=C)C)OCC)NCC(C(N1CCC(C#C)C1)=O)C 20010,CC1CN(C(c2ncccc2C(F)(F)F)=O)CC1NC(=O)Cn1cncn1 20011,CC1=C(C)CC(C(=O)NCCC(C)(C)CNC(C2CC3CC3C2)=O)CC1 20012,C1(NC(C(C)C#N)=O)CN(C(c2ccc(CN3CCOCC3)s2)=O)CC12CC2 20013,c1(C(N2CCC3(C(CNC(CCC(=C)Cl)=O)C3)CC2)=O)coc2c(OC)cccc12 20014,CC(C)CC(C)(CNC(=O)CCOC1CCN(C)C1)NC(C1CC(F)(CO)C1)=O 20015,CCCCC(C(=O)N1CC(COC)(NC(C2CCCCN2C)=O)C1)NC(N)=O 20016,CC(C)CC(CC(=O)O)NC(c1cnc(C2CCC2)s1)=O 20017,c1(CC)nnc2cc(NCC=CCNC(=O)CCC3CC(OC)C3)ncn12 20018,C(CCCC(=O)NCC(C(C)C)NC(=O)C=Cc1ccc(C(N)=O)o1)SC 20019,C1(NC(c2ccc(C)o2)=O)COCCC1NC(C1(F)CC=CCC1)=O 20020,N1(C(C2N(C(C)=O)CCCC2)=O)CCC(C)C(NC(=O)Cc2cnco2)C1 20021,c1(C(N2CC(OC)(CNC(=O)CCOCC(C)C)C2)=O)cc2c(C)[nH]nc2s1 20022,N1(C(C(c2cccc(F)c2)C)=O)CCN(C(=O)C(O)C2CCC2)CC(C)(F)C1 20023,c1(C(=O)NC2CCN(C(=O)C=Cc3cccs3)CC2F)ccnc2cc[nH]c12 20024,c1(C(=O)NC2CCN(C(CC(C=C)C)=O)CC2)cc(Cl)ncc1O 20025,C1(C(N2CCC(CN(C)C(c3cnco3)=O)C2)=O)CC2CC(C1)CS(=O)(=O)C2 20026,O=C(CC1CCc2ccccc21)N1CCC2CCN(C(=O)C=C(Cl)Cl)C2C1 20027,c1(NC=O)ocnc1C1(C(=O)OC)CCC1.C12(CC1O)COC2.CCOC.OC 20028,N1(C(c2cccc(C)c2)=O)CCN(C(=O)COC2CCOC2)CC1CC(F)F 20029,CC(=O)C(C)CC(C)C(=O)N1CCN(C(=O)C#CC2CCC2)C(CO)C1 20030,N1(C(CCC(=C)C)=O)CCC(NC(=O)CC2(CSC)CC2)(OCC)CC1 20031,C1(C)(NC(Cc2nc(CC)sc2)=O)CCN(C(c2cc(C)ccc2F)=O)CC1 20032,Cn1cc2c(n1)CC(CN1CCCC(C(c3ccccc3)O)C1)CC2 20033,N1(C(C2CC(OC)C2)=O)CCC(NC(=O)C=CC(C)(C)C)C1C(C)(C)C 20034,C(=O)(CCC(=O)N(C)C)N(C1CCN(C(CCCSC)=O)C1)CC1CCCC1 20035,Cn1cc(C(=O)NCCC2(NC(=O)C(O)C3CCC3)CC2)c(-c2cnccn2)n1 20036,C(=O)(CC(C(F)F)NC(=O)CC1CC(F)(F)C1)NCC1N(C)CCOC1 20037,C1(N(C(c2ccn(CCC)n2)=O)C)CCC(NC(=O)COCC2CCCC2)CC1 20038,C1(NC(c2nc(C)oc2)=O)CCCCC12CCN(C(C1CSC1)=O)C2 20039,C(=O)(C(CC1CCCC1)C(C)C)NCC1(NC(C=C(C)C2CC2)=O)CCOCC1 20040,c1(C(N2CCC(C(F)(F)F)(OC)C2)C(=O)NCC)ccc(OC)cc1Cl 20041,C1(n2c(-c3ccc(CC4CCC4)o3)nc(CCCN(C)C)n2)CCOC(C)(C)C1 20042,CC1CCCC(C(=O)NCCCOCCC(=O)NCc2ccn(CCF)n2)C1 20043,C(=O)(C1=CCCCCC1)NC(C)CCCCNC(=O)CNC(C1CCCCC1)=O 20044,c1(CSCC(=O)N(C)CC2CN(C(=O)C(C3CCCCC3)O)C2)ccccc1 20045,c1(C(N2CCCC(CCNC(c3cnn(C)c3Cl)=O)C2)=O)cc(F)cc(Cl)c1N 20046,C=C(C)CC(C(=O)N(C)CC1COCCO1)NC(=O)C=C1CCOCC1 20047,N1(C(C(=O)NCCC(C)NC(=O)C(C)(C)c2cccs2)C)CCP(C)(=O)CC1 20048,CCCCC(O)C(=O)NC1C2CC1N(C(c1cc(-n3cccc3)ccn1)=O)C2 20049,C1(C(=O)NCC2CC(OC)C2)(NC(c2cnncc2C)=O)CCN(C)C1 20050,Cc1ccc(C(=O)NCC(CNC(=O)COC(F)F)C(F)(F)F)cc1Br 20051,N1(C(CC)=O)CC(N(C)OC)C1.c12n[nH]cc1C(=O)NC2 20052,C(=O)(CCC(F)(F)C(F)F)NC1CCC(CCNC(c2c(C)cnnc2O)=O)C1 20053,N1(C(C(COC)(C)OC)=O)CCC2(CC1)CN(C(C1(C(C)C)CCC1)=O)C2 20054,c1(C(C)OC)cn(CC2C=CCN2C(c2cc(C(C)=O)on2)=O)nn1 20055,N1(C(CC(C(C)C)O)=O)CCC(C2(O)CCN(C(=O)CN3CCCC3=O)C2)CC1 20056,c1(OC)c(C(=O)NC(CNC(=O)Cc2ccc(C)nc2)CO)ccnc1Cl 20057,c1(C(=O)NCC2CC(CNC(CSS(C)(=O)=O)=O)OC2)cc2ccnc(Cl)c2s1 20058,c1(C(=O)NCCCC2(NC(COC(CC)C)=O)CC2)cnc(C)c(C(C)=O)c1 20059,c1(CC(=O)N(c2cccc(OC)c2)C(C)C)cccc2ccncc12 20060,C(c1ccc2c(c1)OCO2)=CC(=O)OC1COCCC1c1ccccc1 20061,C1(CNC(C2COC3(CCC3)C2)=O)CN(C(=O)C2=CCCSC2)CC12CCC2 20062,c1(C(=O)NC(C2(O)CN(C(=O)C(C)(F)F)C2)C)ccn2nncc2c1 20063,Cc1nnc2ccc(C(=O)NCCNC(C34CCCC3CC4)=O)cc2c1C 20064,Cc1cc(C(=O)NCC2CN(C(c3cnnc(O)c3)=O)CCCO2)cc(C)c1N 20065,CCCC(C)(O)CC(=O)NCC=CC(N1C(CO)CC1CO)=O 20066,C1(C)(C(=O)NCCCCC(C)C)CCCN(C(C2CCCN(C)C2)=O)C1 20067,C#Cc1c(Br)cc(Br)c(NC(C2CCCCN2C(=O)OC(C)(C)C)(C)C)c1Br 20068,CCC(C)(C)CC(=O)N(C(CC(F)F)C(=O)N1CC(N(C)C)C(F)C1)C 20069,C(CC(=O)NCCN(C(=O)CC1(C)CCC1)C(C)C)OCCC 20070,CCC(COC)C(=O)N(CC(C)(C)C(=O)NCC(C)C(=O)OC(C)C)C 20071,N1(C(C=CC)=O)CC(C)(C)CC1C(=O)NCC1COCCO1 20072,C1(C(N(C)CC2N(C(C3CC=C(C)CC3)=O)CCC2)=O)CCC(=O)C(C)C1 20073,C(CCC(C)(C)C)(C(=O)NC1CCS(=O)(=O)C1)N(C(Cc1nc(C)sc1)=O)C1CC1 20074,C(=O)(C1CCCc2nc[nH]c21)N(CC(C)NC(C1(C)CC2(CCC2)C1)=O)C 20075,CC1CCC(C(=O)NC2CC3(CCC3)C2O)N(C(=O)Cn2cc(CO)nn2)C1 20076,N1(CC(=O)NC2CCCC(NC(c3ccnc(S)c3)=O)C2)CCNC(=O)C1 20077,c1(C(=O)NC2C(C(=O)NCCN(CC)CC)CC2)cccc(C)c1O 20078,c1(OC)cncc(C(=O)NCC(C)(CO)NC(=O)Cc2nc(C3CC3)cs2)n1 20079,c1(C(=O)NC(CC)CNC(=O)CCCOC2CCOCC2)c(C(C)=O)cnn1C 20080,C1(F)(CNC(C(CC)=CCC)=O)CCC(NC(=O)C(C)(C)c2cscc2Cl)C1 20081,Cc1ccc(OCC(=O)NC2CCCC2NC(c2cc[n+]([O-])cc2)=O)cc1 20082,c1(CC(=O)NCC2(COC)CCCN2C(=O)CSC(C)(C)C)c(C)cccc1C 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20239,C(CC1=CCN(C(C2(C3CCOCC3)CC2)=O)CC1)NC(C(C)(C)C(N)=O)=O 20240,c1(C(=O)NC(CC2CN(C(C=CSC)=O)C2)C)ccccc1[N+](=O)[O-] 20241,c1(C(C)C)occc1C(N1CCCC1C1(NC(C2C3COCC23)=O)CC1)=O 20242,n1(CC=C)cc(C(=O)NCC(C)(F)CNC(=O)C(=O)NCC2CC2)cn1 20243,C1(CC)CN(C)c2ccccc2CN1C(=O)C(N1CCN(CC(=O)NC)CC1)=O 20244,C(=O)(C1CSc2ccccc21)N1CC(COC)(CNC(C2(C)COC2)=O)C1 20245,CN1CC=C(C(=O)OCCCOCc2ccccc2F)C1 20246,C1(NC(Cc2c(C)cnn2C)=O)CC2(C1)CC(CN=c1[nH]nc(C(N)=O)s1)C2 20247,C(=O)(CC(F)(F)F)NCC(C)(CO)NC(c1ccn(CC)n1)=O 20248,C1(NC(c2cccc(C)c2)CN(C)C)COCC(=O)N1C(=O)Nc1ccccc1 20249,n1(C(C)C)ncc(C(N2CCC2C(=O)NCC2(Cl)CC2(F)F)=O)n1 20250,Cc1cccc(CNC(=O)CC(C(C)C)NC(c2cn(C(C)C)nn2)=O)c1C 20251,C12(C(N(CCCNC(C3(COC)C=CCC3)=O)C3CC3)=O)CC(C)(C1)OC2C 20252,c1(CNC(C(C2CN(C(c3cn(CC)nn3)=O)C2)OC)=O)cccc(C)n1 20253,S(=O)(=O)(c1ccc(Cl)c(C(F)(F)F)c1)NC1CC(C(=O)Nc2cncnc2I)C1 20254,C1(COC)(NC(=O)C(F)OC)CCN(C(=O)C(c2ccccc2)OCO)CC1 20255,CN1CCN(C(c2cnc(C(F)F)nc2)=O)C(CNC(C2CCC3CC3C2)=O)C1 20256,Cc1nc2c(NC(c3ncccc3C(=O)Nc3nccs3)=O)cccn2n1 20257,Cc1ccccc1OCC(=O)NCCN(C1CC1)CC1(C)CC1 20258,N1(C(C2CN(C(C)=O)C3C2C3)=O)CC(CNC(=O)CCNC(N)=O)C2(CC2)C1 20259,C1(CNC(Cn2c(C)ncc2)=O)CC(C)N(C(=O)CN2C(=O)CCC2=O)C1 20260,C(C(C)(C)CC(=O)NC1(C(=O)NCCC(O)C(=O)OC)CCCCC1)OC 20261,C(C(=O)NC(C)CC)(C(C)OC)NC(CCN(CC#C)C)=O 20262,c1(CN2CC(NS(C)(=O)=O)C2)csc(Cl)n1 20263,C1(NC(c2cc(CC)ncc2)=O)CN(C(C2CCCCO2)=O)CC1(F)F 20264,O=C(C1=CN=C2N=CNN2C1)N1CCCC1C1CCN(C(=O)C(O)C2CCC2)C1 20265,CCC(CC(=O)N(CC(CC)n1cccn1)CC(=O)NC(C)C)OC 20266,C1(C(N(C(C(C)C)CO)C)=O)C2CC3C(C2NC(c2c[nH]c(=N)o2)=O)C13 20267,c1(C(=O)NCCN(C(=O)C(CO)OC)CCOC)ccc(C#N)cc1O 20268,c1(CC(=O)N(C(C)C)CCNC(C2(CCF)CC2)=O)ccco1 20269,c1(NC(CCC(F)(F)F)c2c(Cl)cccc2)nc(N2CC3CC3C2)nc2sccc12 20270,c1(C(=O)OC)cc(=NC2CCCC(N3CCOCC3)C2)c2ccccc2[nH]1 20271,Cc1cc2cc(C(=O)NCC3CCCN3C(=O)C=C3CCN(C)C3)oc2cc1C 20272,c1(C(=O)NCC(C)NC(C2(Cc3cccc(Cl)c3)CC2)=O)cnc2scnc2c1 20273,c1(C(=O)NCC2CN(C(CC(CC)OC)=O)C3C2C3)cc(Br)c(C)cc1C 20274,c1(C(c2n(CCC)nnn2)NCc2nc(C)n(C)n2)ccc2c(c1)OCC(=O)N2 20275,c1(C(=O)NC(CC)CN(C(=O)CSc2ccnn2C)CC)ccccc1C(C)C 20276,c1(C(N(CC(C)(C)NC(CCNC(=O)OCC)=O)C)=O)cc(C)c(Cl)cn1 20277,C(C(O)CS(C)(=O)=O)N(C=O)Cc1c(C)nn(Cc2ccccc2)c1 20278,CCCCC(CC(=O)N1CCCCCCC1)NC(=O)CN1CCCC1 20279,Cc1cccc(C(N2CCC(F)CC2C(=O)NCCN2CCCC2)=O)c1O 20280,N(C1CCC(NC(=O)Cc2ccccc2O)c2ccccc21)C(=O)C=CCF 20281,c1(OCC(=O)NCC2C(NC(c3sc(CC)c(C)c3)=O)CCC2)cccc(Cl)c1C 20282,Cc1nc[nH]c1CC(=O)N(CC(C)O)CCNC(=O)C(O)C1CCC1 20283,CON=CC(=O)NCc1cc(C(=O)NCCCC(C)O)co1 20284,C(CNC(=O)Cn1nccc1C(F)F)(CCCC)NC(CCCNC(C)=O)=O 20285,C12(CNC(c3c(C)cc[nH]3)=O)CCCC1CN(C(=O)CN(c1ccccc1)C)C2 20286,C#CC1(C(=O)NC(CC)CCCCC)CCN(C(C2C3CCC(C3)C2C)=O)CC1 20287,C1(NC(c2c(C)coc2C2CC2)=O)CC(F)CN(C(C2CCCOC2)=O)C1 20288,Cc1nc2nccc(NC(C3C(NCc4ccccc4)CC(F)(F)C3)=O)n2n1 20289,Cc1[nH]c(=N)sc1C(=O)NCC1CCC(F)(CNC(c2ncccc2Cl)=O)C1 20290,C1(NC(c2c(-c3cc(C)on3)ocn2)=O)COC2(CCN(C(=O)CCF)C2)C1 20291,C1(c2cn(C(C(=O)OC)C)nn2)CN(C(c2ccc(C(C)(C)C)[nH]2)=O)CCN1 20292,c1(C(=O)NC2C(CO)CCN(C(c3c(C#N)ccs3)=O)C2)cc(S(C)(=O)=O)co1 20293,Cc1cccc2c1CC(C(=O)NCC1(C)CCCN1C(C13CC(F)(C1)C3)=O)O2 20294,N1(C(Cc2cc(C)[nH]n2)=O)CCCCC12CC(NC(=O)CC(C)CF)C2 20295,CCC(CC)CC(=O)NCC(C)(CC(C)C)NC(=O)CC1(O)CCCC1 20296,N1(C(c2c(CNC(c3c(C)[nH]c(C)c3C)=O)n[nH]c2)=O)CC2(C1)NC(=O)NC2=O 20297,N1(C(CC(C=C)CC)=O)CC2(C(=O)NOCCC(F)(F)F)CC1CCO2 20298,CC1(CNC(C2CCCC(F)C2)=O)CCN(C(=O)CCC(=O)NC2CCCC2)C1 20299,Cc1cc(C(=O)NCC2CN(C(=O)CN3CCCS3(=O)=O)C2)ccc1Cl 20300,N1(C(c2n(C)ccc2)=O)CC2(CCCC(CNC(=O)C(F)CC3CCCC3)O2)C1 20301,C=CCCC(C(=O)NCC1(C)CCCO1)NC(c1ccccc1Cl)=O 20302,c1(CC)ccc(C(=O)NC2(CNC(=O)CC3CC34CC4)CCCC2)cn1 20303,C1(NC(C(c2cn(C)nc2)NC(C2CC(F)(CF)C2)=O)=O)CCC(F)(F)C1 20304,CS(C)(=O)=NC(=O)C(=O)NCC(F)CNC(C1CCOC1)=O 20305,C1(CCNC(c2cnn(CC3CC3)c2)=O)CC(F)(F)CN1C(=O)Cc1ccno1 20306,N1(C(c2c(N)ccc(C)c2)=O)CC(NC(=O)CC2OCCCO2)C2CCCCC12 20307,CCCCC(=O)N(C1CCN(C(C2(c3ccnn3C)CC2)=O)C1)C 20308,c1(C(=O)NCCC(C)NC(C2CC(C(C)C)C2)=O)ccc2cc(O)ccc2c1 20309,CC(C)C(O)(C(=O)OCC1C(CNC(=O)OC(C)(C)C)C1(F)F)C(F)(F)F 20310,C(C(C(C)C(C)C)NC(=O)Cc1ccc(C)cc1)NC(c1ccc(CCC)[nH]1)=O 20311,CC1(Cn2cc(CSCC(F)(F)F)nn2)CCCCC1(F)F 20312,C#Cc1ccc(C(N2CCC(C(=O)NCC(O)COC)(CC)C2)=O)o1 20313,N1(C(c2cc(F)cc(Br)c2)C(=O)NC)CCC2CCCCC12 20314,c1(C(N(CCNC(C2(C)CC=C(C)CC2)=O)C)=O)cc(Cl)c(F)cc1Cl 20315,c1(-c2n(CC)c(N(CC(C)C(=O)NC)C)nn2)ccc(S(C)(=O)=O)cc1 20316,C(=O)(C#Cc1ccccc1)NCC1CC(C(=O)NC2CCN(C(C)=O)CC2)C1 20317,c1(C(C)C)ccccc1C(=O)NC1CC1CNC(=O)C=C1CC1 20318,C1(NC(C(CSC)(C)NC(=O)Cn2cnnc2)=O)CCN(OC)CC1 20319,N1(C(CC(C)SC)=O)CCCC(C(=O)NCC2(n3ccnn3)CC2)C1 20320,N1(C(CN(C2CC2)CC)=O)CC2CC(C(=O)NCc3cnc(C)cc3C)(C2)C1 20321,CN=c1nc(N2CCC(C)(CO)C2)[nH]c(=NCC2(c3cnn(C)c3)CC2)[nH]1 20322,c1(C(N2CC(C)C(CCNC(=O)CCS(C)=O)C2)=O)cc(F)c(F)c(C#N)c1 20323,c1(C(N2C(C(=O)Nc3ccc(Cl)cc3)CC(C)C2)=O)c(F)cc(Cl)cc1Br 20324,C1(CNC(C=CC(=O)OCC)=O)CC2CCC1N(C(=O)C(C)C1CCOC1)C2 20325,C(=O)(CC1=CCN(C)CC1)NC1CC2CN(C(c3c(NC)cccc3)=O)C(C1)C2 20326,n1(CC)cnc2c(NC(C)(C)CF)nc(N3CCC(CC(C)C)C3)nc12 20327,C1(NC(c2cc(COC)[nH]n2)=O)CCCCC1CNC(=O)Cc1ccns1 20328,CN1CC(CC(=O)NCCOCCNC(=O)CC=C(Cl)Cl)C(O)C1 20329,c1(C(N2CCC(N(C)C(C3(C)CCCC3)=O)C2)=O)cc(F)c2cn[nH]c2c1 20330,N1(C(Cc2cc(C)nn2C)=O)CCCC(C)(C(=O)Nc2cccnc2C)C1 20331,C1(CCCC)CCCN1C(=O)C(C1CCC1)NC(=O)C=CCC1CCCC1 20332,c1(CC)cc(N2CCCC(NC(C3CCC(=O)N(C)C3)=O)C2C)nc(CC)n1 20333,CCC(CC(=O)N1CC(C2CC2C(=O)N(CC(C)C)C)C1)C(C)(C)C 20334,C1(NC(C(C)OCC)=O)CCCCN(C(C2(C)CCN(C)CC2)=O)CC1 20335,C(=O)(C1CCCc2nc[nH]c21)N1CCC(NC(=O)C=Cc2ccsc2)C12CC2 20336,Cc1nc(NC2CCN(CCNC(C3CCS(=O)(=O)N3)=O)CC2)ncc1Br 20337,CCCCCCCCCCCC(=O)N(CC(C)NC(C1(OC)CCSC1)=O)C 20338,C1(NC(c2cc(CC)c(OC)cc2)=O)C2CC(CN(C(C3CC3F)=O)C2)C1CO 20339,Cc1cccc2c(CC(=O)NC3COCC3NC(C3CC4(CCC4)C3)=O)c[nH]c12 20340,C1(CN=[N+]=[N-])CCCN1C(C1C=CCN1C(=O)CC1OCCCO1)=O 20341,C1(CC)(CC)CCN(C(=O)CCCNC(C2CC(n3cncn3)C2)=O)CC1 20342,C(CC1=CCN(C(C2CC(=O)OC2(C)C)=O)CC1)NC(CC(C)CN(C)C)=O 20343,C1(CC(=O)NC(c2nc(C)cs2)CC)CN(Cc2ccc(C(=O)O)s2)CCO1 20344,Cc1cc(CCNC(C23CC2CCN3C(=O)CCc2ncccn2)=O)nn1C 20345,N1(C(C(CC)C#N)=O)CC2CCOC2(C(=O)OC)C1 20346,C1(CCC)CCN(C(=NCc2cc(Cl)ccc2OC)NC2CC2C)CC1 20347,C1(C(=O)NCCOCCC)CC12CCN(C(=O)CCC(C)(C)F)C2 20348,Cc1ccc(C(F)(F)C(=O)NC2CCC(NC(C3CC(=O)N(O)C3)=O)CC2)cc1 20349,c1(C(N2CCOC(C)(C)CC2)C(=O)NC)cc(Br)c(OC)nc1C 20350,C=CCCCC(C(=O)N1CC(=O)N(C)C(=O)C1)NC(c1nc(C)ccc1C)=O 20351,O=C1NCCCCC1NCC(C1CCCCC1)C1CCC1c1ccc(F)cc1 20352,N1(C(C(CC)C)=O)CCC(O)(CN(C(=O)CCc2nc[nH]n2)C)C1 20353,Cc1cc(C2C(C(=O)O)CCC3C(C2)C3C#N)ncc1S(=O)(=O)N1CCCSC1 20354,O=C(CC1=CSC2=NCCN12)NCC1CCCCN(C(=O)C(F)OC(F)(F)F)C1 20355,c1(OC)ccc(C(N2CC(O)(C(C)NC(=O)C(O)Cn3cncn3)C2)=O)o1 20356,CCC(C(=O)N1CC2CC1(C(=O)NCCC1(COC)CCC1)C2)C(F)(F)F 20357,c1(CC)occ(C)c1C(=O)NCC1CCCC(NC(C2(CC)CC2)=O)C1 20358,c1(C(N(CCCNC(C2CC2Cl)=O)CC2CCCC2)=O)sc(F)cc1Cl 20359,CN1CCN(C(=O)Cc2n[nH]c(=N)s2)CC1CNC(C1CCCCC1CO)=O 20360,C(CC(=O)N1CCC(OC)C(C)(C)C1)(C(F)(F)F)NC(c1ccc(OC)cc1)=O 20361,C1(NC(c2c(C)n[nH]c2)=O)C2CCN(C(=O)C=CC(=O)NC3CC3)CC12 20362,Cc1ccnc(C(=O)NCC2(F)CC(NC(=O)C(O)Cc3ccc(F)cc3)C2)c1 20363,Cc1cccc(CC(=O)NCCC2CCCCN2C(=O)Cc2cccnc2)c1 20364,c1(C(CNC(c2ccc(C)cc2)Cc2ccccn2)=O)ccc(F)c(C)c1Cl 20365,N1(C(C2(CC=C)CC2)=O)CC2(CO)CC1(C(N1CCOC(C3CC3)C1)=O)C2 20366,CC1CN(C(C2(CO)CCCC2)=O)CC(C)C1NC(c1cc(C2CC2)cs1)=O 20367,N1(C(c2n(CC)ncc2)=O)CC2CCC(NC(=O)CC3CC(C)(C)CO3)CC2C1 20368,c1(C(=O)NC2CCN(C(=O)Cn3ncnn3)C(C3CC3)C2)noc2c1CCCC2 20369,C1(C#N)(C(=O)NCC(CC)NC(=O)CCc2c(Cl)cncc2Cl)CCCOC1 20370,c12ncc(Br)cc1C(=O)N1CCC2CC1.C1(COC)CCCN(c2nccs2)C1 20371,c1(C(N2CC3(OCC(NC(c4ccco4)=O)C3)C2)=O)c(F)ccc2occc12 20372,C1(NC(C(CNC(C)=O)(C)C)=O)CCN(C(=O)CC2(S(C)(=O)=O)CCC2)CC1C 20373,S(=O)(=O)(C1CC1)NCCNC(=O)NC1CC(CCC(=O)OC)C1 20374,C1(C(=O)NC2CCCC(C(N(CCCC(C)C)CCO)=O)C2)CC2(C1)CC(O)C2 20375,C1(C(N(CCCC(=O)NC)C)=O)C(C2CC2)CCN1C(C1CCCC1)=O 20376,C1(CNC(CS(C)(=O)=O)=O)CC2(CCN(C(c3cccc(C#N)c3F)=O)CC2)C1 20377,C1(C(=O)NC2CCN(C(C)=O)C2)CC(N=[N+]=[N-])CN1C(=O)Cc1cn[nH]c1 20378,C1(NC(c2cc(F)cs2)=O)CN(C(c2cnc3ccnn3c2)=O)C2(CCOC2)C1 20379,c1(C(=O)Nc2cn(C)c(C(N3CC4CC4C3)=O)n2)ccc(F)c(F)c1[N+](=O)[O-] 20380,N1(C(c2c(CC)nccc2)=O)CCC2(C1)CN(C(c1cc(Br)c(F)cc1C)=O)C2 20381,N#Cc1ccc(CN2CCC3(CN(C(c4cnc(O)[nH]4)=O)C3)C2)c(F)c1 20382,CC(CN(C)C)CCC(=O)NCC(O)CNC(C12CCC(CC1O)C2)=O 20383,c1(C(=O)NCCN(C(c2nccc(OC)c2F)=O)CC)cnn2c1CCC2 20384,C#CCCCC(C)C(=O)NCc1ccc(CNC(=O)C(C)(C)OC(F)(F)F)cc1 20385,c1(C(N2CC(OCCC(=O)NC(CCC)CC)C2)=O)cc2occc2[nH]1 20386,N1(C(CN2CC(C)C2)=O)CCOC2(CCN(C(=O)C3=CCCCCC3)C2)C1 20387,c1(OCC)cnc(C(=O)NC2CCC2NC(c2ccon2)=O)cn1 20388,C#Cc1ccc(C(=O)NC2CCCCN(C(c3scnc3CC)=O)C2)cn1 20389,c1(C(=O)Sc2ccccc2-c2cn(C3CCOC3)nn2)cc2cc[nH]c(=O)c2s1 20390,CC1C(NC(=O)C(C)NC(N)=O)CCCN1C(C1CC12CCCC2)=O 20391,C1(NC(c2scc(CNC(C(C(CC)C)N(C)C)=O)c2)=O)CCN(C)CC1(C)C 20392,c1(C2(C(=O)NC(c3ccccc3)CNC(CC(C)F)=O)CC2)cccnc1Cl 20393,N(C1CCCc2cccc(C)c21)Cc1cc(C)cc(Cl)c1 20394,N1(CC(C)C)CC(C(N2CC(CNC)C2)=O)CC1=O 20395,N12CCCC(C1)N(CCF)C(=O)C2=O.C12(C(=O)NCCOC)CC(C1)C(C)O2 20396,c1(CN(C)C(C2CCN(C(c3ccc(F)cc3Cl)=O)C2)=O)ccc(C#N)cc1 20397,C=CCC(C)(C)CC(=O)NCc1ccccc1CNC(C1NC(=O)CC1C)=O 20398,N1(C(C2C(=C)C2C(=O)OC)=O)CCC(COCC(=O)OC)C(O)C1 20399,O=C(N=c1nc(-c2ccsc2)[nH]s1)c1cncc(OC2CCOCC2)c1 20400,C1(CC(N2CC(O)(CNC(=O)C(c3ccc(F)cc3)(F)F)C2)=O)CCCC12CC2 20401,C12(NC(c3cccc4nonc34)=O)CCCN(C(C3CC(F)(F)C3)=O)CC1C2 20402,Cc1cc(C(N2CCC(CCNC(c3csc(Cl)n3)=O)CC2C)=O)nc(C)n1 20403,N1(C(CC2CC(C)(C)C2)=O)CC2(CC(NC(C3(C)CNC(=O)C3)=O)CO2)C1 20404,Cc1cc(F)c(N(CC(=O)NC(CC2CC2(F)F)C(=O)OC(C)(C)C)C)nc1Br 20405,c1(OC)cc(Br)c(CN2CCCC2CCC(=O)Nc2ccnc(F)c2F)cc1O 20406,c1(CC)[nH]ccc1C(=O)NC.C12CCCN1C2=O.C12CCC1C(=O)NCC2 20407,Cc1ccc(N2CCNC2=O)cc1NC(c1cn(CC(C)N)nn1)=O 20408,C1(NC(c2scc(C)n2)=O)CCN(C(=O)Cn2c(C)ccc2C)CC1F 20409,c12nc(c(C)s1)N(CCNC(c1ccccc1Cl)=O)CCNC2=O.CO 20410,CC(C)CCC(C(=O)NCC(=O)NCCO)NC(=O)CC(O)CN(C)C 20411,N1(C(C2(C(C)C)CCCN2C(C2CC2C#N)=O)=O)CC(C)(C2CCC2)C1 20412,c1(N2C(C(C)(C)NC(Cc3n(C)ncc3)=O)CCC2)cc(C2CC2)ncn1 20413,C1(O)(CN(C)C(c2ccc(C(C)(F)F)cc2)=O)CCN(C(C2CC2F)=O)C1 20414,N1(C(c2c(=N)cc[nH]c2)=O)C2CCC1CN(C(=O)CC1CC(=O)NC1=O)C2 20415,c1(COC)cccc(NC(c2nc(C(C)NC(c3nn[nH]n3)C3CC3)sc2)=O)c1 20416,N1(C(C=C(CCC)C)=O)CC(NC(c2ccc(O)cc2)=O)CC1(C)C 20417,C1(NC(C(C)c2cccs2)=O)CN(C(c2cncn2C2CC2)=O)CC1C1CC1 20418,c1(OC)ccc(-n2nnc(C(=O)Nc3cnnn3C(C)C)c2C)cc1 20419,c1(C(=O)NC2(C)CCCN(c3cnc(C#N)cn3)C2)cc2n(n1)CC1(CC1)C2 20420,c1(C(c2nnnn2C)Nc2ccc(OCCC)cc2C)ccc2c(c1)CCC2 20421,C1(C(N(C2CCN(C(CNC(N)=O)=O)CC2)CCO)=O)CCCC2(CCOC2)O1 20422,CCCC(O)C(=O)NCCCN(C(=O)C(CCSC)OC)C1CC1 20423,C1(N(C(=O)CCCc2sccc2C)CC)CCCN(C(C2CCCCC2)=O)C1 20424,C#Cc1cccc(CNC(C2CCCCN(C(=O)CC3CCCC(C)O3)C2)=O)c1 20425,C1(NC(C(CC)C(C)C)=O)CC2(CCCN(C(=O)COCCN(C)C)CC2)C1 20426,N1(C(c2n(CC)ccn2)=O)C2CCC1CC(C(=O)Nc1cnn(CC(N)=O)c1)C2 20427,c1(C(=O)NC(C(=O)NCCOC)C2CCCO2)cnc(O)c(F)c1 20428,O=C1CC(C(=O)N2CCCOCC23CCC3)c2ccccc21 20429,C1(CC)CCN(C(=O)Cc2cc[nH]c2)C(C(=O)N(C)CC2CCCC2(C)C)C1 20430,c1(C(=O)NC2CC(NC(CCc3onc(C)n3)=O)C2)ccc2c(c1)COC(=O)N2 20431,c1(CC(=O)NCC(COC)N)cc(F)ccc1C(=O)OC 20432,c1(OCC(=O)NCC(C)CNC(=O)Cc2ccon2)ccc(C#N)cc1Cl 20433,C1(CC(=O)NCCCN(C(C=CC(CC)C)=O)C)CC(O)C1(C)C 20434,NS(=O)(=O)CCC(=O)NCCC1CCN(C(=O)CN2CCN(C3CC3)C2=O)CC1 20435,CCCC(CC(C)C)C(=O)NC1CCN(CCCNC(=O)C#CC(C)C)C1 20436,c1(C(N2CCCC2Cc2cccc(Cl)c2)C(=O)NC)ccccc1OC 20437,N1(C(C23CC(C(=O)OC)(C2)C3)=O)C2CCC1CC(NC(c1cc3occc3s1)=O)C2 20438,N1(C(C2(CNC(C(C)N3CCCC3)=O)CC=CC2)=O)CCCNC(=O)C1 20439,c1(C(=O)NC(C2CN(C(=O)CCC3OCCO3)CCO2)C)ccc(C(F)F)cn1 20440,C=C=C(C)CC(=O)NCC(CC1CC1)C(=O)N1CCC1CF 20441,c1(C(N2CC(CNC(c3c(CC)n[nH]c3)=O)OCCC2)=O)scc2c1CCCC2 20442,c1(N(C(C(=O)OC)=O)C)cc(C)c(CCCN(CCN2CCNC(=O)C2)C)cc1F 20443,N1(C(CC(C)F)=O)CCCCC12CN(C(=O)C(=O)NCCOC(C)(C)C)C2 20444,C1(C(=O)NCC2CC(O)(CNC(C=C(CCC)C)=O)C2)CCCC(C)(C)O1 20445,C(=O)(C1=CCc2ccccc21)NC(C)CN(C)C(c1sccc1S(C)(=O)=O)=O 20446,C1(NC(CSc2ccc(OC)cc2)=O)CCN(C(=O)CCCCCBr)CC1F 20447,c1(C(=O)NC2CC3CN(C(c4scc(COC)c4)=O)CC32)cncc2nc[nH]c12 20448,Nc1cc(C(=O)NCC(CO)NC(=O)COCCCF)c(F)c(F)c1F 20449,C1(NC(C2(C)CCN(C)C2)=O)CC2CC(NC(c3occc3C3CC3)=O)C2C1 20450,c1(C(=O)NCC2(O)CCCN(C(C(C(C)O)(C)C)=O)C2)cccn2nccc12 20451,C(c1ccc2c(c1)OCO2)=CC(=O)NC1(CNC(C(CCCC)C)=O)CCOC1 20452,C1(OC)CC(CC(N2CC(N(C(=O)CCN3CCC(C)CC3)C)C2)=O)C1(C)C 20453,CC(C)=C=CC(=O)NCc1cnn(C)c1C(=O)NCCc1ccnc(O)c1 20454,c1(CCNC(C2(COCC)CCOCC2)=O)ccc(OC)c(Cl)c1OC 20455,c1(OC)c(C(=O)NCCC2CN(C(C3CCCC(F)C3)=O)C2)c(C)nn1C 20456,C12(NC(C(CC)N3CCCC3=O)=O)COC(CNc3ncc(F)cn3)(C1)C2 20457,c1(C(N2C3C(NC(C4C(CC)C4)=O)C(C3)C2)=O)ccc(S(=O)(=O)CC(N)=O)cc1 20458,c1(C(=O)NCC(C(C)C)NC(Cn2c(C)nnn2)=O)ccc(N=S(C)(C)=O)s1 20459,C(CN=[N+]=[N-])(C(=O)Nn1cncn1)NC(CCC1C(C)(C)C1)=O 20460,C1(CCC(=O)NC(c2cncnc2)C)CCN(C(=O)CN(C2CCC2)C)C1(C)C 20461,C1(CNC(=O)C=Cc2cc[nH]c2)CC2CCC1N2C(C1(CO)CCOCC1)=O 20462,FC1(F)Oc2cccc(CN3CCOC(c4cc(F)ccc4F)C3)c2O1 20463,c1(C(N(C2CCN(C(CCCC#C)=O)CC2C)C)=O)ccc2cccnc2c1 20464,c1(C(=O)NCC2(O)CCCN(C(c3c(C)cnnc3)=O)C2)cc2ncccc2o1 20465,Cc1c([N+](=O)[O-])c(C(=O)NCC(n2cccn2)C)nn1C 20466,CCCC(C(O)C(=O)N1CCOC(C)(C)CC1)NC(c1ccc(CO)cc1)=O 20467,C(C)(CO)(C(=O)NC1CCOC(C(=O)NCC(C)CC2CCCC2)C1)OC 20468,c1(C(=O)NC2CN(S(C(C)C)(=O)=O)CC2C#N)ccc(C#N)c(F)c1F 20469,CCCC(O)C(=O)N1CCC(OC2CN(C(C3COCCN3C)=O)C2)CC1 20470,C12(C(=O)NC3(C)CCCCC3)CC(CO)(CN1C(C1(C#N)CC3CC3C1)=O)C2 20471,C1(C(=O)NCC2CC(F)(CNC(=O)C(O)CSC)C2)(OC)CCOCC1 20472,c1(C(=O)NC(CCN(C(Cc2ncc(CC)[nH]2)=O)CC)C)scc(C)c1Cl 20473,CN1C(=O)CN(CC(=O)NCCCNC(=O)CCc2cc(Cl)no2)C1=O 20474,N1(Cc2nnc(C)o2)CC2CC2(NC(=O)CC2CCC(C(F)(F)F)O2)C1 20475,N1(C(C(C=C)O)=O)CC(CNC(c2cnn(CC(C)C)c2C2CC2)=O)C(O)C1 20476,n1(CCCC(=O)NC2CC(F)(CNC(COCCC#C)=O)C2)c(C)csc1=O 20477,N1(C(c2nnc(C(C)(C)C)s2)=O)CC2(CCN(C(=O)C=CI)CC2)C1 20478,C(CC(=O)NCC1CC(O)C(O)C1)(C(F)F)NC(c1n(CC)nc(C)c1)=O 20479,n1(CCCC(=O)N(CCCNC(=O)CO)CC2CCCC2)cnc2ccccc12 20480,Cc1c2ncnc1N1CCCC(C1)N2C.c1(NC(C)C)cc(C(F)(F)F)n[nH]1 20481,N1(C(CC(C)SC)=O)CCC(C(N2CCC(c3nc[nH]n3)C2)=O)(CO)CC1 20482,CC1CC(C(N2CCC(C)(CNC(c3cnn(CCF)c3)=O)C2)=O)CCO1 20483,C1(NC(c2ccccc2C(F)(F)F)=O)CCN(C(c2nccs2)=O)CC1F 20484,N1(C(C2CN(CC)C(=O)C2)=O)CCCC2(C1)CN(C(=O)CC1CC(C)C1)CCO2 20485,c1(C(N2CC(c3cnc4ccc(F)cn34)C2)=O)ccc(=O)n2c1CCC2 20486,C1(OC)C(Nc2nccc(N3CC4CC3C4)n2)CC1(C)C 20487,C(=O)(C1=CC2(CCOC2)C1)N(C(C)CNC(Cc1nc(CC)sc1)=O)CC 20488,c12cn(C)nc1C(c1nnnn1C(C)(C)C)CCC2.CC(CCC1CC1)N 20489,CCC(C(=O)NCC(C)(C)CNC(C1CC12CC2)=O)n1ccnc1 20490,N1(C(c2c(OC)scc2)=O)CCC(NC(C2CCC3(CCC3)O2)=O)C2(CCC2)C1 20491,CC(C)CCCCC(=O)NC1CN(C(C2(c3ncccc3F)CCC2)=O)CC1O 20492,c1(SCC)ccoc1C.CCC(C)(c1nccs1)NCCCN 20493,C1(C(N2C(CN(C(C3CC(=C)C3)=O)C)COCC2)=O)OCCCC1(C)C 20494,C=C=C(C)C(=O)NC1CCCC1n1cc(C(C)(C)OC)nn1 20495,C(C(=O)NC(C1CCCN(C(=O)Cc2[nH]cnc2C)C1)C)(C(F)(F)F)OC(C)=O 20496,C1(C)(CNC(c2ccc(OCC)cc2)=O)CCC(O)CC1.C1C(=O)N1C1CC1 20497,N1(C(C2(CC#C)CC2)=O)CC(N(C(=O)CN2CCC(C(N)=O)CC2)C)C(F)C1 20498,Cc1cc(F)ccc1N1CCC(NC(=O)NC(c2ccns2)C)C1 20499,N1(C(C2=CC(C)C2)=O)CCC(CNC(c2cnc(Cl)s2)=O)C1(C)C 20500,C1(NC(=O)CSC(F)F)CCCC12CCN(C(=O)CNC(c1ccccc1)=O)C2 20501,CC1(C)CN(C(=O)C2=COCC2)CC1NC(C1C2CCCC12)=O 20502,N1(C(C(C(C)NC(CN(C(C)=O)C)=O)C)=O)CCC2(CC1)CC(CO)C2 20503,C=CCC(F)(F)C(=O)N1CCC(F)(CNC(C2(C)CC(F)C2)=O)CC1 20504,C(=O)(C(C)(F)C(F)(F)F)NC(CC)CN(C(c1cccc(C)c1N)=O)CC 20505,Cc1ccc(CN2CC3C(C2)N3C(=O)C(c2ccccc2)C)c(C)c1 20506,c1(C(N2CCC(COC)(NC(=O)C=Cc3ccncn3)C2)=O)ccc(Cl)cc1O 20507,CCC(CC(=O)NC(C(=O)N(C)Cc1ccco1)C1(O)CCC1)OC 20508,C1(CNC(C2CC2F)=O)COC2(COCCN(C(c3cnoc3C3CC3)=O)C2)C1 20509,c1(C(=O)NCC(CC=C)NC(=O)C=Cc2ncc(C)[nH]2)ccc(Br)cc1N 20510,C(=O)(C(O)CC(F)(F)F)NC(C(=O)N(CCOCC#C)C)CCSC 20511,c1(OCCC(=O)NCC(CO)NC(CC(C)N(C)C)=O)ccc(F)cc1 20512,C1(CC(=O)N(C(C(=O)N(C(CC)CC)CCO)C)C)CNC(=O)O1 20513,c1(CCNC(C(CC2CC2)NC(C(COC)C)=O)=O)ccccc1F 20514,c1(C(=O)NC(CN(C(c2cc(C(=O)OC)ccn2)=O)CC)C)cc2cccnn2n1 20515,C1(C(N(C2CCC(NC(C3(CO)CCCO3)=O)CC2)C)=O)C2CC3C(C2=O)C13 20516,C(C(C)(C)CS(=O)(=O)N1CC(n2ccnn2)C(C)C1)OC 20517,C1(NC(Cc2c(C)n[nH]c2C)=O)COC2(CCCN(C(=O)CCN3CCC3)C2)C1 20518,N1(C(C2CC(O)(CNC(C(CCN(C)C)O)=O)C2)=O)CC2CC=CCC2C1 20519,c1(NC(=O)NC(C)Cc2cccc(C#N)c2)ccc(C(C)C)c(Cl)c1Cl 20520,CC1CN(C(C2(CF)CCC2)=O)CC1CCNC(c1csc(-c2ccsc2)n1)=O 20521,C(=O)(C#CC1CCC1)NC(CCNC(c1cnc(SC)n1C)=O)C 20522,C12CC13CCN(CC3)C2=O.C12(NC(C(C=C)O)=O)C3C4C1C1C2C3C41C 20523,c1(C(N(CC(O)CNC(C2(F)CCOC2)=O)C)=O)ccc(OC2CC2)cc1 20524,c1(C(=O)OC)cc(C)c(C(=O)NCC2CCC2NC(=O)C(F)C(C)C)o1 20525,CCC(C)CC(CO)N=c1ccc(Br)c(S(=O)(=O)N2CCS(=O)(=O)C(C)(C)C2)[nH]1 20526,N1(C(c2sc3ccn(C)c3c2)=O)CCC2(CCN(C(c3cc(F)cs3)=O)C2)C1 20527,C1(CNC(C(COC)N(C)C)=O)CCC(NC(C2(C)CCCS2)=O)CC1 20528,C12(C)CCCN(C1)C2=O.C1(NC(COC)=O)CCN(C(=O)C(C)C)CC1 20529,CCCC(CCC)N(C(=O)CC1CN(C(=O)CCCC2CCCO2)C1)CC 20530,C12(C(=O)OC)CCC(C(=O)N(CCCNC(C34CCCCC3C4)=O)C)(C1)C2 20531,N1(C(C2C(CN(C)C)C2)=O)CCC(C)(NC(C2CC23CCOCC3)=O)CC1 20532,c1(C(=O)NCCOCCN(C(CC(CCC)C)=O)C)c(C)nc(CC)nc1C 20533,C1(CNC(C2(C)ON=C(C)C2)=O)CC2(CO1)CN(c1cc(O)nc(O)n1)C2 20534,CC1CN(C(C2(NC(c3ccc(Cl)s3)=O)CCSC2)=O)CC(C)(C)O1 20535,c1(C(=O)NC2CCC(CNC(CCCOC)=O)C2)sc(Cl)c(Cl)c1OC 20536,C1(NC(c2nc(C)oc2C)=O)CC(C)CN(C(C2(C)CCC2)=O)C1 20537,S(=O)(=O)(c1ccc(CC(=O)NCC2C(NC(C3CCN(C)C3C)=O)C2)s1)NC 20538,C1(CNC(=O)CCCc2ccsc2)CC2COCC2N1C(=O)CCCCCO 20539,C(=O)(CCC1=CCCCC1)NC1(CO)CCCN(C(CCN(CCC)C)=O)C1 20540,N1(C(=O)CN2CCCC2=O)CCCC2CN(c3cc4nncn4cn3)CC12 20541,C1(C(=O)NCc2cncc(OC)n2)(COC)C=CCN1C(C1CCC(=O)O1)=O 20542,C1(NC(C(c2ccccc2)C)=O)CCN(C(=O)C(C2CC(F)(F)C2)O)CC1F 20543,C1(CC(=O)NC2(CC#C)CCN(C(COCC#C)=O)CC2)COCC2(CCC2)O1 20544,C1(C(N2CC(CNC(COC)=O)C(C)C2)=O)CCCCC1C1CC1 20545,C1(C(=O)OC)CSCN1C(C1CC(C)(NC(=O)CC=C(C)C)C1)=O 20546,c1(CC)ccc(C(=O)NC2CCC2NC(c2cccnn2)=O)cc1CC 20547,c1(CNC2(c3nnnn3-c3ccccc3)CC(C)(C)C2)ccc(O)cc1Cl 20548,Cn1nc(O)cc1C(=O)NCc1ccccc1CNC(=O)C=C(C)C(F)F 20549,CCCCCCCC(=O)N1C2CCC(C2)C1CNC(c1ncccc1C(C)=O)=O 20550,C1(CCOC)(NC(=O)C(F)=CC2CC2)CCN(C(c2cnc(C)n2C)=O)C1 20551,c1(CSC)noc(CNC(=O)Cn2cc(CC(=O)Cn3cncn3)nn2)n1 20552,CCS(=O)(=O)CCCOc1ccc(C)cc1F 20553,C1(C(N2CC(C)C(NC(c3ccc(F)cc3Br)=O)C2)=O)CC(=O)NC(=O)N1 20554,O=C(CC1CC12CC2(F)F)Nn1cnnc1 20555,N1(C(C2(COC)CC2)=O)CC(CCNC(=O)C=Cc2ncc[nH]2)C(C)C1 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20609,CC(C)CCC(C)N(C(=O)CCOCCNC(=O)CC1CC2CCC1O2)C 20610,N1(C)C(C)CC1(C)N=NC(C(C)(C)C=O)CC 20611,CC(C)CC(CC(=O)N(C)CC1CCCCC1)NC(=O)CC(C)C(F)(F)F 20612,CC1CC(NC(=O)C=C2CCN(C)C2)CN(C(c2nccc(Cl)c2O)=O)C1 20613,N1(C(C(CC)SC)=O)CC2(CC)CC1(CNC(c1ccncc1OC(C)C)=O)C2 20614,C(CC(CC)C(=O)NCCCCC1CCN(C(C2CCOCC2)=O)CC1)=CC 20615,c1(C(N2C(C)CCC(CC(=O)NCCN(CC)CC)C2)=O)cc2ccncc2[nH]1 20616,CC1CN(C(c2snc(Cl)c2Cl)=O)CC2(CCN(C(=O)CCc3nccs3)C2)O1 20617,c1(C(CNC(=O)C(CC)SC)NC(c2c(CC)csc2)=O)ccc(C(C)C)cc1 20618,C1(NC(CN(CCOC)C(C2CCC(F)(F)C2)=O)=O)CCCC(F)C1 20619,C12(C(=O)NCCCN(C(c3nc(C(C)=O)sc3)=O)C(C)C)CCC(C1)C(C)O2 20620,c1(C(N2CC=CC(NC(c3cc(OC)ncc3)=O)C2)=O)ccc(C)c2c1CCC2 20621,c1(CCOC)nc(=NC2CN(C(=O)C(C)(C)CC3CC3)CC23CCC3)s[nH]1 20622,C1(CCCC)CN(C(c2ccc(OC(C)=O)s2)=O)CCN1C(C1CC2(CC2)C1)=O 20623,C1(NC(C(N2CCSCC2)C)=O)COCCN(C(=O)CCCc2ncco2)C1 20624,O=C(CS(=O)(=O)CCO)NC1CCN(C(=O)Cc2ccc3c(c2)CCC3)C1 20625,CCCC(C)C(=O)N(Cc1cccnc1)Cc1cccc(NC(C2CC2F)=O)c1 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20661,c1(C(N2C(C)CCC2C)C(=O)Nc2ccccc2-c2cnn(C)c2)ccc(Cl)cc1F 20662,C12(C(N3C(C)CC(CNC(c4c(C(C)C)noc4)=O)C3)=O)CCC(CC1)C2(C)C 20663,c1(NCc2ccc(CC)s2)[nH]c(=NC2CC(NC3CC3)C2)nc2c1ncn2C(C)C 20664,C(=O)(C(C#N)C(C)(C)C)N1C(C2(NC(c3c(C)ccc(CC)c3)=O)CC2)CCC1 20665,C(CCC1CC1)(CN=c1ccc2c([nH]1)CCC2)OC(F)F 20666,Cc1c(C(=O)NC2CC(N(C(=O)CCC3CCCC(O)C3)C)C2)nnn1C(C)C 20667,N1(C(C(C)S(N)(=O)=O)=O)CCCC(C2CN(C(C3(c4ccncc4)CC3)=O)C2)C1 20668,C(=O)(CC(C)C(C)(C)NC(c1sccc1F)=O)N(CCn1c(C)ncc1)C 20669,N1(C(CN2C(=O)CSC2)=O)CCCOC(CNC(=O)CC2CCCOCC2)C1 20670,CC1OC2CCC1(C(=O)NC1CCCC(CC(=O)NCC3NC(=O)NC3=O)C1)C2 20671,CC(C)CC(=O)NCC1CC1CNC(=O)C(N1CCNC1=O)C 20672,C1(OCCNC(c2c(C)ocn2)=O)CCN(C(c2ccc(C3CCCO3)[nH]2)=O)CC1 20673,c1(NC(C(n2cc(C=CC)nn2)C)=O)ccc2oc(N(C)C)nc2c1 20674,N1(C(C)C)CCCC(NC(=O)C(C)N(C(=O)C(C)(C)CF)C2CC2)C1 20675,Cn1nc2c(c1C(=O)NCC1(O)CN(C(c3cc(C4CC4)ccn3)=O)C1)CCC2 20676,N1(C(C(C(=O)OC)C)=O)CC2(CCC(C(=O)Nc3nc(C4CC4)cs3)O2)C1 20677,CC(C)CC(O)C(=O)NCC=C1CCN(C(C2(C#N)CCC2)=O)CC1 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20819,C1(CN(C(=O)CC2(O)CCCO2)CC)CCCCN1C(=O)C#CC1CC1 20820,CN1CCC(C(C)NCc2nncs2)C1 20821,N1(C(c2cscc2C)C(=O)NCC=C)CCCCC(CO)C1 20822,Nc1c(C(=O)NCC(C2CCCC2)NC(=O)C(c2ccccc2)F)cccc1F 20823,CCC(C#N)C(=O)N1CCC(O)(C(C)NC(C2CCC(C)CC2)=O)C1 20824,C1(C(=O)NC(C)CC2CN(C(C3CCC34CC4)=O)C2)(OC)CCCCCCC1 20825,N1(c2cncc(-c3cc(N)cc(F)c3)n2)CC(S(=O)(=O)C2CCOCC2)C1 20826,C1(OC)CN(C(=O)COC2CC(F)(F)C2)CC1NC(=O)C(CCSC)OC 20827,C(C)(C(C(=O)NC1CCCC(CNC(c2sccc2SC)=O)C1)N(C)C)OC 20828,CC#CCCC(=O)NC(C1CCCN(C(C2CN(C)C2)=O)C1)C 20829,C1(N(CC)CC2CCC(C)(c3cccc(Br)c3)CC2)CCCCC(O)CNCC1 20830,C1(C(N(C(C)C)CCNC(=O)CCCCc2cnn[nH]2)=O)CCCCN1N=O 20831,C(=O)(C1=CCC2(COC2)OC1)NCC1C(NC(c2c(C)nccn2)=O)CCC1 20832,C(=O)(C1CCc2cccnc21)N1CC(N(C)C(c2ccc(F)cc2C2CC2)=O)C1 20833,C1(C(=O)NCCC(=O)N(C2CCCCCC2)CC)CCCCC1OC 20834,C1(CCNC(c2cnc(C(C)C)o2)=O)CSCCN1C(c1cccn1C)=O 20835,Cc1cc(C(=O)NCCC2CCN(C(=O)C(c3cccnc3)C)CC2)nn1C 20836,Cc1ccc(C=CC(=O)NC(C2CCCN2C(=O)C(C)Cn2cccn2)C)cc1 20837,N1(C(=O)NC2CC(C)=C(C)CC2)CCc2c(ccc(C)c2Br)C1 20838,C12(C(=O)NC3C(NC(C4N(S(C)(=O)=O)CCCC4)=O)CC3)CCC(CC1)CO2 20839,C(=O)(C(=O)CCc1ccccc1)NCC1CN(C(C(N2CCCC(O)C2)C)=O)C1 20840,N1(C(CCOC(C)=O)=O)CC=CC(C(N2CCC(O)C2C(C)(C)C)=O)C1 20841,CC(CCC(=O)OC1CCC1)NC(=O)CCC(=O)NC1CC1 20842,N1(C(C(C)(C)CO)=O)CCC2(CCC2)C(NC(C2CC(F)(F)C2)=O)C1 20843,C1(C(N2CCC(N(CCC)C(C3CCC3CF)=O)C2)=O)OC(C)(C)OC1(C)C 20844,c1(N2C3CN(C(c4ccc(F)cn4)=O)C(CC3)C2)c(Br)cncc1[N+](=O)[O-] 20845,C1(C(=O)NC(C)C2CC2)CC2(CC2)CN1C(c1cccc(N2CCCC2=O)c1)=O 20846,c1(C(N2CCC(OCCNC(c3nc(CC)sc3)=O)C2)=O)oc(CC2CC2)nc1C 20847,c1(C(=O)NC2C(C)N(C(c3cccnc3N)=O)CC2)ccc2c(c1)COC2 20848,c1(CN2CCCC(F)(CO)C2)ccc([N+](=O)[O-])cc1Br 20849,C1(NC(CN(C)C)=O)CCCCC12CCN(C(=O)Cc1c[nH]nc1O)C2 20850,C1(NC(C2(CC(C)=O)CC2)=O)CN(C(=O)Cc2cn(C)cn2)C2(CCOCC2)C1 20851,c1(N2CCN(C(C(Cc3ccc(C)cc3)C)=O)CC2)ccc([N+](=O)[O-])s1 20852,C1(N(C(c2ccc(OC)cc2)C(=O)NC(C)(C)C)C)CCOC2(CCSCC2)C1 20853,C(=O)(C#CC1CCOCC1)N1C(CNC(C(C)OCCN(C)C)=O)CC(O)C1 20854,CCCCCS(=O)(=O)CC(=O)NC(C)C(CO)NC(=O)C(C)CC(C)(F)F 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20872,CC1(C)CN(C(=O)Cc2cccnc2Cl)C(CNC(C2(C)CC2C(F)(F)F)=O)CO1 20873,c1(CC)cc(C)c(C(=O)N(C2CCC(NC(c3cn(C)[nH]c3=N)=O)C2)C)o1 20874,c1(C(N2CCC(CC(N3CC(C)C(=O)CC3)=O)C2)=O)c(F)cccc1C#N 20875,CCCCCC(=O)N1CC(O)CC1C(=O)N(CC(C)(CO)CO)C 20876,c1(OC)ccc(N)c(C(N2CCC3(NC(=O)C(N)=O)CC3C2)=O)c1 20877,Cc1cc(F)cnc1-c1cn(C2CN(c3n[nH]c(O)n3)C2)nn1 20878,C(=O)(CC(C)CC(C)C)NCc1cccc(NC(c2c(OC)n(C)nc2C)=O)c1 20879,c1(C(C(=O)NC)N(CC(=O)OC)C2CC2)cncn1C(C)C 20880,c1(C(=O)NCC(CN(C(C2(OC)CCOC2)=O)C)(C)C)ccc(CO)cc1.C(N)=O 20881,C(C)(C(=O)NC(C1CCCC1)CNC(=O)CCOC1CC1)SCCCC 20882,O=C1CC(C(=O)NCCCCCC2CCN(C(=O)C(O)C(F)F)CC2)NC(=O)N1 20883,c1(C(=O)NCC(C2CC2)NC(C(CCC)(C)O)=O)cc2c(C)cccc2[nH]1 20884,C1(CC=C)(C(N2CCC(C(F)F)C2)=O)CCN(C(=O)CCOC2CCCC2)C1 20885,N1(C(C2CCCN(C(=O)C(O)C3CCC3)C2)=O)CCOCCC1C1CC1 20886,Cc1c(Cl)ccc(C(=O)NCCC2CCN(C(c3ccc(=O)oc3)=O)CC2)c1O 20887,C1(NC(CCOCCC)=O)CC(C)(C(=O)NCc2cc(C)[nH]n2)C1 20888,c1(C(=O)NC(C(C(=O)NCCCCN(C(C)C)C)C)C)cc(F)ccc1F 20889,C1(CNC(CCn2c(C)ccc2C)=O)CC2(CC(NC(C3CCNC3=O)=O)C2)C1 20890,Cn1cc(C(=O)N(C2CCCC(NC(=O)Cc3ccccc3)C2)C)c(O)nc1=O 20891,Cc1cc(C(=O)NC2CCC2CNC(=O)CNS(N)(=O)=O)cc(F)c1 20892,c1(C(N(C(CNC(c2nc(C(C)=O)sc2)=O)C)C)=O)ccc(CCO)cc1 20893,C1(NC(c2nc(OC)oc2)=O)CCCN(C(=O)Cc2c(N)nc(C)nc2O)CC1 20894,c1(C(N(CC(CC)NC(c2oc(C)nc2C(F)(F)F)=O)C)=O)cnc(O)cc1C 20895,c1(CC(=O)NCC(CC)NC(=O)CCCCN(C)C)nnc2n1CCOC2 20896,c1(C(C(=O)N(CC(CC)NC(=O)C=Cc2cscn2)C)(F)F)ccccc1C 20897,C(=O)(C(C)(C)C(C)O)NC(C1CCCCO1)C(N1C(C(=O)OC)CC1)=O 20898,C12(CNC(CCC#C)=O)CC(CN1C(=O)CC1CCCCC1)C2 20899,c1(CC)c(Cc2nnc(-c3cccc(C)c3Cl)o2)cccc1C1CCCC(=O)N1 20900,c1(OC)ncc(C)cc1C(N1CC(N(C(=O)CN2CCCC2C)C)C(O)C1)=O 20901,c1(CC(=O)NCCCNC(c2ccc(F)s2)=O)nsc2ccccc12 20902,c1(C(=O)NCC(CC)NC(C2(C)CC2Br)=O)ncc(C)cc1C(F)(F)F 20903,N1(C(CC)=O)CCC(C)C1CNC(=O)Cn1cnccc1=O 20904,c1(C(N(C2CN(C(C34CC(C(F)F)(CO3)C4)=O)C2)C)=O)cnccc1Cl 20905,N1(C(CCCC(C)C)=O)CCC2(CC1)CC2NC(=O)Cn1nnc2ccccc12 20906,C1(C(N2CCN(C(=O)CNC(=O)C(C)OC)CC2)=O)(NC(C)=O)CCC(C)CC1 20907,C(=O)(CCCCC1CC1)NCc1ccc(C(N2C(CC(N)=O)CC2)=O)s1 20908,N1(C(CCC#C)=O)CC2CN(C(c3ccc(C#N)c(F)c3)=O)CCC2(CO)C1 20909,n1(C(CC)CC)nc(CCN2CCC(C)CC2)nc1-c1cnc(C(F)(F)F)nc1 20910,CC1(C(=O)NC2CCC(NC(c3ccnc(O)c3)=O)C2)CC2CC2C1 20911,C(C(C)(C)CNC(C1(CCCC)CC1)=O)N(CCC=C)C(C12CCC1C2)=O 20912,C(c1cccc(F)c1F)=CC(=O)N(CC(CN(C(C(C)c1ncco1)=O)C)O)C 20913,c1(C(N2CCCN(C(C(C(C)O)(F)F)=O)CC2)=O)nccc2[nH]ccc12 20914,C(=O)(C1=C(C)C(C)(C)OC1=O)NCC12OCC(CC)(C1)C2.C12(CCC1)C(=O)NC2 20915,n1(CC(=O)N(CCNC(c2ccc(CC)cc2)=O)CC)cccc(C)c1=O 20916,C1(NC(c2nc(CC)sc2)=O)CCN(C(=O)C(C)OCC(C)C)C12CC2 20917,c1(CN2CC(CNC(C3CC3F)=O)OCC2)cnc(Cl)c(F)c1 20918,c12ccc(cn1)C(=O)NC2.C1(CC)OCCC1C(=O)NCCC(=O)NC1CC1 20919,c1(NC(c2c(C(C)C)cn(C(C)C)n2)=O)cccc([N+](=O)[O-])c1Cl 20920,C(CCCCCC(=O)N1CC(NC(c2c(C)ccnc2C)=O)CC(C)C1)SC 20921,CC1CN2CCN1CC2C(N1CCN(C(c2cc(O)cc(N)c2Cl)=O)C(C)C1)=O 20922,N1(C(C2CC2F)=O)CCC(NC(C2(c3ccc(F)cc3)CCC2)=O)CC1 20923,N1(C(Cc2c(C)occ2)=O)CCN(C(=O)CCN(C)CCO)C(CC(F)F)C1 20924,C(C)(CCC(=O)N1CCC(C)(CNC(c2cncc(CO)c2)=O)C1)SC 20925,C(=O)(CCCCC(F)(F)F)N1CCC(CNC(C2CCN(CC)C2)=O)C(F)(F)C1 20926,c1(OC)ccccc1-c1c[nH]cc1C(=O)NCC(C)CNC(=O)CC(C)O 20927,N1(C(C(CC=C)(C)C)=O)C2CCC1CC(NC(=O)C=Cc1nc(C)c(C)[nH]1)C2 20928,C1(NC(C(COC)C)=O)CC(C)N(C(=O)CCC(=O)c2ccc(OC)cc2)C1 20929,C(=O)(C(Cn1cccn1)NC(=O)CC(C)C)NC(C#C)(C)C 20930,Cc1cccc([N+](=O)[O-])c1NC(C)CCNC(C1(CF)CCC1)=O 20931,c1(C(=O)NC2C(NC(C(CC)=CC)=O)CCC2)c(C)ccc(C)c1N 20932,C=CC(C)(CCOC)C(=O)NCC1(CNC(=O)CCCC)CC12CCC2 20933,C(=O)(C(C)CCC(C)(C)C)N1CCCC(CCNC(C(C)C2CCC2)=O)C1 20934,c1(-c2cn(-c3ccc(CNC(COCCC)=O)cc3)nn2)ncc(F)cn1 20935,c1(C(N2C(C)(C(N3CCC(C)(F)C3)=O)CC2)=O)c(Cl)cncc1Cl 20936,c1(NCC2(O)CCN(C(Cc3cccc(C)c3F)=O)CC2)cc2nncn2cn1 20937,Cc1ccc(CCNC(=O)C(=O)NCc2n[nH]c3c2CCC3)c2ccccc12 20938,c1(N(C)C)ncc(C(N2CCCC(CCNC(=O)CC3(CO)CC3)C2)=O)cn1 20939,CC(C(=O)N1CCC(C)(CNC(=O)CCC(C)CN(C)C)CC1)C(F)(F)C(F)F 20940,C(C(C(=O)NCCCF)NC(c1cc(C(F)F)[nH]n1)=O)N(C)C 20941,N1(C(C(C(C(CC)C)O)C)=O)CCC2(CC1)CCN(C(C13CC(F)(C1)C3)=O)CC2 20942,C1(N(C(C(N2CCOCC2)C)=O)C)CCC(NC(=O)CC(C)(C)C)CC1 20943,C1(OCC)CCN(C(C2CC3CC3N2C(=O)CCN(C)C)=O)CC1 20944,c1(-c2scc(C)n2)ccc(OCP(C)(C)=O)cc1.c1(C(NO)=O)ccccc1 20945,c1(OC)cc(C(N2CCC(F)(C(=O)Nc3cnc(C(C)(C)C)nc3)C2)=O)nn1C 20946,Cc1cc(CNC(=O)NCc2cnn(C(C)(C)C)c2)on1 20947,C1(CCC(=O)OCC)CCN(C(c2csc(C3CCCNC3)n2)=O)CC1 20948,c1(C(C)C(=O)NC2CN(C(=O)CN(C)CCO)CC2O)ccc(Br)cc1F 20949,N1(C(CC(C)(C)C2CC2)=O)CCC2(CCCCN(C(=O)CCC3CCCO3)C2)C1 20950,C1(C(=O)NCCCCNC(C2(C)CC(C#N)C2)=O)CCC2(CCOCC2)O1 20951,C1(C(=O)NCC2C(CNC(COCC=C)=O)C2)CCC(C(=O)OC)O1 20952,C1(C)(NC(CC2CC(C)C2)=O)CCN(C(=O)CC2CCNC(=O)C2)CC1 20953,C1(NC(C2(CC)COC2)=O)CCC2CN(C(c3cc(C)cnc3C)=O)CC2C1 20954,c1(NC(N(C)C)=O)ccccc1CSC1C(NC(=O)CCc2ccon2)C1 20955,C1(C(N2CC(CNC(C(n3cc(Cl)cn3)C)=O)C2)=O)CCCN(C(N)=O)C1 20956,CCCCCCCCC(=O)N1CCN(C)C(CNC(C2C3CCC(F)(F)C23)=O)C1 20957,C1(C(=O)NC2CC(C#C)C2)CC2C=CC1N(C(=O)C(C)(C)C(=O)N(C)C)C2 20958,Cc1cc(Cl)c2c(c1)CCN(c1nnc(C3COCCO3)n1CCC#N)C2 20959,C(=O)(CCC1CCc2ccccc21)N1CCC(CNC(CCCCC)=O)C1 20960,C(=O)(C1CC(=O)c2c(F)cccc21)N1C2CN(C(CC3(C=C)CC3)=O)C(CC2)C1 20961,c1(C(N2CC(C(C)NC(C3C(COC)C3)=O)C2)=O)nc(O)nc(O)c1F 20962,C(=O)(CC(C1CC1)NC(=O)CCCn1cnnn1)NCCC=CC=C 20963,C=C(C)CCC(=O)NC12CC(CNC(c3cncc(-n4cnnn4)c3)=O)(C1)C2 20964,CCC(C(=O)NCC1CN(C(c2cc(C(C)C)[nH]n2)=O)C(C)(C)C1)C(C)(F)F 20965,C(CC(C)C(F)(F)F)NC(c1n(CC(=C)C)nnn1)C(C)(C)C1CCCCO1 20966,C1(NC(=O)CC2CCC2)CN(C(c2[nH]ccc2C2CC2)=O)CC1CC1CC1 20967,c1(CCCC(=O)NC2(CS(C)(=O)=O)CC2)ccccc1.CN1CC1 20968,N1(C(=O)OC(C)(C)C)CCC(C(=O)NCC=CC=CBr)C1C1CC1 20969,N1(C(CCc2c(C)noc2)=O)CCC(C)(C)C1CNC(c1cc(F)cc(F)c1)=O 20970,c1(N2CCCCC(CC)C2)ccncc1S(=O)(=O)NC(c1ccnc(C)c1)CO 20971,c1(C2C(C(N3CCC(N(C(C(CC)SC)=O)CC)CC3)=O)C2)cc(F)ccc1C 20972,CC1CN(C(c2cccc(F)c2F)=O)CCN1C(c1ccncc1Br)=O 20973,CC1(C)CCC(O)(C(=O)NCC(O)CNC(C2CCC=CO2)=O)CC1 20974,N1(C(CCCC=C)=O)CCC2(CC1)CN(C(=O)CN(C1CCC1)C)C2 20975,c1(COC)ncc(C(=O)NC(C)(C)C(C)NC(C2C(C)C2C)=O)c(=N)[nH]1 20976,c1(C(=O)OC)nn(C)cc1C(=O)NCCC(O)CNC(c1ccc[nH]1)=O 20977,c1(C(N2CCC(C(CNC(C(C)NC(=O)NC)=O)(C)C)C2)=O)cn(CCF)nn1 20978,C1(CNC(C2CC(C(C)(C)C)C2)=O)CCCCCN1C(C1CC12CC2)=O 20979,c1(C(=O)NCCC(C)N(C)C(C2CC(O)C2)=O)c[nH]c2cc(Br)ccc12 20980,c1(N(C(C)CCNC(C2CCCC(O)C2)=O)C)snc(Cl)c1C#N 20981,Cc1nncc(C(N2CC3CCC3(CNC(c3cncc(N)n3)=O)C2)=O)c1C 20982,c1(C(=O)NCC(CN(C(C2CCC3CC23)=O)CC)(C)C)cn2ccnc2s1 20983,C(C)(C)(CCC(=O)N1CCCC(NC(c2nn(C)nc2Br)=O)C1)OC 20984,C#CC1(O)CC(C(N2CCCC(CCC(=O)NC(COC)CCOC)C2)=O)C1 20985,CCCCCC(C(=O)NC1CC1NC(=O)CN1CCCCC1=O)C(C)C 20986,c1(C(C(N2CC(C)C(NC(=O)C3=CCCC3C)C2)=O)=O)ccc(F)cc1F 20987,c1(C(=O)OC)ccc(F)c(-c2cnc(SC)s2)c1OC 20988,c1(CC(C(N2CC(NC(Cc3nc(C)[nH]n3)=O)(CO)C2)=O)C)ccccc1C 20989,c1(C(N(C)CC2(CNC(C3(O)CCOC3)=O)CC2)=O)ccc(C2=CCCC2)cc1 20990,C1(NC(c2c(CC)cno2)=O)CCC2(CC1)CN(c1nc(C3CC3)ns1)C2 20991,N1(C(C=C(CCC)C)=O)CC2(C1)CN(C(=O)C(CCC)NC(N)=O)CC(C)(C)O2 20992,c1(C(C(N2CC(CNC(C3(OC)CC3)=O)C(OC)C2)=O)(C)C)ccc(Cl)cc1F 20993,C(CCOCC)(C(=O)NCCSCCOC)NC(C(C=C)OC)=O 20994,c1(N2CCC(COC)(NC(C3CC(=O)NC3(C)C)=O)C2)nc(C2CC2)nc(=N)[nH]1 20995,C1(C(=O)NCC2(C)CCN(C(C(C(=O)OC)C)=O)CC2)CCn2ccnc2C1 20996,Cc1ccc2c(c1)c(CCNC(c1cc3c(cc1Br)NC(=O)CO3)=O)cn2C 20997,C(=O)(C1CCc2c[nH]nc21)N1CC(C(=O)Nc2c(O)ccc(CC(=O)OC)c2)C1 20998,C(CS(=O)(=O)c1ccc(COC)cc1)N(C(C(C=CCCC)O)=O)c1ccccc1 20999,C1(C(=O)NC(C)CCN(C)C)C=CC(NC(=O)CC(=O)OC)C1 21000,c1(NC(C2C(CCOC)C2)=O)cc(OCC(=O)OC)cc(O)c1 21001,FC1CCCCCC1N=c1[nH]c(=NCC2CC3(CCOCC3)CO2)[nH]c2c1SCC2 21002,N1(C(CN(C)CC)=O)CCC(C(C)C(N2CCCC2CC(CO)C(=O)OC)=O)C1 21003,C1(NC(CNC(C)=O)=O)C(C)CN1CCN(C)CC.C(C)(C)C 21004,C=CCN=C(NCc1cc(O)cc(O)c1)N1CCC2OCCCC2C1 21005,N1(C(C(CC)c2cccnc2)=O)CCC(NC(c2cc(SC)on2)=O)C1C1CC1 21006,CC1Cc2cc(CC(N3CCCC(CNC(C4COC4)=O)CC3)=O)ccc2O1 21007,C1(C(=O)NCC2(OC)CN(C(=O)C(C)N3CCCC3)C2)CC2(CCO1)CC2 21008,Cc1nn(C)c(C(=O)NC2CC23CC(NC(=O)C(C)(C)C(=O)N(C)C)C3)c1Br 21009,C1(NC(c2occ(C)c2)=O)CCCCC1NC(C1CCC(C(N)=O)O1)=O 21010,c1(NCc2ccc(CO)o2)ccc2nc(-c3cccc(OC(F)(F)F)c3)sc2c1 21011,C1(C(N(CC(CC)NC(c2c[nH]nc2-c2ccco2)=O)C)=O)C(C)C1(F)F 21012,N1(C(c2cc(C)n(C)c2)=O)CC2(CC(NC(c3cccc(F)c3O)=O)C2)C1 21013,CCCCC(O)CNC(C1CC(C)N1C(=O)Cn1cnnc1)=O 21014,CC1(C)CCCC1C1CCN(C(N2CCCC3CC(O)CCC23)=O)C1 21015,C1(CNC(=O)Cn2cncn2)CC(NC(=O)CNC(=O)C2CC2)C(O)C1 21016,c1(C(C)NCC2CCCC(C)O2)cc(Cl)ccc1F 21017,c1(OC)ccc(C(=O)NCC2CC(CNC(c3ncccn3)=O)C2)cn1 21018,C1(NC(C(CC)C)=O)CCCCN(C(c2cnc(C(F)(F)F)cn2)=O)C1 21019,CC1(F)CC(N=c2[nH]c(N3C4CCC3CNC(=O)C4)nc3c(F)cccc23)C1 21020,C(N=c1nc(N2CCC(C3CCC3)C2)c2ncccc2[nH]1)c1c(C)cn(C)n1 21021,C1(C(=O)NC2CC(CC)OCC2)CCN(C(c2cn(C)nn2)=O)C12CC2 21022,c1(OC)nc(N2CCCC2CNC(=O)C(F)(F)c2ccccc2)cc(C)n1 21023,CC1(C)NC(=O)CCC1NC(C1CNC(=O)CN1C(=O)C=C1CCC1)=O 21024,c1(NC2C(C)(C(=O)OCC)CCCC2)ccc(S(N)(=O)=O)cc1F 21025,c1(C(C)C)nc2ccccc2nc1SC1CCN(C)CC1 21026,c1(OC)cc(F)c(Cl)cc1C(N1CCC(NC(C2CN3CCN2C(C)C3)=O)C1)=O 21027,C1(C2CCN(C(=O)C3=CCCSC3)CC2)(NC(C2CCCN2C(=O)C2CC2)=O)CC1 21028,c1(OC)ccc(F)cc1NC(C1CC1C(=O)Nc1ccc(Br)c(F)c1)=O 21029,C#CCC1CC(=O)NCC(=O)CC(=O)N1.c1(C(=O)OC)cc(C(C)(C)C)ccn1 21030,c1(CCC(=O)NC2(C)CC(NC(Cn3c(C)cnc3)=O)C2)ccccc1N(C)C 21031,c1(OCC)cccc(C(=O)NC(C2CCN(C(=O)Cc3conc3C)CC2)C)c1 21032,c1(C(=O)NC2(COC)CN(C(=O)Cc3ccsc3C)C2)cnc2c[nH]nc2c1 21033,CC(CC(=O)N1CC(C)(C)CC1CNC(C1CCc2ncnn2C1)=O)C(F)(F)F 21034,Cn1cncc(C(=O)NCCOCCOCCNC(=O)C(C)(Cl)Cl)c1=O 21035,c1(C(N2CCC(F)(CNC(C3CCC3F)=O)CC2)=O)ccc2c(c1)CNC2=O 21036,N#Cc1ccc(C(N2CCCC(NC(=O)C=CC3CCOCC3)C2)=O)nc1 21037,N1(C(c2c(C)cn(C)n2)=O)CC(C(F)(F)F)OCC1CNC(c1csnc1C)=O 21038,C(CCCCCCCO)=CC(N1C(CCNC(CCCC#C)=O)CSCC1)=O 21039,N1(C(C2CCN(CC#C)CC2)=O)CC(O)C(O)C1CNC(=O)CCCCCO 21040,C1(NC(C(C)NC(C)=O)=O)CN(C(C2(c3ccc(F)cn3)CC2)=O)CCC1CO 21041,CCC(C)CC(=O)NC1CC(F)(CNC(=O)CCCCN(C)C)C1 21042,C(=O)(CC(O)C1CCCC1)NCCOCCN(C)C(c1csc(CC2CC2)n1)=O 21043,CC1CCC(F)(C(=O)NCC2(C)CCCN2C(c2ccc(CCF)cc2)=O)CC1 21044,Cc1cc(OC(=O)CN2CCCC2)ccc1N1CCCC1=O 21045,C=CCC(C)(C)CCNC(C1CCOC1CNC(=O)C(C)(C)CC1CC1)=O 21046,N1(C(c2c(CCC)nns2)=O)CCN(C(c2ccc(C(C)F)cc2)=O)CC1CC 21047,C(=O)(C1CCCn2cncc21)NCC(CNC(c1sc(C)c(O)n1)=O)(C)C 21048,C(=O)(C(O)CC(C)C)NCC1CCC(NC(CCSCCCC)=O)CC1 21049,S(=O)(=O)(c1cccc(N2CCCC(CCO)CC2)n1)NCC(CC)C(C)C 21050,C1(C(=O)NCC(N(C)C(C2CC(F)C2)=O)C2CC2)CCOC(C)(C)C1 21051,N1(C(C(C)(C)NC(N)=O)=O)CCN(C(=O)CCc2cnc[nH]2)C(CC(F)(F)F)C1 21052,C(=O)(C(C)(C)C(=O)NCC1COCC1NC(=O)C1=CCOCC1)N(C)C 21053,C1(C(N2CCC(C(CNC(=O)CCc3cn[nH]c3)F)CC2)=O)CCC(F)(F)CC1 21054,c1(NCC2CCCN(C(C3(CC#C)CCCCO3)=O)C2)cc(C)nc2ncnn12 21055,n1(C(C)C)ncnc1CNC(=O)C=CC(c1cnn(C)c1)=O 21056,N1(C(C2CN(S(CC)(=O)=O)C2)=O)CC2CCCC2(NC(=O)CCC2(C)CC2)C1 21057,CC1CCN(C(c2c(Cl)n[nH]c2C2CC2)=O)CC1N(C(=O)CCC1CC1(F)F)C 21058,CC(C)CCCC(=O)NC1(CF)CCN(C(c2coc3c2CSC3)=O)C1 21059,CC(C(=O)N1CC2(CC2)CC1CNC(=O)Cc1cnccc1Cl)C(C)(F)F 21060,C(=O)(C(C)(CC)C(=O)NS(CCCC(C(C)C)NCC(=O)OCC)(=O)=O)OCC 21061,C1(C(NOCCCN(C)C)=O)C=CCN(C(C2CCCO2)=O)C1 21062,C(=O)(CCCCCCS(N)(=O)=O)N1CCCC(CNC(C(C(C)C)OCC)=O)C1 21063,C1(C(N2CC(OC)C(C(N3CCC(N(C)C)C3C)=O)C2)=O)CCC2(CC1)CC2 21064,c1(N(C)C2CC2)ccc2nc(CC=O)[nH]c2n1.C1(NC)CC2CC1C1CCCC21 21065,C#CCC(O)C(=O)NCC1CCCCN1C(=O)CCCSCc1ccc(C)cc1 21066,S(C(F)(F)F)CC(=O)NC1CC(N(C(CNC(C)=O)=O)C)C1 21067,c12c(OC)cc(cc1OCC(F)F)OCC(C)(C)N2.C(=O)(COCC(F)F)OC 21068,N(C1CC(C)Sc2ccccc21)OC.c12nc3n(n1)CC(CC3)NC(=O)C(=O)N2 21069,C(CC(N)=O)(C(=O)NC1CC1NC(=O)CC1CC1)NC(CC(C)C)=O 21070,C1(O)(C(CNC(COCC(C)C)=O)C)CCN(C(=O)Cc2nc(=N)[nH][nH]2)C1 21071,c1(SC)ncccc1NC(=O)CC1CCN(C(c2[nH]c(C)nc2C)=O)C1 21072,C1(C(=O)NCCCC)CCCN(C(c2cn(CC)nn2)=O)C1CC 21073,C1(CNC(C=COCC)=O)CN(C(=O)C(C)CN(C)C(=O)OC(C)(C)C)CCO1 21074,c1(C(N2CC(C#N)(CF)C2)=O)nc2ccccc2s1.C12CCN1C2 21075,N1(C(CC2CCC(C)C2)=O)CC2CC(N(C(=O)CSC(F)(F)F)C3CC3)(C2)C1 21076,c1(C(CC(=O)N(CCNC(c2cn(CC)nn2)=O)C2CC2)C)ccc(F)cc1F 21077,C1(C(N)=O)CN(C(c2coc(C(F)F)n2)=O)CCC1NC(C1(C)CCC(=O)C1)=O 21078,c1(C(=O)NC2CCCC2NC(C2(F)CCS(=O)(=O)C2)=O)cc2n(n1)CCCN2 21079,Cn1nc(CNC(C23CC2CCN3C(=O)NC2CCCC2)=O)c2c1CCC2 21080,c1(C(C)NCC(COCC)C)cc(C(=O)OC)c2n1CCOC2 21081,N1(C(CCSCC)=O)CCC(C2CCC2)(CNC(c2cc(=O)n(C)o2)=O)CC1 21082,CC(C)C(C(=O)N(C)CC1CCN(C(=O)CC(C)O)C1)c1ccc(Cl)cc1 21083,CN1CCCC(O)(CC(=O)NC2CC(CO)N(C(c3cc(Cl)ncc3O)=O)C2)C1 21084,c1(CC(=O)N(C2CC(NC(C3COC(=O)N3C)=O)C2)C)ncncc1Cl 21085,Cc1ccc(F)cc1CC(=O)NC(C)CCCC(=O)N1CC(CO)CC(C)C1 21086,CC(C)C(C(=O)NCCNC(C1(Cc2cccc(Cl)c2)CC1)=O)c1ccn(C)n1 21087,CC(C)CC(O)C(=O)NC1CCN(C(=O)CN2CCN(C)CC2)C1C(C)(C)C 21088,C1(CNC(C2OCC(C)C2)=O)CC2COCC2N1C(c1c[nH]cc(F)c1=O)=O 21089,N1(C(C)=O)CCC(NC(=O)C(C(C)C)NC(C2CC(=O)C2)=O)CC1 21090,C1(NC(C(C)NS(C)(=O)=O)=O)C=CCN(C(c2cc(-c3ccoc3)on2)=O)C1 21091,N1(C(C(CC#C)O)=O)CCn2nc(CNC(C3(O)CCCC(C)(C)C3)=O)cc2C1 21092,C1(C(=O)NC(C2CCCCC2)C2CCC2)CNC2(CCC2)CO1 21093,N1(C(C2CCN(C(C)=O)CC2)=O)CC(C)CN(C(=O)COc2ccsn2)CC1C 21094,Cn1c(C(=O)NC2CCCN(C(c3ccc(S(C)(=O)=O)s3)=O)C2)ccc1[N+](=O)[O-] 21095,N1(C(CCC=C)=O)CCC(CN(C)C(C2NC(=O)CC2C)=O)CC1 21096,C1(NC(c2c(OC)nsc2)=O)CC(C(=O)NC2CCNC(=O)C2)C1(C)C 21097,C12(O)CCCN(C1)CC=CCC(=O)NC2.C(C(C)C(=O)OC)SC 21098,c1(N2CCC(C)C(NC(c3cc(C4CC4)no3)=O)C2)ncc2c(c1C#N)CCC2 21099,CC1CCCCC1(C(=O)O)NC(=O)OC(C)(C)C.c12cscc1NC2.C1(=O)NC1 21100,CC1CCN(C(c2nn(CC(F)(F)F)nc2Br)C(=O)NC(C)C(=O)OC)C(C)C1 21101,C(=O)(C(C)(F)C(C)(C)F)NCC(C(C)C)NC(c1ccc(OC)c(C#N)c1)=O 21102,C1(C(=O)NC(C2CCCC2)CNC(C2CCCO2)=O)(SC)CCC1 21103,C(CNC(=O)CCCC1(NC(c2ccc(CO)o2)=O)CCC1)(C(F)(F)F)OC 21104,Cc1sc(O)nc1C(=O)NCC12CC1CN(C(C13CCC1CC3)=O)C2 21105,c1(C(C(=O)NCCCCCNC(=O)CC2(O)CC2)O)cccc([N+](=O)[O-])c1 21106,CCCCCCCC(=O)NCC1(F)CC(NC(=O)CCc2cnco2)C1 21107,C(CC(C(=O)N1CC(CC)(OC)C1)NC(C1CCNC1=O)=O)=CC 21108,N1(Cc2cn[nH]c2)CCN(Cc2ccnc(Cl)c2)CC1.C123CC(C1)(C2)NC3=O 21109,c1(OCC)ncc(C(=O)NCCC(O)CNC(=O)CCC2CCCOC2)s1 21110,N1(C(C(n2c(C)ccn2)C)=O)CCC(CCNC(=O)Cc2ccsc2)CC1 21111,CCS(=O)(=O)CC(=O)NCC(C)(C)CN(C)C(C1CC2CC(=O)C1C2)=O 21112,C1(C(=O)NCC(C)NC(=O)COCC2CCOCC2)Cc2ccccc2S1 21113,c1(NC(=O)CCc2ccccn2)ncsc1C(=O)Nc1ccsc1C(=O)O 21114,C(=O)(C1CCCc2scnc21)NC1C2N(C(c3ncc(C)cc3F)=O)C(CC2)C1 21115,C(=O)(CC(O)CC(C)C)N1CC(NC(C2N(CCC)CCC2)=O)C(O)C1 21116,N1(C(c2ccc(CC)o2)C(=O)NCC2CC2)CCCC(CN2CCOCC2)C1 21117,CC1(C)NC(=O)OC12CCN(C(=O)C(=O)NC1CCN(CCF)C1)C2 21118,N1(C(c2cncc(C)c2C)=O)CCC2CN(C(=O)C(O)C3CC3)CC12 21119,c1(-c2c(C)ccc(CO)c2)ccc2[nH]c(C(N3CCCC(O)C3C)=O)nc2c1 21120,C1(NC(C(CCC)N(C)C)=O)CC2CCC1CC2NC(=O)CN(C)CC 21121,N1(C(CCc2ccc(C)o2)=O)CCOCC1CNC(c1ncoc1C(C)C)=O 21122,CCC(CC(=O)NC1CN(C(=O)Cn2cnc([N+](=O)[O-])n2)CC1O)C(C)(C)C 21123,C12(CNC(C(C)OCCC=C)=O)CC(NC(=O)C=Cc3ccncn3)(CO1)C2 21124,N1(C(C2C(CC)C2)=O)CC(CNC(c2ccc(=O)n(CCO)c2)=O)CC(C)(C)C1 21125,C1(CC(=O)NCC2CC2c2ccc(Cl)cc2)CCN(C(C2(CO)CCC2)=O)CC1 21126,c1(C(=O)NC2CCC(NC(=O)COC3CCCC3)CC2)ccn2cnnc2c1 21127,c1(CC)ccc(C=CC(N2CCN(CCNC(C3CCCC3C)=O)CC2)=O)cc1 21128,N1(C(=O)CCCCC2CC2)CCCN(C(C2C3CCC23)=O)CC1 21129,C1(CNC(C2(C)CC2)=O)CN(C(=O)COc2ccc(CC#N)cc2)C2(CCC2)C1 21130,c1(C(N2CC(NC(CC(C(=O)OC)C)=O)C(C)(C)C2)=O)ccn2cncc2c1 21131,CN1CCOC2CN(C(C3CCN(C(C4(CO)CC(C)(C)C4)=O)CCO3)=O)CC12 21132,C=CC1CCC1C(=O)N(C1CN(C(=O)C=CC(CC)=CC)C1)C 21133,c1(C(=O)NCCN(CCC)C(c2oc3ccccc3c2Cl)=O)ccc2nncn2c1 21134,Cc1noc(C)c1C(=O)OC(c1cc[nH]n1)=O.N12CC(C(C)C1)N(CCO)CC2=O 21135,c1(CCN2C(C)CC(NC(=O)C(=O)N(C)C)C2)ccc([N+](=O)[O-])cc1O 21136,c1(C(C(=O)NC2CCCC2)N(CC(COC)C)C)ccncc1F 21137,N1(CC(=O)N(C2(CNC(=O)CCOC3CCOCC3)CC2)C)CCN(C)CC1 21138,c1(C(C)O)ccc(C(=O)NCC2CCCCN2C(=O)C(F)=CC2CC2)cc1 21139,C(=O)(CCCC(=O)NCC(CO)NC(c1cccc(C2CCCC2)c1)=O)N(C)C 21140,N1(C(CCSC)=O)CC2CCC(CNC(=O)C(C)(C)c3ccno3)C2C1 21141,C1(CNC(c2cscn2)=O)CN(C(c2ccc(F)cc2F)=O)C2CCN1C2 21142,Cn1cnnc1CCCC(=O)NCC1C=CCN1C(c1cnc(C(F)F)s1)=O 21143,C(C(=O)Nn1cccn1)C1C(C)CCC1.C12(CCCCC1)C(=O)N2 21144,C1(CCC)(NC(=O)Cc2ccc(OC)c(Cl)c2)CCN(C(=O)C2=COCC2)CC1 21145,c1(CC(N2CC(C(C)NC(=O)C=CC(F)(F)F)C2)=O)n[nH]cc1Br 21146,C1(O)(CNC(C2CC3CC3C2)=O)CCN(C(C2COCCN2CC(F)F)=O)CC1 21147,C(CC(O)CC(=O)NC1CC(O)(CNC(=O)CCc2ccccc2)C1)SC 21148,C1(C(=O)NCCC(C)N(C)C(c2cc(O)nc(Cl)c2)=O)CC1C1(C)CCOCC1 21149,C(C(CC(C)C)C(=O)NC1(C(=O)NCC#CC(F)(F)F)CC1C)OC 21150,c1(C(=O)NC2CC3(C(NC(c4c(C)onc4)=O)C3)C2)cc2c(o1)CCCC2 21151,C1(NC(=O)NC(C(CSC)(C)C)=O)CCC2(CC1)CC2C#N 21152,C1(COC)(CNC(C2CCC2(C)C)=O)CCN(C(c2cc(Cl)nnc2O)=O)CC1 21153,C(CC(F)F)(C(=O)NN(C)c1ncccc1Cl)N(C)C(=O)OC(C)(C)C 21154,c1(CC(N)C(=O)NCCc2nc(C(F)(F)F)no2)cccc(Br)c1 21155,c1(C(N2CC3C(CNC(c4c(CNC)onc4)=O)(C3)C2)=O)cc(OC)c(O)c(Cl)c1 21156,C1(NC(C2CN(CCOC)C(=O)C2)=O)CN(C(C2(C)CCCCC2)=O)CC12CC2 21157,C1(NC(CC)=O)CCCCC12CCCN(C(c1ccc(C3CC3)cn1)=O)C2 21158,c1(C(=O)NC2COCCN(C(C(COC)(C)C)=O)C2)ccc2ccccc2c1F 21159,Cc1ccnc(C(=O)NC2CC(NC(=O)CCn3cc(Cl)cn3)C2)c1 21160,N1(C(c2c(C)ncc(Cl)c2)=O)C(C)CC2CN(C(C3(F)CCOC3)=O)CC12 21161,C1(C(=O)NCCc2cn(C)cn2)(CNC(C(C=CC)O)=O)CCCCC1 21162,c1(C(N2CCC3(CC2)CC3)C(=O)NC(CC)C)ccc(C)c2c1CCC2 21163,N1(C(C(CC)OC)=O)CC2CCC(NC(c3cnoc3C)=O)CC2C1 21164,CS(=O)(=O)C1CN(C(C2(F)CCC2)=O)CC1NC(c1cn2cc[nH]c(=O)c2n1)=O 21165,N1(C(CCN(CC=C)C(C2CC2F)=O)=O)CCC2(CCCO2)CC1 21166,C1(=O)CCC(C)(C)CNOCCC(COC)N1.C(C)(C)(C)OC(C)=O.CO 21167,c1(C(COC)NC(C2CC(O)(CO)C2)=O)ccc(F)cc1 21168,c1(NC(C(C2CC(NC(c3cccs3)=O)C2)F)=O)ccc(-c2nn[nH]n2)s1 21169,Cc1cc(C)c(CC(=O)NC2C=CCN(C(c3n[nH]cc3C)=O)C2)c(C)c1 21170,C1(NC(CC2(NC(C)=O)CC2)=O)C2CC1CN(C(=O)CNC(C1CC1C)=O)C2 21171,N1(C(c2ccn(C)n2)=O)CC(CNC(=O)COc2ccccc2)C2CC12 21172,N1(C(C=C(CCC)C)=O)CCC(C)(C(=O)NC(c2cnn(C)c2)CO)C1 21173,CC12CC(NC(C3CCC3(C)C)=O)(C1)C1(CCN(c3ncnc(Cl)c3Br)CC1)O2 21174,c1(C(=O)NC(C)CNC(=O)C(F)(F)c2csc(Cl)c2)cnc(N)cn1 21175,N1(C(c2cccc(CC=C)c2)=O)CC(C)C(NC(=O)CNS(=O)(=O)NC)C(C)C1 21176,CCC(C)(CCC(=O)OC)NC(c1cc(CCN)on1)=O 21177,C1(O)(CC(=O)NCc2ccc[nH]2)CN(C(c2ccsc2)=O)C1 21178,N1(C(CCC)C(=O)NCCCC(=O)OCC)CC(C)CCC12CC2 21179,C(=O)(C1CCCc2nnn(C)c21)NC(CNC(CCCCC)=O)CC(F)(F)F 21180,CCCCC(O)C(=O)N1CC(c2ocnc2CNC(C2(C)CCCN2C)=O)C1 21181,C1(NC(c2coc(C(F)(F)F)n2)=O)CCCCN(C(=O)COCC2CCOC2)C1 21182,C1(CC)CN(S(=O)(=O)CC2CC(C)(C)CO2)CC(C)S1=O 21183,N1(C(C2C(CC)CCN2C(c2ccnc(C)n2)=O)=O)CCc2ccsc2C1 21184,c1(C(=O)NC2CCN(C(C(CC)NC(N)=O)=O)C2(C)C)ccc2c(n1)CCCN2 21185,C12(C(=O)NC(c3ccc(N4CCOC4=O)cc3)C)CC(C1)C(C(F)(F)F)N2 21186,CCCC(CC(C)C)C(=O)NCC(=C1CN(C(C2CN(C)CC(C)O2)=O)C1)F 21187,Cc1ccc2c(c1)CC(NC(c1ccc(F)cc1)CC1CC1)C2 21188,C(CC(C)CCS(=O)(=O)NCC1COC2(CCCC2)C1)OC 21189,N1(C(C2CC(C)C2)=O)CCOC2CCN(C(=O)Cn3cnc([N+](=O)[O-])c3)CC12 21190,N1(C(c2c(CC)nn[nH]2)=O)CC2CC1CN2C(C1CC1OCCOC(C)(C)C)=O 21191,C(C(=O)NCC1CCCCN1C(=O)CC1CCC(=O)N1C)(C(C)(C)C)SC 21192,C1(CC(=O)N(C(C)C(=O)NC2CC(=O)N(CC)C2)CCC)CCC(C)(C)C1 21193,N1(Cc2c(C)onc2)CC(NC(=O)C(=O)NC2CCC3CC3C2)CCC1C 21194,N1(C(C(COC)(C)C)=O)CC2(CCC(CNC(c3cc(COC)cs3)=O)O2)C1 21195,c1(C(N2C(CCNC(CCSCCCC)=O)CCC2)=O)cn(C)nc1OC 21196,C(CC(C)(C)C(=O)N1CCC(C)(CNC(=O)CCC(C)(F)F)C1)SC 21197,c1(C(N(CCN(C(C2C(C)CCC2)=O)C)C)=O)ccc2cccnc2c1N 21198,c1(C(N2CC(C)(NC(C3C(SC)CCC3)=O)C2)=O)nn(C)c(C(F)(F)F)c1Cl 21199,C1(N(C(c2csnc2N(C)C)C(=O)NC)C)CCCN(c2cnn(C)c2)C1=O 21200,C1(CC)CN(C(=O)C(CNC(=O)OC(C)(C)C)CC2CC2)CC1C 21201,n1(CC)cc(C(O)CNC(=O)NCc2cnc(C)s2)cn1 21202,C(N=c1ccnc(NCC2CCCC(F)C2)[nH]1)C1(OC)CC(C)(C)CC1 21203,C(=O)(CC(C)(C)N(C(=O)CC1CCC=CCC1)C)N(CCCCCO)C 21204,c1(C(N2CCC(NC(C3(C)CCC(C)C3)=O)CC2)=O)cnn2c1OCC2 21205,C1(C)(CNC(Cc2nc(CC)sc2)=O)CC(F)(F)CN1C(c1scnc1C)=O 21206,N1(C(CC(CC)SC)=O)CCC(C)C(CNC(c2nccc(Cl)c2F)=O)C1 21207,c1(C2(C(=O)NC(CC=C)C3CC3CC=C)CCC2)ccc(F)cn1 21208,C1(NC(=O)CCOC2CCCC2)CC(O)(CNC(=O)CCC2CCOC2)C1 21209,C=CC1(NC(C23CC2CCN3C(c2sccc2F)=O)=O)CCCC1 21210,Cc1occc1CC(=O)NC1CCN(C(c2cn(C3CCCC3)nn2)=O)C1 21211,C#Cc1ccc(F)c(C(N2CCC(CNC(C3CCC(C)(C)OC3)=O)CC2)=O)c1 21212,c1(CC(N2CC=C(CNC(CC(C)F)=O)CC2)=O)ccc(S(N)(=O)=O)s1 21213,N1(C(C(C)Cc2ccccc2)=O)CC2CN(C(c3coc(O)n3)=O)CC2C1 21214,c1(C(N(C2CC(NC(c3ccc(Cl)cn3)=O)C2)C)=O)cnc2[nH]c(O)nc2c1 21215,c1(C(=O)NC(C(C)NC(C2CCCN2C=O)=O)CO)ccc(Cl)c(N)c1Cl 21216,c1(OC)ccc(CC(=O)NC2CN(Cc3nccnc3Br)CC2F)c(C#N)c1 21217,C(CCN(C)C(C1CCS(=O)CC1)=O)(C(C)C)NC(C1(OC)CC(C)C1)=O 21218,C=CC1CN(C(=O)C(C)(C)n2ccc(C)n2)CC1NC(=O)CC1C(=O)NN=C1C 21219,C(C)(CCCC(=O)N1CC(N2CCNC2=O)C1)NC(c1[nH]cc(C)c1C)=O 21220,C(=O)(C(CC(F)F)NC(c1ccc[n+]([O-])c1)=O)NC(CCC)CCO 21221,CCC(C)C(O)C(C)C(=O)NC1C2CCN(C(=O)C(O)C(C)(C)C)CC12 21222,C1(CNC(CCN(CCC)C)=O)C2CCCC1N(C(c1cccc(O)c1F)=O)C2 21223,C1(CNC(C2CC(O)(N(C)C(=O)OC(C)(C)C)C2)=O)CC2CC(C1)CC(F)(F)C2 21224,CC1CN(C(c2cnn3ccsc23)=O)CCC1NC(C1CN2CCN1CC2)=O 21225,c1(C(=O)NC2CC(C)CN(C(=O)CCc3cnccn3)C2)ccc2[nH]ccc2c1 21226,c1(NC(N2CCCC(NC(C(C)C3CCCC3)=O)C2)=O)ccc(Cl)nc1Cl 21227,C(c1ccc(C(F)(F)F)cc1)=CC(N1C(CNC(CCOCC#C)=O)CCC1)=O 21228,C#CCC(O)C(=O)NC(CCOCC)C(=O)NCCC1CCCCO1 21229,CC1(C)C(C(=O)O)CC1CNCc1cc[nH]c1C(=O)O 21230,CCC(CCOC)C(=O)NC1(c2cccc(C)n2)CCCC1 21231,Cc1c(NC(=O)CC2CCN(C(=O)Cc3cccnc3)CC2)cnn1C1CC1 21232,c1(C(N2CCC(COC)(NC(c3cncs3)=O)C2)=O)c(C)oc2nc(Cl)ccc12 21233,C(=O)(CC1=CCCC1)N(C(C(=O)N(C)Cc1snc(C)n1)C)C1CC1 21234,C1(C)(C(=O)NCC2C(NC(C3C(C(=O)OC)C3)=O)C2)CCc2ccccc2C1 21235,C1(CNC(c2c(C)nc(CO)o2)=O)C2CCC(C2)N1C(=O)CCn1cccn1 21236,C1(C(N2C(CNC(CCCCOCC)=O)CC(O)C2)=O)(OC)CCC(C)(C)C1 21237,C1(NC(CC(C)OC)=O)CCC(C)N(C(=O)C=CC2CC2)C1 21238,c1(C(=O)NC(c2ccc(C)cc2C)CC(=O)OC(C)C)ccc2sncc2c1 21239,c1(OCC)ccc(Br)c(NNC(=O)C2Cc3c(F)cccc32)c1 21240,C(O)(CC(=O)NCC1(CC2CC2)CC1)(C(F)(F)F)c1ncc(C)o1 21241,c1(-n2cc(C(=O)NC(CN3CCCC3)CO)nn2)cccc(Br)c1 21242,C1(C(N2C(C)(CNC(c3cccc(F)c3N)=O)CCC2)=O)CN(CP(C)(C)=O)C1 21243,N1(C(c2c(CC)cco2)=O)CCCCCC(NC(=O)C2=CCCS2)C1 21244,CCCCC(C)CCC(=O)NCC(C1CCOC1)NC(=O)CC#N 21245,c1(C(=O)NC(c2ccccc2OC)CNC(CCCCC)=O)cc(F)cc(Cl)c1 21246,Cc1nn(C)c(C)c1NCCC(N1CC(CN(c2ncccn2)C)C1)=O 21247,N12CCCCC1C(=O)N(C(CO)C1CCC1)CC2.c1(CC(=O)OC)nn[nH]n1 21248,CC1CN(C(=O)Cc2ccccc2F)CCN1C(=O)CCCOC(=O)C(C)(C)C 21249,CC(C)(O)C(F)C(=O)N1CCOC(CNC(C2CCCCO2)=O)C1 21250,C(=O)(CCOCCN(C(=O)Cc1ccsn1)C)N(CC(=O)NC(C)C)C 21251,c1(OC)cccc(-c2nc(C)c(C(=O)NCC3CC(NC(C4CCO4)=O)C3)[nH]2)c1 21252,c1(C(=O)NCC2(C(N(CC(O)CO)C(C)C)=O)CC2)csnc1Cl 21253,C1(NC(CONC(c2cn(CC)nn2)=O)=O)CCCCCC1CO 21254,S(=O)(=O)(c1cnn(C)c1)NCC(N1CCC(C)(NC(c2c(C)ocn2)=O)C1)=O 21255,C1(C(=O)NC2CCC(CC(=O)NC3(C)CC(O)C3)C2)CC2C(C1)C2(C)C 21256,CC1(C)OCc2c1n[nH]c2C(=O)NCC1CC(NC(=O)C(F)CC2CCCC2)C1 21257,c1(C(=O)NC(C2OCCN(C(CSCC#C)=O)C2)C)ccc(C#N)cc1OC 21258,c1(C(=O)NC(C2CN(C(=O)CC(C)(C)N(C)C)C2)C)ccc(Cl)nc1 21259,CC(CNC(=O)CSC)(CO)NC(=O)C(CC1CC1)NC(c1cccnc1)=O 21260,c1(-c2nc(CC(C)CCO)on2)c(Cl)cccc1Cl.C1CCCCCC(=O)O1 21261,C(=O)(C1CCOc2ccccc21)NCC(C1CCCN1C(C1C=CCC1)=O)(C)C 21262,C(CC(=O)NC(C)CCCCO)(C(C)C)NC(c1nc(COCC)oc1)=O 21263,c1(C(N2CCC(CCOC)(NC(C3(C)CCCCO3)=O)C2)=O)ccnc(Cl)c1O 21264,C1(C(=O)NC2CC(F)C2)CCCCCC1NC(C1(CO)CCOC1)=O 21265,c1(C(N2CC(C)OCC2C)=O)nc2ccccn2c1C1=CCOCC1 21266,c1(CC)cc(C(=O)NCCSCC(=O)NCC2(C#N)CC2)no1 21267,c1(C(N2CCN(C(CC=C=C)=O)CC2C)=O)cc(Cl)cc2nc(C)[nH]c12 21268,N1(C(c2cnn(CC)n2)=O)CC(C2CCCCN(C(=O)CC3CC4(CC4)C3)C2)C1 21269,S(=O)(=O)(c1[nH]c(=NC2CCCC(C(C)(C)C)C2)ccc1Br)NCCCNC(C)C 21270,c1(C(=O)NCC2(CCNC(COC(C)C)=O)CC2)cncc2c(O)nccc12 21271,CCC(CC)CC(F)C(=O)NC(C12CCC(CC1)C2)CNC(=O)C(C)(C)O 21272,N1(C(c2c(-c3c(C)cccc3)noc2C)=O)CC2CCCCC12c1ccccc1 21273,C#CCC(O)C(=O)N(CCCNC(=O)C(O)CCN(C)C)CC1CCCC1 21274,N1(C(C(CCC)CC)=O)CCCCCC(NC(c2coc(COC)n2)=O)C1 21275,Cc1cncnc1NCC1CN(C(=O)C(C)Cc2ccc(Cl)cc2)CCO1 21276,C1(C(N(C(CC)CC)C)=O)CC(F)CN1C(=O)CC1COCCO1 21277,C1(CNC(C(C)OCC2CC2)=O)CC(C)CN(C(=O)CC2CSCCO2)C1 21278,NS(=O)(=O)C1(C(=O)NCCC2(O)CCN(C(C3C4COCC34)=O)C2)CCC1 21279,Cc1nc2ccc(C(=O)NCC3C4CN(C(c5csc(C)c5)=O)CC34)cc2s1 21280,N1(C(CN(C)C(c2c[nH]c3nccc-3c2)=O)=O)CCC2(CC1)CC2C#N 21281,O=S(=O)(c1ccc(NOc2ccc(Br)cn2)cc1)OC(F)(F)F 21282,C1(CNC(C2CC(C)C2)=O)CCCCC1NC(c1cnccc1Cl)=O 21283,C1(O)(CC=C)CCN(C(=O)C(CO)NC(=O)C(CN(CC)CC)OC)CC1 21284,c1(NC(N2CCC(CC(=O)NC)C2)=O)nc2ccccc2n1C(C)C 21285,c1(C(=O)OCC)cc(CCNC(=O)Cc2nn[nH]n2)nc(O)c1 21286,Cn1nc(C(F)(F)F)c(Br)c1CN1CCC(C)(CO)CC1 21287,C1(NC(CC2(C=C)CC2)=O)CC(=O)N(C2CN(C(=O)Cc3c[nH]ccc3=O)C2)C1 21288,C1(C)(CNC(CCOC)=O)CCC(NC(C2(F)CCCC2)=O)C1 21289,C12CCOC1C(=O)N2.C1(NC(C(C)OCC)=O)CCCC1C(=O)OC 21290,C1(C(N2C(C(=O)NCC3CCOC3)CC=CC2)=O)CC2(C1)CC2(F)F 21291,C1(NC(=O)CCC2CC2)CCC2(CCN(C(c3csc(Cl)c3Cl)=O)CC2)C1 21292,c1(OC)cccc2scc(C(N3CC4C(NC(=O)C(C)N(C)C)C4C3)=O)c12 21293,c1(NCC(n2cccn2)OCC)[nH]c(=NCC2CC2(C)C)nc2sccc12 21294,C1(C2CCN(C(C3CCC(F)CC3)=O)CC2)(NC(C(CC)C(C)C)=O)CCC1 21295,C(CNC(c1nc(C)no1)=O)(C(C)(C)C)NC(CNC(CCNC(C)=O)=O)=O 21296,c1(C(=O)O)ccc(CN2CCC(CC(N3CCC(O)C(O)C3)=O)C2)cc1Cl 21297,C1(COC)CC(C(=O)NC2(N)CC2)N(C(C2CCC2)=O)C1.c1(S)ccccc1 21298,C1(NC(c2cc(C(=O)OC)ncc2)=O)CN(C(=O)C(F)C(F)(F)F)CCC1F 21299,CC(C(=O)NCC1CCN1C(c1cncc(C(F)(F)F)n1)=O)C(C)(F)F 21300,c1(C(N2C(CNC(=O)C(F)CC3CCC3)CCCC2)=O)cccc(C#CCO)c1 21301,C1(C(=O)NCC23CC2CN(C(=O)Cn2ccnn2)C3)CCC2(CC1)OCCO2 21302,C1(CNC(C=C(CC)CC)=O)(COC)CCCN1C(C1(CCF)CC1)=O 21303,C1(C)(C(=O)NC(C)CN(C)C(C2CCN(C)S2(=O)=O)=O)CCC(F)(F)CC1 21304,C(=O)(CC(=O)N(CC(C)CNC(c1cocc1C)=O)C)OCC 21305,N1(C(C)Cn2nccn2)CCN(C)CC(O)C1.C12(CCOCC1)C(=O)N2 21306,N1(C(C(C)(C)C(F)F)=O)CCCC(O)(CNC(C23CCC(C2)C3)=O)CC1 21307,c1(C(N2CCCCC2CCNC(C)=O)C(=O)NC)cc2cccnc2s1 21308,c1(C(=O)ON)nccc(CC2CCN(C(CCC)=O)C2)n1.C(C)(C)(C)O 21309,O=C(CCC(=O)c1cccs1)NCC(O)CCNC(c1ccn(C2CC2)n1)=O 21310,c1(C(=O)NCc2cc(C)oc2C)cc2cc(Cl)sc2[nH]1 21311,c1(CNC(C2CCCN(C3CCNC3=O)C2)=O)ccc(I)c(F)c1 21312,C1(CC)CN(C(=O)C(C2CCOCC2)O)CCC1NC(=O)C(O)C(C)(C)C 21313,C(=O)(CC(C)(C)CC(F)(F)F)N1CCCC(C(=O)NCc2cc(C)no2)C1 21314,C1(NC(CCCc2cc(C)no2)=O)CCN(C(=O)C(C)SC(F)(F)F)CC1O 21315,C(=O)(C1CCCc2cncn21)N(CCNC(c1nc2nccc(C)n2n1)=O)C1CC1 21316,c1(C(=O)NC(C2CCN(C(C(C)=C3CC3)=O)CC2)C)ccc2c(C)nn(C)c2n1 21317,c12ccc(cc1)S(=O)(=O)Nc1cc-2ccn1.CC1(CON)CC1 21318,C1(NC(CCc2cc(OC)no2)=O)CN(C(=O)CCC(C)C)C(C)(CC)C1 21319,N#CC1CN(C(=O)CSc2ncccn2)CC1NC(c1ccc2ncnn2c1)=O 21320,C1(CNC(C(=O)NC2CCN(CCC)C2)=O)CCCC(C(F)(F)F)CC1 21321,Cn1[nH]c(=NC(=O)C2CCCN2C(C2(C(F)(F)F)CCC2)=O)cc1Cl 21322,C1(C(N2CC(C)C(F)C2)=O)N(C(c2cc(C(N)=O)c[nH]2)=O)CC12CCCC2 21323,N1(C(C(C)N(C(C2(CC#C)CCOC2)=O)C2CC2)=O)CCOC(C)(C)C1C 21324,N1(C(Cc2c(C)n[nH]c2)=O)CC2CC(NC(c3nnn(C)c3N)=O)C(C2)C1 21325,N1(C(CS(CC)=O)=O)CC(S(=O)(=O)N2CCN(C(=O)C(C)(C)C#N)CC2)C1 21326,C(=O)(CCC(N)=O)Nc1nc(NC(C2CCN(C(CN3C(C)CC3)=O)C2)=O)sc1 21327,C(C)(c1cccc(C(F)(F)F)c1)=CC(=O)NC(CCC)(C)C 21328,C1(c2cnc(CC)nc2)NC(=O)N(CC)C2=C1C(=O)NC21CCSC1 21329,C(=O)(CCc1ncc[nH]1)NC1C(NC(CNC(=O)NC)=O)C1 21330,C1(COCC=C)CCCN(C(=O)N(C)CCC2CCCCC2)C1 21331,C1(NC(CCC2CCN(C(c3c(C)nc(C)o3)=O)C2)=O)CC2(CCCC2)C1 21332,C1(CN(C(=O)Cc2cncs2)C)CCCCN1C(=O)Cn1ncccc1=O 21333,c1(C(CC)C)cc(C(=O)NCc2ncc(-c3cccs3)[nH]2)on1 21334,N1(C(CCCNC)=O)CCc2nc(C3=CCSCC3)sc2C1.CO 21335,c1(C(=O)NC(C)CCNC(=O)C=CC2CCCC2)cnc2ncnn2c1O 21336,N1(C(C#CC(=O)N(C)C)=O)CCN(C(=O)CCC2CCCCO2)CC1CCO 21337,CCC(C(=O)N1CC(OCC(N)=O)C1)NC(c1cc(CO)[nH]n1)=O 21338,C1(NC(CC(CC(C)C)C)=O)CCC2CN(C(=O)CN=S(C)(C)=O)CCC2C1 21339,n1(C)nnnc1C1CC1.C1(CCC)CN(C(=O)CNC(=O)C(F)C2CCCC2)C1 21340,CC(C)(C)C(C#N)C(=O)NCC1(NC(C2CCC3(CCCC3)C2)=O)CC1 21341,c1(CC)cnn(CC(=O)NC2CC(CNC(=O)C(C)O)C2)c1 21342,N1(C(C(N2CCCCC2=O)C)=O)CCC2CN(C(c3cn(C)cn3)=O)C2C1 21343,CCC(C)(C)CC(=O)NC1CCCC(NC(=O)CSCc2ccc(F)cc2)CC1 21344,N1(C(CCc2cc(C)no2)=O)CC(NC(=O)CNS(N)(=O)=O)C(O)C1 21345,C1(F)(CNC(c2c(C)snn2)=O)CCN(C(c2cc(C(C)(C)C)[nH]c2C)=O)C1 21346,Cn1nc(C2CC2)cc1C(C1(C(C)(F)F)CC1)=O 21347,c1(OC)cccc(F)c1C1CCCN1CC(C)Nc1ccnc(Cl)n1 21348,CC(C)CCCCC(=O)N1CC(C2CC2)(C(=O)NCC2CC23CC3(F)F)C1 21349,Cc1cc(CC(=O)N(C(C)C(=O)NC2CC=CCC2)C2CC2)no1 21350,CN1CCN(C)C(C(N2CC(C(N3CCC(C(F)(F)F)C3)=O)C(C)(C)C2)=O)C1 21351,n1(C(C)C(C)(C)C)nc(-c2cccc(Cl)c2)nc1C1CC2CC2C1 21352,C=C=CC(C)C(=O)N1CC2C(NC(=O)CC3CCN(C)CC3)C2C1 21353,Cc1csc2ccc(C(N3CCCC3(C)CNC(c3nn(C)cc3C)=O)=O)cc12 21354,N1(C(CCCN(C)C(C23CCC(CO2)C3)=O)=O)CC2(CCC(=O)O2)C1 21355,C12(CCNC(C3CC(SC)C3)=O)CCC(CC1)N(C(c1cncn(C)c1=O)=O)C2 21356,c1(N2CCC(C)(CC)C2)ccc(S(=O)(=O)NC(c2ncccc2F)C)cn1 21357,CCC(C)(C)C(O)C(=O)NCC1CC(C)CCN1C(c1cc2c(nn1)CCC2)=O 21358,Cc1ccc(C)c(C(N2CC(CNC(=O)CC=CC(C)(C)C)C(O)C2)=O)c1 21359,C1(NC(CC2(C)N(C(c3cc(C)sc3)=O)CCC2)=O)CC2CC3C(C2)C13 21360,c1(COC)cc(C(N2CC(NC(=O)C(N3CCC(O)CC3)C)C=CC2)=O)c(C)o1 21361,C1(C(N(C2CCCOC2)CCC)=O)CCN(C(c2c[nH]nc2C2CC2)=O)CC1 21362,c1(NCCNC(=O)NC2CCC3(CC2)COC3)cc2c(cc1Cl)COC2 21363,C1(C(=O)NCCCCCNC(c2c(CC)csc2)=O)CCCNS1(=O)=O 21364,c1(CN=C(NC(C=C)C)NC(C)COC)cc(O)cc(Br)c1 21365,c1(OCCOC)ccc(COC=O)cc1.C12CC(C1)CNCC2.C(C)(C)(C)O.N 21366,C1(N(CC(=O)N(CC(C)N(C(C)=O)C)C)C(=O)OC(C)(C)C)CCCN1N=O 21367,C1(NC(c2ccc(OC)nc2)=O)C2CCN(C(=O)CCn3cnnn3)C2C1(C)C 21368,c1(C(=O)NC2CN(C(c3ccc(SC)s3)=O)C(C)C2)ccc(F)cc1C#N 21369,C(CCC(C)(C)C(=O)NCc1c(F)cccc1F)NC(CCC(C)=O)=O 21370,C1(CNC(=O)CCOC2CCOC2)CCCN(C(c2cc[nH]c2)=O)CC1 21371,c1(NC(c2ccc(-c3ccc(C)o3)cc2)=O)ccc(Cl)c(Br)c1Cl 21372,N1(C(C2C(OCC)C2)=O)C2CCC1CN(C(=O)C(C)Sc1ccccn1)C2 21373,C1(NC(C(=O)NC2CCN(c3ccc(COC)s3)CC2)=O)CCC(=O)C(C)C1 21374,N#CC1CCN(C(=O)CC2(CNC(=O)CC3CCOC3)CC2)C1 21375,c1(C(N2CCC(NC(CCCN(C)C)=O)(CO)CC2)=O)ccc2nonc2c1 21376,CC1CCn2cc(C(=O)NCC3(O)CN(C(=O)C(O)C(F)F)C3)nc2C1 21377,O(N1CCC(CC(=O)NC2CCN(C(c3csc(C)c3C)=O)CC2C)CC1)CC 21378,c1(CC)nc(CC(=O)N(C)CCN(C)C(C2CC2(C)C)=O)cs1 21379,N1(C(C2N(N=O)CCC2)=O)CC(NC(=O)C(F)(F)C(F)(F)F)CC2(CC2)C1 21380,N1(C(C(CC)CN(C)C)=O)CCC(C=CC(=O)NCCCCCN=[N+]=[N-])CC1 21381,c1(OC)cc(NC(C2CC2C(N2CC(OC(C)=O)C(F)C2)=O)=O)c(Cl)cc1Cl 21382,C1(NC(C(CC)=CC)=O)CC2(C1)CC(NC(C1CCC(C)(CC)O1)=O)C2 21383,C1(NC(Cc2cccc(OC)c2)=O)CCCN(C(=O)CS(C)(=O)=O)CC1 21384,N1(C(C(=O)NCCCOCC2CC2)CC2CCCCO2)CCCC(F)CC1 21385,C(=O)(C(C)(F)C(C)(C)F)Nc1c(F)ccc(CSCCCC)c1 21386,CC1=CC(NC(=O)C(C2(O)CCC2)NC(=O)CC(C)=C(C)C)CCC1 21387,N1(C(c2ccc(OCCC)cc2)=O)CCOCC(NC(=O)CC2CCC(=O)O2)C1 21388,C1(N(C(C(n2ccc(C)n2)C)=O)CCF)CCCN(C(c2nc(=N)cc[nH]2)=O)C1 21389,CC(CCNC(C1(S(C)(=O)=O)CC1)=O)CCNC(=O)CNC=O 21390,c1(C(N(CC(CNC(C(CC=C)CC=C)=O)C)C)=O)cccc2oc(O)nc12 21391,c1(OC)cc(OC)cc(C(N2CCCN(C(C3CC34CCCC4)=O)CC2)=O)c1 21392,C(C(C(=O)N1CC(NC(N)=O)C1)C(C)(C)C)NC(Cn1ncc(C#C)c1)=O 21393,c1(N2CCC(=C)C2)ccc(S(=O)(=O)N(CCCN2CCCC2)CC)cc1Cl 21394,c1(C(c2n(CC(=C)C)nnn2)NC(c2ccccc2F)CF)noc2c1CCC2 21395,N1(C(CC=CC=C)=O)CC(NC(=O)C(F)n2cccn2)CC(C)(C)C1 21396,c1(C(=O)NCC(C)N(C(c2cnc(O)n2C)=O)CC)c(C)cncc1C 21397,N1(C(c2c(C)cn(C)c2)=O)Cc2[nH]nc(C(N3CC(F)(CF)C3)=O)c2C1 21398,C(=O)(CCCC(=O)NOC(C)(C)C)NCC(CC)N(C(CC=CC)=O)C 21399,C1(NC(c2cnnn2C2CC2)=O)CC2CC(C1)N(C(C1SC3C=CC1CC3)=O)C2 21400,c1(C(N(CC2N(C(c3cn(CCC=C)nn3)=O)CCC2)CC)=O)cc(Cl)cn1C 21401,N1(C(C(C)(C)c2cscn2)=O)CCC2C(C1)CN2C(C1CCCOC1)=O 21402,N1(C(c2cnc(C(C)=O)c(C)c2)=O)CCCC2(CC(NC(c3cnco3)=O)C2)C1 21403,C(C(F)(C(=O)N1CCCCC1C(C)C)C(C)C)NC(c1nc(CC)oc1)=O 21404,N1(c2cc(SC)nc(C)n2)CCC(CNC(C2CCOC(C)C2)=O)C(F)(F)CC1 21405,N1(C(C2CN(CC)C(=O)C2)=O)CC2(CCCCN2C(=O)C(C)CSC)C1 21406,c1(OC)cnccc1C(=O)NC1CCCCC1NC(=O)COCCSC 21407,C1(NC(Cc2cnc(C)s2)=O)CN(C(C2CC3CCC2O3)=O)CC1C 21408,C12(NC(=O)CCCF)CCC(CNC(C34CC=CC(C3)OC4)=O)(CC1)CC2 21409,N1(C(c2ccn(CCN(C)C)n2)=O)CCN(C(c2cc(CN(C)C)on2)=O)CC1 21410,c1(N2CCC(S(=O)(=O)NC3(CC4CC4)COC3)C2)nc(C2CC2)nc2cc[nH]c12 21411,C=CCC(CNC(=O)CC(CC)C1CCC1)C(=O)NCc1cnc(C)cn1 21412,c1(C(=O)NC(CC)CNC(=O)CC(C)C2CCCCC2)nccc2cccnc12 21413,C1(NC(c2c(OC(C)C)nccc2)=O)CN(C(C2CCC3CC23)=O)CC2(CC2)C1 21414,C1(NC(C(CSC)(C)C)=O)CN(C(C2CN(C(N)=O)C2)=O)CC2CC12 21415,O(NC(=O)C(CC#CC)N(C(=O)C=Cc1ccncc1)CC)CCCC#C 21416,c1(C(=O)NCC(CC)NC(c2cccc(N)c2C)=O)cccc2[nH]cc(Cl)c12 21417,c1(C(=O)NC2CCC(C)N(C(c3nc(Cl)cs3)=O)C2)c(F)cc(O)cc1F 21418,c1(CC)noc(CCC(=O)N2CCC2CNC(=O)C(F)(F)c2nccs2)n1 21419,c1(CN2C3CN(C(CCN(C(C)=O)C)=O)C(C3)C2)cnc2cc[nH]c2c1 21420,N1(C(CCN(C(CCC=CCC=C)=O)C2CC2)=O)CCN(C)C(=O)C1 21421,c1(C(=O)NC(CN(C(C2C(c3n(C)ncc3)C2)=O)C)(C)C)cc2ncccc2o1 21422,C(=O)(C(CCOC)NC(C1CCN(C)C1C)=O)N1CC(N(C)CC)C1.CC 21423,c1(C(N(C(C)CCNC(c2cn(C3CCC3)nn2)=O)C)=O)cccc(=O)n1C 21424,c1(C(C)NC(=O)N(CC(=O)NC2CCOC2)C2CC2)ccncc1F 21425,C(=O)(C1CCCc2cncn21)NC(C)CCNC(=O)C(c1cc(F)cc(F)c1)O 21426,C12CC(C(O)C1)N(C)C2.C(C(=O)N(C)C)N(C(=O)C=CC(=O)N(C)C)CCC 21427,c1(OC)cccc(C(=O)C(=O)N(C)CCOCCN(C)C(C2CC2C#N)=O)c1 21428,C1(CC(=O)NCC2CC2CN(C(F)F)C2CC2)CCCCO1.c12cc(cs1)C2=O 21429,C(=O)(C1=CC(O)C(NC(=O)CN2CC3CCC2C3)C1)NC(CCC(C)C)C 21430,C(C)(C)(CCC(=O)N1CCC(C(=O)NCc2cnc(C)o2)(CO)CC1)OC 21431,C1(C(=O)NC2C(NC(=O)CCF)C2)COc2ccccc2C1 21432,C1(O)(C(C)NC(c2cc(C3CC3)ns2)=O)CCN(C(C2CCN(C)C2=O)=O)CC1 21433,N=c1cc[nH]cc1C(N1CCN(CCCNC(C2CCCS2)=O)CC1)=O 21434,C12(C)CN(C1)C(=O)C(C)CC1CN(C1)C2=O.c1(CC(=O)N(C)C)cccs1 21435,c1(C(N2CC3(CN(C(CN(C)CC)=O)C3)C2)=O)cccc2[nH]nc(O)c12 21436,N(C1CCCc2sc(Cl)cc21)C(CCn1cc(CNC)nn1)=O 21437,c1(C(N2CCC(CN=c3[nH]cncc3F)(F)CC2)=O)cccc2c(I)n[nH]c12 21438,C1(NC(C(C)c2ccsc2)=O)CN(C(c2ccnnc2O)=O)C(C)(C)C1 21439,c1(C(=O)NC2CCN(C(C(C(C)C)NC=O)=O)C2)cccc2nc(O)oc12 21440,C1(CCCNC(C=CC=CCC)=O)CCCN1C(c1cc(C)c[nH]1)=O 21441,C1(C(=O)NCC2CN(C(C3CN(C(=O)NC)C3)=O)C2)CC(C)(C)O1 21442,C(=O)(C#CC1(C)CCCO1)NC1CCN(C(CN(C)S(N)(=O)=O)=O)CC1C(N)=O 21443,C1(NC(CN2CC(C)(C)C2)=O)CC2CC1CC2C(=O)NCCCCCO 21444,C1(C)(C(=O)NC(C=C)C2CC2)CCN(C(=O)COC2(C)CCC2)C1 21445,N1(C(CS(=O)(=O)NCC)=O)CCN(C(c2scc(C)c2C)=O)CC1CC 21446,Cc1cc(Cl)ccc1NC(C12CCC(C1)OC2)=O 21447,N1(C(C2(C(C)C)CCC2)=O)CC(C(N)=O)(CNC(=O)Cc2cnsc2)C1 21448,c1(SCC(N2CCC(NC(Cn3cnc(C#N)n3)=O)C2)=O)n[nH]c2ccccc12 21449,c1(OC)cccc(S(=O)(=O)NNC(=O)C2CC(F)(F)C2)c1 21450,C1(C(=O)NC2(C)CCCCC2)CCC2(CCN(C(C3CCNC(=O)C3)=O)CC2)O1 21451,N1(C(COCCC(C)C)=O)CCC2CN(C(C34CCCC3C4(F)F)=O)CC2CC1 21452,c1(C(=O)NC2CC(CNC(CC3(C#N)CCC3)=O)C2)ccnc2[nH]nnc12 21453,CC1(C)NC(=O)CC1C(=O)NC12CC(C1)N(C(=O)Cn1cc(C3CC3)nn1)C2 21454,c1(OC)ccc2c(c1)OCC(c1nnnn1C)(NC(C(C)O)C(F)(F)F)C2 21455,C12(C(=O)NCCC3CC(NC(=O)CSc4ccc(Cl)cc4)C3)COC(CCO1)C2 21456,C1(C(=O)NCC(CC(=O)NC)C)CCN(C(c2occc2C(C)C)=O)CCO1 21457,C(=O)(C#CC1(C)CCCO1)NCC(C)CNC(c1ccccc1C1CC1)=O 21458,C1(F)(C(=O)NC2CC(CCNC(C=CC(C)C)=O)C2)CCCOC1 21459,N1(c2c(C(=O)OC)cc(C)cn2)CCC2(CCCCC2NC(=O)C(C)CF)C1 21460,CCC1=C(C(=O)N2CCC(C(C)NC(c3cc(C)ccc3C)=O)C2)CCCO1 21461,C=CCC(CC(C)C)C(=O)N1CCC(C)(NC(=O)CCC2CCC(=O)NC2)CC1 21462,c1(CC(=O)NC(C)CC(C)NC(c2ncoc2C2CC2)=O)ccc(F)c(Cl)c1F 21463,N1(C(C(CNC(C2(C)CC(=C)C2)=O)C)=O)CC(C)C(C)C1C 21464,C(C(C)(C)CCNC(=O)CC1CC=CCC1)NC(C1C(C(=O)OC)COC1)=O 21465,c1(NC(C2CCN(C(C(c3cccnc3)C)=O)CC2O)=O)cnn2ccccc12 21466,N1(CC(=O)NCC(O)CNC(c2ncccc2O)=O)CCCCC1=O 21467,Brc1c[nH]c2ncc(NCCCCCOc3ccccc3)cc12 21468,C1(CNC(C(CC)(C)COC)=O)CCC2(CN(C(c3cc(F)cc(Cl)c3)=O)C2)O1 21469,C1(NC(C2CC(C)(C)OC2)=O)CCN(c2ccc(C#N)nn2)CC1O 21470,C1(C(=O)NCCC(C(N2C(CN(C)C)COCC2)=O)O)CC(=O)CC(=O)N1 21471,C1(NC(C(=Cc2cccnc2)C)=O)C2CCC1CN(C(c1ccns1)=O)C2 21472,O=C(C(Cc1ccoc1)NC(C1(CO)COC1)=O)NCC(F)(F)Cl 21473,Cn1ncc(Cl)c1-c1cc(C(=O)NCc2cn(CC3COCCO3)nn2)on1 21474,C(=O)(C1CCCc2nn(C)cc21)N(CCCNC(=O)COC1CCCOC1)C 21475,C1(C(=O)NCc2ccc(C(=O)OCC)o2)C(Cl)(Cl)C12CC2 21476,C1(C2CC2)(NC(C(c2cccc(C)c2)C)=O)CCN(C(=O)CCN(C)CCO)C1 21477,N1(C(C2CCN(C(C3C(OC)C3)=O)C2)=O)CCC(C2CCC2)C1 21478,c1(C(C)C)cc(NC2CN(C(=O)CCc3cncs3)CC2(C)C)nc(C(C)C)n1 21479,Cc1cccc2c1CCCN2C(=O)NCC1COC(C)(C)OC1 21480,c1(CC(=O)N(C(C(=O)N(CC(O)CF)CC)C)C2CC2)ccc(C)nc1 21481,c1(C(=O)OC)ccc(CC(N2CC3C(NC(C4CC4C)=O)C3C2)=O)cn1 21482,C1(CC(=O)N(C2CCCN(C(c3nc(OC)c(C)s3)=O)C2)C)CC2CCC1CC2 21483,c1(C(=O)NC(CCNC(C(C(CC)C)O)=O)C)c[nH]c2cccnc2c1=O 21484,N1(C(CC(=O)NC)=O)CCCC2C(NC(c3ccon3)=O)C(C)(C)C12 21485,N#Cc1ccc2c(c1)C(=CC(=O)NC1(C(O)C(F)(F)F)CC1)C2=O.N1CC(CF)C1 21486,C=CCC(O)(CC=C)C(C)NC(C1CCC(F)(F)C1)=O.c12cc3c1cccc3[nH]2 21487,C(=O)(C1=NOCC1)N1CC(C(=O)NOC(C)CC)(CC=C)C1 21488,C(=O)(CCCCCN1CCOCC1)NC(c1cn(CCO)nn1)CCC 21489,C1(C(=O)NC(CC)C)CCN(C(=O)C(=O)NC2(Cl)CC2)CC1 21490,N1(C(C2(OC)CC2)=O)CC=CC(NC(c2c[nH]nc2C2CC2)=O)C1 21491,CC(C)C(CNC(C1CC2CCCC2C1)=O)C(=O)NCC(C)(F)C(C)(C)F 21492,C1(O)(CNC(C(CNC(C=C=C(C)C)=O)OC)=O)CC2C=CC1C2 21493,c1(C(=O)NC23CCC(CC2)CC3)coc2c1CN(C(C1CC(O)C1)=O)C2 21494,C1(C)(C(=O)NC(C2CCCO2)CC)CN(C(=O)CCCCNC(C)=O)C(C)(C)C1 21495,N1(C(CC2(OC)CN(C(=O)C(O)C3CCCC3)C2)=O)CCCCCCC1C 21496,C=CCCC(F)(F)C(=O)NC(CO)CCCCNC(c1cnsn1)=O 21497,c1(C(N2CC(O)C2)=O)ccccc1F.C(=O)(C(=O)NC(C)(C)C)N(C1(C)CC1)C 21498,CCCCCCC(C)C(=O)NC1CC1NC(c1cc(C)cc(F)c1N)=O 21499,c1(C(=O)NC(CNC(Cc2c(C)non2)=O)CO)ncc[nH]c1=O 21500,c1(-c2cn(C3C(C(N4CCCC4CC(F)F)=O)C3)nn2)cccc(C(=O)O)n1 21501,C1(CNC(CC(CC)OC)=O)CN(C(=O)CCc2nc(C)no2)CCC1(F)F 21502,N1(C(c2ccc(CN(CC)CC)o2)=O)CC(CCNC(c2ccsc2)=O)C(C)C1 21503,c1(C(=O)NCCn2c(C)ncc2[N+](=O)[O-])ccc2ncc(Br)cc2c1 21504,c1(C(=O)NC(CNC(C2CCC3CC23)=O)CO)cc2c(c([N+](=O)[O-])c1)OCO2 21505,n1(CC)nc(C)c2cc(C(=O)NCC(C)(CO)NC(C3CC4CCC4C3)=O)sc12 21506,N1(CC)CC(NCc2cnc(Cl)c(F)c2)CC(C)C1 21507,N#CC1(C(N2CCC(C(=O)NCC(O)C(F)(F)F)C2)=O)CC12CCC2 21508,C1(CCNC(CN(c2ccncc2)C)=O)CN(C(=O)CS(C)(=O)=O)CCCO1 21509,C=CCC(C)(C)CC(=O)NCCNC(=O)C(c1ccc(OC)cc1)NC(C)=O 21510,C1(CCNC(C2C(C(=O)OC)CCC2)=O)CCN(C(c2nc(O)c(C)s2)=O)CC1 21511,C1(C2CCN(C(=O)CCCCC(F)F)C2)(NC(=O)Cn2cccn2)CC1 21512,N1(C(C2C(CCC)CCC2)=O)CCC2(CC1)CCN(C(=O)CCN(CC)CC)C2 21513,c1(CC(C(=O)NCC(CNC(Cc2nc(C)[nH]n2)=O)CO)C)ccccc1F 21514,c1(C(=O)NCC(C)(C2CC2)NC(=O)CSC(=N)N)cnc2nccn2c1 21515,CC1C(C)N(C(=O)C2=CCCOCC2)CCN1C(=O)C(O)CC1CCCC1 21516,c1(CC(=O)NCC2(O)CN(C(c3oc(C)c(CO)c3)=O)C2)cccc([N+](=O)[O-])c1 21517,CC(C)C(C(=O)NCC(n1cc(-c2cccc(C(F)(F)F)c2)nn1)C)C(C)C 21518,S(=O)(=O)(c1ccc(Cl)nc1C)NCC1CCN(C(CCCC)=O)CC1 21519,N1(C(COC2CN(C(c3snc(C)c3N)=O)C2)=O)CC2CC(C)(C)C2C1 21520,C(C(CC(C)C)C(=O)NCCc1c(C)noc1C)NC(C=CCN(CC)CC)=O 21521,c1(OC)ccc(C(=O)NCC(C)(C2CC2)NC(c2cccn(C)c2=O)=O)c(C)c1 21522,CC1(C)COCCC1C(=O)NC1CCC(NC(=O)CCCC2CCCC2)C1 21523,c1(C(C(N2CC(OC)C(NC(c3csc(CO)n3)=O)C2)=O)C)ccc(F)cc1F 21524,C1(CC=C)(NC(=O)CCc2ccc(C)s2)CCN(C(C2CCO2)=O)C1 21525,c1(C(N(C)CC2COCCN2C(c2cn[nH]c2)=O)=O)noc2c1CCCCC2 21526,C1(C(NOCCC(c2cccnc2OCCN(C)C)C)=O)C2CC3C(C2=O)C13 21527,Cc1scnc1C(=O)N(CC(C)C(=O)NCCN1CC2CC2C1)C 21528,C=C(Br)CC(=O)NCCC1CCN(C(C2CC2F)=O)C1 21529,N1(C(=O)Cc2cncc(F)c2)CC2CC(C1)N(C(=O)COc1cccnc1)C2 21530,OC1(Cc2ccc(-c3nnc(C(F)F)o3)nc2)CC(O)C12CCC2 21531,Cc1cc(C(=O)NC2(CNC(=O)CC3CCOC3=O)CC2)c2ccccc2n1 21532,CCC(CC(=O)NCCCOCCC(=O)NC1C(CO)CC1O)C(C)C 21533,CC1=CC(NC(=O)COC(C)(C)CNC(C2(C)CCOCC2)=O)CCC1 21534,CN1CCN(C(C2COCC2NC(=O)C=Cc2cocn2)=O)CC1=O 21535,c1(CN2CCN(C(c3ncc(C)o3)C(=O)NC3CC3)CC2)cncc(Br)c1C 21536,N1(C(C(=O)Nc2ccc(OC)cc2OC)CC2CCC2)CCn2ncc(Cl)c2C1 21537,C(CCC(=O)NC(c1ccccc1)CNC(=O)Cc1ncccn1)=CC(C)C 21538,Cc1[nH]c(C)c(C(=O)NC2CCCC2NC(C2CC23CCC3)=O)c1C 21539,CC(C(=O)NC1CCC(N2CCN(C(c3ccc(C4CC4)s3)=O)CC2)C1)C(C)(C)O 21540,C1(NC(=O)CCc2cscn2)CCOCC1NC(=O)CCC(=O)N1CCCCC1 21541,CC1(C(=O)NC2CC(CNC(=O)CC3CCCC34CC4)C2)CC(C#N)C1 21542,CC1CN(C(=O)Cn2cc(CNC(=O)C3=CCCCO3)nn2)CC(C)(C)O1 21543,c1(OCC)nn(C)cc1C(N1CCC(N(c2cc(C(C)C)ncn2)C)CC1)=O 21544,C(CCC(CO)NC(=O)CC1CC(O)C1(C)C)NC(c1nc(COC)sc1)=O 21545,N1(C(Cn2c3cccc(C)c3cc2)=O)CCC2(NC(=O)CCF)CCCCCC12 21546,C(=O)(C1=CCCSC1)NC1(C)CN(C(C2CCN(C3CC3)CC2)=O)C1 21547,C12COCC1NC2=O.c1(CCC(=O)N(C23CC(C2)C3)C)cnn(C)c1 21548,c1(C(N(c2cn(CCNC(=O)Cc3nc(=N)[nH][nH]3)cn2)CCOC)=O)nnnn1C 21549,Nc1cc(C(N2CC(NC(=O)CCNC(c3ccsc3)=O)C2)=O)cc(F)c1 21550,CC(C(=O)NCCNC(c1ccns1)=O)C(F)F 21551,c1(CC(C(=O)NC(COCC)C(C)C)N2CCC(C(=O)OC)C2)ccc(Cl)cc1 21552,N1(Cc2scc(C)n2)CCOCC(NC(c2ccc(C#N)s2)=O)C1 21553,N1(C(c2cccc(CNC(C(C)(C3(C)CC3)OC)=O)n2)=O)CCOCCC1C 21554,c1(C(=O)NC2(CC=C)CCN(C(=O)CS(=O)CC)CC2)ccc2c(c1)CC(=O)N2 21555,C1(CC)CCC(C(=O)NCCC(C)NC(=O)C=C2CCC(C)C2)C1 21556,CCC1=C(C(=O)NC2CC(NC(c3cc(NC(C)=O)cnc3C)=O)C2)CCCO1 21557,C(CN1CCCC1)(CN=c1[nH]c2c(c(=NCCF)[nH]1)SCC2)N(CC)CC 21558,CC1C2CCC(C2)C1C(N1CCCC(C)(C(=O)NC2CC23CC(O)C3)C1)=O 21559,C1(CCNC(C(C)NC(CC)=O)=O)CCN(C(c2cn(C)cn2)=O)C1 21560,C(C(CC(F)(F)F)NC(C1(C)CC1(Cl)Cl)=O)NC(c1c(CC)oc(C)c1)=O 21561,O(NC(=O)CCC1CCCO1)CC(=O)NCC1(NC(=O)CC2CCNC2=O)CC1 21562,Cn1ncc2cc(COC(=O)CCn3cc(CN4CCC(F)C4)cn3)cnc12 21563,N1(C(CCc2cnc(C)o2)=O)CCC2CCCC12C(=O)NC1CCCC(C)(C)C1 21564,C1(CNC(=O)C2=NOCC2)CCN(C(C2CCC3C(C2)C3(F)F)=O)CCC1(F)F 21565,N1(C(c2c(C)ccc(C)n2)=O)CCOCC12COCCN(C(c1ccco1)=O)C2 21566,c12ccn3ncc(c3n1)C(=O)NCC1CCCN1C2=O.C1(C(=O)NC)(SC)CC1 21567,c1(CC(N2C(CNC(C(CCC)O)=O)CC(F)C2)=O)ccc(S(=O)(=O)CC)cc1 21568,C(C(=O)NCC1CC2(CCC2)CN1C(=O)CC(C)CF)(c1ccccc1)=C(C)C 21569,N1(C(c2cc(C)sc2)=O)CCC(C2CCCN2C(=O)CC2(O)CCOC2)CC1 21570,C(=O)(C(C)(C)CCCC(C)=O)NC(C(C)O)CO 21571,c1(C(N2CCN(C(C(COC)C)=O)CC2CF)=O)ccc2c(c1)CC(C)(C)C2 21572,c1(C(N2CCCN(CCN(S(C)(=O)=O)CCO)CC2)=O)cccc2cccn12 21573,c1(N2CC(C)C(NC(=O)C(C)(C)C(F)(F)F)CC2)nc2ccc(F)cc2s1 21574,c1(-c2nc(CCSC)nn2-c2ccn(C(C)C)n2)c[nH]c2cccnc2c1=O 21575,C1(C(=O)NC2CN(C(=O)Cn3cccn3)CC23CC3)C2C3CC4C1C1C2CC3C41 21576,Cc1cc(NC(c2ccc(-c3ccccc3)nc2)=O)ccc1F 21577,N1(CC(Br)=C(C)C)CCC2(CC1)CC2C(=O)NCc1nnc(C)s1 21578,O=C(CC1CCOc2ccccc21)NC1C=CCN(C(c2c[nH]nc2F)=O)C1 21579,c1(C(N2CC(OCC)C(C)C2)C(=O)NC)ccc(C(F)(F)F)cc1Cl 21580,N1(C(c2ccc(SC)o2)=O)CCCCC(CCC(=O)NCC2COCCN2C)C1 21581,c1(CC(=O)NCC(C)(C2CC2)NC(c2nonc2N)=O)csc2nc(C3CC3)cn12 21582,c1(C(=O)NC2CN(C(C3CC(O)C3)=O)CC3(CC3)C2)ccc2nnc(O)n2c1 21583,C1(CNC(C2C(C=C)C2)=O)CN(C(=O)CCC(=O)OCC)CC12CC2 21584,C1(NC(c2cocn2)=O)CN(C(C2CCCC3(CC3)C2)=O)CCC1F 21585,N(C1COc2cc(Br)ccc21)CCNc1cc(C(=O)OCC)c(I)cc1 21586,N1(C(C(CC)CCOC)=O)CCC2(CC2)CC1C(=O)NCC(C)(O)CO 21587,CC(C)CCN(CCC(C)C)C(=O)CC1CC1CNC(=O)C(C)OC1CC1 21588,c1(OC)ncccc1C(=O)N(CC(C)NC(c1ccc(-c2ccccn2)o1)=O)C 21589,c1(OC)cc(Cl)c(C(N2CCC(C(C)O)C2)C(=O)Nc2ccccc2Cl)cc1Cl 21590,C1(C)(NC(C2(CC)CCN(C(C3CCN(CC)CC3)=O)C2)=O)CCC(=O)N(C)C1 21591,C1(NC(c2scc(CC)c2)=O)(COC)CCN(C(c2cc(SC)c(C)o2)=O)CC1 21592,NCC(O)C(=O)NS(=O)(=O)Cc1ccc(CN2CC(C(=O)O)C2)o1 21593,c1(C(=O)NCC(C2CCCOC2)OCC)cnc2ccccn12 21594,C1(CNC(CCC(=O)NC)=O)CN(C(=O)CC(C)(F)F)CC12CCC2 21595,C1(C(=O)NCCc2scc(C(C)C)n2)CCCC1S(C)(=O)=O 21596,c1(OC)cc(C(=O)NCC2CC2CC(N2CCCC2CF)=O)on1 21597,C(CN=S(C)(C)=O)NC1(c2n(C3CCC(C(=O)OC)C3)nnn2)CS(=O)(=O)C1 21598,n1(C2CCC(C)C2)nc(CC2CCOCC2)nc1-c1cnon1 21599,C(c1ccccc1F)=CC(=O)N(CCC)CCNC(C1CC2(C1)CC2F)=O 21600,c1(CC(=O)N(CCN(C(C2CCC(CO)CC2)=O)CC)CC)sc(C)nc1C 21601,C1(C(=O)NCCCCCOC)CCN(C(=O)C2=C(C)CC2)C1C(C)C 21602,CC1(C(N2CCCC(CNC(=O)COc3ccccc3F)C2)=O)CCC(F)(F)C1 21603,C1(CNC(C2(C)CSC2)=O)CCCCN1C(C1CC(C(N)=O)C1)=O 21604,N1(C(COCCOC)=O)CCOC(c2cn(CCCC3CCOC3)nn2)C1 21605,c1(-c2nc(C3CCCC(=O)O3)n(C3CCCSC3)n2)cc(F)cc(F)c1 21606,N1(C(c2ccn(C(C)C)n2)=O)CCC(CNC(c2cccc(CC#N)c2)=O)CC1 21607,c1(C(=O)NCC2N(C(CC=C)=O)CCN(C)C2)ccc2n[nH]c(C)c2c1Cl 21608,C1(CCCCNC(C(C=CC)O)=O)CCN(C(=O)CCSC(F)(F)F)CC1 21609,C1(NC(C(C)=CCC)=O)C=CCCC1C(=O)NCc1nn(C)cc1CO 21610,CC1=NOC(=O)C1CC(=O)NCC1(CNC(C2(C)CCOCC2)=O)CC1 21611,C(=O)(C(F)(F)CCn1cccn1)NCC(C)CN(C)C(c1cc(=O)cc[nH]1)=O 21612,c1(C(N2CC(CCNC(C=CC(C)C)=O)OCC2)=O)cccc2c1C(C#N)C2 21613,N1(C(c2n(C(C)C)nnc2)=O)CCC(O)(C(C)NC(=O)CCc2ncco2)C1 21614,O=C(C1CCCc2scnc21)N1CCCNC1=O 21615,CC1CCN(C(C2C(C(F)F)C2(C)C)=O)CCN1C(=O)CSc1ccccc1Cl 21616,C(=O)(C(C)CC(N)=O)N(C(C(C)O)C(=O)N(CCCCN(C)C)C)C 21617,C1(C(=O)NC2(CC=C)CN(C(=O)Cc3csc(Br)n3)C2)CC=C(C)CC1 21618,C(CN=C(NCC(C1CNC(=O)C1)(C)C)NC(C)CC=C)OCC#C 21619,c1(NC(C)=O)ccc(Br)cc1C(=O)NC1CCC1NC(=O)CCCC#N 21620,CC1C2C(CCN2C(=O)CC2CCCC(=O)C2)CN1C(=O)CC(O)C(Cl)(Cl)Cl 21621,C(=O)(CS(=O)(=O)CC(F)(F)F)N(CC(C)O)CCNC(c1c(OC)nn(C)c1)=O 21622,Nc1cnc(Br)c(C(=O)NCCNC(=O)CC2(C3CC3)CC2)c1 21623,c1(CC)nc(N2CC(F)CC2CNC(=O)C(C)OCC(C)C)cc(C#N)n1 21624,C1(CNC(C2(CCCC)CCC2)=O)CN(C(C2(F)CC=CCC2)=O)CC12CCC2 21625,N(C1c2ccccc2OCC1C)C(c1ncnc2cccc(C)c12)CCC 21626,C(=O)(C(C)S(C)(=O)=O)N(CCCN(C(c1c(CCC)occ1)=O)C)C 21627,C1(C)(CC)C=C(C(=O)N2CC3CC(NC(c4cccc(=O)n4O)=O)C3C2)C1 21628,CCC(CCCC(=O)N(CC(=O)NC)C)NC(c1cc(C(N)=O)co1)=O 21629,CC1CC(NC(C2CCCN(CCNS(C)(=O)=O)C2)=O)CCS1 21630,N1(C(C)C)CCCC(C(=O)O)C1=O.c12ccccc1S2 21631,C1(C(=O)NC(C(C)C)(C)C)CC(=O)CN1C(=O)CCc1ccncc1 21632,C1(CNC(C=CCC)=O)CCC2CN(C(=O)CCC(=O)NC)CCC2C1 21633,c12cccc(c1)CO2.C(=O)(CP(C)(C)=O)NC(CNC(c1c(C)non1)=O)C 21634,N1(S(=O)(=O)Cc2nnc(Cn3cccn3)o2)CCCC(CN=[N+]=[N-])C1 21635,c1(CC)cc(Cl)ccc1C(=O)NCC1(F)CCN(C(=O)C=CCO)C1 21636,c1(CC)ccc(CC(N2CCN(Cc3cc(-c4ccccc4)n[nH]3)CC2)=O)cc1 21637,C(C(C(=O)N1CCN(C(=O)C=C2CCSCC2)CC1)C(C)(C)C)OCC=C 21638,Cc1nn(C2CCC2)cc1C(=O)NC(C(C)NC(c1ccc(Cl)[nH]1)=O)C(C)C 21639,O=C1CCCC(C(=O)NCCCNC(c2csc(C3CCCCC3)c2)=O)O1 21640,Cc1c(CC(=O)NC2CN(C(=O)CCc3cc[nH]n3)C2)ccc(Cl)c1Cl 21641,CC1(C)CC(C(=O)NCC(C)(C2CC2)NC(C2CCCCC2CC(N)=O)=O)=NO1 21642,N1(C(C(c2cnn(C)c2)NC(C=CCC)=O)=O)CCC(C)(O)C(O)C1 21643,c1(C(C)(C)NC(CCCC)Cc2ccccc2)cnn2cccnc12.C(=O)C(CC)C(C)C 21644,C1(CNC(C(CC)N(C)C)=O)CCC2CN(C(=O)C=C(C)c3cccs3)CC12 21645,N#CC12CC(C(=O)NC3CC(C(N4CCCC4c4ncc[nH]4)=O)C3)(C1)C2 21646,c1(NC(C)CCCCO)cc(S(=O)(=O)NCC2CC2c2ccco2)ccc1C#N 21647,Cc1ncc([N+](=O)[O-])cc1C(=O)NCCNC(C1CC(C2CCCC2)C1)=O 21648,N1(C(C2C(CCC)CCC2)=O)CCSCC1CCNC(=O)Cn1nnnc1C 21649,C1(C)(CC)CC(NC(=O)C=CC(C)NC(=O)CNc2ccncc2Cl)CCO1 21650,N1(C(C(=O)NCc2n(CC(C)C)ccc2)=O)CCC(C(=O)O)C1C(C)C 21651,n1(CCOC)nc(C(N2CCC(C(C)NC(C3(CCO)CC3)=O)C2)=O)ccc1=O 21652,C=CCC(Cc1ccccc1)C(=O)N1CC(Cc2cc(OC)ns2)C1 21653,C1(CS(C)(=O)=O)CCCC1(c1nnnn1CCc1nccs1)NCCNC(N)=O 21654,C1(CC(=O)NCCCC2(NC(C(C)C#N)=O)CC2)CCCCN1C 21655,N1(CC(=O)OCC)CC(CNC(=O)CCCOc2ccccc2)OC2COCC12 21656,c1(C(=O)NC2CCC(CNC(C3NC(=O)OC3)=O)C2)cccc(Cl)c1Br 21657,n1(CC)cnc2c(N3CCC(C)=C(C)C3)[nH]c(=NCc3ccncc3N)nc12 21658,c1(C(N(C2CCN(C(C3COCCC3(F)F)=O)C2)C)=O)nc(O)nc(O)c1N 21659,c1(C(=O)OC)ccc(Cl)c(C(F)F)c1.c12nc(no1)CNC2=O 21660,N1(C(c2n(CC)ncc2)=O)CC2CCCC1(CNC(c1conc1C1CC1)=O)C2 21661,C(c1ccccc1)=CCC(=O)NC(C)(C)CNC(=O)Cc1csnn1 21662,Cc1cc(CN2CC(NC(=O)COc3ccccc3F)C2)ccc1Br 21663,C1(C(=O)NCC2CC(NC(C(n3ccc(C)n3)C)=O)C2)CCOC(C)(C)C1 21664,N1(C(c2nc(Cl)c(Cl)s2)=O)CC2CCN(C(c3ccncc3)=O)C2C1 21665,C1(C(=O)NC(CC)(C)CNC(=O)Cc2cn[nH]c2)CC(C)CCO1 21666,Cc1nc(Br)sc1C(=O)NC(C1(F)CCCC1)C1CCCC1 21667,N1(C(C=CC(=O)OCC)=O)CC2(C=C(C(=O)N(C3CCN(C)C3)CC)CO2)C1 21668,c1(OC)cc(C)c(C(=O)NC2CC3(C2)CC3NC(=O)CC2CCCN2C)cc1Cl 21669,C1(C(N(C)CCOCCNC(=O)C=CC2CCCC2)=O)CCCCC1C(F)(F)F 21670,Cc1ccnc(C(=O)NC2CC2CNC(c2snc(O)c2Cl)=O)c1N 21671,C(=O)(CC1OCCc2ccsc21)N1CCN(C(C(CC=C)N(C)C)=O)C(C)C1 21672,c1(C(=O)NCC2C(NC(C(COC)OC)=O)CC2)cc(=O)n(C)cc1Br 21673,CCC(C(=O)NCC1CCC(NC(c2ncccc2Cl)=O)CC1)C(C)(C)CC 21674,N1(C(C2(SC)CC2)=O)CCOCC(NC(=O)C=CSc2ccccc2)C1 21675,C(=O)(C(C)(F)C(C)(C)F)NCCCOCCN(C(c1cnc(C(C)C)nc1)=O)C 21676,C1(C(=O)NCC2CCCN(C(c3ncccn3)=O)C2)Cc2n[nH]cc2C(=O)N1 21677,CCC(CNC(=O)CCS(N)(=O)=O)(CC)C(=O)NCC1CCOC(C)(C)C1 21678,Cc1ccc(C(=O)NC(C)CN(C(=O)CC2COC(=O)N2)C)c2c1CCC2 21679,c1(NC(C2NCCN(C(C(C)O)=O)C2)=O)cc(F)c(Cl)c(Cl)c1 21680,c1(CC(=O)N(C2CCN(C(=O)C#CC3(C)CC3)C2)CC)c(Br)ccc(F)c1F 21681,CCC(CC(=O)NC1CCC(NC(c2ccc3nc(C)[nH]c3c2)=O)C1)C(C)(C)C 21682,C=C(C)CCC(C)NC(c1cccc(Cn2cc(CN(C)C3CC3)nn2)c1)=O 21683,c1(C(=O)NCC2C(C)(C)C(NC(c3n[nH]cc3Cl)=O)C2)ccc2c(c1)OCCO2 21684,N1(C(C(CC)(C)C)=O)CC2CC(C1)CN(Cc1cc(I)c(OC)cc1Cl)C2 21685,C(CCNC(=O)C(C)CO)(C(=O)NCCCN1CCCC1)OC 21686,c1(C(=O)OCC)c[nH]c(=NCC2(F)CCN(C(C3CC3(C)C)=O)CC2)cc1C 21687,c1(CNCc2c(OC)nc(C)cc2)[nH]c2ccccc2c1Cl 21688,CCC(C)C(C(=O)N1CCC(C(F)(F)F)C(NC(c2ccnn2C)=O)C1)OC 21689,Cc1ccc(C2CCN(CC=CCC3CCCCN3C(=O)C(F)(F)F)C2)nc1 21690,Cc1onc(CC(=O)NCC2(C)CCCN(C(c3coc(Cl)n3)=O)C2)c1C#N 21691,C1(C2CCOCC2)(C(=O)NCC2(NC(C34CCCC3C4Br)=O)CC2)CC1 21692,c1(C(=O)NC(CC(C)NC(C2CCC(=O)N2)=O)C)ncccc1OC(F)F 21693,c1(OC)cc(F)cc(C(N2CCC(N(C)C(C3CC(CC(F)F)C3)=O)C2)=O)c1N 21694,C1(NC(C=CC(C)(C)SC)=O)CCCN(C(C2CCCCCO2)=O)C1 21695,S(=O)(=O)(c1ccc(CBr)cc1)N1CC2N(C(CSC)=O)C2C1 21696,C(CO)(CCCCNC(c1ccc(=O)n(CC(C)O)c1)=O)NC(C(C)OCC)=O 21697,C1(NC(C)C)CCN(C(=O)OC(C)(C)C)CC1C(=O)Sc1ccncc1Cl 21698,n1(CC)cc(S(=O)(=O)N2CC3CC2CC3NC(=O)Cc2ccc(Cl)cc2Cl)cn1 21699,n1(CCNc2c(C)c(N(C)CC3CC(O)C3)ncn2)cnc2c1CCCC2 21700,N1(C(c2c(=N)cc[nH]c2)=O)CCCC(NC(c2ccsc2Br)=O)C(F)C1 21701,c1(C(N2CCN(C3CNC3)CC2)=O)csc2c1CCNC2 21702,CC(CC(F)(F)F)C(=O)NC(CC(=O)N(CC(O)C(C)(C)C)C)C(F)(F)F 21703,c1(C(=O)NCCC(CC)(C)NC(=O)CCC(C)(C)C)ccc(C#N)cn1 21704,c1(C(=O)NC(C(C)(C)NC(Cc2c(C)nn(C)c2)=O)C)ccc2c(c1)CN(C)C2 21705,C(c1cccc(Cl)c1)=C(C(=O)NC1(C)CCN(C(C(C)OCCOC)=O)CC1)C 21706,C1(NC(c2cnn[nH]2)=O)CCC2CN(C(c3cccn4ccnc34)=O)CC2C1 21707,C1(CNC(C2N(CC)CCC2)=O)C2CCC1CN(C(C1CCC1)=O)C2 21708,c1(CC(=O)OC)ccc(C(=O)NC(C)CC(C)NC(=O)Cc2cccs2)c(C)c1 21709,N1(C(C(c2n(C)cnc2)O)=O)CCC(F)(CNC(C2CCC3(CCC3)O2)=O)CC1 21710,N1(Cc2c(OC(C)C)ccc(OC)c2)CC(C)C(P(C)(C)=O)C1 21711,c1(C(C(C)NC(c2ccsc2Br)=O)NC(C=C(C)C)=O)ccccc1 21712,C(=O)(CC(C(=O)OC)C(C)C)NC1(CO)CCCN(C(C2(COC)CC2)=O)C1.OC 21713,S(=O)(=O)(c1cccs1)NCC(=O)NC1CC(NC(C=CC(=O)N(C)C)=O)C1(C)C 21714,C1(NC(C2CCC2(F)F)=O)CC2(CCN(C(C3(C4CC4)CC3)=O)CC2)C1 21715,c1(N(C)CC)nnc2c(C(N3CCc4cc(Br)cnc43)=O)ccc(C(F)(F)F)n12 21716,C1(NC(C(F)=CCC)=O)CC2CC(C1)N(C(C1CC1[N+](=O)[O-])=O)C2 21717,C(=O)(CC(CC1CC1)NC(C1C2CN(C)CC12)=O)NCCC(=C)C 21718,N1(C(CCC(=O)N(C(C)C)C)=O)CCC2(NC(=O)CC(O)C(C)C)CCCC12 21719,c1(CC)nc(-c2nc(CN3CC(C)OC(C)C3)nn2C)ccc1Br 21720,C(C)(C(=O)NC1CCC1NC(=O)COCCCOC)OCC=C 21721,CN1CC(C)(C)CC1C(=O)NC1CCCN(C(c2cnc(C#N)s2)=O)C1 21722,Cc1ccc(C(=O)NC2CCN(C(=O)Cn3cc(CO)nn3)C(C)C2)c(O)c1 21723,c1(CSCC(=O)NC2C(NC(C(C)C)=O)CCC2)ccc(O)cc1 21724,Cc1c(C(=O)NCC2CCCC(NC(C34CC(CO3)C4)=O)C2)cnc2ccnn12 21725,C12CCCN(C1)C2=O.c1(C(C(=O)N(C2CCCC2O)CC)C)ccn(C)c1 21726,N1(CC(=O)NC2C=CC(CC(=O)NC3COC(=O)C3)C2)C(=O)CNC1=O 21727,N1(C(C(C)(C)C2CCCC2)=O)CCC(CNC(=O)COCC2CCOC2)C(O)C1 21728,c1(C(N(C(=O)CN2CCCC2C)CCOC)=O)cc(I)c(F)cc1F 21729,CC1CC(NC(c2ccc(C3CC3)nc2)=O)CN(C(c2cnc(S)n2C)=O)C1 21730,CCC(CC)C(C)C(=O)NCC1(F)CC(CNC(=O)CC2=CCOCC2)C1 21731,c1(C(C)C)ccc(C(N2CCC(CF)(NC(=O)CC3CCCC3(F)F)C2)=O)cc1 21732,Cc1nc(CC(C)C)sc1C(=O)NCC1CN(C(C2OC(C)CC2C)=O)CCO1 21733,CC(C(O)C(=O)NC(CNC(=O)CN(C)C(N)=O)C1CC1)c1ccc(Br)cc1 21734,CC1CC(NC(C2CCC2)=O)CCN1C(=O)C(=C1CCCCC1)F 21735,Cc1cc(C)n(-c2ccc(-c3nccn3C(c3ccc(F)cn3)C(C)C)cn2)n1 21736,C12(CNC(c3cnn(C(F)(F)F)c3)=O)CCC1CCN2C(=O)Cc1cccs1 21737,C(=O)(N=c1ccn(C(C)C)[nH]1)C1(CC=C)CN(C(=O)C(c2ccn(C)c2)C)C1 21738,N1(C(C2CC(NC(CC3(C)OCCO3)=O)C(O)C2)=O)CCCC(C)(C#N)C1 21739,C(C(C)CN=c1[nH]c(=NC(C)c2cnn(C)c2)[nH]c2ccsc12)SC 21740,N1(C(CCCCOC)=O)CCCC(C)C1CCNC(=O)C=CC1CCOCC1 21741,c1(C(=O)OCC)cc2cc(NCC3CCCC3N)ccc2s1 21742,c1(C(=O)OC)nccc2cc(-c3ccc(OC)c(C(=O)OC)c3)ccc12 21743,CC(C)CC(CNC(=O)CC(C)NC(c1ccccc1)=O)NC(C1CC(F)C1)=O 21744,N1(C(C(C=C)O)=O)CCOCC1CC(=O)NC1(CCO)CCCC1 21745,Cc1cc(N)ccc1C(=O)NC(C)(C)CCCCNC(=O)CC1CCCOC1 21746,N1(C(CCCC#C)=O)CCC(O)(CCNC(c2coc(COC)c2)=O)CC1 21747,CC1CN(C(c2ccc(C3CCC3)nc2)=O)CC1NC(C1(F)CCOC1)=O 21748,Cc1ccc(S(=O)(=O)NCC(=O)N(CC(N2CC(CO)C(O)C2)=O)C)cc1 21749,C(C(CC(F)(F)F)NC(=O)CN1C(=O)CCC1=O)NC(CC(C)c1ccco1)=O 21750,c1(NC(Cn2c(CC=C)nnc2S)=O)cc2scc(Cl)c2[nH]1.C1CC1OCC=CC 21751,c1(C(=O)NCCC2CC(NC(C3ON=C(C(C)C)C3)=O)C2)cncc2c[nH]nc12 21752,S(=O)(=O)(c1cccnc1NCCc1nncs1)NC1C(C)CCCC1 21753,C=CCCCCC(=O)N(C(C)CCNC(=O)C(N1C(=O)CCC1=O)CC)C 21754,C1(C)(CNC(Cc2c(C)nc[nH]2)=O)CCCC1NC(c1cnc(C(F)F)cn1)=O 21755,C=CCC(C(=O)NC1(COC)CC1)OC.N12CCN(CC1)C(=O)C=CC2 21756,c1(C(CNC(C=C(COC)C)=O)NC(=O)C(C)Cn2ccnc2)ccc(F)cc1 21757,c1(SCC(=O)NCC2(Nc3cc(OC)nc(SC)n3)CC2)nc2ccccc2s1 21758,CCC(C)(C)C(=O)C(=O)NC1CC(C)N(C(=O)CN2CCC2)C1 21759,Cc1ncc(N)cc1C(N1CC(CNC(C2CCCCCN2C)=O)C(F)(F)C1)=O 21760,c1(SC)ccc([N+](=O)[O-])cc1C(=O)NCCCC(C)(C)NC(=O)CC1(CO)CC1 21761,CCCCC(CNC(c1c(C)nsc1N)=O)NC(=O)CCN(CC)CC 21762,c1(OC)ccc(NC(=O)CCCc2cn(C3(COC(C)C)CC3)nn2)cc1.C1CC1 21763,c1(C(N2CC(F)(C(=O)NC(CC(=O)NC)C3CC3)C2)=O)cccc(CO)c1 21764,CC(C)S(=O)(=O)CC(=O)N1CC(CNC(=O)C(C)c2ccco2)C2(CC2)C1 21765,c1(C(F)(F)F)cc(CNCC2(NC3CC3Br)CC2)ccn1 21766,C(=O)(C(C(F)(F)F)C(F)(F)F)NC1(C2CN(C(c3ncc(CC)cn3)=O)C2)CC1 21767,N1(C(CCSCC)=O)CCN(C)CC1C(=O)NCc1nnn(C)n1 21768,c1(CC)cc(N(C2CNCC2O)C(=O)C(c2ccccc2)N(C)C)nc(C)n1 21769,CC1CC(NC(C2CCN(C(=O)CCC(C)(C)C)CC2CO)=O)CC(C)O1 21770,C(=O)(CC(C)(C#N)C(=O)Nc1nc(CN2CCCC2)n[nH]1)OC(C)(C)C 21771,C12(CCCC1)CNC2C1CC12CC2.c1ccc[nH]1 21772,N1(C(C(C)OC2COC2)=O)CCCC1CNC(c1ccc(F)o1)=O 21773,c1(CCC(=O)NCCCN(C(C(CCC)NC(C)=O)=O)CC)ccc(C)cc1C 21774,C1(CNC(C(C)(C)OC(C)=O)=O)CCC2(CN(C(=O)C(C)C(C)(F)F)C2)O1 21775,c1(C(=O)NCCNC(C2C(C)(C(F)F)C2)=O)ccn2nccc2c1 21776,C=CCCC(C(=O)NCC1(CO)CC2CC2C1)NC(c1ncccc1N)=O 21777,C1(NC(C2(CNC(C(C)N(C)C)=O)CCCO2)=O)CC2(C1)CC(O)C2 21778,c1(C(=O)NC2CN(C(CC=C=C)=O)C(C)C2)ccc(C(C)=O)c(Br)c1 21779,CCC(C(=O)NCC1(OC)CN(C(=O)C(C)c2ccsc2)C1)SCC 21780,C1(CN(C(C2C=CCCC2)=O)C2CC2)C2CN(C(=O)COCC(F)F)CC12 21781,C1(CNC(C2Cc3nccnc3C2)=O)CC2(CCC2)CN1C(=O)Cn1ccnn1 21782,C(=O)(C#CC1CCCOC1)NCC1CN(C(C(C)N(C)C)=O)CC1C(F)(F)F 21783,C1(NC(c2c(CC)occ2)=O)CC2CC1N(C(c1cc(Cl)nn1C)=O)C2 21784,C1(CC(=O)NCc2cccc(F)c2)CC2(C1)CN(C(=O)Cc1cnns1)C2 21785,C1(NC(C(=O)OCC)Cc2ccc(F)cc2)CC(=O)N(C(=O)OC)C1 21786,c1(C(N2CCC(CNC(C(C)OCC(C)C)=O)C2)=O)c2c(c[nH]c1=N)CCC2 21787,N1(C(c2ccn(CC)n2)=O)CC2CN(C(=O)CC(c3cccc(F)c3)C)CC2C1 21788,C(c1cc2c(cc1OC)CC(C)O2)=CC(=O)NC(CNC(C(CC)N(C)C)=O)C 21789,c1(C(=O)NC2C(NC(CCCC(=O)OC)=O)CC2)cn2cc(C)c(C)cc2n1 21790,C=CCC(C)(C)CC(=O)N1CCC(C)(C)C1C(=O)NC1CCNC(=O)C1 21791,C1(C(=O)NC(C2CC2C(N2CCC2(CO)CO)=O)C)COc2ccccc2O1 21792,C1(C(=O)NC2(CCCC(=O)NC3CC4CCC3C4)CCC2)OC2CCC1C2 21793,C12(C(=O)NCC(CC=C)(C)C)CCCC1N(C(=O)COC1CC=CC1)CC2 21794,N1(C(C2(CCC=C)CN(C(C3SCC=C3C)=O)C2)=O)CCC(F)(C#N)C1 21795,c1(NC(C(N2CCC(C(=O)OC)C2(C)C)=O)=O)ccc(N=[N+]=[N-])cc1 21796,CCCCC(O)CC(=O)NC1(COC)CN(C(c2ccc3c(c2)C(C)CO3)=O)C1 21797,N1(C(C(CC(C)C)=O)=O)CCC2(CC1)CC2CNC(=O)CCCc1cccs1 21798,C1(C(N2CC(CN(C)Cc3c(C)ncs3)C2)=O)CC(=O)N(C)C1c1cccnc1 21799,C1(C(=O)NCc2c(C)cn(C)n2)CN(C(=O)C(CO)C(C)(C)C)CC1C1CC1 21800,n1(C(C)C(N2CC=CC(NC(=O)C(C)(F)F)C2)=O)c(S)nc2ccccc2c1=O 21801,c1(NC(=O)CC2CCN(C(c3ccc(Cl)c(F)c3)=O)C2)nc(Br)cnc1Cl 21802,c1(C(N2CCC3(CNC(=O)O3)C2)C(=O)NCCC#N)cn2cc(Cl)ccc2n1 21803,c1(C(N(CCCNC(C(C2CCOCC2)OC)=O)C(C)C)=O)cn(C)[nH]c1=N 21804,c1(OC)cc(F)c(C(=O)NC2CC2NC(c2cccc3c2COC3)=O)cc1N 21805,C1(C(=O)OCC)CC2CSCC(C1)C2NC(=O)Nc1cc2ccc(C)cc2[nH]1 21806,C(=O)(CCN=c1[nH]c(N(C2(CNC)CCCCC2)C)nc2cc[nH]c12)NCC 21807,C(=O)(C1CCCn2nccc21)N1CC2(C(NC(C(CC)OC)=O)CCC2)C1 21808,N1(C(CN(C(=O)CCc2cc(Cl)no2)C)=O)CCN(C(c2ccoc2)=O)C2CC12 21809,C(=O)(C#CC1CCOCC1)NCCCC(C)(C)NC(c1c(CC)n[nH]c1)=O 21810,N1(C(C2CCC(O)C2)=O)CCC(C(=O)NCc2noc(C3CC3)n2)CC1 21811,O=C(CS(=O)(=O)CC1CCCO1)NCC1CNCC2(CC2)C1 21812,N1(C(CC(COC)COC)=O)CCCCC12CN(C(c1cc(O)ncn1)=O)C2 21813,c1(CNC(C(C2CCCOC2)OC)=O)ccc(C#N)s1 21814,N(C(=NCCCCl)NC1CC(=O)N(c2ccccc2F)C1)C(C)CC#N 21815,Cc1nn(C)cc1CC(=O)NCCC1CSCCN1C(=O)CC(C)(C)C1CC1 21816,N1(C(C=C2CCC(C)CC2)=O)CCC(NC(=O)COCCF)C(CO)C1 21817,C1(C(N(C)CC2(C)CCCO2)=O)C2CC1N(C(C1CCOCC1)=O)C2 21818,c1(C(N2CCC(C(=O)Nc3ccc(C)cc3)C2)=O)cc2c(cc1Cl)NC(=O)C2 21819,C1(n2cc(CC=C)nn2)CCN(C(=O)Cn2cc(C(C3CC3)C3CC3)nn2)CC1 21820,C(=O)(C(C1CC1)OC)N(CC(=O)NCC(C1CCCC1)NC(C)=O)CCC 21821,C(=O)(C(c1cccs1)NC(=O)C(C)n1cccn1)N(CCF)CC 21822,c1(SC)nc(Cl)c(CN2CC(C(N3CC(F)C(F)C3)=O)CC(F)C2)c(Cl)n1 21823,N1(C(CCN(CCC)C)=O)CCCC(N(CCF)C(c2cc(CC)oc2C)=O)C1 21824,N1(C(C2(OCC)CCOCC2)=O)CC(NC(c2cnccc2C)=O)CC(O)C1 21825,c1(C(N(C)CC2N(C(C(F)=C(C)C)=O)CCCC2)=O)ccc2c(c1)C(=O)C(=O)N2 21826,c1(N(C(C)=O)C)ccccc1C(=O)N(CC(C)CNC(=O)CC1OCCCO1)C 21827,C(C(CNC(=O)C=C1CCC1)C(F)(F)F)NC(C(CC)(C)OC)=O 21828,N1(C(C(CCC)C)=O)CCCCCC1CNC(=O)CCc1c(F)cccc1Cl 21829,CC(C)CC(O)C(=O)N1CCCC(C(C)C(=O)NCCC(=O)NO)C1 21830,C(=O)(C(C)(O)CC(C)C)NCC(CNC(c1c(C)nc(Br)s1)=O)F 21831,N1(C(c2c(C)nn(C)c2Cl)C(=O)NC2CC(C(=O)OC)C2)CCS(=O)(=O)CC(C)C1 21832,c1(C(=O)NCC(C(C)C)NC(c2c(SC(C)C)cccc2)=O)ccc([N+](=O)[O-])s1 21833,N1(C(C(C)CC2CCCC2)=O)CCCC(O)C1.C12(CC1)C(=O)N2 21834,C(=O)(CCC(=O)N1CC(OCCCNC(C2(C)CC2(F)Cl)=O)C1)NC 21835,c1(C(N2C(C)(CC(=O)N(C)C)CCC2)C2(C(=O)OC(C)=O)CC2)cccc(F)c1N 21836,c1(CN(C(=O)NC2CC3CC3N2C(=O)C(C)(C)C)CC)oc(C)nc1C 21837,c1(CC(N2CCC(C(N=c3[nH]nc(CCC)s3)C)C2)=O)sc2ccccc2c1C 21838,CC(C(=O)NC1CC(NC(=O)C(C)N2CCC2)C1)S(C)(=O)=O 21839,c1(C(=O)NCC(CNC(C2(CCC)CC2)=O)C)cnc(C(C)(C)C)[nH]1 21840,C=CCCCCCCCC(=O)NCCOCCNC(=O)C(c1c(C)n[nH]c1C)C 21841,C=CC(C)(CC)C(=O)NCC1(F)CC(NC(=O)C=CC)C1 21842,CCCCCCN(C(C1CCCCS1)=O)NC(=O)C(C)OCCN(C)C 21843,c1(C(N2CC(CNC(c3cc(Br)no3)=O)C3C2C3)=O)ncc2ccccn12 21844,N1(C(CCNC(COC)=O)=O)CCCN(C(C2CC2[N+](=O)[O-])=O)CC1C 21845,C1(CNC(=O)CC2CCOC2=O)(NC(C2CCSCC2)=O)CC(F)(F)C1 21846,O=C(O)CC1CCCc2ccc(C(=O)NC(c3ccccc3)CO)cc21 21847,C(CCCC(=O)OC)OCC1(NC(C)=O)CCN(C(C2(n3cccn3)CC2)=O)C1 21848,CC1=C(C(=O)NCC2(C)CCC(NC(=O)Cc3cncn3C)C2)COCC1 21849,c1(C(=O)NCC2C(NC(c3ccc(F)cn3)=O)CC2)cccc(F)c1Br 21850,c1(C(N2CC3C(NC(C4(O)CC(F)(F)C4)=O)C3C2)=O)ccc(Br)cc1F 21851,c1(C(N2CC(CNC(c3cncc(F)c3)=O)C(O)C2)=O)coc2c1C(O)CCC2 21852,N1(C(C2CCC(=C)CC2)=O)CC2(CC2)CC1C(=O)Nc1cn(C)nc1C(N)=O 21853,c1(CN2CC(C(=O)Nc3cnc(Cl)cc3I)SCC2)c(F)ccc(Cl)c1Cl 21854,c1(C(=O)NC(CNC(COCc2ccc(C)cc2)=O)CO)cc(Br)c(C)cc1F 21855,C(=O)(CCCN=[N+]=[N-])N(CCC(C(C)C)NC(C1(C)CC=CCO1)=O)C 21856,Cc1cc(NCCCCC(C)NC(=O)C(F)(F)CN(C)C)n2nc(C)nc2n1 21857,N1(C(Cn2cc(C(=O)O)nc2)=O)CCCC2C1CCN2C(=O)C=C1CCC1 21858,Cc1cc(C(=O)N(C)CC2CCN(C(=O)C(F)C(C)C)CC2)ccn1 21859,c1(OC(C)C)ccc(C(=O)NCCN(C)C(C23CCCN2CCC3)=O)c(O)c1 21860,C(=O)(C(C(C)C)n1cccc1)NC(C1CCN(C(c2cc(OCC)no2)=O)C1)C 21861,c1(NCC(N2CCC=C(Br)C2)=O)ccc(-c2nn[nH]n2)cn1 21862,CCS(=O)c1ccccc1C(=O)NC1CC(NC(C2CC2C)=O)C1 21863,N1(C(C2(NC(=O)NC)CCCC2)=O)CC(C)N(C(=O)Cc2cc(C)on2)CC1C 21864,CCC(C)C(C)C(=O)NCCOCCOCCO.C1=CC(=O)N2CC1C2 21865,c1(CC)nc(C(=O)NCCC2CN(C(=O)C(C(C)OC)N(C)C)CCO2)c(N)s1 21866,c1(C(N2C(COC)(CNC(=O)CC(F)F)CCC2)=O)ccn2nccc2n1 21867,C(CCC(C)(C)C(=O)N1CCC2(CC2)C1)NC(c1cnc(C)s1)=O 21868,c1(CN2CC3(N(C(c4ccc(O)cc4)=O)CC3)C2)c[nH]c2ncccc12 21869,CS(=O)(=NC(=O)c1ccc2n[nH]c(Br)c2c1)c1ccncc1 21870,C(CS(C)(=N)=O)NC(C(n1cc(CCC2CCOC2)nn1)C)=O 21871,O=C(C1=CCCOC1)NC(C1C2CN(C(c3ccc(=O)oc3)=O)CC12)c1ccccc1 21872,C1(CNC(c2ccc(NC)cc2)=O)CC(C(=O)NC2(C3CC3)CC2)=NO1 21873,N1(C(C2N(S(CC)(=O)=O)CCCC2)=O)CCOCC(CNC(=O)CCSC)C1 21874,c1(CN2CCC(C)(C(=O)Nc3[nH]nc(OC)c3C#N)CC2)c(F)ccc(F)c1C 21875,Cc1cc(NC(c2ccnnc2C)=O)ccc1NC(c1cc(F)n[nH]1)=O 21876,c1(CN2CC(C)CC(NC(c3ccc(OC(C)C)cc3)=O)C2)c(Cl)ccc(Cl)c1Cl 21877,CC(C)C(C(C)NC(c1cn(C(C)C)cn1)=O)NC(=O)CCC1CCC1 21878,Cn1cc(C(=O)NC2CC(C)(CNC(c3cccc4c3OCC4)=O)C2)ccc1=O 21879,C12(CNC(C3(CCC=C)CC3)=O)CCCC1N(C(c1ccc(F)cn1)=O)CCC2 21880,Cc1ccnc(-n2cc(C(C)N(C(=O)CCc3cn[nH]c3)C)nn2)n1 21881,CC1CCN(C(=O)NC2CC3(C2)CC2(CC2)C3)CCN1S(C)(=O)=O 21882,N1(C(CNC(CC)=O)=O)CCOC(CC(=O)NCC2(O)CCSC2)C1 21883,C1(C2(O)CN(C(=O)C(C)OC3CCOC3)C2)(CNC(C(C2CC2)OCC)=O)CC1 21884,N1(C(CCC(C)C#N)=O)CCC(S(C)(=N)=O)C1 21885,N12CCC(CC1)CC2=O.n1(C(C)(C)C)cc(-c2cn(CCC3CC3)nn2)cn1 21886,CP(C)(=O)CC(=O)N1CCOC(CCNC(=O)CC2CCC(=O)O2)C1 21887,c1(C(=O)NCC2C(C(=O)NCc3c(C)occ3)OCC2)cnc(S)nc1 21888,N1(C(C(CCC)CC)=O)C2CCCC1CN(C(C1(CCCC)CC1)=O)C2 21889,c1(C(N(CC(C(C)(C)C)=O)C(=O)CN2CCC(CO)CC2)=O)ncn2ccccc12 21890,N1(C(C(CCN(C)C)NC(C2C(C)=CCS2)=O)=O)CCCC2(CCCC2)C1 21891,c1(CCC(N2C(C(CNC(C3(CCC)CC3)=O)(C)C)CCC2)=O)cncc(C)c1 21892,C1(NC(C(F)OC)=O)COC2(C1)CN(C(=O)CN(C)C)C2 21893,c1(OC)cc(F)c(C(=O)NCCCNC(C2CCS(=O)(=O)C2)=O)cc1Br 21894,C12(NC(=O)Cc3cnccn3)CCCN(C(C3CC3(Cl)Cl)=O)CC1C2 21895,c1(CC(N2CCC(O)(CNC(c3[nH]cc(CC)c3)=O)C2)=O)cccc2sccc12 21896,c1(C(=O)NCCc2nc(CC)[nH]n2)oc(CNC(C2(OC)CC2)=O)nc1C 21897,c1(C(N2CCCC(C(C)NC(c3nc(C)[nH]n3)=O)C2)=O)cc(C#N)c(C)cn1 21898,C1(CNC(=O)COCC(F)F)CN(C(c2ccc(Cl)cn2)=O)C2CCN1C2 21899,c1(SC)cc(N2CCSCC2CCNC(=O)CC2CCC(=O)N2)nc(SC)n1 21900,N1(C(CN(C)C(C2CCN(C)C2)=O)C(F)F)CCN(C(c2cnnn2Cl)=O)CC1 21901,CC1CC(C(=O)NCC2(F)CN(C(c3c(F)cccc3Br)=O)C2)=NO1 21902,C1(NC(CC2(NC(C(CC)n3ccnc3)=O)CCC2)=O)CN(C)C2(CCC2)C1 21903,C1(CC(=O)NC(CC(C)NC(COCC(=O)OC)=O)C)CCC(=O)N1C 21904,C(C(C)C(F)C(=O)NC(c1snnc1C)C)NC(c1nn(CC)c(O)c1)=O 21905,C1(C2CCN(C(=O)CCCCCn3cnnn3)C2)(NC(c2c(C)coc2)=O)CC1 21906,N1(C(=O)CN2CCOCC2)CC2CC1CN2CCN1CCOC1=O 21907,C(CC(C(N)=O)NC(C1CC1CNC(c1ccc(F)cn1)=O)=O)OC 21908,c1(C(N2CCC(NC(C)C)C(C)C2)=O)ccc2c(c1)CCC(C)(C)O2 21909,N1(C(CNC2CC2)=O)Cc2[nH]nc(C(C)NC(=O)C=Cc3ccccc3)c2C1 21910,c1(C(=O)NCC2(O)CCN(C(c3c(C(C)C)nn(C)c3)=O)C2)cc2n(n1)CCC2 21911,C1(CNC(c2c(CC)ocn2)=O)CC(F)(F)CN1c1nnc(C(=O)OC)s1 21912,C(=O)(CC(C)(C)COC)NC(c1ccc(CNC(C(CC)(C)C)=O)cc1)C 21913,c1(CN(c2coc(Br)c2)CC)cccc(CNC(=O)CNC(C2(CO)CC2)=O)c1 21914,N1(C(c2cnc3cnccn23)C(=O)NC(CC)C)CCc2cc(C#N)ccc21 21915,N1(C(Cc2cc(C)nn2C)=O)CC(NC(C2(n3cc(Cl)cn3)CC2)=O)CC(C)C1 21916,c1(N(C)C)cccc(C(N2CCCCC2CNC(=O)CCC2CCCO2)=O)c1 21917,C(=O)(NNc1nc(C)nc(Cl)c1C)c1cc(OC)cc2c1OCC2 21918,c1(C(=O)NCC(C)(C)O)n[nH]c2c1CCN(C(c1cccc(F)c1O)=O)C2 21919,C1(C)(NC(C(CCC)O)=O)CCN(C(=O)CCC2CC2(F)F)CC1 21920,c1(C(N2CCC(CNC(CN(CC)CC)=O)(OC)C2)=O)c(C)ccc(F)c1N 21921,C1(C(=O)Nc2c(-c3oc(C)c(NS(C)(=O)=O)n3)cccc2)CCCC(=O)N1C 21922,c1(C(=O)NCC2CCC(NC(c3cnnc(Cl)c3)=O)C2)ccc2nn[nH]c2n1 21923,C(=O)(CC(Cl)Cl)N(C)CC=CC(=O)N1CCC1 21924,N1(C(C2CC(C)C2)=O)CC2CCC1(CNC(C1CCC=CCC1)=O)CC2 21925,N1(C(C(C)OC)=O)CCC2(CCCN2C(=O)CNc2cccc(F)c2)C1 21926,CCCCC(C)CCC(=O)N1CC2CC(O)C1C2NC(c1ccoc1Cl)=O 21927,N1(C(C(N2CCC(OCCOCC)C2)=O)=O)CCC(F)(NC(=O)NC)C1 21928,C1(C(=O)NC2CC(N(C(CCNC(C)=O)=O)C)C2)Cc2ccccc2S1 21929,N1(C(c2c(C)noc2C)=O)CCC(CNC(=O)Cc2ccccc2)C(C)C1 21930,Cc1cc(NCCN)n2ncc(C)c2n1.C1(C(C(=O)N)C)CCCCC1 21931,CC1CC(NC(c2ccc(N(C)C(=O)C3CC3)cc2)=O)CN(C(=O)C(F)Cl)C1 21932,c1(C(CC)N(C2CNC2)Cc2ccccn2)ccc(Br)cc1 21933,C1(C(N(CCCNC(Cc2n(C)ccn2)=O)C2CC2)=O)CC2CCCC2C1 21934,CN1CCC2(CCN(C(CCc3ccccc3F)C(=O)NC3CCC3)C2)C1 21935,N1(C(C=CC(C)C)=O)CCC2CC(NC(C3CC(=O)N3)=O)CCC2C1 21936,C1(C)(OCC)CCN(C(C2CC23CC(NC(=O)C(C)C2(O)CCC2)C3)=O)CC1 21937,C(=O)(CCCC(C)(C)NC(c1ccncn1)=O)NC(CCN(C)C)(C)C 21938,C(=O)(C(O)CC(C)C)NCC1(COC)CN(C(=O)CCC2(C#N)CCC2)C1 21939,c1(C2(C)CC2NC(N2CCC(Sc3cccs3)CC2)=O)cccc(Cl)c1 21940,C(=O)(C(=O)CCC(C)C)NC(CCN(C(C(=Cc1ccccn1)C)=O)C)C(C)(C)C 21941,C1(NC(c2cn(C(C)C)nc2O)=O)CN(C(c2c(O)cccc2O)=O)CC1(C)C 21942,C1(C(N2CCCC(CCNC(Cn3c(C)csc3=O)=O)C2)=O)CS(=O)(=O)CCO1 21943,C(CC(C(C)(C)C)NC(c1coc(Cl)c1)=O)N(C(=O)CC1CCOCC1)C 21944,C(=O)(C1=CC2(CCOCC2)C1)NCC1CCC(CNC(CCC2C(C)C2)=O)CC1 21945,N1(C(c2c(OC)cc(OC)nc2)=O)CC2CC(C1)N(C(C1CCC3(CC1)CC3)=O)C2 21946,CC1C(CN(CC(N2CCC(C3(C)OCCO3)CC2)=O)C)CCN1C 21947,N1(C(CC2COCC(C)O2)=O)CCN(C(c2cccc(C(C)C)c2)=O)C(CO)C1 21948,c1(C(=O)NCC2(NC(C(C)OCC)=O)CCOC2)cnn2ccn(C)c12 21949,C(=O)(C1=CC2C=CC(C1)C2)NCCC(C(=O)NC1CC1CC(C)(C)C)OC 21950,CC1(C)CCCC(C(N2CCC3(CC3C(=O)NCCOC(=O)C3CC3)C2)=O)C1 21951,C(=O)(C(C(C)C)C1CCC1)NCC(NOCCCC=C)=O 21952,C1(NC(=O)CSCc2cn(C(=O)OC)nn2)CCCCC1NC1CC1.C1C(=O)N1 21953,c1(CCCC(=O)NC(C)CNC(C2CCC2(F)F)=O)ccc(F)cc1 21954,CN1C(=O)C2CN(C(C3CCN(c4ccnc(Br)n4)CC3)=O)CC2C1=O 21955,c1(C(N2C(C)CN(C(c3c[nH]nc3F)=O)CC2)=O)ccc2c(c1)OCCNC2=O 21956,c1(C(CC(=O)N(CC(CC)NC(=O)CC(C)C)CC)O)ccccc1OC 21957,C1(CC=C)(NC(=O)CC(C=C)OC)CCN(C(=O)C(C)CN(C)C)C1 21958,Cc1cc([N+](=O)[O-])cc(C(=O)NC(C)CN(C)C(C2CC3CC2CC3O)=O)n1 21959,c1(-c2nnn(C)n2)ccc(NC2CCOC(c3ccc(F)cc3)C2)cc1Cl 21960,N1(C(=O)CCC2CCC2)CCC2(CC1)CCN(C(C1(CC3CC3)CC1)=O)C2 21961,C(=O)(N=c1cc(C)n(C2CC2)[nH]1)C1(OC)CCN(C(=O)CC2C=CCC2)C1 21962,N1(C(=O)NCCC(c2ccc(F)cc2)C2CC2)CCS(=O)CC1c1ccccc1 21963,C(=O)(CC(C)C(F)(F)F)NC1C2(C)CN(C(CCC(CC)OC)=O)C1C2 21964,Cn1cnc(NC2CC(CCNC(c3cccc[n+]3[O-])=O)C2)c(Br)c1=O 21965,c1(CC(N2CC(NC(C3C(C)C3C)=O)(CO)C2)=O)ccc(C#N)cc1 21966,C(C(C)C)(C(O)C(=O)NC(C)(CSC)C(=O)NC(c1cccc(C)n1)C)OC 21967,C1(O)(CC(N2CC(C(=O)NCCCOC)(Sc3ccccc3)C2)=O)CCOCC1 21968,N1(C(C(C)c2ccsn2)=O)CCC(CCNC(C2CCCC2)=O)C(F)(F)CC1 21969,C1(CNC(c2c(C)nns2)=O)CCN(C(=O)CN2CCC(=O)CC2)C(C)C1 21970,C1(C(N(CCNC(C(C)SC)=O)C)=O)CCNC(=O)C1 21971,CN=c1nc(N(C)Cc2cncs2)[nH]c(=NC2Cc3ccc(Cl)cc3C2)[nH]1 21972,c1(C(=O)NC(C)CNC(c2conc2C2CCC2)=O)n[nH]c(C2CC2)c1Br 21973,c1(NC(C(=O)NCCNC(c2cncc(OC)c2)=O)=O)ccc(OC)c(OC)c1 21974,C1(NC(C2(C)CCCC2)=O)CCOC(C(=O)NCCCCC2CCCCC2)C1 21975,N1(C(N(C)C)=O)c2ccccc2CCC1C(=O)NCC1CCCN1C1CC1 21976,C1(NC(CC(C)N(C)C)=O)CCC(C)N(C(C2(C#N)CCOCC2)=O)C1 21977,Cc1cc(C(=O)NC2CN(C(c3cnc(C(C)(C)CF)o3)=O)CC2C)nc(O)c1 21978,C1(CC(=O)OCC)CN(C(C(=O)NCCC#N)C2CC2CC)C2(CC2)CO1 21979,C(CC(=O)N(CCNC(C1(n2ccnn2)CC1)=O)C1CC1)=CCC 21980,c1(C(=O)NCCC(C)N(C(C2C(CC)OCC2)=O)C)c[nH]cc(Cl)c1=O 21981,Fc1cc(OCC(Cc2ccccn2)Sc2ccccc2)cc(Cl)c1 21982,N1(Cc2cccc(C(=O)NCc3c(C)noc3C)c2)CCC2(CC1)OC(=O)NC2C 21983,c1(OC)cc(C2(C(=O)NCC#CCNC(=O)CCCSC)CCCC2)ccc1C 21984,c12c(nc3c(CC)cccn13)c(=O)[nH]c1ccccc21.N1(CC(=C)C)CC(C)C1 21985,c1(C(N2CCC(F)(CO)C2)=O)cc2ccc(-c3cccc4c3CCC4)cn2n1 21986,N1(C(c2c(CC)nco2)=O)CC2CCC(N(C(=O)C(C)CC(F)F)C)C2C1 21987,c1(C(=O)NCC2COCCN2C(=O)C2=C(Cl)CC2)noc2c1COCC2 21988,C1(O)(C(N(C(CN(C(c2ccc(OC)s2)=O)C)C)C)=O)CCN(C(=O)N(C)C)C1 21989,C1(CCNC(c2cncc(NC(c3cocn3)=O)c2)=O)CCc2ccccc2C1 21990,C1(CNC(COC)=O)CC2CCC1N2C(=O)Cc1ccc(OC)c(O)c1 21991,c1(CCC(=O)NC2CC(CNC(C3CC(F)(F)C3)=O)C2)ccccc1 21992,c1(CC(=O)NCCN(C(=O)CC2CC2(Cl)Cl)CCC)ccnc(Cl)c1F 21993,C1(CCC)CCCN(c2nnc(-c3ccccc3Cl)n2CCC(=O)N(C)C)C1 21994,N1(C(C(C)(C)OC)=O)CCN(C(c2ccc(F)cc2Cl)=O)C(C(C)C)C1 21995,Cc1ccc(C(=O)NCC2(NC(C3CC(F)(F)C3)=O)CCOC2)nc1O 21996,N1(C(CC(=O)NCC)=O)CCN(C(c2c[nH]c(=N)o2)=O)C(C(C)C)C1 21997,CCC(CCC(=O)NC1(CNC(c2ccc(CC)c(O)c2)=O)CCC1)OC(C)=O 21998,N1(C(c2ncc(CC)cn2)=O)CCCC(O)(CNC(C2CCCC(=O)N2C)=O)C1 21999,N1(CC(=O)NCC(C)N(C(c2ccc(Cl)cc2)C(N)=O)C)CCCCCC1 22000,N1(C(C2C(C(=O)O)C23CC3(F)F)=O)CCc2c(I)n[nH]c2C1 22001,N1(C(CCCCOC)=O)C2CCC1CC(CNC(=O)CC1CC(C)=NO1)C2 22002,CCC(C)C(C(=O)NCCN(C)C(C)=O)NC(=O)C(=O)N(C)C 22003,C12CCN(C(=O)C3CCCN3C1=O)O2.C1(CC(=O)OC)(NC2CC2)CCC1 22004,c1(C(N2CC(CC(=O)NC3C(C(=O)OC)CCC3)C2)=O)cc(C)cc(C)c1 22005,C1(CNC(c2c(CN(C)C)ccs2)=O)CCN(C(c2cnns2)=O)CCC1(F)F 22006,CC(CC(C)(F)F)C(=O)N1CCC(NC(c2cnc3scnc3c2)=O)C1C 22007,CN1CCC2(CC1)CN(C(C1CCN(C(C3(C)CC=CC3)=O)CC1(C)C)=O)C2 22008,c1(C(N2CC(NC(c3cc(-c4ccccc4)on3)=O)C2)=O)csc(O)n1.C1CCC1 22009,c1(-c2ccc(C)s2)ccc(=NC(=O)C2CCC2(C)C)[nH]n1 22010,c1(OC)cc(Br)cc(C(N2CCN(C(C3CC3F)=O)C(CO)C2)=O)c1OC 22011,N1(C(C(C)Cc2ccc(Cl)cc2)=O)CC2CCC(C1)N2Cc1ccc(F)nc1 22012,c1(NC(CNC(C2(SC)CC2)=O)C(C)C(C)C)ncc(Cl)cc1[N+](=O)[O-] 22013,CS(=O)(=O)c1ccc(S(=O)(=O)N2CCOC3(CCC(NC(=O)CN)CC3)C2)cc1 22014,N1(C(c2ccc(C)nc2)=O)CCC(C2CN(C(c3c[nH]cc(Cl)c3=O)=O)C2)CC1 22015,CCN=C(NCCC1CCCCO1)NC1CC(=O)N(C(C)(C)C)C1 22016,N1(C(CCOC(CC(C)C)C)=O)CCC(C2(NC(=O)CN(C)C(N)=O)CC2)C1 22017,c1(CNC)cnn2c1CN(C(=O)CCc1cn(-c3cccc(C)c3)nn1)CC2 22018,C1(C(=O)NCC(C)NC(CC(OCC)OCC)=O)CC(=O)N(C2CC2)C1 22019,c1(C(=O)NCCC(C)NC(Cc2ccc(C)c(F)c2)=O)ccc2c(n1)OCCO2 22020,c1(C(=O)NC2(CC=C)CCN(C(=O)COCC)C2)c(C)nc2ccccn12 22021,C1(Cc2nc(C(C)OCC)nn2-c2c(C)cc(C)cc2Cl)CCCCC12CCC2 22022,C1(C(=O)NC(CC)C)CC(=O)CN1C(=O)C(c1ccccc1)F 22023,C(CCCCC(=O)N(C1CCC(NC(C2CCCC(C#N)C2)=O)CC1)C)OCC 22024,c1(CCNC(C(C2CCC2)NC(c2cc(Cl)n[nH]2)=O)=O)ccncc1F 22025,c1(C(N2C(CCNC(c3cnnc(O)c3)=O)CCCC2)=O)ccc(O)nc1Cl 22026,Cc1ccc(CCN(CCC#N)C(=O)NC(C)CC(F)(F)F)cc1 22027,c1(C(=O)NCC(C)CN(C)C(c2cc(F)c(N)cc2F)=O)cnc2[nH]cncc1-2 22028,C1(C(C)(C)O)CCCN(C(=O)C(N2CCNCC2)C2CC2)C1 22029,C(=O)CC(C)(C)C(C)(F)F.N1(CC)CCC(c2cn(CC(F)(F)CO)nn2)CC1C 22030,c1(C(=O)NC2C(NC(c3c(C)nn[nH]3)=O)CC2)cc(Br)c2ccccc2c1 22031,c1(CNC(C(C2CCCCC2CN)CC)=O)ccc(Cl)c(Cl)c1C 22032,Cc1cc(C)c(NC(C2CCCC(NC(=O)Cc3ccccn3)C2)=O)c(C)c1 22033,N1(C(C2N(C(C(C)=CC3CC3)=O)CCN(C)C2)=O)CCC2CCC(C1)N2C 22034,CCCC(C)(C)C(=O)NCC(C)(O)CNC(=O)CSc1ccc(C(C)C)cc1 22035,C1(Cc2nc(C)sc2)CCN(N2CCOCC3(CC3)C2)C1 22036,N#CC12CCC(C(=O)NCC3CCN(C(C4CC5(CC5)CO4)=O)CC3)(CC1)CC2 22037,N1(C(C2C(OC)CCC2)=O)CC2CC2(NC(c2cncc(-n3ccnn3)c2)=O)C1 22038,c1(C(N2CCN(C(=O)C3=CSCS3)C(CF)C2)=O)ccc2oc(S)nc2c1 22039,Cc1cnccc1C(=O)NC(C1CN(CC2CCC(C)O2)C1)C 22040,c1(C(=O)NCC23C(CN(C(C(CSC)C)=O)C2)C3)cccc(=O)n1C 22041,C1(CNC(c2ccc(Br)o2)=O)C2CN(C(C3CC4CCC3O4)=O)CC12 22042,Cc1cc(C(=O)NC(C)(CNC(=O)C2=CCC2)C2CC2)nn1C(C)C 22043,CCC1=NOC(CC(=O)NC(CCC2CC2)C(=O)NCC(C)C(=O)NC)C1 22044,C1(CNC(C(C)c2cccs2)=O)CCN(C(=O)CCS(N)(=O)=O)C1(C)C 22045,Cc1ccc2c(N3CCn4ncnc4C3)nc(=NCCCCC(N)=O)[nH]c2c1 22046,C12CCCCN1C2=O.c1(N(C(=O)C(F)=CC2CC2)CC)ccnnc1C 22047,C(=O)(C(C(C)C)N1CCCCC1)NCCN(C1CCCC1)C(C1CC(C)C1)=O 22048,CC(C)(C(=O)N1CC(C2CN(C(=O)Cc3ccon3)C2)C1)C1=CCSCC1 22049,C#CCC(C(=O)NCC(C)Cn1cccn1)NC(=O)Cc1cccnc1O 22050,C1(C(=O)NCC(C)C2CCC2)CCN(C(c2c[nH]c(=O)cn2)=O)C1(C)C 22051,C1(C)(C(=O)NCC2N(C(CNC(C)=O)=O)C3CCC2C3)CC(C(C)(C)C)=NO1 22052,Cc1cccc(C(=O)N(CC(C)NC(=O)CSCc2ccccc2)C)n1 22053,N1(C(C2CC3(CCN(C(C(C=C)C)=O)C3)C2)=O)CCCC2(CCCC2)C1 22054,C(=O)(C1=CNS(=O)(=O)N=C1C)N1CCCC(NC(C(CCC)=CCC)=O)C(F)C1 22055,Cc1ccc(C(=O)NC(C2CN(C(=O)C(C)c3cccs3)C2)C)nc1C 22056,C1(N(C(C=C(CC)CC)=O)C)CCN(C(C2CC(c3cccc(F)c3)C2)=O)CC1 22057,Cc1cncc(C)c1C(=O)NC1(CC=CC(N2CCC(CC3CC3)C2)=O)CCC1 22058,C(=O)(C(CC(C)C)N(C)C)NCC(CCC)NC(=O)CCc1ccc[nH]1 22059,N1(C(C(CNC(CSCCC)=O)CC(C)C)=O)CC(C)OC(C)(C)C1C 22060,c1(NC2CC=C(C)CC2)ccc(S(=O)(=O)N2CCCCC2C(C)CO)cn1 22061,N1(C(C2C(=C)CC2)=O)CC2CC(NC(c3ccc(NC(C)=O)cc3OC)=O)C1C2 22062,N1(C(c2c(C)c(F)ccc2Cl)=O)CC2CC3CC2C1C3NC(c1ccn(C)c1)=O 22063,Cc1ccn2ncc(C(=O)NC3CC(C)N(C(=O)CCCc4ccsc4)C3)c2c1 22064,c1(CCNC(c2cccc(NC(=O)NC)c2)=O)c[nH]c2cc(F)c(Cl)cc12 22065,CCC(C)(CNC(c1ccnc(C)c1C)=O)C(=O)NC1(CCF)CCC1 22066,N1(C(CNC(C2CC(SC)C2)=O)=O)CCN(C(C2CC2F)=O)CC1 22067,CC1CC2(CCN(C(=O)CC3CCCC3)CC2)CN1C(=O)CCCCC(C)(C)C 22068,Cc1cnn(C(C)C(=O)NC2CCC2NC(c2ccn(C3CCCC3)n2)=O)c1 22069,C1(O)(CC=C)CCN(C(c2conc2CNC(C2CC(=O)C2)=O)=O)CC1 22070,c1(C(N2C(C(=O)Nc3cc(O)nc(O)n3)CC3CC32)=O)ccc([N+](=O)[O-])cc1O 22071,n1(C(C)C)cnc(C(=O)NC(c2ccnn2C)C(=O)NCC2(C)CC2(C)C)n1 22072,c1(C(N2CC(O)(C(C)NC(C3CCOC3)=O)C2)=O)coc2c1CCCC2 22073,C1(C(N(CCCN(C)C(=O)C2CC2)C)=O)CCC2(CCOC2)O1 22074,CN1CCN(C(c2ccsc2C#N)=O)CC1C(=O)NCC1CCCC(C)(C)C1 22075,C(=O)(CCCC(=O)N1CCN(C(=O)CC2CCCSC2)C(C2CCC2)C1)N(C)C 22076,C1(c2cn(-c3ccn(C(C)(C)C)n3)nn2)COCCC1OCc1ccccc1 22077,c1(CSCCC)ccc(C(=O)NC2(CNC(C3CCOC3)=O)CCOC2)o1 22078,c1(C(CC(=O)NCC(CC=C)NC(=O)C=CO)NC(C)=O)ccc(F)cc1 22079,Cc1oc(-c2ccc(F)cc2)nc1CC(=O)NCCC1CCC(O)CC1 22080,c1(N2CCC(C(=O)OCC)(NC(=O)OC(C)(C)C)C2)c(Cl)cc(SC)cc1Cl 22081,C(CC1C=CCC1)(C(=O)N(C)C)c1onc(C(c2ccccc2)(C)C)n1 22082,C(=O)(CCCCC#N)N1CC(C(=O)NCCCC(=O)OC)C(C(C)C)C1 22083,C(CNC(=O)CN(C)C(C)C)(CCNC(=O)CCc1nccn1C)OC 22084,c1(C(=O)NC2CN(C(C3(CC)CCOC3)=O)CC(F)C2)c(O)ccc(F)c1F 22085,C(c1c(C)coc1C)=CC(N1CC(O)(C(C)NC(C=C(C)C2CC2)=O)C1)=O 22086,Cc1ncccc1C=CC(=O)NC1(CCCNC(c2nccn2C)=O)CC1 22087,c1(NCC(C)(C)C2CCC2)[nH]c(=NCCc2ccn(C(F)F)n2)nc2scnc12 22088,N1(C(CNC(NCC)=S)=O)CC2(C1)CN(C(C1CCC(=O)N1)=O)CC2CO 22089,C(C(C(=O)NC1CCCCC1)N1CCC2CCC12)(C1CCCC1)OCC 22090,c1(OCC)c(C(=O)NC2CCN(C(c3ccc(C)cc3O)=O)C2)cccc1F 22091,C1(CCNC(=O)Cc2nnc(-c3ccco3)o2)(NC(COC)=O)CCCC1 22092,CC(=O)C(C)CC(C)C(=O)N1CCC(C)(C)CC1C(=O)NCC(C)(C)C 22093,c1(-c2ccc(F)c(C)c2F)cccc2c1CCN(C(C1C3COCC13)=O)C2 22094,C1(CNC(=O)CCN2CCC2)CCN(C(C23CC(C(F)F)(C2)C3)=O)CC1 22095,CN1CCOC(C(=O)N(C2CC2(C)C)CCOC(C)(C)C)C1=O.C(=O)OC 22096,Cc1cccc(C)c1C(c1ccccc1)NC(=O)C(N1CCC(C)C(CO)C1)=O 22097,c1(CCC)nc(CCCNC(N2CCCC2CC(C)(C)C)=O)cs1 22098,C(C(C)(C)CC(=O)N(C1CC(C(N2CC3CCC3(C)C2)=O)C1)C)OC 22099,c1(OC)cc(Br)c(CNCC2COCCN2C=O)cc1O.c1ccc(F)c(Cl)c1 22100,C1(CC=C)(NC(c2cnc(C(F)F)s2)=O)CN(C(c2cc(C(F)F)cs2)=O)C1 22101,Cc1cc(C)c(CN2CCC(N(C(=O)C(C)C)C)C2)cc1C 22102,c1(CC)ncc(C(=O)NC2CCCN(C(=O)CCC#CC)C2CC)c(C)n1 22103,c1(C(N2CCC(C)C2)=O)onc(-c2ccc(F)cc2)c1-c1ccccc1 22104,C1(C(N2CCC2c2cn(-c3cnnc(O)c3Br)nn2)=O)CC2CC1CN(CCO)C2 22105,Cc1cccc2c1CCC2NC(c1cnc2n1C(C)CCC2)=O 22106,N1(C(COC)=O)CC2CCC(C1)N2Cc1c(C(F)(F)F)cccc1F 22107,CC(C)CC(CNC(=O)CC1CCC(=O)C1C)C(=O)NCC(C1CC1)N(C)C 22108,Cc1cc(C(=O)NCCc2ccn(C)n2)nn1C(C)(C)C 22109,c1(C(N2CC(N(C(C3CN(CC(C)C)C3)=O)C)C2)=O)ccc2c(O)ncnc2c1 22110,c1(C(=O)NCC2CC(NC(c3occ4c3CCCC4)=O)C2)ccnc2[nH]cnc12 22111,c1(C(=O)NCCCCC2CN(C(C(C(C)O)(F)F)=O)C2)cc2ccsc2n1C 22112,c1(CNC(C(C)N(CC)CC)=O)ncoc1C1CN(C(C2CCCS2)=O)C1 22113,N1(C(Cc2cc(CC)no2)=O)CCC2(CCN(C(C3CCC(C4CC4)C3)=O)C2)C1 22114,C=C(Cl)CCC(=O)NCC1CCN1C(c1ccnn1C(CC)CC)=O 22115,C(=O)(C1CCc2nccn21)NC(C)C(C)(C)C(=O)NCc1ccnc(O)c1 22116,C(CC(C(=O)Nc1cn[nH]c1)NC(=O)C(CCC(C)(C)C)OC)OCC 22117,C1(CC)CN(C(C2(O)CC3(CCOCC3)C2)=O)CC2(CCCOC2)O1 22118,C12(NC(C(C)=CC3CC3)=O)CCC1CN(C(c1ccsc1C)=O)C2 22119,Cc1cc(NC(C)CC(C)NC(=O)Cc2c(F)cccc2F)n2nc(C)nc2n1 22120,C(=O)(CS(=O)(=O)N1CCOCC1)NCCCN(C(=O)C(C)N1CC(C)C1)CC 22121,c1(N(C2CC3(CCNCC3)C2)C(C2(F)CCCOC2)=O)ncc2[nH]ncc2n1 22122,c1(C(CC)C(=O)NC2CCC2NC(c2sncc2C)=O)ccc(Cl)cc1 22123,CC1CCC(NC(=O)Cc2cn[nH]c2)CN1C(c1ccc(O)nc1Cl)=O 22124,Cc1cc(NC(C23CC2CN(C(c2ccno2)=O)C3)=O)c(F)c(Br)c1 22125,C1(NC(C2C(=C)C2)=O)COC2(C1)CN(C(c1cccc3nncn13)=O)C2 22126,N1(C(c2c(NC(COC)=O)cccc2)=O)CCC(NC(=O)C(C)OC)C(CO)C1 22127,C1(CC(=O)N(CC(CC)NC(=O)Cn2cnc(C)n2)C)CCCCC(=O)N1 22128,c1(CNC2CCC(C(=O)NCc3ccn(C)n3)CC2)c(Br)ccc(Cl)c1F 22129,N1(C(C(C)C#N)=O)CCC2(CC(NC(=O)C=Cc3ccccc3F)C2)C1 22130,c1(C(=O)NC2(C(=O)OC)CC2(C)C)cc(Br)ccc1Cl 22131,C(=O)(CS(=O)CCC(F)(F)F)N1C2(CNC(CC=CCC)=O)CCC1CC2 22132,c1(C2C(C(=O)NCCCC(C)NC(=O)CCC(=O)OC)C2)c(F)cccc1F 22133,N1(C(C(CCCC)C)=O)CCC2CCCC12C(=O)NCC1CC2(CCC2)C1 22134,c1(C(=O)NC2CN(C(C(C=C)(C)CC)=O)CC2(C)C)cnc2onc(C)c2c1 22135,C1(C(N(CCCNC(c2c(OC)nsc2)=O)C2CC2)=O)CCSC(C)C1 22136,Cc1cnc(C(N2CCCC(CN(C)CCc3cnn(C)c3)C2)=O)cn1 22137,c1(CC(N2C(NC(CC3CN(C)C3)=O)CCC2)=O)ccc(OC(C)(C)C)cc1 22138,C(C)(C(=O)N1CCC(N(CCO)C(C2CC(C)C2)=O)CC1)(C(C)C)OC 22139,C(CCN=c1cccc(S(=O)(=O)NC(c2ccc(C)s2)C)[nH]1)SCC 22140,C(=O)(CCCCC(=O)NOC(C)(C)C)N1CCC(C(=O)NC2(C)CSC2)(OC)C1 22141,C(=O)(C1=CCCOCC1)NC1CCCC(CC(=O)NOCCCC2CC2)C1 22142,Cc1cc(C)c(CNC(=O)C(c2ccoc2)NC(c2cccc(O)n2)=O)cn1 22143,c1(C(N2C(CN(C(c3ccc(CC)o3)=O)CC)CCC2)=O)c(C)nnn1CC 22144,C1(NC(C2(SC)CC(O)C2)=O)CC2CCC(C1)N2C(=O)CCCCSCCC#N 22145,N1(C(c2nc(C(C)C)oc2)=O)CCC(NC(C2(C(F)(F)F)CC2)=O)C2CC12 22146,C1(C(=O)NC(C(C)NC(c2cc(C)n(C)c2C)=O)C)CN(C)CCN(C)C1 22147,N1(C(c2c(C)snc2)=O)CCC(NC(=O)CC(C)c2cccnc2)C(F)(F)CC1 22148,C1(C(=O)NCc2ccc(C)cn2)CCCCC1(C)NC(=O)C(C)OCCN(C)C 22149,c12cc(ccc1C)C(=O)NOC2.CCCCS(=O)(=O)NC(=O)CC(C)C(=O)OC 22150,C#Cc1ccc(C(N2CCCC(CCN(C)C)C2)C(=O)NCC)cc1OC 22151,c1(CC)conc1C(=O)NC1(c2nnc(C(C)C)s2)CCOC1 22152,N1(C(c2c(CNC(CCC(C)OCC)=O)nnn2C)=O)CCCC12CCCC2 22153,Cc1ccc(SCC(=O)NCC(C)N(C(=O)CCCNC(C2CCC2)=O)C)cc1 22154,c1(C(N2CC(N3CCC(OCCCCC)CC3)C2)=O)ccc2nonc2c1 22155,N1(C(Cc2ccn(C)n2)=O)CC(F)CC1C(=O)NC(c1nn[nH]n1)C1CC1 22156,C1(N(CCOC)C(c2ccncc2)=O)CCN(C(=O)C(C)(C)n2cccn2)CC1 22157,c1(NC(C)=O)cccc(C(N2CCN(Cc3nc(-c4nc[nH]n4)no3)CC2)=O)c1 22158,C1(CNC(=O)C(=O)NCC(F)(F)F)CCC(Nc2cccc(F)c2)CC1 22159,C1(Nc2ccc(COC(C3CCOCC3)=O)cc2)CCC2CC1CN2 22160,c1(C(N(C2CCN(C(C3CC3COC)=O)CC2)CC)=O)ccc2c(c1)CC2 22161,c1(SC)cc(NC23CCC(NC(=O)C(C(C)C)SC)(C2)OC3)nc(SC)n1 22162,c1(C(N2C(C)C(C)N(C(=O)CN3CC4CC4C3)CC2)=O)cccc2c1CCC2=O 22163,c1(C(=O)NC2(C(N3CC(C)(CC=C)C3)=O)CCCCC2)cnc(C)c(C#N)c1 22164,N1(C(Cc2ccc(C)s2)=O)CCN(C(=O)C=Cc2ccoc2)C(C)C1C 22165,C(=O)(C(CC=C)C(C)C)N1CC(CC#C)C(C(=O)NCC(C)(O)CC)C1 22166,C(=O)(C(C)CCCC(C)C)NC(C=CC(N1C(CO)CC(OC)C1)=O)C 22167,c1(CC(=O)N(C)CCNC(c2cnccc2Br)=O)cc(S(N)(=O)=O)cn1C 22168,C1(NC(c2cc(C#N)no2)=O)CN(C(=O)C(Cl)=CCl)C2(CCCCCC2)C1 22169,c1(C(=O)NC(C(C)C)CCNC(=O)CC2NC(=O)NC2=O)ccc2[nH]ccc2n1 22170,N1(C(C(CC)N(CC)CC)=O)CC2(C1)CN(C(C1(C(F)F)CCCC1)=O)C2 22171,C1(C(=O)NCC(O)CNC(=O)Cn2ccnc2)(SC)CCOCC1 22172,c1(C(N2CCCC(c3cn(C4CCOC4)nn3)C2)=O)cc2scc(Cl)c2[nH]1 22173,C1(NC(COCC)=O)CCN(C(c2cc(C)n(-c3nccs3)c2C)=O)C(C)C1 22174,c1(NC)cnc(C(N2CC3C(C(=O)NCCn4ccnc4)C3C2)=O)cn1 22175,N1(C(CC2CCN(C)C2=O)=O)C2CCC1CN(C(=O)C1=CCCS1)C2 22176,C12(CNC(C(C=C)O)=O)CC3CC(CC(C3)C1NC(=O)CCC(=O)N(C)C(C)C)C2 22177,CCCCCC(C)CC(=O)NCC1CCC2(CN(C(C3CC(C)(CC)C3)=O)C2)O1 22178,CN1CCOc2cc(CN3CC4CC3CN4C(c3ccc(O)cc3Br)=O)ccc21 22179,N1(C(c2cc(C(=O)OC)on2)=O)CCC2(CC(NC(c3cc(C)ns3)=O)C2)C1 22180,CC1OCCCC1C(=O)NCC1(CNC(c2cccc(OC(F)F)c2)=O)CC1 22181,C1(O)(CN(C(c2c(C)con2)=O)C)CCN(C(=O)C(C)c2ccco2)C1 22182,C1(C)(C(N(C2CCC(OC)C2)C)=O)CCN(C(=O)CCc2cnc(C)o2)CC1 22183,N1(C(CCn2ncc(C)c2)=O)CC(CNC(C2CCC(=O)NC2)=O)CC(C)(C)C1 22184,C(C(CNC(C1C(C)C1C)=O)CO)NC(CC1(OC)CC1)=O 22185,CC1c2cc(C(=O)NCCC3CCN(C(c4cnco4)=O)CC3)ccc2OC1C 22186,N1(CC)CC(C(=O)NC23CC2CN(C(c2cc(F)cs2)=O)C3)CCC1=O 22187,C1(NC(C2(CC#C)CCCO2)=O)COCCN(C(C2CCCCS2(=O)=O)=O)C1 22188,c1(CN2CC(F)(C(=O)NCCc3ccc(OC)cc3)C2)cc(F)cc(Br)c1Cl 22189,C(=O)(CC(F)(F)C(F)F)N1C(CNC(CCc2onc(C)n2)=O)CCC(C)C1 22190,N1(C(c2c(SC)csc2)=O)CC2CCCC2(NC(C2OCCC2(C)C)=O)C1 22191,N1(C(CC=C)=O)CCC(NC(c2ocnc2C2CC2)=O)C(C)C1 22192,Cc1cn(C2CCN(C(=O)C(=O)NCCCCN3CCC(C(=O)O)C3)C2)cn1 22193,C(C(=O)N(C1CCC(NC(=O)CN2CCC3CC23)CC1)C)(C(C)(C)C)NC(C)=O 22194,C1(CNC(CCN2CCC(C)CC2)=O)CC2(CC2)CN1C(=O)CCCC#N 22195,S(=O)(=O)(CC(=O)NC1(C)CC(C(=O)NC2CC23CCC3)C1)NCC 22196,N1(C(C(C)NC(=O)NC)=O)CCN(C(=O)C(C)=C(C)C)CC1CC1CC1 22197,Cc1cc(C(N2CCOCC2CS(C)(=O)=O)=O)ccc1C#N 22198,N1(C(c2c(CC)oc(C)c2)=O)CC(Nc2ncncc2Cl)CC(F)C1 22199,C(=O)(C(C)S(C)(=O)=O)NCC(N1CCN(C(c2c(OCC)nccc2)=O)CC1)C 22200,c1(C(=O)NC(C2CN(C(CC3C(C)CCO3)=O)C2)C)c(F)ccnc1Cl 22201,C1(S(C)(=O)=O)(C(=O)NCC(CN(C(C2CC(O)C2)=O)CC)(C)C)CC(O)C1 22202,c1(C(=O)NCC2CC(F)CN2C(C2CCCC23CC3)=O)cnn2cnnc2c1 22203,Cc1nc(CCNC(c2cccnc2-n2nccn2)=O)c(C)o1 22204,c1(CC)c(C(N2CCN(C(CNC(=O)C(C)O)C(F)F)CC2)=O)nnn1CC 22205,C1(N(C)C(C2CCOC2)=O)CCCN(C(c2cc(O)ccc2Br)=O)CC1 22206,C(=O)(C(O)CCC(F)(F)F)N1C(CN(C(=O)CCc2ncc(C)[nH]2)CC)CCC1 22207,C1(NC(C2C(C)(C)C2)=O)CC(NC(=O)CNC(N)=O)C12CCC2 22208,N(C1CCCn2ccnc21)C(C(CCNC(c1ncc[nH]1)=O)OC)=O 22209,CC(C)C(CC(=O)N1CC(N(C)C)C1)NC(C1CCC(C2CC2)C1)=O 22210,C1(NC(CC(CCC)O)=O)CCCCN(C(c2cccc3cnsc23)=O)CC1 22211,c1(-c2nn(C(C3(C)CC3)C)c(COC(F)(F)F)n2)ccc(F)c(Cl)c1 22212,C1(CCNC(Cn2ccc(C)n2)=O)CCN(C(C2CC2C(C)(F)F)=O)CC1 22213,C1(C(=O)NCc2ccnnc2O)CC2CCCC2N1C(C1CC12CCCC2)=O 22214,N1(C(CC2(CSC)CC2)=O)CC2CCN(C(c3cncc(O)c3)=O)CC(C2)C1 22215,C1(C(=O)NC2N(C(N)=S)CCC2)CC2(CCN(S(=O)(=O)C3CC3)CC2)C1 22216,c1(CC(=O)NCC(C)CNC(=O)Cn2cnc(C#N)n2)cc(F)ccc1F 22217,c1(N2CCC(C)C(CO)C2)nc2cc[nH]c2c(=NCC2CSC2)[nH]1 22218,N1(CC(=O)NCC2CCC2NC(C2C3CNC(=O)C23)=O)CCN(C2CC2)C1=O 22219,CC#CC1CCN(C(=O)CC2CCCC2NC(=O)C(O)C(C)(C)C)CC1 22220,C1(CC(=O)NC2CCN(C(c3cnc(C(=O)OC)s3)=O)C2)CCN(CCF)CC1 22221,N1(C(C(C2CC2)OCC)=O)CCC(C)(NC(=O)Cc2ccn(C3CCCC3)n2)C1 22222,c1(OC)cccc(F)c1C(=O)NCC1CN(C(=O)Cc2csc(C)n2)CCC1C 22223,C(=O)(C(O)CC(F)(F)F)NCC1N(C(CSc2nc(C)[nH]n2)=O)CCCC1 22224,C1(CCCNC(c2c(CC)noc2)=O)CCCCN1C(=O)C=CC1CCOCC1 22225,c1(C(=O)NCC(CNC(C2CC(C#N)C2)=O)F)nc2ncccn2n1 22226,C1(CC(N2CCCC2)=O)(C(=O)OC)CCN(C(=O)CC2CCCS(=O)(=O)C2)CC1 22227,Cc1c(C(N2CCOC(C(=O)NCC(C3CCCC3)C)C2)=O)cnn1C 22228,C1(NC(C(C)n2cnnn2)=O)CCCCCN(C(c2cn3ccnc3cn2)=O)C1 22229,c1(OC)ccc(C=CC(=O)NC2CCCCC2CNC(C2CC2C)=O)c(OC)c1 22230,Cc1cc(NC(=O)N(C2CC2(F)F)C)cc(F)c1Br 22231,Clc1cc2c(cc1CNCCCc1cn[nH]c1)OCCO2 22232,c1(C(=O)Nc2ncc(C(F)F)c(C(F)(F)F)n2)cccc2c(Cl)c(Cl)sc12 22233,c1(NC(N(CCC(C)(C)C)CCOC)=O)ccnc(Br)c1 22234,N1(C(C2CC(=C)C2)=O)CC(CNC(c2ncccc2C(C)=O)=O)C(O)C1 22235,C1(NC(CN(CC(C)(C)C)C)=O)(CNC(=O)C=CC(F)(F)F)Cc2ccccc2C1 22236,C12(CNC(=O)COCC3CCCCO3)CC1CN(C(c1cc(CO)on1)=O)C2 22237,Nc1cc(C(=O)NCC(c2cccc(Cl)c2)NC(c2csnc2Cl)=O)cc(F)c1 22238,N1(C(C2(COC)N(C(C(C)SCC)=O)CC=C2)=O)CCN(C)C(C)C1 22239,CCC(CCC(=O)N(C(C)CC(N)=O)C)NC(C1(C)CCCCC1)=O 22240,C#Cc1cccc(C(=O)NCC2COC(CNC(=O)C(C)(C)c3ccsc3)C2)c1 22241,C1(C(N2CC(NC(C(C)OCC=C)=O)C2)=O)CCC(=C(F)F)CC1 22242,CCCCC(CNC(C1(C(N2CCCC2)=O)CC1)=O)NC(=O)C=C1CCN(C)CC1 22243,c1(OC(C)C)cc(C(N2CCN(C(C3CC3(C)C)=O)CC2C)=O)cc(Br)c1 22244,c1(C(C(=O)NCC2CCCO2)N(C)CC2(C(=O)OC)CC2)n[nH]cc1C 22245,N1(C(c2cc(C(C)C)no2)=O)CCC(C(C)(C)C)(CNC(=O)C(C)C(F)F)C1 22246,c1(CN2CCC3(CN(C)C3)C2)ccc2c(C(=O)O)n[nH]c2c1 22247,c1(C(N(C(CNC(c2ccc(CNC(C)=O)o2)=O)C)C)=O)occ2c1CCOC2 22248,CON1CCC(NC(C2(NC(=O)COCC3CCOC3)CC2(C)C)=O)CC1 22249,c1(C(=O)NC2CC(NC(C3(CC)CCNC3=O)=O)C2)cn2cccc(Br)c2n1 22250,c1(C(N2C(CN(C(CCCC)=O)C)CCCC2)=O)cnc(C2CC2)[nH]c1=N 22251,Cc1cc(CCNC(=O)C(=O)NC2CC(N(C)C)C2(C)C)c(C)s1 22252,CC(Cn1ccnc1)C(=O)NC1C=CCC1 22253,C(=O)(CS(=O)(=O)C(C)C)N1CCC(N(C(=O)CCn2ccnc2C)CC#C)CC1 22254,N1(C(c2ccn(C3CC3)n2)C(=O)NC(CC)C)CCc2c(cc(C#N)n2C)C1 22255,C1(CC(=O)NCC(C)(CO)NC(=O)C=CC2CCC2)CCCCCCC1 22256,CC(c1ccc(F)cc1)=CC(N1CC(NC(c2c[nH]nc2[N+](=O)[O-])=O)C(C)C1)=O 22257,N1(C(c2ccc(C)o2)=O)CCCC2CN(C(c3cc(N)ccc3C)=O)CCC12 22258,C(=O)(C1=CC2CC(C1)CC2O)NC1C2CN(C(c3ccc(OC)cc3C)=O)C1C2 22259,C1(C(N(C)CCOCCN(C(=O)C(F)(F)c2cscn2)C)=O)CCCC(F)C1 22260,CC1CC(C2CN(C(c3ccoc3CNC(C3(O)CCOC3)=O)=O)C2)=NO1 22261,C1(C(=O)NC(C2(O)CCN(C(=O)C(C)(C)N(C)C)C2)C)CCC(=C(F)F)CC1 22262,N1(C(C(CC)=O)=O)CCC2CN(S(=O)(=O)c3ccccc3F)CC2CC1 22263,CC1(C(=O)NC2C3CC(NC(C4C5CCCCC45)=O)CC23)CCC2(CC1)CC2 22264,c1(OC)nc(C(N2CCCCC(NC(=O)CN3CCSCC3)C2)=O)ncc1F 22265,c1(C(=O)NCC(c2ccccc2F)(F)F)c[nH]c2cc(Cl)ccc12 22266,N1(C(C(C2CCCCC2)NC(c2cn(C)c(=O)cc2)=O)=O)CC2(C)CC1CCO2 22267,Cc1cnccc1C(C)C(N1CC(NC(=O)CCc2cncnc2)CC1C)=O 22268,CC1(F)CN(C(C2CC(N3CCC3)C2)=O)CCN(C(C2(C(F)F)CC2)=O)C1 22269,N1(C(C(C)C2CCCO2)=O)C(CNC(c2n[nH]cc2Cl)=O)CC2COCC12 22270,c1(C(=O)NC(CC=C)(C)C(F)F)n[nH]c2c1CN(C(c1nnn(C)c1CC)=O)C2 22271,N1(C(CN(C(C)C)C)=O)CCC2(CC2NC(=O)COC2CCCCCC2)C1 22272,CC1(C)CC(O)CCN(C(c2cc(F)cs2)C(=O)NC2CCOCC2)C1 22273,c1(C(C(=O)NCCSC)N(C(=O)C=C(C)C(=O)OC)CC)ccccc1 22274,c1(NC(C)=O)ccc(C(=O)NC2COCC2NC(=O)CCc2cncs2)cc1 22275,N1(C(C(CO)OC)=O)CCC(NC(=O)C2=C(Cl)CCC2)C1(C)C 22276,N1(C(C(C)N(C(=O)CC2OCCO2)C2CC2)=O)CC(CO)C(O)C1 22277,C1(CC)CN(C(=O)C=CC(C)NC(C2(C)COCCO2)=O)CC1F 22278,n1(C(C)C)cc(Br)cc1C(=O)NC(C)CCNC(C1(O)CCSC1)=O 22279,Cc1c(C(N2CC3CN(C(=O)CCC(C)(C)C)C3C2)=O)cccc1O 22280,c1(C(=O)NC2C(C)CN(C(=O)C(F)(F)CC3CCCO3)C2)c(N)cccc1Cl 22281,c1(C2(C(=O)NCC3C(CNC(C(C)N(C(C)=O)C)=O)C3)CC2)ccc(C)cc1 22282,CCCCC(C(=O)NC(c1csc(C)n1)C)NC(C1CC(C)(O)C1)=O 22283,C1(C(=O)OC)(NC(C)C(c2ccccc2)NCc2ccccc2)CC(C)(C)C1 22284,CCC(C)CC(C(=O)NCCOCCC1CC1)NC(=O)C1=CCOC1 22285,N1(C(Cc2cccc(OC)n2)=O)CCC(C)(C)C(NC(c2ccc(F)cn2)=O)C1 22286,c1(-c2scc(C(C3COC(C)(C)O3)c3ccc(F)cc3)n2)ccc(Cl)cc1F 22287,Cc1ccc(C)c(CNC(C2CC(O)(CNC(=O)C(O)Cc3cnc[nH]3)C2)=O)n1 22288,CC(C(C)C(=O)N1CCOCC1C(C)O)NC(=O)C(C)CC1CCCC1 22289,Cc1cc(C(=O)N(C)CCNC(c2cn(C)nc2C(F)F)=O)[nH]c1C 22290,c1(CC(=O)NC2COCCN(C(=O)C(F)CC3CCC3)C2)nc2c([nH]1)CCCC2 22291,Cc1cc(NC(=O)C(C2CCOCC2)O)ccc1NC(=O)C(C1CCC1)N(C)C 22292,C1(C(=O)NCCCOCCNC(C(C)Cn2ccnc2)=O)NC(=O)OC1C 22293,N1(C(Cn2cc(C(C)O)nn2)=O)CC(NC(c2cccn2C)=O)C2CCCC12 22294,C=CCC(CNC(=O)C(C)OCC1CC1)C(=O)NC1(CO)CC2CCCC12 22295,N1(C(C2CCN(CC)CC2)=O)CCC2(CC1)CC(N1CCC(F)(F)CC1)C2 22296,c1(C(=O)OC)cc(C(=O)NCC(O)CNC(c2sc(N(C)C)nc2C)=O)c(C)o1 22297,C(C(F)(F)CN(C(=O)CCCN(C(=O)C(O)CN1CCCC1)C)C)OC 22298,c1(C(=O)NC(C)CN(C(=O)C=Cc2c[nH]cn2)C)cc2c(Cl)cc(Cl)cc2[nH]1 22299,CC(C)C(C)C(CNC(c1cccc(N2CCCC2=O)c1)=O)NC(=O)C=C(Cl)Cl 22300,OC1(F)CCN(C(=NCC2(O)CCCOC2)NCC2CCCCO2)CC1 22301,C1(NC(C2C(CC)C2)=O)COCCN(C(c2cc(C)nnc2O)=O)C1 22302,c1(OC)cc(C)c(C(=O)NCC2CN(Cc3cc(Cl)ccc3C)C2)c(C)c1 22303,Cc1nn(C)c(C)c1C(C)C(N1CCCC(CNC(=O)C#CC2(C)CC2)CC1)=O 22304,Cc1cc(CCC(=O)N(C(C)CCNC(=O)C=CC2CCCO2)C)n[nH]1 22305,c1(N(C2CCCN(C(CCC(C)C)=O)C2)CCO)nc2cc(Cl)cc(Cl)c2o1 22306,CC(C)(CO)C(=O)N1CCC(CCC(N2CCC(O)C2)=O)C1 22307,CC1(CNC(C2CC3CCC3C2)=O)CCN(C(=O)Cc2ccc(CO)cc2)C1 22308,CC1CN(C(c2ccc(OCCF)cc2)=O)CC1NC(=O)CCC1CC1(Cl)Cl 22309,C1(NC(C(COCC)C)=O)CN(C(c2cc3ccccc3[nH]2)=O)CC(C)(C)C1 22310,c1(OC(c2c(Cl)ccc(OC)c2)=O)ccc(S(C)(=O)=O)cc1Cl 22311,n1(CC(=O)NCC2CC2NC(C2CC2c2cccc(Cl)c2)=O)cccnc1=O 22312,C12(C(=O)NCCCc3cc(C)no3)CCCC1CCN2C(c1cc(O)cs1)=O 22313,c1(C(=O)NCCCNC(c2nnn(C)n2)=O)ccc(O)c(Cl)n1.C1C=CC1 22314,C(=O)(C(C(C)C)C(C)C)N(C)CC1(C)C(NC(C(C(CC)O)C)=O)CCC1 22315,N1(C(Cc2c(C(C)C)cccc2)=O)CC2CC(CNC(=O)C(C)(O)C3CC3)C2C1 22316,c1(C(=O)NCC(C2CC2)NC(C(OC)OC)=O)ccc2cccnn12 22317,C1(C(=O)NC2(CO)CCCN(C(=O)CCCC3CC3)C2)(OC)CCS(=O)(=O)C1 22318,N1(C(CCCC(C)O)=O)CC(NC(c2coc(C3CCC3)n2)=O)CC2(CC2)C1 22319,N1(C(c2cn(CC)nc2C)=O)CC(NC(=O)Cc2ccns2)C(N=[N+]=[N-])C1 22320,Cc1ncnc(N2CC3CC3(CNC(c3cc(F)ccc3Cl)=O)C2)c1Br 22321,C(c1cncc(O)c1)=CC(=O)NCC(CNC(c1ccc(CCO)cc1)=O)OC 22322,CC(=Cn1ccnn1)C(=O)NN=c1[nH]ccnc1-c1ccccc1 22323,c1(CCC)ccc(S(=O)(=O)N(CCO)Cc2ccsc2)cc1Br 22324,Cc1nn(C)c(C)c1C(C)NC(c1nnnn1C1CCCCC1)C1(C)COC1 22325,C1(NC(c2ncn(CC)c2)=O)CCCC(NC(=O)Cn2nnc(C3CC3)n2)CC1 22326,N1(C(C(CCC=C)(F)F)=O)CCC2C(CCCN2C(=O)CC(F)(F)Cl)C1 22327,C1(C2CC2)(CNC(C(C)OCCOCC)=O)CCN(C(C2CC3(CC3)C2)=O)C1 22328,CC1OC2(C(=O)NCC3CC4CC4N3C(=O)Cn3cnnc3O)CC1C2 22329,c1(C(=O)NC2C(OC)CN(C(c3cn(C4CC4)nn3)=O)C2)ccc(F)cc1O 22330,N1(C(C=CCC)=O)CC2C(NC(=O)CCSc3ccccn3)C2C1 22331,C=CC(C)(C)CC(=O)NC1CCCN(C(C2CCC(c3nc[nH]n3)O2)=O)C1 22332,Cc1c(C(N2CC3CC2C3C(=O)Nc2csc(C(F)(F)F)n2)=O)cccc1F 22333,N1(C(c2c(C)nc(C(C)C)s2)=O)CC(NC(c2ccnc(CO)c2)=O)C2CC2C1 22334,C=CCC(CC(=O)NCC1(CCC)CCC1)NC(=O)CCCF 22335,C(=O)(CS(=O)(=O)N(CC(F)(F)F)C(C)(C)C)N(CC(C)NC(=O)C(F)CC1CC1)C 22336,N1(C(C(c2cn(C)nn2)NC(C2CC(C#C)(O)C2)=O)=O)CCC(O)C(F)(F)C1 22337,c1(C(=O)NCC2CC(NC(c3cccnn3)=O)C2)cnc(S)nc1 22338,C12(CNC(COCC#C)=O)CCC(CC1)N2C(C1(C)CNC(=O)C1)=O 22339,n1(CCC)c(C)cc(C=C(C#N)C(=O)NCC2CCNC3(CC3)C2)c1C 22340,N1(C(=O)CS)CCC(CNC(=O)C=Cc2ccccc2)C(O)C1.C1COC(=O)C1 22341,c1(C(=O)NC2CC(NC(=O)CNC(c3ccsc3)=O)C2)ccc2c[nH]nc2c1 22342,N1(Cc2ccc(OC(C)C)cc2)CC2C(CCNC)(C1)C(F)(F)C2(F)F.C(C)C 22343,N1(C(C2N(CC)CC2)=O)CCC(NC(C2CCC2(C)C)=O)C(F)C1 22344,N1(C(C(C)n2ccnc2)=O)CCCN(C(=O)C2=CCCS2)C(c2ccccc2)C1 22345,C1(O)(CNC(CCN(C(=O)C2=CCOCC2)C)=O)CC2CCC1C2 22346,C1(C(=O)NC2CCCOC2)C=CCN(C(=O)C(O)CC2CCCC2)C1 22347,C(=O)(C(C(C)(C)O)NC(c1cccn(C)c1=O)=O)NC(C(=O)OC)CO 22348,c1(N2CCCC3(CC(NC(CCC(C=C)(C)C)=O)C3)C2)nc2ncc(Cl)cc2s1 22349,N#Cc1cc(F)c(CN2CCSCC2C(=O)NCc2ccc(F)c(Cl)c2)c(Cl)c1 22350,Cc1ccc(CC(N2CCCC(O)(CNC(=O)C(C(C)O)N(C)C)C2)=O)cc1C 22351,N1(C(c2c(SCC)nn(C)c2)=O)CCN(C(=O)C(C)(F)CCC)CC12CCC2 22352,C(=O)(CCC(CC)OC)NC(CC#C)C(=O)NCCC1CCOCC1 22353,n1(CC)cc(CC(=O)NC(C(=O)NC(CO)C2(O)CC2)C2CCOC2)cn1 22354,CC(C1CCCCC1)=CC(=O)NC1CN(C(=O)CCOC2CC2)CCC1C 22355,c1(C(=O)NC2CCC(CNC(C(n3ccc(C)n3)(C)C)=O)C2)cccn(C)c1=O 22356,C(=O)(C(C(=O)NC1CC2(C(=O)NC3CCOCC3F)COC1C2)C(C)C)OCC 22357,n1(CC(=O)NC2CC(C)(NC(C(CC)O)=O)C2)nc(-c2ccccc2)oc1=O 22358,c1(CNC(c2cnc(S)nc2)=O)ccc(C(=O)NCCC(O)CCO)cc1 22359,c1(CNC2CC(C(=O)NC3(CCC)CCNC3=O)OCC2)ccc2n[nH]cc2c1 22360,N1(C(C(CC#C)(C)NC(=O)CCC#CC)=O)CC2(CNC(=O)C2)C1 22361,N1(C(CC(C)OC)=O)CCC(O)(CN(C(=O)CCCN(C)C(C)=O)C)CC1 22362,C1(C(=O)NC(CC)C(C)(F)F)CN(C(=O)C(C)O)CC1C1CC1 22363,c1(C(=O)NCCN(C(=O)CC2COC3CC2C3)C2CC2)cc([N+](=O)[O-])ccc1Cl 22364,C(C(C)(C)CN=c1ccnc(N2CCOC(C3CCCO3)C2)[nH]1)OCC 22365,CC1(C)CN(C(=O)C=CC=CCO)CC(CNC(=O)CC2CC3(CCC3)C2)O1 22366,Cc1ncc(Cl)c(C(N2CC3C(CN(C(=O)C(C)(C)O)C)C3C2)=O)n1 22367,N1(CC2(F)CCN(C(C3(CCC=C)CC3)=O)CC2)CC(C)N(C)CC1C 22368,c1(C(N2CC(C(=O)NCc3ccc(OC)nc3)C(C)C2)=O)cccc(C#N)c1 22369,c1(C(C)=O)cc(S(=O)(=O)NC)c(C)o1.N12C(=O)CCC1NC2 22370,C(=O)(C1=CC2CCCC12)N(CC(CNC(c1n[nH]c(CC)c1Br)=O)(C)C)C 22371,C1(CNC(C(CC)(C)C)=O)C(O)C(O)CN1C(=O)C=Cc1ccnn1C 22372,c1(CC)nn(C)c(C(=O)NC2C3CN(C(=O)CCS(=O)(=O)N(C)C)CC23)c1Cl 22373,c1(C(=O)NC2C3CN(C(C4(CF)CC4(F)F)=O)CC23)cccc2cnccc12 22374,C1(C2CC2)(C(=O)NC2C(C=C)COC2)CN(C(=O)CC23CCC(CC2)C3)C1 22375,C1(C(N2C(c3n(C)ncc3)COCC2)=O)CCc2nnc(C(F)F)n2C1 22376,N1(C(CNC(C(C)(C)C)=O)=O)CCC2CCCC12C(N1CCCC(C)(CO)C1)=O 22377,Cc1nsc(N)c1C(=O)NC1CCCC(CNC(C2(CO)CC2)=O)C1 22378,C1(CCCNC(=O)CSc2cccnc2)CCCCN1C(c1cccnc1)=O 22379,c1(CC(N2CCC(N(C(CC(CC)SC)=O)C)C2)=O)c(F)cccc1Cl 22380,C1(CC(=O)NCC(C23CCC(CC2)C3)NC(c2ccon2)=O)CCCNC1=O 22381,CC1CN(C(C2(c3ccccc3Br)CCC2)=O)CCN1C(C1C=CCCC1)=O 22382,C1(C)(C(=O)NCC(CNC(CCn2ncc(C)c2)=O)(C)O)COCCO1 22383,C(CNC(C1(c2ncco2)CC1)=O)(CC(=O)N1CCOC(C2CCC2)C1)OC 22384,N1(C(C(CC)OC)=O)CCOC(C(=O)NCC2(F)CC(CO)C2)CC1 22385,CCC(C(=O)OC)C(=O)NC1CC=C(C(=O)NCCc2nc(C)no2)C1 22386,c1(NC(CC(=O)N2CCCC2)c2cccnc2)ncnc2[nH]cc(Cl)c12 22387,Cc1ccc2c(C(=O)NCC3CC3NC(c3cc(N(C)C)ccn3)=O)n[nH]c2c1 22388,C1(COC)(CNC(=O)CC#N)CCN(C(c2ncccc2C)=O)C1 22389,c1(C(=O)NCCC2(O)CN(C(C34CCCC3CC4)=O)C2)cnc2n1CCOC2 22390,S(=O)(=O)(c1ccc(C2CC2)s1)N(C(=O)C(N)Cc1ccc(Br)cc1)CC(=C)C 22391,N1(CCCC)CCCC(NC(c2ccc(C(C)C)cc2)C(N)=O)C1 22392,C(=O)(C1=CNC2=NCCCC2=C1)N1CC(CNC(C(C(=O)OCC)(C)C)=O)C1 22393,c1(OCOC)cccc(C(=O)NC(C)CNC(=O)C(F)C(C)C)c1 22394,Cn1cc(C(N2CCC(CNC(c3nocc3C3CC3)=O)C2)=O)nc1C(F)F 22395,N1(C(c2c(C)cc(C)s2)=O)CCCC1C1CCCN1C(=O)CCN(S(C)(=O)=O)C 22396,c1(C(N(CC(C(=O)NC(CC=C)(C)CC=C)C)C)=O)ccc2cccnn12 22397,C(=O)(C1=C(Cl)CCC(C)C1)NCC1(NC(C2CCCC(C(=O)OC)C2)=O)CCC1 22398,C1(NC(CC2CN(C)C2)=O)CCCC(NC(=O)C=Cc2cccc(F)c2)CC1 22399,c1(CC)nc(=N)[nH]c(=NC2C3CC2CN(C(=O)C(C)SC)C3)[nH]1 22400,CC(C(=O)NCC=CCNC(c1cnc(N)c(-c2ccccc2)c1)=O)C(C)(F)F 22401,N1(C(c2cn(CC)nn2)=O)CC2(CCC2NC(=O)CC2CC3(CC3)CO2)C1 22402,Cc1ccc(C2(C(N3CCC(NC(=O)CCC4CC4)C3)=O)CCOCC2)cc1 22403,C(=O)(C(CC(F)F)C1CCC1)NCC1C(NC(c2n(CCC)ncc2)=O)CC1 22404,CC1=C(C(=O)N(CC(=O)NC2N(C)CCCC2(C)C)C(C)(C)C)C(=O)OC1(C)C 22405,CC1CC(NC(=O)C(C)(C)N2CCOCC2)CCN1C(C1C(F)(F)C12CC2)=O 22406,C1(NC(CCOCC)=O)CN(C(=O)C=CC2CCOC2)CC12CC2 22407,c1(CC)c(C(=O)NC2CCCCC2NC(=O)C=NOC)cccc1C 22408,c1(C(=O)NC2CC3CC(NC(CCCSC)=O)CC32)ccc2c(c1)ncn2C 22409,C1(NC(C(N2CCOCC2)C)=O)CN(C(C2CC2c2ccccn2)=O)C(C)(C)C1 22410,c1(C(N(C(CNC(C2C(OC)C2)=O)C)C)=O)ccc(-c2ccccc2)[nH]1 22411,N1(CC)CCC(NC(C2CCOCC2NC(C2CC2Cl)=O)=O)C1=O 22412,C12(NC(CC3(OC)CC3)=O)CCCC(NC(=O)CCc3nccn3C)(C1)C2 22413,C(=O)(C(CC)C(C)(C)CC)N1CC2=C(CN(C(C(CC)OC)=O)C2)C1 22414,C(=O)(C#CC(C)(C)C)NCCNC(CC(C)c1ccncc1)=O 22415,N1(C(CSC)=O)CCC2(NC(=O)CC3CCCC3C)CCCC12 22416,N1(C(C2(C)CC(C)C2)=O)CCC(C2(O)CN(C(C3C4COCC34)=O)C2)CC1 22417,c1(CC)cc(F)ccc1CC(=O)N(C(C)CNC(c1sccc1C#N)=O)C 22418,C1(NC(=O)CC2=CCCC2)CCC2(CCCN2C(C2COC2)=O)CC1 22419,c1(CSc2nc3ccc(C(=O)OC)cc3o2)nc2ccc(Br)cc2n1C 22420,C1(F)(C(=O)NCC2C(NC(=O)Cc3sc(O)nc3O)C2)CS(=O)(=O)CC12CCC2 22421,c1(CNC(C(C2CN(C(=O)CN3CC4CC4C3)C2)OC)=O)cn(C)cn1 22422,c1(OC(F)(F)F)cccc(CNCc2c[nH]nc2C(F)(F)F)c1 22423,n1(CC)nc(C(=O)NC(CCF)C(N2CCCC(C(N)=O)C2)=O)cc1C 22424,N1(C(CC=C=C)=O)CC(CCNC(c2ccnc(Cn3cnnc3)c2)=O)OC(C)C1 22425,C1(C(N2CCC(C(C)C)(CO)C2)=O)C2CCC(C2)N1C(=O)C(C)(C)C 22426,N1(CC)CCCCC1C(=O)NCC(CNC(c1cn(CCC2CC2)nn1)=O)CO 22427,Cc1[nH]ccc1C(=O)NCc1cn(CCNC(=O)CC2COCCO2)nn1 22428,N1(C(C2N(C(C)(C)C)CC2)=O)CCC(NC(c2cnn(C3CC3)c2Cl)=O)C(F)C1 22429,C1(NC(c2c(COC)cco2)=O)CCN(C(=O)C(CSC)OC)C(C)C1 22430,c1(Cn2cc(CCCNC(c3c(CC)ocn3)=O)nn2)ncccc1C 22431,Cc1cc(C)[nH]c(=NCC2(NC(c3cccn4c(O)nnc34)=O)COC2)n1 22432,C1(CC(=O)NCC(C)(C)NC(c2cncc(COC)c2)=O)NC(=O)CNC1=O 22433,CC(N=c1[nH]c2ccccc2s1)C1CCN(C(C2CC23CC3)=O)C1 22434,CCCCC(O)CC(=O)NC1(CO)CC(O)C1.c1(CC)cn(C(C)C(=O)O)nn1 22435,n1(CC)cc(Cl)cc1C(=O)NC1(CNC(C23COCC(C2)C3)=O)CCCC1 22436,c1(C(N2CC3C(NC(c4c(OC)ccs4)=O)C3C2)=O)cc(Br)cc2cc[nH]c12 22437,c1(C(N2CCOCC2)C(=O)NC2(CNC(=O)Cc3ccccc3)COC2)cc(Cl)cs1 22438,CCS(=O)c1ccccc1C(N1CCN(C(c2cc(C)cs2)=O)CC1)=O 22439,C(=O)(CC1CCOc2ccccc21)NC1C2(CC(NC(C(C)(C)C(N)=O)=O)C2)C1 22440,N1(c2nnc(CCOC)s2)CCC(CNC(C2CCCN2C(C)C)=O)CC1 22441,Cc1ccc2c(=NCCCC3CC3)[nH]c(=NC3CC4CC4C3)[nH]c2c1 22442,N1(C(C2CC(C)(C)C2)=O)CC(CNC(=O)CC2=CCCCC2)C2(CCOCC2)C1 22443,c1(OC)ccc(NC(C(CCC)OC)c2nnnn2CC2CCCO2)cc1SC 22444,N1(C(C(CC)(C)C)=O)CCC(NC(=O)Cc2cc(Cl)ccc2O)C(C)C1 22445,c1(C(=O)NCCCC(C)(C)NC(c2c(C)nn(C)c2)=O)cnn2c(N)ccnc12 22446,C(=O)(C(=O)C(C)(C)C)N(C(C(=O)Nc1ccsc1)C1CC1c1cccc(I)c1)C 22447,N1(C(=O)CN2CCOCC2)CCCC(CCC(=O)NCC23CC(CO)(CO2)C3)C1 22448,c1(CCC(=O)NCC2(OC)CN(C(=O)C(C)CO)C2)ccc(C#N)cc1 22449,C(C(CC(C)C)C(=O)N(C(C)CCNC(c1cnc(Cl)n1C)=O)C)OC 22450,Cc1cc(N2CCC(C(C)NC(C3CCCC(O)C3)=O)C2)c(Br)cc1[N+](=O)[O-] 22451,c1(C(=O)NC2(CCNC(=O)CCF)CC2)c(Cl)ccc(Br)c1F 22452,C12(NC(CN(C)C)=O)CCCCCC1N(C(c1coc(Br)n1)=O)CC2 22453,Cc1cnn(C)c1C(N1CC(CCNC(=O)CCC=CBr)C1)=O 22454,C1(C(C)C)CCC(C(=O)Nc2cccc(C(N)=O)c2)N1C(=O)CN1CCOCC1=O 22455,CC1(C)CCc2n[nH]cc2CN1C(=O)NCC1CCCCS1(=O)=O 22456,c1(OC)cc(CCCNCC(C)(C)C2(O)CNC2)cc(F)c1 22457,c1(-c2c(C)c(N3CCn4c(C)cnc4C3)ncn2)cccc2c1OCCO2 22458,CC(C)(O)CC(=O)NCCn1ccc(C(=O)NCC2(CC3CC3)CCC2)c1 22459,Cc1cc2nc(NCC3(O)CCCN(C(C4(C)CC(C)(C)C4)=O)C3)cc(=O)n2o1 22460,N1(C(CC2(COC)CC2)=O)CCC(F)CC1C(=O)NC1CCC(C)(C)CC1 22461,C1(NC(C(=O)NC(c2ccccc2)CC=C)=O)CCCCC1N1CCOCC1 22462,N1(C(c2cc(C)oc2C)=O)CCC2(CCC(NC(C3CC(F)(F)C3(C)C)=O)C2)C1 22463,C1(NC(=O)Cc2cccnc2Cl)C2CC(CN(C(=O)C=CC(=O)N(C)C)C2)C1CO 22464,N1(C(C)C)CCCC(C(N2CCCCC2CCNC(C2OCCC2(C)C)=O)=O)C1 22465,C(=O)(C(C)CC(F)F)N1C(CCNC(c2c(C)[nH]c(=N)s2)=O)CCCC1 22466,C(=O)(C(C)CC(C)(F)F)NC(CCNC(CCc1ccc(OC)cc1)=O)C(C)C 22467,C(CCCC(C)C)NC(C(C1CCN(C(c2c(C)scn2)=O)C1)(C)C)=O 22468,C1(C(=O)NCCC(=O)NCCCNC(C23CSCC2C3)=O)(CO)CCCCC1 22469,c1(C(=O)NC(C)C(=O)Nc2cncc(-c3ccco3)c2)nc2ccccc2s1 22470,N1(C(c2c(C)cc(SC)o2)=O)CC(NC(c2coc(C)n2)=O)CC1(C)C 22471,C1(CC)(NC(=O)CC(O)C2CCCC2)CN(C(C2(NC(N)=O)CC2)=O)C1 22472,c1(CC(C)C(=O)NCC2CCN(C(=O)COCCO)CC2)ccc(O)c(O)c1 22473,c1(C(N(CCN(C(=O)C(=O)NCCC(N)=O)CC)CC)=O)cccc(CC)c1F 22474,N=c1ncn(CC(=O)NCCC(O)CNC(=O)CCn2cc(Cl)cn2)[nH]1 22475,C1(NC(C2(N(C)C)CCCC2)=O)CN(C(=O)CC2CCC23CCC3)CC1C(F)F 22476,c1(N2CC(C(C)O)OCC2)ncnc2c1ncn2CC1CCC2(COC2)O1 22477,CCC(CC)(CC)C(=O)N1CC(C)(c2cn(-c3ccc(C(C)(C)C)cc3)nn2)C1 22478,CCC(CC)CC(=O)NCC12CC1CN(C(=O)CC1(C)CC1(F)F)C2 22479,C12(C(N3CCC(C)(NC(c4c(CC)noc4)=O)C3)=O)CCOC1CC(=O)NC2 22480,C(=O)(C(COC)OC)NC1(C(N2C(C(=O)OC)CC2)=O)CSC1 22481,C12=NC3=NC(CCCN1C(=S)NCC(F)F)C(=C(CCC)C(C)CCCN2C)N3 22482,c1(C(C)C)ncncc1C(=O)NCC1CC(NC(=O)CC(C)C2CC2)C1 22483,N1(C(CC2(N(C)C)CCC2)=O)CCOCC(NC(c2cc(Br)no2)=O)C1 22484,c1(OCC(N2C(C)CCC(C(=O)OC)C2)=O)ccc([N+](=O)[O-])cc1 22485,C1(N(C(=O)C=CBr)C)CCCCN(C(=O)C(C)(C)c2cnn[nH]2)C1 22486,C1(CNC(C)=O)CCCN(C(C2(n3cc(CC(C)O)nn3)CC2)=O)C1 22487,c1(C(=O)NCC(C)(C2CC2)NC(c2ccc(CC)[nH]2)=O)ccc(=O)n(C(C)C)c1 22488,c1(CCC(=O)NCC2(C(=O)OC)CC2(F)F)cccc(F)c1Br 22489,C1(NC(C(=CC2CCCC2)C)=O)CN(C(=O)C(Br)=C(C)C)CCC12CCC2 22490,N1(C(Cc2c(C)n[nH]c2)=O)CC(CNC(=O)CCC2CCCO2)C(C)(C)C1 22491,C(=O)(CC(C)(C)C(=O)N1CC2C(CNC(C3CCS(=O)CC3)=O)C2C1)OCC 22492,O(NC(=O)C(F)C(C)CNC(C1C2(CC2)C12CC2)=O)C(CC(C)C)C(=O)O 22493,c1(NCC)ncc(C(=O)NCC2CCC(C(=O)OC(=O)C#CC(C)C)C2)cc1Cl 22494,c1(CC(=O)NCC2CC(O)(NC(C(COC)NC(C)=O)=O)C2)c(O)ncnc1O 22495,c1(C(=O)N=c2cc(-c3cccc(Cl)c3)o[nH]2)csc2ccc(F)cc12 22496,CCCC(C)CC(=O)NC(C)C(C)NC(c1onc(OC)c1Br)=O 22497,c1(OCC)cccnc1C(=O)NCCC(C)N(C(=O)C=Cc1ccc[nH]1)C 22498,C1(C)(CNC(C(CC)O)=O)COCCN(C(c2cc(F)c(O)c(Cl)c2)=O)C1 22499,c1(C(N(C)CC2CCCC2NC(=O)Cn2ccc(C(F)(F)F)n2)=O)nsnc1O 22500,N1(C(CC2CC(C)C2)=O)CC2(CNC(c3cnn(C)c3Cl)=O)CC1CO2 22501,C(CN=C(NC1CCS(=O)(=O)C1)N1CC2C(C)C2C1)OCC(=O)OC 22502,c1(C(=O)NCC(CO)NC(C(C2CC2)OC)=O)c[nH]c(=N)nc1C 22503,c1(C(=O)NC2(C)CC(C(N3CCCN(C(C)=O)CC3)=O)C2)cc2ccccn2c1 22504,CC(C)CC(O)C(=O)NC1(C(=O)NC2CCCCCC2C)CC1(C)C 22505,CC(CC(C)(C)C)C(F)C(=O)NCC1C2CN(C(=O)Cn3ncnn3)CC12 22506,N=c1[nH]c2cccc(C(=O)NC3C4CN(C(c5cscc5Cl)=O)CC34)c2o1 22507,C(CC1C(=O)N1)OCC=C.C(C)(C)(C)OC(=O)N(CC(C)C)C 22508,CCCCCC(O)C(=O)N1CC=CC1CNC(=O)CNC(C1CCC1)=O 22509,c1(CC(=O)NC2CCCC2Cn2cc(-c3ccncc3)nn2)ccc(F)nc1F 22510,C(=O)(C1CCCn2cnnc21)N(CCC(C(C)(C)C)NC(C)=O)C 22511,C1(C(=O)NCc2cn(-c3cncc(C(F)(F)F)c3)nn2)(OCC)CC2CCC1C2 22512,c1(-n2ncc(C)c2)cncc(C(=O)NC(C2CNCCN2C)c2ccccc2)c1 22513,C1(C(=O)NCc2n(CC)nnc2C)N(C(=O)C(C)n2cccn2)CCCC1(C)C 22514,c1(C(N2CC(C(Cn3cc(COC)nn3)F)C2)=O)ccc2nc(Cl)nn2c1 22515,c1(C(=O)NCC2CCCN(C(C(CC)C(=O)OC)=O)CC2)ncnc2c1CCC2 22516,c1(-n2c(CCC#C)nc(C(C)CCC)n2)ccc(S(=O)(=O)N(C)CC)cc1 22517,N1(C(CC(C)=C(C)C)=O)CC2CC(CNC(C3(C4CC4)CC3)=O)C2C1 22518,N1(C(c2n[nH]c(C)c2O)=O)CCC(C2CC2)(CNC(=O)COc2ccccc2)C1 22519,C1(C(=O)NCC(CC)C)CC(C)CN(C(C2CCC(O)CN2C)=O)C1 22520,N1(C(CN(C(=O)COCC2CCCO2)CC#C)=O)CC2COC(=O)C2C1 22521,N1(C(CC2CN(C(C(CC#C)C3CC3)=O)CC2C)=O)CCCSCC1C 22522,c1(C(N2CCC(O)(CCNC(CSCC=C)=O)C2)=O)cccc(C(N)=O)c1F 22523,c1(C(C)SCC)nc(-c2ccc(C(C)C)cn2)n(CC2CCSC2)n1 22524,C1(C)(NC(CCCNC(C)=O)=O)CCCN(C(=O)CC2CCCC2(F)F)C1 22525,N1(C(CC(C)(C)C)=O)CCC2CN(C(c3cc(F)cc(F)c3O)=O)CCC2C1 22526,C1(C(=O)Nc2cnc(Br)s2)CCN(Cc2ccc(OCCO)cc2)CC1O 22527,C(C(O)(C(F)(F)F)c1ccccc1)NC(C(C)(C)Oc1ccccc1)=O 22528,N1(C(c2c(CCC)n[nH]c2)=O)CC=CC(NC(c2cnco2)=O)C1 22529,Cc1cc(C)n(CCC(=O)N(C)CC2CCN(C(=O)C(C)N(C)C)CC2)n1 22530,C(=O)(CS(=O)(=O)Cc1cccs1)NCC(C)NC(C1CSCC(=O)N1)=O 22531,c1(C(=O)NCC2CN(C(C(CC)=CCCC)=O)C2)cncc2ncccc12 22532,C(CCC)(C(=O)N(C1CCN(C(=O)CCn2cccc2)C1)CC)=CCC 22533,c1(-n2cc(NCC3CCCN(C(C(COC(C)C)O)=O)C3)nn2)ccc(C)c(Cl)c1 22534,Cc1cc(C)n(CC(N2CCC(N(C)C(c3cccc(CS(C)=O)c3)=O)C2)=O)n1 22535,C1(C(=O)NC(C(=O)OC)C)CN(C(c2ccc(COC(C)=O)s2)=O)CCC1O 22536,N1(C(C(F)=CC)=O)CC(C)N(C(c2ccc(-c3cscn3)cc2)=O)CC1C 22537,O=C(C1=CC2CCCCC12)NC1C2CN(C(c3ccc[n+]([O-])c3)=O)CC12 22538,N1(C(c2scc(OC)c2)=O)CCC(C)(CNC(=O)CC(C)(C)C)C1 22539,N1(C(c2ccn(CCNC(C3(CC)CCC3)=O)c2)=O)CC(S(N)(=O)=O)C1 22540,CC1(CNC(=O)CC2CCCCC2)COCCN(C(C2CC3CC(=O)C2C3)=O)C1 22541,N1(C(CSCC)=O)CC2CCCC2(CNC(=O)C2=NOC(c3ccccc3)C2)C1 22542,c1(CNc2scc(-c3ccc(C)cc3)c2)cc(F)c(I)c(F)c1 22543,N1(C(c2c(C)nsc2)=O)CC(NC(c2ncc(Cl)c(N)c2Cl)=O)CC2(CCC2)C1 22544,C(CN=c1[nH]cc2ncnc-2[nH]1)=CCNC(CC(CC)OC)=O 22545,C1(C(=O)NC(CC)C(N)=O)CCN(C(C2CC(=O)NC2(C)C)=O)C12CCC2 22546,C1(N(C)C(c2cc(Cl)c[nH]2)=O)CN(C(C2COC(=O)N2)=O)CCC1O 22547,C1(N(C(=O)C(O)C2CN(C(C3CCCC3F)=O)C2)CC)CCCCC1 22548,CC(C)CCCC(C)CCNC(=O)N(C(C)(C)C)Cc1ccc(Cl)cc1 22549,c1(C(=O)NCCC2(O)CCN(C(=O)CSC(F)F)C2)cnn2ncccc12 22550,C(=O)(C(C)(O)COC)NC1CC(C)(NC(c2ccc(CC)cc2)=O)C1 22551,c1(C(N(CCCNC(=O)C(C)C(F)F)CC)=O)cc2c(cc1N)CCCC2 22552,C1(C(=O)NCCC(N)=O)CCC(NC(=O)Cc2cccc(Cl)n2)CO1 22553,Cc1cc(NC(=O)C(C)CNC(=O)Cc2cnccc2C)c(C)c(C)c1 22554,N1(C(C2(C)CCCO2)=O)CCOC2(CCN(C(c3cc(C4(C)CC4)n[nH]3)=O)C2)C1 22555,C1(C(=O)NCC=C2CCSCC2)(NC(C(c2cncnc2)C)=O)CC(O)C1 22556,O=C(CCCCCl)NCc1ccc(CNC(c2cccc(O)c2)=O)cc1 22557,c1(CN2C(C(=O)Nc3nnc(C)o3)CC(F)C2)c(C)[nH]c2ccccc12 22558,c1(CN2CC(C(=O)NCC34CC(C3)C4)C2)cc(O)c(O)c(O)c1 22559,C1(C(N(C(CCNC(c2nc(C)sc2)=O)C)C)=O)CCC(C)CC1 22560,c1(C(=O)NC2(CNC(c3csc(-c4cccs4)n3)=O)CC2)ncc[nH]c1=O 22561,C1(NC(c2nccc(CC)c2)=O)CC2CC1N(C(c1ccc(F)c(N)c1)=O)C2 22562,c1(SC(c2nc(-c3sc(Cl)nc3Cl)no2)C)ccc(=O)n(-c2cccc(Br)c2)c1 22563,C=CCC(CNC(=O)CC1(C#N)CC1)C(=O)NC(C)Cc1nncn1C 22564,C(=O)(C1=CC2(CCOCC2)C1)NCC(C)CNC(=O)C(CO)C(C)(C)C 22565,C(C(C)(C(=O)N(C(C)CCNC(c1n[nH]c(C)n1)=O)C)OC)OC 22566,N1(C(c2ccc(C(F)F)c(C)c2)C(=O)NC)CCC(C)C(F)(F)C1 22567,N1(S(=O)(=O)c2cnccc2N2C3CCC2CC2(CC2)C3)Cc2ccccc2CC1CO 22568,N1(C(C(CC)(C)O)=O)C2CCC1CN(C(c1cc(O)ccc1Br)=O)C2 22569,C1(NC(COC(C)=O)=O)CC(CNC(c2ccc([N+](=O)[O-])[nH]2)=O)C12CCC2 22570,CN1CCCC1(C)C(=O)NCc1cccc(NC(C2CC2[N+](=O)[O-])=O)c1 22571,N1(C(c2ncc(NC)nc2)=O)CC(C)C(C)(CNC(=O)CN(C)C(C)C)C1 22572,Cc1ccc(C(N2CCCC2CNC(=O)CC2COC(=O)N2)=O)c(C2CC2)n1 22573,Cc1cc(C(N2CCCCC2CNC(=O)CNC(=O)C(C)C)=O)cc(C(F)F)c1 22574,Cc1oc([N+](=O)[O-])cc1C(=O)NCCC(C)(C)NC(=O)C=CC1CCCO1 22575,C(=O)(C1=C(C)S(=O)(=O)CC1)NC1CN(C(Cn2ncc(C#C)c2)=O)C(C)(CC)C1 22576,C1(C)(CC(=O)N(CCC(C)NC(COCC(C)C)=O)C)CCCC1 22577,c1(CC)ccc(O)c(CNC(C2C(C(=O)O)CN(CC(C3CC3)OC)C2)=O)c1 22578,N1(Cc2cccnc2)CCOC2CN(c3ccncn3)CC12.Cc1nn2cc1-2 22579,c1(NC(C2N(C(c3c(C)nn[nH]3)=O)CC(O)C2)=O)ncc(Br)cc1F 22580,Cc1cc(C(N2CCCC(C)C2CNC(=O)C2=C(Cl)CC2)=O)cc(=O)n1C 22581,c1(C(=O)NC2CC(NC(CCCOC)=O)C2)cc(C)c(Br)cc1C 22582,N1(C(c2ccc(COC)[nH]2)=O)CCN(C(c2cc(C)cc(C)c2)=O)CC1CCO 22583,C#CCC(C(=O)NC1(CNC(=O)C(=Cc2cccnc2)F)CC1)C1CC1 22584,C1(NC(c2ccc(OCc3ccc([N+](=O)[O-])cc3)o2)=O)CCC2(CCC2)C1C(=O)O 22585,CCC(CC)(CC)C(=O)NC1CN(C(=O)CS(=O)(=O)CC)CC1O 22586,C1(S(C)(=O)=O)(C(=O)NC2CC(NC(c3nc(OC)nc(O)c3)=O)C2)CC(O)C1 22587,C#CC1CCN(C(=O)C(C)(C)c2csc(Br)n2)C1 22588,Cc1cn2c(C)c(C(=O)N(C)CCN(C(=O)CCC(C)C#N)C)nc2s1 22589,C1(C(=O)NCCNC(N)=O)CCC(O)CN1C(=O)Cc1cccc(O)c1 22590,S(=O)(=O)(c1ccccc1Br)N1CCN(C(C2C(C#C)C2(C)C)=O)CC1 22591,c1(C(=O)NCC(C)NC(=O)CC2CC3CC3C2)ccccc1 22592,CC1COC2(C1)CN(C(=O)C(C1(C)CC1)NC(C1CN(C)CCO1)=O)C2 22593,C1(C2CC2)(CNC(CCSCC)=O)CCN(C(c2cn(C)nc2Cl)=O)C1 22594,N1(C(=O)CCCN2CCCCC2)CCc2nc[nH]c2C12CCN(C(C1CC1F)=O)C2 22595,C1(CSCC(=O)NCC2CC2C(=O)NCC2(Br)CC2)CCCO1 22596,Cc1nc(N(C2CCC(NC(C3CCCOC3)=O)CC2)C)cc(C(C)C)n1 22597,C1(O)(CC(=O)NCC(CC)NC(=O)C(C)(C)OCC(F)(F)F)CCCCC1 22598,C1(NC(c2cc(Cl)nnc2O)=O)CN(C(=O)COCC(F)(F)F)CC1C1CC1 22599,CC(C)(CC(=O)NCC1CCCCN(C(C2CCC(N=[N+]=[N-])C2)=O)C1)CC(F)F 22600,C1(F)(C(=O)NCC2N(C(C)=O)CCC2)CCN(C(C2(C)CCN(C)C2)=O)C1 22601,N1(C(C2(CCC)CC2)=O)CCC(F)(F)C(CNC(C2(N(C)C)CC2)=O)C1 22602,CC1=CC(C)CN(c2cc(C)nc(NC(C3CCOC3)COC(C)C)n2)C1 22603,c1(C(N2C3C(NC(Cc4c(OC)ccnc4)=O)C(C3)C2)=O)cncc2nc[nH]c12 22604,C(CC(C(=O)NCc1cscc1C)NC(c1ccsn1)=O)OCC 22605,C1(CNC(c2c(C)cc[nH]2)=O)CCCCN(C(=O)CC2CC3(COC3)C2)C1 22606,c1(C(N(C)CC2N(C(C(C=C)C)=O)CCCC2)=O)cc(CC)ccc1F 22607,CCC(C)(C)CCCC(=O)NC(CC)CCCC(=O)NC1(C2CC2)CC1 22608,c1(C(N(C2CCN(Cc3cc(OC)ns3)C2)C)=O)cc(F)c2ncccc2c1 22609,C1(C(=O)NCC(C)CN(C)C(c2nccnc2O)=O)CS(=O)(=O)CC12CC2 22610,C12CCN(CC1(F)F)C(=O)C(=O)Nc1cc(Cl)sc1NC2=O.S(C)(=O)(=O)N(C)C 22611,C(C(C)C(C)(C)C)NC(C1CCCN(Cc2ccccc2)C1)C 22612,C1(NC(C2(OC)CCN(C(C(CC)N(C)C)=O)C2)=O)CCCOC12CCC2 22613,c1(C(=O)NCCCCN(C)C(C2CC(=O)N(O)C2)=O)coc2c(F)cccc12 22614,C1(CNC(=O)NCC(c2ccc(F)cc2F)SC)CC(S(C)(=O)=O)C1 22615,CCC(CO)CCNC(=O)C(C)C(C)NC(=O)CCC1CCCC1 22616,C=CCC(CC)C(=O)N1CCCOC(CNC(c2nccc(C)c2N)=O)C1 22617,c1(C(=O)NCCCN(C(CCNC(N)=O)=O)C2CCCC2)nocc1Cl 22618,c1(C(C(=O)NCCCF)N(C2CN3CCC2CC3)C)ccc(Br)c(Cl)c1 22619,c1(CC)c(NC(C2CC(NCc3n[nH]c(C)c3C)C2)=O)cnn1C 22620,c1(OC)ccc(C(=O)NCC(C(C)C)NC(=O)C(C)=CC2CC2)c(C)c1OC 22621,c1(C(N2C3C(NC(C(c4ccccc4)OC)=O)C(C3)C2)=O)ccc(=O)n(O)c1 22622,c1(C(N2C(C)CC(NC(=O)C(C)(C)N(C)C)CC2)=O)ccccc1S(C)(=O)=O 22623,C1(O)(C(C)NC(C2(CO)CCCCC2)=O)CCN(C(c2nccnc2N)=O)CC1 22624,c1(C(N2C(CCNC(CN(C)C3CC3)=O)CCCC2)=O)ccnc(C#N)c1 22625,CC1=C(C(=O)NC(C2CCN(C(c3ncccc3N(C)C)=O)C2)C)CCO1 22626,Cc1cccc(C(N2CC(CC(=O)N(CC(C)C(F)(F)F)C)C(C)C2)=O)c1O 22627,c1(C(=O)NC(C)(C)CCNC(c2cc(CO)on2)=O)ccnc(F)c1O 22628,N1(C(c2c(C)cccc2)=O)CCC2(COC(CNC(c3ccc(O)nc3)=O)C2)C1 22629,C(CN=C(NC1CCCCC1)N1CCP(C)(=O)CC1)c1cc(CC)c(O)cc1 22630,N(C(=S)N1CC(S(=O)(=O)C2CC2)C1)CC(C)Cc1ccccc1 22631,C(C)(C(C(=O)NCc1nccn1C1CC1)C(C)C)NC(C#CC(C)C)=O 22632,c1(C(N2CC(NC(c3[nH]n(C)c(=O)n3)=O)C(O)C2)=O)occ2c1CCOC2 22633,C(CNC(c1cc(CO)c(C)o1)=O)(CC(F)(F)F)NC(c1c(NC)nccc1)=O 22634,c1(N(CCC(=O)NC)C)nc(=NCC(CO)C2CCC2)[nH]c2cccnc12 22635,c1(OC)cccc(C(=O)NC2CC(CC3(C(=O)N)CC3)C2)c1.c1(C)ccccc1 22636,N1(C(CC(=C)Br)=O)CCC(NC(=O)COCCCC)C(F)C1 22637,c1(CC)cccc(CC)c1C(=O)NCC=CCNC(c1ccc(O)c(OC)n1)=O 22638,N1(C(c2cncc(C)c2)=O)CC2CC1CN2C(=O)C(C)Cc1cccc(Br)c1 22639,C1(OC)CCCC1NC(=O)CCN(C(=O)C(C)OCCOC)CCO 22640,C(=O)(C1=CCCOCC1)N1CCC(NC(C2(COC)CCOC2)=O)CC1 22641,C=CCC(CC)C(=O)NC1CN(C(c2cn(C(C)C)nn2)=O)CC1(C)C 22642,C1(C2CCN(C(c3ccc(C#N)nc3O)=O)CC2)(NC(COCC)=O)CCC1 22643,c1(C(=O)NC2CC(C)(NC(COC(C)(C)C)=O)C2)cc(F)c2c(c1)CCC2 22644,C(C(=O)N(C)CC1CC(F)CN1C(C1CCC(C)O1)=O)(C(C)C)OC 22645,c1(C(C(=O)N(C2CCCCC2)CCNC(CCC(N)=O)=O)O)ccc(F)c(F)c1F 22646,C(CO)(CCCNC(c1cnn(C)c1)=O)NC(C(C1CCOCC1)C)=O 22647,c1(C(=O)NC(CCNC(c2n(CC)nnc2)=O)C)cc2c(s1)COCC2 22648,N1(C(c2ccc(C#C)cn2)=O)CCC2(CC(NC(=O)C3=NOCC3)CO2)C1 22649,c1(C(N(CCCOC(C)=O)C(C)C)=O)nc2cc(F)ccc2s1.CCC1C(=O)N1 22650,c1(-c2c(C)onc2)ccc(Br)cc1OC(=O)C(C)C.N12CCC(CC1)C2 22651,N1(C(C(CCC)F)=O)CC2CCC(C(N3CCc4c[nH]nc4C3)=O)(C2)C1 22652,c1(SC)ccc(CC(N2CC(C(N3C4COCC3C4)=O)CC2C(F)(F)F)=O)cc1 22653,C1(C(=O)NCCC2CCN(C(=O)CCc3ncc[nH]3)C2)CCCC(CF)C1 22654,C(CCCCCCC(=O)NC1(CO)CCN(C(c2cn(CCO)nn2)=O)C1)SC 22655,C1(CC)(Cc2ccccc2)COCCN1C(=O)CCCN1CCC(N(C)C)C1 22656,C1(C(=O)NC2CCC(CNC(c3c(C)cnnc3)=O)CC2)CCC2(C1)CC2(F)F 22657,N1(C(CCP(C)(C)=O)=O)CCOC2CN(C(=O)C=C(C3CC3)C3CC3)CC12 22658,N1(C(CCCCC(N)=O)=O)CCC2(CCCN2C(c2cn(CC(F)F)cn2)=O)C1 22659,Cc1cnsc1C(=O)NC1(C(=O)NOCC2CC(=C)C2)CCC1 22660,C1(C(C)(C)NC(C2C(F)(C(=O)OC)C2)=O)CCN(C(c2ccon2)=O)CC1 22661,N1(C(C=CCN(C)CC)=O)CC(O)CC1C(=O)N(CCN=[N+]=[N-])C 22662,c1(OC)ccc(C(C(F)(F)F)NC(c2coc(C(C)OC)n2)=O)cc1 22663,c1(C(=O)NC(C2CCN(C(C=CC)=O)C2)C)cc2c(c(S(N)(=O)=O)c1)CCC2 22664,C1(Nc2nccc(C)n2)CCC2(CCC(=O)N2)CC1 22665,c1(C(N2CC(CC=C)(NC(c3nc(C)nn3C)=O)C2)=O)nc(C2CC2)oc1C 22666,N1(C(C(=O)NCC=C)c2cn[nH]c2)CC2C(OC)CS(=O)(=O)C2C1 22667,C1(CC(=O)NC23CC(NC(=O)C(F)F)(C2)C3)CCCC(C(=O)O)C1 22668,c1(NC(C)=O)cnc(C(=O)NC2CC2C(=O)NCc2ccc(C(C)C)cc2)cn1 22669,C1(C(N(CC(O)CF)C)=O)C(C)CCN1C(=O)C(C(C)C)SC 22670,C1(N(C(CC(CC)OC)=O)C)CCN(C(=O)CCN2CCOCC2=O)CC12CC2 22671,CC(CS(=O)(=O)c1ccccc1)NCc1nnc2cccnn12 22672,c1(C(N2CCOCCC2)=O)cc(-c2cccc(Cl)c2Cl)n2nccc2n1 22673,Cc1cc(=NC(=O)C(C)(C2CC2)N(C)C(c2ccoc2C)=O)[nH]n1C 22674,c1(C(N2CC3C(NC(C(CCC)O)=O)(C3)C2)=O)cc(OC)ccc1C 22675,C12(C(N3CCC(OCCNC(C(C)n4cnnn4)=O)C3)=O)CCCCC1C2(F)F 22676,c1(C(=O)NCC2CC3CN(C(C(C)OCC)=O)CC32)c(F)cc(C)cc1Br 22677,Cc1nnc2n1CC(N=c1nc(N(C)Cc3ccn(C)n3)c3c([nH]1)CCC3)CC2 22678,Cc1oc(C)c(C(=O)NC2CC2CNC(=O)CCc2ccc(N(C)C)nc2)c1C 22679,C1(NC(CCOC)=O)COCC1C(=O)NC(C)CC1CCCO1 22680,c1(C(=O)NCC2(C(N3C(C(=O)NC)CCC3)=O)CCCC2)cncc2[nH]ccc12 22681,N1(C(Cc2cc(C)no2)=O)CCC(CNC(C2CCC(C)(C)O2)=O)C(F)(F)C1 22682,C1(CNC(CCCCNC(N)=O)=O)CCN(C(=O)CC2CCCOC2)CC1(F)F 22683,c1(OC)ccc2c(C(=O)NC3CC(C)CN(C(c4[nH]ccc4C)=O)C3)c[nH]c2c1 22684,Cc1nc(NC2CN(C(c3nc(N(C)C)nc(=N)[nH]3)=O)CC2C)cc(O)n1 22685,N1(C(CCC2CC(C)C2)=O)CCC(C)(C)C(C(=O)NCC2(C)CC(C)(C)C2)C1 22686,c1(OC)ccc(F)cc1CC(=O)NCC=CCNC(=O)C(c1cnccn1)C 22687,N1(C2C(NC(C(CC)F)=O)CCC2)CCN(C(C2CC(O)C2)=O)CC1 22688,C(=O)(C1c2ccccc2CCCN1Cc1cc(Cl)ccc1Br)OC 22689,C=C(C)CC(C(=O)NC(CCC1CC1)C(=O)N1CC(OC(F)F)C1)OC 22690,CC1CN2CCN1C(C(N1CCCC1C1CCN(C(=O)CC3CC3(Cl)Cl)C1)=O)C2 22691,N1(C(CCCCOC)=O)CC(O)CCC1C(=O)NCCCc1ccco1 22692,Cc1cc(S(N)(=O)=O)sc1C(N1CCC2C(CCN2C(=O)C#CC(C)(C)C)C1)=O 22693,N1(C(c2ccc(C)cc2Cl)=O)CCCC2CCN(C(c3onc(C)c3C)=O)CC12 22694,c1(OCC)ccc(C)nc1C(=O)NCC1CN(C(=O)CC2COC(=O)C2)C1 22695,N1(C(CN(CCC)C)=O)CC2CCC1CN2C(=O)Cc1c[nH]c2ncccc12 22696,CCCC(CC)CCN1CCCC1C(N1CCCCC1)=O 22697,c1(C(N2CCC(NC(CCn3c(C)ncc3)=O)C2)=O)cc2scc(C)c2[nH]1 22698,C=CC1(C(=O)NCCN(C2CC2)CC)CCN(C(=O)CCCC2CC2)C1 22699,c1(C(=O)NCC2(C)CCC(NC(c3ncn(C)c3)=O)C2)ccnc2ncccc12 22700,C12(CNC(c3ncc(SC)s3)c3nnnn3CCC3CC3)CC1CCC2(F)F 22701,N1(C(C2=C(C)CC2)=O)CC2COCC2(C(=O)NC2CCCC(O)C2)C1 22702,O=C(CC1CCN(S(=O)(=O)c2cccnc2)C1)N=c1cc(C2CCOC2)[nH][nH]1 22703,c1(CC=C)cccc(C(=O)NCCN(C(=O)C=C(C)C)CC2CC2)c1 22704,c1(CC(=O)NCC(C)(C2CCC2)NC(CC2(OC)CC2)=O)nc(F)c(F)cc1F 22705,c1(C(N2CC(C(=O)NCC(C)(C)C3CC3)(COC)C2)=O)ccc2cccnn12 22706,Cc1coc(C2CC2)c1C(=O)NCC1CC(NC(c2coc(CF)n2)=O)C1(C)C 22707,C#CC1CN(C(=O)CCNC(C2CC2OC)=O)CCN1C(=O)Cc1nc[nH]n1 22708,CC1CCn2c(C(=O)NC(C)CNC(C3(N4CCOCC4)CCC3)=O)cnc2C1 22709,Cc1ccc2occ(C(=O)NC3CCC(CNC(c4cscc4C)=O)CC3)c2c1 22710,C1(NC(CC(C)C2CCCCC2)=O)CC2(CCCN(C(C3CC(=O)C3)=O)C2)C1 22711,c1(CC)ccccc1CC(=O)NCC(C)(Cn1cccn1)NC(=O)CN1CCC1C 22712,C1(C(N2CC3C(NC(C4(C)CCOCC4)=O)(C3)C2)=O)CN2CCN1CC2 22713,c1(CC(N2CC(O)(C(C)NC(COC(C)C)=O)C2)=O)noc2cc(F)ccc12 22714,n1(CCC(N2CC(NC(C3(C(CC)(F)F)CC3)=O)C3C2C3)=O)cc([N+](=O)[O-])cn1 22715,N1(C(Cc2coc3ccc(C)cc32)=O)CC2CCCC(C1)N(C(=O)C(N)=O)C2 22716,CCCCCC(F)C(=O)N1CC2CC1C2C(N1CCC2CC12C)=O 22717,N1(C(CCC2(NC(c3c(CC)cno3)=O)CCC2)=O)CC(C)SC(C)C1 22718,C1(NC(CCOCCOCC)=O)CCN(C(c2c[nH]cc2C(C)(C)C)=O)CC1F 22719,N1(CC2CC(C(=O)OC)C2)CCOC2(CCC(F)(F)CC2)C1 22720,N1(c2scc(C(=O)NC3CN(C(C4CC4CC(F)(F)F)=O)C3)n2)CCCNC1=O 22721,c1(OC)ccc(C(C(=O)NC(C)COC)OC)cc1 22722,CCCC(C(=O)NC1CN(CC)CC1C)NC(C1(CC)CCCC1O)=O 22723,c1(C(CCNC(CC2CCN(Cc3nnc(C)o3)CC2)=O)C)ccccc1C#N 22724,CC(C)C(O)C(=O)NC1CC12CC(NC(=O)C=Cc1ccsc1Br)C2 22725,O=C(CC1=CCN(C(C2(O)CCOC2)=O)CC1)Nc1cncc(C2CC2)c1 22726,c1(C(=O)NCc2occc2C(=O)NC2CN(c3ccncc3)C2)ncc(F)cc1F 22727,c1(C(C(=O)OCC)C#N)ccc2c(c1)nc(Oc1cc(Cl)cc(Cl)c1)n2C 22728,C1(C(=O)NCc2ccc(C(N(C)CC3(O)CCC3)=O)cc2)CC(C)(C)OC1(C)C 22729,CC1=C(C)CC(C(N2CCOC(C(=O)NCC3(O)CCC(C)(C)C3)C2)=O)CC1 22730,c1(OC)cc(C(=O)NCC#CCNC(=O)CCc2ccc(Cl)nc2)ncn1 22731,C1(N(C)C(=O)Nc2ccc(Br)s2)CCCN(CCC(=O)Nc2ccccc2Cl)C1 22732,CCC(CC(=O)N1CCC(CCNC(=O)C(C)(CC)OC)C1)C1CCC1 22733,CC1(C)Cc2cccc(C(=O)NCC3CC(NC(C4(C)CC4)=O)C3)c2O1 22734,Cc1ccn2cnc(C(=O)NCCCC3CCCN3C(C3CCCOC3)=O)c2c1 22735,C(=O)(CC(C)(C)CC(=O)NC1CC12CC(NC(=O)C(O)C1CCC1)C2)OC 22736,N1(C(Cn2ncc(C)c2)=O)CCC(CNC(=O)CC(C)C(F)F)C(F)(F)CC1 22737,c1(C(N(C2CCN(C(=O)C=CS(C)=O)C2)CC)=O)ccccc1Cl 22738,C1(CNC(CSCCCC)=O)CC2(CCC2)CN1C(=O)CC(C)n1cccn1 22739,O=C(C(F)C(F)(F)F)NC1CCC(NC(c2cccnc2C(=O)NC2CC2)=O)CC1 22740,C1(N(c2ccccn2)C(N2CCCC2Cc2nccn2C)=O)(CC)CCCC1O 22741,C1(NC(Cc2nc(CC)sc2)=O)CCN(C(c2ccncc2Cl)=O)C(C)C1 22742,c1(C(=O)NC(c2ccccc2)CNC(C(C=C)O)=O)nc2ncccc2cc1C 22743,CCCC(O)CC(=O)N(C1CCCN(C(=O)Cc2nccn2C)C1)C 22744,C1(C(N2CC(O)(C(F)C(=O)NCCCCO)C2)=O)(CC)CCOC1 22745,C1(C(=O)NCC(CN(C)C(c2ccc(CO)cc2F)=O)O)CC2(COCCO2)C1 22746,N1(C(CCCCC(=O)NC)=O)CCC2(C1)CN(C(=O)C(F)n1ccnc1)CCO2 22747,N1(CCC(=O)NC(C(C)NC(c2c(C)onc2Cl)=O)C)CCSC(C)(C)C1 22748,S(=O)(=O)(c1ccc(=NCC2CNC(=O)CO2)[nH]c1)NC(c1n(C)cnc1)CO 22749,CCC(CO)(C(=O)N1CC=CC(C(=O)NOC(C)C)C1)OC 22750,Cc1cc(NC(=O)N(C2CC2)Cc2ccc(C)c(F)c2)c(=O)n(C)c1 22751,c1(OCC(=O)N(CCC(C)NC(=O)C(C)(Cl)Cl)C)ccc(F)cc1 22752,C1(CC(=O)NC(CNC(C2(COC)CCC2)=O)(C)C2CC2)C=NN(C)C1=O 22753,c1(CC=C)ccccc1C(=O)NC(C)(CSC)C(=O)NCCOC(F)F 22754,C(C(C(C)(C)C)NC(=O)Cn1c(C)csc1=O)NC(C1C(CC)C1)=O 22755,C(=O)(C(O)C(C)(C)C)N1C(C(=O)NC(COC)COC)CC2CC21 22756,C1(NC(=O)C=Cc2cccs2)CCN(C(C2(C(F)F)CCCCO2)=O)CC1CO 22757,C1(C2CCC(=O)NC2)(C(N2C(C)CN(C(C3CCC(C)CC3)=O)CC2)=O)CCC1 22758,c1(-c2cccc(N(CCCC(=O)O)C)c2)ccc(N)cc1F 22759,C1(NC(c2ncc(C)[nH]2)(C)C)CNCC(O)C1 22760,c1(CC(=O)NCC2CC(NC(c3c(=N)cc[nH]c3)=O)C2)cc(O)nc(O)n1 22761,c1(CNC(c2c(C)c(C3CC3)on2)=O)cnn2c1CN(C(=O)CCC1CC1)CC2 22762,c1(OC)cc(O)nc(O)n1.C1(NC(C2CCCC(SC)C2)=O)CNC(=O)C1 22763,C1(NC(c2ccc([N+](=O)[O-])nc2)=O)COC2(CCN(C(C3CCC3)=O)CC2)C1 22764,C12CCCC(CC1)C(=O)N2C(N1CC=CCC1)=O.C(C)(C(F)F)=CC(=O)OC 22765,c1(NC(C2(C(C)C)CC2)=O)cc(OC2CC2)ncc1C1=CCCCC1C 22766,C1(OC)CC(NC(c2cn(C(C)(C)C)nn2)=O)CN(C(=O)CC2C=CCCC2)C1 22767,C(=O)(C(CCF)NC(=O)OC(C)(C)C)NCC(N(C(CC=C)=O)C1CC1)C1CC1 22768,C1(CNC(c2cn(CC)nc2)=O)CCC(NC(=O)CN2CCSCC2)CC1 22769,C1(NC(C2CCC(C)(C)OC2)=O)CC1C1CCN(C(c2ccoc2Cl)=O)CC1 22770,c1(CC)onc(C(F)(F)F)c1C(=O)NCC(c1cccnc1)NC(=O)OC(C)(C)C 22771,O=C(CC(Cc1cccs1)NC(=O)CC1CCC1)NCc1cc[nH]n1 22772,c1(N2CC(C(=O)NCC)C2)ncc(C)c(C)n1 22773,c1(C(N(CCNC(=O)Cc2cn(CC)nc2C)CC)=O)cnccc1C#N 22774,CCCC(C(=O)NCC1CCC(NC(C2CC2CC(C)(C)C)=O)CC1)NC(N)=O 22775,N1(C(CC=C=C)=O)CC2CC1CCC2NC(=O)Cc1scnc1C 22776,c1(OCC)ccc(-c2ccc(NC(=O)Nc3cc(C)cc(C)c3)nc2)c(C)c1 22777,N1(C(Cc2c(C)cccc2C)=O)CC2CCC(C1)C(NC(C1CC(F)(F)C1)=O)C2 22778,N1(C(c2cn(CCOC)nc2)=O)CCOC2(CCN(C(=O)C3=COCC3)CC2)C1 22779,C1(NC(CCCC#C)=O)CCN(C(=O)COc2ccc(C)cc2C(C)C)CC1C 22780,Cc1c(NC(=O)C(C2CCOC2)NC(C2C3CN(C)CC23)=O)cccc1C#N 22781,CC1CC=C(C(=O)NC(CN=[N+]=[N-])C(=O)NCC2CCN(C)CC2)CC1 22782,C1(C)(C(=O)NC(c2cccnc2)C)CCCO1.C1(=O)C=CCN1 22783,c1(C(N(CC(C)NC(C(COC)N(C)C)=O)C)=O)sc(C)c(Br)c1OC 22784,C1(N(C(COC(C)C)=O)C)CCCCN(C(c2cn(C)nc2C2CC2)=O)C1 22785,c1(NC(CCCCc2cccc(OC)c2)=O)cccc(SC(F)(F)F)c1F 22786,Cc1c(C(=O)NC(C)(C)CN(C)C(C2(C)CC2F)=O)nc(O)c2ccccc12 22787,N1(C(CC2OCC(C)(C)OC2)=O)CC2(C1)CN(C(c1coc(O)n1)=O)CCO2 22788,c1(OCC=C)ccccc1C(N1CCCC1(C)C(=O)NCc1ccccn1)=O 22789,C1(CNC(C=CC(C)=O)=O)CC2CCC(C1)N2C(=O)CCCc1cccnc1 22790,Cc1ccc(C(F)C(N2CCCCC2CNC(=O)CN(C)C2CC2)=O)cc1 22791,C1(CNC(=O)C(O)Cc2cnc[nH]2)C2CN(C(C3CC(F)(CF)C3)=O)CC12 22792,C1(C(=O)NC2(CC)CC2)CCN(C(C2(CC)CN(C(=O)OC)C2)=O)C1 22793,N#Cc1c(Cl)ccc(Br)c1SCC1=NOC2OCCCC12 22794,C1(NC(C=CC=CCC)=O)CCC(O)CN(C(=O)CCC2CCN(C)C2)C1 22795,c1(C(=O)NCC(CNC(Cc2c(C)n(C)cn2)=O)C)ccc(S(N)(=O)=O)nc1 22796,CC(CC(C)(C)C)C(=O)NCCSCc1cn(-c2ncc(Cl)cc2Cl)nn1 22797,C(CNC(=O)NCc1cc(C)c(F)c(C)c1)(CCS(C)(=O)=O)OC 22798,N1(C(c2cnn(CC)n2)=O)CCCC(NC(c2cccc(C)c2Cl)=O)CC1 22799,C1(CC)CN(C(=O)CN2CCCCCC2)CCC1NC(c1c(C)nn(C)c1N)=O 22800,c1(C(N(CC(CC)NC(C=CCC)=O)CC)=O)cnn2cccc(Br)c12 22801,N1(CC(=O)NC2CCCC2CNC(C2CC(CF)C2)=O)CCOCC1 22802,C1(CN(C(=O)CCCN(C)C(C)C)CC)CCN(C(c2cc(C)cs2)=O)CC1 22803,CC1CCc2sc(CNC(=O)Nc3nc4ccccc4nc3C3CC3)cc2C1 22804,c1(C(=O)NCC2CCN(C(c3c(CC)cc[nH]3)=O)C2)ccc(F)cc1C 22805,C(=O)(CC(O)C(C)C)NC(CC=CC)C(=O)NC(c1ncccc1F)C 22806,C1(CN(C(=O)C(c2cnn(C)c2)O)C)CCN(C(=O)C(C2CCOCC2)=O)CC1 22807,C(=O)(C1Cc2ccc(C)cc21)N1CCC(N(C(CCCC(=O)NCC)=O)C)CC1 22808,C1(CNC(C(C)C2CC2)=O)CN(C(=O)Cn2ncc3ncccc23)CCC1(C)C 22809,c1(C(N2CCC(C3N(CC(CC)C)CCC3)CC2)=O)cc(C#N)[nH]c1C 22810,C1(C(=O)NC2CC(C)C2)CC2(CCN(C(C3CCCCS3)=O)C2)C1 22811,C(=O)(C(C)CC(=O)NCCCc1cncc(C(=O)OC)c1)OC 22812,c1(C(=O)NC(C(=O)OC)Cc2c(OC)cccc2Cl)cccc2c1CCC2 22813,c1(C(C)(C)C)nc(=NCC2CCCCN2C(=O)Cn2cncn2)s[nH]1 22814,C1(NC(c2cc(C)n(C(C)C)n2)=O)CCN(C(=O)Cc2ccco2)CC1F 22815,c12c(Cl)cc(cc1Cl)OC(=O)CS2.c1(C(N(C(C)=O)C)C)nnc(C)o1 22816,CCC(C)C(C)C(=O)N(C)CC1CCCCN1C(C1CCCC(C)CC1)=O 22817,CC(C)(C(=O)NCCC1CN(C(C2CCS2(=O)=O)=O)C1)c1ccccc1 22818,Cc1cc(N2CCC(NC3CCSC(c4cnn(C)c4)C3)CC2)ccn1 22819,n1(CC(N2CCCC(N(C(C3CC3CF)=O)CC)C2)=O)cc([N+](=O)[O-])cn1 22820,CC1(CNCc2cccnc2Br)CCN(Cc2ccccc2)C1 22821,Cc1ccc(C(N2CCCC(C)C2C)C(=O)NC2COC2)cc1[N+](=O)[O-] 22822,c1(C(=O)NCC(C)(C)NC(CC(=C)C)=O)ccc(CC)nc1C 22823,Cc1nc2nccc(C(=O)NC3CCCC(CNC(C4CN(C)C4)=O)C3)n2n1 22824,N1(C(=O)C2=C(Cl)CC2)CCC2(CCCN2C(C2CC3(C2)CC3F)=O)C1 22825,c1(C(=O)NC2(CO)CCN(C(=O)CC3C=CCC3)C2)cccc2ccsc12 22826,Cc1ccncc1C=CC(=O)NC1CC(NC(=O)CC2CS(=O)(=O)C2)CC1O 22827,CC(CCCC(=O)NOC1CCOCC1)NC(c1cc(=N)[nH][nH]1)=O 22828,C(=O)(C1=C(C)C(C)(C)OC1=O)N1C(CCOC)CN(C(=O)Cc2cccs2)CC1 22829,C1(C)(C(=O)OC)COCCN1C(=O)C(=O)N(C(C)C)Cc1ccc(Cl)c(Br)c1 22830,C1(C(N(CCN(C(=O)CC2CCC(=O)N2)C(C)C)C)=O)CCNC(=O)C1 22831,N1(C(CCC(C)C)=O)CCC2CN(C(=O)Cn3cc(C4CC4)nn3)CC2C1 22832,C1(C(=O)NCC(C)NC(C(C)NC(c2ccco2)=O)=O)C(C)(C)OC1(C)C 22833,CCCC(CC(C)C)C(=O)N1CC=CC1C(=O)NCC(=O)OC 22834,C1(C(=O)NCCC2COCCN2C(c2cnc(SC)n2C)=O)(CC)CC(C)(C)C1 22835,Cc1nc2cncc(C(=O)NCC3CN(C(C4C(Cl)(Cl)C45CC5)=O)CCO3)c2[nH]1 22836,C(=O)(C1CCCn2ncnc21)NC1CC(C)N(C(c2cnc(C(C)(C)C)s2)=O)C1 22837,C(=O)(CCCc1ccncc1)N(CC(CC)NC(=O)C(C)(C)SC)C 22838,N1(C(C(C)(C)CF)=O)CCC2(CCCC2CNC(c2ccnc(O)c2)=O)CC1 22839,S(=O)(=O)(c1c[nH]c(C(=O)NCC2CC(C)N(C(C3C4CCC3CC4)=O)C2)c1)NC 22840,CC1CCN(C(c2cn(CCNC(c3cnsn3)=O)nn2)=O)C(C)C1 22841,N1(C(C2(C=C)CCC2)=O)CCCC(CC(=O)NCCC2CCCN2C)C1 22842,c1(CNC(C23N(C(COC(C)(C)C)=O)CCC2CC3)=O)nccn2nccc12 22843,C(=O)(C1=Cc2ccccc2OC1)N(CC(C)NC(=O)CCN1CCCCC1=O)C 22844,c1(OC)ccc(NC(=O)C(C)C(c2ccc(N3CCCC3SCC)cc2)C)cc1 22845,c1(CC(N2C(COC)CN(C(=O)CC3CC3(F)F)CC2)=O)ccc2c(c1)OCO2 22846,c1(C(C)=O)cc(O)cc(O)c1C(=O)NCC12CC1CN(C(c1cc(O)n[nH]1)=O)C2 22847,c1(OC)cc(C(=O)N(CC(C)NC(c2c(C)nc(C)n2O)=O)C)ccc1C 22848,C1(F)(N(C(C(CC)C2CCC(=O)N2)=O)c2nn[nH]n2)CCN(C(=O)OC(C)(C)C)C1 22849,C(CNC(C1(C(F)F)CC1)=O)(C(C)C(C)C)NC(c1cc(C)c(C)[nH]1)=O 22850,N1(C(CC)=O)CCCC2(CNC(C3CCCC(=O)C3)=O)CCCC12 22851,C1(C(=O)OCC)CC(F)CN1C(=O)CCCCc1cn(C2CCOC2)nn1 22852,N1(C(c2cn(CC)nc2)=O)CCC(C)(C)C1CC(N1CC(C)(C#N)C1)=O 22853,S(=O)(=O)(c1cccc(-c2nnc(C(N)C3CC3)o2)c1)N(C)C 22854,C1(NC(Cc2c(C)cco2)=O)CN(C(=O)CC2CCCOC2)CC2(CC2)C1 22855,C(c1ccc2c(c1)COCC2)=CC(N1C2CN(C(C(C(C)C)F)=O)CC1CC2)=O 22856,O=S(c1ccc(NC2COc3c(Cl)cc(Cl)cc32)cc1)C(F)(F)F 22857,c1(C(=O)NC23C(CN(C(CC4(NC(C)=O)CC4)=O)C2)C3)cc2nc[nH]c2cn1 22858,CCC(CC)CC(=O)NC(c1nn(C)cc1O)C 22859,C1(C(=O)NCC(=O)NC(C(C)NC(=O)CCC2CC2)C)CCCCC1 22860,Cc1ccc([N+](=O)[O-])c(C(=O)NC2CCCN(C(c3c(C)n[nH]c3C)=O)C2)c1C 22861,CCC(CC)CCCC(=O)NC(C1(O)CCN(C(c2noc(CC)c2C)=O)C1)C 22862,C1(NC(c2csc(Cl)n2)=O)CC(O)CN(C(c2ccc(OCC3CC3)nc2)=O)C1 22863,C12(CNC(C(CC=CC)CC)=O)CCCC(CN1C(=O)CCc1cncnc1)C2 22864,N1(C(C2C(=C)C2C(=O)OC)=O)CC(=O)NCC1C(=O)N(CCC)CC 22865,C1(NC(C2C(C)(C)C2)=O)CCCN(C(c2ccn(-c3ccc(O)cc3)n2)=O)C1 22866,C=CCC(C)(C)CC(=O)NC1CCC(N(C)C(c2cc3ncccc3s2)=O)CC1 22867,C1(NC(c2nc(C)sc2)=O)CN(C(C2C=CCC2)=O)CC12CCS(=O)(=O)CC2 22868,C(=O)(C1CCCn2cnnc21)NCC1(O)CN(C(c2n(CC)ncn2)=O)C1 22869,C1(C(=O)NCC2N(C(c3ccnc(C)c3N)=O)CCC2)CCc2ccccc2O1 22870,C1(C(C)NC(=O)Cc2cn[nH]c2)CCN(C(c2cnnn2C2CCCC2)=O)CC1 22871,N1(C(c2c(C)ccnc2)=O)CCC2(CC1)CC(NC(C1CCN(C)C1C)=O)C2 22872,c1(OC)c(CC(=O)NCCN(CC(C)O)C(C2CCCCS2)=O)cccc1F 22873,C(CC(=O)N1CCN(CC(C)(C)NC(C2CC3CC2C3)=O)CC1)(C(F)(F)F)OC 22874,c1(C(=O)NCC2CN(C(CC=CCC)=O)C3C2C3)ccc(O)c(CO)c1.C1CS1 22875,C(C)(N=c1cc(C)nc(N2CCC(C)C2)[nH]1)c1[nH]nc(C(=O)OCC)n1 22876,N1(C(c2ccc(CN(C)C)o2)=O)CCC(CO)(CNC(C2CCS(=O)(=O)C2)=O)C1 22877,c1(C(N(CC(C)NC(=O)CSCc2cccs2)CC)=O)cc(CCO)on1 22878,CCC(C)(C)C(C)NC(C1CCN1C(=O)C(C)NC=O)=O 22879,C=CC1OCCC1C(=O)NCCC1CC(NC(=O)CCC2CC2C)C1 22880,c1(OC)cc(Cl)c(C)cc1C(N1CC=CC(NC(c2cc(SC)c(C)o2)=O)C1)=O 22881,Cc1cn(C)nc1C(=O)NC(CC1CCCC1)C(=O)NC1CCOCC1F 22882,C(=O)(C1COc2ccccc21)N1C(CNC(c2n[nH]c(C)c2O)=O)CC(F)(F)C1 22883,CC(C)C(O)C(C)C(=O)NCC1CCOC1C(N1CC2CC(CO)C(C2)C1)=O 22884,N1(C(c2ccc(CCC)s2)=O)CCC2CN(C(c3ncc(F)cn3)=O)C2C1 22885,C(=O)(CC(O)CC(C)C)N1C(CN(C(c2c(C)[nH]c(C)c2C)=O)C)CC(F)C1 22886,c1(C(N2CC(CNC(CC=C=C)=O)C(O)C2)=O)c(-n2cccn2)cccc1F 22887,c1(C(=O)NC2CN(C(=O)CC3CC4(CC4)CO3)C2)ccc2c(c1)CNC2=O 22888,C1(C(N(CCC=C)CC)=O)CCCCCC1Nc1ncc(CC)cn1 22889,c1(C(=O)NC2C(F)CCN(C(C3CC(=C)C3)=O)C2)ccc2nc(C(F)F)[nH]c2c1 22890,C1(NC(c2n(C(C)C)ncc2Br)=O)CCCCCN(C(=O)C(C)C2CC2)C1 22891,c1(C(=O)NCCCCC(CO)NC(CC2(OC)CCC2)=O)ccc(C#N)c(O)c1 22892,N1(C(C(C2CCC2)OC)=O)CCCC(C)(C)C1C(N1CC(O)C(C2CC2)C1)=O 22893,c1(C(N2C(C)CC(NC(C(C(=O)OC)(C)F)=O)C2)=O)ccc2ncnc(O)c2c1 22894,CCCCCCCCCCCCCCCOC(C1CC(=O)NC2CCCCC12)=O 22895,c1(C(=O)NC(c2cn(CC3(C)CCCC3O)nn2)CCC)ncc(Cl)cc1Cl 22896,c1(-c2scc(C(N3CCC(NC(CCC=C)=O)C3)=O)n2)ncccc1F 22897,C1(CNC(COCCCOC)=O)CCC2CN(C(c3ccoc3C(C)C)=O)CC12 22898,c1(COCC(=O)N)cc(C2CC2)on1.C1(C2CC2)CCCC1.C12CC(C1)NC(=O)C2 22899,Cc1oc(CNC(C2CN(C)C2)=O)nc1C(=O)N(C)CCC1CCC1 22900,c1(CNC(C2C=CCCC2)=O)ccccc1-n1cc(CC2CC(CF)C2)nn1 22901,C12(CNC(C3C(C(=O)OC)C3)=O)CC(NC(=O)CCC(C)N(C)C)(CO1)C2 22902,N1(C(CNC[Si](C)(C)C)=O)CC(O)CC1CNC(C1(C(F)(F)F)CC=CC1)=O 22903,C12(COC)CC(C(=O)NCC(C3CCCN3C(=O)C(C)CN(C)C)(C)C)(CO1)C2 22904,C1(CC(=O)Nc2cnsn2)CCCN1C(=O)CN1CCCC1 22905,c1(OC)cc(C(=O)N(C(C)CNC(c2noc(CO)c2C)=O)C)cc(F)c1 22906,Cc1nnn(CC(=O)NC2(CNC(c3ccn(CC(F)F)n3)=O)CCC2)n1 22907,N1(C(C(C)(C)SC)=O)CCC2(CC1)CC2NC(c1cnn(CCCOC)c1)=O 22908,c1(CC)nc[nH]c1C(=O)NCC1(Cn2cc(CCCN(C)C)nn2)CC1 22909,Cc1csc(Cl)c1C(=O)N(C)CC1COCCN1C(c1cnccn1)=O 22910,c1(C(=O)NC2C=CC(C(=O)Nc3c(O)ccc(C)c3)C2)cc2cccc(F)c2s1 22911,c1(OC)ncccc1-c1cn(C2CCC(C(N3CCC(CC4CC4)C3)=O)C2)nn1 22912,c1(C(=O)Nc2c(CC(=O)N(C(C)(C)C)C)nccc2)nn(C)c2ccc(Br)cc12 22913,CC(C)CC(C(=O)NCCOCCN(C)C(c1cc2c(nn1)CCC2)=O)C(N)=O 22914,N1(C(c2occ(C)c2)=O)CC2OCCN(C(C3CCCCS3(=O)=O)=O)C2C1 22915,N1(Cc2cc(C(C)C)no2)CCc2c(C(=O)OC(C)(C)C)cccc2C1 22916,N1(C(CCCCC)=O)CC2(C1)CN(C(C1CCCC1)=O)CC2CO 22917,C(=O)(C(CCCC)C(C)C)N1CCC(C(=O)NCC(C)OCC#C)C1C(C)C 22918,C1(C2(NC(c3c(CCCC)ocn3)=O)CC2)CCCCN1C(=O)C=CC(F)(F)F 22919,Cc1cn2c(C(=O)NCC3CC3CNC(=O)C=C3CCOCC3)c(C)nc2s1 22920,CC1(C)C(C(=O)NCc2ccc3c(c2)CC3)CCN1C(c1c[nH]c(=O)cn1)=O 22921,N1(C(CCC(C)C)=O)CC(C)CN(C(c2cccc(C(C)(C)C)c2)=O)C(C)C1 22922,c1(C(N2C(C)CCC(NC(c3cncn3C)=O)C2)=O)cc2c(s1)CCCCCC2 22923,N#Cc1ccc(NC(=O)CNC(=O)CC2CNCCO2)cc1Cl 22924,N1(C(CC(C(C)C)C)=O)CCC(N(C)C(C2CC3(C2)CC(O)C3)=O)C2(CC2)C1 22925,C(=O)(C(CCC(C)C)NC(C1CN2CCN1CC2)=O)NCc1ncc(OC)cn1 22926,CC(O)CCC(=O)NC1CCC(N(C(=O)CCc2ccccc2C(N)=O)C)CC1 22927,C1(CC#C)(C(=O)NC2CCC2NC(C2CN(c3nncs3)C2)=O)CCCCO1 22928,C1(C)(COC)CC(NC(c2cc(N)ccc2Cl)=O)CN1C(=O)CCCC1CC1 22929,c1(C(C(=O)NC2C(NC(c3occ(C(=O)OC)c3)=O)CC2)O)ccc(F)cc1C 22930,CC(C)CC(C(=O)NC(COC(C)C)C(=O)NC1CC(C)(C)OC1(C)C)C(N)=O 22931,C(=O)(CC(C)c1ccncc1)N(CCNC(=O)CCSC(F)(F)F)CC 22932,Cc1ccc(C(=O)N(C2CN(C(C3CC4(CC4)CN3C)=O)CCC2O)C)cc1Cl 22933,c1(C(C)NC(=O)OC(C)(C)C)c(NC(=O)C(=Cc2cscn2)C)sc2c1CCCC2 22934,c1(C(=O)NCC23OCC(CNC(=O)CCF)(C2)C3)sc2sccc2c1Cl 22935,CCCCC(CNC(c1cc(C#N)c[nH]1)=O)NC(=O)COCC1CCOC1 22936,c1(C(N2C(CC(C)(C)C)CCC2)=O)cc(C(F)(F)F)ccc1Br 22937,CC1=C(C(=O)NC2CC2CNC(C2(C)CCC2)=O)CCCC1 22938,N1(C(C(n2cc(Cl)cn2)C)=O)CCCC1Cn1cc(C2CCCCO2)nn1 22939,c1(OC)cc(C(N2CC(C)CC(C)C2)=O)ccc1NC(=O)CC(C)O 22940,c1(C(c2n(CCOC)nnn2)NCC(c2cccs2)C)nc(C)c(C)[nH]1 22941,CC1CCN(C(=O)Cn2ccnn2)C(C)C1NC(c1cccc(C(F)(F)F)c1)=O 22942,c1(CNc2c(C(=O)NCC)nccc2)oc2ccccc2c1C 22943,C(c1ccc2ccccc2n1)=CC(=O)NCC(F)CNC(=O)CC1COCCO1 22944,N1(c2nnc(C)s2)CCC2CC(C(N3CCC(c4nncn4C)CC3)=O)C2C1 22945,C1(C2CCC2)(C(=O)NCC2(C(C)(C)C)CCN(C(c3cnns3)=O)C2)CC1 22946,N1(C(c2c(C(C)C)nn(C)c2)=O)C(CNC(=O)COCC2CC2)CC2COCC12 22947,c1(C(=O)NC(C(C)NC(=O)CC2CCC2)(C)C)ccc2c(c1)CCN2S(C)(=O)=O 22948,CC12CC(C(N3CCC(F)(CNC(=O)C4=CCCOC4)C3)=O)(CCO1)C2 22949,C1(NC(C2CCN(OC)CC2)=O)CCC2(CC1)CCN(C(=O)Cc1cnoc1)C2 22950,N#CC1(C(N2CCC3(CC(NC(C4CNC(=O)N4)=O)C3)C2)=O)CC2(CCC2)C1 22951,C(C)(C)(CCC(=O)N1CCCC(COC)(NC(=O)Cc2ccco2)C1)OC 22952,C12(C(=O)NCC3CN(C(C4CCCC45CCC5)=O)CCO3)C3CC(CC13)C2(F)F 22953,c1(C(=O)NCCCN(CCCNC(C2C(C)C2C)=O)C)csc(Cl)c1 22954,N1(C(C2CCC(=O)O2)=O)CCCC2CN(C(c3noc4c3COCC4)=O)CCC12 22955,C#CCCCC(C(=O)NC1CCC(F)(F)CC1)N1CC(C)CC1c1ccccc1 22956,CC(C(=O)NC(C1(C(N2CCOCC2CC2CCC2)=O)CC1)C)C(F)F 22957,C(C1c2ccccc2CCN1C(C1CCCS1)=O)NC(COCCCC)=O 22958,Cc1ccc(F)cc1NC(C1C2CC2CN1C(=O)CCc1nncn1C)=O 22959,C(=O)(C(C)(O)CCSCc1ccccc1)N1C2C(NC(CCCOC)=O)C(C2)C1 22960,C1(C(N(C)CC2CCCCN2C(c2nonc2N)=O)=O)Cc2ccncc2C1 22961,c1(C(=O)NC(c2ncccc2F)CC)cc(C(C)C)cc(C(C)C)c1 22962,S(=O)(=O)(c1ccc(F)c(F)c1)N1C(C(=O)NCc2ccc(Br)cn2)CC2CC21 22963,Cc1cc(O)cc(C)c1CC1CCCCC1c1nc(CSCc2ccccc2)no1 22964,CC1(C#N)CCN(C(=NC2CCC2)NC2CCN(S(C)(=O)=O)C2)CC1 22965,CCC(C)C(O)C(C)C(=O)NCC(C)=CC(N1CCC(O)(C(F)F)C1)=O 22966,c1(C(N2CCC(C3(NC(C(C)=C(C)C)=O)CC3)C2)=O)ccc2ncccc2n1 22967,c1(OCC)ccc(Cl)nc1C(N1CC(NC(C2CC2c2ccccc2)=O)C1)=O 22968,N1(C(c2c(CC)cno2)=O)CC(N(C(=O)C(C2CC2)SC)C)C2(CC2)C1 22969,N1(C(C2CC(CC)C2)=O)CCN(C(c2coc(Br)n2)=O)C(CCOC)C1 22970,c1(C(N2CC(C(=O)NCc3ccc[nH]3)OCC2)=O)ccc2ccncc2c1 22971,CCCC(C)(O)C(=O)NC1CC(CC(=O)NCC(C)(C)CC(C)C)C1 22972,C1(C(C(=O)O)NC(c2nc(CCP(C)(C)=O)sc2)=O)CC2C=CC1C2 22973,C1(N(C(=O)CN(C)C2CC2)C)CCN(Cc2ncccn2)CC1 22974,c1(SC)ccc(CN(C(c2cc(C)ns2)C(=O)NCCCF)C2CC2)cc1 22975,C=C(CNC(=O)C(C)(C)C1CCCC1)CCN(C(=O)CC1(C(F)(F)F)CC1)CC 22976,C(N=c1[nH]c2c(F)cc(Cl)cc2s1)C1CC(NC(c2c(CC)nc[nH]2)=O)C1 22977,C1(CNC(C(CC=CC)C)=O)CN(C(c2cc(Cl)cs2)=O)CC1(F)F 22978,c1(C(=O)NCCC2CN(C(C3CCCS3)=O)CCO2)coc2c1COC2 22979,N1(C(C(CC)OCC)=O)CC(NC(C2CC(=O)N(C(CC)CC)C2)=O)C(C)C1 22980,Cc1nc2[nH]c(C(N3CCC(C)(NC(C4(COC(C)C)CC4)=O)C3)=O)cc2s1 22981,N1(C(C2N(CC)CC2)=O)CCC2(CC1)CC2CNC(=O)CN1CC(C)(C)C1 22982,Cc1cc(NCCc2ncc(Br)cn2)ncc1S(=O)(=O)NC(C)(C)C1CC1 22983,C1(NC(C2C(NC(Cc3n(C)ccn3)=O)COC2)=O)CCCCC12CC2 22984,N1(C(c2cc(OC)nc(F)c2)=O)CCN(C(c2ccc(Cl)cc2Cl)=O)CC(O)C1 22985,c1(OC)ccc(F)c(C(c2nnnn2C(C)C)NCC(Cl)(Cl)Cl)c1F 22986,C1(CNC(=O)CC2=CCCC2)CC2CCC1N(C(=O)CC1CCC3CC3C1)C2 22987,N1(C(c2c(-c3cn(C)nc3)onc2)=O)CC=C(CCNC(=O)CC2CCC2)CC1 22988,C1(O)(C(C)NC(C(C)OCC=C)=O)CN(C(=O)C=Cc2ccc[nH]2)C1 22989,c1(COC)ccccc1NC(=O)CCC(=O)NC(c1cccc(C(F)(F)F)c1)C 22990,c1(C(N2CCCC(CCNC(C(CN(CC)CC)F)=O)C2)=O)cnc(O)cc1O 22991,c1(C(=O)NCCC(CNC(C(C2CCC2)OC)=O)C)ncccc1Br 22992,c1(OC)cncc(C(=O)NCC(C)Oc2ccc(C(C(C)C)SC)cc2)n1 22993,c1(CNC(CN(C)C(c2nnc(-c3c(F)cccc3F)s2)=O)=O)cc2c(s1)CCC2 22994,CC1CCC(C)N1CC(=O)NCc1ccc(C(=O)O)cc1 22995,c1(OC)ccc(C(N2CC3CC3(NC(c3cc(C4CCC4)[nH]n3)=O)C2)=O)c(N)c1 22996,N1(CC(=O)NC2(C)CC(NC(=O)CC3C=CCCC3)C2)CCCS1(=O)=O 22997,c1(C(=O)NC2CC3CC(NC(=O)CO)CC32)cc2ccccc2o1 22998,c1(NC(COC(C2CSC2)=O)=O)cccc(CC2CC2)c1 22999,c1(C(=O)NCC(C)(CC)NC(c2cnc(OCC)s2)=O)cc(OC)cc(Cl)c1F 23000,C1(C(N(CC(CN(C(=O)CC2CC(F)(F)C2)C)O)C)=O)CCC(F)(F)CC1 23001,CC(C)CC(F)C(=O)NCC1C2CCC(C2)N1C(=O)CNC(C1CCCC1)=O 23002,c1(OC)cc(F)cc(C=CC(=O)N(C(C)CNC(=O)C2=CCOC2)C)c1 23003,CCC(C)(CCNC(=O)Cc1nocc1C)NC(=O)COC1CCOCC1 23004,N1(C(c2cc(CCC)ncc2)=O)CCCC(C2CC2NC(C2CC=CCO2)=O)C1 23005,c1(C(=O)NCCN(C(C2CN(C)CC2c2cccnc2)=O)CC)ncc[nH]c1=O 23006,C(=O)(C(C(C)(C)S(C)(=O)=O)N(C)C)N1CC(C)C(CNC(=O)OC(C)(C)C)CC1 23007,N1(C(C(C)(C)NC(C2C(C)C2)=O)=O)CCc2ncccc2C1 23008,N1(C(CC2CCC(=O)N2)=O)CC2CC3CC2C1C3NC(=O)C1=CCC1 23009,CC(C)(O)C(C(=O)NOC1CC1)NC(c1ccc(=O)n(C)c1)=O 23010,C(=O)(C(O)CCCC)NCC1OCCN(C(C2(C=C)CC2)=O)C1 23011,N1(C(C=CC)=O)CCC2CN(C(C3CCN(c4nccn4C)C3)=O)C2C1 23012,C1(Cn2cc(CNC(c3cscc3-c3ccccc3)=O)nn2)CCC(C(=O)O)C1 23013,c1(NCc2cc(C)c(Cl)cc2)cc(Br)ccc1S(=O)(=O)N1CCCNC(=O)CC1 23014,N1(C(c2n[nH]cc2Br)C(=O)NCc2cccc(OC)c2)CCNC(=O)C1CCO 23015,C12(C(=O)NCCCOC)CC(NC3CN(C(=O)CCC4CCCC4)C3)(C1)C(C)O2 23016,c1(C(C(C)C)NC(=O)Nc2ccc(CCC(=O)OC)cc2)ccc2c(c1)OCCO2 23017,C1(OC)CN2CCCC2(C(=O)NC2CC(NC(c3c(Cl)cccc3Cl)=O)C2)C1 23018,N1(C(c2n[nH]c(C)c2C)=O)CC2CN(C(C3CCC([N+](=O)[O-])CC3)=O)CCC12 23019,N1(C(c2ccn(C(C)C)n2)=O)CCCC1C1CCCN1C(C1CC(O)C1)=O 23020,N1(C(C2C(CNC(C3CCCS3)=O)CC2)=O)CC(F)(F)C(F)(F)C1 23021,C#Cc1ccc(C(=O)NC2CN(C(=O)Cc3sc(C)nc3C)CC23CC3)cc1F 23022,CC1=CCSC1C(=O)NCC(C1CC1)N(C)C(c1cnc(C(C)C)[nH]1)=O 23023,Cc1ncnc(C(N2CCC(NC(=O)CC3C=CCCC3)C2C)=O)c1C 23024,C1(NC(CC)=O)(CNC(C2CCN2S(C)(=O)=O)=O)CCC(C)(C)CC1 23025,C1(O)(CC(=O)Nc2ccccc2Cl)CCN(Cc2ccc(O)nc2)CC1 23026,c1(C(N2C(CNC(C3N(C)CCCC3)=O)CC(O)C2)=O)ccc(N)c(Cl)n1 23027,C1(CN(C(CC(=O)OCC)=O)C)CN(C(C2(C)CCN(C)C2)=O)CCO1 23028,c1(C(=O)NCc2cn(C3CCN(C(C=C(CC)C)=O)C3)nn2)ccccc1C 23029,Cc1cc(N2CC(F)(F)CC2CNC(=O)CC(F)(F)F)n2ncnc2n1 23030,S(=O)(=O)(c1ccccc1Cl)NCCC(=O)N(C)CCNC(c1ccns1)=O 23031,c1(CC(N2CCN(CC3CCCN(C(COC)=O)C3)CC2)=O)csc2nccn12 23032,S(=O)(=O)(c1cccc(=NCC(C)c2cccs2)[nH]1)N(CC(C)C#N)CC 23033,N1(S(CCOC)(=O)=O)CCC(N=c2nc[nH]n3cc(Br)cc23)C1 23034,C1(NC(c2ccn(CCC)n2)=O)CC(CNC(c2cocc2C(N)=O)=O)C1(C)C 23035,C1(CNC(c2cccc(C)n2)=O)CN(C(=O)C(C)(C)C2CCCO2)CCN1C 23036,C1(C(C)C)CCC(NC(c2nc(NS(=O)(=O)CC#N)cn2C)=O)CC1 23037,C1(NC(CCCCCC)=O)CC2CN(C(c3cc(C)n(C(C)CC)n3)=O)CC2C1 23038,c1(C(=O)NCCC2OCCCN(C(C(C)C)=O)C2)ccc2c(c1)C(=O)NCCO2 23039,C1(S(N)(=O)=O)(C(=O)CC2CN(C(=O)OC(C)(C)C)C2)CC1.C12(CC(F)C1)C(=O)N2 23040,C(=O)(CC(C)C(C)(C)C)NCCN(C(C(CC)CC)=O)CC1CC1 23041,C(CO)(C(F)(F)F)NC(C(Cc1cc[nH]n1)NC(=O)CCn1cncn1)=O 23042,N1(C(C=C(C)c2cccs2)=O)CCN(C(c2ccc3cc[nH]c3n2)=O)CCC1C 23043,C1(C(N2C(CCNC(c3nc(C4CC4)cs3)=O)CCC2)=O)CCC2(CCC2)C1 23044,c1(OC)cccc(C(N2CCC(CF)(NC(=O)Cn3cccn3)C2)=O)c1 23045,c1(NC(C2CCN2C(c2cnc(-c3ccccn3)nc2)=O)=O)nc(Br)ccc1Cl 23046,N1(C(CCC=CC)=O)CCCCC(CCC(=O)NCCC(O)CCC)C1 23047,C#CCCCCC(=O)NCC(CC(=O)NCC(=O)OC(C)C)C1CCC1 23048,N1(C(C(CC)C2CCOCC2)=O)CCN(C(c2[nH]c(C)cc2C)=O)CC1CCO 23049,Nc1ccc(NC(N2CC(CC(=O)C(=O)O)C2)=O)cc1Cl 23050,CN1CCCC1C(N1CC(CCNC(C2CC2C2CC2)=O)C1)=O 23051,C1(C(=O)NC(C2CCN(C(=O)C(C3CCC3)C3CCC3)C2)C)CC(F)C(=O)N1 23052,c1(CNC(c2cnc(CC)s2)=O)ccc(CNC(C2COC(=O)O2)=O)cc1F 23053,C1(CC(=O)NCC(C)NC(c2nnc(C(C)(C)C)o2)=O)CCOCC1 23054,c1(SC)cc(F)ccc1C(=O)NCCOCCNC(=O)COCC(F)F 23055,C1(C(=O)NCC(C2CCCC2)C)CCN(C(C2(COC(C)(C)C)CC2)=O)C1CO 23056,N1(C(C(CC)n2ccnc2)=O)CCN(C)CC1C(=O)NOCC(O)CO 23057,CN1CC(NC(c2c[nH]c3cc(F)c(F)cc23)=O)CCc2ccccc21 23058,c1(OC(C)C(=O)NCC2(O)CN(C(=O)Cn3cnnn3)C2)cccc(Br)c1 23059,c1(C(=O)NC2CC(CCNC(c3coc(O)n3)=O)C2)cc(F)c2ncccc2c1 23060,c1(C(=O)NC(C)C(C)(C)NC(=O)CCNC(c2ccsc2Cl)=O)ncc(F)cn1 23061,Cc1ccc(C2CC2C(=O)NCC2CC(C)CCN2C(=O)C(O)C(F)F)c(Cl)n1 23062,c1(C(N2CC(NC(C3C(C(C)C)C3)=O)C3(C2)CC3)=O)cc(Cl)cc2ccncc12 23063,N1(C(CCCOC(C)C)=O)CC2(CC(NC(c3csc4nccn34)=O)C2)C1 23064,C1(CN(C(c2c(CC)con2)=O)CC)CCN(C(=O)Cc2ccccc2Cl)CC1 23065,N1(C(C(CCCOC)NC(=O)CCC(C)SC)=O)CCC2(CCC(OC)C2)C1 23066,CN1CC2C(CCN2C(C2CCCN(C(C3CCCC(N)C3)=O)C2)=O)CC1=O 23067,C(CN=c1ccc([N+](=O)[O-])c[nH]1)N(C(C(CCC)CC1CC1)=O)CC1CCCC1 23068,Cc1ccc(C(=O)N(c2cnncc2C)C2CC3(CNC3)C2)nc1 23069,c1(C(=O)NCC2C(C)CCN(C(C34CC(C)(C3)C4)=O)C2)ccc2nn[nH]c2n1 23070,c1(C(N2CCCN(C(C3CC4CCC3C4)=O)CC2)=O)ncc(F)cc1F 23071,n1(C(C)C)cc(C(=O)NC(C2CCOC2)CNC(c2cc(C(F)F)no2)=O)nn1 23072,N1(C(c2c(OC)cc(F)cc2)=O)CCCN(C(=O)CC(C)C)C(C)C1 23073,C1(NC(c2c(CC)c[nH]c2)=O)CC2CCC1CN(C(=O)CC(C)C(C)C)C2 23074,c1(NC(COc2ccc(C)cc2)=O)cc(N2CCC2)c(Br)cn1 23075,C1(C(=O)NCC2C(CNC(Cn3ccc(C)c3)=O)C2)CCC2(CC2)C1 23076,C1(NC(N2C(COCC)C=CC2)=O)CC2(C1)CC2C(=O)O 23077,N1(C(C2COC(=O)O2)=O)C(CNC(C2CCOC2)=O)CC2COCC12 23078,C1(CNc2cccc(C(F)(F)F)c2)CCC2(CCCC2)CC1 23079,N1(C(c2cnc(C(C)C)nc2)=O)CC(NC(C2CCCC2O)=O)CC(C)(C)C1 23080,N1(C(c2c(C)ccnn2)=O)C2CCCC1CN(C(c1cnc(O)cc1O)=O)C2 23081,CCS(=O)CC(=O)NCC1COCC1NC(=O)CSc1cn[nH]c1 23082,c1(CCC)c(C(N2CCCC(CNC(C3CCCN3CC)=O)C2)=O)nnn1CC 23083,C(=O)(C(CNC(c1cnsc1C)=O)CC(C)C)NC(c1c(C)nc(C)[nH]1)C 23084,Cc1cc(C(=O)NC(C)CCNC(=O)C=Cc2cnccc2C)ccc1C#N 23085,c1(-c2cnc3c(c2)N(C(C=CC=CC)=O)CC3)ccc2c(c1)n(C)c(=O)n2C 23086,c1(CC(=O)NCC2CN(C(c3occc3C3CC3)=O)C2)ccc2n[nH]cc2c1 23087,c1(C(=O)NC(C)CCNC(=O)C(C)C2CCC2)ncccc1C(F)F 23088,n1(-c2cc(C)on2)c(C)cc(C(=O)NCC(C)NC(=O)C(F)C(C)C)c1C 23089,C1(C(=O)NCCN2CCN(C(=O)Cc3ccc(F)cc3)CC2)CCCS1(=O)=O 23090,c1(N2CCC(O)CC2)nc(=NC2CCN(CC(F)F)C2)[nH]c2c1SCC2 23091,CC(C)C(CC(=O)NCCC1CCN(C(=O)CC(C)(C)C#N)C1)c1ccccc1 23092,C1(F)(C(=O)NCC23CC(CNC(C(CC)COC)=O)(OC2)C3)CCC(F)(F)CC1 23093,c1(CC)[nH]c(=N)sc1C(N1CC(CNC(=O)C=COCC)CC1C)=O 23094,C(=O)(C#CC1CCCCO1)N(CCCNC(C(CSC)C)=O)C 23095,C1(C(C)C(=O)NCc2cccc(Cl)c2)CCN(C(C2CCC(=O)C2)=O)CC1 23096,C#CC1(O)CC(C(=O)NC(Cn2ccnn2)C(=O)NC2CCN(CC)CC2)C1 23097,CCC(CCOC)C(=O)NC12CCC(CC1NC(=O)CCC#N)C2 23098,CC1CN(C(C2CC3C=CC2C3)=O)CC1NC(c1cnn(C)c1N)=O 23099,N1(c2c(S(=O)(=O)NC3CC4C(O)C3C4)cccn2)CCOCC2(CCCC2)C1 23100,N1(C(c2ncc(C)c(C)c2)=O)CC(NC(=O)CC2CCCCN2C)C2(CCC2)C1 23101,N1(C(c2ncn(C(C)(C)C)c2)=O)CC2(NC(=O)Cc3ccc(F)cc3)CC1C2 23102,C1(N(C(c2c(C)ocn2)=O)C)CCCC(N(C)C(c2ccon2)=O)C1 23103,C1(n2c(CSCc3ncc(C)o3)nnc2)CCCCCC1 23104,Cc1cccc(C(N2CCOCC2CCNC(=O)CC2CCC23CCC3)=O)c1F 23105,C1(NC(C(=O)NCC(c2ccc(CC)s2)=O)=O)CC2(CCC2)C1OC 23106,Cc1onc(Cl)c1C(N1CCC(Cn2cc(-c3nccnc3N)nn2)C1)=O 23107,C1(NC(COC(C)C)=O)C2CC1N(C(c1ccnc(CN(C)C)c1)=O)C2 23108,N1(C(CC2CN(C(c3c(C)nn(C)c3C)=O)C(C)C2)=O)CC2CCC(C1)N2C 23109,C1(CC(NOCCCCC)=O)CN(C(=O)CC2CCOC2C)CC1C 23110,C1(n2cc(CNC)nn2)CCCN(C(=O)C(C)(C)c2ccc(Cl)s2)C1 23111,C1(NC(COC(C2C(C)OCCC2)=O)=O)CC2CC1C1CC21 23112,C1(CC)CN(C(c2sccc2Cl)=O)CCN1C(=O)Cc1ccc(Cl)nc1 23113,c1(C(N2CC(CNC(C(c3c(C)cncc3)C)=O)C2)=O)cc2c(s1)CCSC2 23114,c1(CC(N2CCCC(NC(C=CC)=O)CCC2)=O)ccc2c(c1)CCCO2 23115,c1(C(C(=O)N(C(CNC(Cc2c(OC)cccc2)=O)C)C)C)cc(C)cc(F)c1 23116,c1(C(=O)NC(CCNC(CCC2CCC(C)O2)=O)(C)C)ccc(Cl)c(F)c1N 23117,C1(CC)C(NC(=O)C=C2CCC(C)C2)CCN1C(c1oc(C(F)(F)F)nc1C)=O 23118,C1(CNC(=O)CC)(NS(C)(=O)=O)CCN(C(=O)CC2CCOC2)CC1.CO 23119,c1(NC(c2nnnn2C2(C)CC2)C2CC(OC)C2)ccc2nn(C(F)F)cc2c1 23120,Cc1cc(C(N)=O)cc(C(=O)N(C)CCN(C)C(c2c(C)cccc2Cl)=O)c1 23121,C(C(=O)N1CCC(F)(CCOC)C1)(C(C)C)n1cc(-c2ccn(CC)n2)nn1 23122,C(C(CCCC)NC(=O)CNS(N)(=O)=O)NC(CSCCCC)=O 23123,CC(C)CCC(O)C(=O)NC(C(=O)Nc1ccc(CO)cc1)c1cccs1 23124,N1(C(C(C(C(CC)C)O)C)=O)CC=C(C(C)(C)C(=O)NCC(C)N(C)C)C1 23125,c1(C(C)NC(c2ccc(OC)c(F)c2N)=O)cc2c(cc1Br)OCCO2 23126,c1(CNC(=O)CNC(=O)Cc2nc(-c3cccc(O)c3)cs2)cc(I)ccc1O 23127,c1(CCC(N2CCCC(F)CC2)=O)ccc(S(=O)(=O)N2CCCC2)cc1 23128,C(=O)(C1CSc2ccccc21)NCCC1CC(NC(c2c(CC)nn(C)c2)=O)C1 23129,N1(C(C)=O)CCOC(C(=O)Nc2cnn(C)c2)C1.C12COCC1C(=O)N2C 23130,C(=O)(C(F)(F)CC(C)C)NC1CC2(C(NC(c3c(C)n(C)nn3)=O)C2)C1 23131,C1(C2CC2)(NC(c2c(C)cc(CC)o2)=O)CCN(C(C2CCCNS2(=O)=O)=O)C1 23132,CC1(NC(C2CCC(n3cc(-c4cncnc4)nn3)CC2)=O)CCCC1O 23133,c1(CN2CCN(C(C=Cc3c(C)cncc3)=O)CC2)c(Cl)cccc1[N+](=O)[O-] 23134,c1(N2CC(CC)C(O)CC2)nc(=NCC(C(C)C)N(C)C)[nH]c2c1COCC2 23135,C1(CNC(c2ncncc2Cl)=O)CCCCN1C(=O)CCc1cccc(Br)c1 23136,c1(C(N2C(c3cn(CCC=C(C)C)nn3)C(C)CC2)=O)cnn(C2CC2)c1N 23137,c1(SC)cc(Cl)nc(NC(N2CCCC(N3CC(C)(C)C3)C2)=O)n1 23138,C1(NC(c2cc(OCC)ncc2)=O)CN(C(=O)C(O)CC(N)=O)CC1(C)C 23139,N1(C(c2cncs2)=O)CC2CCC1C1CN(C(C3(CO)CCC3)=O)CC21 23140,c1(C(=O)NCC2CCCN(C(C3(O)C(C)(C)C3)=O)CC2)nc2ccccn2c1F 23141,c1(C(N(CC(CNC(C2C(C)OCCC2)=O)(C)C)C)=O)nccc2cccnc12 23142,C(CNC(=O)C(O)c1cnc[nH]1)(CCCC)NC(c1ccc(CC=C)s1)=O 23143,C1(CCN(C(=O)C(=O)NC(c2ccccc2)Cc2ccccc2)C)CCNCC1 23144,CC1(CCn2cncn2)CCN(CCC(=O)O)CC1 23145,C#CCCCCCCC(=O)N(CCCCNC(=O)CC(CC)OC)C 23146,CC(CC(=O)NC1CCN(C(c2cc(N)c(O)c(F)c2)=O)CC1)P(C)(C)=O 23147,N1(C(c2ccc(C(=O)OC)o2)=O)CC(NC(=O)Cc2csc(C)n2)C(F)C1 23148,CC1=C(C)C(OC(c2cnc(C3CC3)nc2)=O)CCC1 23149,c1(NC(c2c(C)ccnc2)C)[nH]c(=NCCC(C)(C)F)nc2c1cnn2C 23150,C12(CC(N3CC(C)(NC(c4c(C)cc(SC)o4)=O)C3)=O)CCC(CC1)CC2 23151,C1(CNC(CCCC2C(C)C2)=O)(CNC(=O)C(C)CCO)CCCCC1 23152,c1(C2(NC(C(COCC)n3cc(COCC)nn3)=O)COC2)c(C)[nH]c(C)c1C 23153,c1(SCC)ccc(C(N2CCCC(CCNC(c3ccc(Cl)nn3)=O)C2)=O)cc1 23154,C(=O)(C1=CC2(CCN(C(=O)C(O)Cn3cncn3)C2)C1)N(C(CC(CC)C)C)C 23155,N1(C(C(c2ccc(C)s2)C)=O)CCN(C(c2coc3c2CSC3)=O)CC(O)C1 23156,c1(OC)c(-n2cc(NC(=O)NC(C)CCC(=O)OCC(=O)O)nn2)cccc1F 23157,Cc1ccc([N+](=O)[O-])c(C(=O)NC(CNC(=O)C(C)CF)CC(C)C)c1C 23158,C1(CC)CN(C)C(=O)CN1C(=O)C(C)CNC(c1cc(F)n(C)n1)=O 23159,C1(C)(C(=O)NC2CCC(NC(CC(C)c3ccncc3)=O)CC2)CCN(C)C1=O 23160,C1(CNC(c2c(Cl)nc(OC)s2)=O)CCCCN(C(=O)C(C)C2CC2)CC1 23161,C1(C(N(CCNC(C2N(CCC#C)CCC2)=O)C(C)C)=O)CCCC(=O)N1 23162,CCC(C)C(C(=O)NC1(C)CC(NC(c2cccc(NC(=O)OC)c2)=O)C1)OC 23163,C(C(F)(F)CCC(=O)NC(C)CCc1ccc(C)cc1)n1cc(CCOC)nn1 23164,c1(C(=O)NC2(CNC(C3(OC)CCOCC3)=O)CCOC2)cc2ncccc2o1 23165,C(=O)(CCC#Cc1ccccc1)NC1C(C)(C)C(CNC(C2(CO)CCC2)=O)C1 23166,C1(CNC(C2CC(=O)NCC2)=O)CCCCN(C(=O)CCn2cnnn2)CC1 23167,C1(C(=O)NCC(F)CNC(c2sccc2C2CC2)=O)(COC)CC=CCC1 23168,CC1Oc2c(C(=O)NC3(CCNC(c4cccs4)=O)CC3)cccc2NC1=O 23169,N1(C(c2c[nH]c(=N)s2)=O)CC2CCC(NC(=O)Cc3ccc(F)cc3)(C2)C1 23170,Cc1c(C(=O)NCC(F)CNC(=O)CC2(C(F)(F)F)CC2)cccc1O 23171,CCCCCC=CC=CCC(=O)NC(C)CC(C)NC(=O)CN(C)C 23172,C1(C)(CNC(C(C)Sc2ccccc2)=O)CCCN1C(=O)Cc1cnccn1 23173,C#Cc1ccc(NC(=O)C(CC(F)F)NC(=O)CC=CC)cn1 23174,c1(N2CC(O)(CCNC(CC(CC)C3CC3)=O)C2)ncnc2[nH]cnc12 23175,C(=O)(C(O)CNC(=O)CCC1CC1(F)F)NC1CC(COC)C1 23176,N1(C(C2(c3c(C)ncs3)CC2)=O)CC2(CCN2C(=O)CCCCNC(N)=O)C1 23177,CCCCC(O)CCC(=O)N(CCCCN(C)C(c1ccc2nc[nH]c2c1)=O)C 23178,C12CCN(CC1)C2=O.N1(NC(C(=O)N(CC=C)CCOC)=O)CC(C)(C)C1 23179,N(C1CCc2c(Br)cccc21)C(c1ccncc1-c1cccc2nc[nH]c12)=O 23180,C1(NC(C(CC)SC)=O)Cc2ccccc2C1NC(=O)C(C(C)C)NCC(C)C 23181,c1(CNC(Cn2ncc(CC)c2)=O)cccc(C(=O)NCc2[nH]nnc2C)c1 23182,C1(C(N2CCN(S(CC)(=O)=O)CC2C)=O)CC2(CCO1)CC(F)(F)C2 23183,c1(Cc2nnc(C(CCC)N(C)Cc3ccncc3)o2)ccc(F)cc1 23184,c1(OCCC(=O)NCC2CCCN2C(c2nn[nH]c2Cl)=O)ccccc1F 23185,CC1CCCC(C(=O)NC2(C)CC(C(=O)NCC3CC3C3CCC3)C2)C1 23186,N1(C(C=CC(=O)OCC)=O)CCC2(CC1)CC2c1ccc(F)cc1 23187,C1(NC(=O)COC2CCCC2)CCC2(CCN(C(c3cn[nH]c3)=O)CC2)C1 23188,C1(NC(c2cnn(CC)n2)=O)CCC2(CC1)CC2NC(=O)CCC1CCCCO1 23189,c1(CC(=O)NC(C)C(CO)NC(c2nn(C)cc2N)=O)cnc2cccnn12 23190,S(=O)(=O)(c1c(C)sc(C)c1C)NCC(CCCC)NC(=O)NC(C)(C)C 23191,C1(COC)CCCCN1C(C1CC2CC2N1C(C1CCCCCC1)=O)=O 23192,N1(CC)CCC(NC(=O)C(CC2CCCC2)NC(=O)C=CC(C)(C)C)C(C)C1 23193,O=C1CCc2cc(-c3ccnc(CC(=O)NCc4ccc(O)cc4)c3)ccc2N1 23194,O=C(C1=CCCCCC1)NCC12CCC1CN(C(c1nncs1)=O)C2 23195,CC(CC(=O)NCCC1CCN(C(c2cnc(Cl)cc2N)=O)C1)C(C)(C)C 23196,C1(NC(CCc2c(C)cccc2)=O)CC(O)CN(C(c2cc(CF)on2)=O)C1 23197,c1(C(=O)OC)cnn2c1CC(Nc1nn3cc(CC(C)C)nc3s1)CC2 23198,C(=O)(C(CC(C)C)C(C)C)N(C(C(=O)NC1CC(COC)C1)C)C1CC1 23199,Cc1c(N2CCCC(CNC(=O)CCc3nc[nH]n3)CC2)ncnc1Cl 23200,c1(C(N(CC(=O)NC2(C3CCC3)CCC2)CC#C)=O)c(Cl)nsc1Cl 23201,C12(NC(c3ccc(CC)c(C)c3)=O)CCCC1N(C(c1cncn1C)=O)CC2 23202,c1(C(N2CCN(C(C3C(C)(C)NC(=O)C3)=O)C(CO)C2)=O)cnn2ncccc12 23203,C(=O)(C1Cc2ccc(F)cc21)NC12C(CN(C(CS(CC(=O)OC)(=O)=O)=O)C1)C2 23204,N1(C(C(C2CCCO2)C(=O)OC(C)(C)C)=O)C=CCCC2CCCC12 23205,Cc1cc(CNC(=O)NC2(n3cnnn3)CCCCC2)cnc1Br 23206,C12(NC(Cc3c(C)occ3)=O)CCCN(C(c3ccc(Cl)c(F)c3F)=O)CC1C2 23207,C(=O)(C1=NOC(C(C)(C)C)C1)N1CCCC(N(C(C2C3CCC(F)C23)=O)CC)C1 23208,N1(C(C(COCC)OC)=O)CCN(C)C(C(=O)NOC2CCCC3CC23)C1 23209,c1(NC(=O)NC(c2ccc(N(C)C)cc2)C)c(Br)sc(Cl)c1Cl 23210,C(=O)(C1=CC2C=CC1C2)N1CCN(CC(C)NC(C2=CCCC2C)=O)CC1 23211,C(F)(c1ccccc1)=CC(=O)NC(CNC(C(COC)OC)=O)CC(C)C 23212,Cc1ncncc1C(N1CC(NC(C2CCCCC2)=O)C(C)C1)=O 23213,C1(CC(N2CCN(C3CCN(C(=O)CC4(CO)CC4)C3)CC2)=O)CC2CCC1CC2 23214,C(=O)(C(O)CC(C)(C)C)NCCc1cc(C(N(C)Cc2cc(C)nn2C)=O)no1 23215,C1(NC(C(N2C(C#C)CC2)=O)=O)CC(=O)N(C)C1c1ccc(F)cc1 23216,Cc1ccc2c(c1)C(NC(=O)CN1CC(C)CCC1c1ccccc1)CCC2 23217,N1(C(c2ccc(N(C)C)cc2)C(=O)NCC(=C)C)CC=C(c2ccccn2)CC1 23218,C(CN=c1cc(C)nc(-c2cccc(Cl)c2)[nH]1)NC(CCN(CCC)C1CC1)=O 23219,c1(CC(=O)NC(Cn2cc(C3(C)CCCO3)nn2)CC2CC2)c(F)cccc1Br 23220,N1(C(CC(C)C)=O)C(C(=O)NC(c2c(CN3CCCC3)cncc2)=O)CC2CC12 23221,CC(C)C(C(=O)NCCCCNC(=O)CCC1CCC1)S(=O)(=O)C1CCCCC1 23222,C(=O)(C(F)CC(C)(C)C)OC(C)(C)C.CC1CC2CN1C(=O)NCCC2 23223,c1(C(N2CCC3(CCCN3C(=O)C(F)C3CC3)C2)=O)ccc([N+](=O)[O-])cc1O 23224,C(C1COCc2ccccc21)NC(=O)NC1CCCC(C)(C)O1 23225,C1(C(=O)NC2CC(N(C(c3[nH]cc(C(C)=O)c3C)=O)C)C2)CC(=O)NC1(C)C 23226,CC1ON=C(C(=O)N2CC(NC(=O)Cc3c(Cl)cnn3C)C(C3CC3)C2)C1C 23227,c1(OC)ccc(F)c(F)c1CN1CC(NC(c2ccc(Br)c(CO)c2)=O)C(F)C1 23228,N1(c2nnc(CC)n2C)CC(C)N(c2nc(C)ncc2F)CC1C 23229,C1(NC(C)=O)CCC(C(N2CCC(NC(c3cn(C(C)C)cc3C)=O)C2C)=O)CC1 23230,N1(C(c2c(C)n[nH]c2)=O)CC2CC1(CNC(=O)C(C)(O)Cc1ccccc1)C2 23231,c1(C(N2CC(C(C)NC(c3c[nH]cc3-c3ccccc3)=O)C2)=O)nnc(S)n1C 23232,N1(C(C=CC=CC)=O)CCc2ccccc2C1CNC(=O)CCc1scnc1C 23233,N1(C(c2cncc(C(C)(C)C)c2)=O)CCN(C(c2csc(Cl)c2Cl)=O)C(CF)C1 23234,c1(-c2cc(NC(C3CC3F)=O)sc2)ccccc1-c1ccco1 23235,c1(NC(C(CC)(C)CNC(=O)C(C)NC=O)=O)cnc2ccnn2c1 23236,C(=O)(C1=CC2CCCC12)Nc1cccc(CNC(=O)C=Cc2cocn2)c1 23237,N1(C(c2c(C)cc(F)s2)=O)CCCC2(CCCN2C(c2cncs2)=O)C1 23238,c12c(ncn1C)-c1cncc(c1)NCCCC2.C(=O)(C1CC1)OCC 23239,Cc1cccc(C)c1CC(N1CCCC(NC(C2(O)CCC2)=O)C1)=O 23240,CC1=C(C(=O)NCC2CCCN(C(=O)CCCc3nccs3)C2)CCC(C)(C)C1 23241,c1(C(N2C(CNC(c3noc(CC)c3C)=O)C=CC2)=O)ccc(P(C)(C)=O)cn1 23242,C1(CNC(c2nccn3ccnc23)=O)CCN(C(=O)CSC2CC2)CC1(F)F 23243,S(=O)(=O)(c1cccnc1N1CCC(CN2CCC(O)C2)CC1)N(CC(CC)C)C 23244,N1(C(C2(c3c(C)cccc3)CC2)=O)CC2CC(NC(=O)C(C)NS(C)(=O)=O)C1C2 23245,c1(CC(=O)NCC(=O)NCCC(C)N(C(CCSCC)=O)C)cc(C)no1 23246,Cn1nc(C(=O)N(c2ncccc2Br)C2CC2)c2c1CCCC2 23247,c1(N2CCC(NC(c3nc(Cl)ccc3F)=O)(CF)C2)ncc([N+](=O)[O-])cc1Br 23248,C(=O)(C1=C(CC)OCCS1)NC1CCC(CNC(c2n(C=C)ncc2)=O)CC1 23249,N1(C(C=CCN(CC)CC)=O)CCC2(NC(C3CN(C)C3)=O)CCCCCC12 23250,C1(CC=C)(NC(=O)C=CBr)CN(C(=O)C(C2CCOCC2)OCC)C1 23251,N1(C(C(=O)C2CC2)=O)CCC2(CCCCC2NC(=O)CCCCCF)C1 23252,CCC(CC(F)(F)F)C(=O)N1CC2(CNC(C3CCC(C)CC3)=O)CC1CO2 23253,c1(C(=O)NCCN(C(=O)CC2CCCC23CC3)C(C)C)ccc(C(F)(F)F)cn1 23254,c1(C(N(CC(C)(C)CNC(=O)CC=C(C)C)CC)=O)cc2sc(C)cc2[nH]1 23255,N1(C(CCC2C(C)C2)=O)CC2CN(C(c3ccccc3CO)=O)CC2(C)C1 23256,CC1(C)CCC(CNC(=O)CC2(C3CC3)CC2)N(C(C2(C)CCCS2(=O)=O)=O)C1 23257,N1(C(c2nc(C(C)NC(C=CC(C)(C)SC)=O)oc2)=O)CCc2ncsc2C1 23258,c1(C(=O)NC(C2CC2C(=O)Nc2cncc(Cl)c2)C)ccnc(O)c1 23259,O=C(C(F)C(F)(F)C(F)(F)F)N1CC2(CCCN(C(C3(CO)CC3(F)F)=O)C2)C1 23260,C1(NC(c2cc(CNC(c3cn(C(C)C)nn3)=O)on2)=O)CCc2ncnn2C1 23261,C(C(=O)N=S(C)(=O)c1cnn(CCF)c1)c1cc(CC)c(F)cc1 23262,C#CCCCC(=O)NC1CCOC(C2CCN(C(=O)Cn3ccsc3=N)CC2)C1 23263,N1(Cc2c(OC)nsc2)CCC(C(C)(C)NC2CCCN2C(=O)CO)CC1 23264,c1(C(=O)NC2C(NC(C3(C)CC4CC4C3)=O)CCOC2)cc2nn[nH]c2cc1F 23265,Cc1nc2ccccn2c1NC(N1CC2CC(C1)N2C(C1CCC(F)(F)C1)=O)=O 23266,c1(Cn2cc(CC3N(C(CC4CN(C)C4)=O)CCC3)nn2)ccc(F)cc1 23267,C1(CN(C(=O)C=CI)C)COCCN1C(=O)Cn1cnnc1O 23268,N1(C(C2(C#C)CC2)=O)CCC(C(=O)Nc2cnccc2C)C(C)(C)C1 23269,C(=O)(C(O)CC(N)=O)N(CCCNC(=O)C=C1CCN(C)C1)CC 23270,C(=O)(CCC(C)NC(=O)CC1CC2(CC2)CO1)NCc1c(C)occ1 23271,C1(C)(C(=O)NC(C(C)C)CCNC(c2coc3c2COC3)=O)CCCNS1(=O)=O 23272,c1(N2CC(O)(C(C)NC(c3nn(C(CC)CC)c(C)c3)=O)C2)cc(O)nc(=O)n1C 23273,N1(C(C(n2ccc(C)n2)C)=O)CC(NC(C2CCCC(C)C2)=O)CC(F)C1 23274,C1(CC)(CO)CCCN(C(=O)CC2COCCN2C(c2ccc(C(N)=O)o2)=O)C1 23275,CC(C)CCC(C(=O)NCCCc1ncn(C)n1)NC(C1CC1(F)Cl)=O 23276,N1(C(CC(C)C)=O)CCN(C(=O)C(C)NC(=O)OC(C)(C)C)CC2(C)CCCC12 23277,C1(NC(c2cccc(C(=O)NC)n2)=O)CN(C(c2cc(Cl)c[nH]2)=O)CC1(C)C 23278,C1(C(N2CC(CCCCC)C2)=O)CCN(C(=O)C(C)CCOC)CC1C 23279,N1(C(=O)CC2CC2(Cl)Cl)CCC(O)(C(F)(F)F)CC1 23280,CC1CCN2N=C(C(=O)NC3CCN4CC3C4CCC)NC2=N1 23281,N1(C(=O)OC(C)(C)C)CC(CNCC(C2CC(C)(C)CO2)O)C(F)C1 23282,c1(C(C(=O)NC)N(c2cc(Br)ccc2OC)CC2CC2)cn2c(Br)cnc2s1 23283,N1(C(C(CC)N(C)C)=O)CCCC(C)(CNC(=O)CCc2cnco2)C1 23284,N(C1CCCc2ccc(F)cc21)C(C(CC)OC1CCCCC1)=O 23285,c1(SC)nccc(=NC(=O)CC2CN(C(=O)C=C(C)C)CCO2)[nH]1 23286,CC1OC2(C(=O)NCC3CC(NC(=O)C#CC(C)C)CCO3)CCC1CC2 23287,C(C1CN(C(=O)CC(C)O)Cc2ccccc21)NC(Cc1ccn(C(C)C)n1)=O 23288,N#CC1CN(C(=O)C=Cc2ccc(O)cc2)CCN1Cc1cc(Cl)cc(Br)c1 23289,C1(CC)CN(C(C2CCCC2F)=O)CC1C(=O)NC1CCCC1CN(C)C 23290,C1(CNC(CNC(CC)=O)=O)CC12CCN(C(=O)C(C)(O)CC(C)C)CC2 23291,N1(C(c2ccnc(Br)c2F)C(=O)NCCSC)CC(CO)OCC12CCOCC2 23292,C(=O)(C1=CS(=O)(=O)CCC1)NC1C2(CN(C(C3=NOC(C)C3)=O)C2)CCC1 23293,C1(C(=O)NC2CCOCC2NC(c2cc[nH]n2)=O)(COC)C=CCCC1 23294,c1(C(N2C3CN(Cc4cn(CC)nc4)CC2C3)=O)ccc(C#N)cc1Cl 23295,CC1(C)NC(=O)CCC1NC(c1n[nH]c2c1CN(C(c1sccc1Cl)=O)C2)=O 23296,c1(OC)ccc(C(=O)NC2CN(C(c3sc(Br)nc3C)=O)C2)c(OC)c1 23297,C1(F)(C(N(CC(C)N(C(C(c2cc(F)cc(F)c2)C)=O)C)C)=O)CCN(C)CC1 23298,N1(C(C(C)c2cccs2)=O)CC2(C1)OC1(CO)CC2(NC(C2C=CCS2)=O)C1 23299,N1(CCN(C)C(c2conc2C2CC2)=O)C(=O)CNC1=O.C12CCCN1CC2 23300,Cc1nccc(C(=O)NCCC2(C(=O)NC3CC3C)CC2)c1N 23301,C#CCCCCC(=O)NC1(C)CC(NC(=O)C=Cc2cc(Br)cs2)C1 23302,C(=O)(C(F)C(=O)N1CC(F)CC1C(=O)NC(CC)C1CC1)OCC 23303,CC1CN(C(=O)C=CC2CCC2)CC2(CCN(C(C3CCC(C)(C)O3)=O)C2)O1 23304,O=C(CS(=O)(=O)c1ccncc1)N(C1CCCC1)CC(F)F 23305,O=C(N=c1[nH]nc2n1CCCS2)N1CC2CC1C1OC(C)(C)OC21 23306,CCCS(=O)(=O)CC(=O)N1CCN(C(=O)CCOc2ccccc2F)C2CC12 23307,Cc1cc(=NCC2(N3CCCCC3C)CC2)[nH]c(N2CCc3ncncc3C2)n1 23308,c1(C(=O)NC(CC=C)CNC(c2ccc(CO)cc2)=O)c(F)ccc2n[nH]cc12 23309,N1(C(C2(C#C)CCC2)=O)CCC(C2CCCN(C(=O)C(C)C(C)(C)C)C2)CC1 23310,N1(C(CC(CCC)C)=O)CC2CCC(N(C)C(c3ncc(F)cc3C)=O)C2C1 23311,N=C1NC(=O)C(CC(=O)NCC2(CNC(=O)C(O)Cc3cnc[nH]3)CC2(F)F)S1 23312,C1(CNC(c2c(CC)ncs2)=O)C(O)C(O)CN1C(=O)CN1CCCC1=O 23313,CC12CC(C(N3CC(CNC(C4CCC(F)C4)=O)C3)=O)(C1)C1(CCC1)O2 23314,C(=O)(C#CC1CCOCC1)NC(C1CCCN1C(c1cc(C(F)(F)F)n[nH]1)=O)C 23315,C1(C)(C(N(CCNC(=O)C(c2ccccc2)C2CC2)CC)=O)CC(OC)CN1C 23316,c1(C(N2CC(N(C(c3ccc(CC)[nH]3)=O)C)C(C)CC2)=O)ncn2c1COCC2 23317,C1(CNC(C(Br)=C(C)C)=O)CC2(CC2)CN1C(C1CC(C2CC2)=NO1)=O 23318,c1(C(N(CC(C)NC(C(CSC)C)=O)C)=O)cc2ccc(Cl)cc2c(O)n1 23319,N1(C(c2ccc(C)cn2)=O)CCCC(NC(C2CCCCO2)=O)C1C 23320,C1(CNC(c2c(C)nc(Br)o2)=O)CN2CCCCC2CN1C(C1COC1)=O 23321,c1(CC(=O)NC2CC(NC(C3(c4cccc(Cl)c4)CC3)=O)C2)cc(O)nc(O)n1 23322,c1(C(=O)NC2CCN(C(C(CC)NC(C)=O)=O)CC2F)cc2n(n1)CCNC2=O 23323,N1(C(C(=O)N(C)C2CC2)C2CC2(Br)Br)CCCC(C2CCC2)C1 23324,c1(C(=O)NCC2(F)CC(NC(C3CCSC3)=O)C2)cccc(CC(F)(F)F)c1 23325,CC1=NNC(=O)C1CC(=O)NCC1(CN(C)C(c2ccn(CC(C)C)n2)=O)CC1 23326,CCCC(CNC(=O)CC1(NC(=O)CCCCOCC)CCCCC1)CCO 23327,C(=O)(CS(=O)(=O)CC(C)C)N1CC(O)(CCNC(c2c(C)ccc(C)c2O)=O)C1 23328,C(CCC(=O)N1CC(O)(C(C)NC(=O)C(C2CC2)OC)C1)=CCC=C 23329,C1(CNC(c2ncn(C)n2)=O)CN(C(=O)Cc2n[nH]c(=N)s2)C(C)(C)C1 23330,CC1CCCN1CCCn1cc(CC2COC(=O)C2)nn1 23331,C=CC1(CC(N2CCC2(C)C(=O)OC)=O)CN(C(=O)C(CN(C)C)CC)C1 23332,N(C(=NCCc1csc(C)n1)NC1CC(c2ccccc2Br)C1)C(C=C)C 23333,n1(CC)nnc2cc(C(=O)N(C)CCN(C(=O)CNC3CC3C)C3CC3)ccc12 23334,c1(N2C(C)(CNC(C(N3CCSCC3)C)=O)CCC2)nc(Cl)nc2[nH]c(O)nc12 23335,C1(C(N2CCC(CCCO)C2)=O)CC2CC2N1C(=O)C(O)c1ccsc1 23336,c1(C(N2CC(Cn3cc(-c4scc(C)n4)nn3)OCC2)=O)c(O)ncc2c1CCC2 23337,N1(C(C(CCSC)(C)C)=O)CC2ON=C(CNC(c3coc(C(F)F)n3)=O)C2C1 23338,c1(N2CC(NC)C3(C2)CC3)ncc(C)cc1S(=O)(=O)NCc1cc(Cl)nc(Cl)c1 23339,Cc1nscc1C(=O)NC1CCC(NC(=O)C(C)N2CCC2)C1 23340,c1(N2C(C)C(NC(=O)CC3(CO)CC3)CCC2)ncc2ccnc-2[nH]1 23341,N1(C(C(N2CCN(C)CC2)C)=O)CC2CN(C(C3OCCO3)=O)CC(C1)O2 23342,c1(CSC)cccc(C(=O)NC2(C)CCN(C(c3nncs3)=O)C2)c1 23343,CC(C(O)C(F)F)NC(=O)C(C1CCCC1)NC(=O)CC1(C)CCOC1 23344,C(C)(CN=c1[nH]c(Cl)ncc1F)(C1CC1)NC(C(C(C)C)O)=O 23345,C1(OC)CCN(C(=O)C(CN)C2CCCCC2)CC1(C)C 23346,N1(C(CN(CC)CC)=O)CCC(C)(C)C1CNC(=O)CCc1ccc(C)c(Cl)c1 23347,N1(C(COC)=O)CC2CCCC(NC(C3CCC=CCC3)=O)(C2)C1 23348,N1(C(C(CC=C)C(C)C)=O)CC2(CCN(C(c3cc(C)ns3)=O)CC2)CC1C 23349,N1(C(C(CN(CC)CC)F)=O)CC2CCN(C(c3cc(C)ccc3F)=O)CC2C1 23350,c1(CNCc2occ(CO)n2)cccc2c1OCC2 23351,C(CC(C)(C)CC(=O)N(C(CC(C)C)C(=O)NCCc1cc[nH]n1)C)OC 23352,C1(NC(=O)CC(O)C2CC2)CCCOC12CCN(C(=O)CCC1(O)CCC1)CC2 23353,CC1(C)CC(C(=O)NCC(CC(=O)NCCSC(F)F)C2CCC2)CCO1 23354,c1(OCCOC)ccc(Cl)cc1C(=O)NCC1CN(C(=O)C(C)CF)CCO1 23355,CC(C)C(C)CC(=O)N1CCCCC1CCCNC(=O)Cc1ccccc1O 23356,c1(OC)nccc(Br)c1C(=O)N(C)CCNC(C1CCSC(C)C1)=O 23357,N1(C(c2c(OC)cc(Br)cc2)=O)Cc2[nH][nH]c(=NC(=O)C3CC4C=CC3C4)c2C1 23358,c1(C(N2CCC(OCCNC(CCC#CC)=O)C2)=O)cc(C)c(O)c(C)c1 23359,c1(C2(N(C)Cc3ccccc3OC(F)F)CCC2)[nH]c(=N)c(C#N)cc1C#N 23360,CCCCC(CNC(=O)CCSc1ccccc1)NC(=O)CCC1CCCN1C 23361,C(=O)(C1=NNC(=O)CC1)NCC1N(C(c2cc(CCOC)on2)=O)CCN(C)C1 23362,C1(O)(CC(=O)N(C)CC)CCN(C(=O)C(O)Cn2cncn2)CC1 23363,C1(C(=O)N(C(C)CCNC(=O)C(C(C)O)N(C)C)C)(COC)CCCCO1 23364,CC1=C(C(=O)N2CCCC(N(C)C(c3coc(C(F)F)c3)=O)C2)CCC1 23365,c1(NC(C)=O)cccc(C(=O)NC(C)CC(C)NC(c2ccccc2CO)=O)n1 23366,c1(OCC)ncccc1NC(c1cnn(CCN(C(=O)CC2(O)CCC2)CC)c1)=O 23367,S(=O)(=O)(c1cccc2cnccc12)N1CC2C(C(=O)Nc3cccc(C)n3)C2C1 23368,C(C(CC1CC1)C(=O)NOCC1CCCO1)NC(c1c(OC)ccs1)=O 23369,c1(C(=O)NCC2CN(C(c3c(OC)n[nH]c3)=O)CC2C)cc(F)cc([N+](=O)[O-])c1 23370,CC1(NC(=O)C(C2CCOCC2)SC)CCCN(C(=O)CSc2ccccc2)C1 23371,c1(C(=O)NCC2(O)CN(C(C(C)NC(CC)(C)C)=O)C2)cc(Br)cn1C 23372,CC1(C)CC(NC(c2ccco2)=O)CN(C(C2CC2(F)F)=O)C1 23373,c1(CCC(=O)N(C2CN(C(CN(C)Cc3ccccc3)=O)C2)C)cnc(O)[nH]1 23374,c1(OCC)cccc(C(=O)NCC2(NC3C(C)C3C)CCOCC2)c1[N+](=O)[O-] 23375,C=C1CC2(C1)CC(C(=O)NCC(C)CNC(=O)C(O)C(C)CC)C2 23376,C(=O)(CC(C1CC(F)(F)C1)NC(c1ncoc1C(C)N)=O)OCC 23377,c1(C(=O)OCCC(=O)Nc2ccc(OCC)cc2C)cnc2ccccn12 23378,N1(C(C2CCN(C(C(C(C)C)CN(C)C)=O)CC2)=O)CCCOC(C)(C)C1 23379,C1(CC)CCC(C)CN1C(c1c[nH]nc1CNC(c1cnc(Cl)s1)=O)=O 23380,C1(N(C(=O)CCc2cn[nH]c2)C)CCCN(C(=O)C(C)(C)c2ccccn2)CC1 23381,C1(O)(CC)CCC(NC(=O)CC(C)(C)CNC(C2CCCOC2)=O)CC1 23382,N1(C(C2CCCN(CCC)C2)=O)CCC(NC(=O)CN2C(C)CCC2C)C(F)C1 23383,CC1CCN(C(C2(C)CC2)=O)C1CNC(=O)Cn1cnnc1 23384,c1(C(=O)OC)cc(CC(=O)NC(C)CNC(c2[nH]ccc2C2CC2)=O)cs1 23385,c12cncc(c1)NC(=O)C(=O)N2.C1(OC)COCC1Cc1ccccc1 23386,C1(C(N2CC(NC(C3CCC(C)(C)O3)=O)(CO)C2)=O)CCC2CC2CC1 23387,N1(C(CC)=O)CC2CC1C2CNC(C1(C)CC1(F)F)=O.CCC(=O)NCC=O 23388,c1(-c2nc(Cc3ccc(C)nc3)n(C3CCS(=O)(=O)C3)n2)ccc2nc[nH]c2c1 23389,c1(C(N2CCN(C(Cn3ccc(C)n3)=O)CC2CF)=O)ccc(O)c(C)c1C 23390,C1(NC(C=COCC)=O)COCCC1NC(=O)C(O)CCc1ccccc1 23391,n1(CNC(COCCCOC)=O)cc(C(=O)N(C)CCC2CCOC2)nn1 23392,C(=O)(C1=NOC2COCC12)N1CC(CC=C)(C(N2CC3CCC=CC23)=O)C1 23393,CC1(C)C(C(=O)NCC2(N3CCNC3=O)CC2)CCN1C(=O)C(=O)NC1CC1 23394,C1(CC2(O)CCN(C3CC(=O)N(CC)C3=O)CC2)COC2(CCCC2)O1 23395,C1(C(N(CCCC)CCO)=O)CN(C(C2CCCOC2)=O)C(C)(C)C1 23396,C12(OC)CCC(C(=O)NC(C)(CNC(c3cscc3F)=O)C3CC3)(CC1)CC2 23397,c1(C(=O)NC2CC3CC(NC(C(C(C)(C)O)F)=O)C2C3)ccn2cccc2c1 23398,C(=O)(C(O)(C(C)C)C(F)(F)F)N1CCCCC(NC(c2c(C)scc2)=O)C1 23399,N1(C(CCC)=O)CCN(C(c2occ3c2CCC3)=O)CC1CC(C)(C)C 23400,C1(C(=O)NCC(CNC(C(C=C)C)=O)(C)F)CC(C)(C)CN1C 23401,C(=O)(C(CC(F)F)c1ccccc1)NC(CC)(C)CN(C)Cc1cc(C)cnn1 23402,N1(C(C(C)C)=O)CCN(C2CCC(NC(=O)C(N3CCC(C)(O)C3)=O)C2)CC1 23403,c1(C(C(=O)NC(CCOC)CNC(c2cc(C)sn2)=O)C)cccc([N+](=O)[O-])c1 23404,N1(C(Cc2nc(=N)[nH][nH]2)=O)CCC(NC(C2CC2F)=O)C12CCC2 23405,C1(NC(C2N(CCC(C)C)CCC2)=O)CN(C(=O)Cn2nccn2)CC1CO 23406,N1(C(C(C(C)O)C)=O)CCC(C2(NC(=O)CCc3ccccc3)CC2)C1 23407,C1(NC(NOCC(C)(C)C2CCCC2)=O)CC2(C1)CC(C#N)C2 23408,C(=O)(CC(F)(F)C(F)F)N1CCC(N(C(c2cc(CCC)oc2C)=O)CC)C(F)C1 23409,C(=O)(C(O)(C(C)C)C(F)(F)F)NCC(C)NC(Cc1c(C)ccnc1)=O 23410,C1(CC=C)(C(=O)NC2CCCCC2F)CCN(C(C2CCN2C)=O)C1 23411,C1(CNC(c2cccc(C)c2N)=O)CCC12CCN(C(C1CC13CC3)=O)CC2 23412,c1(NC(C2C(NC(N3CCOC3=O)=O)C2)=O)cnc2ccccc2c1Cl 23413,Nc1cncc(C(N2CCCCC2CCNC(c2cc(CO)ccn2)=O)=O)n1 23414,C1(C(=O)NCCN(C)C(c2ccc(-c3nccs3)cc2)=O)CS(=O)(=O)CC12CC2 23415,Cc1c[nH]cc(C(=O)NCC(F)CNC(c2ccc(N)c(F)n2)=O)c1=O 23416,C1(NC(COCc2onc(C)n2)=O)CN(C(C2CCN2C(C)(C)C)=O)CC1F 23417,Cc1cc(C(N2CCN(C(c3ccc(Br)c(O)n3)=O)C3CC23)=O)nc(C)c1 23418,Cc1cnc2n1CC(C(N1CCCOC(CNC(C3CCSCC3)=O)C1)=O)CC2 23419,N1(C(C(CCOC)C)=O)CCC(NC(C23CC2COC3(C)C)=O)C(C)(C)C1 23420,c1(C(=O)NCCCNC(C(c2cccc(C)c2)(C)C)=O)ccc(F)c2[nH]ccc12 23421,c1(C(=O)NC(C2(C)CCCC2NC(c2nn(C)cc2Cl)=O)C)cccnc1CO 23422,C=CCC(C(=O)NCC1(O)CCCC1)NC(c1sccc1Cl)=O 23423,C1(CC(=O)NC(CCCNC(C2CC(OC)C2)=O)c2ccccc2)CCCCO1 23424,c1(NC(C(CC)C)C)cc(N2CCN(C(C)C)CC2)nc(C(F)(F)F)n1 23425,c1(OC)cccc(CCC(N2CCCC2(C)c2cccc(F)c2)=O)n1 23426,N1(C(c2cnn(C)c(=O)c2)=O)CC(C(N2C3C=CCC2CC3)=O)CCC1(C)C 23427,CCCCC(C(=O)NC(C)CCCCNC(C)=O)N1CCCS1(=O)=O 23428,CC(F)(F)CCCC(=O)NCC(C1CCCCC1)NC(C1OCC1(C)C)=O 23429,C1(CCC#C)CCCN(C(=O)CC(C)(C)OC2(C(=O)NCC)CCN(C)C2)C1 23430,C(=O)(CCCCCc1ccccc1)NCC(CNC(C(C)CN1CCCC1)=O)O 23431,NC(=O)CCC(=O)NCC1(C(=O)NCc2ccccc2F)CCCO1 23432,CC1(C)CCC(C(=O)NC2CC23CCOCC3)CN1C(=O)CC(=O)NC1CC1 23433,CC(C)CCCC(=O)N1CCCCC1CCN(C)C(c1cc(CC(C)C)c[nH]1)=O 23434,CC(C)(F)C(C)(F)C(=O)NC1CCC(CNC(=O)CCC2OCCO2)CC1 23435,c1(C(N2CC(CC)N(C(c3ccc(Cl)cc3)=O)CC2)=O)nn(C)cc1[N+](=O)[O-] 23436,Cc1cc(C#N)nc(NCC(C)(C2CC2)NC(=O)CCc2ccncc2F)n1 23437,C1(N(C(=O)C(C)NC(=O)C2CC2)CCC)CCN(C(=O)CCC(=O)OC)CC1 23438,CCC(CCOC)C(=O)NCCCOCCNC(C1CC(N2CCOCC2)C1)=O 23439,C1(NC(=O)CC2CC(F)C2)CN(C(c2ccc([N+](=O)[O-])o2)=O)C2CCCCC12 23440,c1(C(=O)NC(c2ccc(C)cc2)CC(=O)OCC)cc(F)cc2c1CCC2 23441,Cc1ccc(Cl)c(C(N2CC3(CCC3)CC2CNC(C2(CF)CC2)=O)=O)c1N 23442,c1(OC)cnc(Cl)cc1C(=O)NC1(CO)CN(C(C2CCCC(=O)N2C)=O)C1 23443,C(=O)(C(C)(C)c1sccc1Cl)N(CC(C)NC(=O)CCNC(=O)C=CCl)CC 23444,N1(C(CCCOCCOC)=O)CCOCC(NC(=O)C(n2cnc(C#N)n2)C)C1 23445,c1(NC(COc2ccc(CNC3C(CC)CCC3)cc2)=O)nc(O)sc1C 23446,C1(C(=O)NC2(C)CN(C(C3CCNC(=O)C3)=O)C2)CCN(C2CC2)C1=O 23447,c1(N2CC3N(C(=O)CC4CCC5CC5C4)C(CC3)CC2)nc2ccc(F)cc2s1 23448,C1(CC(=O)NCC(n2nnnc2C(C)(C)C)C)CCCN(C(c2cnns2)=O)C1 23449,CC(CC#N)C(=O)N1CC(n2cc(C(C)(O)CN(C)C)nn2)C1 23450,C(=O)(CC1=CCN(C)CC1)NCCC(C(N1C(C)CS(=O)(=O)CC1)=O)O 23451,N1(CCc2cn(CC3(C)CC3)nn2)CCCN(C(C2CCCC2C(F)F)=O)CC1 23452,C1(CC)CN(C(c2ccc(-c3nnc(C)o3)cc2)C(=O)NC2CCCC2)CCO1 23453,c1(CN(C(C)CN(C(=O)CC2CCCO2)C)C(=O)CC2CC(OC)C2)ccccc1 23454,C#CC1CN(C(=O)CC2CCCCN2C(=O)CC2CCC(=O)C2)CCN1C 23455,Cc1nc2cncc(C(=O)N(C3CCN(C(=O)C(C)(F)C(C)(C)F)C3)C)c2[nH]1 23456,C=CC(C)(C)C(=O)Nc1cccc(CNC(=O)C(c2ccnn2C)C)c1 23457,c1(OC)c(C)cc(C(=O)NC2CCCC(N(C(=O)CSC3CC3)C)C2)cc1C 23458,N1(C(C(C(=O)OC)C)=O)C2CCCC1CC(NC(C1CCC(=O)N1)=O)C2 23459,c1(CNC(CCC2CC(NC(C(C)SC)=O)C2)=O)cc(C)ccc1C 23460,N1(C(c2cnn(CCC)c2C)=O)C2CC1CN(C(c1cccnn1)=O)C2 23461,c1(C(N(CCNC(C2C(COC)C2)=O)C)=O)cccc(Cl)c1O 23462,c1(C(=O)NCC2CCCN(C(c3ccon3)=O)CC2)c[nH]c2ccc(Br)cc12 23463,c1(COC)ccccc1CC(=O)NC(C)CNC(=O)Cc1cc(C)nn1C 23464,c1(C(=O)OC)cccn(O)c1=O.CC(C)COC(C)(C)C1(CO)CC1 23465,c1(C(N2CC(SC)C(NC(=O)CCC(N)=O)C2)=O)cc(S(N)(=O)=O)cnc1C 23466,N1(C(CCC(CC)C)=O)C2CCC1CN(C(=O)CSc1nnc(S)s1)CC2 23467,C(=O)(C(O)C(C)NC(=O)OC(C)(C)C)NC(C1(c2cccc(Cl)c2)CC1)C 23468,C(=O)(CC1OCCc2ccsc21)N(CCCNC(C1CC2C(C1)C2(C)C)=O)C 23469,Cc1csc(C2CCCN2C(=O)CCCOCCN)n1 23470,c1(C(=O)NC(c2c(C)nc[nH]2)c2nnnn2C2(C)CC2)cccc(C(F)(F)F)c1C 23471,N1(C(CSCCNC(Cc2n(C)nnc2)=O)=O)CC2CC2C2CC12 23472,n1(CC(=O)NCC2(CN(C(=O)CCCN3CCCCC3)CC)CC2)ncn(C)c1=O 23473,C(=O)(CCC(CF)CF)NCCn1ccc(C(N2CCC(N(C)CC)C2)=O)c1 23474,N1(C(c2occc2C2CC2)=O)CC2C3CCC(C2C1)N(C(=O)CCF)C3.C1CC1 23475,N1(C(c2cnsn2)=O)CCC2(CCN(C(C3CCCC3CF)=O)CC2)C1 23476,c1(OCC(N2CC(C(=O)Nc3ccccc3)CC(F)(F)C2)=O)ccc(F)cc1Cl 23477,Cc1cc(Cl)cc(C(N2CCCOC(CNC(C34CC3CCC4(F)F)=O)C2)=O)c1C 23478,c1(C(N(C2CC(NC(C34CCC3C4)=O)C2)C)=O)ccc(CO)s1 23479,C1(C(N2CCC(NC(Cc3c(C)ccc(C)c3)=O)C2)=O)(CF)CCC(F)(F)CC1 23480,N1(C(C(C)(C)SC)=O)CC2CS(=O)(=O)CC2(NC(c2ccc3cccnn23)=O)C1 23481,N1(C(c2[nH]cc(C)c2)=O)CCOCC(NC(=O)C(C)(C)CF)C1 23482,CCS(=O)(=O)CC(=O)N1CCN(C(=O)CC2C=CS(=O)(=O)C2)C(CO)C1 23483,c1(CC)ccc(C(=O)NCC2COCC2NC(c2c(C)cncc2C)=O)cc1Cl 23484,C(=O)(CC(F)(F)Br)N1CC(NC(CN(C2CCOC2)C)=O)C1 23485,C1(CC)CN(C(=O)CCC(F)F)CCC1NC(c1nc(-c2cncn2C)no1)=O 23486,C1(NC(c2c(C)nn(C(C)(C)C)c2)=O)CC2CCC1N(c1ncncc1C#N)C2 23487,C1(O)(C(=O)NCC(C)CNC(=O)C(n2ccc(C(F)(F)F)n2)C)CCCCCC1 23488,C1(CNC(C(C2(O)CCOCC2)C)=O)CN(C(c2cc(Br)c[nH]2)=O)C(C)(C)C1 23489,c1(CC(N2C(CNC(CCCOCC)=O)C(C)CC2)=O)ccc(O)cc1Cl 23490,CCCC(C(C)(C)C)NC(=O)CC(C)(C)N(C(=O)CCC1CC(OC)C1)C 23491,c1(CC)ccccc1OCC(N1CCCC1CNC(=O)C(C)(C)c1cnco1)=O 23492,CCCC(C(F)(F)F)NC(C1CCCC(NC(C2(Cl)CC2)=O)CC1)=O 23493,C1(OCCNC(CC2CC(CC)C2)=O)CCN(C(=O)CC2CCOC2C)CC1 23494,c1(C(N(c2ccc(-c3ccc(C)o3)cc2)C)=O)ccc(OC2COC2)cc1Cl 23495,N1(C(C(C(C)C)O)=O)CC2=C(C1)CN(C(=O)C(C)C1CCC1)C2 23496,C1(CNC(CCCC#C)=O)CC(NC(c2nnn(C)c2N)=O)C12CCC2 23497,c1(C(=O)NC2C(C=C)CN(C(C3COC(=O)O3)=O)C2)n[nH]c2cccc(OC)c12 23498,Cc1cc(C(=O)N(CCC(C(C)C)NC(=O)CC2CCCO2)C)c(C)nc1C 23499,O=C(CC1CCc2ccccc21)NC1CC(F)CN(C(C2(n3cnnn3)CC2)=O)C1 23500,CC1CCN(C(=O)C(F)CC2CC2)CCN1C(=O)CC1NC(=O)NC1=O 23501,c1(C(N2C(CNC(COCCOCC#C)=O)CC2)=O)cc(F)cc(F)c1N 23502,c1(NC(c2ccc(CC)s2)=O)cccc(NC(=O)CCc2cncn2C)c1 23503,Cc1cccc(NC(=O)C(c2c(C)noc2C)(C)C)c1O 23504,c1(C(N2CC(CC)C(Nc3nc(C)nc(=N)[nH]3)CC2)=O)cn2cc(C)ccc2n1 23505,CC1CN(C(=O)Cc2cccs2)CC(C)C1NC(c1cccc(N)c1F)=O 23506,C=C1COCCN(C(=O)CC(CC)N(C(=O)Cn2cnnn2)C)C1 23507,C(=O)(C#CC1CCOC1)N1CCCC(N(C(=O)C(Cl)=CCl)CC)CC1 23508,CCCC(C(=O)NC(CC)C(c1ccc(OCC)cc1)=O)N(C)C 23509,N1(C(C2(N(C)C)CCC2)=O)CCCC(CNC(=O)CCc2cnco2)C1 23510,c1(N2CCC(N(C(=O)CCc3nc(C4CCCC4)no3)C)C2)ncc(Cl)cn1 23511,C1(C(=O)NCCCN(C(=O)C(c2cccc(C)c2)O)CC)CCCC(C)(C)C1 23512,c1(NC(CCNC(c2c(C)n(CCO)nc2)=O)C)snc(Cl)c1C#N 23513,O=S(=O)(c1ccc(NCC2=CCCC2)cc1Br)NCc1cscc1Br 23514,N12CCC3(COC(C3)CNC1=O)C2.c1(OC)cc(C(=O)OC(C)(C)C)cc(F)c1 23515,c1(CNC(C2(N(C(C3CC(C)OCC3)=O)C3CC3)CCC2)=O)cc(F)ccc1O 23516,c1(NC(COC2CC(NC(C(C(CC)C)C)=O)C2)=O)cc2cccnc2[nH]1 23517,CCCC(C)(C)C(=O)NCCC1(C)CCN(C(c2cn(CCO)nn2)=O)C1 23518,CC(O)CCCCCC(=O)NC12CC1CN(C(c1cc(N)cc(F)c1)=O)C2 23519,C12CCCC(C1)NC(=O)CN2C(C1(N(C)C)CC1)=O.c1(CSC)ccccc1 23520,Cc1oc(C(C)NC(=O)OC(C)(C)C)nc1C(=O)NCC(C)(C)n1cccn1 23521,C(C)(C(C(C)C)NC(c1ccc(SC)o1)=O)NC(c1ccn(CCCC)n1)=O 23522,c1(NCC(CC)OC)nc(N2CC3CCC(CC3)S2(=O)=O)nc2ncn(C)c12 23523,S(=O)(=O)(c1cnc(NCc2conc2C2CC2)cc1C)N(CCF)CC 23524,c1(C(=O)NC(CN(C(=O)CN(S(C)(=O)=O)C)CC)C)cn[nH]c1 23525,O=C(NNC(=O)c1nccs1)N1CCC(c2cccc(Cl)c2)C1 23526,N1(C(C2N(CC(C)C)CC2)=O)CC(C2(NC(c3cccc(C(F)F)c3)=O)CC2)C1 23527,c1(C(=O)Nc2ccc(C3(NC(COC)=O)CCC3)cn2)ccc2occc2c1 23528,c1(OC)cc(C(=O)NC(C)(C)CNC(=O)C(C(C)O)N(C)C)cnc1O.C1CO1 23529,N1(C(=O)NC(C)CN2CCCCC2)CCC(c2nc(-c3ccccc3)no2)CC1 23530,N1(C(CC2CCCC(C)C2)=O)CC2CC(NC(=O)Cc3ccc(F)cc3F)C2C1 23531,C1(CN)CCN(S(=O)(=O)NC(C2CC(=O)N(C3CCOCC3)C2)=O)C1 23532,CC(C)(O)C(F)(F)C(=O)NCC(C)(C1CC1)NC(c1ccc(S(N)(=O)=O)[nH]1)=O 23533,CC(C)S(=O)(=O)CC(=O)NCC1(NC(c2cccc3cnnn23)=O)CCOCC1 23534,c1(OC)cc(NC(C2CC2C(=O)Nc2cncc(C)n2)=O)ccc1CN(C)C 23535,N1(C(c2cnc(C)o2)=O)CC2CCCC2C1C(=O)NCC(O)CF 23536,C(CCSC)(C(=O)NCCC1(NC(=O)CC2CSCCS2)CC1)OC 23537,c1(C(=O)NCC2C(NC(C(OC)OC)=O)CCCC2)ccc2c(n1)CCC2 23538,c1(C(N2CCN(C(C3CCCCS3(=O)=O)=O)C(CF)C2)=O)ccn2nccc2n1 23539,CC1(C)CN(C(c2cnns2)=O)CC1NC(=O)COCC1CCCC1 23540,C1(C(=O)NCC#CCOC)(CNC(C2CCC(C)(C)C2)=O)CC12CCC2 23541,C(=O)(C1=NOC(CNC(c2cccc(CO)c2)=O)C1)NC(C(=O)N(C)CC)C 23542,N1(C(CC2(CSC)CC2)=O)CCCC(C)(C)C1CNC(c1ccc(C)c(F)c1)=O 23543,N1(C(CCC(=C)C)=O)CC2CCC(C1)N2C(=O)CC(C)(C)CN(C)C 23544,c1(C(N2C(C)CC(CNC(=O)CCN3CCC3)C2)=O)cc2n(n1)CCC2 23545,C(=O)(C1=CCC(F)(F)CC1)N(CCCNC(C1(COC)CCCOC1)=O)C(C)C 23546,c1(C(N2CC(CC(C)NC(=O)C(C)(F)F)C2)=O)ccc2nc(CO)[nH]c2c1 23547,C1(C(N2CCC(F)(CNC(c3ncn(C)n3)=O)CC2)=O)CC2CCCCN2C1 23548,C(=O)(C(CCC(N)=O)n1cc(CCc2nn[nH]n2)nn1)NC(C12CC(CO1)C2)C 23549,Cc1cc(Cl)nc(Cl)c1NC(=O)CC1CCCN1C(c1cc(O)cc(Br)c1)=O 23550,c1(C(N(C)CCC2CCO2)=O)ccc(-n2cccn2)cc1 23551,C1(C(NOCC(C(C)C)O)=O)CCCCCCN1C(C1C2CCC(F)(F)C12)=O 23552,C(=O)(C(C(=O)N1CCC(C(C)(C)NC(C2CCCC2C(C)C)=O)CC1)OC)OC 23553,N1(C(CN(C(C)C)C)=O)CC2ON=C(CNC(=O)COCC3CC3)C2C1 23554,C1(NC(C(n2cc(C)nc2)(C)C)=O)CN(C(c2ccncc2)=O)CCC1CO 23555,Cc1nn(C)c(C)c1CC(N1CCCC(CC(=O)NC2CCC(=O)N(C)C2)C1)=O 23556,C(=O)(C(CC(C)(C)C)NC(=O)CN1CC(=O)NC1=O)NCc1c(C)non1 23557,CCC(C(=O)N1CC(F)(F)CC1CNC(=O)C=Cc1cnccn1)C(C)(C)CC 23558,N(C1CC(C)(C)Oc2ccc(F)cc21)C1CC(S(=O)(=O)N)C1.CCC 23559,n1(CCC)nnnc1C(C(C)(C)c1ccccn1)NCC1CC1C1CC1 23560,CCC(C)(C)C(=O)C(=O)N1CCCC1CNC(=O)C(F)(F)C1CC1 23561,N1(C(CC(OCC)OCC)=O)CC(NC(c2ccc(Br)nc2Br)=O)C(C#N)C1 23562,S(=O)(=O)(c1c[nH]c(=NCCNC(C)=O)cc1C)N1CC(C)=C(C)C(C)C1 23563,CC(C)S(=O)c1ccc(C(=O)N(C)CCNC(=O)C(F)CC2CCCC2)cc1 23564,C1(C(N2CCC(NC(CC=CC)=O)C23CC3)=O)CC(c2ccccc2F)=NO1 23565,N1(C(c2n[nH]cc2-c2ccccc2)=O)CCN2C(=O)OCC2C1 23566,Cc1cnccc1CC(C)NC(=O)C(C)(C)n1cc(COC(=N)O)nn1 23567,C1(C(=O)NC(CC(C)NC(c2cn(C(C)C)nn2)=O)C)CCC(C(N)=O)CC1 23568,c1(C(C)C)ccc(N)c(C(N2CC(C(N)=O)(CNC(=O)CC(C)C3CC3)C2)=O)c1 23569,N1(C(CC=CC=C)=O)CCN(C)CC1C(=O)NCC(C)C(F)F 23570,C1(C)(C(N(C(CNC(=O)C(O)CC2CC2)Cc2ccccc2)C)=O)CCCN1C 23571,N1(C(C=C(CCN(C)C)Cl)=O)CCC(NC(C2CCCN2C(N)=O)=O)C1(C)C 23572,C(=O)(CC(C)(C)CC(=O)N1CCN(C(C2CCc3nnnn3CC2)=O)CC1)OC 23573,c1(C(=O)NCC(CNC(C2CCC(CC)O2)=O)(C)O)c(CC)ncnc1CC 23574,C1(NC(=O)CCC2CCOC2)CCC(NC(=O)CCCn2ccnc2)C1 23575,C1(NC(C2CCc3nncn3CC2)=O)C2CC3CN(C(=O)CC(F)F)C1C3C2 23576,c1(C(=O)NC2C(OC(C)C)C2)cnn(CC(C)O)c1 23577,c1(NC(C2CC23CN(Cc2scnc2Cl)C3)=O)cc2ccccn2n1 23578,Cc1ccc(C(c2nnnn2-c2ccccc2C)NC(C)(C)C)c(Br)c1 23579,N1(C(C2CCN(C(=O)OC)CC2)=O)CCC(C)(C)C1CNC(=O)C(C)N1CCC1 23580,CCCC(CC)CC(=O)NCC(O)CN(C)C(c1ccoc1C1CC1)=O 23581,CC(c1cccs1)=CC(N1CCC(C(F)CNC(C23CC(C)C2C3)=O)CC1)=O 23582,N1(C(C)CCc2ccco2)CCC(CC(=O)NC(c2cccs2)C)C1 23583,N1(S(CC(=O)OC)(=O)=O)CCCC2(CCN(C(c3ncc(OC)cc3F)=O)C2)C1 23584,N1(S(CCCC)(=O)=O)CCc2[nH]nc(C(N3CCOCC3CO)=O)c2C1 23585,C#CCCC(C(=O)Nc1cc(C(N)=O)oc1C)NC(=O)CN(C)CCC 23586,CCC(C)(COC)C(=O)NC1CCN(C)C1=O.c12ncoc1CCNC2=O 23587,N1(C(C(C)CC(F)F)=O)CC(C)(C)OCC1CNC(=O)CC1CC2CCC1O2 23588,Cc1cccc(C(=O)NCC(CNC(=O)CN2CCOC2=O)CO)c1Br 23589,N1(C(c2c(CNC(C=Cc3n(C)cnc3)=O)ccs2)=O)CCC(N=[N+]=[N-])C(O)C1 23590,C(CN=c1ccc2c([nH]1)CCC2=O)C1CC(NC(c2cn(CCOC)nc2)=O)C1 23591,N1(C(CC(CC)C(C)C)=O)CCN(C(c2ccc(C)cc2N)=O)C2CCCC12 23592,c1(C(=O)NC(C2CCN(C(c3cnco3)=O)C2)C)ccn2nccc2n1 23593,S(=O)(=O)(c1cc(C(=O)O)cc(C#N)c1)N1C2CC(SC)C2CC1 23594,C123CC(CN1C(=O)C(C1CCCC1)NC2=O)C3.c1(CN(C)C)coc(CO)c1 23595,CCCC(C)(C)CN=c1[nH]c2c(c(=NCC3CCCCCN3CC)[nH]1)S(=O)CC2 23596,N1(C(=O)OC(C)(C)C)CCN(C(C2CCSC2)=O)C(C2CCC2)C1 23597,C1(C#CC(=O)N(C)CC2CCCN2C(c2cnc(O)s2)=O)(CC)COC1 23598,c1(C(C)C)cccc(C(N2CCC(F)(C(=O)NC(c3ccccc3)C#N)C2)=O)c1 23599,O(C1CCOc2c(F)cc(F)cc21)C(=O)CCCCC1CCCC1 23600,Cc1cc(C(=O)NC2C3CN(C(c4occ5c4CCC5)=O)CC23)c(O)nn1 23601,c1(C(C)(C)C)ncccc1C(=O)NC(Cc1cncc(Br)c1)C(=O)O 23602,N1(C(C2C(OC)(OC)CC2)=O)CC(NC(=O)Cn2nc(C)cc2C)CC1(C)C 23603,C=CCC(CC(F)F)NC(=O)CC1CCCCC1NC(C1CCCSC1C)=O 23604,c1(C(=O)N(C2CCCCC2)CCNC(C2(F)CCCC2)=O)cc(F)cc(F)c1 23605,C#Cc1cccc(C(N2CCN(CCNC(=O)CC3CCC(O)C3)CC2)=O)c1C 23606,C1(c2ccccc2)(C(N(CCCCNC(C=CCC)=O)CC)=O)CC(O)C1 23607,C(=O)(CCCCCC(C)(C)C)NC1CC2(C(NC(c3c(C)cc(N)cc3)=O)C2)C1 23608,C12(CNC(C=CSC)=O)CCCC1N(C(c1cc(C)c(C)c(C)c1)=O)CCC2 23609,CC(C)(C)CC(C(F)(F)F)NC(=O)NCCn1cccn1 23610,Cc1ccc(Cl)c(O)c1C(N1CC(NC(c2ccc(F)s2)=O)CC(C)C1)=O 23611,N1(C(CCS(C)(=O)=O)=O)CCC2(CC1)CN(Cc1ccc3scnc3c1)C2 23612,C1(CC#C)(NC(=O)CCC2(NC(=O)C(C)CN(C)C)CCC2)CCCCC1 23613,c1(C(N2C(C(C)(C)NC(C(F)=CCC)=O)CCC2)=O)cc2cc(Br)cn2cn1 23614,C(=O)(C(C)C(CC)CC)NC(C1CN(c2nc(C(C)C)nc(C)c2F)C1)CC 23615,Cc1cc(C(=O)N(C(C)CNC(=O)CC2CCCOCC2)C)cnc1O 23616,C1(NC(C(N2CCOCC2)C)=O)CC2(CCCN(C(C3C(C)C3C)=O)C2)C1 23617,C12(CNC(COCCCC)=O)CCC(CC1NC(c1ncccc1CSC)=O)C2 23618,N1(C(CC2CC(C)(C)C2)=O)CC2CC(C1)CN(C(C1CC1C(F)(F)F)=O)C2 23619,C1(NC(C2C(C(C)(C)C)C2)=O)COC2CN(C(=O)Cc3cscn3)CC12 23620,C12(CNC(CCC3N(C(C(C=CC)O)=O)CCC3)=O)CC(C)(CCO1)C2 23621,Cc1cccc(Cl)c1CN1CC(O)(CNC(=O)CC2CCOC(C(C)C)C2)C1 23622,N1(C(C)=O)CCC(C)(C(=O)NCC2CCC(NC(=O)C#CC3CC3)C2)CC1 23623,CCCCC(C)C(=O)N(CC(CC)NC(=O)C=CC(F)(F)F)C 23624,N1(C(C2C(C)C2)=O)CCCCC(NC(C2CC3CCC2CC3)=O)C1 23625,C#Cc1ccc(CC(=O)NC(C2CN(c3cc(C(F)F)ncn3)C2)C)cc1 23626,C1(NC(CNC(CC)=O)=O)CC2CN(C(c3cc(C)ccc3C)=O)CC12 23627,c1(OC)cccc(C(N2CCC(CCNC(=O)CSC(F)(F)F)C2)=O)c1 23628,Cc1cc(CN2CCN(C(c3nnnn3C)=O)CC2)c(C)cc1O 23629,CN(C)NC(=O)CCC(=O)N1CCC(NC(C2CC(C(F)F)C2)=O)C1C(C)(C)C 23630,c1(C(N2CCC(O)(CNC(c3n(C)ccn3)=O)C2)=O)c(O)ccc2ccccc12 23631,C(=O)(C1CCCc2sc(=N)[nH]c21)N1CC(NC(C2C(C)C2C)=O)CC2(C1)CCC2 23632,c1(C(N2CC(C(=O)N=c3cco[nH]3)CC(F)(F)C2)=O)c(O)ccc(Br)c1O 23633,CC(C(=O)NC1(CNc2nc3ccc(F)cc3o2)CCOCC1)C(C)S(C)(=O)=O 23634,c12cccc(c1)NC(=O)CC2.C(=O)(C(CC1CCC1)OCC(F)(F)F)OC 23635,c1(C(=O)NCC2C(C)CCN2C(C23CCC(F)(CC2)C3)=O)noc2ncccc12 23636,Cc1cc(CNC(c2coc(CNC(=O)CC3CCN(C)C3)n2)=O)sn1 23637,Cc1c(C(C)NC(=O)C(=O)N(C)C)oc2ccccc12.N12CCOCC(C1)C2=O 23638,CC1CN(C(c2ccc(O)c(F)c2)=O)CCN(C(=O)C=Cc2ccc(Cl)cc2)C1 23639,CC(C(F)(F)C(F)(F)F)=CC(=O)N(CCCNC(c1cc(C)ccc1Cl)=O)C 23640,N1(C(CC=CCC)=O)CCCC(O)(CNC(=O)C=Cc2nccn2CC)CC1 23641,c1(C(N)=O)cc(Cl)cc(Cl)c1NC(C1CNCCN1Cc1cc(Br)cnc1Br)=O 23642,Cc1oc(CO)cc1C(N1CCN(C(C2CNC(=O)C2)=O)CC1)=O 23643,N1(C(Cc2cnc(C)[nH]2)=O)CC2CCC1C1CN(C(C3CCC3)=O)CC21 23644,C1(CCNC(CN(C)C2CC2)=O)CCN(C(C2CC3C(C2)C3(F)F)=O)CC1(F)F 23645,C(C(C#N)Cc1cccs1)NC(C1(CC)CC1)C 23646,C1(C(N2CCC(C(C)NC(=O)CCc3cncn3C)CC2)=O)CCC2(CCC2)C1 23647,C12(CNC(CCOCCCOC)=O)CCN(C(=O)CC(C)(C)C)CC1C2 23648,c1(OC)ncnc(C)c1C(=O)NCC1CCN1C(C1CC(F)(F)C1)=O 23649,c1(C(=O)NC2CC(CNC(c3c(CC)occ3C)=O)C2)ccc(C)c(C)c1O 23650,c1(C(=O)Nc2cnn(C3CC3)c2)cc(C2CC2)no1.O=CCCNCC1CC1 23651,C1(C(N(CCCCCNC(=O)CCN2CCCCC2=O)C)=O)CCC2(CCOC2)O1 23652,c12cc(cc(Cl)n1)C(=O)N2C1CCNC1=O.C1(C(=O)NC)Cc2ccccc2C1 23653,C1(C(=O)NCC2CCN(CCC)C2)CC(N=[N+]=[N-])CN1C(c1scnc1Cl)=O 23654,Cc1oc(C)c(C(N2CC(N(C(=O)CC3CC4COCC34)C)C2)=O)c1C 23655,c1(C(C)C)nnc(C(=O)NC2CC(n3ccnn3)C2)o1 23656,N1(C(c2ccc(OC)c(F)c2F)=O)CCCC2(CCCN2C(C2C=CCC2)=O)C1 23657,N1(C(c2cc(C)nc(C)c2)=O)CC(C)CN(C(c2nc(Cl)sc2Cl)=O)C(C)C1 23658,N1(C(c2cnc(OC)s2)=O)CC2CCC1C(CNC(=O)CCCC(N)=O)C2 23659,Cc1cc(Br)ccc1C(=O)NC1CCC(NC(=O)C(C)(F)F)C1 23660,c1(C(=O)NCCN(C(=O)CC(O)c2ccccc2)CCOC)nocc1C 23661,C1(CC(=O)NCCC2CCN(C(C3(C)CCCC3)=O)C2)CCCC1(F)F 23662,C1(NC(c2noc(CC)c2C)=O)CCC12CCN(C(=O)Cc1cc(C)no1)CC2 23663,N1(C2SCCN(C(C3CCCCCC3)=O)C2)CCN2CCCCC1C2 23664,c1(C(N(C)CC2CN(C(c3cc(I)cnc3Cl)=O)C2)=O)ccc2c(c1)COC2=O 23665,N1(C(C)=O)CCCC(C)(C(=O)N(C2(c3ccc(Br)cc3)CC2)C)C1 23666,c1(N2CC3CC(NC(c4cccc(C(C)C)n4)=O)C3C2)ncnc2c1CCO2 23667,N1(C(C=CC=CC)=O)CCC(NC(c2cc(C(N)=O)cs2)=O)C(O)C1 23668,N1(C(=O)OCC(CC)OC(C)(C)C)CCC(O)(NC(=O)OC(C)(C)C)C1 23669,N1(C(c2c(Br)cc(C)s2)C(=O)NC(C)(C)C)CCCc2ncccc2C1 23670,C(C(=O)NOCCN(C)C)N(C(=O)CC1(C)OCCO1)C(C)C 23671,c1(OC)cc(Br)ccc1C(c1nnnn1C)NC1(C2CCCCO2)CC1 23672,CC(C)CCC(=O)NC(C)CCC(=O)NCCCc1ncn(C)n1 23673,S(=O)(=O)(c1c[nH]c(C(=O)NC2CCN(C(=O)C(C)(C)C#N)C2)c1)NCC 23674,N1(C(C(C)c2ccsc2)=O)CCCC(O)(CCNC(=O)C(C)(Cl)Cl)C1 23675,C(=O)(C(O)CC(F)F)N1C(C(C)(C)NC(c2cc(C)n(C)n2)=O)CCC1 23676,C(=O)(C1=CCC(NC(c2cnn(C)c2Cl)=O)C1)N(C)CC1CC(F)(F)C1 23677,CC(C)(C)C(CN=c1ccn2c(Br)cnc2[nH]1)NC(c1ccc(F)o1)=O 23678,c1(C(=O)NCCCN(C(CCCOCC)=O)CC)ccc(N)c(N)n1 23679,C12(CNC(C(C)C3CCC3)=O)CC1CN(C(c1nccn1C)=O)C2 23680,C1(NC(N(C2CCC(C)CC2)CCCC)=O)CCNC(C2CC2)C1 23681,N1(C(Cc2ccc(C)nc2)=O)CC(C)(C)C(NC(c2cnc(O)s2)=O)C(C)(C)C1 23682,C(CC(C)(C)C)(C(=O)N(CCNC(=O)C1CC1)Cc1ccccc1)OC.C1CC1 23683,N1(C(=O)OC(C)(C)C)CC2COCC2(C(=O)NC(C)(C)CN2CCOCC2)C1 23684,c1(C(=O)NCC2C(CNC(C34CCC(OC)C3C4)=O)C2)[nH]c2ccccc2c1C 23685,C(CN=c1ccnc(NC(c2c[nH]c(=N)s2)C)[nH]1)N(C(C)C)CC 23686,c1(CC(=O)NCC2CCN(C(C3ON=C(C)C3)=O)C2)ccc(F)cc1[N+](=O)[O-] 23687,C1(OCC)CCCN(C(C2CC(C)=NO2)=O)C1.c12nc(cs1)CNC2=O 23688,C(=O)(C(C)(C)CC(C)=O)NCC(=O)NCC(=O)N(CC(C(CC)C)(C)O)CC 23689,C1(C(N(CCC)CCNC(=O)Cc2ccsc2Br)=O)CC(C)N(C)C1 23690,CC1(C)CN(C(=O)CCc2nccs2)CC1CNC(c1cc(CO)[nH]n1)=O 23691,N1(C(C(C)OCCCC)=O)CC(C(N2CC(C(C)(C)O)C2)=O)CC(C)C1 23692,C(=O)(C#CC1CCCCO1)NCCN(C(C)C)C(c1ccc(OCCF)cc1)=O 23693,c1(C(N2C(C(C)NC(C3CC(C#N)C3)=O)CCCC2)=O)cc2cc(F)ccc2o1 23694,CCCCC(F)C(=O)N1CCCCC1C1(Cc2ccc(F)cn2)CC1 23695,NS(=O)(=O)c1ccnc(C(=O)NCC2CN(C(=O)CC3CC4(CC4)C3)CCO2)c1 23696,Cc1ccc(C(C)C)cc1OCC(=O)NCC(CC(C)C)NC(=O)C1=CCC1 23697,C1(C(N2C3CN(C(c4ncn(C)c4)=O)C(CC3)C2)=O)CCC(S(C)(=O)=O)CC1 23698,N1(C(COCCCC(C)C)=O)CCC2(C1)CN(C(C1CC1C#N)=O)C2 23699,CCC(O)CCN=c1[nH]c(N2CCN(C)C(C)(C)C2)nc2cccnc12 23700,c1(CCC)nc(C(N2CCC(CNC(c3cn[nH]c3)=O)C2)=O)co1 23701,c1(C(=O)NCC2C(NC(C(C)C#N)=O)C2)ccc(C2CC(F)(F)C2)cc1 23702,N1(C(Cn2nc(C)n(CC)c2=O)=O)CCC2C(C1)CN2C(=O)C=C1CCC1 23703,C(CC(C)C(=O)NCC1CCC1NC(c1c(C)nsc1Br)=O)OC 23704,C12(NC(C=CC(=O)OCC)=O)CC1CN(Cc1cccc(CO)n1)C2 23705,C1(CC(=O)NCc2cccc(O)c2)CCCCN1C(=O)CN1C(=O)CNC1=O 23706,C1(NC(C2C(=O)NCC2)=O)CC2CC(C1)N(C(=O)Cc1cnsc1)C2 23707,C12(C(N3CC4C(NC(c5cc(O)ccc5Cl)=O)C4C3)=O)CC3CC1C2C3O 23708,N1(C(C(COC)C)=O)CCC2(CCC(NC(C3CCC(F)C3)=O)CC2)CC1 23709,c1(C(N(CC(C)NC(=O)CC2CC3CCC2O3)C)=O)c(Cl)csc1Cl 23710,CC1CN(C(C2(c3ccccc3F)CC=CC2)=O)CC1NC(=O)CCF 23711,C(=O)(C(CCC)N(C)C)NCC(C)(C)NC(COCCOCC#C)=O 23712,N1(C(C(C(CC)C)O)=O)CC2(CC(NC(C3CCCCN3N=O)=O)CO2)C1 23713,N1(Cc2c(COC)noc2)CCC(CNC(c2nccnc2CN(C)C)=O)CC1 23714,c1(CC(=O)N(C(C)C(C)(C)O)C)ccc(NC(=O)OC(C)(C)C)nc1 23715,C1(NC(C(C)(C2CC2)NC(C)=O)=O)CN(C(=O)Cc2ccc(CO)cc2)CC1O 23716,c1(C(=O)NCCCN(C(C2C(C)=CCS2)=O)C(C)C)cn2cccnc2n1 23717,c1(C(=O)NCC(=C)CCNC(=O)C=CCOC)noc2ncccc12 23718,c1(CC(N2CC3(CCN(C(CC(CC)C)=O)C3)C2)=O)ccc(Cl)c2cccnc12 23719,c1(OC)ccccc1OCC(=O)NC(CNC(c1cn(C)nc1C)=O)C1CCC1 23720,CC(CC(=O)N1CCC(CNC(=O)C(c2cc(F)cc(F)c2)O)C1)C(C)(C)C 23721,c1(C(N2CCN(C(=O)C#CC3CCCCC3)CC2)=O)cnc2ncnc(O)c2c1 23722,Cc1ccc(SCC2CCCN2C(c2c[nH]c(C#N)c2)=O)cc1.C12(CC1)C(=O)N2 23723,C(C(F)(C(=O)N1CCCC(C)C1CO)C(C)C)NC(C(C)N(C(C)=O)C)=O 23724,CC1=C(C(=O)NC2CC3CC(NC(=O)C(O)CN(C)C)CC23)SCCO1 23725,N1(C(c2nn(CC)c(O)c2)=O)CCC2(CC1)CC2CNC(=O)CC(O)CC(C)C 23726,C1(C(=O)NCC2C3CN(C(C4(C)CCCCC4)=O)C2C3)CS(=O)(=O)CC(=O)N1 23727,O=C1CCN(C(C23CC(CO2)N(C(=O)C(C)(C)C2CCCO2)C3)=O)CCN1 23728,N1(C(c2c(C)nc(O)[nH]2)=O)CCC(NC(c2cc(C(F)(F)F)no2)=O)CC1C 23729,CC1CC(C(=O)NCc2ccc(C(=O)NCC3(O)CC3)cc2)CC(C)C1 23730,N1(C(CC2(OC)CCC2)=O)C2CCC(C2)C1CC(=O)NC1(CO)CCCCCC1 23731,C(CCCCC(=O)NC1CC2CC(NC(C3CCS3(=O)=O)=O)CC12)SC 23732,Cc1nn(CC(=O)NCCCC(=O)NCCC2CCCO2)c(=O)o1 23733,C1(CNC(C2C(=O)NCC2)=O)CC2CC2N1C(c1ccn(CC(F)F)n1)=O 23734,n1(CC(=O)NCC(CNC(C2CC3CCC(C2)O3)=O)OC)nc(C)c(C)c1C 23735,C1(NC(C2(C)CC(NC(c3c(C)noc3)=O)C2)=O)CCOC2(CCC2)C1 23736,C1(O)(CN(C(=O)C(F)=CC2CC2)C)CCN(C(c2ccc(C(F)(F)F)[nH]2)=O)C1 23737,c1(C(=O)NCC2CCC(NC(C3C(C)(C)CC3)=O)C2)cc2c(F)c(F)ccc2[nH]1 23738,c1(C(=O)NCC(CN(C)CC2CCC(=O)N2)O)ccc(C(F)(F)F)cc1[N+](=O)[O-] 23739,c1(CC(=O)NC2CCC(CNC(=O)CC3CCCCC3)C2)cc(C(F)(F)F)co1 23740,C1(F)(CNC(c2ccc(C#C)cc2)=O)CC2CCC(C1)N2C(=O)C=CC(=O)NC 23741,Cc1cc(C)n(-c2ccc(-c3nc(-c4ccn(C)c4)n(CCC(C)C)n3)nc2)n1 23742,c1(C(=O)NC2(C)CCN(C(C3C(C)C3)=O)C2)cnc2c(c1)CNC(=O)N2 23743,C(=O)(C(O)CCNC(C1CCCC1F)=O)N(CCCC=C)C 23744,C1(CN(C(COCCSC)=O)C)COCCN1C(C1CC1c1nccn1C)=O 23745,N1(C(C(CSC)C)=O)CC(NC(=O)C(CO)NC(=O)C(F)(F)F)CC(F)C1 23746,c1(CC(CNC(Cn2c(C)nnn2)=O)NC(C2(SC)CC2)=O)ccc(C#N)cc1 23747,N1(C(C=CC=CCC)=O)CC(NC(c2cnc(C)nc2CC)=O)CCC1C 23748,CC(C)CC(F)C(=O)NCC1(C)CN(C(c2c(Br)cnn2C)=O)CC1C 23749,N1(C(C(C)C(C)(F)F)=O)CCCC2(CCCN2C(c2cnc3ccccn23)=O)C1 23750,C1(CCOC)(NC(=O)Cc2cccnc2Cl)CCN(C(C23CC4CC2C3C4)=O)C1 23751,N1(C(c2c(C)nc(C)s2)=O)CC2(CC(NC(c3n[nH]c(C)c3[N+](=O)[O-])=O)CO2)C1 23752,c1(OC)cc(Br)c(COC(c2cc3c(s2)CCNC3)=O)cc1OC 23753,N1(C(c2c(CC)nc(C)[nH]2)=O)CC(NC(C2(C)CCN(C)C2)=O)CC12CCC2 23754,c1(CC)cc(C(=O)NC2(C)CC(NC(=O)CC3CC(OC)C3)C2)ccc1C 23755,c1(CC(=O)NCC(CNC(CC(=O)OC)=O)OC)ccc2ncsc2c1 23756,C1(C(=O)NCCCNC(C=C(C)C2CC2)=O)CN(C)CC(C)O1 23757,C1(C(=O)NCCCNC(C2(CC=C)CCC2)=O)NC(=O)CC1C(F)(F)F 23758,N1(C(Cc2ccc(C)s2)=O)CCC(C2CC2)C1CNC(=O)COc1ccsn1 23759,c1(CNC(=O)NC(C)CC2=CCCCC2)ccc([N+](=O)[O-])c(N)c1 23760,CCC(CC)CCCC(=O)NC(CC1CCC1)C(N1CC(O)CC1CO)=O 23761,CC(C(=O)NC1C=CC(CC(=O)NCCCCNC(N)=O)C1)C(F)F 23762,C1(CC)CCCCN(C(=O)CCCN(C(=O)C(=O)C(C)(C)CC)C)CC1 23763,C(=O)(C(C)S(N)(=O)=O)N1CC(c2cn(CCOCC)nn2)(O)C1 23764,C(CCS(C)(=O)=O)N(C)C(=O)NC(c1cscc1Cl)(C)C 23765,CCCC(C(O)C(=O)NCC1(O)CCN(C)C1)NC(c1ccccc1CC)=O 23766,N1(C(c2ccc(OC)cc2F)=O)C2CCC1CC(NC(=O)C(C)CS(C)(=O)=O)C2 23767,C#CCCCC(=O)N1CCC(C(F)C(=O)Nc2cnn(CCC)c2)C1 23768,c1(C(=O)OC)cnc(SC)[nH]c1=NCCCC(C)(C)NC(=O)CC(C)SC 23769,N1(C(c2c(N)cnc(Cl)c2)=O)CCCC(NC(=O)Cn2cc(CO)nn2)C(F)C1 23770,C(C(C)(C(=O)NC(CNC(=O)CCc1cc(Cl)cs1)C(C)C)OC)OC 23771,c1(CC(N2C(CCNC(CC(CC)C3CC3)=O)CCCC2)=O)ccc(C)c(C)c1 23772,Cc1c(C(N2CCC3(CC3C(=O)Nc3cc(O)nc(O)n3)C2)=O)ccc(Br)c1F 23773,C1(CC=C)(C(=O)NC2CC(C(C)NC(c3cscc3Cl)=O)C2)CCOC1 23774,N1(C(C2(C)CCOC2)=O)CCC(C(F)F)(CNC(c2ncc(F)cn2)=O)C1 23775,C(=O)(C(C)Cn1ccc(C)n1)NCCCN(C(=O)C(C)c1ccon1)CC 23776,C1(C(=O)NCC2(O)CCN(C(c3c(C)cc(F)s3)=O)C2)SC2C=CC1CC2 23777,C#CC1(O)CCN(C(c2cnc(CNC(=O)C(C)(C)C(O)CC)nc2)=O)CC1 23778,c1(C(=O)NC(C(C)NC(C(C)NS(CC)(=O)=O)=O)CO)cccc(N)c1F 23779,c1(C(=O)NCC(C)N(C)C(C2COCCN2C)=O)cccc(C(F)F)n1 23780,N1(C(=O)NCCNC(C2(C(C(=O)OCC)C3(C)CC3)CC2)=O)C(=O)CCCC1=O 23781,Cc1cncc(C=CC(=O)NC2CC2NC(=O)C(c2cc(Cl)ccc2Cl)(F)F)c1 23782,Cn1cnc2nc(N3CC(C)(C)CC3CNC(=O)C(C)(C)C(F)F)nc(O)c12 23783,Cc1nc2cccc(C(N3CC=CC(NC(C4(Cl)CC4)=O)C3)=O)c2s1 23784,C(=O)(C=C1SCC(=O)N1C)NC(CC)CNC(c1cc(C(C)C)c(C)s1)=O 23785,N1(C(c2cnn(C)c2Cl)=O)CCCC(NC(=O)CC2CCCOCC2)CC1 23786,Cc1cc(C(=O)NCC(C)NC(=O)C(C)C2CCC2)ccc1C(C)C 23787,C(=O)(C(C)(CC1CCC1)OC)NCC1C(NC(CCNS(CC)(=O)=O)=O)CC1 23788,Cc1nnc2ccc(C(N3CCN(C(=O)COC4CCC4)CC3C(C)C)=O)cn12 23789,c1(C(N2CCC(C(C)NC(C=C=C(C)C)=O)C2)=O)cccc2c[nH]nc12 23790,C(=O)(CC(O)CC(C)C)N(CC(CNC(C(CSC)OC)=O)O)C 23791,C1(CC(=O)N(CCOCC)C)CN(C(=O)CC2(COC)CCOCC2)CCO1 23792,Cc1nn(CC(=O)NC2CC3C(NC(=O)C(c4cnccn4)C)C3C2)c(=O)o1 23793,c1(C(C(N2C(CN(C(C(F)=CCC)=O)C)CCC2)=O)O)ccccc1F 23794,N1(C(c2c(CC)noc2)=O)CC2COCC2(C(=O)NCC(O)C2CCC2)C1 23795,c1(C(C(=O)OCC(=O)N(CC)CC)C)c(F)cccc1F 23796,C1(C)(C(=O)NCCn2cc(CNC(C(C(C)C)F)=O)nn2)CCCCC1(F)F 23797,C1(C(=O)NCCCOC2CCN(C(c3cnc(C)s3)=O)CC2)CC(C(C)C)=NO1 23798,C(C(CCC)C(=O)N1CCC1(C)CC)NC(C(C=C)(C)C)=O 23799,c1(C(N2CCN(C(CC(C=C)C)=O)CC2C2CC2)=O)ccn2ncc(C)c2n1 23800,N1(C(c2n(CCC)ncc2)=O)CC2(C)CC1C2NC(c1ccc(=O)oc1)=O 23801,C(C)(C)(C(=O)N1CCC(CCNC(=O)Cc2[nH]cnc2C)C1)OCC 23802,c1(C(=O)NCC2CC(C)N(C(=O)CC3C=CCCC3)C2)ncc(Cl)cc1Cl 23803,c1(C(=O)NC2C(CN)CCC2)ccc(F)c2cccnc12 23804,c1(CC)ncsc1C(=O)NC1(CN(C(=O)CC(F)F)C)CC1 23805,CCCCC(Cc1ccccn1)NC(=O)NCc1ccc[nH]1 23806,C1(C(C)(C)C)CC(C)(CC(=O)NC(C(=O)NC2C=CC(CO)C2)C2CCCC2)C1 23807,N1(C(C(CC=C)(F)F)=O)CCC2CN(C(=O)CC3CCCN3CC)CC2CC1 23808,C1(NC(CCOC(C)C)=O)CC2CCC1CN2C(=O)CC1(C#N)CCOCC1 23809,Cc1c(C(N2CCC(C(F)(F)F)C2(C)C)=O)cc([N+](=O)[O-])cc1[N+](=O)[O-] 23810,CCC(C)C(O)C(=O)NCC1(NC(=O)C2=NOC(C3(O)COC3)C2)CCCC1 23811,c1(C(=O)NCc2cccc(CN(C(C(C)CO)=O)C)c2)onc2c1CCCC2 23812,N1(CC2CCC(C(=O)OCC(C)C)CC2)CCC(CN)C(F)(F)C1 23813,C=CC(C)CC(=O)NCC1(OCC)CN(C(c2ncn(C)n2)=O)C1 23814,c1(C(=O)NC(CNC(CN(C)CC)=O)C)ccc(C(=O)NC(C)(C)C)cc1 23815,c1(OCC)nc(Cl)cc(=NC(=O)C2CC(F)CN2Cc2cccc(I)c2F)[nH]1 23816,c1(C(N(CC)CC2CCCN2C(=O)C=CS(C)=O)=O)cnn2cccnc12 23817,c1(C(N2CC(C)(CNC(c3c(C)c[nH]n3)=O)OCC2)=O)cc2c(s1)CCCC2 23818,c1(NC(C2C3CN(C(c4c(C)cns4)=O)CC32)=O)ccc(O)c(C)c1 23819,S(=O)(=O)(c1cccnc1[N+](=O)[O-])N(C)CP(C)(C)=O 23820,c1(C(C)=O)ccc(CC(=O)N(CCCCN(C(=O)Cn2nccc2C)C)C)s1 23821,N1(C(CCOCC)=O)CC(CNC(=O)CN2CCSCC2)CC(C)(C)C1 23822,C1(O)(CCNC(=O)Cc2ccoc2)CCN(C(=O)Cc2cc(C3CC3)no2)C1 23823,C1(C(=O)NC23C(CN(C(COCC)=O)C2)CC3)Cc2cc(F)ccc2O1 23824,C1(C)(NC(C2CC(CNC(c3c(C)nsc3C)=O)C2)=O)CC2CCC1C2 23825,N1(C(C=CC(CC)=CC)=O)CC2CCC1C2NC(C1CN(C)C1)=O 23826,C1(N(C(c2c(C)nsc2)=O)C)CCC2CN(C(C3CC(=O)C3C)=O)CC12 23827,S(=O)(=O)(c1cnccc1N1CCS(=O)(=O)C(CO)C1)NC(c1ccc(Br)cc1)C 23828,C1(CNC(C(CC#C)(C)C)=O)CC(O)C(O)CC1C(=O)NCC(C)C(C)C 23829,c1(CN(CCCOc2ccc(C)cc2)C=O)c(Br)cc(F)c(F)c1F 23830,c1(NC(CC)CO)cc(Br)ccc1S(=O)(=O)NC1CCCN(C)C1 23831,CCCC(C)CC(=O)N1CCCC1(C)C(=O)N(CCCOCC)C 23832,C1(C2CCOCC2)(NC(c2scc(C)c2)c2nnnn2C2CCOCC2)CC1 23833,N1(C(c2c(C)ncn2C)=O)CCC(NC(C2CC2(C)C)=O)C(CO)CC1 23834,CCC(c1cccc(Cl)c1)=CC(=O)NCC(C)(C)NC(C1CCC(C2CC2)C1)=O 23835,C(=O)(C(O)CCCCCCCCC)NC1CN(C(CC(C=C)CC)=O)C1 23836,N1(C(C(C2CCCC2)OCC)=O)CCC(CNC(c2cnc(O)o2)=O)CC1C 23837,N1(C(C=CC=CC)=O)CCN(C(=O)Cn2c(C)c(C)sc2=O)C(c2ncc[nH]2)C1 23838,Cc1cc(C(=O)NCC(C)(CC(C)C)NC(=O)C(C)Cn2ccnc2)c(C)cn1 23839,CC(c1ccccc1C)=CC(=O)NC12CC(NC(c3ccsc3)=O)(C1)C2 23840,N1(C(=O)N(C23CC(C(F)F)(C2)C3)c2ccccn2)CC=CC12CCOCC2 23841,C(=O)(CS(=O)CCC(F)(F)F)N1CCC(NC(C(CC)=CCCC)=O)CC1C 23842,c1(C(=O)NCC(CC)NC(c2cn(CCF)nn2)=O)c(OC(F)F)cccc1F 23843,c1(C(N(C2CCC(NC(CCC=C)=O)C2)C)=O)sc2nc(C)nc(C)c2c1C 23844,Cc1ccc(-n2ccnc2)c(C(=O)NC2C=CCN(C(C3CC3C#N)=O)C2)c1 23845,c1(CC(N2CC(C3CCN(C(=O)C(=O)NC4CC4)CC3)C2)=O)cccc(O)c1 23846,Cc1cc(S(=O)(=O)N2CCC(OC(F)(F)CF)CC2)ccc1Br 23847,CC1=CC2CCCC(C1)N2C(=O)NCCCNC1CCC1 23848,CC#CCC(C(=O)N(c1ccc(O)cc1C)C)NC(=O)C(C)NC(N)=O 23849,C1(C(N2CC(C)C(C(=O)NCCC3=CCOCC3)C2)=O)CC2CCC(C1)N2C 23850,c1(C(N(CCN(C(C(CCCOC)C)=O)C)C)=O)cccc2c1C1CCC2CC1 23851,N1(C(C2(CCNC(C(CC)C)=O)CCCC2)=O)CC2C=CCC(C2)C1 23852,c1(NCC(c2ccc(C)cc2)O)cc(C(=O)O)ccc1C(N)=O 23853,C12(CNC(Cc3ccc(C)c(Cl)c3)=O)CCC(CC1)N(C(=O)C(O)CC(F)(F)F)C2 23854,c1(NCC(C2CCCCC2)NC(C2C(C)(Br)C2)=O)cnc2ccccc2n1 23855,S(=O)(=O)(c1c(C)ccc2ccccc12)NC(CC)C(c1ccc(F)cc1)=O 23856,c1(ONC(C(N(C)C)C2CC2)=O)ccc(Cl)c(C(N)=O)c1 23857,N1(CCCCCC)CC(NC(c2cc(C(=O)NC(C)(C)C)n[nH]2)=O)C(C)C1 23858,CCS(=O)(=O)CC(=O)N1CCC(NC(=O)CCCOC(=O)CCC)C1.C(C)(C)C 23859,c1(OC)ccccc1CC(=O)NCC1CCN1C(C1CCCN1c1nccs1)=O 23860,c1(N2CC(CC=C)(NC(=O)CNS(=O)(=O)C3CC3)C2)ncc2c(ncn2C)n1 23861,c1(CC(=O)NC2CCC(N(C(C=CCC)=O)C)C2)cnn(C)c1C(=O)OCC 23862,C1(C(=O)NC(c2ccn(C)n2)CO)(NC(Cc2c(C)ccs2)=O)CCN(C)C1 23863,C(C)(C(=O)N1CCCC(C)(CNC(=O)CCC2CCCCC2)C1)(C(C)C)OC 23864,N1(S(c2c(NC(CCC)CCCO)nccc2)(=O)=O)CCc2cc(C)cc(C)c2C1 23865,C1(CNC(c2n(CC)ncc2)=O)CC(OC)CN1C(c1cn(C2CC2)nn1)=O 23866,C(=O)(C1=CCCOC1)NC1CCCN(C(C(C)(C)Cc2ccccc2)=O)C1 23867,c1(C(=O)NCC2N(C(C(C(CC)C)O)=O)CC(F)C2)c2n(c(=O)n1C)CCCC2 23868,N1(C(CCCC(CC)C)=O)CCN(C(=O)CC(F)(F)C(F)(F)F)C2COCC12 23869,Cc1nccc(CNC(=O)CCC2CCCCN(C(C3(C)CCCC3)=O)C2)n1 23870,CCCCC(C(=O)NC)NC(C12CC1CCN2C(c1cc(C)ccc1O)=O)=O 23871,c1(CNC(c2cnc(O)c(Br)c2)c2n(CCC)nnn2)ncc(C(N)=O)cc1C 23872,n1(CC(C)(C)C)ccc(=NC(=O)c2ccc(C3CCNCC3)s2)[nH]1 23873,C1(C(=O)NC2(C)CN(C(C(C)c3ccco3)=O)C2)CN(C(N)=O)CCO1 23874,C(=O)(CCCCC(F)F)N(CCNC(c1nc(COC)sc1)=O)C(C)C 23875,C(=O)(C#CC(C)(C)C)N1C(C)(NC(N2CC(CCCCC)C2)=O)C=CC1 23876,CC(CN=C1NCC2(CCCC2)CN1)CC(F)(F)F.C1(COC)CC1 23877,N1(C(C(c2ccnn2C)NC(Cn2c(C)ccn2)=O)=O)CCC(C2CCC2)CC1 23878,C(=O)(CCC(F)(F)F)NC(C1(O)CCN(C(c2nn(C)cc2Cl)=O)C1)C 23879,C1(C)(NC(COc2ccc(C)cc2)=O)CCN(C(C2CC(C)OC2C)=O)CC1 23880,c1(OC)cc(NC2CCN(C(=O)C(C)C(C)O)C2)ccc1[N+](=O)[O-] 23881,N1(C(C(CCF)NC(CCCOCC)=O)=O)CC2CCC2(CO)C1 23882,N1(C(C(C2CC2)OC)=O)CC(C)(NC(=O)COC2CCCCC2)C1 23883,C(=O)(C(F)C(C)CNC(c1cncc(OC)n1)=O)NCc1n(CC)cnn1 23884,c1(C(=O)NC(CC(C)NC(=O)Cc2ccon2)C)ccc2cccnc2c1 23885,N1(C(CCC(=O)OC(C)(C)C)=O)CC2(C1)CN(C(c1cnn(CCF)c1)=O)C2 23886,N1(C(c2c(C)nn(C)c2C)=O)CC(NC(c2cnn(CCO)c2)=O)CC2(CC2)C1 23887,C1(CNC(c2c(COC)cco2)=O)C2CCCC1N(C(=O)Cc1csnc1C)C2 23888,CCCCCCCC(F)C(=O)NCCn1cc(CC(CO)C2CC2)nn1 23889,Cc1c(C(N2CCCC2C(C)NC(C2CCCN2C)=O)=O)cnn1CCO 23890,S(=O)(=O)(c1cccc(S(N)(=O)=O)c1)NC(c1ccc(C)c(S(N)(=O)=O)c1)=O 23891,N1(C(C(C)N(C(=O)C2=NOCC2)C)=O)CC(F)CC1C 23892,C1(NC(=O)C(C)(C)C)CN2CC1CNC2=O.c1(COC)ccccc1 23893,C(CNC(=O)Cc1c(Cl)cnn1C)(CCCC)NC(CSCC=C)=O 23894,C(c1ccc(F)cc1F)=CC(=O)NCC1(NC(C(CCSC)OC)=O)CCC1 23895,C(=O)(CCCCC(=O)OC(C)(C)C)NC1C(NC(C2CC(C)OCC2)=O)CCC1 23896,C(=O)(C1=CC2CCC(C1)C2)N(CC(CC)NC(C1CCC([N+](=O)[O-])CC1)=O)C 23897,C(C)(C)(CCN=c1nc(C#N)[nH]cc1Cl)NC(C(c1ccc(OC)cn1)(F)F)=O 23898,C1(CC)CN(C(c2nc(C3CCCCC3)cs2)=O)CCN1 23899,C1(C(=O)NC2CC(NC(Cn3c(C)ccc3C)=O)C2)CC(S(C)(=O)=O)C1 23900,Fc1ccccc1CN=C(NCc1ccco1)NC1CC12CCCC2 23901,c1(C(N(CC(CNC(COC(C)=O)=O)C)C)=O)c(Br)c(C)nn1C 23902,CC1SCCCC1C(=O)NC1CCN(C(=O)C=Cc2cnccn2)CC1 23903,N1(C(C(C)(C)O)=O)CCC(C2CCN(C(C3(C(C)(F)F)CC3)=O)CC2)C1 23904,N1(C(CCCOCC)=O)C2CCC1C(C(N1CCC(C(C)(C)C)CC1)=O)C2 23905,N1(C(CCOCCC)=O)CCN(C(=O)Cc2nocc2C(C)C)CCC1C 23906,C=CC(CC)CC(=O)NCCN(CC(C)O)C(c1cn(CCC(C)C)nn1)=O 23907,CCC(C)CCC(=O)N1CC(COC)(NC(=O)C(C)Cc2ccc(N)cc2)C1 23908,C(C)(C(=O)N(CC(=O)OC(C)CN1CCCC1)CC1CC1)OCC(C)C 23909,C#Cc1cc(C(c2nnnn2C)NCC2CCCCC2C)cc2c1OCO2 23910,Cc1ncccc1CCC(=O)NCCOCCCNC(=O)Cc1ccc(O)nc1 23911,C1(C(C(=O)NCCC(=O)OCC)N(CC(C)SC)C)CCCC(C(=O)OC)CC1 23912,C1(NC(CC(C)F)=O)CN(C(c2ccc3scnc3c2)=O)CC12CCOCC2 23913,c1(C(=O)NCC2(O)CCN(C(C3(SC)CC3)=O)C2)cnc2nc(C)ccc2c1O 23914,N1(C(C2C(C(=O)OC)CCCC2)=O)CCOC2(C1)CN(C(C1(O)CCC1)=O)C2 23915,c1(C(=O)NCC2CCCN2C(c2ccc(O)cc2)=O)cc(Br)cc2c1OCC2 23916,C1(NC(c2ccn(CC)n2)=O)CC(NC(=O)C=CC(F)(F)F)C12CCC2 23917,c1(C(C)=O)cc(Br)cc(C)c1NC(C1CN(C(=O)C(C)(C)Br)CC12CC2)=O 23918,Cc1ncnc(C(N2CCCC(N(C(=O)CCC3CCCCCC3)C)C2)=O)c1C 23919,Cc1noc(C)c1CC(=O)NCC(C1CC1)N(C)C(C1CC2C=CC1C2)=O 23920,N1(C(c2cc(C)no2)=O)CCC(C)(CNC(=O)CNC(c2ccncc2)=O)CC1 23921,C1(C(=O)OC)(C(=O)NCCOC2CCN(C(C3CC=CCO3)=O)C2)CC=CC1 23922,C(N=c1[nH]c2ccc(Cl)cc2c(=NCC(C(C)C)OCCO)[nH]1)SC 23923,CCC(C)(C)CC(=O)NCC1OCCC1C(=O)Nc1cc(OC)ccc1O 23924,n1(CC)cc(C(=O)NC(c2cccnc2)C(=O)NCC2CCCS2)c(C)n1 23925,C(=O)(CCCCC(N)=O)N1CCC(C(C)NC(C2(C)CCNC(=O)C2)=O)C1 23926,c1(NC(C2(CNC(=O)CCc3ccsc3)CC(=C)C2)=O)ccc(CC)nc1 23927,C(=O)(NNC(=O)N1CCCC1C(F)(F)F)c1n(C)ncc1 23928,c1(CCC)cccc(C(=O)NC(C)CCCNC(=O)CC2CC3(CC3)C2)c1 23929,C1(COC)(NC(=O)CNC(N)=O)CCN(C(c2ncncc2Br)=O)CC1 23930,c1(C(N2C(C)CCN(C(=O)CC(O)CN(C)C)CC2)=O)cccc2c1CCC2=O 23931,CC(C)C(C)(C)C(=O)NCc1cc(C(=O)NC(C2(CO)CC2)C)n[nH]1 23932,O=S(=O)(c1ccc(NCC2(CO)CCCCO2)cc1Br)NCc1cc(F)ccc1F 23933,C1(NC(C(CC=C)CC)=O)CCC2(CC1)CC(NC(c1ccoc1)=O)C2 23934,c1(SCC(=O)NCC2(OC)CCN(C(C(CC)SC)=O)C2)nc2ccccc2[nH]1 23935,c1(C(N2CCN(C(C(CCC)OC)=O)C(C)C2)=O)sc2ccccc2c1Cl 23936,CC1(C)CCCC(CC(=O)NCC(C)(O)CNC(C2CC(O)C2)=O)C1 23937,CC1CC(C(N2CCCN(C(C3CC(NS(C)(=O)=O)C3)=O)CC2)=O)CCC1C 23938,N1(C(=O)NC(c2c(C(=O)OC)scc2)C2CC2)CC(CN(C)C)C(F)C1 23939,c1(CC)nnc(COC(c2cc(-c3ccccc3)on2)=O)s1 23940,C1(NC(COCCOC)=O)CC(NC(c2sccc2C#N)=O)C12CCC2 23941,C1(N(C)C(c2cccnc2S)=O)CN(C(=O)C=CC2CCCCC2)CC1(C)C 23942,C(c1cccc(F)c1)=CC(=O)NC(CNC(=O)C(F)(F)CC1CC1)CO 23943,C1(C(=O)NC(C(=O)NCCCC)C)OCCOC1C 23944,CCS(=O)(=O)CC(=O)NC1(C)CC(NC(c2c(C(F)(F)F)coc2C(C)C)=O)C1 23945,c1(NS(C)=O)ccc(C2C(C(=O)NC(=O)CNCC(=O)OC(C)(C)C)C2)cc1 23946,Cc1c(C(=O)NCC2(C)CCCN2C(c2ccc(N)cc2F)=O)cccc1C#N 23947,N1(C(C2(CCC=C)CC2)=O)CCC(NC(=O)CC2CC(C)=NO2)C2(CCC2)C1 23948,N1(C(C(CCCCC)F)=O)CCn2nc(C)cc2C1 23949,C1(N)(C(C)(C)C)CCN(C(C2CC(=O)CCO2)=O)C1 23950,N1(C(c2c(COC)occ2)=O)CC2C(NC(=O)CCc3nc(C)c(C)o3)C2C1 23951,Cn1nnc2c1C(c1nc(-c3ccc(Cl)s3)nn1CC(F)F)CCC2 23952,Cn1cnc(C#N)c1C(=O)NC(c1cccc(Cl)c1)CNC(=O)CS(C)(=O)=O 23953,CCC(C)C(C(=O)NCCCC(C)(C)NC(C1C2CCC1(C(F)(F)F)C2)=O)OC 23954,c1(C(N2CCC(N(C(CCC3N(C)CCC3)=O)CCO)C2)=O)nccc2occc12 23955,C(CC1CC1)(C(=O)NOC1CCC1)NC(CC(CN(C)C)O)=O 23956,N1(C(C2C(C)N(C)CC2)=O)CCC2CN(C(=O)COC(F)F)C(C)C12 23957,c1(C(=O)NCC2N(C(CC#N)=O)CCOC2)cccc2c1OCC2 23958,C(C(=O)N1CC(NC(=O)Cc2c(F)cncc2Cl)CC(O)C1)(C(C)(C)C)SC 23959,c1(OC)cc(NCc2cc(O)nc(O)n2)nc(OCCOC)n1 23960,c1(-c2c(OCC(F)(F)F)ccnc2)ccc2c(c1)CN(Cc1cnc(O)c(Br)c1)C2 23961,C1(C(N2C(CC)(CO)CCC2)=O)CN(C(c2cccc(Br)c2)=O)CCC1O 23962,C12(CC(=O)N(C)CC3CCC(CNC(C(=O)NCC)=O)CC3)CCC(CC1)OC2 23963,CCC(CC)C(C(=O)N1CCC(F)(F)C(CNC(C2CC3(CSC3)C2)=O)C1)OC 23964,N1(C(CCC(=C)C)=O)CCS(=O)(=O)C(CCNC(c2coc(CC3CC3)n2)=O)C1 23965,c1(CNC(C2(C(F)(F)F)CC3C=CC2C3)=O)cc(O)ccc1O 23966,c1(C(=O)NCC2CN(C(COCCC)=O)C2)c[nH]nc1-c1cnn(C)c1 23967,c1(OC)ccc(C(=O)NC2CC(C)CN(C(c3c(C)cnn3C)=O)C2)c(F)c1Cl 23968,O1NC(=O)C(CCSC)NC(=O)CCC1.C1(C(=O)OC)CC1(C)C(F)F 23969,C1(C(C(=O)N(C2CN(C(C3(C(F)F)CC3)=O)C2)C)O)CCCCCC1 23970,c1(C(=O)NC2CCC(NC(C=CC3=CC(C)(C)C3)=O)C2)[nH]cc2c1CCC2 23971,C(=O)(C(F)C(=O)NCCCOCCCNC(=O)Cc1ccc(O)cc1)OCC.CC 23972,c1(CC(=O)NCc2cnn(CC)c2C)ccc(Br)cc1OCC(F)F 23973,C1(CN(C(CCC#C)=O)CC)CCCCN1C(c1ccc(C(F)F)nc1)=O 23974,C1(C(=O)NCC(c2cccc(Cl)c2)OC)CCCC(=O)N1 23975,CCC(C)CCCCC(=O)N(C1CCCN(C(c2cnc(S)n2C)=O)C1)C 23976,Cn1ncc2c(C(=O)NCC3CCN(C(C4(F)CCOC4)=O)C34CC4)ccnc12 23977,C(=O)(CCCCNC(c1ccn(C(F)F)n1)=O)NC(C=C)CO 23978,CCC(C)CCCCC(=O)NC(C1CN(C(=O)C(C)O)C1)C 23979,CS(C)(=O)=Nc1ccc(C(N2CCN(C(=O)C(C3CCCO3)C3CC3)CC2)=O)s1 23980,C1(C(=O)NOCC2CCCO2)(C(C)C)CCCN1C(=O)C(C1CCOCC1)F 23981,c1(C(=O)NC(CC(C)NC(C(CC)=CC)=O)C)c(C)c[nH]c1CC(N)=O 23982,c1(-c2n(-c3c(OC)nccc3)nc(CC3CC3)n2)cc2c(OC)cccc2[nH]1 23983,C#CC1CCCCN1N1CCN(Cc2ccc(-c3ccccc3)cc2)CC1 23984,Cc1cc(Cl)c(C(=O)N(CC(O)CNC(C2Cc3nccn3C2)=O)C)cn1 23985,c1(N(C2CSC2)C(=O)NCC2C(CC)C2)ccc(Br)s1 23986,C1(C(N2CC(C3(NC(C(c4ccnn4C)C)=O)CC3)C2)=O)CS(=O)(=O)CC(=O)N1 23987,N=c1cc(C(N2CCN(C(=O)C=CC3CCOC3)CC2CCO)=O)[nH]c(=N)[nH]1 23988,Cc1nc(-c2ccccc2)sc1C(=O)NCC1CC1CNC(=O)CNC=O 23989,C1(N(CCC(C)C)C)CN(C(=O)C=CC(c2ccc(F)cc2)=O)CCS1 23990,c1(C(=O)NCC2(F)CC(NC(C(C(C)C)F)=O)C2)sccc1S(C)(=O)=O 23991,c1(Nc2n(C(c3nnn(C)c3C(F)(F)F)C)nnn2)ncccc1OCC(F)F 23992,c1(OCCC)ccnc(C(N2CC(CNC(C3(OC)CCSC3)=O)C(C)C2)=O)c1 23993,CCCC(CCC)C(=O)NC12CCC(CN(C(=O)CCC(=O)NC)C1)C2 23994,C1(C(C(=O)N(C(COC)C)C)C)CCN(C(c2ccns2)=O)C1 23995,n1(CC(COC)OC)c(N(CCCS(C)(=O)=O)C2CC2)nnc1-c1coc(C)n1 23996,c1(CCC(N2CCN(C(c3ccc(F)o3)=O)C3CC23)=O)ccc(Cl)c(F)c1 23997,c1(C(=O)NC(CC)(CNC(C2(C)CNC(=O)C2)=O)CC)ccc2occc2c1 23998,c1(NC(C2N(C(C(C(CC)O)(F)F)=O)CCC=C2)=O)cnc2ccccc2c1 23999,N1(C(C(CCC)C)=O)CCN(C(c2cc(C(N)=O)c[nH]2)=O)C2CCC12 24000,C(=O)(C1=C(C)N(CC)C(=O)NC1c1sncc1Br)N1CCN(CCC)CC1 24001,c1(C(N2CCC(C(=O)NCCC(CCC)C)(OC)C2)=O)ncc2ccccn12 24002,N1(C(C(Cc2ncn(C)c2)O)=O)CCCC2(CCN(C(=O)CNS(N)(=O)=O)C2)C1 24003,CP(C)(=O)c1cncc(CNC(=O)NC(c2ncccc2F)c2ccccc2)c1 24004,C#CCC(CC(=O)NC1(CC=C)CCOC1)NC(c1cnc(OC)cn1)=O 24005,C=CC(C)(C)CC(=O)NC12COC(C1)C(NC(C1CCCC1(F)F)=O)C2 24006,c1(C(=O)NCC(CNC(C2=C(C)OCCS2)=O)CO)ccc2c(c1)OC(C)(C)C2 24007,C1(C(=O)OCC2CC(=O)N(C(c3ccsc3)=O)C2)CCCN(C2CCCC2)C1 24008,n1(CC(=O)NC2CN(C(c3ccc(NC(C)=O)nc3)=O)C2)c(C)cc(C)nc1=O 24009,c1(CC(N2CCCC2c2cccc(OC(F)F)c2)=O)c(F)cc(Cl)cc1F 24010,c1(C(=O)NCC(CNC(=O)Cc2cncc(C)c2)OC)cnn2c1NCCC2 24011,c1(C(=O)NCCNc2sc(C(=O)OC)c(C)n2)ccc(Br)c(C)c1N 24012,N1(C(CC(C)SC)=O)CCCC(C)(NC(=O)C(=Cc2cnn(C)c2)C)C1 24013,C(=O)(CCC(=O)C(C)(C)C)NCC1C(C)CCCN1C(C1CCCCC1(C)C)=O 24014,c1(C(N2CC(CNC(C3C(C(C)C)C3)=O)C(F)(F)C2)=O)c(S(C)(=O)=O)cnn1C 24015,C1(CC(=O)NC(CC=C)CNC(=O)C=CCC)COC(C)(C)CO1 24016,N1(C(CCC(C)=O)=O)CCC2(CCCN2C(c2nn(C)c(C)c2Br)=O)CC1 24017,N1(C(CCNC(C)=O)=O)CC(C(F)(F)F)CC1CNC(=O)CC1CCCC12CC2 24018,C1(CNC(Cc2c(C)noc2)=O)CCN(C(=O)CC(C)n2ccnc2)C(C)C1 24019,C1(NC(Cc2cc(C)sc2C)=O)CC12CCN(C(c1nccnc1N)=O)C2 24020,N1(C(c2c(C)cc(N)cn2)=O)CCC2CC(CNC(=O)C#CC3CC3)CCC2C1 24021,N1(C(c2ccnc(C)n2)=O)CC2CC(NC(c3csc(C(C)(C)C)n3)=O)CC2C1 24022,C1(NC(c2c(SC)csc2)=O)CC2CCC1(NC(=O)CC(C)(C)C#N)C2 24023,C(=O)(C(C)CC(F)(F)F)NCCCCCNC(c1ccc(OCC(C)C)nc1)=O 24024,c1(OCC(=O)NC23CCN(C(N)=O)CCC2C3)cccc2ccccc12.O=C1CN1 24025,CCCCC(C)CCC(=O)NCC(CC)NC(C1CCN(C)C1CC)=O 24026,c1(OC)cc(O)c(CNc2cnc(F)cc2C(N2CCC2CO)=O)c(Br)c1 24027,CC1CN(C(=O)CC(=O)N(C)C)C(C)CN1C(=O)CC1CCCNC(=O)C1 24028,Cc1c(NCCCCN2CCCC2)ncnc1NC1CCCCC1CC(F)(F)F 24029,N1(C(C(C)(C)NC(C)=O)=O)CCC2(CCCCC2NC(=O)COCCO)C1 24030,CCC(CC(=O)N1CC(CC(=O)NC2CCN(C)CC2C#N)CC1C)CC(C)C 24031,c1(C(=O)NCCN(C(c2cc(C)ccc2N)=O)CC)coc2c(Cl)cccc12 24032,c1(NC2(COC)CC2(c2cc(F)c([N+](=O)[O-])c(F)c2)C)c(Cl)cc(Cl)cc1C#N 24033,N1(C(CCC2(C)CCC(=O)N2)=O)CC2CCC(C1)C(NC(=O)C(F)C1CCC1)C2 24034,C12(C(=O)NCC(CCOC)NC(c3ccsc3C(F)F)=O)CCC(OC)C1C2 24035,C1(CNC(Cc2ccc(C(=O)OC)s2)=O)CN(C(c2ncnc(C)n2)=O)CC1C 24036,Cc1ccc2c(C(=O)NCC(C(C)C)NC(C3CN(C)CCO3)=O)onc2c1 24037,C=CCCC(C(=O)NCCC(O)C(F)F)NC(=O)C(=O)NC1CC1 24038,c1(C(=O)NC2C(NC(CC3(C=C)CCC3)=O)CCCC2)cc(F)c2[nH]nnc2c1 24039,c1(OC)cc(C(N2CCCC2CNC(C2C(C#N)C2(C)C)=O)=O)cc(Cl)c1 24040,c1(C(N2C(CNC(C(C)CC(N)=O)=O)(CO)CCC2)=O)cnn2cccnc12 24041,c1(C(N2CCC(N3CCN(C(C(C)O)=O)CC3)C2)=O)n[nH]c2ccc(Cl)cc12 24042,Cc1ncc(C=CC(N2CC(F)(F)CC2CCNC(=O)C(C)C(F)F)=O)c(O)n1 24043,c1(-c2n(CCOCC=C)c(N(CC(C)C(C)C)C)nn2)ccc2cccnc2n1 24044,C1(NC(CSCC=C)=O)C2CC3CN(C(=O)CC4CCCC(C)(C)CC4)C1C3C2 24045,c1(CC)nc(CC(=O)NCC2CC2NC(=O)CC2(NC(C)=O)CC2)cs1 24046,C1(NC(C(C)C(C)(F)F)=O)CCC2(CC1)CCN(C(=O)CN1CC3CC3C1)CC2 24047,C#CC1CN(C(C2(NC(c3cnc(Cl)n3C)=O)CCCC2)=O)CCN1C 24048,N1(C(CC(=C)C)=O)CCC(OCCNC(=O)CCc2nnc(C3CC3)o2)CC1 24049,Cc1ccc(C=CC(=O)NCCCC2CCCN2C(=O)CN(C)C)nc1 24050,C1(CNC(CC(C)C)=O)CCCCN(C(c2cc(=N)[nH]c(=N)[nH]2)=O)C1 24051,C(=O)(CCC(C)NC(=O)CC(C)(C)n1cc(-c2cc(C)ncn2)nn1)OC 24052,c1(N(C(C)C)Cc2cccc(C)n2)nc(=NCCc2cccs2)[nH]c2c1CCC2 24053,C(CC(COC)N=c1[nH]c(=NCC2(C(N)=O)CC2)[nH]c2c1SCC2)OC 24054,N1(C(C(CC#C)O)=O)CC2(CNC(=O)CCCOCCCOC)CC(F)(C1)C2 24055,CC(C)(C#N)C(=O)NCCc1ocnc1CNC(=O)CCc1nncs1 24056,C1(CN(C(N(C2CC(S(C)(=O)=O)C2)CCO)=O)C2CC2)CC2(CCOCC2)CO1 24057,N1(CCOC)CC(NCc2cnn(-c3ncc(Br)cn3)c2)C(C)C1 24058,CC1(C)OCC2CC12C(N1CCN(C2CCN(C(C3OCCO3)=O)CC2)CC1)=O 24059,c1(C(=O)OC)ccc(NC(C2(CNCC3CNCCO3)CCC2)=O)cc1 24060,C(=O)(C(C)CC(C)(C)C)N(C(C)C(=O)NCCCC(N)=O)CC 24061,C1(NC(C2(CC=C)CC2)=O)CS(=O)(=O)C2CN(C(C3CC(OC)C3)=O)CC12 24062,N1(C(CCC=C=C)=O)CC2(C1)CN(C(c1cc(C)nc(C)n1)=O)C2 24063,c1(C(C(=O)NC(C)CN(C)C(c2cnc(Cl)[nH]2)=O)(F)F)ccc(Br)cc1 24064,C1(NC(=O)C(=O)NC(C2CCCCO2)CC2CC2)CC(C2CC2)(C2CC2)C1 24065,C12(CNC(c3c(C)cccc3)=O)CCCC1CCN2C(=O)Cc1cnn(C)c1C 24066,c1(OC)cc(OC)cc(CN2CCC(O)C(C(=O)Nc3ccc(C)c(F)c3)C2)c1 24067,C1(CC(=O)NCC2(C)N=C(C)SC2)CC(C)(C)CN1C(=O)CCC1CCCCC1 24068,c1(CNC2(c3nnnn3C3CCCCC3)CC(C)(CO)C2)ccc(C#N)cn1 24069,C(=O)(C(C#N)C(C)C)NCC1(C(=O)NCCc2ncc[nH]2)CC(=C)C1 24070,C1(C(=O)N(CC(O)C2CCC2)C)(CC)CN(C(=O)C(C)CN(C)C)C1 24071,Cc1nc2sccn2c1C(=O)NC1CN(C(c2cccc3oncc23)=O)C1 24072,C12CN(CC1(F)F)C(=O)c1cn2nn1.C1(CNC(C)=O)CCN(C)C1(C)C 24073,C(=O)(C1=CCCCC1)NCC(C)(C1CC1)NC(c1cnc(OCC)s1)=O 24074,C(CC(O)C(=O)NC1CC(NC(=O)CCSc2ccccc2)C1)SC 24075,c1(CC(=O)NCCOCCN(C(=O)C(O)CF)C)ccccc1OC(F)F 24076,c1(NC)nc2c(c(=NCC3CC4C=CC3O4)[nH]1)CCC2.C1(=O)CCCCC1=O 24077,c1(CNC(C2CC(=C(F)F)C2)=O)cccc2ncccc12 24078,C1(C(N(CCC(=O)NCCCc2ccccc2)C(C)C)=O)COC(=O)N1C 24079,c1(C(=O)NCC(COC)O)n[nH]cc1CNC(=O)CN1CCCC1C 24080,C1(C)(C(=O)NCCCOCCNC(C(C)c2cc[nH]n2)=O)CC=CCO1 24081,c1(C(N2CCC(O)(CN(C(C3C(OCC)C3)=O)C)C2)=O)cnc2cnccc2c1 24082,C(=O)(N1CC(O)CCO1)C1(CC)CCN(C(=O)C(O)CC[S+](C)C)CC1 24083,C1(CNC(c2cc[nH]c2C2CC2)=O)CCC2(CN(C(C3CCSC3)=O)C2)O1 24084,C1(C)(C(=O)NC2CCC(CNC(c3cc(CC)oc3C)=O)C2)CC(C(C)C)=NO1 24085,C1(NC(C(C=C=C)C)=O)CC(F)CN(C(=O)Cc2cc(Br)nn2C)C1 24086,CC1CCCC(CCNC(=O)CC2CC(O)CN2C(c2cnn(CCF)c2)=O)C1 24087,N1(C(CCCCOC)=O)CC(CNC(=O)C2=NOC(C(C)(C)C)C2)C(F)(F)C1 24088,N1(C(C(C)CC(N)=O)=O)CCCC2(CCN2C(=O)CCN2CCCCC2)C1 24089,Cc1nn(CCF)cc1NC(=O)CCC1CCN(C(C2C3CCCOC23)=O)C1 24090,Cc1cc(C)c(CC(=O)NCC(F)CNC(=O)C(c2ccccc2)=O)s1 24091,C(CC(O)C(=O)N1CC=CC1CNC(=O)CSC(C)C)SC 24092,C12(NC(C3CC4CCC3C4)=O)CCC(CC1)N(C(c1cnc3occc3c1)=O)C2 24093,n1(CC)nnc(C(=O)NCc2csc(CNC(c3cc[nH]n3)=O)n2)c1C 24094,c1(C(=O)NCC(CO)NC(CC2CC(=O)NC2)=O)cccc2nccnc12 24095,Cc1nc(C2CC2)ncc1C(=O)NC(CCNC(=O)C(C)NS(C)(=O)=O)C(C)C 24096,CC(C)(C)CCCC(=O)NC1CCN(C(=O)CC2(CCCO)CCCC2)C1 24097,c1(C(c2nnnn2CC2CCCO2)(C)NC2CCOCC2)nc2c(s1)CCCCC2 24098,CC1CCCN(C(c2c[nH]c(=O)cn2)=O)C1CNC(C1CC(Cl)(Cl)C1)=O 24099,N1(C(C2(C(F)(F)F)CC2)=O)CCC2CN(C(=O)C(F)(F)Cl)CC2C1 24100,Cc1cc(O)c(Cl)cc1C(N1CCC(C(C)(C)NC(c2ccncc2)=O)C1)=O 24101,N1(C(CCCC=C)=O)CC(C(N2CCCC2CSC)=O)C2(CC2)C1 24102,CC(CCC(=O)N1CCOC(CCO)C1)NC(=O)C=C1CCC1 24103,N1(C(CN(C(C)=O)C)=O)CC(C(N)=O)(CNC(C2(c3ccno3)CCC2)=O)C1 24104,Cc1coc(C)c1C=CC(N1CC(O)(CCNC(C2COC(C)C2)=O)C1)=O 24105,C1(N(C(C=CC)=O)C)CN(C(=O)C(C)N(CC(F)(F)F)C)CC1(C)C 24106,c1(C(=O)NC(CN(C(c2nscc2C)=O)CC)C)cnn(C(C)(C)C)c1 24107,c1(C(=O)NCC2(NC(CSCC)=O)CCOC2)[nH]nc(NC)c1Br 24108,C1(C(N(C2CCN(C(=O)OC(C)(C)C)CC2)C2CC2)=O)SC2C=CC1CC2 24109,CC(C)C(C)CC(=O)NCC1CCCC(CNC(=O)C=Cc2ccncn2)C1 24110,C1(C(N2CCC(N(C(=O)CNC(c3cccs3)=O)C)C2)=O)CC2(CC(=O)C2)C1 24111,Cc1c(C(N2CCN(C(c3c(Cl)cnn3C)=O)C3CC23)=O)cccc1O 24112,c1(COC)ccc(C(=O)NCC2CC(CNC(=O)CCc3cncn3C)CO2)o1 24113,N1(C(c2c(CC)ccc(Br)c2)=O)CCCN(C(=O)CC2CC(C)C2)CC1C 24114,c1(C(N2CC(N(C)C(C3CN(Cc4ccccc4F)C3)=O)C2)=O)nnc(O)nc1O 24115,C(=O)(CC(C1CC1)NC1CCCN1C(=O)CCCN(C)C)OC 24116,S(=O)(=O)(c1cnc(NCCN2CCC(C)(C)C2)c(Cl)c1)NC(C(OC)OC)C 24117,C1(C)(C(=O)NCCCNC(C2(C)CC(C(F)(F)F)C2)=O)CC2CC2C1 24118,C(=O)(C(O)CC(F)F)N1CC(O)(CCNC(CCC2C(C)=NOC2=O)=O)C1 24119,C1(CCOC)CCCCC1NC(C1(CCOC)CN(C(=O)CC2CCCO2)C1)=O 24120,C1(CC(=O)NC2(C)CN(C(c3cnc(O)c(F)c3)=O)C2)CC2(CCCC2)CO1 24121,N1(C(C(C)CC(F)(F)F)=O)CC2N(C(c3ccn4ccnc4c3)=O)CCC2(C)C1 24122,c1(C(N(CCCN(C)C(C2(F)CC3(CCC3)C2)=O)C)=O)ccc(F)c2c1CCC2 24123,c1(C(=O)OC)c[nH]c(=NCC23CCC(CNC(=O)CC(C)(C)C)(CC2)OC3)cn1 24124,C1(C(=O)NCCC(C)NC(c2cc(Cl)cc(Cl)c2N)=O)OCC2COCCC12 24125,N1(C(COCCOCC#C)=O)CCCC12CCCN(C(=O)C=CCC)C2 24126,CC1(C)C2CCC(C2)C1(C)C(=O)NCc1ccccc1CNC(c1csnn1)=O 24127,C1(C(N(CCN(CC)CC)C)=O)C2CC3C(C2NC(=O)C(C)(C)n2ccnn2)C13 24128,c1(C(=O)NCCNC(C2CC(=O)N(C3CCS(=O)(=O)C3)C2)=O)ccc2c(c1)CC2 24129,c1(C(=O)NCCNC(C(C(C)C)c2cc(C)no2)=O)cc(C)ccc1S(N)(=O)=O 24130,c1(C(=O)NC(CNC(C2(CSC)CC2)=O)COC)ccncc1N=[N+]=[N-] 24131,c1(CN2CCC(N(C(C3CCN(C)C3)=O)CC)C2)cccc(Cl)c1Cl 24132,N1(C(C2(CC)COC2)=O)CCC(C2CCCN(C(=O)C=CCO)C2)CC1 24133,N1(C(c2c(C#C)c[nH]n2)=O)CCC(C2CC2)C1CNC(C1C=C(C)CS1)=O 24134,CC1CN(C(C2(Cc3ccc(F)cc3)CCCO2)=O)CCN1C(=O)C(F)F 24135,c1(C(C)C)ccc(C=CC(=O)NC23CCC2CN(C(=O)CC2CC(F)C2)C3)cc1 24136,Cc1nc2cnn(C)c2cc1C(=O)NC1CCCN(C(=O)CC(O)C(C)C)CC1 24137,c1(C(=O)NCCC(CNC(c2ccnn(C)c2=O)=O)O)c2c(nn1C)CCSC2 24138,CC1CC(NC(C2CN(C)C(=O)N2)=O)CCN1C(=O)Cc1nnc(O)s1 24139,c1(CCC(=O)NC2CCOCC2NC(C2CCOC2=O)=O)ccccc1F 24140,C1(O)(CNC(C2(NC(C(C)Sc3ccccc3)=O)CC2)=O)CC2CCC1C2 24141,C(=O)(C1=C(C#N)CCC1)NC(CC(=C)Cl)C(=O)N1CCCC(CCC)CC1 24142,c1(C(N2CCCC(CN(C(C3(C=C)CC3)=O)C)C2)=O)cc2cc[nH]c(=O)c2s1 24143,C1(C2CCCO2)CCC(NC(=O)NCCNC(=O)C2CC2)C1 24144,c1(CC(=O)NCC2C=CC(NC(C(CCC)N(C)C)=O)C2)cc(C)ccc1F 24145,C1(NC(c2nccc(CNC(C(C)C#N)=O)c2)=O)Cc2cscc2C1 24146,CCC(CC(=O)NC(C)(CO)C(=O)N1CCC(N2CCC2)CC1)C1CC1 24147,c1(C(=O)NC2CN(Cc3c(Br)ccc(OCC)c3)C2)ccc(O)c2ccccc12 24148,C12(C(=O)NC3CC4C(NC(c5c(C(C)C)cco5)=O)C4C3)CCC(C1)C(C)(C)O2 24149,C(=O)(CCCCCF)N1CCC(Cn2cc(C3(OCC)CCOC3)nn2)C1 24150,C1(C(N(C)CC2CCN(C(Cc3nnc(C)o3)=O)C2)=O)CC(F)(F)CS1 24151,C1(C)(C(=O)NCCCOC(C)C)CCCN(C(=O)CC2CCOCC2)C1 24152,C1(NC(COCCC)=O)CCC2(CCN(C(c3cc(CC)ccc3N)=O)C2)C1 24153,CC1(C)CCCC1CCNC(=O)C(=O)Nc1ccc(CN2CCCCC2)cc1 24154,S(=O)(=O)(c1ccc(NC(C)CCC(C)C)cc1Br)NC1(C)c2csc1n2.CC.CC 24155,O=S1CCC(CCNCc2n[nH]c(Br)n2)C1 24156,C(=O)(CCS(N)(=O)=O)NCCC(C)NC(C(c1cccc(C)c1)SC)=O 24157,c1(COC)cscc1C(=O)NC(C1(C(=O)CNC(c2ccccc2)=O)CC1)C.C 24158,Cc1ccn(CC(N2CCC(F)(CNC(=O)CC(=O)NC3CC3)C2)=O)c(=O)c1 24159,c1(N2CCC(CCCO)CC2)[nH]c(=NCC2(CF)CCC2)nc2scnc12 24160,CCC(C)(CO)C(=O)NC1CCCCCC1NC(=O)Cn1cc(C(=O)NC)nn1 24161,N1(C(CCOC(C)C)=O)CCN(C(C2CCC(=O)NC2)=O)C2(CCC2)C1 24162,N1(C(C(C)OCC#C)=O)Cc2nccn2CC(NC(=O)C2=CCC(C)(C)C2)C1 24163,c1(CNC(c2ccon2)C)cccc(-n2cncn2)c1 24164,N1(c2nc(NCC(C)(C)C)c3c(n2)scc3)CCCC(C2CC2(F)F)C1 24165,c1(CC(N2CC(CNC(COCC#C)=O)C(OC)C2)=O)c(OC)cccc1O 24166,C(=O)(CCC(C(=O)N(CCCNC(c1cnn[nH]1)=O)C)N(C)C)OC 24167,c1(NC(=O)Nc2cccc(C(F)F)n2)ccc(N=Nc2ccccc2)cc1 24168,CC1CN(C(=O)Cc2csnn2)CCC1NC(c1ccc(C(F)(F)F)cc1N)=O 24169,C1(C(=O)NC2CCC(NC(CC3(CN(C)C)CCC3)=O)CC2)OCC2CCCC12 24170,c1(NC(C2C3CN(C(c4ccnnc4O)=O)CC23)=O)ncc(Cl)nc1Cl 24171,N1(C(C)=O)CCCC2C1CCCN2C(=O)CC(F)(F)CS(C)(=O)=O 24172,C1(C(=O)NC2C(O)CCN(C(c3n(CCC)ncc3)=O)C2)CCn2cnnc2C1 24173,c1(C(=O)NC2C(NC(C3CCC(C(=O)OC)CC3)=O)C2)cc(C(F)F)cc(F)c1 24174,C1(C)(CNC(C(C)OCc2ccc(OC)cc2)=O)CN(C(c2cocn2)=O)CCO1 24175,c1(CNC(N2CCC(c3ccncn3)C2)=O)cc(O)ccc1F 24176,N1(C(c2c(OC)c[nH]n2)=O)CC2OCCN(C(C3CC34CCSCC4)=O)C2C1 24177,C1(N(C(=O)CC2CC23CC3)CC)CCN(C(=O)CC2OCCO2)CC1 24178,c1(CNC(C(COC)OC)=O)ccc(CCNC(c2c[nH]c(C#N)c2)=O)cc1 24179,C(=O)(C(O)C(C)(C)C)N1CCC(C(=O)NC(c2cncnc2)C)(CC)C1 24180,C12(NC(C=C(C)CN3CCOCC3)=O)CC(CNC(C3(C(N)=O)CCCC3)=O)(C1)C2 24181,CC1CCn2cc(C(=O)NCCC3=CCN(C(=O)Cc4nc[nH]n4)CC3)nc2C1 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24216,c1(OC)cc(F)ccc1C(=O)NC(C)CNC(C1CC=C(C)CC1)=O 24217,C1(C(=O)OC)CCN(C(=O)C2CN(C(=O)CN3CC4CCC3C4)CC23CC3)O1 24218,C1(CNC(=O)CCc2nc[nH]n2)COC(CNC(=O)CSC2CCCC2)C1 24219,N(C(=NCCCCl)NCC1CC12CCSCC2)C(c1ccc(OC)cc1)CF 24220,C1(CNC(CNC(CC)=O)=O)CN(C(=O)CCCC(C)=O)CC1(F)F 24221,C(C(=O)NCCC(C(C)C)N(C)C)(C(C)(C)O)NC(C(CCOC)C)=O 24222,c1(C(N(CCOC)CCNC(=O)CNS(=O)(=O)CC)=O)nc(C)nn1C 24223,C1(OC)(CNC(=O)CCc2ncnn2C)CN(C(c2ccc(C(C)(C)C)[nH]2)=O)C1 24224,c1(CN2C(NC(=O)C(O)CCC)CC(=C)C2)c(Cl)nc(SC)nc1Cl 24225,C1(CNC(C(CSCC)C)=O)CCCCN(C(c2c[nH]c(=N)nc2SC)=O)C1 24226,c1(CC(=O)N(C)CC2CN(C(c3c(CC)occ3)=O)C2)ccccc1C(N)=O 24227,c1(CN(CCC)CCNC(=O)Cc2csc(C)n2)cc(C)ccn1 24228,N1(C(c2cn(C)nc2C(F)F)=O)CCC(NC(C2(C)C=CCC2)=O)C(F)C1 24229,C(=O)(C(F)C(C)(F)F)N1CC(C)(C(=O)NC(C2CC2(C)C)CC)C1 24230,C(C1=CCN(C(c2ccc(Br)cc2F)=O)CC1)NC(C1CC12CCCC2)=O 24231,C(=O)(CC(C)C(F)F)NCCCC1CCN(C(C2(CC)CC(F)(F)C2)=O)CC1 24232,c1(C(=O)NC(CC2CCOCC2)C(=O)N2CCC2CO)ncnc(O)c1F 24233,c1(C(=O)NC2CC(NC(c3cnc(OCC)s3)=O)C2)nccc(OC)c1N 24234,CC(C)C(C)(O)C(=O)NC(Cc1ccccc1Br)C(=O)N(C(C)C(=O)N(C)C)C 24235,c1(C(CC)NCC2CCC(C)O2)ccc(O)c(Br)c1 24236,c1(C(=O)NCC2N(C(C(C(=O)OCC)F)=O)CC2)c(F)ccc2nc[nH]c12 24237,C(CC(C)(c1nnnn1C(C)(C)C)NCC1(C)CC1(C)C)OC 24238,C(CCC(=O)N1CCCC1CN(C)C)(C(C)C)NC(C=Cc1cc(C)no1)=O 24239,c1(C(=O)NCCC2(C)CCN(C(=O)CCC3CC3)C2)ccn2ccnc2c1 24240,Cc1cc(C(=O)NCC2(CNC(=O)C=Cc3cncs3)CC2(F)F)ccc1O 24241,CC1C2CC(C2NC(c2ccc(Br)o2)=O)N1C(c1cncc(C(N)=O)c1)=O 24242,C1(CCC)CN(C(=O)C(C2CCCCC2)C)CCN1C(c1cc(C)n(C)c1)=O 24243,N1(C(C2C(C)OCCC2)=O)CCN(C(c2cc(S(C)(=O)=O)co2)=O)C2CCC12 24244,C1(C(N2CC(C)C(C)(C(=O)O)C2)=O)CC(F)(F)C12CCCC2 24245,c1(C(=O)NC2C3(CC(NC(=O)COCC(F)F)C3)C2)ccc2cnnn2c1 24246,C1(C(=O)OC)CC2CC1CC2NC(=O)Nc1cc(C(F)(F)F)cc(C)c1 24247,CC1CCN(C(=O)CCc2c(F)cccc2F)CC1NC(=O)C=C1CCCCC1 24248,N1(C(CC)CC(=O)OC)C(=S)NC(c2ccc(Br)c(N)n2)C2=C1C(C(C)(C)C)NC2=O 24249,C1(NC(c2c(Cl)cn(CC)n2)=O)COCCN(C(=O)C(C)Cn2ccnc2)C1 24250,c1(C(=O)NCCN(C(C(CC)C(=O)OC)=O)CC)cc2ccccc2o1 24251,C1(C)C(=O)N1.C1(CN(CC)CC)CC(CNC(=O)CCSCC(N)=O)C1 24252,N1(C(C2CC(=C)C2)=O)CCC(CF)(NC(c2cnc(C3OCCO3)s2)=O)C1 24253,c1(N2CC(C)(C)SCC2)nc(N2CCOC(C)(C3CC3)C2)nc2c1SCC2 24254,C1(C(=O)NCc2n[nH]c(-c3cccc(Cl)c3)n2)CCCC2(CC2)C1 24255,c1(CNC(C2CCC2C(=O)N(C)C)=O)ccc(CNC(CC2C(C)C2)=O)cc1 24256,Cc1c(CC(=O)NCC2(CCNC(=O)CC3CC=CC3)CC2)ncn1C 24257,N1(C(CNS(C)(=O)=O)=O)CC2COCCC2(NC(c2ccn3cncc3c2)=O)C1 24258,Cc1cccc(C(=O)N(C2CCC(NC(C3CN(C)C(=O)N3)=O)CC2)C)n1 24259,N1(C(C(CC)Cl)=O)CCC2(CCC(C(=O)Nc3ccccc3C(C)O)O2)CC1 24260,c1(NC(COC(C)(C)C)CO)ccc(S(=O)(=O)N(C2CC2(Cl)Cl)C)cc1Br 24261,C1(C(=O)NCCOC2CN(C(C(C=C)O)=O)C2)CCC2C(CC1)C2(F)F 24262,N1(C(c2c(C)ccs2)=O)CCC(NC(=O)C(c2ccc(F)cc2F)C)C(F)C1 24263,C=CC(CC(=O)NCC1(C)CCCC1C)c1ccc(OC)cc1 24264,C(=O)(C1=C(Cl)CCC1)N(C1CCN(C(=O)C(c2cccnc2)OC)CC1)CCC 24265,c1(OC)ccc(Cl)c(C(N2CCCC2CCNC(C2CC(C)(C)CN2C)=O)=O)n1 24266,c1(CC(=O)NC2CC2CNC(C2CS(=O)(=O)C2)=O)cc(F)c(F)cc1F 24267,C(CN=C(NCc1cccc(-c2cc[nH]n2)c1)NCc1cccs1)C1(C)CC1(Cl)Cl 24268,C1(C(=O)NC2(CF)CCN(C(c3nccc(CC)c3)=O)C2)CCCCS1(=O)=O 24269,c1(C(=O)OC)cnc(NCC2CC(C)N(C(=O)CN(S(C)(=O)=O)C)C2)nc1 24270,c1(C(C(N2CCC(O)(C(C)C)C2)=O)(F)F)ccc2c(c1)OCO2 24271,Cc1cncc(C(=O)NCC2CC2CNC(c2ccc(=N)[nH]c2Cl)=O)c1Cl 24272,N1(C(c2cc(C)nn2C)=O)CCN(C(c2c(C)coc2C)=O)CC12CC2 24273,c1(C(N2CC3CC2CO3)=O)ccc2nc(-c3ccnc(OC(F)(F)F)c3)sc2c1 24274,N1(C(C2CCC(C(C)C)CC2)=O)CCCN(C(=O)C(CO)NC(N)=O)CC1 24275,Cc1cc(C)nc(SCC(=O)N(C2CCN(C(=O)C(C)C(C)(C)C)CC2)C)n1 24276,Cc1ccc(Br)c(F)c1C(N1CC2CC1C2C(N1CC2CC1CC2(F)F)=O)=O 24277,C(=O)(CC(O)C(C)C)NC(CCOC)C(=O)NC12CC1CN(C)C2 24278,N1(C(CN(C(=O)C(O)C(F)(F)F)CCC)=O)CC2(COCC(=O)N2)C1 24279,c1(C(=O)NCC(CCNC(CC2CCCC(C)(C)C2)=O)O)cnn2cccnc12 24280,N1(C(=O)NCc2c(CC)ccc(F)c2)CCc2cc(OC)ccc2C1C 24281,c1(C(N(C2CCN(C(C3CCSCC3)=O)C2)CC)=O)nc(OC(C)C)ccc1Cl 24282,c1(C2(C(=O)NCCNC(C3(C#N)CC3C(F)(F)F)=O)CC2)ccc(O)cc1 24283,C(C(=O)N1CC(NC(=O)CC2(CO)CCC2)C(C)C1)(C(C)(C)C)NC(C)=O 24284,c1(NC(CN(C(=O)COC(=O)CC2CCCO2)C)=O)cccc2ncccc12 24285,C1(N(C(C(C)SCC)=O)CCCN(C(C)C)C2CC2)CCCC1n1ccnn1 24286,C(C(CC(C)C)C(=O)N(C)Cc1c(C)cnn1C)NC(CC(C=C)C)=O 24287,C1(NC(C(CC)NC(C)=O)=O)COCCC1C(=O)N(CC)Cc1cnco1 24288,N1(C(C(CC)C)=O)CCN(C(=O)CNC(c2ccccc2C)=O)CC1 24289,c1(CC)cccc(C(=O)NCC2CCCN(C(C3(C)CC3(C)C)=O)C2)c1N 24290,c1(NC(CC(CC)n2cc(NC(N)=O)nn2)=O)ccccc1C#N 24291,C1(NC(C2CCOCC2)CCOC)CCC(C2CCC2)CC1 24292,c1(CNC(Cc2ccc(C)o2)=O)ccc(C(=O)NCc2ccoc2)cc1 24293,N1(C(c2c(CC)cco2)=O)CC2CC(C1)CN(C(C1CC(=O)OC1(C)C)=O)C2 24294,c1(C(=O)NC2CCC(CNC(C3C(=C)C3C(=O)OC)=O)C2)c(F)cc(Cl)cc1F 24295,N1(C(CC2(CNC(c3n(CC)ncc3)=O)CC2)=O)CC2(CC2)CC1C(=O)NC 24296,C(=O)(CCCCCN=[N+]=[N-])N1CC(CC)N(C(=O)CC(C)c2cnn(C)c2)CC1 24297,CCC(C)C(O)CC(=O)N(CCCCCNC(C1(C(=O)N(C)C)CC1)=O)C 24298,c1(C(=O)NCC(CN(C(C(C)SCC)=O)C)O)ccn(CCN(C)C)n1 24299,c1(CC)cccc(C(=O)NC2CC(NC(=O)CC3CCCO3)CC2O)c1 24300,c1(OCCCC)ccc(CNC(=O)C(=O)NCC2CCC(O)C2)c(O)c1 24301,c1(C(N2CCC(C)(CNC(C3CC(SC)C3)=O)CC2)=O)cc2cc(Cl)cnc2[nH]1 24302,CC1(C)CCCOC1CC(N1CCOC(CNC(C2CC(=O)N(O)C2)=O)C1)=O 24303,N1(C(C(C2CCC2)OC)=O)CC(CNC(C2CCCCC2O)=O)C(C)C1 24304,Cc1cc(C(N2CCC(CNC(c3ccc(O)nc3)=O)C(C)C2)=O)[nH]c1C#N 24305,C1(C(N2CCC(N(C(C(c3ccccc3F)C)=O)CCO)C2)=O)C(C)(C)C1(F)F 24306,Nc1ccc(CCCC(=O)NC2CCOC(CNC(=O)COC(F)(F)F)C2)cc1 24307,Cc1ccc(S(=O)(=O)N2CCN(CC(=O)NC3CCCC3)CC2)nc1 24308,Cc1ncnc(C(N2CC3CC3(CNC(C3CC3(Cl)Cl)=O)C2)=O)c1C 24309,C=CC1CCCCN1C(=O)Cn1cc(CNC(c2cc(C(C)=O)c[nH]2)=O)nn1 24310,c1(C(=O)NC2CC(NC(CC3(C(=O)OCC)CCC3)=O)C2)ccc(C)cc1 24311,c1(CC(=O)NC(CNC(C2C(CC)CCO2)=O)(C)CC)cnn2ccccc12 24312,N1(C(c2c(CC)con2)=O)CC(NC(C2CCC(C(F)(F)F)CC2)=O)C2(CC2)C1 24313,c1(N2CC(OC)C(F)C2)nc(Nc2cc(N)ccc2C)c2cnn(C)c2n1 24314,n1(CCOC)cc(C(=O)NCC(C2CC2)NC(=O)CC2CCCCCC2)c(C)n1 24315,Cc1ccc2oc(C(=O)NC(C3CN(C(C4CCC4(C)C)=O)C3)C)c(C)c2c1 24316,c1(C(=O)NC2CN(C(C(CCOC)OC)=O)C2)ccc(S(N)(=O)=O)[nH]1 24317,N1(C(c2c(C)ncc(Cl)c2)=O)CC2(CCN(C(=O)C3=CCCCC3)CC2)CC1C 24318,N1(C(C(C)(C(C)C)OCC)=O)CCCN(C(c2cnc3c[nH]nc3c2)=O)C(C)C1 24319,C1(C(C)C)CCOC1C(=O)NCCCN(C(=O)C(C1(O)CCCC1)F)C1CC1 24320,N1(C(CC(C(C)C)O)=O)CCCCC12CC(NC(=O)COC1CCCOC1)C2 24321,C1(C(C(=O)N(CC(O)CNC(c2cc(O)cs2)=O)C)O)CCS(=O)(=O)CC1 24322,Cn1cc(CNC(C2C3(CC(NC(=O)CC45CCC(CC4)C5)C3)C2)=O)ncc1=O 24323,C(=O)(CC(F)(F)F)N(CCOC(c1nsc(CCN(C)CCOC)n1)=O)C 24324,CC(N=c1[nH]c(N(C)Cc2ccoc2)nc2c1CCC2)c1cc(Cl)cc(Cl)c1 24325,C(=O)(C1OCCc2ccccc21)N1CC(CC)(CNC(=O)C(CSC)N(C)C)C1 24326,C1(CNC(c2cnc(C(C)C)[nH]2)=O)CCC(CNC(C2CCN(C)C2)=O)CC1 24327,FC1(F)CCC1CN1CCOCC1.C(CC1=NOCC1)c1nnnn1C1CC1 24328,C(=O)(C1CCc2c[nH]nc21)NC(C(NOCC)=O)c1ccccc1 24329,C(C)(CCC(=O)NC1CC1CNC(c1cnc(-c2ccccc2)[nH]1)=O)OC 24330,C1(CNC(CN(C2CC2)CC)=O)CC2(CCN(C(C3(CC(C)C)CC3)=O)CC2)CO1 24331,c1(-n2c(C)ncc2)ccc(CC(N)C(=O)N2CCCC2c2cccnc2)cc1 24332,c1(C(=O)NC(CC)CN(C(=O)C(F)C(F)(F)F)C)c(F)cc(C#N)cc1F 24333,C1(CNC(CN(C)CC)=O)(CO)CCCN(C(c2cc(C)nc(O)n2)=O)C1 24334,C1(CNC(Cc2cc(C)[nH]n2)=O)(CO)CCN(C(c2sccc2C#N)=O)C1 24335,c1(C(=O)NCC(CC=C)NC(=O)C(F)(F)C(F)F)cc(N)c(O)c(F)c1 24336,n1(CC2CC2)cc(COC(C=C(C=CC)C)=O)c(CCOC)n1 24337,C(=O)(C1=NOC(C)C1)NCc1scc(CNC(c2c(C)cco2)=O)n1 24338,C1(C(=O)NC(C)C(C)NC(c2cnoc2-c2ccoc2)=O)CCCC2(CC2)C1 24339,CC1(C)CC(C(=O)Nc2cnc(Cl)nc2)N(C(C2CC(=O)OC2(C)C)=O)C1 24340,C1(C(N2CCC(C#C)(O)C2)=O)CC12CCN(C(C13CCCC(CO1)C3)=O)CC2 24341,n1(C(CC)C)ccc(=NC(=O)CC(CC(C)C)NC(C2C=CCCC2)=O)[nH]1 24342,N1(C(C(C)CN(C(=O)CCC2OCCO2)C)=O)CCC(CO)CC1 24343,N1(C(c2c(COC)cc[nH]2)=O)CC2CC(NC(C3CN(C(C)C)C3)=O)CC(C2)C1 24344,N1(CCCNC(C(C)OC)=O)CCC(NC(=O)C(C)(C)O)C1 24345,C(=O)(C1CCCc2scnc21)N1CCC(CNC(c2n(C)c3c(c2)scc3)=O)C1 24346,C(C)(CN=c1cc(COC)nc[nH]1)(C(C)C)NC(c1ccc(CC)cc1)=O 24347,C(C)(Cc1ccccc1)(C(F)(F)F)N(CC(N1CCN(S(C)(=O)=O)CC1)=O)C 24348,C12CCC(F)(C1)CNC2=O.c1(C2C(N(C(=O)C(C)C)CC)C2)ccc(Br)s1 24349,C(=O)(C(CC)(CC)c1ccccc1)NCC(CCCC)NC(=O)OC(C)(C)C 24350,C1(C(=O)NCCN(C(=O)CN(C)Cc2ccccc2)C(C)C)CN(C)CC(C)O1 24351,C1(CC(=O)OC(C(=O)NCc2c(C(=O)OC)cccc2)=O)COC2(CCCCC2)O1 24352,Nc1cccc(C(N2CC3(C2)CN(C(=O)Cc2c(F)cncc2Cl)C3)=O)c1O 24353,C(C(F)(C(=O)N(C1CCCC(C)C1)CC)C(C)C)NC(COCCC=C)=O 24354,N1(C(C2C(C)(C)C2(F)F)=O)CCC(NC(c2ccnc(N(C)C)c2)=O)C12CCC2 24355,N(C(=NCCF)NCC1CC2CCC1O2)CC(N1CCCCCC1)(C)C 24356,C#CCCCCCCCNC(=O)C(CC(N)=O)NC(=O)C(C(C)C)NC(C)=O 24357,C12(C(=O)NCC3(C(F)(F)F)CCC3)CC(CNC(C(C3CCC3)OC)=O)(C1)C2 24358,C1(C(NOC(C=O)CC(NOC(C(C)C)CO)=O)=O)COC(=O)N1C 24359,C1(NC(=NCC=C)NCCS(=O)(=O)NCC2CCC2)CC2(C1)CC(F)(F)C2 24360,N1(C(c2n(CC)ccc2)=O)CCC(C2CCCN(C(=O)C(=O)C(C)CC)C2)CC1 24361,C12(NC(C=CC)=O)CC(CNC(=O)CC(C)c3ccccc3)(C1)OC2(C)C 24362,c1(C(N(C)CC2CN(C(Cc3scc(C)c3)=O)C2)=O)ccc(Br)nc1C 24363,N1(C(c2n(CC)cnn2)=O)CCCCC(N=c2ccc(C(F)(F)F)n[nH]2)C1 24364,C1(NC(c2cnc(CC)[nH]2)=O)(CNC(c2cc3c(s2)CCC3)=O)CC2CCC1C2 24365,c1(C(=O)NCCC2N(C(C(N3CCOCC3)C)=O)CCC2)cc2ccccn2n1 24366,C1(CNC(c2c(C(C)(C)C)nccc2)=O)CC(O)CN1C(C1CCS(=O)(=O)N1)=O 24367,C(=O)(C(CO)C(C)(C)C)N1CC(CCNC(=O)Cn2ccc(O)nc2=O)(OC)C1 24368,N1(C(CCCC#C)=O)CCC(C(=O)NCC2(O)CCC(C)C2)C12CCC2 24369,c1(CC(=O)NCCC2CCCN2C(=O)CCc2cn[nH]c2)cn(C2CC2)cn1 24370,c1(C2N3CCCC3CNC2=O)cc(Cl)ccc1Cl.c1(C(=O)NCCO)cccs1 24371,N1(C(C(COC)OC)=O)CC(CNC(c2cccc(-n3cccc3)c2)=O)CC1C 24372,Cn1cc(C=CC(=O)NC2(C(=O)N(CCO)CC3CC3)CC(F)C2)nn1 24373,N1(C(c2cnc(C)c(N)c2)=O)CCC2(CCCC2CNC(C2(Cl)CC2)=O)CC1 24374,c1(C(=O)NCC2C(CNC(C(C)(C)OC(C)C)=O)C2)cn2c(n1)CCCC2 24375,c1(C(N2C3C(NC(c4c(C)nncc4)=O)CC(C3)C2)=O)c(F)cc(N)cc1F 24376,c1(OC)ccc2ccnc(C(C)NC(=O)C(=O)NCC3CCNCCO3)c2c1 24377,C(N=c1nc(N2CCCC(CF)C2)cc(C)[nH]1)C1N(CCC)CCCC1 24378,Fc1cc(Cc2nc(-c3cccc(Cl)c3)nn2CC2CCCCCC2)ccc1Cl 24379,N1(S(C)(=O)=O)CCOC(CNC(=O)Nc2ccc(NCc3ccccn3)cc2)C1 24380,C1(CNC(c2ccc(OCC)cc2)=O)CCC(C)CN1C(c1cccc(O)n1)=O 24381,C1(CCNC(c2c(C)ocn2)=O)CCCN(C(C2CCCOCC2)=O)C1 24382,c1(C(=O)OCC)cc(C(=O)NCC(CO)NC(=O)C(F)=C2CCC2)[nH]c1C 24383,C1(NC(C(c2cccnc2)C)=O)CC12CCN(C(C1CC(N=[N+]=[N-])C1)=O)C2 24384,C1(CC)(CC)CC(NC(C2CC2C2CC2)=O)CN1C(=O)CCCF 24385,C(C(=O)N1CCC(NC(=O)CCc2ccccn2)C1C)(C(C)C)SC 24386,c1(C(=O)NC(C)CCCNC(c2cn(C3CC3)cn2)=O)cccc2nc[nH]c12 24387,N1(C(C)(C)C)CC(C(N2CCC2CNC(C2(c3ccsc3)CC2)=O)=O)CC1=O 24388,Cc1ccc(C(N2CCC(NC(=O)CN3CSCCSC3)C2)=O)cc1OC(F)F 24389,N(C(=NCC(C(C)(C)C)OC)NC1CCN(C(=O)C(C)C)CC1)C(COCC)C 24390,CCC(CC(=O)NC1CC=C(C(=O)NCCCC2CCC2)C1)C(F)F 24391,C1(C(N(CCCF)C)=O)(NC(=O)CCC2CCOCC2)CCSC1 24392,c1(C(N2CCC(NC(C(C=C)O)=O)C(F)C2)=O)c(C)cc(O)cc1C 24393,Cc1cc(C(N2CC3(NC(c4nnc(S)n4C)=O)CCC2C3)=O)cc(N)c1O 24394,C1(C(N2CC(NC(CCN(CCC)C)=O)C3(C2)CC3)=O)CCC2(CC1)CC(O)C2 24395,C(=O)(C1=NNC(=O)CC1)NC1C(NC(c2c(C)ccnc2O)=O)CCCC1 24396,CC1(C)CN(C(=O)C2=CCCCO2)CC1C(=O)NC1CC2C=CC1C2 24397,c1(OC)cccc(C(=O)NCC(C)CNC(c2cnc(CC(C)C)s2)=O)c1N 24398,c1(C(N2CC(N(C(C(C)OCC#C)=O)C)C(C)(C)C2)=O)cncc(C=C)c1 24399,C#Cc1ccc(C(=O)NC(C2CCCN2C(c2ccc(=O)n(O)c2)=O)(C)C)nc1 24400,C(=O)(CC(C)C(C)(C)C)NCC1N(C(C(CC(=O)OC(C)(C)C)O)=O)CCC1 24401,c1(NC(C2C(C(N(CC#C)C)=O)C2)=O)cc(Br)cc(F)c1OC 24402,c1(C(=O)NC2CC(OC)CN(C(C3C(=C)C3)=O)C2)c[nH]c2c(C)cccc12 24403,Cc1c(C(=O)NCC2(CN(C(=O)C(C)CS(C)=O)C)CC2)ccc2c1CCC2 24404,c1(N(C(=O)C2=CCCC2)CC#C)cccc(C(N2CCC(N(C)C3CC3)C2)=O)c1 24405,c1(OC)nc(CCNC(=O)C(COC2CCCC2)NC(=O)OC(C)(C)C)sc1C 24406,CC1COCCCN1C(C1CC(O)CN1C(=O)Cn1cnnc1)=O 24407,c1(C(=O)NCC(CNC(c2cc(CC)on2)=O)(C)O)c(C)[nH]cc([N+](=O)[O-])c1=O 24408,N1(C(C2C(NC(=O)Cc3ccccc3[N+](=O)[O-])C2)=O)CCc2cc(O)ccc2C1 24409,C1(C(N2CCC(C)(CNC(C3N(C)C(=O)CC3)=O)C2)=O)C(F)(F)C12CCC2 24410,c1(CC(=O)N(CC(CC)NC(C(C)SCC)=O)C)cccc2ncccc12 24411,Cc1n[nH]c(C)c1C(C)CC(=O)N1CCCC1Cn1cncn1 24412,C(=O)(N=S1(=O)CCNC(CNC(=O)OC(C)(C)C)C1)c1nc2c(ccc(C)c2)n1C 24413,N1(C(COC(C)=O)=O)CC=C(C(C)(C)C(=O)N(C)CC2OCCC2(C)C)C1 24414,C1(C(c2cn(Cc3nncn3C)nn2)C)CCN(Cc2cnoc2)CC1 24415,C1(C(=O)NCC2(c3ccccc3)OCCO2)Cc2ccncc2C1 24416,C(CC(C(=O)NCc1ccc(F)cc1)NC(C1CCS1(=O)=O)=O)=CC 24417,C12(NC(C3OCCC(C)C3)=O)CC(CNc3cc(CC4CC4)ncn3)(C1)OC2C 24418,Cc1ccnc(C(=O)NCc2ncc(C(=O)NC(c3cn(C)cn3)C)cn2)c1F 24419,c1(OC)cc(CN2CCC2C(=O)NC2CC2)cc(F)c1OC(F)F 24420,c1(C(N)CNC(c2cccc(C(F)(F)F)c2)C(F)F)ccccc1Br 24421,N1(C(C(C)NC(c2nc(C)oc2C)=O)=O)CCCC12CCCOC2 24422,c1(N2CCCC(C(=O)OCC)C2)ncnc2c1ncn2CC(COC)CCCC 24423,c1(CSC2CN(C(C)=O)C2)cn(CC(C)O)nn1 24424,CC1CC(c2nnnn2CSc2ccccc2)(NCC2(CO)COC2)CS1 24425,N1(C(C2CC(C)(CC)C2)=O)CC=C(CC(=O)N2CC(F)(F)CC2CO)CC1 24426,N1(C(C(c2ccccc2F)C)=O)CCN(C(=O)CC=C(Cl)Cl)C2(CC2)C1 24427,N1(C(c2nc(C)oc2)=O)CC2(C1)CN(C(=O)C(C)OCCN(C)C)CCO2 24428,C1(C(=O)NC(CNC(c2nc(C)sc2)=O)(C)Cn2cccn2)CCC(O)CN1C 24429,Cc1nc2ccc(-c3cncnc3C(=O)NCc3ccsc3)cc2[nH]1 24430,N1(CC(N2CC(F)(C(=O)OCC)C3(C2)CCC3)=O)CCc2ccccc2C1 24431,C1(C(=O)NC(C)C(=O)Nc2cccc([N+](=O)[O-])c2)NCCC12CCCCC2 24432,Cc1csc2c(NC3CCC(N(C)C(C4CCC(CO)CC4)=O)CC3)ncnc12 24433,c1(CC)cc(F)c(C(N2CC3(CCC3NC(C3CCCN3C=O)=O)C2)=O)cc1F 24434,c1(OCCCCC)ccc(NCc2cn(C3CCOCC3)nc2C)cc1 24435,C(=O)(CC(C)(C)C(F)F)NC(C(N1CCC(NC(=O)C)C1C)=O)CCF.CO 24436,C(CC(CC)C(=O)N1CCCC(NC(C2CCC(N(C)C)CC2)=O)C1)=CC 24437,N=c1[nH]n(Cc2cn(CC3(F)CCOC3)nn2)cc1Br 24438,c1(C(N2CCC(NC(C3(COC)CC3)=O)C2)=O)c(C)nc2sc(C)nn12 24439,C1(N(C(c2c(C)scc2)=O)C)CCCC2CN(C(c3cnc(C4CC4)[nH]3)=O)CC12 24440,C1(c2ccccc2)(C(=O)NCC(C)NC(c2cc(C(=O)C(C)C)c[nH]2)=O)CCCO1 24441,c1(C(=O)NCCC2CC(NC(c3cncc(CO)c3)=O)C2)cnc2n1CCS2 24442,CC(C)C(C(=O)NCC(C)N(C)C(C1(C)CC1)=O)c1ccncc1 24443,CC1CCC(CO)CN1C(c1cc(C(C)(C)C)no1)C(=O)NCc1ccco1 24444,Cc1nc(C(=O)N(C)C)ccc1C(=O)NCCN(C)Cc1ccnn1C 24445,n1(CC)nc(C)cc1C(=O)NCc1ocnc1C(=O)NC12CC(F)(C1)C2 24446,c1(C(=O)NC2C(NC(=O)Cc3csc(Cl)c3)COC2)cnc(S)nc1 24447,Cc1ccc(CN(C2CC(c3ccccc3)C2)C)s1 24448,C1(CC(=O)NC(C(C)NC(CNS(CC)(=O)=O)=O)(C)C)COCCN1C 24449,CN=c1[nH]ccc(C(N2CCC(C)(C)C2CNC(C2CCC(C)CC2)=O)=O)c1N 24450,c1(OC)cc(C(=O)NCc2cnc(Br)s2)c(NCc2cccc(F)c2Br)cn1 24451,CCCCC(CCCC)C(=O)OC1C=CC(C(=O)OC)C1 24452,C#CC1CCCC(c2nnnn2C2CCCC2)(NC2(C)CCC(C)=C(C)C2)C1 24453,c1(C(N(CCNC(C2C(C)C2(F)F)=O)C2CC2)=O)cccc(C2CNC(=O)C2)c1 24454,c1(C(N2CCCCC(NC(c3scc(OC)c3)=O)C2)=O)cnc2nncn2c1C 24455,N1(C(C2CCCC(OC)C2)=O)CC2(CCN(C(=O)C(C)NC=O)C2)C1 24456,N1(C(CCCC(N)=O)=O)CCC2(CC1)CN(C(c1cnn(CC3CC3)c1)=O)C2 24457,c1(CC)ccc(C(=O)NCCC2CCN(C(=O)CCCC#N)C2)cc1Br 24458,C1(NC(C2(CC)CC(OC)C2)=O)CN(C(=O)CC(C)OC)CC1N=[N+]=[N-] 24459,c1(NC(c2cn(C3CCCCC3)nn2)=O)ccc2c(O)ncnc2c1 24460,C(=O)(C(C)C(F)(F)C(F)F)NC1(CCCNC(c2cc(CC)c(F)cc2)=O)CC1 24461,c1(C(N2CCC(N(C(CCC=C)=O)CCO)C2)=O)cc2n(n1)CC1(CC1)C2 24462,n1(Cc2cc(C)cc(F)c2)nc(-c2cncc(F)c2)nc1C1=NOC(C)C1 24463,CC1CN(C)CC1NC(C1CCN(C(c2ccoc2Cl)=O)C1C)=O 24464,c1(N(C)CCn2c(C3(SC)COCC3C)nnn2)ccc2nnn(C(C)(C)C)c2c1 24465,CC(C)C(C(=O)NCC(C1CCCC1)NC(c1ccc(C2CC2)s1)=O)c1cn[nH]c1 24466,CN1CC(F)CC1C(=O)N(S(C)(=O)=O)CCC1CC1 24467,CCCCC(CO)NC(=O)CC1CC(NC(=O)CN2CCNC(=O)C2)C1(C)C 24468,C1(C(=O)NCCCN(CC)CC)(CO)CCOC1.C(=O)CCC1CC1 24469,Cc1cc(Cl)c(C(=O)NCC2(C)CCCN2C(=O)CSCc2ccncc2)cn1 24470,c1(OC)cc(NC2CN(C(=O)C(=O)NC(C)(C)C)CC2C(F)(F)F)ncn1 24471,c1(C(=O)OC)[nH]c(=NCC(c2ccccc2F)NC(=O)COC(F)F)sc1C 24472,CC1CCCC(N=c2nc(N3CC4CCC3CC4)c3c([nH]2)CCC3)C1 24473,C1(COC)(NC(c2cocc2C)=O)CCN(C(=O)C(C#N)C(C)C)CC1 24474,c1(CC(=O)NC(CC(C)NC(CCOCC(C)C)=O)C)ccc(F)cn1 24475,c1(CC(=O)NCC=CCNC(C=CCCC)=O)csc(Nc2ccccn2)n1 24476,CCC(C)C(C(=O)NC(C)CC(N)=O)N(C)C(c1ccnc(NC)c1)=O 24477,C1(C(N2C(CNC(=O)CN3CSCC3=O)CCCC2)=O)CCC=CCCC1 24478,N1(C(c2cccc(CC)c2)C(=O)NC)Cc2nccn2CC(C(=O)OC)C1 24479,C(=O)(CCC(CF)CF)N1CC(CC(C(=O)NCC(F)(F)F)F)C1 24480,C1(NC(Cc2c(C)scc2)=O)CN(C(=O)C(C2CCOCC2)C)C2(CCC2)C1 24481,C(CS(=O)(=O)c1ccc(F)cc1)NC(c1nnc(-c2ccc(Cl)cc2)o1)C 24482,C1(C(=O)NC2COCC2F)(COC)CCCNCC1 24483,c1(CC(=O)NC2(C(=O)NCC)CCC2CO)ccc(OCC)cc1Cl 24484,Cc1ncc2n1CCC(C(=O)NC(C)CNC(=O)CCc1ccc(CO)cc1)C2 24485,C1(C(=O)NC(C(N2CC(CC)OCC2)=O)Cc2cnc[nH]2)CC1C1(C)COC1 24486,c1(C(C(=O)NC(C)CN(C(=O)CSC(F)F)C)C)cccc(O)c1 24487,C(C(CC(C)C)C(=O)N(C)Cc1ccncc1)NC(C(CCC)CC)=O 24488,Cc1cccc(CC(N2CCC(NC(=O)C(C)CF)C(O)C2)=O)c1F 24489,N1(C(C2(C)CCCO2)=O)CCC2(CCC2NC(c2cn3c(n2)COCC3)=O)CC1 24490,c1(CCCC(=O)NC(CNC(C2CCOC2)=O)C2CCC2)ccccc1Cl 24491,C(=O)(C1=C(F)CN(C(=O)CN2CCC(OC)C2)CC1)N1CC(CC)OCCC1 24492,C(=O)(CC(C)(C)c1ccccc1)NCC(CCOC)NC(=O)C(F)=CCCF 24493,C1(C(N2C(CC(=O)NC)CC2)=O)CC(N=[N+]=[N-])CN1C(=O)Cn1ccnc1 24494,N1(C(CC(C(C)C)NC(CC(=O)OCC)=O)=O)CCn2ccnc2C1C 24495,c1(C(=O)NCC(C2CC2)NC(CC2C(C)(C)C2)=O)cocc1Br 24496,N1(C(c2ccc(C)cc2)=O)CCC(NC(C2CCC(CO)CC2)=O)C(F)C1 24497,C=CC1(CC(=O)NCC(C2CCN(C(C3CCC(=O)O3)=O)CC2)F)CCCCC1 24498,n1(CC=C)nc(-c2cccc(Br)c2)nc1C1CCCC1O 24499,C(=O)(C(F)C(C)CNC(c1ccc(F)c(O)c1)=O)N1C(COC)C=CC1 24500,C(=O)(C(C)(C)C(=O)Nc1cc(F)cc(F)c1)NCC1(O)CCN(C(COC)=O)C1 24501,Cc1ccc(F)cc1C(N1CCCC(N(C(=O)CC2(O)CCCCCC2)C)C1)=O 24502,C(=O)(C(F)C(F)(F)F)Nc1cccc(NC(CC(SC)SC)=O)c1 24503,Cc1c(Br)cnn1CC(=O)NCCCN(C(=O)C(O)c1ccco1)C1CC1 24504,CC(C)CS(=O)(=O)CCC(=O)NCC(C)CN(C(=O)CP(C)(C)=O)C 24505,CC1(C)CC(CC(N2CC(CC(F)F)C2)=O)N(C(=O)OC(C)(C)C)C1 24506,C1(C(=O)NC(C)COCC2CCC2)CC(F)(F)CN1C(=O)CCC1CC1 24507,CCCCCC(CC)C(=O)NC1C2CCC1N(C(=O)C=Cc1cccc(Cl)c1)C2 24508,c1(NC2CCCN(C(C(CCC)(C)C)=O)CC2)ncc([N+](=O)[O-])cn1 24509,N1(C(CN(CCOC)C(C2C=CCS2)=O)=O)CC=CC12CCCCC2 24510,N1(C(c2cc(F)cc(C)c2N)=O)CCOC2(C1)CN(C(C1CN(C)C(=O)N1)=O)C2 24511,Cc1cc(CCC(N2CCOC(CN(C(=O)C(C3CC3)C3CC3)C)C2)=O)nn1C 24512,N1(CCC)CCCC(C(N2CC(N(C)C(C3(C)CC3)=O)C2)=O)C1 24513,N1(C(c2cn(CCF)nn2)C(=O)NCCOCC)Cc2ccc(F)cc2CC1C 24514,C1(C(=O)NCCN(C(C(CC=C)C(C)C)=O)C)CCOC2(CCOCC2)C1 24515,c1(C(=O)NCC2CN(C(c3cc(C)no3)=O)CC2O)c(C)ncnc1O 24516,c1(-c2c(C(=O)Nc3ccc(F)cc3O)n[nH]c2)ccc(S(=O)(=O)N2CCCC2)cc1 24517,C1(NS(CC=C)(=O)=O)CC2(C1)CN(C(c1cc(I)ccc1O)=O)C2 24518,C1(CC(=O)NCCCC(C)NC(Cc2cccc(OC)c2)=O)CCCC(C#N)C1 24519,CC1(C)CN(C(=O)CCn2ccnc2)CC(C)(C)C1NC(c1ccc[nH]1)=O 24520,C1(NC(=O)C=CCN2CCOCC2)CCN(C(=O)CCc2cn[nH]c2)CC1F 24521,C(=O)(CC(O)CC(C)C)N1C(CCC)CN(C(=O)CC(C)F)CC1 24522,c1(OC)cc(F)c(C(N2CCC3C2CCN3C(c2cccc(Cl)n2)=O)=O)cc1F 24523,C1(c2c(C)cco2)NC(=S)N(CC2(CF)CCC2)C2=C1C(=O)NC2c1ccccc1 24524,C(C(=O)N1OC2CCC1CC2)N(C(=O)C(CCCC)N(C)C)CC#C 24525,C1(NC(=O)CCc2ncc(F)cc2F)CCC2(CC1)OCc1ccccc12 24526,C(C)(CCCNC(=O)C(C)Sc1nncn1C)NC(C1(CCC=C)CC1)=O 24527,c1(NCc2c(OC)cccc2)ccc(NC(=O)NCc2cccc(F)n2)cc1F 24528,Cc1cc(O)cc(=O)n1CC(N1CC(CNC(=O)CCC(C)(F)F)C2CC12)=O 24529,C1(NC(C)=O)CN2C(C)(C1)C2.C1(C(=O)NC(C)C)(NC(=O)COC)CC1 24530,C=C=CCCC(=O)NCc1cc[nH]c1C(N1CCC(O)CC1)=O 24531,CCCC(C)CC(=O)N1CC(NC(=O)CCCc2ccccc2)C(O)C1 24532,N1(C(c2cccc(CC)c2)=O)CCN2C(=O)C(NC(=O)Cc3cncs3)CC2C1 24533,c1(CNCC2=CCN(C(CNCCC)=O)C2)ccc(=O)oc1 24534,N1(Cc2nccc(C(=O)OC)c2)CCC(NC(=O)Cn2cc(Cl)cn2)C(C)(C)C1 24535,C(=O)(C(O)C(C)CC)NCC(C1CCCC1)NC(CNS(CCCC)(=O)=O)=O 24536,N1(C(C(CC)NC(N)=O)=O)CC2CC2C1C(=O)NCc1nccn1C(C)C 24537,c1(NC(CC(C)F)=O)sc2c(c1C(=O)Nc1ccccc1)CCCC2 24538,c1(OC2(C(=O)NCC(c3cccc(F)c3)C)CC2)ccc(Cl)cc1 24539,N1(C(=O)Cc2cnc3cccnn23)CCc2c(Cl)ccc(Br)c2C1 24540,N#Cc1c(N2CCC(F)(CNC(C34CC=CCN3CCC4)=O)CC2)cccc1F 24541,c1(C(N2CCC(O)(CCNC(C(C)C)=O)C2)=O)nc(N(C)C)nc(=N)[nH]1 24542,Fc1cc(Cl)cnc1-c1nnc(N2CC3CN(CC(F)(F)F)C3C2)s1 24543,C(=O)(C(C)(CNC(=O)CCc1nc(O)n[nH]1)CC)NCC(N(OCC)C)=O 24544,C(=O)(C(C)C(C)CC)N(CC(CNC(c1nc(C(=O)NCC=C)sc1)=O)(C)C)C 24545,c1(C(=O)NCC2OCCCN(C(CCSCCC)=O)C2)cccc2nc(O)[nH]c12 24546,N1(C(CC(=O)NC)=O)CCC2(CC1)CCN(C(c1ccc(CC(C)C)cc1)=O)C2 24547,c1(C(=O)NC23CCN(C(=O)Cc4nc[nH]n4)CC2C3)ccc2ccsc2c1 24548,N1(C(CCCOC)=O)CC2CCCC(N(C(=O)CC3CCCC34CC4)C)C2C1 24549,CC#CCCCC(=O)NCCOCCCNC(=O)C(c1ccn(C)n1)C 24550,C(=O)(C(CCC(C)C)NC(c1ccnn1CCC)=O)NC(C=C)C1CCC1 24551,CCC(O)C(C)C(=O)N1CCCC1CN(C)C(C1CN(C2CCOC2)C1)=O 24552,c1(OC)ccc2nc(N3CC(CO)(NC(c4c[nH]nc4C4CC4)=O)C3)sc2c1 24553,N1(C(c2c(SC)cn(C)n2)=O)CC(C)(CNC(=O)C(F)(F)C2CC2)CC1(C)C 24554,N1(C(C2=CC(C)(C)C2)=O)CC2(C1)CN(C(c1cccc(=O)n1O)=O)CC2CO 24555,CCC(C)(CO)C(=O)NC1CC(CNC(=O)C(C(C)C)n2cnc(C)c2)C1 24556,C1(C(N2CCC(CNC(c3ccc(CO)o3)=O)C2)=O)CCC=CCCC1 24557,c1(OC)cccnc1C(=O)N(C(CNC(=O)CCSc1nnnn1C)C1CC1)C 24558,N1(C(C2CCN(C)C2=O)=O)C(CC(=O)NC(c2ccsc2)(C)C)C2CCCC12 24559,C(C(C)(O)CC)NC(C1C(=C)C1C(=O)OC)=O.N12CC(C1)C(OC)C2=O 24560,CC1CCCC1CC(=O)N(C)CCN(C(=O)CCCc1n[nH]c(=N)s1)C 24561,C(=O)(C(C)(C)C(C)(C)C)N1CCC(F)(C(N(C2CC(=C)C2)C)=O)C1 24562,Cc1ncnc(C)c1CC(N1CCC(F)C(NC(C2CCC3CC2CO3)=O)C1)=O 24563,C1(C(=O)NC(C)(C)CC(N)=O)(CC)CCN(C(c2cc(C(C)=O)on2)=O)C1 24564,N1(C(C2C(C)CCN2C(=O)CCC(N)=O)=O)CC2(CCCCCC2)C1 24565,c1(CCC)[nH]nc2ccc(C(=O)Nc3cccc(N)c3C(=O)O)cc12 24566,c1(-c2c(C)ccs2)ccc2c(c1NC(=O)Cn1cccn1)OCO2 24567,C1(NC(C(CC2CC2)OC)=O)CC2CC(C1)CN(C(=O)Cc1ccc(O)cc1)C2 24568,CC(CC(N)=O)C(=O)N1CCC(CNC(c2cccc(C3(O)COC3)c2)=O)C1 24569,CCC(F)(F)C(=O)N1CCOC(CCNC(c2cnnn2C2CCOCC2)=O)C1 24570,N1(C(C(C)n2cnnn2)=O)CCOC2(CCCN(C(c3cc(Cl)ncn3)=O)C2)C1 24571,c1(OC(C(=O)N(CCN(C(=O)CC2CC3CC3C2)C(C)C)C)C)cccnc1 24572,N12CCC(O)(CC1)CC2=O.c1(C(=O)Nc2ccc(CO)nc2)cc2ccoc2s1 24573,Cc1cccc(C(N2CC(CCNC(c3cc(C)ccn3)=O)C(C)C2)=O)c1 24574,C(=O)(C1=CC2CCCCCC12)NCCCN(c1ncnc2sccc12)C 24575,N1(C(=O)C=C2CCC2)CC(CNC(C23CCC2C3)=O)CC12CCOCC2 24576,CCC(CNCC1(C(=O)O)CC(C)C1)(CN(C)C)CC 24577,C1(C(N2CC(OC)(CNC(=O)C(C)(C)c3ccccn3)C2)=O)CC1C1CCCC1 24578,C(CCC(=O)N1CC2(CCC2(C)C)C1)(C(C)C)NC(c1cccc(CC)n1)=O 24579,c1(C(=O)NCC(CC)(CC)NC(=O)C(O)CN(C)C)nc2n(c1Cl)CCCC2 24580,N1(CC(N2CCC(CNC(C(c3ccccn3)C)=O)C2)=O)CCC(=O)CC1 24581,CC1CC(CNC(c2cnc(C3CCC3)s2)=O)CN1C(c1cncc(F)c1)=O 24582,c1(C(=O)NCCNC(C2CCN3CCCC3C2)=O)cccc2c1OCCO2 24583,c1(CN(C)C(c2ccnn2C2CCCNC2)=O)cccc2c1OC(F)(F)O2 24584,N1(C(c2c(CC)c[nH]n2)=O)CC2CCCN(C(=O)C(C)O)C2C1 24585,N1(C(CSC(=N)N)=O)CCn2ncc(C(=O)NCc3ccc4nncn4c3)c2C1 24586,C1(NC(CC2CC(NC(c3cn(C)nn3)=O)C2)=O)CC2CCCC(C1)C2 24587,c1(C(C)CNC(=O)C(=O)NCC2CC2[N+](=O)[O-])cncc(F)c1 24588,Cc1cc(C(=O)NC(c2ccccc2)C(C)NC(=O)CCc2nccs2)nc(O)n1 24589,N1(c2nc(CC)nc(C)c2)CC2(CCCC2NC(c2ccc3c[nH]nc3c2)=O)C1 24590,N1(C(C(CC)OC)=O)CCCC(F)(C(=O)Nc2cn(C)nc2C#N)C1 24591,C1(C(=O)N(CC)CC)(OCC)CCN(C(c2ccc(C)o2)C)CC1 24592,N1(C(C(C)c2ccco2)=O)CCCN(C(c2ccc(Br)s2)=O)CC1CO 24593,C1(NC(=O)C=Cc2cnc[nH]2)CC2CC(NC(=O)CCc3cscn3)CC2C1 24594,Cc1cc(C(=O)NCC2(C)CCCN(C(c3nnn(C)c3N)=O)C2)ncc1Cl 24595,C(C1CCN(C(C2CCCC(=O)N2C)=O)CC1)=CC(=O)NCc1c(CC)nccn1 24596,C1(NC(C(Cc2cc[nH]n2)NC(CCCCN(C)C)=O)=O)CCC(N=[N+]=[N-])CC1 24597,Cc1nc(-c2ccn(C)n2)sc1CC(N1CC(NC(=O)C(C)C(C)C)C1)=O 24598,C1(CC(=O)NCCC2CCN(C(C3(O)CC(F)(F)C3)=O)C2)CCCOCC1 24599,c1(C(=O)NC2CCC(NC(Cc3cc(C)on3)=O)C2)cc2c(C)cc(F)cc2[nH]1 24600,N1(CC)CCOC(C(N2CCOC(CNC(=O)CC(F)(F)Br)C2)=O)C1 24601,CCN=C(NCC(CO)C(C)(C)C)N1CCC(COc2cccc(C)c2)CC1 24602,C(=O)(CC(C(F)F)NC(c1c(O)noc1C)=O)Nc1ccc(OC)nc1 24603,Cc1oc(C)c(C(=O)NCCC(O)CNC(c2cnn(C(C)(C)C)c2C)=O)c1C 24604,Cc1ccc(F)c(CN=c2[nH]c(-c3cccc4[nH]ncc34)cs2)c1F 24605,N1(C(C2CC(N(C)C)C2)=O)CCC(NC(C2CCC(F)(F)CC2)=O)C(O)C1 24606,N1(C(CN(CCC)C)=O)CC(C(=O)NCc2ccnc(Cl)c2)C2(CCC2)C1 24607,C1(C(N(CC(C(=O)NC)C)C)=O)CCCC(NC(=O)C(C)OC)CC1 24608,C(C)(C)(CCC(=O)NCc1ccoc1)NC(C(CC)NC(N)=O)=O 24609,Cc1nccc(C(=O)NCCOC2CCN(C(C3CCC(C)NC3=O)=O)C2)c1C 24610,c1(C(=O)NCC2C(C)CN(C(c3cccc(C(N)=O)c3)=O)C2)c(F)ccnc1F 24611,N1(C(C(CC)NC(c2cnnn2C)=O)=O)CCOC(C)CC1 24612,C1(CNC(CSCC)=O)CCC(C)CN1C(c1ccnn1CC(C)C)=O 24613,C1(C(C)(C)NC(=O)C=C2CC2)CCCN(C(c2ccc(C(N)=O)cn2)=O)C1 24614,C1(NC(=O)C(O)C2CCCC2)CC2CN(C(c3occc3C3CC3)=O)CC2C1 24615,C(CC(=O)N(CCCCNC(c1csc(-c2ncc[nH]2)n1)=O)C)(C(F)(F)F)OC 24616,c1(NC(CN(C(=O)C(C)c2cccs2)CCC)=O)cscc1C 24617,C(C1=NOC2CCCC12)NC1CNCCC(O)C1 24618,Cc1ccc(C(=O)NC2CCN(C(=O)CC3(C)OCCO3)C2)cc1[N+](=O)[O-] 24619,C12(C(N(CC(C)NC(=O)C3=COCCC3)C)=O)CCOC(C)(C1)C2 24620,Cc1c(C(=O)N(C2CCN(C(=O)C(C)(C)c3cccnc3)C2)CCO)ncn1C 24621,N1(C(CC=C=C)=O)Cc2ccnn2CC(NC(=O)C(C)CCOC)C1 24622,C(=O)(C(C)(C(F)(F)F)c1ccccc1)NC1C(CNC(CC=C)=O)CCCC1 24623,N1(C(C(=C(C)C2CC2)F)=O)Cc2ccccc2C(NC(=O)CC2CCC2(F)F)C1 24624,CC(C)C(C)(C)C(=O)NCC(CC1CCCC1)C(=O)N(C1CCCN(C)C1)C 24625,c1(C(N2CC3(N(C(Cc4c(C)nc(C)s4)=O)CC3)C2)=O)ccc2oc(C)nc2c1 24626,c1(N2CCC(CC(C)C)C2)nc(=NCC2CC(C)(C)C2)[nH]c2c1ncn2C 24627,N1(C(C(C(C)C)NC(=O)OC)=O)CCCC(O)(CNC(C2SCCS2)=O)CC1 24628,C1(n2ncc(CN3CCCC3=O)c2)CCCN(C(C2(C(N(C)C)=O)CCCC2)=O)C1 24629,Cc1occc1C(=O)NC1CC(C)(NC(c2ccon2)=O)C1 24630,CC1(C)CN(C2CC2)C1c1nccn1C(c1ccccc1Cl)C1CC1 24631,C1(CCN(C(CC(C)F)=O)C)CCN(C(=O)CC2CCC23CCC3)CC1 24632,c1(NC(C2N(Cc3cnc(C)nc3Cl)C3C(C2)C3)=O)ccc(O)c([N+](=O)[O-])c1 24633,c1(C(=O)NCCC(C)NC(c2cc[nH]n2)=O)cc2c(s1)CCCNC2=O 24634,c1(C(=O)NCCC(C)NC(=O)C2=CCCS2)ccnc(SC(C)(C)C)c1 24635,c1(NC(C)C)ccc(C(=O)NCC2CCCN2C(c2ncc(Cl)n2C)=O)cc1 24636,c1(C(N2C(CNC(=O)Cc3ccc(C(=O)O)cc3)CC2)=O)cc2c(s1)CCCC2 24637,C1(F)(c2cn(CCC(C)C)nn2)CCN(C(C2CC3(CC3)CO2)=O)C1 24638,C1(C(=O)NC2(C(COC)O)CC2)C(NC(C2CN(C(C)C)C2)=O)C1(C)C 24639,N(C(=NCCC(C)=O)NCc1nc2c(s1)CCC2)C1C(CCC)CCCC1 24640,Cc1cn2c(n1)CC(C(N1CC(C)(NC(C3CC34CCOCC4)=O)C1)=O)C2 24641,C(=O)(CCCC(F)(F)CO)N1CC(NC(=O)CC23CCCN2CCC3)CC(C)C1 24642,c1(C(COC(C2(CCC=C)CC2)=O)=O)nnn(C)c1N 24643,N1(C(c2c(C)scc2)=O)CCC2(CC1)CC2NC(=O)C1=CCC1 24644,C1(C(N2CCCCC2CN(C(=O)C(C)NC(C)=O)C2CC2)=O)(COC)CCCCC1 24645,N1(C(C(=CC2CCCC2)C)=O)CC2CC1CN2C(=O)CC1NC(=O)CNC1=O 24646,Cn1cc2c(n1)CCCC2C(=O)N1CCCC(CNC(=O)Cn2cccc2)C1 24647,c1(C(=O)NC2CCCN(C(C3C(C)C3)=O)C2)ccc2c(c1)CC2 24648,c1(CC(=O)NCC2(C)CCC(NC(=O)CN3CCSCC3)C2)ccc2c(c1)CC2 24649,C1(NC(c2ccc(NC(C)=O)cc2)=O)CC2(C1)CN(C(c1ncnn1C)=O)C2 24650,C1(CC(C(=O)OCC)NC(=O)COC(C)CC)CCC(C)(C)CC1 24651,N1(C(COC)=O)CCCC2CN(C(c3ncc(C)cc3C)=O)CCC12 24652,N1(C(c2cc(OC)ns2)=O)CCCC2(CCN(C(c3ocnc3C)=O)C2)C1 24653,c1(CC)cccc(C(=O)NCCC2CCN(C(=O)CS(=O)(=O)NC)C2)c1O 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24672,N1(Cc2cn(CC(C(C)C)CO)nn2)CCC2(CC1)CN(C(=O)C1CC1)CCO2 24673,C1(C(C(=O)NCc2c(C(C)(C)C)ocn2)(C)O)CCC(F)(F)CC1 24674,CCC(CC(=O)NCC=CC(N1CCC(OC(C)C)CC1)=O)SC 24675,n1(C(C)(C)C)ncc(C(=O)NC2(CNC(=O)CC3C=CCC3)CCC2)c1N 24676,C1(CC(=O)NCCC(CCNC(CCCCSC)=O)C)CCCCCCC1 24677,c1(NC(=O)OCC)ccc(C(=O)N(C)CCNC(=O)CC2CCCN2C)cc1F 24678,c1(N)cc(C(F)(F)F)nc(Cl)n1.C1(CC(=O)N(C)CCNC2CC2)(CC)CC1 24679,N1(C(C(C)NC(N)=O)=O)CCN(C(=O)Cc2csnn2)CC12CC2 24680,c1(CC)nccnc1C(=O)NC(CNC(c1ccccn1)=O)C1CC1 24681,C(=O)(CC(CC=C)NC(=O)CC1(O)CCC1)NC1(CC=C)CC=CC1 24682,c1(C(=O)NC(C)C(=O)N(C(C)(C)CC2CC2)CCO)cc2ccccc2[nH]1 24683,C1(C(C(=O)OC)F)CCN(S(=O)(=O)CC2CCC(C(F)(F)F)O2)C1 24684,N1(C(c2c(C(C)C)noc2)=O)CCC(C)(NC(C2(n3ccnn3)CC2)=O)CC1 24685,C12(C(N3C(C)(CC#C)CC3)=O)CC(C)(CN1C(=O)CCC=CCC=C)C2 24686,CC(F)(F)CCC(=O)NN1CCCC1C(=O)NCC1(CCO)CCC1 24687,c1(NC(C(COC)NC(c2ccccc2)=O)=O)cc(O)c2ccccc2n1 24688,C1(C(=O)NC2CCC(OC)C2)CCN(C(=O)CCc2cnco2)C1C 24689,C1(C(N(CCCC)CCOC)=O)C=CCN(C(C2(OC)CCOCC2)=O)C1 24690,C1(C(=O)NCC(C)N(C2CCN(CC(F)(F)F)C2=O)C)CC(=O)N(C)C1 24691,O=[SH](Cc1c(-c2cccc(Cl)c2)ccnc1O)(CCO)c1ccccc1 24692,c1(OCC)ccc(C(=O)NC2CCC2NC(=O)CC(n2nc(C)cc2C)C)nc1 24693,CC1CCC(C(=O)NCC(=O)NCc2ncccc2F)CC1 24694,c1(C(N2C(COC)CN(C(C3CCCOC3)=O)CC2)=O)c[nH]c2ncnc(O)c12 24695,c1(C(=O)NC2CCN(C(c3cccc4nccn34)=O)C2)ccc2c(c1)COCO2 24696,C1(C(=O)NC(CN(C(CS(=O)(=O)NC)=O)C)C)CCCC(=O)N1C 24697,C12(C)COC(COC)(C1)C2.C1(N(CCC)C=O)CCN(C(C2CC2(F)F)=O)CC1 24698,Cc1c(CNC(N2CCCC2C2OCCO2)=O)cccc1S(C)(=O)=O 24699,N1(C(C#CC)=O)CCC(CCNC(=O)CC(c2ccc(C(F)(F)F)cc2)C)CC1 24700,C(C(=O)NCC1CC(C)N(C(=O)CCn2cnnn2)C1)(C(C)C)OCC 24701,Cc1ccc(C(=O)NC2(C)CCN(C(C3(C)CCN(C)C3)=O)CC2)c(C)c1 24702,c1(C(N(CCCN(C)C(c2cnn3c2OCCC3)=O)C)=O)ccn2ncccc12 24703,C(CCC(CO)NC(c1cn(C)nc1C(C)C)=O)NC(C(Cn1ccc(C)n1)C)=O 24704,c1(OC)ccccc1C(N1CC2CC1C2NC(c1cnn(C2CCC2)c1)=O)=O 24705,c1(C(N(CCCNC(C2CC3(CC3)CO2)=O)CC)=O)cc(Cl)c(N)cc1F 24706,n1(CCC(N2CC(NC(CCSCC)=O)C(O)CC2)=O)ccc2ccccc12 24707,N1(C(C(=O)N(C(C)C)CC2CCCO2)=O)CC2(CC(O)c3nccn32)C1 24708,N1(C(C(CC)N(C)C)=O)CCCCC12CN(C(=O)C(O)(C1CC1)C1CC1)C2 24709,C1(C2CCN(C)CC2)(C(=O)NC2C(OC)CN(C(C3CC(F)(CO)C3)=O)C2)CC1 24710,C(=O)(C(C)N(OC)C(=O)CCCCCN(C(=O)CSCc1nc[nH]n1)C)OC 24711,CC(C)CCN=C(NCC1COC1)NCC1CC12CCOC2 24712,CCS(=O)(=O)C=CC(=O)N1CCC(CCNC(c2cncc(N)c2)=O)C1 24713,N1(Cc2c(C)c(F)ccc2)CCC2(CCCC2C(=O)NC2CCOCC2)C1 24714,c1(C(N(CCOC)CCNC(C2CC3CCC2C3)=O)=O)cc(F)c(F)cc1Cl 24715,c1(C(=O)NCC2(CNC(C3C(OC(C)=O)C3)=O)CC23CCC3)cc(C)nnc1O 24716,N(C(=NCc1csc(C(F)(F)F)n1)NCc1ccccc1)CC1C(C)CCC1 24717,C#CC(CNC(=O)C(C1CC=CCC1)NC(=O)CNC(=O)NC)CC(C)(C)C 24718,N1(C(C(CCC)OCC)=O)CCN(C(c2ccc3nncn3c2)=O)C2CCC12 24719,N1(c2cc(C)nc(NC3CCc4c[nH]nc4C3)n2)CCCC2(CCCC2)C1 24720,c1(NC)cnncc1C(N1CCC(O)(CN(C)C(C2CC=CCC2C)=O)C1)=O 24721,c1(CC)nc(CCN2CCOCC2)nn1-c1ccn(C)n1 24722,N1(C(C2CCN(C)C2)=O)CCC12CCCN(C(c1ccnc(OCCO)c1)=O)C2 24723,N1(C(C(F)=C(C)C)=O)CC2COCCC2(NC(c2ccc(S(C)(=O)=O)[nH]2)=O)C1 24724,N1(C(c2n[nH]c(CC)c2[N+](=O)[O-])=O)CC(C2CCCN(C(=O)C#CC3CC3)C2)C1 24725,N1(C(C(C)OCC=C)=O)CCCCCC1CC(=O)NCCCSC 24726,c1(C(N2C(CN(C)C(C3CC=CCO3)=O)CCC2)=O)cc(Br)ccc1O 24727,CCC(CO)C(=O)NCC(=O)NC.C1CCCCn2cc(nn2)CN1C 24728,C(=O)(CCCCC(=O)N(C)CC1(CNC(c2cnc(N)cn2)=O)CC1)NC 24729,Cn1cc(N)c(C(N2CCCC2)=O)n1.C12CCN(C1)C(=O)N2Cc1ccc(Cl)s1 24730,S(=O)(=O)(c1ccnc(N2CCC(c3ncccn3)C2)n1)N(C)C 24731,c1(C(N2CCC(NC(C(C=C=C)C)=O)CC2)=O)cc(Br)c2ncccc2c1 24732,c1(CN(C(c2cscc2Cl)C(=O)NC2(C)CC2)CCOC)ccccc1 24733,C1(CC(=O)NCCCCC2CN(C(CCc3n(C)cnc3)=O)C2)CCC=CCC1 24734,Cc1ccc(F)c(OCC(=O)N(CC(C)NC(c2ncn3c2CCC3)=O)C)c1 24735,C1(C#N)(C(=O)NC(C(C)C)CNC(=O)CC2CC2C)CC2CC2C1 24736,n1(CC(N2CC(N(C)CC)C2)=O)cc(CNC(=O)C(C2CCOC2)OC)nn1 24737,Cc1cc(Br)cc(C(N2C3CCC2C(NC(=O)CN(C)C2CC2)C3)=O)c1N 24738,c1(C(=O)NC2C(C)CCN(C(c3cnc(C)o3)=O)C2)cc2c([nH]1)CCCC2 24739,N1(C(CSCCOC)=O)CCC2CCN(C(c3cc(C)nnc3O)=O)CC2C1 24740,c1(NC(C2CN(C(CCS(C)(=O)=O)=O)CC(F)C2)=O)ncnc2sc(Br)cc12 24741,Cc1c(C(=O)NCCOCCNC(=O)CC(C)n2ccnc2)ccn1C(C)C 24742,CCCC(C(=O)N1CC(NC(C2COCCOC2)=O)CC1CO)OC 24743,c1(OC)cc(C(=O)NC(C)CN(C(=O)C(C)CC2CCC2)C)ccc1SC 24744,CC1(C)C(CNC(C2(C(F)F)CCC2)=O)CCN1C(C1(CCF)CC1)=O 24745,c1(-n2cc(CNC(c3nccnc3Br)C)nn2)cn(C)nc1C(F)(F)F 24746,N1(C(c2c(OC)csc2)=O)CC(C)(CNC(C2CC3CCC2CC3)=O)CC1(C)C 24747,C1(C(=O)NCC(CNC(C(C)Cc2ccncc2)=O)F)C2CC3C(C2=O)C13 24748,N1(C(C(CC#C)NC(=O)CCC(F)(F)F)=O)CC(C)(C)CCC1C 24749,C1(C(N(C2CCN(C(C3C(OCC)C3C)=O)C2)CCC)=O)CC(=O)CO1.OCC 24750,Cc1ncc(N)cc1C(=O)N(C1CCCN(C(C2CC3CCC2CC3)=O)CC1)C 24751,CN1CCN(C(=O)C(C)(C)C(N)=O)CC1c1cn(C2(CO)CCOCC2)nn1 24752,c1(NCC)cccc(C(=O)NC(C)CNC(=O)CSC(C)(C)C)c1 24753,C1(NC(c2c(CC)cncc2)=O)COC2(CCN(C(c3cn(C)c(C)n3)=O)C2)C1 24754,C1(C(=O)NC(CC=C)CO)CN(C(c2ccns2)=O)CC1C(C)C 24755,C1(C(N(CCCN(C(=O)C=C2CCCC2)C)C)=O)CCC2COCCC2C1 24756,c1(C(N2CCC(NC(C(C)c3cccs3)=O)C23CC3)=O)cnc2ccnn2c1 24757,C(=O)(C1Cc2ccccc21)NCC1C(NC(CCCc2ccc(C)cc2)=O)C1 24758,N1(C(CCc2ccc(C)s2)=O)CC(C)CC1C(=O)Nc1cccc(F)n1 24759,C1(C(=O)NC(CNC(c2n(C)ncc2)=O)C(C)(C)C)CCCCN1N=O 24760,N1(C(C2CN(C(c3cc(C)ncn3)=O)CC2F)=O)CC(O)CC(O)C1 24761,c1(OC)cc(Cl)ccc1CN1CC(=O)NC(C)C1.C12(CCC1)CC(=O)N2 24762,N1(C(C(C)C2CCOC2)=O)CCOCC(NC(C2(C(=O)OC(C)(C)C)CCC2)=O)C1 24763,N1(C(CCOC)=O)CCOCC(CNC(c2cccnc2OCC(F)F)=O)C1 24764,C=CCCCC(C(=O)NOC(CO)C(C)C)NC(c1csc2nccn12)=O 24765,Cc1cc(CC(=O)NC(C)CCNC(=O)CC2CCOC(C(C)C)C2)c(C)o1 24766,c1(CN(C(CN(c2ccccc2)CC(C)C)=O)C)c(Cl)nc2sccn12 24767,N1(C(C2=CCC(NC(C(CCC)=CCC)=O)C2)=O)CC2CCCCC12C 24768,C1(C(=O)NC(C2CCCC2)CNC(C2NC(=O)OC2)=O)CCS(=O)CC1 24769,CC1(C)CC2(CN1)CC(NC(=O)C(N1CCN(c3ccncn3)CC1)=O)C2 24770,c1(C(c2cnc(C)s2)(C)CNC(=O)Nc2ncnn2C)cccc2ccccc12 24771,N1(C(c2n(CCCC)ncc2)=O)CC(NC(c2cc(O)ncn2)=O)CC(O)C1 24772,N1(C(C(c2ccnn2C)NC(c2ccc(OC)nn2)=O)=O)CCC(O)C(O)C1 24773,CC1CCc2n[nH]cc2C1C(=O)NC1CC2CCC(C1)N2CCS(C)(=O)=O 24774,c1(C(N2C(CNC(CCC)=O)COC(C)(C)C2)=O)cc2cc(Cl)cc(C)c2[nH]1 24775,n1(CC(=O)NC2C(NC(C(C)C(C)O)=O)CCCC2)ccc(=O)n(C)c1=O 24776,N1(C(C(C)CC(C)(C)C)=O)CCC2(CC1)CCN(C(C1COC(=O)N1)=O)CC2 24777,c1(C(N2CCC(CN(C(Cc3ccc(C)s3)=O)C)CC2)=O)cc2c(ncn2C)s1 24778,N1(C(c2csc(-c3ccccn3)n2)=O)CCC2C(CCCN2C(=O)C2CC2)C1 24779,N1(C(=O)NC(CCC)C(=O)OC)CC(OC)CC(C)C1 24780,CC1CCN2N=C(C(=O)N(CCCNC(C3CNC(=O)C(C)(C)C3)=O)C)NC2=N1 24781,C1(c2cc(C)no2)CCCCCN1C(=O)CC1CCN(C(=O)C2CC2)C1 24782,CCC(CC)C(C)C(=O)NCC1C2CN(C(C3CCC(C)=C(C)C3)=O)CC12 24783,c1(C(N2CCC(C)(NC(C3CC(c4ccccc4)CO3)=O)C2)=O)cnc(O)c(F)c1 24784,C1(CCOC)CCCN(C(c2ccc(NCC(N)=O)cc2)=O)C1.C1(C)CC(=O)N1 24785,N1(C(C(C2CC2)OC)=O)CCC2C(C1)NC(=O)CN2C(c1cncn1C)=O 24786,c1(-c2c(C)ccnc2)cccc2c(C(=O)NCCCO)n[nH]c12 24787,C1(C(=O)NC(C(C)NC(c2ccn(C3CCCC3)n2)=O)CO)CCOC(C)(C)C1 24788,c1(C(=O)NCC2N(C(CN(C(C)=O)C)=O)CCCC2)ncc(Cl)cc1Br 24789,C1(C(=O)NCC(C(C)C)NC(c2ccc(C(=O)OC)cc2)=O)CC(C)(C)CN1C 24790,C1(CC(N2CCC(OCC)CC2)=O)CN(C(=O)CN2CC(=O)NC2=O)CCC1C 24791,N1(C(c2ccc(C#C)cc2OC)=O)CCCC12CCCN(C(C1(F)CC1C)=O)C2 24792,O=C(CCCC(F)F)NCC12CC1CN(C(=O)Cn1cnc(Br)n1)C2 24793,C1(NC2C(C)(NC(=O)Nc3ccccn3)CCC2)CCC2(CC1)CC2C(=O)O 24794,N1(C(CCOCC#C)=O)CC=CC1CNC(=O)C(C)OCCN(C)C 24795,Cc1ccn2ncc(C(=O)NCC(C(C)C)NC(=O)CN3CC4CC4C3)c2c1 24796,N1(C(C=Cc2c(C)ncs2)=O)CCN(C(c2oc(CO)nc2C)=O)C(C)CC1C 24797,C12(C(=O)NC(C(C)C)(C)CNC(=O)C=CC(F)(F)F)CC(C)(C1)OC2C 24798,Cc1c[nH]c(=NC(=O)c2cc(C)c(OCc3ccccc3)c(Cl)c2)cn1 24799,c1(C(=O)NC2(CNC(C(C)OC3CCCCCC3)=O)CC2)ccc(P(C)(C)=O)o1 24800,c1(C(=O)OC)ccc(C(=O)NCC(C)NC(=O)CCCSC)cc1Cl 24801,c1(C(N2CC(N(C)Cc3cc(F)ccc3Cl)C2)=O)cc(F)c2cn[nH]c2c1 24802,c1(C(N(CCN(C(=O)CC2C=CS(=O)(=O)C2)C)C)=O)cccc2c1OCC2 24803,C1(C(=O)NC(N)=O)CC(F)(CNC(=O)C(C)NC)C1.c1(C(n2cnnn2)C)cc(Cl)no1 24804,c1(C(=O)NCC2N(C(C3C(C)CCC3)=O)CCOC2)nn2c(c1Br)CCC2 24805,c1(SC)nc(N2CCC(C(=O)NCc3c(F)cccc3F)C(O)C2)cc(C)n1 24806,c1(OC)cc(C(C)(C)C)cc(C(C)(C)C)c1OC1CC1(c1ccc(C)cc1)C 24807,Cc1cnncc1C(=O)NCC1C(C(=O)NCC2CN3CCC2C3)C1(C)C 24808,C1(CC)CN(c2nccc(C(C)C)n2)CCN1C(=O)CCc1cncs1 24809,C(=O)(CC(C)CCC(=O)NC1CN(C(c2ccc3oc(O)nc3c2)=O)C1)OC 24810,c1(CNC(CCSCCC)=O)ccc(CN(C)C(c2ccncc2F)=O)cc1 24811,CS(=O)c1ccccc1CC(=O)NCC1CC2(CC2)CN1C(C1CSC1)=O 24812,CC1CN(C(=O)C(F)(F)c2cscn2)CCC1N(C(=O)CSC(F)F)C 24813,c1(NC(C2C3CN(C(C(C)Cc4ccc(F)cc4)=O)CC32)=O)c(Br)ccnc1Cl 24814,Cc1n[nH]cc1CC(=O)NC(CO)C(C)NC(=O)CC(C)n1cccn1 24815,Cc1ncnc(C)c1NC(=O)CC1CC(F)CN1C(=O)Cn1cccnc1=O 24816,C1(F)(C(=O)NCC2(NC(Cc3ccc(C(N)=O)cc3)=O)CC2)CC12CCCCC2 24817,C1(C(N2CC(C(C)C)N(Cc3ns[nH]c3=O)CC2)=O)CCC(=O)C(C)C1(C)C 24818,C(=O)(CC(C)C(F)F)N1CCC(CN(C(c2ccnc(C(F)F)c2)=O)CC)CC1 24819,CCC(C)(C#N)C(=O)NCc1ccc(C(=O)NC2(CO)CC(F)(F)C2)cn1 24820,c1(C(=O)NC(CNC(=O)C(F)OC(F)(F)F)C2CC2)cc2c([nH]1)CCOC2 24821,S(=O)(=O)(c1ccc(-c2ccccc2)cc1)N1C(C(=O)NCC#CCOC)CC1 24822,Cc1cnn(C)c1CNC(=O)N(c1nnc(C(C)C)s1)C 24823,C1(NC(C2CCCCCN2C(C2CC(F)(F)C2)=O)=O)C2CCC(F)(F)C12 24824,CON=CC(=O)N1CCC(C(=O)Nc2ccc(O)c(F)c2)O1 24825,N1(c2snc(C)c2C#N)CC2C3CCC(C2C1)N(C(C1CCC(=O)NC1)=O)C3 24826,c1(C(N2CC(NC(c3ccc(S)cc3)=O)CC(C)C2)=O)ccc2c(c1)CCCC2 24827,CCCCC(O)CC(=O)NCC1CCCN1C(c1cnc(C(C)C)s1)=O 24828,N1(C(C=NOC)=O)CC(NC(C2CCNC(=O)C2)=O)CC2(CCC2)C1 24829,CCC(C)(CO)C(=O)N1C(C(=O)NCCCC2CCCCO2)CCC1C 24830,Cc1cccc(-n2nnc(OC3CC(F)CN3C(=O)OC(C)(C)C)c2CO)c1 24831,c1(N2CCC3(CN(C)C3)C2)ccc(Br)c(S(=O)(=O)NC2C(CO)CCC23CCC3)n1 24832,CC(C)C(C)(C(N)=O)NC(C1CC2CC2N1C(C1CC2C=CC1O2)=O)=O 24833,c1(N2CCC(NC(N3CCCCC3c3ncc[nH]3)=O)C2)ccc(Br)nc1 24834,c1(OC)ccccc1C(=O)NCC(=O)NC1CC(O)(C(=O)NC2CC2F)C1 24835,c1(C(=O)NC(CNC(C2C(c3n(CC)cnn3)CC2)=O)(C)C)cc(N)ccn1 24836,c1(C(N2CC(NC(CC(C)C(F)F)=O)C2)=O)ccc([N+](=O)[O-])c(Cl)c1 24837,c1(CC)nn(C)cc1C(=O)N(CC(O)CNC(=O)C(C)Cc1cccc(F)c1)C 24838,c1(C(N2C(CC)CCCC2)C(=O)NC2CCOC2)cc(=O)n2ccccc2n1 24839,C(c1ccc2cc(OC)ccc2c1)=CC(=O)NCCNC(CCC(=C)C)=O 24840,c1(C(=O)NCC2CCN(C(C(C)=C3CCCC3)=O)C2)cccn2c(C)ccc12 24841,Cc1csc(S(=O)(=O)NCC2CCCS2(=O)=O)c1 24842,C(=O)(C1CCCc2nc[nH]c21)NCC(CNC(c1nc(OCC)sn1)=O)(C)OC 24843,C1(C(=O)NCC2C(NC(c3nc(OC)c(C)s3)=O)CC2)CCc2ncnn2C1 24844,c1(OC)cc(N2CC3CN(C(c4ccco4)=O)C3C2)nc(C)n1 24845,C=CCC(CNC(=O)C=C(C1CC1)C1CC1)C(=O)NCCN1CCCC(C)C1 24846,c1(CN2C(C3CCN(C(CCC(C)C)=O)CC3)CCC2)ccc2n[nH]cc2c1 24847,N1(C(c2c(C)nn(CC(F)F)c2)=O)CC(NC(=O)C=Cc2cnc[nH]2)CC(O)C1 24848,C(=O)(C(O)C1=CCCCC1)NC1CC(CC(=O)NCc2n(C(C)C)ncc2)C1 24849,C(CNC(=O)CCCN(C)C(C)C)(C(C)(C)C)NC(CCN(C(C)=O)C)=O.CCO 24850,Cc1nn(C2CCOCC2)cc1NC(C1CCCCC1c1ccncc1)=O 24851,C(=O)(C(C#N)C(C)(C)C)NC1(c2ccc(Br)cn2)CN(C(C(C)(C)C#N)=O)C1 24852,Cc1n[nH]c(C)c1C(C)C(=O)N(CC)CC1CCCN1C(=O)CC1CCOCC1 24853,c1(N(C2C3CCC2CNC3)Cc2n(C)ccc2)nc(Cl)c(Br)cc1O 24854,N1(C(C(OC)OC)=O)CCCC(NC(c2ccc(OC)cc2C(F)(F)F)=O)CC1 24855,C(=O)(C(CSC)CC(C)C)N1C(C(=O)NC2(CC)CCCCC2)(C(C)C)CCC1 24856,C1(CNC(C(C)n2cccn2)=O)CC2CC2N1C(=O)C=CCN1CCOCC1 24857,Cc1cccnc1C(=O)NC1CC(C(=O)N(C2CC2)CC2CC2)C1(C)C 24858,c1(OC)cc(F)c(CN2CCCC(C(C)NC(c3ccc(Cl)cc3)=O)C2)c(F)c1 24859,c1(CC)cc(C(=O)NCCCCCN2CCN(C(C3(O)CC3)=O)CC2)cc(Cl)n1 24860,c1(C2(C(=O)NC3CC4CC4C3)CCCC2)ccccc1Br 24861,c1(C(=O)NC2CC(C)(CNC(CC=C)=O)C2)cccc(OC)c1 24862,Cc1ccc(C(=O)NCCc2cc(C(=O)NCCCCN(C)C)no2)c(C)c1 24863,c12cc(ccn1)N2.c1(C(C(C)n2cccn2)NC(=O)NCCOC)ccccc1 24864,C#CCC(C)(C(=O)NCc1c(OC)noc1C)NC(=O)C(CC)CCOC 24865,O=C(C1=NOCC1)NC1(C2CCCCN2C(=O)C(O)CC2CCCCC2)CC1 24866,C(CCCCCN)N(C(=O)C(N)CC1CCS(=O)(=O)C1)C 24867,C1(NC(CCN(C(C)=O)C)=O)CCCOC12CCN(C(C1C3COCC13)=O)CC2 24868,c1(C(C)C)cc(C(=O)NC2(CO)CN(C(C3(C)CNC(=O)C3)=O)C2)nn1C 24869,c1(C(=O)NC(CNC(C2CN(C)C(=O)N2)=O)CO)c(F)ccc2[nH]ccc12 24870,c12cccc(c1)NC2.c1(CNC(C2CC(F)(F)C2)C)ccccc1 24871,c1(C(=O)NCC(CC)NC(C2C3CC(=O)CC23)=O)nc(C)oc1C 24872,C(C(=O)NC(CC1CCCC1)C(=O)N(C)CC1CCN(CC)C1)(C(C)C)SCC 24873,c1(OC)ccccc1OC(C)C(=O)NCCC(C)NC(c1c[nH]c(C#N)c1)=O 24874,C1(C(=O)OCC)CCN(C(C2CN(C(c3ocnc3C3CC3)=O)CCS2)=O)CC1 24875,C#CC1(O)CC(C(N2CCC(COC)(NC(c3c[nH]nc3C(F)F)=O)C2)=O)C1 24876,C12(C(N3CC(CC)(CC)C3)=O)CCCC1CCN2C(=O)CCC1OCCO1 24877,CN1CCC(CC(=O)NC(C)(CNC(=O)CN(C2CCC2)C)C2CCC2)CC1 24878,N1(C(C2CC23CCCC3)=O)CC2CCC1C(CNc1cc(F)ncn1)C2 24879,C1(NC(c2cc(C(C)C)[nH]n2)=O)CC2CC1N(C(C1(C(F)F)CCC1)=O)C2 24880,CCC(C(=O)N1CC(CO)(NC(C2COCCN2CC2CCCC2)=O)C1)C(C)C 24881,Cc1cc(C(N2C3CC2CN(C(c2c(O)cccc2Br)=O)C3)=O)cc(Br)c1 24882,Cc1ccc2cc(C(=O)N(CCNC(=O)Cc3ccc(C)s3)C(C)C)cnc2c1 24883,c1(COC(C2(C(F)(F)F)CCC(COC)CC2)=O)ccc2c(c1F)CCC2 24884,Cc1cc(Cl)c(C(=O)NC(C)(CNC(=O)CC2(O)CCCOC2)CO)cn1 24885,c1(OC)cc(C=CC(N2CCC(NC(=O)C(F)CC3CCCC3)C2)=O)sn1 24886,c1(N(C(c2c(=N)cc[nH]c2)=O)C(c2cc(F)ncc2Br)=O)ccc2c(c1)CNC2 24887,N#Cc1ccc(Cl)c(CNC(=O)NC2CCOC23CCCC3)c1 24888,c1(COC)n[nH]c(=NC2(CNC(=O)CCc3c(N)cnn3C)CCCCC2)s1 24889,O=C(CN1C(=O)Cc2ccccc21)NC1CCCCN(C(=O)C(F)C2CC2)C1 24890,C1(NC(CCCSC)=O)CCC2CCN(C(=O)C=Cc3cncn3C)C1C2 24891,c1(C(=O)NC(c2cccc(C)c2)CNC(C2(CO)CC2)=O)ccc2scnc2c1 24892,C1(C(=O)NC(C2CN(C(c3ccc(C(F)F)o3)=O)C2)C)CCC(CC(C)(C)C)C1 24893,Cn1nc(C(N2CC(CNC(c3cnoc3C3CCC3)=O)C2)=O)cc1Cl 24894,CC1CC2(C(N3CC(SC(C)(C)C)C3)=O)CC12 24895,C1(C(=O)NC2(CC(=O)NCC(CNC(N)=O)O)CC2)CC=CCO1 24896,c1(C(=O)NC(CN(C(c2ccc(F)c(O)c2)=O)CC)C)ccc(C)cc1OC 24897,N1(C(c2ccc(C(C)C)cc2)=O)CCC(NC(=O)CC2COC(=O)C2)C1(C)C 24898,CC(CC(=O)N1CCC(N(CC(C)C)C(=O)CC2CCC(O)C2)CC1)C(F)(F)F 24899,C(CC(C(=O)NC(C)C(C)n1cccn1)NC(=O)Cc1oc(C)nc1C)OCC 24900,c1(C(N2CC(O)(C(C)NC(CCC(=C)C)=O)C2)=O)nc(Cl)ccc1Cl 24901,c1(OCC)ccc(CN(C2CCC2(F)F)Cc2ccccn2)c(C)c1 24902,N1(C(CC2CCN(C(CNC(N)=O)=O)CC2)=O)CCCC(C2CCC2)C1 24903,c1(CN2CCC(NC(C(c3ccnn3C)C)=O)C(O)C2)ccc(F)c(C#N)c1 24904,C12(C(=O)NCC3C(NC(c4cccc(OCCF)c4)=O)CC3)CCC(CC1)CO2 24905,C(C(=O)NCCCC(C)NC(=O)CCNC(c1ccco1)=O)(C(C)(C)C)SC 24906,Nc1nc(NC(=O)NCCS(=O)(=O)Nc2c(Cl)nsc2Cl)ccc1O 24907,C=CC(C)(O)CC(=O)N1CCC(C(C)(C)C(=O)N(C2CCOC2)C)C1 24908,N1(C(Cc2c(C)non2)=O)CCC(C)(CC(N2CCC(CC(=O)N(C)C)C2)=O)C1 24909,CC(O)C(C)C(=O)NC1(CNC(=O)CCCc2cccs2)CC1 24910,N1(C(CC2N(CC)C(=O)CC2)=O)C2CCC1CN(C(C1CN(S(C)(=O)=O)C1)=O)C2 24911,C(=O)(CCCCC#N)NCC1CN(C(C=CCOC)=O)C(C)C1 24912,C1(NC(C(C)(C)OCC)=O)CC2CC(C1)N(C(c1ccnc(Cl)c1N)=O)C2 24913,c1(OC)nc(Cl)ccc1C(N1CCCCC(NC(C2CCN(C)C(C)C2)=O)C1)=O 24914,C(=O)(C1=CCC(C)CC1)NC1(CF)CCN(C(C(CCC)NC(N)=O)=O)C1 24915,C(=O)(CCCC(N)=O)N1CCC(NC(CCC2CCC(C)O2)=O)CC1 24916,CCN=c1[nH]c(C(N2CC3CC(NC(c4cncc(Cl)c4)=O)C3C2)=O)cs1 24917,CCC(C)(COC)C(=O)NC1C=CCC(C(=O)NCC(C)C(C)O)C1 24918,C1(C)(C(=O)NCC(C2CCCCC2)NC(C(C(C)C)CO)=O)CC2CCC(C1)S2 24919,N1(C(C2CCN(c3ccccc3)C2)=O)CCc2sccc2C1c1ccc(Cl)cc1 24920,c1(NC2CC3CN(C(CC(CC)C4CCC4)=O)CC32)ncnc2cccc-2n1 24921,Cc1cnc(C(N2CC3CC2C3CNC(=O)CCS(C)=O)=O)c(F)c1 24922,c1(OC)ccc(C)cc1C(=O)NCCN(C(C1CCC1CNC(=O)C(C)C)=O)C 24923,c1(NCC)ccc(Cl)cc1C(N1CCC1CNC(c1cccnc1C)=O)=O 24924,N1(C(CC(CNC(=O)C(n2cc(C)cn2)C)OC)=O)CCC(C)(C)C1C 24925,c1(C(CO)NC(C#C)C)ccc(OC)c(OC(CC2(C)CCN(C(C)=O)C2)=O)c1 24926,Cc1cccc(CO)c1C(=O)NCCN(C(=O)C(F)C(C)C)CC1CC1 24927,N1(C(c2n[nH]c(C)c2C)=O)CC(C)(C(=O)NCC(c2ccccc2)O)CC1(C)C 24928,C1(C(N2CCC(C3N(C(CCC(=C)Cl)=O)CCC3)C2)=O)CCc2cnc(C)n2C1 24929,C=C=CC(C)C(=O)NC1(C(F)F)CC(NC(=O)CCCOCCOC)C1 24930,N1(C(c2ccc(C3CC3)s2)=O)CC2CCCC(N=c3ccn(CCF)[nH]3)C2C1 24931,CCC(CCCC(=O)N1CC2COCC2O1)NC(C1(C)CCCCC1C)=O 24932,N1(C(CCCOCC=C)=O)CCN(C(=O)C(CO)C2CC2)CC1c1cn[nH]c1 24933,CC1CCN(C(=O)CCc2nc[nH]n2)C1CNC(c1cc(O)ncn1)=O 24934,N1(CC(=O)N(CCC)CC2CC2)CC(c2ccccc2C)OCC1C 24935,CCCCC(C)C(C)(c1nnnn1CC1CCCO1)NCc1ccc(SC)cc1 24936,c1(C(N(C(CCNC(C=NOC)=O)C)C)=O)cccc2c(C)coc12 24937,C=CC(CCC)CC(=O)N1CC=CC1CNC(=O)COC1(C)CCCC1 24938,C1(NC(C2CC(=C)C2)=O)CC2CCC1CN(C(c1cn(C3CCOC3)cn1)=O)C2 24939,C(=O)(NNC(=O)c1cc(-c2cccn2C)[nH]n1)N(C(c1ccc(Cl)cc1)C)CCO 24940,C1(COC)(NC(=O)CCNC(N)=O)CCN(C(C2CC3(CSC3)C2)=O)C1 24941,N1(CCC2CCC(C)O2)CCN(C(C2CCCC2)C)CC1 24942,c1(C(N2CC(NC(C3(SC)CC3)=O)C(C)C2)=O)cnn2c1CCCC2 24943,C1(CC(=O)NC)CN(C(CCC2CC2)C(=O)NCCSC)CCO1 24944,c1(C(N(C2CCN(C(=O)CCc3ncco3)CC2)C)=O)ccc(F)c2c1OCC2 24945,O=C(CC1CCOc2ccccc21)NC1CN(C(=O)Cc2nccc(Br)c2)C1 24946,Cc1cc(CNC2CC2C(N2CC(O)CC2(C)C)=O)c(C)cc1O 24947,C1(C(C)C)CCCCC1CNC(N1CC(C(C)(C)S(C)(=O)=O)C1)=O 24948,CCC(CNC(=O)C(C)(C)c1ccccc1)(CC)NC(=O)CN(C1CCSC1)C 24949,C1(CC)CN(C)CCCN1C(=O)C(CC(N)=O)NC(=O)C(C(C)OC)N(C)C 24950,c1(CC)ccc2c(c1)C(CC(=O)Nc1ccsc1C)C(=O)N2 24951,c1(OCC)ccc(CN(C(=O)C(CC)n2cccn2)CCCC(=O)O)cc1 24952,C1(OC)CC(C(=O)N(C2CC3CNC2C3)Cc2cscn2)CCC1O 24953,Cc1cc(CNC(=O)C(CC2CCC2)NC(=O)C(C)C#N)no1 24954,c1(CC(N2C(CCP(C)(C)=O)CCCC2)=O)ccc(Cl)c(Br)c1 24955,CC1(CNC(c2cncc(N)n2)=O)CCCN1C(=O)CSC(=N)N 24956,C=CC1(C(=O)NCCc2ocnc2CNC(=O)C(C)SC(C)C)CCOCC1 24957,c1(C(=O)NCC(C)CNC(=O)CCCn2ccccc2=O)cc(Cl)ccc1N 24958,CCCC(C)C(=O)NC1CC(F)(C(=O)NC2(O)CN(C(=O)OC(C)(C)C)C2)C1 24959,C1(C(N)=O)CCC(C(N2CC(CCO)(CNC(c3cc(CO)[nH]n3)=O)C2)=O)CC1 24960,n1(CC)cnnc1C1CN(C(=O)NOC(C)C(=O)OCC(C)C)C1 24961,N1(CCC)CC(C(=O)NC(C)(C)C(C)NC(=O)C(c2ccc(F)cc2)=O)CC1=O 24962,C1(NC(CCNC(C)=O)=O)CC2(CCN(C(C3CC3Cl)=O)CC2)C1 24963,c1(C(C)(C)C)ccc(N)c(C(=O)NCC=CCNC(=O)C=CC2CCC2)c1 24964,C1(NCC2(C(CC)=O)CC2)CN(C(=O)C(Br)=C(C)C)CC1C1CC1 24965,N1(C(c2c(Cl)cn(C)n2)=O)CCCC2CN(c3nc4ccc(Br)cc4s3)CCC12 24966,C=CCC(CC=C)C(=O)NC(CN(C)C)C(=O)NCC(=O)NCC1CCC1 24967,C1(CNC(C=C(CC)C)=O)CN(C(c2cc(C)[nH]n2)=O)CC12CCC2 24968,C(CC(O)CCc1ccccc1)NC(CCNCCCC(=C)Br)=O 24969,c12cc(c(F)c(F)c1)NC2=O.C1(=CC(=O)NCC(CC)OC)CCSCC1 24970,N1(C(c2cc(C)n(C3CC3)n2)=O)CC(CN(C(=O)Cc2cscn2)C)C2(CC2)C1 24971,N1(C(C(COC(C)(C)C)(C)C)=O)CC2CC(NC(=O)CCC3CCOC3)C1C2 24972,c1(NC(=O)N(C2C(C(N3CCCC(O)C3)C)C2)CCCl)ccccc1O 24973,N1(C(c2cc(C)n(C)c2)=O)CC2CCN(C(c3ccnc4cc[nH]c34)=O)C2C1C 24974,C1(NC(c2cn(CCC)nc2)=O)CS(=O)(=O)CC1NC(=O)C=Cc1csc(C)n1 24975,c1(C(N2CCC(NC(c3c(CC)cno3)=O)C23CC3)=O)noc2c(F)cccc12 24976,C(=O)(C(C)(C)CN1CCOCC1)NCC(CNC(C1(n2nccn2)CC1)=O)OC 24977,Cc1ccnc2sc(C(=O)NCC=CCNC(=O)Cc3ccc(O)c(F)c3)c(C)c12 24978,CC1CN(c2nnnn2CC#CC(F)(F)F)C(C)C1C 24979,C(=O)(CCOCCCOC(C(=O)OC1(CC(=O)O)CC1)c1cnsc1)OCC.OC 24980,C12(C(=O)NCC3C(NC(CN(CC)CC)=O)CCCC3)CCCN(CC1)C2 24981,CC(C)CC(CNC(C1OCCC1C(C)C)=O)C(=O)Nc1ccccc1N=[N+]=[N-] 24982,c1(CC)oc(C(=O)NCC2CN(C(=O)CC3C=CCC3)C2)cc1C 24983,C1(NC(c2n(C)c(S)nc2)=O)CN(C(c2noc3c2CCCC3)=O)CCC1(C)C 24984,C(C(O)CC(=O)N(C1CC1)CC)NC(CCOC)=O.C(C=O)SCO 24985,CN1CCC(N=c2[nH]c(=NCC3(C)CC4(CCC4)C3)c3sccc3[nH]2)C1 24986,C(c1ccc(Cl)c(Cl)c1)=CC(=O)NC1(C)CC(NC(CC(C)N(C)C)=O)C1 24987,C1(NC(C(C2CC2)OC)=O)CCN(C(c2cn(CC(=O)N(C)C)nn2)=O)C1C1CC1 24988,C(C(c1ccccc1)NC(=O)CCF)(C(C)C)NC(c1c(OC)nsc1)=O 24989,C(C(=O)NC1(CCNC(c2cscc2Cl)=O)CC1)(C(C)O)NC(C)=O 24990,C1(NC(c2[nH]nc(C(=O)OC)n2)=O)C2CC3CN(C(c4ccccc4)=O)C1C3C2 24991,c1(NC(c2nc(-c3ccc(OC)nc3OC)c(F)cc2)=O)ncnc2c1ccn2C 24992,C(=O)(C1=Cc2cc(Br)ccc2SC1)NC1CCN(C(C)=O)CCC1(F)F 24993,c1(C(N2CCC3(C(C(=O)Nc4ncc(Br)s4)C3)CC2)=O)c(F)c(F)cc(F)c1F 24994,c1(OC)ccc(CC(=O)NCC(C)NC(C2(N(C)C)CCCOC2)=O)cc1 24995,CCC(C)(CC)NC(C1CC(CCNC(=O)CC(=O)N(C)C)C1)=O 24996,C12CCCCN(C1)C2=O.C1(C(C)(C)C)CCC(N(C)C)N1C(C12CC(F)(C1)C2)=O 24997,C1(C(=O)NC(c2ccc(OC)c(F)c2)C)CC12CCN(c1ccncn1)CC2 24998,C(=O)(C(C)CS(=O)(=O)NC1CCC(SC)C1)OC 24999,CCC(c1ccccc1)=CC(N1CCC(C)C1CNC(c1c(C)coc1C)=O)=O 25000,C1(CNC(CCN(CC#C)C(C2CC(C)CO2)=O)=O)CCCOCC1 25001,c1(-c2ccc(OC(C(CC)(C)O)=O)cc2)cc(C)c(Br)c(Cl)c1 25002,N1(C(C(C(C)C)=O)=O)CCCCC(CCC(=O)N(C(CC2CC2)CO)C)C1 25003,N1(C(=O)Cc2cccs2)CCC2(CCN(C(c3cc(Cl)c4n[nH]cc4c3)=O)C2)C1 25004,C1(C(=O)NCCCN(C(c2c(N)cccc2Cl)=O)CC)CCn2c(cnc2C)C1 25005,C(N=c1cc(C(N)=O)nc[nH]1)C1CN(C(Cc2nc(=N)[nH][nH]2)=O)C1 25006,C=CC(O)C(=O)N1CCC(n2cc(CNC(=O)C(=O)NCC(F)(F)F)nn2)C1 25007,C1(NC(c2ccsn2)=O)COCCN(C(=O)CCc2ccsc2)C1 25008,c1(CC(=O)N(CCNC(C2C(=C)CC2)=O)C)cc(F)cc(Br)c1 25009,C(=O)(C1SCc2cccnc21)NCC=CCNC(c1cc(CCC)[nH]n1)=O 25010,C(=O)(C1CCc2c(F)cccc21)NCC(c1cc(OC)ns1)=O 25011,C1(C(=O)NC2C(C(=O)NC(C(C)C)c3nc[nH]n3)OCC2)CCOC(C)C1 25012,C(=O)(C(C)(C)CNC(=O)CCCOC(C)C)NCC(C1CC1)OCC 25013,c1(C(=O)NC2(C3N(C(C=CC(CC)C)=O)CCC3)CC2)cccc(C(F)F)c1OC 25014,c1(OC)cc(I)c(C(N2C3COCC2C3)=O)cc1OC 25015,c1(CNC(=O)COCCNC(=O)CCc2cnco2)nncs1 25016,N1(C(C2OCC(C)(C)C2)=O)CCC(CNC(=O)Cn2ncc(O)nc2=O)C(O)C1 25017,N1(C(c2coc(C)n2)C(=O)NCCOCC)CCCC(C)(C)C1CO 25018,c1(N(C)C)nc(C(=O)NCC2CCCN2C(=O)CCc2nc[nH]n2)[nH]c(=N)n1 25019,C=CCC(C(=O)NCC(CCOC)NC(c1[nH]nc2ncccc12)=O)C(C)C 25020,c1(C(=O)NC2CCN(C(C3(F)C(C)C3)=O)C2)cc(O)nc2cc(F)ccc12 25021,C1(NC(CN(C(=O)CN2CCCC2C)CC)=O)COCCOC1 25022,C(C(CNC(=O)CC1CCN(C(c2nc[nH]n2)=O)C1)C(C)C)OC 25023,C1(C(=O)NC(CCCNC(COC(CC)C)=O)C)CCCC(O)C1 25024,c1(C(N2CC(O)(C(C)NC(c3ncn(C(C)C)c3)=O)C2)=O)ccc2c(c1)COC2 25025,C1(OCC)CS(=O)(=O)C2CN(C(=O)C(C)(C)Cc3ccc(Cl)cc3)CC12 25026,CC1(CCC#N)CCCN1C(C1CCC(NC(=O)CCC2CC2(F)F)C1)=O 25027,C1(COC)(CNC(=O)C=Cc2cn[nH]c2)CCN(C(=O)C(C)(CO)N(C)C)C1 25028,Cc1cc[nH]c(=N)c1C(=O)NC(CNC(=O)C(C)c1cccs1)C1CC1 25029,c1(OC)ccc([N+](=O)[O-])c(C(N2CC(F)CC2C(=O)NCC2CCOC2)=O)c1 25030,C1(C(=O)NC(C(=O)N(C)CC)C)COCCN(C(c2c(C)nn(C)c2N)=O)C1 25031,S(=O)(=O)(c1cc(C)ccc1C)N(CC(CC)CC(C)C)C1CCNCC12CC2 25032,c1(C(N2CCCCC2C2CCN(Cc3ccsn3)C2)=O)ncc(C(F)(F)F)cc1F 25033,c1(OC)cc(OC)cc(COC(N2CCN(CC(N3CCCCC3)C)CC2)=O)c1 25034,c1(C(=O)NC(CNC(C(C(C)C)(C)O)=O)CO)coc(S(N)(=O)=O)c1 25035,CCCCC(CC)C(=O)N1CCCC(NC(c2ccc(OC)nc2C)=O)CC1 25036,C1(OCC)CN(C(=O)C(=Cc2c[nH]cn2)F)CC1CNC(c1cn(C)nc1Cl)=O 25037,c1(C(N2CCCC(NC(C3CC3(F)F)=O)C2)=O)c(OC(F)F)cccc1Br 25038,c1(C(N2CC(NC(c3scc(OC)c3)=O)C2)=O)n[nH]c2ccccc12 25039,Cc1cc(C(=O)NCC2CCCC2C(N2CCCC(C#N)C2)=O)cc(O)n1 25040,c1(C(N2CCCC2)=O)ccc2c(c1)CCN(Cc1cccc3c1CCCC3)C2 25041,CC(C)(C)C(C(=O)N1CCC(NC(=O)CC2CCC3CC23)CC1)N1CCOC1=O 25042,Cc1cccn(CC(N2C3CCC2(C2C(CNC(=O)C(O)C(C)C)C2)CC3)=O)c1=O 25043,N1(C(C(CCC)=CCC)=O)CCC2CC(C1)CN(C(=O)CCc1cnoc1)C2 25044,c1(OC(=O)NC(c2nnnn2C2CCOC2)CC#N)ccc2ccccc2c1 25045,c1(SC)cc(NC(=O)CN2CCSC(c3ccccc3)CC2)ccc1OC 25046,N1(C(C(C2CCN(C(CCCOCCC)=O)C2)C)=O)CCCC2C(O)CC12 25047,N1(C(C(N2CC(C)C(NC(=O)C(F)(F)F)CC2)=O)=O)CC(C)(C)C(F)(F)C1 25048,c1(C(=O)NC(C2CC2C(N2CC(O)CC(O)C2)=O)C)ccc(C#N)c(C)c1 25049,C1(NC(C(C)C(F)F)=O)CC2CCCC(C1)C2NC(=O)Cn1ccc(O)nc1=O 25050,C(CCCC(C)(C)C(=O)NNC(=O)c1ccco1)NC(c1cc(C)cc(C)c1)=O 25051,Cc1nc(=N)[nH]c(C)c1C(N1CC(NC(c2ccc(C(C)C)cn2)=O)C(C)C1)=O 25052,c1(C(N2C3(CNC(C(COCC)C)=O)CC(C2)C3)=O)cccc(C)c1C 25053,C(=O)(CC(C)C(F)(F)F)N1C(C(N2C(COC)COCC2)=O)CC2CC21 25054,C1(F)(C(=O)NCc2ccc(C)s2)CCN(C(C2CNC(=O)N2)=O)C1 25055,N1(C(C2CCCC(C(N)=O)C2)=O)CCCC(C)(CNC(c2ccc(CO)o2)=O)C1 25056,N1(C(CN(CC)CC)=O)CCCCC(N=c2ccc(C(F)(F)F)n[nH]2)C1 25057,NS(=O)(=O)CC(=O)NC1CN(C(C2CC(Cc3ccc(F)cc3)C2)=O)CC1O 25058,c1(C(=O)NCC2N(C(c3cc(C)[nH]c3C)=O)CC=C2)cn(C)c(=O)nc1O 25059,N1(C(c2ccc([N+](=O)[O-])[nH]2)=O)CC(C2CCCN(C(=O)C3=CCCC3)C2)C1 25060,Cc1ccc(C)c(C(C)N(C)C(c2cc(-c3ccccc3)[nH]n2)=O)c1 25061,c1(C(=O)NCC(C(C)C)NC(C2CCc3c[nH]nc3C2)=O)cncc2ccsc12 25062,C1(NC(c2cnn(-c3ccncc3)c2)=O)CN(C(=O)C=CBr)C2(CCC2)C1 25063,C(=O)(CC(C)(C)CC(=O)NCC1(C2CC2)CCN(C(=O)Cc2ccsc2)C1)OC 25064,C(=O)(C1CCCc2ncc(C)n21)NC(CC)CNC(c1cn(C2CC2)cn1)=O 25065,C(=O)(CC(F)(F)CC(=O)NC(C)CN(C(=O)COCC1CCCOC1)C)OC 25066,N1(C(C(C=C)OC)=O)CCCC(CC(=O)NCC(C)CN(C)C)C1 25067,C(=O)(C1CCCCc2ccccc21)N1CC(O)(C(C)NC(CCCOC)=O)C1 25068,c1(CC)cc(C(=O)N(C2CCN(C(c3cnn(C4CC4)c3C)=O)C2)C)cc(O)n1 25069,NS(=O)(=O)CC(=O)NCCCN1CCC(NC(=O)CC(F)(F)F)C1 25070,c1(C(=O)NC(CC)CNC(=O)Cn2cnnc2)ccc2nc(CO)[nH]c2c1 25071,c1(CC)[nH]nc(C(=O)NC(CCC2CCC2)C(=O)NC(c2cnc(C)s2)C)c1C 25072,N1(C(C2(COC)CC=CC2)=O)CC2OCC(C(=O)N(C)CC#N)C2C1 25073,CC(c1cccnc1)=CC(=O)NCC1CC2CCC1N2C(=O)Cc1ccco1 25074,c1(C(=O)NCCN(C(=O)C(=O)NOC)CCC)ccnc(OC(C)(C)C)c1 25075,c1(C(=O)NCC2C(CNC(Cc3c(C)ocn3)=O)C2)cc(O)cc(Br)c1 25076,CC(CC(=O)NCC1C(C(=O)Nc2cccnc2)C1(C)C)C(F)F 25077,CCCC(CC1CCCC1)C(=O)NCC1CCN(CC(O)COC)CC1 25078,c1(OC)cc(F)c(F)cc1C(N1CCC(C)(C(=O)O)CC1)=O 25079,c1(OC)ccc(C(=O)N(C)CCNC(=O)C(C)S(N)(=O)=O)cc1S(=O)(=O)NC1CC1 25080,C(=O)(C(C(C)(C)C)NC(=O)CO)NCC1(NC(CCC(C)OC)=O)CCC1 25081,C(=O)(C(C)(C)C(O)CC)N1C2C(NC(c3cccc(CC=C)c3)=O)CC(C2)C1 25082,c1(C(N(CCNC(c2cc3ccccn3n2)=O)CC)=O)ccc([N+](=O)[O-])cc1Cl 25083,C1(C(=O)NC2(CCO)CN(C(CC3(NC(C)=O)CC3)=O)C2)CCOCC12CCC2 25084,CCCC(C(=O)NC1CCCN(C(c2ccc(F)c(C(F)F)c2)=O)C1C)C(C)C 25085,Cc1nn(CC(F)F)c(C)c1C(=O)N(CC(C)(C)N(C)C)CCCC1CC12CC2 25086,CC1CCC(NC(c2ccc(C#N)n2C)=O)CN1C(c1cnc(C(F)(F)F)s1)=O 25087,C1(CNC(c2c(C)coc2C)=O)CC2(CCN(C(C3(O)CC(C)(C)C3)=O)CC2)C1 25088,N1(C(CCC(=C)C)=O)CCCC(CO)(NC(=O)CCSc2ccc(C#N)cc2)C1 25089,c1(OC)ccnc(C(N2CC(CC(F)C(N3CCCC34CC4)=O)C2)=O)c1 25090,CC1(C)C(C(N2CC(CNC(=O)C(c3ccccc3)O)C2)=O)CCS1(=O)=O 25091,c1(C(C2(OC)CCOC2)NC(CCC)C2CCCC2)nnnn1CCC1CC1 25092,CC1CN(C(C2CCC(F)(F)CC2)=O)CC(C)CN1C(=O)Cc1cnccc1Cl 25093,C1(NC(=O)CNC(C2CCCC2)=O)CC2CN(C(C(CC)NC(C)=O)=O)CC2C1 25094,c1(OCC(N2CCCC(c3cn(-c4ncc(C)s4)nn3)C2)=O)cc(C)cc(Cl)c1 25095,C1=C(C(c2nnnn2CC2CCC2)NC2(C(=O)N)CC2)CCCC1.C1CCCO1 25096,C1(C(=O)NC(C2CCN(C(CC(C)C)=O)C2)C)Cc2ccccc2N1C 25097,c1(OCC)ccc(C2(C(=O)NCC3C=CCN3C(=O)CCCOC)CCC2)cc1 25098,c1(C(=O)NC(C2CCCN2C(=O)Cc2ccc(Cl)s2)C)csc(-c2nc[nH]n2)n1 25099,c1(-c2ccc(CN(C(CCC)C)Cc3ccncc3)s2)c(F)cccc1Cl 25100,c1(OC)cnc(F)c(C(=O)N(C(C)CN(C)C(c2cncc(COC)c2)=O)C)c1 25101,S(=O)(=O)(c1cnn(C)c1)N1C(C(=O)NC(C(=O)OC)C(C)O)CC2CC21 25102,CCC(C)CC(=O)C(=O)NC(C)(C)C(=O)NC(C1CSC1)C 25103,CC1(C)CCCOC1CC(=O)NC1(C)CN(C(=O)C(c2ccccc2F)O)C1 25104,N12CCCCC(C1)N(C(C1CC(OC)C1)=O)C(=O)C2.N1(CC)CCN(C)CC1 25105,C12(C(N3CCC(=CCNC(=O)CN4CCCC4)CC3)=O)CCN(C1)S(=O)(=O)C2 25106,C1(CCNC(CCCOCCOC)=O)CCCN(C(=O)Cn2cnnc2)CC1 25107,CC(C(=O)N1CCC(N(C)C(C2CCCN2CC(F)(F)F)=O)CC1)C(F)(F)F 25108,N1(C(CCOCC#C)=O)CC2CCC1C1CN(C(c3ccnc(CO)c3)=O)CC21 25109,CCCCCCCC(=O)NC1C(C)CCN(C(=O)COc2ccc(O)cc2)C1C 25110,CC1CCN(C(=O)C(=C2CCCCC2)F)CCN1C(=O)COc1ccon1 25111,c1(C(N2CCC(C(=O)OC)(CO)C2)C(=O)NC2(C)CC2)cc(C)c2c(c1)CCC2 25112,c1(OCC)ccc(C2(CNC(c3n(CC)nnn3)c3ccon3)CC2)cc1 25113,N1(C(CN(C(=O)CCC2CC(C)C2)CC)=O)CC(CO)OCC1C 25114,C1(CNC(CC=C(C)C)=O)CN(C(=O)CC2CCCCCC2)CC12CCC2 25115,C(=O)(CC(C)CC(C)(C)C)NCC1=CCN(C(C(c2cccc(C)c2)O)=O)CC1 25116,N1(C(C(C)OCCC=C)=O)CCCC1C=CC(=O)NCc1ccc(C)cc1 25117,Cc1noc(C(F)F)c1C(=O)NCCNC(=O)C(C)Cc1ccccc1F 25118,N1(C(CC(C)NC(C(C)O)=O)=O)CCCC(C(C)C)CC1 25119,c1(NC(CCOCCNC(C(COC)OC)=O)=O)ccncc1F 25120,N1(C(C(C)n2cnnn2)=O)CC2CCCC(C1)N2C(c1cnc(F)c(F)c1)=O 25121,c1(CC)n[nH]c(CC)c1CC(N1CCC(N(C(=O)C(C)CN(C)C)CC)CC1)=O 25122,c1(CC(C)C(=O)NC2CCN(c3ccnc(C(F)(F)F)n3)CC2)ccc(Cl)cc1 25123,C1(=CC(=O)NCC(C)(C)CNC(C23CSCC2C3(F)F)=O)CN2CCC1CC2 25124,CC1CCN(C(C2(O)CC2)=O)CC1NC(c1coc(-c2ccccc2)n1)=O 25125,C#CCCC(O)C(=O)NCC(c1ccccc1)N(C(=O)Cc1sc(C)nc1C)C 25126,Cc1scc(CNC(=O)C(C2(O)CN(C(c3ccn(C)c3)=O)C2)F)c1C 25127,c1(OC)ncc(NC(=O)CNCC2CCN2C(=O)C(C)CC(C)C)c(C)n1 25128,O=S(=O)(c1cnn2ccc(=NCCN3CCCOCC3)[nH]c12)NC1(CO)CCC1 25129,C(=O)(N=c1[nH]nc(CC2CC2)s1)NCCOC(CNC(C)=O)(C)C 25130,c1(CNC(c2nc(C)oc2C)=O)cc2n(n1)CCN(C(=O)C(F)(F)C1CC1)C2 25131,CCCC(C(=O)N1CC(O)(CCNC(=O)C(=O)N=S(C)(C)=O)C1)S(N)(=O)=O 25132,CC(CC(F)(F)F)C(=O)NCc1occc1C(N1CCC(C)(N(C)C)C1)=O 25133,CC1CC(C(N2CC(CCNC(c3ccc(=N)[nH]c3)=O)C2)=O)CC(C)C1 25134,CCC(CCCC(=O)N(C)CC1(CC)CC1)NC(=O)CCC(=O)NCC 25135,N1(C(C2C(CNC(C(C)=O)=O)CC2)=O)CCCC1CCC(C)C 25136,N1(C(c2c(C)n[nH]c2)=O)C2CCCC1CC(NC(=O)CC1CCC3CC3C1)C2 25137,Cc1[nH]nc2cc(C(N3CC4CC3CN4C(C3CC(=O)N(OC)C3)=O)=O)ccc12 25138,C1(C2CC2)(OC)CN(C(=O)CC2CN(C(=O)CCCF)C(C)(C)C2)C1 25139,CC1CCN(CC2CCN(C(=O)OC(C)(C)C)C(C)C2)CC1C 25140,C1(C)(C(=O)NC2C(CNC(C)=O)CC(C)(C)CC2)CC(F)(F)C1(F)F 25141,C=CC(C)(C)CC(=O)N1C(C)CCCC1C.C1C(=O)N1 25142,N1(C(c2ncc(NC)nc2)=O)CC2CCCC2C1C(=O)NCCN1CC=CC1 25143,C1(CC(=O)NC2CN(C(c3ccc(C)o3)=O)C2)COCCOC1 25144,C(=O)(C(C)CC(N)=O)N1CCC(CC=C)(C(=O)NCCCc2nccs2)C1 25145,c1(CNC(CSC)=O)ccc(CC(C)NC(C2(C)CS(=O)(=O)C2)=O)cc1 25146,C(N=c1[nH]c(=NC2CCSC2C)[nH]c2cc[nH]c12)c1ncn(C(C)C)n1 25147,C(CC(C)N=c1[nH]c(=N)[nH]c(=NC(C)c2cc(Br)n(C)n2)[nH]1)SCC 25148,Cn1c(C(N2CC3CCN(C(=O)COCC4CC4)C3C2)=O)cnc1[N+](=O)[O-] 25149,N#Cc1cc(NCCc2cccc(F)n2)cc([N+](=O)[O-])c1Cl 25150,Cc1nc(C(=O)NCC(O)CNC(=O)C(C)(C)C(N)=O)ccc1[N+](=O)[O-] 25151,N1(C(CC(C)c2ccncc2)=O)CCSCC1C 25152,Cn1ncc2ncc(C(N3CC4CCC3CN4C(c3cc[nH]c(=N)c3)=O)=O)cc12 25153,c1(C(N2CC(=C(CNC(C(C)Cc3ccco3)=O)F)C2)=O)cccc(Cl)c1Cl 25154,C(=O)(CCCCN(C)C(c1cnnn1C)=O)N(CCN=[N+]=[N-])C 25155,Cc1cc(O)cc(C)c1CS(=O)(=O)NC1CCN(CC2CC2)CC1.c1(O)cnccn1 25156,C1(C(N(CCNC(C(C=C)OC)=O)C(C)C)=O)CN(C)CC(C)O1 25157,C(=O)(C(CCCC#N)N(CC(F)Br)C)OCCCc1ccc(OC)c(OC)c1 25158,Cn1ncc(Cl)c1C(=O)NCCC1CCCN1C(C1CN(C2CCOCC2)C1)=O 25159,C1(C)(CC)CCN(C(C2CCCC2NC(=O)CC(C)N(C)C)=O)CC1 25160,N1(C(CC2CC(OC)C2)=O)CC2(COC(CNC(=O)C(O)c3ccsc3)C2)C1 25161,C(CC(C(=O)NC1(SC)CCC1)OC)NC(=O)CC1C(N(C)C)CC1O 25162,CC1CC(CC(=O)NCCN2CCCC2)CN1C(c1ccc(=N)[nH]n1)=O 25163,C(CC(=O)N1CC(c2ncc[nH]2)C1)(C(F)F)NC(C(C1CCOCC1)C)=O 25164,C1(C2CCN(Cc3ncc(C)s3)CC2)(NC(C(C(CC)C)OC)=O)CC1 25165,C(C)(C(=O)N1CC(C(C)NC(c2coc(C(F)F)n2)=O)C1)(C(C)C)OC 25166,C(=O)(C(C(C)(C)C)N1CCCC1)NC(C(C)C)(C)CNC(=O)Cn1ccnn1 25167,C(C(CC(=O)N(C1CCOCC1OC)C)NC(c1cncc(CO)c1)=O)OC 25168,CC(=O)CCC(=O)NC(Cn1ccnn1)C(N1CCC(F)(CF)C1)=O 25169,c1(C(=O)OCC)ccc(=NCCCNCCCN2CCC2)[nH]c1.C 25170,c1(C(C(N2CCN(CC)C(C)C2)=O)=O)cc(OC)c(OC)c(C)c1OC 25171,C1(C(=O)NC(C2C(C(=O)NC3CC(OC)C3)C2)C)CC(C)(O)C1 25172,CON(CCO)C(=O)CC(C(F)F)NC(=O)C(C1CCOCC1)F 25173,C1(C(=O)NCC(CNC(C(N2CCC(O)CC2)C)=O)O)CCCCC1(F)F 25174,c1(C(=O)NCC#CCNC(c2c(C(C)C)n(C)nc2)=O)cc(Cl)c(Cl)cc1O 25175,C(c1ccccc1)=CC(=O)NCC(=O)NC(C(C)NC(C(C=C)O)=O)(C)C 25176,CC1(CNC(=O)C=Cc2cnc[nH]2)CCN(C(c2ncc(Cl)cc2Cl)=O)CC1 25177,C1(CC(=O)NCC2(CO)CCC2)CC2CCC1N2C(c1cnc2n1CCC2)=O 25178,C1(NCc2cn(C)nc2C2CCCC2)CC(O)C12CC(F)(F)C2 25179,Cc1ncccc1C(=O)NCC(C)(C)C(=O)NCC1(n2nccn2)CC1 25180,c1(CC(=O)NC(C2CCN(C(=O)CC3CCC3(F)F)C2)(C)C)c(F)cccc1F 25181,c1(CC(N2CC(NC(CC(CCC)O)=O)C3(C2)CC3)=O)c[nH]c2cccc(Cl)c12 25182,N1(C(c2ccsc2Cl)=O)CCC2C(C1)CN2C(c1cnnc(O)c1)=O 25183,c1(CC)ccc(C(N2CCC(CCNC(c3cn(CC)nn3)=O)C2)=O)c(O)c1 25184,CCC(CC)CCC(=O)NC1C2CC(NC(=O)C(C)CC(N)=O)CC12 25185,C(=O)(CN=S(C)(C)=O)NC(c1cnn(C)c1)C(N1CC(CN(C)C(=O)C2CC2)C1)=O 25186,c1(CN2CC3N(C(c4c(OC)cncc4)=O)C3C2)c(C)cc(C)cc1C 25187,c1(COC)cc(C(=O)NC(C)(CNC(=O)Cc2nccn2C)C2CC2)no1 25188,O=C1COc2cccc(C(=O)NOC3CC(O)C3O)c2N1 25189,c1(C(=O)NCC2N(C(C(n3ccc(C)n3)C)=O)CCC2)ccc(C)cc1[N+](=O)[O-] 25190,c1(C(=O)NC2(C(=O)NC(CCC=C)C)CC2(C)C)cc(O)n(CC)n1 25191,C1(C(=O)NCC(C)CNC(=O)CNC(c2ccco2)=O)(CC)CCCCO1 25192,N1(C(CCc2cc(C)[nH]n2)=O)CC2(CCN(C(c3cc(F)ccc3Cl)=O)C2)C1 25193,C1(C(C)NC(=O)C(C)N2CC(C)C2)CCCN1C(=O)CCCN1CCOCC1 25194,N1(C(C(C)(C)n2cccn2)=O)CCC2(CCC2)CC1 25195,C#Cc1cccc(NC(=O)CC(C)CNC(=O)CCSCC(F)F)c1 25196,C1(NC(CN2C(=O)CN(C)C2=O)=O)CCC2(CC1)CC2Nc1ncncc1Cl 25197,C(=O)(C(CC(C)C)C(N)=O)NC(CCNC(c1ccc(CC)cc1F)=O)(C)C 25198,c1(CCC)cc(NC(=O)Nc2ccc(-c3cc(OC)ccn3)s2)n(C)n1 25199,C1(CCC(=O)NCc2ccc(Br)cc2)CCCCN1C(=O)CCc1ccncc1 25200,N12CCC(O)CC1C(=O)NCC2=O.C1(NC(CN(C)C)=O)CC(OC)C1.C1(C)CC1 25201,C1(NC(C(CC)N(CC)CC)=O)CC2(C1)CC2C(=O)Nc1cnn(C)c1SC 25202,CC1(C)CCCC(O)(C(=O)NC2CN(C(c3nocc3Cl)=O)C3(CCC3)C2)C1 25203,C(C)(CCC(=O)NC(c1ncccn1)C)NC(CCCOC)=O 25204,N1(c2n(CCOC)c(C3(OC)CCSC3)nn2)CCCC(O)(COC)C1 25205,CC1CCN(C(C2CCCC2)=O)C1c1cn(-c2cccc(OCCO)c2)nn1 25206,C1(O)(CNC(c2c(C)snn2)=O)CCN(C(c2cccc(Cl)c2)=O)CC1 25207,C(N=c1nc2sccc2c(NCc2cc(C3CC3)on2)[nH]1)c1n(C)nnc1 25208,CCC(CC)C(C)C(=O)N1CC(NC(c2ccc(N)c(SCC)c2)=O)C(C)C1 25209,C1(C(=O)NCCOC2CCN(C(=O)C(F)n3ccnc3)C2)CC2(C1)CC21CC1 25210,Nc1cc(C(=O)NCC2CCN(C(=O)Cc3cc(C(F)F)cc(F)c3)C2)cc(N)c1 25211,n12c3c(cc(cc3)c1=O)C1(C2)CCCC1.O=C(N=c1nc[nH]s1)C1CCCO1 25212,C1(C)(CC(=O)NC23CCC(CC2)N3Cc2n(C)c(S)nn2)CCS(=O)(=O)N1 25213,C#Cc1cnn(C)c1C(N1CC(C)(NC(=O)CC2CC(O)C2(C)C)C1)=O 25214,n1(CC(=O)NC2CCC(F)(CNC(C=CCCC)=O)C2)cnc2ccccc12 25215,C1(C)(C(N(C)CC2CN(C(=O)CN3CCCC3)CCO2)=O)Cc2ccccc2N1 25216,C12(CNC(C(C)CF)=O)CCCC1N(C(C1COc3ccccc3O1)=O)CCC2 25217,C1(C(N(CC(=O)NCCNC(C)=O)CCC)=O)CC12CCC2 25218,c1(CNc2cn(C(C)(C)C)nn2)scnc1C1=CCN(c2ccc(Cl)cc2)CC1 25219,N1(C(c2cnc(CC)s2)=O)C2CCC1CC(N(C)C(c1cc(C)ncc1C)=O)C2 25220,CCC(CNC(c1ccc(C2(O)COC2)cc1)=O)(CC)NC(=O)C=CC(C)(C)C 25221,N1(C(CCNC(=O)OC)=O)CC2(CCC(NC(=O)C(C)C(O)CC(C)C)CC2)C1 25222,Cc1nn(C)c(N)c1C(N1CCC(OCC(=O)NC(C)C(O)C(C)C)C1)=O 25223,C(=O)(CC(C)(C)C(C)(F)F)N(CC(C)NC(c1ccc(NC(N)=O)cc1)=O)CC 25224,c1(C(=O)NC(C(C)(C)NC(C=CCCC)=O)C)ccc(C2(CC)CC2(F)F)cc1 25225,CCCC(CC(C)C)C(=O)N1C(C(=O)NCCC(=O)OC(C)C)C2CC(O)C1C2 25226,C1(CNC(=O)Cc2cnc[nH]2)CN(C(=O)C(N)=O)CC1O 25227,N1(CC)CC(NC(C2(F)CCN(C(c3nc(Cl)cs3)=O)C2)=O)CCC1=O 25228,CCCCC(O)C(=O)NC1(CCNC(c2[nH]ccc2C2CC2)=O)CCCC1 25229,Cn1cc(-c2cnn3cccnc23)cc(C(N2CCC(CCCO)CC2)=O)c1=O 25230,S(=O)(=O)(c1c[nH]ccc1=NC1COCC(C)(C)C1)N(C(C(CC)C)C)CC 25231,C1(NC(c2n(CC=C)nnn2)c2cc(C)on2)CCn2nnnc2C1 25232,C1(C(=O)NC2CC(NC(C34CCC(CC3)CC4)=O)C2)CCCC2(CCCCC2)C1 25233,c1(C(N2CCC(NC(COCC#C)=O)C(O)C2)=O)cc(C)c2[nH]nnc2c1 25234,CC1CC(C(=O)NCCC2CC(NC(=O)C3=CCCCO3)C2)CC(C)C1 25235,C1(=C(CO)NC(=O)CC2CCOCC2)CCN(C(=O)CCCOC(C)(C)C)CC1 25236,c1(C(C)(C)C)[nH]cnc1C(=O)NCC(C1CC1)NC(c1cn(CC(F)F)cn1)=O 25237,CC(C)C(C)(CNC(C1SCCS1)=O)NC(=O)Cc1csc(-c2ccoc2)n1 25238,c1(C(=O)NCCCNC(C(C)OCCC#C)=O)cc2cnn(C)c2s1 25239,C1(NC(C2CC23CCC3)=O)CCC(O)CN(C(c2ccc(-c3csnn3)cc2)=O)C1 25240,N1(C(C=CC(C)(C)SC)=O)CC2CCC1CC2NC(=O)CC(O)CN(C)C 25241,C1(N(C(c2cc(C)oc2)=O)C)CCCN(C(C)C(=O)N)C1C.N1(C(C2CC2)=O)CCCC1 25242,c1(NCCCCN(CC(=O)NCCc2cscn2)CC)cccc(C(C)(C)C)c1 25243,c1(C(N(CCNC(c2ccc(Br)o2)=O)CC)=O)ccncc1Br 25244,C1(CC(=O)NC(CNC(=O)CCCNS(C)(=O)=O)C(C)C)(C(=O)OC)CCN(C)CC1 25245,c1(CCC)cc(C(=O)NC2CN(C(=O)CCC(=O)OCC)CC2C)ccn1 25246,C1(CC(=O)NCC2C(NC(CN(C)CCO)=O)CCC2)CCC(F)(F)CC1 25247,N12CCC(CC1)C(=O)NCC2=O.C(=O)(C(F)(F)F)NC1(c2cccnc2)C(C)(C)C1 25248,C1(C2CC2)(C(=O)NC(C#C)C(C)(C)C)CN(C(C2CC(=O)CC(=O)N2)=O)C1 25249,Cn1ncnc1CNC(c1occc1Br)c1nnnn1C1CC1 25250,c1(SC)c(NC(=O)N(CC(F)(F)F)C(c2ccc(OC(F)F)cc2)C)cnn1C 25251,c1(C(=O)NC2CC(N(C(C34CC(C(C)C)(C3)C4)=O)C)C2)cn(C)[nH]c1=N 25252,C1(NC(c2ccn(C)c2)=O)CC(NC(c2nnc(S)n2C)=O)C12CCC2 25253,N1(CC)CC2CC1CN2C(=O)C=CC(C)NC(C1(C(C)C)CC1)=O 25254,C1(NC(CCCC#CC)=O)COC2(C1)CN(C(=O)C(c1ccc(Br)cc1)C)C2 25255,C(C)(CSC)(C(=O)NOCCCC(=O)OC)NC(c1cccc(CC)n1)=O 25256,Cn1ccc2cccc(C(=O)NC3(C)CCN(C4CCNC4=O)C3)c12 25257,C(CCN(C(=O)CC1CC2(CC2)C1)C)(C(C)(C)C)NC(c1c(C)cno1)=O 25258,C(=O)(CCCCCCNC(c1coc(CO)c1)=O)NCC(c1c(C)ncnc1)=O 25259,CCCCC(C)CCC(=O)NC(COCC)C(=O)N(C1CC=CC1)C 25260,N1(C(C2N(CC)CCC2)=O)CC(C)(C)C(NC(C2CCOCC2)=O)C(C)(C)C1 25261,N1(C(C(C)NC(C2CC(CC)(CC)C2)=O)=O)CCC2(CC1)CC2CCCC1CC1 25262,c1(-n2cc(C3CCCN(C(C(CC=C)C)=O)C3)nn2)ccc(Cl)nc1C(F)(F)F 25263,c1(C(N(CCNC(C=C(CC)C)=O)CCOC)=O)cccc(F)c1Br 25264,C1(C(=O)OC)(CC)CCN1C(C1CC(C)N1C(=O)OC(C)(C)C)=O 25265,CCC(O)C(F)(F)C(=O)NCC(C1CCN(C(c2ccncc2F)=O)CC1)C 25266,C1(CC)C(C(=O)NC2CCN(C(=O)Cn3nc(C)oc3=O)C2C)CCN1C 25267,C(=O)(C(C)C(O)C(C)C)NC(C(=O)NCC(COC(C)=O)C)(C)C 25268,N1(C(C2(CO)CC2c2cccs2)=O)CCC(c2nc(-c3ccccc3)no2)CC1 25269,c1(C(=O)NCC(C)NC(C2(F)CCOC2)=O)nc(Br)c2c(F)cccn12 25270,N1(C(CCc2ccc(C)o2)=O)CCCC2CN(C(=O)C(C)(C)C(C)(C)O)CCC12 25271,S(=O)(=O)(c1cccc(Cl)c1F)NC1CCC(C(N(C)Cc2ccc(O)cc2)=O)C1 25272,c1(C(CO)NC2CC(C)(CC)C2)ccc(F)cc1F 25273,N1(S(C)(=O)=O)CCC(NC(=NCc2ccnc(Br)c2)NCC2CCOC2)CC1 25274,C(CC(=O)N(C)C(C)C)OC1C(C)C1.C1(=O)C(C)N1 25275,C1(F)(C(=O)NCC2CC(N(C)C)C2)CCCN(C(c2c[nH]nc2C2CC2)=O)C1 25276,c1(C(N2C3CN(C(C4(C=C)CC4)=O)C(C3)C2)=O)cc2ccc(OC)cc2s1 25277,C(CCCCC(=O)NCC1CCCC(C)(C)C1)N(C(=O)C1=CCCCC1)C 25278,CC1(C)CN(C(c2c(O)cc(F)cc2F)=O)CCN(C(=O)CCc2cn[nH]c2)C1 25279,C(=O)(C1=C(C#N)CCC1)NCC1CN(C(c2c(C)nc(N(C)C)s2)=O)C(C)C1 25280,c1(C(N2C3C(NC(=O)CCC4CCCO4)C(C3)C2)=O)n[nH]c2c1CCC2 25281,C1(NC(C(C)OCC(C)C)=O)CC2CC(C1)CN(C(C1(O)CC(C)(C)C1)=O)C2 25282,O=C1CC2CN(C(=O)C(c3ccc(OCCCN4CCOCC4)cc3)=O)CC2N1 25283,C=C(Cl)CC(C(=O)NCC1COCC(C)O1)NC(=O)COc1cccnc1 25284,n1(CC)cc(Br)cc1C(=O)OCc1nnc(C2CCOCC2)o1 25285,Cn1cc(Cl)c(C(N2CC(O)(CCNC(C34COCC3C4)=O)C2)=O)n1 25286,C1(CC)CCN(C(c2[nH]ccc2CNC(=O)CCCCSC)=O)C1C 25287,c1(C(=O)NC2CC3(C2)CC(Br)C3)cc(S(=O)(=O)N2CCC2)c[nH]1 25288,C1(C(=O)NC2C(NC(C=C(C)C)=O)C2)CCC(OC2CCOC2)CC1 25289,N1(C(c2c(C)nsc2)=O)CCC(C)C(NC(C2(F)CCCCC2)=O)C1C 25290,N(C(=NCCc1cnccc1OC)NC1CC1C1CCC1)CCC(=O)NC 25291,c1(C(=O)NC2C(NC(c3c(C)nc(C)s3)=O)CC2)cccc2oc(O)nc12 25292,C#Cc1c[nH]nc1C(=O)NC(C)CC(C)NC(=O)Cc1ccc(F)cc1 25293,C1(C(=O)OC)CC2(C1)CC(C(=O)NCC(CNC(c1sccc1SC)=O)CO)C2 25294,C1(CCC)(NC(=O)CCC2CC2(F)F)CCCN(C(c2cc(Cl)no2)=O)C1 25295,Cc1nc(NC(C2CCC(F)CC2)=O)sc1C(=O)NC(C)(C)C 25296,C=Cc1cnn(C)c1C(=O)NCc1cccc(NC(C2(C)CCC(C)C2)=O)c1 25297,C1(NC(C(C)OC(C)=O)=O)CC(C(=O)NCC2CC2c2ccoc2)C1(C)C 25298,C1(C(N2C(C3(NC(COCCC)=O)CC3)CCC2)=O)CC(=O)N(CC(F)(F)F)C1 25299,CCCCCC(O)CC(=O)N1CCOC(CNC(=O)C(CC)C2CCOCC2)C1 25300,c1(CNC(C2C(C(=O)OCC)C=C2)=O)cccc(OC)c1.C12CCN(C1)CCN2 25301,C(=O)(C(CNC(C1CC1(F)Cl)=O)N(C)C)N(CCCCO)CC 25302,C1(NC(c2ccc(OC)o2)=O)CC2CC1CN(C(=O)Cc1ccc(F)cn1)C2 25303,c1(C(NOC(C2CC2c2ccccc2)=O)=O)cnn(CCc2nn[nH]n2)c1 25304,c1(CC)nc(C(N2CCC(CCNC(C34CC(O)C3C4)=O)C2)=O)co1 25305,N1(C(C2N(CC)CCC2)=O)CCCC(CNC(=O)CN2CCC(OC)C2)C1 25306,Cc1ccc(CC(=O)NCCCCCNC(C2CN(C)C(=O)CCO2)=O)cc1C 25307,c1(NC(CNC(c2cc(CC)n(CCO)n2)=O)C(C)C)ncnc2cnccc12 25308,c1(C(=O)NC(CCNC(C(C)SC(C)C)=O)C)ccc2c(c1)NC(=O)CN2C 25309,N1(C(C=CCC(C)(C)NC(c2cnn(C)c2Cl)=O)=O)CCC(O)(CO)CC1 25310,c1(-c2c(NOC)cccc2)nc(S(C)(=O)=O)nc2c1ncn2C 25311,N1(C(CN(C(C)=O)C)=O)CC(NC(=O)C=C2CCC(C)CC2)CC12CCCOC2 25312,c1(C(=O)NCC(C(N2C(C)(CC)CC2)=O)N(C)C)nc(C)ccc1C 25313,C1(CNC(CC(CCOC)(C)C)=O)CCC2CN(C(=O)C3=CCCO3)CCC2C1 25314,C(=O)(C(CNC(=O)Cc1cncn1C)N(C)C)NCC(N(C)C)C1CC1 25315,S(=O)(=O)(c1ccc(NCc2ccc(Cl)o2)nc1)N(C)Cc1sccc1C(F)F 25316,c1(C(=O)NCC(C)(C)NC(c2c(SC)cc(F)cc2)=O)cc2ccc(F)cc2o1 25317,C(=O)(C1OCCc2c(O)cccc21)NC1C(C)(C)CN(C(=O)CCOC2CC2)C1 25318,c1(OC)c(NC(c2cnn(CCN(C)C)c2)=O)cccc1SC 25319,C1(CN(S(CC)(=O)=O)C)COCCN1C(=O)C(N1CC(O)C(F)C1)=O 25320,C(=O)(C1CCCn2cnnc21)NC(C)(C)CCNC(=O)CCOCC1CCCO1 25321,C1(CNC(CCNS(CC)(=O)=O)=O)C(C2CC2)CCN1C(=O)CC(C)(F)F 25322,Cc1ccc2c(c1)C(C(=O)NC(C)CNC(c1ccc(CO)cc1F)=O)C2 25323,CC1(C(N2CCC(C)(NC(c3cc(F)cnc3O)=O)C2)=O)CCCCC1(F)F 25324,Cc1cccc2[nH]cc(C(=O)NCC3CC3NC(c3nnc(O)nc3O)=O)c12 25325,C1(NC(c2[nH]cc(CC)n2)=O)CCC2(CCN(C(=O)CC(C)CC(C)(C)C)C2)C1 25326,c1(C(C)N)ccc(NC(=O)CN(CCCC#N)C(=O)CC)cc1 25327,Cc1cc(C(N2CCC(N(CCO)C(c3cn[nH]c3)=O)C2)=O)n2ncnc2n1 25328,c1(-c2ccc(C(N3C(C(C)NC(C=CC)=O)CCC3)=O)s2)cccc(F)c1 25329,Cc1cccc(OCC(=O)NC(CNC(=O)C2=CCCSC2)CO)c1C 25330,C1(O)(CCNC(c2n[nH]cc2F)=O)CCCN(C(c2sccc2C(F)F)=O)C1 25331,C1(NC(C(CC=C)OC)=O)CC(NC(C23COCC2C3)=O)C12CCC2 25332,C1(Cn2cnc(C(=O)O)n2)CCN(Cc2cn(CC3COCCO3)nn2)CC1 25333,c1(CNC(C(CC)(C)C)=O)cc2n(n1)CCN(C(=O)CN1CCCNS1(=O)=O)C2 25334,C1(F)(CNC(=O)C(F)=CC2CC2)COCCN(C(c2ncsc2C2CC2)=O)C1 25335,C1(C2=CCN(C(=O)Cc3c(C)ncnc3C)CC2)(C(=O)OC)CCC1 25336,O(NC(=O)C(CC(N)=O)NC(c1ccc(C)s1)=O)CC=C(C)C 25337,C1(C)(CNC(CC2N(C(CCn3ccc(C)n3)=O)CC(F)C2)=O)NC(=O)NC1=O 25338,c1(C(=O)NC(CNC(C(CC)F)=O)(C)CO)cccc(NCC)c1 25339,c1(-n2cc(CNC(c3ccc(C(CC)C)cc3)=O)nn2)cc(C)c(F)cc1Cl 25340,N1(C(c2ccc(C(C)C)s2)=O)CCC12CN(C(=O)CC13CCCC1C3)C2 25341,CC1(CNC(=O)CCC2(NC(=O)C=CC(=O)N(C)C)CCCC2)CCCCC1O 25342,c1(C(N2CC(Cc3cn(CC4(O)CC=CC4)nn3)C2)=O)ccn(CC(F)F)n1 25343,N1(C(=O)NCC(c2cnn(C)c2)C)CCC(C)C1c1ccc(CC(F)(F)F)cc1 25344,C1(CCOC)(C(=O)NCCCCCNC(C)=O)CCCCO1.C12(CC1)C(=O)N2 25345,C1(CNC(C2C(C)=C2)=O)C2CN(C(=O)COc3ccccc3)CC12 25346,C(CN=C(NCC1(O)CCN(C)C1)N1CCC(SC)C1)SCCC=C 25347,C#CC1CN(C(=O)CC2CCC(C)(C)CO2)CCN1C(c1nnsc1CC)=O 25348,N1(C(C(C)NC(=O)NC)=O)CCC(CCCCNC(C2C(F)(F)C23CC3)=O)CC1 25349,N1(C(CC(CCCC)O)=O)CCOC2(CCN(C(c3cnn4c3CCC4)=O)C2)C1 25350,c1(NC(C2N(CC)CCC2)=O)nc(OC)ncc1F.N12CCC(C1)C2=O 25351,C(C(CC(=O)N1CCC1c1cccnc1)C1CCC1)NC(=O)C(C1(O)CCCC1)F 25352,C1(CNC(c2c(C)nn[nH]2)=O)CC(F)CN1C(c1sccc1C(F)F)=O 25353,C1(O)(CNC(C2CC2c2ccncc2)=O)CCCN(C(C2(F)CCC2)=O)C1 25354,N1(C(c2c(C)nccn2)=O)CCC(C2CCCN(C(=O)C(C)(F)F)CCC2)CC1 25355,c1(C(=O)NC2CC(CCNC(CC(COC)C)=O)C2)cnn2ccccc12 25356,C(=O)(CC1=CCOCC1)N1C(CN(C(=O)COCP(C)(C)=O)CC)CCC1 25357,c1(C(=O)NC2CN(C(C(CCC)N(C)C)=O)C2)ccc(C(C)C)cc1F 25358,CC1(C(=O)NCC(C2CCN(C(=O)CCC3CCC3)CC2)F)CCNC1=O 25359,c1(C(N(CC(C)NC(CCCCCC)=O)C)=O)sc2cc(C(C)C)ccc2c1Cl 25360,Cc1cc(C(=O)NC2CC(NC(C3(C4CCCO4)CCC3)=O)C2)sn1 25361,C(=O)(CCCCC(C)(C)C)NC(C(C(C)C)NC(=O)C=Cc1ccc(F)cc1)C 25362,N1(C(c2ccc(CC)[nH]2)=O)CC(C)N(C(=O)COCCc2ccccc2)CC1C 25363,CC(C)(CS(C)(=O)=O)C(=O)NCCC1CCN(C(=O)Cn2ncnn2)CC1 25364,C1(C(N2C(c3cn(CC4CCC(=O)O4)nn3)CCC2)=O)CC2CCCC2C1 25365,CC(CC(C)NC(=O)CCCF)NC(=O)C(CC1CC1)NC(=O)OC(C)(C)C 25366,C1(COC)CCCCN1C(=O)CCN(C(=O)CCc1ccc[nH]1)C(C)C 25367,CC(C)(F)CCC(=O)NCC1(C)CCCN1C(C1COC(=O)O1)=O 25368,CCCCS(=O)(=O)CC(=O)NCC1CCN1C(c1ccn2ncccc12)=O 25369,C1(C(=O)NCC(COC)NC(c2cnc(C3CC3)s2)=O)CNC(=O)N1C 25370,C=CCC(C)(C(F)F)NC(=O)C(n1cc(-c2ccc(C)cc2Cl)nn1)C 25371,C1(NC(c2ccn(CCOC)n2)=O)CN(C(=O)CNS(=O)(=O)C2CC2)CC1C 25372,S(=O)(=O)(c1ccc(OC)cc1O)NC1CCC(NCc2ccc(OCC)nc2)C1 25373,Cc1cc2[nH]c(C(=O)NCC(C(C)C)NC(=O)CCCCCN(C)C)cc2o1 25374,c1(C(=O)NCC(C2CCCC2)C)cn(CCNC(c2cc[nH]n2)=O)cn1 25375,N1(C(c2cnc(C(C)C)[nH]2)=O)CCC(C2CCN(C(=O)CC3CC=CC3)C2)C1 25376,N1(C(c2n(CC#C)cnn2)=O)CC(CNC(C2(C)CCCCC2)=O)CC12CCC2 25377,N12CCN(CC1)CC(C)NC2=O.C1(NC(CC=CCC)=O)CCC(C)CC1 25378,n1(CC(N2CC(N(C(=O)C(O)CC(C)(C)C)C)C2)=O)c(O)nc2ccccc12 25379,c1(C(=O)NC(CC(C)NC(CC(CC)(F)F)=O)C)cc(S(N)(=O)=O)c[nH]1 25380,c1(C(=O)NCCC(C)NC(c2cccc(F)n2)=O)cccc(Cl)c1Cl 25381,Cc1cc(C)c(C(=O)NCCC2CCN(C(=O)C(c3ccccc3)O)C2)s1 25382,C1(C(=O)NC2CCC(NC(c3cc(C#N)on3)=O)CC2)C2CCC3C(C2)CC13 25383,Cc1cnc(C(N2CCC(C)C(NC(c3ccc(C#N)cc3)=O)C2)=O)c(F)c1 25384,C(=O)(C(C(C)O)NC(N)=O)NC(CC)CN(C(=O)C(C)c1ccon1)C 25385,C1(C(N2C(C(=O)OC)CCC2C(F)(F)F)C(=O)NC)CCC2(CC2)C1 25386,C1(C(N2C(C(C)NC(C3CC=CCC3)=O)CCC2)=O)CCC(C)(F)CC1 25387,Cc1nsc(C(=O)NCC2CC(F)CN2C(=O)CC2CC(F)(F)C2)c1N 25388,N1(C(c2c(CC)cc[nH]2)=O)CCCC(CN(C)C(c2coc(C(F)F)c2)=O)C1 25389,Cc1nc(NCC(C)(C)C(C)O)cc(=NCc2ccc3ncsc3c2)[nH]1 25390,c1(C(=O)Nc2cccc(CNC(c3c(C)noc3C)=O)c2)c(C)oc(C)c1C 25391,C(CNC(c1cnc(SC)s1)=O)(C(C)(C)C)NC(c1cn(CC(CC)O)nn1)=O 25392,Cc1cc(F)cnc1C(=O)N(C)CCNC(C1C(C)(C)C1(F)F)=O 25393,C1(CC(=O)NC(C(C)(C)C)CNC(=O)C=Cc2ccco2)CCCC2(CC2)C1 25394,N1(C(c2c(CNC(C(C)SC(C)C)=O)nccc2)=O)CCc2nnnn2CC1 25395,C1(O)(CNC(C2CCN(C(C)=O)C2)=O)CCN(C(c2cnoc2C2CC2)=O)CC1 25396,c1(C(=O)NC2C(C)(CNC(C3(O)CCOCC3)=O)CCC2)nnc(O)cc1O 25397,C1(CN(C(C(=O)Nc2ccc(CCCC=C)cc2)=O)CC)Cc2ccccc2O1 25398,c1(CN(C(C(=O)N(CC(C)O)CCNC(C)=O)=O)C)ccc2c(c1)OCCO2 25399,N1(C(c2snc(OC)c2Br)=O)CCCC(CNC(=O)CSC(C)C)CC1 25400,C(=O)(CCCCNC(c1nnn(C)c1C)=O)N(CC=C)CC 25401,C1(N(C(CCCOC)=O)C)CC2CCC(C1)N2C(C12CCCC1C2(F)F)=O 25402,C(CC=O)(CC)NC(C=CCCC)=O.C12(F)CC1C(=O)NC2=O 25403,N1(C(c2cc(CNC(c3ccco3)=O)no2)=O)CC2CC1CO2 25404,N1(C(C(CC(=C)C)C)=O)CCC2CCN(C(c3c[nH]c4nccc-4c3)=O)C2C1 25405,C1(C(N(CCCNC(c2c(C)oc(Cl)n2)=O)C(C)C)=O)CCOC(=O)CC1 25406,C(=O)(C1=C(CC)OCCS1)NCC(C1CC1)NC(c1oc(CC)c(C)c1)=O 25407,C(=O)(CC1COc2ccccc21)NCC(C)CNC(=O)Cn1cc(C2CC2)cn1 25408,C(C(C)CC(=O)N1CCCCC1C(C)(C)CNC(c1cc(C#N)on1)=O)OC 25409,N1(C(C2(CNC(Cc3ccc(C)o3)=O)CCC2)=O)CCCC(C)CC1 25410,c1(SC)cncc(C(=O)NC2CC(NC(C3CC3(F)F)=O)CC2O)c1 25411,C12CCC3(CC13)C(=O)N2.N1(C(c2ccc(COC)o2)=O)CCCC(C(N)=O)C1 25412,c1(CCC)cc(C(=O)NCC(O)CCNC(=O)Cc2cccn2C)ccn1 25413,CC1c2cc(O)c(O)cc2CCN1C(c1ccc(NCc2ccccc2)cc1)=O 25414,c1(C(=O)NCC2C3CN(C(C4(CCCC)CC4)=O)CC32)cc(CC)nnc1C 25415,c1(CCC(=O)NC2CN(C(CCC(=C)Cl)=O)CC(C)C2)cccc(S(N)(=O)=O)c1 25416,C1(CNC(CN(C)CCO)=O)CN(C(C2CC3CCCC3C2)=O)CC(C)(C)O1 25417,C1(C(C(C)C)NC(C=CC)=O)CCN(C(=O)CN2CC(=O)NC2=O)CC1 25418,c1(C(=O)NC2CCC(CCNC(c3oc(C)c(CO)c3)=O)C2)cccc(F)c1O 25419,Cc1cc(CN2CCC(C(C)NC(C3COCCN3C)=O)CC2)ncn1 25420,N1(C(=O)C=CBr)CCC2CN(C(=O)CSCC3CCCCO3)C2C1 25421,N1(C(C2(CO)CCCO2)=O)CCC(F)(C(=O)NCc2n[nH]cc2C2CC2)CC1 25422,CN1C(=O)CC(C(C)(C)CNS(=O)(=O)Cc2nc(Cl)sc2Cl)C1=O 25423,C12(CC(=O)N(C3CCN(C(c4ccc(CC#N)cc4)=O)C3)C)COCC(C1)C2 25424,N1(C(CNC(CC)=O)=O)CCC(C(=O)Nc2cc(Cl)ccc2-n2ccnc2)CC1C 25425,N#Cc1c(NC(C2CCCN3CCCC23)=O)sc2c1CCCCC2 25426,c1(OCC)ccc(C(C)NC(C23CC(CNC)(C2)C(C)O3)=O)cc1OC 25427,C(=O)(C1SCCc2sccc21)N(C(C)(CNC(=O)CCc1ncc[nH]1)C1CC1)C 25428,C12(NC(c3cnc(=N)[nH]c3)=O)CCN(C(c3cnn(C4CCCC4)c3)=O)CC1C2 25429,CN1CCCC1CC(=O)NCCOCC(=O)NC1CCN(CC2CC2)C1 25430,C(=O)(C1CCCc2nn[nH]c21)N1CC2CC(NC(=O)Cn3ncccc3=O)C2C1 25431,Cc1cc(C(N2CCC(NC(=O)C(=O)N(C)C)C(CO)CC2)=O)cc(C)c1C#N 25432,c1(C(N2C(CNC(c3c(C)ccc(OC)c3)=O)CC2)=O)cn(C)c2ncccc12 25433,CCCCCC(O)C(=O)NC(C)CN(C(=O)C(c1ccc(=O)n(C)c1)(F)F)C 25434,N1(C(c2cc(C)sc2)=O)CC(C)CN(C(c2ccn(C)c2C)=O)C(C)C1 25435,C1(CC=O)(OC)CN(C(C(C(=O)N2CC(Cn3ccnn3)C2)C2CCC2)=O)C1 25436,c1(CC)c(C(=O)NC2COCC2CNC(C2(CC(C)C)CCC2)=O)ccn1C 25437,c1(C(=O)NCC(CC)C#N)nc(CNC(c2cnn(C(F)F)c2)=O)oc1C 25438,Cn1c(NCC(C2CCCC2)NC(=O)CC=C(Cl)Cl)cc(=O)n(C)c1=O 25439,c1(C(=O)NC2C(C)(CC)C2)cc(CNC(C2(CC)CCCC2)=O)[nH]n1 25440,N1(C(C2(S(C)(=O)=O)CCC2)=O)CC2CCC1CN2C(=O)CN1CC2C=CC1C2 25441,CC1CCCC1NC(=O)CCCN(C(=O)CC1CCCC1)C 25442,c1(CNC(c2cc(C)[nH]n2)C)ccc(CN2CCC(C)CC2)cc1 25443,N1(C(CCCC#C)=O)CCC(NC(=O)CC2CCC(=O)N2C)C12CC2 25444,C1(CCC)CC(C(=O)N(C(C)CCNC(=O)C(C)C)C)C1 25445,N1(C(COC)=O)CC(OC)C(NC(=O)Cn2cc(-c3ccc(C)cc3)nn2)C1 25446,c1(C(=O)NCC(CO)NC(CC(CC)C2CC2)=O)cc(C)ncc1C 25447,N1(C(CC=C)=O)CCC2CCCC12C(=O)NC(c1ccnn1C)C 25448,c1(C(COC(CCCCC)=O)=O)ccc(N2C=CC=CC(C(F)(F)F)C2=O)cc1 25449,CS(=O)C1CN(C(=O)CC2CCN2C(c2csc(Cl)n2)=O)C1 25450,c1(C(=O)NCCCC2(CNC(C(C)N(C)C)=O)CCCC2)cnc2ccoc2c1 25451,CC1CNC(C)(C)CN1C(=O)Cc1ncc(Br)s1 25452,C=CC1(C(=O)NC2CCC(NC(=O)C(C)=CCC)CC2)CCCCC1 25453,C(=O)(CCCN=[N+]=[N-])N1CCC(N(C)Cc2c(C(=O)OC(C)(C)C)occ2)CC1 25454,N1(C(CSCC)=O)CC2CC1(C(=O)NCCc1nc[nH]n1)C2 25455,C1(CNC(CCc2n(C)ccc2)=O)C(O)C(O)CN1C(C1CCNC(=O)C1)=O 25456,c1(C(=O)NC2(C3N(C(C4CC(OC)C4)=O)CCC3)CC2)cnc2ncccc2c1 25457,N1(C(CSCCCC)=O)CCC(C)(CNC(=O)C2=NOC(C(C)(C)C)C2)CC1 25458,C(=O)(CC(CC(C)C)NC(C12CCC(C)(C1)OC2)=O)N1CC(C)(CC=C)C1 25459,N1(C(C)C)C(=O)CCC1C(=O)NCCCNC(=O)CC1CC2(COC2)C1 25460,C1(C)(C(=O)NC2C(NC(C)=O)CCC2)Cc2ccc(Br)cc2C(=O)O1 25461,Cc1ncncc1NC(C1CC1NCc1cccc(CO)c1)=O 25462,N1(C(C(C)N(CCCC)C(=O)COC)=O)CCN(C(=O)CCOC2CCCC2)CC1 25463,C1(C(C)C)(C(=O)NCCC2(NC(C3CC34CCCC4)=O)CCCC2)CNC(=O)C1 25464,Cc1cc(CCC(=O)N(CCNC(=O)CC2(C)CC2(F)F)C(C)C)on1 25465,C1(NC(C(C(C)C)(C)C)=O)CC2CCC1CN(C(=O)CC1CCCCC1O)C2 25466,c1(C(=O)NCCCC2(NC(CCn3ncc(C)c3)=O)CC2)cc2ccncc2s1 25467,N1(C(c2c(C)cn(C)c2)=O)CCC(F)C(NC(c2cc(C)n(C(C)(C)C)n2)=O)C1 25468,c1(NC2C(CC)CN(C(=O)C(F)(F)F)CC2)ccnc2cccnc12 25469,Cc1nn(C)c(C)c1C(C)C(=O)NC1CC(CCNC(=O)CC2CCCOC2)C1 25470,c1(OC)cc(CNC(=O)NC2CN(C)C2Cn2cccc2)ccc1OC(C)C 25471,N1(C(c2c(C)csc2)=O)C2CCCC1CN(C(C1CCc3n[nH]cc3C1)=O)CC2 25472,C1(C(=O)NC2(C)CCCC2)CN(C(C2(C#N)CC(=O)C2)=O)CC1(F)F 25473,N1(C(c2ccc(C)nc2O)=O)CC2(C1)CN(C(=O)C(C1CCC1)C1CCC1)CCO2 25474,C1(C(N2C3C(NC(COCCC)=O)C(C3)C2)=O)CCCC2CCCN12 25475,c1(C(=O)NCCN(C(C(CC#C)O)=O)C2CC2)ccc(OC)c(C)c1 25476,c1(NC(C2N(C(COC)=O)CC2)=O)ccc([N+](=O)[O-])c(C(=O)OC)c1 25477,N1(C(C(=O)NCC=C)C(C)C2CCOC2)CCN(Cc2ccccc2F)C(=O)C1 25478,c1(OC)cc(N)c(C(N2CC(NC(=O)Cn3cncn3)C3CC23)=O)cc1F 25479,C1(C(N2CC(S(C)(=N)=O)C2)=O)(NC(c2scc(OC)c2)=O)CCC(C)(C)C1 25480,c1(N2CC(N(C(c3ccn(CCOC)n3)=O)C)C2)ncnc2[nH]c(C)nc12 25481,c1(C(=O)NCC2CC(NC(C(C=CC)O)=O)C2)cc2n(n1)CCCC2O 25482,Cc1ncc(Cl)cc1NC(=O)CCC1(NC(=O)Cc2cccnc2C)CCC1 25483,c1(-n2cc(C(C)(C)NC(c3ccc(C(C)=O)cn3)=O)nn2)ccc(Cl)c(C)c1 25484,C1(=O)CC(Cc2cccs2)N1.c12cc(n(C)n1)NC2=O.C(C(C)C)N(CC)CC 25485,C(=O)(CC(C)(C)N(C)C(C1(Cl)CC1)=O)N1C(CC)CCC1 25486,C1(C#N)(C(=O)NCCCCCN(C(c2c(C)n[nH]c2)=O)C)C(C#N)C1(C)C 25487,C1(c2nc(C3CCCC(COC)C3)on2)CCCC12CCC2 25488,N1(C(c2c(SC)n(C)nc2)=O)CCCC(C2CN(C(C34CC(CO)(C3)C4)=O)C2)C1 25489,C=CCC(CNC(=O)C(C#N)CCC)C(=O)N1CCC(OC(C)=O)C1 25490,c1(SC)cc(N(C2CNCC2C#N)Cc2cc(Cl)sc2Cl)ncn1 25491,c1(C(=O)OC)ccc2nc(C(=O)OC(CC(C)C)c3cccs3)sc2c1 25492,C1(CNC(c2ccc(Cl)[nH]2)=O)CC(F)CN1C(C1CCS(=O)(=O)C1)=O 25493,CN1CCC(=CC(=O)NC2CC(CCNC(c3n[nH]cc3Br)=O)C2)CC1 25494,Cc1nc(N2CCC(c3cc(F)cc(Cl)c3)C2)ccc1[N+](=O)[O-] 25495,CC1(CNC(C2(C(F)F)CCC2)=O)CN(C(c2cc(Cl)ccc2N)=O)CCO1 25496,C=CCCC(C(=O)N1CCC(CN=[N+]=[N-])CC1)NC(=O)CCC(C)(C)C 25497,C1(CC(F)F)(C(=O)NCC(CNC(=O)Cc2cnco2)OC)CCOCC1 25498,C12(CNC(CC(c3cccs3)N(CC)CC)=O)CC1CN(C(=O)CCCOC)C2 25499,N1(C(C2CCC(C)O2)=O)CCC2(CCC2NC(=O)Cc2ccco2)CC1 25500,Cc1cc(NC2CC(CNC(=O)CCC3(O)CCC3)C2)c(Br)cc1[N+](=O)[O-] 25501,CC(C)(C)CCCCCC(=O)N1CC2CN(C(=O)CC3(C)CC3(F)F)CC2(C)C1 25502,C1(C(=O)NC(CCSC)C)CCN(C(=O)CCCC2CCCO2)O1 25503,C1(CC(=O)NCC2CC(OCC)C2)CCN(C(=O)CC2(C)CCC2)C1 25504,c1(C(=O)NC2CN(C(Cc3ccc(OC)cc3)=O)C(C)C2)c(C)nn(C)c1F 25505,c1(N2CCC(C(F)(F)F)(N(C)CC)C2)cc(C)[nH]c(=NCCc2cnn(C)c2)n1 25506,C(=O)(C1Cc2c(Cl)cccc21)NC1C(F)CCN(C(c2ccc(CC)s2)=O)C1 25507,c1(NC(=O)NCc2c(C)occ2)nc(O)c2cnn(-c3ccccc3)c2n1 25508,C(=O)(C1CCc2cccnc21)NC1(COC)CN(C(C2(C(CC)(F)F)CC2)=O)C1 25509,c1(CC(=O)NC2CN(C(C(CSC)O)=O)C(C)CC2)cccc([N+](=O)[O-])c1 25510,C(=O)(C(C)(CCC(F)(F)F)c1ccccc1)NCc1nc(C)c(C)[nH]1 25511,c1(C(N(CC(C)CNC(c2cnsc2)=O)C)=O)cc2c(nc1O)CCCC2=O 25512,C1(n2ncc(C)c2)CCN(C(=O)COc2cnn(C)c2)CC1.C12CC1CNC2=O 25513,c1(OC)cc(CN2CCN(c3nc(N(C)C)cc(C)n3)CC2)ccc1Cl 25514,C1(C(=O)NCCc2c(C)nn(C)c2)CN(C)CCN1C(=O)CC1CC(C)C1 25515,C=CCC(CNC(=O)Cn1cc(C)cn1)C(=O)NCC1(CO)CC12CCC2 25516,C1(N(C(=O)CCc2cnoc2)CC)CCCN(C(=O)CC=C(C)C)C1 25517,c1(COC)nc(NCCc2c[nH]nc2O)cc(=NC2CCCC(C)C2)[nH]1 25518,c1(CCN(C2(CC(=O)N(C(C)CC(C)C)C)CC2)C(C)=O)ccccc1 25519,C1(NC(c2cc(CCNC(CCSCCC)=O)on2)=O)CC(CO)C2CC12 25520,c1(OCC)nc(C(=O)NCC2CN(C(C3(C)CC3)=O)CC2OC)cc(O)n1 25521,N1(CC)CCc2sccc2C1.C(C)(C(=O)OC)N(CC(F)(F)F)CCCOC 25522,C(CCCCC(=O)NCC(CNC(C1CC(C)(C)O1)=O)OC)OCC 25523,N1(C(C(C)(CO)NC(C)=O)=O)CC2(C(=O)Nc3cnccc3C)CC1CO2 25524,N1(C(CCc2cccc(OC)n2)=O)CC(N=[N+]=[N-])CCC1(C)C 25525,C=CCCCCCC(=O)N1CCC2(C(=O)OC)CC2C1.n12nc(C)cc1NC(=O)C2 25526,n1(CC(=O)NCCCNC(CC2CC(CC)C2)=O)c(C)cc(C)cc1=O 25527,CC1CCN(CC(C)(C)COC(C2(c3ccc(C(C)C)cc3)CC2(F)F)=O)CC1 25528,c1(NC(C(CC)C)C)ccc(S(=O)(=O)NCCc2cccc(F)n2)c(Br)c1 25529,C1(C(N(CC(C(=O)NCC2CN(C(=O)OC)C2)C)C)=O)CCCC(=O)CC1 25530,CC1(C)COc2c(C(=O)NCC3CCN(C(c4csc(C#N)c4)=O)C3)cccc21 25531,N1(C(c2nccc(C#C)c2)=O)CC2CCCCC2(NC(c2cnco2)=O)C1 25532,c1(CN2CCC(CC(=O)N(CC)Cc3ccco3)C2)ccc(Cl)c(Cl)c1 25533,C1(CN(C(C2CC2CC(C)C)=O)CC)CCCCN1C(=O)CC1(OC)CCC1 25534,Cc1ccc(C(=O)O)cc1CNC(c1cnn(C2CCC2)c1C)C 25535,N1(C(c2c(CCC)cccc2)=O)CC2CCC2(CCNC(=O)C2=CCCCC2)C1 25536,C(=O)(CCCCCC(=O)NC(C)CNC(=O)CC1CCC2(CC1)CC2)OC 25537,C1(OCC)CCN(C(=O)C=CC(C)(C)NC(=O)CCOC(C)=O)CC1C 25538,C12(CCNC(CCc3c(C)noc3)=O)CCC1CN(C(c1cncs1)=O)C2 25539,Cc1cc(CNC(=O)NCc2ccc(CC(C)C)cc2)ccc1O 25540,CCCC(O)CC(=O)NC1CN(C(c2ccnn2CCC(F)(F)F)=O)CC1O 25541,c1(C(=O)OCC(c2n(C)nnc2)=O)cc2cc(Br)cn2cn1 25542,n1(CCC2C(OC)CCCC2)cc(C(=O)ON(C(=O)CCS(N)(=O)=O)C)c(=O)cc1C 25543,c1(C(=O)NC23CC(CNC(C4(C)CCN(C)CC4)=O)(C2)C3)cnc2ncccn12 25544,C12(NC(C(C)N(C(C(CC)=CCCC)=O)C)=O)CCN(CC1)CC2 25545,c1(N(CCNC(C(CCCC)C)=O)C2CC2)ccc([N+](=O)[O-])cn1 25546,N1(C(C(C(=O)OCC)OC)=O)CCC2(CCN(C(=O)C=Cc3ccco3)CC2)C1 25547,C1(OC)(CNC(N2CCCC2(CO)CO)=O)CCCSC1 25548,C1(NC(c2n[nH]cc2Br)=O)CC2CC(NC(C3CC34CC4)=O)C2C1 25549,C1(C#N)(C(N2CC(C)(c3cn(C4(O)CCOCC4)nn3)C2)=O)CC2CCC1C2 25550,CS(=O)c1ccccc1C(=O)NC1C=CC(CNC(=O)Cc2ccns2)C1 25551,C(CC(CC)(CC)NC(=O)C(O)CSC)NC(c1cn(CCCC)nn1)=O 25552,c1(NC(=O)NCC2(C#N)CC2)ccc(C(F)(F)F)cc1Cl 25553,C=CC1(C(N2CCC(OC(C)C)CC2)=O)CCN(C(=O)C(CC)N(C)C)C1 25554,Cc1cc(C(N2CCCC2CNC(C2(C3CCC3)CCC2)=O)=O)nc(C)n1 25555,c1(C(N2CCN(C(COCc3ccc(C)cc3)=O)CC2)=O)cnc(F)cc1C 25556,c1(OCC)ccc(Cl)c(Cl)c1.C1(C)(CCCC)CC1C(=O)NCCN(C(=O)C)CC 25557,c1(NC(=O)CC2COCCN2C(=O)NC2CCC(CO)CC2)cnnc(Cl)c1Cl 25558,c1(CCN(C)C)ccccc1C(=O)NC1CC(CCNC(C2OCCO2)=O)C1 25559,CCC(C)C(C(=O)N1CCCC1(C)CNC(C1CCOC1)=O)OC 25560,c1(-c2cc(C)sc2)nc(COc2cccnc2)nn1C(c1ccc(Cl)cc1)C 25561,c1(CC(N2CC(CC(C)NC(c3c(CCC)n[nH]c3)=O)C2)=O)cnccc1OC 25562,c1(OC)cc(C(=O)NCCCCNC(=O)C(F)Cc2ccccc2)c(O)c(Cl)c1 25563,c1(OCC)c(OC)cc(C(=O)NC2CCN(C(=O)C(F)F)CC2F)cc1Cl 25564,C1(NC(=O)C=C2CCCCC2)CN(C(C2CCN(C(CC)=O)C2)(C)O)C(C)(C)C1 25565,N1(C(c2c(C)scn2)=O)CC(C)CN(C(c2ncncc2Cl)=O)C(C)C1 25566,N#Cc1cc(CN2CCCC2CC(=O)NCCC2CCCCC2)ccc1F 25567,N1(C(CC(=O)NC)=O)CCC(NC(=O)CCNC(=O)Cc2ccccc2)C1C 25568,c1(C(N2C(CNC(c3ccc(CC)cc3)=O)CC(F)C2)=O)cccc2occc12 25569,Cc1cc(C(=O)NC(C2CCCN(c3nnc(C(F)F)s3)C2)C)nn1CCO 25570,C1(NC(CC(C)c2ccco2)=O)CCC(CNC(=O)CCc2ccc[nH]2)CC1 25571,N1(C(C(CCC=C)(F)F)=O)CCC2(CC1)COC(CNC(=O)CNC(N)=O)C2 25572,c1(C(=O)NCCC(C)NC(=O)C(C)(F)C(C)(C)F)cc2ncccc2[nH]1 25573,C1(CNC(COC2(C)CCOCC2)=O)CCCCN(C(=O)CCn2cncn2)C1 25574,CCS(=O)c1ccccc1C(N1CCCN(CCNC(C2CC2C)=O)CC1)=O 25575,N1(C(c2n(C)ncc2Br)=O)CCC2(CC1)CC(NC(=O)C(C)(CO)CO)CO2 25576,C1(NC(c2cc(C)sc2)=O)CCCN(C(=O)CN2CCC(=O)NC2=O)CC1F 25577,Cc1nc(N)c(CC(=O)NC2CCCC2NC(=O)CC(C)P(C)(C)=O)c(O)n1 25578,Cc1nc2cc(C(=O)NCC(CNC(c3cn(C)cn3)=O)CO)cnc2[nH]1 25579,c1(NCCSC2C=CC(CC(=O)N(CC)CC)C2)cccc(C#N)c1F 25580,C(C)(CNC(C1(C2(C)OCCO2)CC1)=O)(CC)NC(C=C(CC)C)=O 25581,N1(CC)CCCN(C(c2ccccc2C(C)(C)C)C(=O)NC2CCOC2)CC1 25582,Cc1cc(F)cc2c1CN(c1cnncc1Oc1ccccc1)CC2 25583,c1(C(=O)NC2CN(C(Cc3nc(=N)[nH][nH]3)=O)CC2O)cccc2ccccc12 25584,n1(CC)cnc2c(NCc3ccnn3C)[nH]c(=NC3CCOC(C)C3)nc12 25585,Cc1ccn2c(C(=O)NC(C34CCC(CC3N)C4(C)C)=O)cnc2c1C 25586,N1(C(CCOC)=O)CCOCC(C)(CNC(c2ccc(CS(C)(=O)=O)cc2)=O)C1 25587,C1(NC(C2C(C3C(C)C3)C2)=O)CCN(C(=O)Cc2ccccc2F)C1(C)C 25588,n1(CC)cc(CC(=O)NC(CNC(=O)C=CCN(C)C)CCOC)cn1 25589,Cc1ccccc1OCC(=O)NC1CN(C(=O)CCC2NC(=O)NC2=O)CC1O 25590,c1(C(=O)NC2CC(N(C)C(C3CC34CCCC4)=O)C2)c[nH]c2ccc(Cl)cc12 25591,c1(C(=O)NCC(C)CNC(C2COC(=O)N2C)=O)ccc(C(O)CF)cc1 25592,C1(C(=O)NCCCN(C(C(C)SC)=O)C(C)C)CC(=O)N(c2ccccc2)C1 25593,N1(C(C)=O)CC2CC1CN2C(=O)COC1CN(C(C2C3CCC(=O)C23)=O)C1 25594,C(=O)(CC(C)C(C)(C)NC(=O)CSC1CC1)NCCCCCCC=C 25595,C(=O)(C1=C(Cl)CCC1)N(CCC)CCNC(=O)CNC(c1cnccn1)=O 25596,N1(C(C=C2CCC(C)C2)=O)CCC(C2(NC(c3cc(F)c(F)c(F)c3)=O)CC2)C1 25597,c1(SCC=C)ccccc1NC(=O)COC(C1CC(C)OC1C)=O 25598,N1(Cc2cn(CCCCCN)nn2)CCOc2ncccc21 25599,C1(CC(=O)NCC(COCC)(C)C)CC(C)N(C(=O)Cc2cnccc2C)C1 25600,CC(CC(=O)N1CCN(CC(N2CC(F)(F)CCC2C)=O)CC1)C(C)(C)C 25601,c1(C(=O)OC)cc(C)cnc1NC(CNC(=O)C=Cc1cccnc1)CO 25602,c1(C(N(C)CC2CCC2(F)F)=O)cnc(N(C)C)nc1 25603,C(CN=C(NCC1CCCO1)NCc1c(Br)cnn1C)N(CC)CC 25604,C1(CNC(C2(CCCC)CC2)=O)CCCCCN1C(c1ccccc1OC)=O 25605,CN1CCC(O)(CNC(=O)CCN(CCCO)C(C2(F)CCCCC2)=O)CC1 25606,Cc1cc(O)c(C(=O)NCCCN(C(=O)COCCCF)C)cc1Br 25607,C(CC(C)C)(C(=O)NC(C1CCOC1)C)NC(C=CC=CCC)=O 25608,C=CCN=C(NCc1ccc(F)cc1)NC1CCCN(CC(F)F)C1 25609,N1(C(C2C(C(C)C)C2)=O)CC2CN(C(=O)C3=CCCC(C)(C)C3)CC2C(F)(F)C1 25610,N1(C(=O)CCc2cc[nH]n2)CC2CN(C(c3ncc(Cl)s3)=O)CC2C1 25611,Cc1ncnc(C(N2CCC(CN(C)C(c3n[nH]cc3C(F)(F)F)=O)C2)=O)c1C 25612,N1(C(CCC(=C)Cl)=O)CCC(CNC(c2cc(Br)ncc2OC)=O)C12CCC2 25613,N1(C(C(C)NC(C)=O)=O)CCC(C2OCCC2NC(c2ccns2)=O)CC1 25614,C(C(F)(F)F)(C1CCCCC1)NC(=O)NC(c1cscn1)C 25615,N1(C(C(C)(C)C2CCOC2)=O)CC2C(CNC(=O)C(N)=O)C2C1 25616,Cc1ccc(C=CC(=O)NCC(O)CN(C(=O)CN2CCCCC2)C)c(C)c1 25617,c1(C(=O)NC2(CNC(C(CCOC)OC)=O)CCOC2)cnc(C2CC2)cc1C 25618,C1(F)(CNC(c2ccccc2)=O)CCN(C(=O)CCNC2(O)CCCCC2)C1 25619,C(=O)(C(C)C1=CCCC1)N(C)CC1CN(C(CSC(C)C)=O)CC12CC2 25620,CC(CC(=O)N1CCN(C)CC1)C(C)(C)NC(=O)CCCCN=[N+]=[N-] 25621,C1(O)(CN(C)C(c2scnc2C2CC2)=O)CCN(C(=O)CCc2cnc[nH]2)C1 25622,CC1CN(C(=O)C(C)(C2CC2)N(C)C(c2cncc(CO)c2)=O)CCS1=O 25623,C(CNC(c1ccc(N2CCC(C)(C)C2)cc1)=O)(CCS(C)(=O)=O)OC 25624,C1(C(N2CC3C(CNC(CNC(C(C)(C)C)=O)=O)C3C2)=O)CC2(CCOCC2)C1 25625,C1(C(=O)OCC)(NC(C2CCC2)=O)CCC1.C12CC(C1)C(=O)N2C.C1CC1C 25626,C(=O)(C1=NOC(C(F)(F)F)C1)OC(=O)COC1CCC(Oc2ccncc2)C1 25627,C1(NC(CSCC)=O)CN(C(c2csc3nnsc23)=O)CCC1C 25628,C(C1CCCCC1)=CC(=O)NC1(C2N(C(C3CC(N(C)CC)C3)=O)CCC2)CC1 25629,N1(Cc2ccc(C(=O)OC)[nH]2)CC2CCN(C(c3ccc(C#N)c(F)c3)=O)CC2C1 25630,c1(OC)cccc(F)c1CCNC(CO)CF 25631,c1(C(=O)NCC2N(C(CCC)=O)CCCC2C)cc2ccccn2c1 25632,Cc1cc(C(N2CC3CC3(NC(=O)C=CC3CCC3)C2)=O)c(S(N)(=O)=O)s1 25633,C(C)(CNC(=O)CC1(CC)CCC1)(CO)NC(C(F)=CC)=O 25634,c1(C(=O)OCC)cccc(C(=O)OC(C(CCSCC)(C)C)=O)c1O 25635,N1(C(c2sc(C)c(O)n2)=O)CC2COCCC2(NC(C2OCC3CCCC23)=O)C1 25636,c1(C(C)C(=O)NC2CCC(NC(C3CC(Cl)(Cl)C3)=O)CC2)ccc(C#N)cc1 25637,Cc1ccc(F)c(C(=O)NCc2occc2C(=O)NC(C)C(F)F)n1 25638,C1(N(C(=O)CN2CCS(=O)CC2)C)CN(C(C2CCCCCC2)=O)CC12CC2 25639,C=CCC(C(=O)NC(C)CC(C)(C)OC)NC(C1(CO)CCCCC1)=O 25640,c1(C(N2CC(CN(C(C(CCSC)O)=O)C)OCC2)=O)ccc(=O)n(CCO)c1 25641,S(=O)(=O)(c1cccc(S(=O)(=O)N2CC3CN(C)CCC23)c1)NCC(=C)C 25642,c1(C(N2C(CNC(c3c(C)cco3)=O)CN(C)CC2)=O)ccc2nccn2n1 25643,C1(C(=O)NC(CCCC)CNC(=O)COC2(C)CCC2)Cc2nccn2C1 25644,Cc1nn(C)c(C)c1C(C)C(=O)NC(CNC(c1cc[nH]c(=N)c1)=O)C(C)(C)C 25645,C1(CC(=O)NC(CC=C)CNC(=O)CCOC2CCC2)CCC2(CC1)COC2 25646,CC(CCCO)N=c1[nH]c2c(c(=NCC3OCCC3(C)C)[nH]1)COC2 25647,Cc1cc(C(=O)NC2CC3(C2)CC3NC(=O)CC2CN(C)CC2O)cc(C)c1Cl 25648,c1(CC(=O)NCC2C(NC(c3c(C(C)(C)C)ncs3)=O)C2)cccc(F)c1O 25649,C1(CC(=O)NC(C(C)(C)NC(c2c(C)con2)=O)C)CCOC(C(C)C)C1 25650,C1(OC(=O)CC2SC3=NCCN3C2=O)C=C(c2ccc(Cl)cc2)CCCC1 25651,CCCC(CCCNC(C1CC(C)OC1C)=O)NC(c1ccnn1CCC)=O 25652,C1(NC(c2n(CC)ccc2)=O)(CF)CCN(C(=O)C=C(C)C(C)C)C1 25653,N1(C(c2nc(NC(C)=O)sc2)=O)CC(NC(C2CCC(=C3CCC3)CC2)=O)C(C)C1 25654,c1(C(=O)NCCN(C(CCc2c(C)nn(C)c2C)=O)C)nc(=N)[nH]c2ccccc12 25655,C(CN=C(NCC(=O)OC)N1CCC(O)C(C)C1)Sc1c(OC)nn(C)c1 25656,C(C(CC(C)C)C(=O)N(C1CCCC1O)C)NC(c1cc(C)oc1)=O 25657,C1(N(C(CC2C(C)CCC2)=O)CCO)CCN(C(=O)C(CO)NS(C)(=O)=O)CC1 25658,C1(CNC(=O)C=Cc2cccs2)CCN(C(c2cn(C(F)F)cn2)=O)CC1 25659,c1(CCC(=O)NC2(C)CC(NC(COCC)=O)C2)ccc(C#N)cc1 25660,C(=O)(CCC(C)(C)N(C)C)NC1CC(CNC(c2ncc(OC)nc2)=O)C1(C)C 25661,N1(C(CNC(=N)N)=O)CC2(CCCC2NC(=O)Cc2c(Cl)cccc2Cl)C1 25662,C1(CC)CC(O)CN1C(=O)CCCCN(C)C.c12cc(on1)CNC2=O 25663,c1(OC)cc(OC)cc(C(=O)NCc2csc(CNC(=O)C(C)SC)n2)c1 25664,C1(CNC(CC(C)SC)=O)CN(C(C2CC=CCC2)=O)CCC1C 25665,CCCCC(CC(=O)NC1CC2(C1)CC2(F)F)NC(c1cccc(CC)n1)=O 25666,CC1CCN(C(=O)C(=O)N(C)C)C(C)C1NC(c1cc(CC(F)(F)F)[nH]n1)=O 25667,C(c1cc2ccccc2o1)=CC(N1CCC(C(C)NC(COCCC)=O)C1)=O 25668,c1(C(=O)NCC(CC=C)NC(C2CC(O)CN2C)=O)c(F)ccc(C)c1Cl 25669,N1(C(C(C2CCOCC2)OC)=O)CCC(C(F)CNC(=O)CSC)CC1 25670,c1(OC)cnc(C(F)(F)F)cc1C(=O)NC1(CF)CCN(C(=O)C(O)C(C)C)C1 25671,N1(CC(=O)NC(COC)C2(C)CC2)C(=O)CCC1=O.C12CCC(C1)C(=O)NCC2 25672,C=C(Cl)CC(C(=O)NC(c1cn(C)nc1C)C)NC(=O)Cc1ccc(F)cc1 25673,c1(C(=O)NCC2(NC(C3C(C(C)C)(CC)C3)=O)CC2)cc(O)cs1 25674,Cc1ccc(C)c(C(N2CC3C(CNC(c4cnn(C5CCC5)c4)=O)C3C2)=O)n1 25675,C1(NC(C2C(C(=O)OC)CCC2)=O)CN(C(=O)C(C)CC(F)(F)F)C2(CCC2)C1 25676,CC1CN(C(=O)C(N2C(C)CCC2C)C)CCN1C(=O)CCCC(C)O 25677,CCCC(CCC)=Cc1nc(C2(C(=O)N(C)C)CC2)no1 25678,N1(C(C(CCOC)OC)=O)CCC12CN(C(=O)C(CC(C)C)NC(C)=O)C2 25679,CN1C(=O)OC2CN(C(C3(F)CN(C(c4ccncc4Cl)=O)C3)=O)CC12 25680,N1(C(CCC#C)=O)CC(N(C(=O)CN(C)C)C)C2(CC2)C1 25681,N1(C(CC(C)(C)SC)=O)CC(CNC(=O)C(C)C(C)(C)C)OC(C)(C)C1 25682,C1(C(N(CCN(C(CCOCCCOC)=O)C(C)C)C)=O)CCC(N=[N+]=[N-])CC1 25683,N1(C(C2CCC(=C)CC2)=O)CCC2(CC(NC(=O)CCOCC(C)C)C2)C1 25684,C=CC1COCC1NC(=O)C(O)CCNC(=O)CCOCC(F)F 25685,CC(C)CC(C(=O)NCC1C2CCOCC12)N(S(C)(=O)=O)C1CC1 25686,c1(NCC2(CCC)CC2)nc2ccccc2nc1NCc1cc(Br)ccc1N 25687,C12(c3cn(CCOC)nn3)COC(CN1C(=O)C(C1(OC)CCCOC1)(F)F)C2 25688,c1(C(C)=O)ccc(C(=O)NCC=CCC(=O)NCCCCCC)[nH]1 25689,c1(C(CNC(C(CC)=CC)=O)CNC(c2cnn(CCF)c2)=O)cccc(C)c1 25690,C(CC(N)=O)(C(=O)N1CCCC1c1nc[nH]n1)NC(C(C)c1cccs1)=O 25691,C1(NC(c2occ(C)c2)=O)CCCCCCC1NC(c1cnn(C2CC2)c1)=O 25692,c1(CC)ncc(C(N2CCCC2CCNC(=O)COC2CCCCC2)=O)s1 25693,O(NC(=O)CC1(C)CCN1C(C1(OC)CCOC1)=O)CC(=O)OCC 25694,C(C(CC(C)C)C(=O)NCC1CCCN(C(C2CC(=O)N(C3CC3)C2)=O)C1)OC 25695,C1(C(C)NC(=O)CCOc2ccc(Br)cc2)CCc2ccccc2C1 25696,N1(C(C=CSC)=O)CC2CCC1C1CN(C(=O)CCn3cc[nH]c(=O)c3=O)CC21 25697,CN1C(=O)NCC1C(=O)NC(C1CCCC1)CNC(=O)C=CC1CCOC1 25698,C#CCCC(O)C(=O)NC1(C)CN(C(=O)C2=CSCCO2)C1 25699,O(P(=O)(CCCNC(=O)Cn1cc(C2(C)CSC2)nn1)OOC(C)C)CC 25700,Nc1nccnc1C(=O)NCC(c1ccccc1)CNC(C1COCC1CF)=O 25701,CC1C(NC(c2ccsc2C(F)F)=O)CC2CCC1N2C(C1CN(C)C(=O)N1)=O 25702,c1(C(=O)NC2CCCC2C(=O)NCC2(O)CCCC2)ccc(F)c(F)c1O 25703,c1(C(N(C2CCN(C(c3scc(C)c3)=O)CC2)CCO)=O)ccn2ncccc12 25704,C1(NC(C(F)(F)C2(OC)CCC2)=O)CC2CCC1(NC1(CO)CCCO1)C2 25705,N1(CCC(=O)NCC2(C(N3CCC3CC3CC3)=O)CCCO2)CCCCC1 25706,C(COC)(C(=O)NOCC(=O)NC(C)C)NC(c1c(CC)cns1)=O 25707,N1(C(CN(C(C(C)OCC2CC2)=O)CC2CC2)=O)CCC(O)C(C)(C)C1 25708,c1(C(N2CCCC(F)(CNC(c3ccncc3F)=O)C2)=O)cccc2nn[nH]c12 25709,Cc1nc(C(=O)NCC(c2ccccc2F)NC(=O)C=CC2CCC2)c(C)s1 25710,N1(C(=O)CSC2CC2)CCOC(c2ccccc2)C(O)C1 25711,N1(C(c2cccc(I)c2)C(=O)NC2(C)CC2)CCCC(O)(c2cccc(F)c2)CC1 25712,n1(CC)ncc2cc(C(=O)NC(CNC(c3nocc3Cl)=O)CC(C)C)cnc12 25713,c1(NC(C(=O)NCC(N2CCOCC2)C2CC=CC2)=O)cccc(CO)n1 25714,C(CCC(C)(C)C(=O)NCC1CCC2(CCC2)C1)NC(COCCOCC)=O 25715,C#CCCCCC(=O)N1CCC(CO)C(NC(c2ncccc2Br)=O)C1 25716,C1(CC(=O)OC)CCN(CCCCc2ccccc2Br)C2(CC2)C1 25717,CCCC(C(=O)NCc1cc(C)ns1)NC(=O)CC1CCOC1(C)C 25718,C1(CCN2CCCC(O)C2)CC(C(=O)NC(C2(C)CCCC2)=O)=CC1O 25719,CCCC(CCC)CC(=O)NC(C(=O)N(C)CC)C1CCOC1 25720,c1(C(=O)NC2CN(C(C(CCC)N(C)C)=O)C2)nc2ccccc2[nH]1 25721,c1(C(N2CCC(NC(C=CC)=O)(CO)C2)=O)cc2c(=O)n(C)c(=O)n(C)c2n1C 25722,N1(C(C(CCSC)O)=O)CC(NC(=O)Cc2ccc(C)s2)C(C2CC2)C1 25723,c1(C(=O)NC2C(C)(C)C(CC(=O)NCc3ccco3)C2)ccc2c(c1)CC2 25724,C1(COC)(NC(=O)CNC(N)=O)CCN(C(=O)CCc2ccncc2Br)C1 25725,N1(C(CCC2C(C)(C)C2)=O)CCC(OCCNC(c2sccc2F)=O)C1 25726,C1(NC(C2CC(C)CC(C)C2)=O)CCOC12CCN(C(=O)OC(C)(C)C)CC2 25727,C1(C(=O)O)CN(C(c2cnc(OCC(F)F)cn2)=O)C2(CCC2)C1 25728,c1(C(=O)NCCC2(CNC(C3(C)C(C)(C)C3)=O)CC2)cccc(OC(F)F)n1 25729,C(CCN=c1[nH]c(=NCC2COC(C)(C)CO2)[nH]c2c1CSC2)NC(C)=O 25730,c1(C(N(CC)CC2CCCN2C(c2occc2F)=O)=O)[nH]c(O)nc1C 25731,c1(N2CC=CCC2)nc(=NCC2CN(S(C)(=O)=O)C2)[nH]c2c1CSC2 25732,c1(C(=O)NC(CC)CNC(=O)C(c2cccs2)SC)ccc(-c2ccncc2)s1 25733,c1(CNC2CC(CC(N3CCN4CCCCC4C3)=O)C2)cn2cc(Br)ccc2n1 25734,C(=O)(C(C)(C)Nc1ccccn1)NCCCN(C(=O)CN1CC(C)(C)C1)C 25735,N1(CC(=O)NCC2C(NC(C(C3CCC3)OCC)=O)C2)CCC(C(N)=O)CC1 25736,Cc1nc2c(C(=O)NCC3CCCN3C(=O)C=Cc3sccc3C)cccc2o1 25737,c1(C(=O)N(C2CCCN(CC(F)(F)F)C2=O)C2N(C)C(=O)CC2)ncc(F)cc1F 25738,c1(NC(C2N(CC)CCC2C)=O)ncc(C)cc1Cl 25739,Cc1cccc(C(C(=O)O)NC(c2ccccc2C(N)=O)=O)c1 25740,C1(CNC(=O)NC2C(C)SCCC2)CN(C(=O)OC(C)(C)C)CC1(F)C(=O)O 25741,N1(C(CC=C)=O)CCCC2(CCN(C(=O)C=Cc3ccc(OC)cn3)CC2)C1 25742,CCCCC(CCCC)C(=O)NC(C1CCCN1C(=O)CS(=O)(=O)NC)C 25743,C(=O)(C1=NOC2COCC12)N(C)CC1CCCC1NC(c1cnccc1Cl)=O 25744,CC1CCN(C(C2CC2C2CC2)=O)CCN1C(c1cc(Cl)nnc1O)=O 25745,N1(C(CNS(CC)(=O)=O)=O)CCCC(O)(CN(C(=O)Cn2nccn2)C)C1 25746,N1(C(C(C=C)CC)=O)CC(NC(=O)CN(C)CCO)CCC1C 25747,C(=O)(C(O)CC(C)(C)C)NCC1(CNC(CCCOC(C)=O)=O)CCCS1 25748,Cn1cc2c(C(=O)NC3CCCN(C(=O)CCc4nc(=N)[nH][nH]4)C3)cccc2n1 25749,CC1CC(CCNC(c2cccs2)CO)C1 25750,C(N=c1[nH]c2c(c(=NC3CCC4CCC34)[nH]1)CCCCC2)C1(COC)CCCC1 25751,c1(SC)ccc(C=CC(=O)NCC2(COC(C)C)CC2)s1.C12CC1CNC2=O 25752,S(=O)(=O)(c1ccc(Nc2cn(C)nc2OC)nc1)N1CCC(CCCC)C1 25753,n1(CC(=O)OC(CNC(C(C)OCC#C)=O)C)cc(Cn2ccnc2)nn1 25754,N1(C(CCOCCOCC)=O)CC(OC)C(NC(=O)CCCON)C1 25755,Cc1nc2ccsc2c(=NCCNC(=O)C(C)Cc2ccc(F)cc2)[nH]1 25756,C1(C(=O)NCCOC(C)C)(CNC(C2CC(OC)C2)=O)CCCCC1 25757,N1(Cc2cccc(C#N)n2)Cc2ccc(NC(C3CCOCC3)=O)cc2C1 25758,C1(N(C(C(C(=C)C)(C)C)=O)C)CC2CCC(C1)N2C(=O)C1=CC2CCCC12 25759,CCC(CC)CCC(=O)N1CCC(N(C(=O)C#CC2CCC2)CC)C1 25760,N1(CC(N2C(c3nc(=N)[nH][nH]3)CCC2)=O)CCC2(CC1)CC2C(=O)O 25761,N1(C(C(CCOCC)NC(c2ccns2)=O)=O)CC2C3CCC(O3)C2C1 25762,C1(OC)CCN(CC(N2CC(NC(C3SCCS3)=O)C(C)C2)=O)CC1 25763,C1(C2CCC2)(N(CCCSC2CCCC2)C)CC1 25764,C1(C(=O)NCCCC(C)NC(=O)Cc2cccc(F)c2)COCC2(CCC2)O1 25765,N1(C(c2c(C)sc(Cl)n2)=O)CCN(C(c2ncc[nH]2)=O)CC(O)C1 25766,N1(C(CN2C(C)CC2)=O)CCC(F)C(NC(c2cc[nH]n2)=O)C1 25767,c1(C(=O)Nc2cc(F)ccc2F)n[nH]c2c1CN(C(C1(F)CC1)=O)CC2 25768,C1(CNC(C=CC(CC)C)=O)(NC(=O)CCC(C)(F)F)Cc2ccccc2C1 25769,CCCCCC(=O)NC1CCC(CNC(c2cc(-c3cccc(O)c3)on2)=O)C1 25770,c1(C(N(C(CN(C(c2c(C)cccn2)=O)C)C)C)=O)ccc(F)c2occc12 25771,c1(C(=O)NCC(CO)NC(c2cc(C)no2)=O)cc(C(C)=O)oc1C 25772,c1(NC(C2(CCC=C)CN(C(=O)CC3CCC(=O)N3)C2)=O)cncnc1OC 25773,C(CO)(C(=O)NCC1CC1C1CC1)NC(C(F)=CCC)=O 25774,N1(C(c2[nH]n(C)c(=O)n2)=O)CCCC1C1CCCCN1C(=O)C(N)=O 25775,CCS(=O)CC(=O)NCCCC(C)(C)NC(=O)C(C)NC(c1ccoc1)=O 25776,CC1CN(C(=O)C=CS(C)=O)CCCN1C(c1cncc2ccsc12)=O 25777,CN1CCN(c2nccc(Cc3ccccc3)n2)CC1(C)C 25778,c1(C(N2CC(C(C)NC(c3c(C)ncn3O)=O)C2)=O)cccc2[nH]ccc12 25779,C(C)(c1ccc(F)cc1F)=CC(=O)NC(CC)CNC(C1CCS(=O)(=O)N1C)=O 25780,C12CCN(CC1)Cc1cn(nn1)CC2.c1(C(=O)OC)ccc(C2CC2(Cl)Cl)cc1 25781,Cc1cc(C2CCCO2)cc(C(=O)NC(CNC(C23CC(C2)C3)=O)CC(C)C)n1 25782,c1(CCC)cc(C(=O)NC2CC23CC(NC(c2nn(C)cc2C)=O)C3)n(C)n1 25783,c1(C(=O)NC2C(NC(=O)C=C3CCC3)C2)[nH]n(-c2ccccc2)c(=O)c1Br 25784,N1(C(C2CC(=O)N(Cc3ccccc3Cl)C2)=O)C2CCC1CC1(C2)CC1(F)F 25785,c1(CC(=O)NC2C(NC(Cc3nnc(C)s3)=O)CCCC2)cccc(O)c1F 25786,CCCS(=O)(=O)CC(=O)N(CC)CC1CCN(C(C2CC2CF)=O)CC1 25787,CC(CS(C)=O)C(=O)NCCOCCNC(c1cc(N)cc(O)c1)=O 25788,c1(C(=O)NC23C(CN(C(CSC)=O)C2)C3)c(Cl)oc2ccccc12 25789,C(=O)(CCCCCC#N)NCc1c(CN2CC(C)OC(C)C2)cccc1 25790,C(=O)(C1=C(Cl)CCOC1)N1CCC(C(=O)NCC(CC)C(C)(F)F)C1 25791,C(=O)(CC(C)(C)O)NCC(C)NC(C1(n2cncn2)CC1)=O 25792,CC1(C)CCc2ccc(C(N3CCC(NC(C4CC4C(N)=O)=O)C3)=O)cc2O1 25793,N1(C(CNC(CCC)=O)=O)CCN(C(c2cc(Br)sc2C)=O)C(C)C1 25794,C1(C(C(C)C)NC(=O)C(Cl)=CCl)CN(C(=O)C=Cc2cn(C)cn2)CCO1 25795,n1(CCC(=O)NCC(C2CC2)NC(=O)CC2CCCCC2)cnc([N+](=O)[O-])c1 25796,C1(C(C)NC(C(C)(C)OC)=O)CCCN(C(=O)CC(C)(F)F)C1 25797,C=CCCC(C(=O)NC(C(N)=O)C1CCCC1)NC(c1cc(Cl)n[nH]1)=O 25798,Cc1cc(-c2cn(CC3C(C)CCN3C(C3CC=CCO3)=O)nn2)c(Cl)cc1F 25799,c1(C(N2CC(CCNC(C(CCCC)C)=O)C(C)C2)=O)nccn2cc(C)nc12 25800,N1(C(N2CCC(Cc3cc(C(=O)OC)[nH]c3)CC2)=O)CC2C3CCC(C3)C12 25801,C1(C2CN(c3nnc(C)s3)C2)CN(C(c2coc(-c3ccccc3)n2)=O)CCO1 25802,N1(C(c2sc(CCC)c(CC)c2)=O)CC2(C1)CN(C(=O)C(C)(C)CCC)C2 25803,C1(C)(NC(COC2CCN(C(c3cccc(CC)n3)=O)C2)=O)CCCCC1C 25804,C1(NC(C(=Cc2ccncc2)C)=O)CS(=O)(=O)CC1NC(c1cnc[nH]1)=O 25805,Nc1ccc(C(=O)NC2CCC(CNC(C3CC4CCC(C3)O4)=O)CC2)cc1F 25806,C1(NC(c2c(CC)cno2)=O)C(C)CCN(C(c2nc(C)c(C)nc2C)=O)C1C 25807,CS(=O)(=O)CC(=O)NC1CCOC(CNC(=O)CCc2ncc[nH]2)C1 25808,N1(C(CC(CC)(F)F)=O)Cc2nccn2CC(NC(=O)C(F)C(C)C)C1 25809,c1(C(=O)NC2CCCCCN(C(CC=C)=O)C2)n[nH]c2cc(Br)ccc12 25810,Cn1cnc(I)c1C(N1CCC(c2ccncc2)CC1)C(=O)NC1CCOC1 25811,Cc1cncc(C=CC(=O)NC2(CNC(C3CC3C(C)C)=O)CCC2)c1 25812,Cc1[nH]nc(C(=O)N(C)CC2CN(C(c3ocnc3C(F)(F)F)=O)CCO2)c1F 25813,C(=O)(CCCC(C)O)N(CC(C)(C)Nc1nccc(CC(=O)OC)n1)C 25814,N1(C(c2cc(COC)no2)=O)CC2CN(C(=O)C(C)CS(C)(=O)=O)CC2C1 25815,c1(C(=O)NCC2CC(C)(C)CN2C(=O)Cn2cnc(=N)[nH]2)cc2c[nH]cnc-2n1 25816,Cc1c(C(N2CC(O)CC2CNC(=O)CC2CN(C)CC2O)=O)sc2nccn12 25817,c1(CNC(C2C(C)C2)=O)cc(C(N2CCCC2c2nc[nH]n2)=O)n[nH]1 25818,N1(C(CCOC)=O)CCC(NC(c2cc(C(C)C)n(C)n2)=O)C1c1ccccc1 25819,N1(C(COC2(C)CCC2)=O)CC2CC1C2NC(=O)C(C)(C)C1CCCO1 25820,CC1CCn2cc(C(=O)NCC(CO)NC(c3c[nH]c(Br)c3)=O)nc2C1 25821,N1(C(C(C)CF)=O)CC=CC(NC(c2cnn(C(C)(C)C)c2Cl)=O)C1 25822,CCCCS(=O)(=O)CC(=O)NCCCN1CCN(C(=O)C2=CS(=O)CCC2)CC1 25823,C#Cc1ccc(C(=O)NC(C)CN(C)C(c2cscn2)=O)c(OC)c1 25824,C1(CNC(C2CN(C(N)=O)C2)=O)CN(C(c2cc(F)ccc2Cl)=O)CC1(F)F 25825,C1(C(=O)NC(CSC)(C)C)C2CC2CN1C(=O)C(C)OCC(C)C 25826,C1(NC(c2ccn(C)n2)=O)CN(C(=O)CC2CC(C(C)(C)C)=NO2)CC2(CC2)C1 25827,N(C1COc2ccccc21)C(c1[nH]c(=NCc2cnc(CCC)s2)sc1)=O 25828,c1(C(c2nnnn2C2CC2)NC2C(CCOC)C2)cccc(C(C)C)c1 25829,N1(C(c2ccc(=NC)[nH]c2)=O)C2CCC1C1CC1(NC(=O)CC(C)C(F)F)C2 25830,N1(C(=O)NC(Cc2c(C)ncs2)C)CCCC(C(=O)OC(C)(C)C)C1 25831,C(C)(C)(C#CCCC)NC(CCN(CC#C)C(C1CCCC(O)C1)=O)=O 25832,C(C)(CCCCNC(C12CC(C)(C1)C2)=O)NC(c1c(C)ocn1)=O 25833,C1(COC)CN(C(=O)CCN2CCCC2)CCN1C(c1sncc1C)=O 25834,c1(NC(C2N(C(c3ccc(C)cn3)=O)CC2)=O)cc(F)c(O)cc1C 25835,Cc1ccccc1C1(C(N2CC(O)(CNC(c3nn[nH]c3Cl)=O)C2)=O)CCC1 25836,C1(C(N2CC(CNC(CCOCC#C)=O)(OC)C2)=O)CCOC(CC)C1 25837,N1(C(CCCS(C)(=O)=O)=O)CCC2(CC1)CCN(c1ncnc(=N)[nH]1)C2 25838,c1(C(=O)NC(C2CN(C(=O)CCCCC(N)=O)CCO2)C)cc(Cl)c(F)cc1F 25839,c1(SC)ccn2c(-c3ccc(Cl)cc3Cl)nnc2c1 25840,c1(C(=O)NC2CCCCN(C(CC(=C=C)C)=O)C2)c(F)cc(O)cc1F 25841,c1(C(=O)NCCCN(C(=O)C2=CC(C)(C)C2)C(C)C)ccc2c(c1)C(=O)NC2=O 25842,c1(C(=O)NC2CCN(CCC(N)=O)CC2)cc(Cl)cc(F)c1Br 25843,N1(C(CCNC2C3(CC(N)C3)C2)=O)CC(=O)Nc2ccccc21 25844,c1(CC)nn(C)cc1C(=O)NCC=C1CCN(C(C2(OC)CCCC2)=O)CC1 25845,c1(OC)ccc(F)c(C(=O)N(C2CCN(C(=O)C(C)C3CC3)C2)C)c1OC 25846,C1(NC(CCc2c(C)noc2)=O)CC(C)N(c2nc(-c3ccccc3)ns2)C1 25847,N1(C(C2C(OC)(OC)CC2)=O)CCCCC(NC(c2sccc2CN(C)C)=O)C1 25848,S(=O)(=O)(c1ccccc1F)NCC(=O)NC(CNC(CCCCNC(C)=O)=O)C 25849,c1(C(=O)NC(CNC(C(C)C2CC2)=O)(C)C2CCC2)cc(-c2cnn(C)c2)on1 25850,c1(C(=O)NCC2N(C(c3cc(C)n(C)c3C)=O)CC=C2)ccc(S(N)(=O)=O)cc1 25851,C12CN(CC1(C)C)C2=O.c1(C(N(C(CC)C)C)=O)ccc(O)nc1Cl 25852,C1(NC(C2CCC(C(=O)OC)CC2)=O)CCN(C(C2CCC(=O)N2)=O)CC1CO 25853,C(C(C)(C)C(C)(C)O)NC(C1N(C(C(C)=C(CC)C)=O)CCC=C1)=O 25854,N1(C(c2nnn(C)n2)=O)C2CCC1CC(NC(=O)CCC1CC1)C2 25855,C(=O)(C1CCc2nccn21)NCCCCCCC(=O)N1CC2CC(N(C)C)C2C1 25856,C12(CNC(C(=O)Nc3ccc(-c4cc(C)ncc4)cc3)=O)COC(C1)C(N)C2 25857,C1(CNC(c2cc(C(C)C)no2)=O)CC(C)CN(C(=O)C(CO)N(C)C)C1 25858,c1(NC(c2ccccc2-c2co[nH]c2=O)=O)c(O)ccnc1F 25859,c1(C(N2CC(C(C)NC(=O)C(C3(O)CCCC3)F)OCC2)=O)cc2occc2s1 25860,C(=O)(C(CO)C(C)(C)C)N(C(CNC(CCCC=C)=O)C1CC1)C 25861,c1(OC)ccc(C(N2CC(F)CC2C(=O)Nc2ccnc(Br)c2)=O)c(Br)n1 25862,C=CC(CCC)CC(=O)NCC1(O)CC(NC(=O)Cn2ccccc2=O)C1 25863,C(C(O)CC(=O)N(C)CC1(O)CCC1)NC(CNC(CC(C)C)=O)=O 25864,N#Cc1cnccc1N1CCCCC1NC(=O)CCOCCOCCCO 25865,c1(C(=O)NCC2C(C)CN2C(=O)CC2OCCC2(C)C)cc2ccccn2c1 25866,c1(C(=O)OC)c[nH]c(=NC(CNC(=O)Cc2cnnn2C)C(C)C)cn1 25867,C(=O)(C1CCCn2nccc21)NC(CNC(CCC=C=C)=O)C(C)(C)C 25868,N1(C(=O)CCc2cc(F)ccn2)CCC2C1CCN2C(=O)CCC12CC(F)(C1)C2 25869,c1(NC(c2c(SC)cc(Br)cc2)=O)ccc(S(=O)(=O)N2CCOCC2)cc1 25870,CC(C)CC(CNC(=O)C1=C(Cl)CCC1)C(=O)NC1CCCC(O)CC1 25871,Cc1ccc2[nH]c(=NC(C)C3CCN(C(c4cnc(O)o4)=O)C3)sc2n1 25872,c1(CNC(C(C)(C)C2CCC2)=O)cccc2c1CN(C(C1(C(C)(F)F)CC1)=O)C2 25873,N1(S(c2cc(C)c(Cl)s2)(=O)=O)CCCc2c(O)cccc21 25874,C(=O)(CS(=O)(=O)C(C)(C)C)N1CCCC(C)(NC(=O)CCC(=O)N2CCCC2)C1 25875,c1(CC)ccc(C)c(C(N2CCCCC2C(C)NC(c2nnc(C)s2)=O)=O)c1 25876,N1(C(C(C)OC(C)C)=O)CCN(CC(=O)Nc2scnc2Br)C(=O)C1 25877,Cc1ncc(CC(=O)NCC(C(C)C)NC(=O)C(C)CSC(F)(F)F)[nH]1 25878,c1(Cc2n(-c3cc(OC)ncc3)nc(C3CC3)n2)c(F)cccc1Br 25879,N1(CCCC(=O)N(CC(CC)NC(=O)C(N)=O)C)C(=O)c2ccccc2C1=O 25880,c1(NC(C2CCCN(C(C3CC3C3CC3)=O)CC2)=O)cc(Cl)ncc1[N+](=O)[O-] 25881,c1(C(N2C3C(NC(=O)Cc4ccns4)CC(C3)C2)=O)ncnc2c1CCCC2 25882,CCCC(C)(C)CC(=O)NCCC1(O)CN(C(c2ccsc2-n2cnnn2)=O)C1 25883,Cc1ccc2cc(C(=O)NC3CCCN(C(c4ccn(C)c4)=O)C3)nn2c1 25884,C1(OC)CN(C(=O)CC2(O)CCOCC2)CC1NC(C1(n2nccn2)CC1)=O 25885,c1(C(=O)NC2C(NC(CC(CC)C(C)C)=O)CC2)c[nH]c2cccc(Cl)c12 25886,CN1CC2C(NCC(=O)N=S(C)(C)=O)CCCN2C1=O 25887,c1(C(=O)NCC(CNC(C)=O)NC(=O)CO)sccc1SC 25888,c1(C(N(CC(CN(C)C)O)C)=O)sccc1C1CC1.c12cnn(c1)CNC2=O 25889,C1(NC(CN(C(=O)CC(C)n2cccc2)CCC)=O)CC12CCOCC2 25890,c1(NCC2CCC(=O)NC2)ccc(S(=O)(=O)NC(Cc2nccs2)CO)cn1 25891,c1(C(=O)NC(CCN(C(C(C)CC(N)=O)=O)C)C(C)(C)C)ccc2occc2c1 25892,CN1CC2CCC(NS(=O)(=O)Cc3ccc(-c4cccc(C(N)=O)c4)cc3)C2C1 25893,c1(C(C(=O)NCC(C)CN(C(=O)CCC2(C#N)CCC2)C)O)cnn(C)c1 25894,c1(C(=O)NC2CCCC(CNC(C(C)(F)F)=O)C2)ncc(C(N)=O)cc1Cl 25895,c1(CN(C(C)=O)CC2CCCN2C(=O)COCC2CC2)cccc(C)c1 25896,N1(C(c2ncc(OCC)nc2)=O)CC2CN(C(=O)CCc3cccc(C)n3)C2C1 25897,c1(C(=O)NC2CC(C)SC2)c(CNC(c2cc(=N)[nH][nH]2)=O)cnn1C 25898,CCCC#CC(C)(C)NC(c1oc(CNC(C2CCC2C(N)=O)=O)nc1C)=O 25899,C1(CN(C(C2(COC)CCOC2)=O)C)CCN(C(=O)CC(C)c2ccco2)CC1 25900,Brc1cc(I)c(CN2CCC(N3CCC3)CC2)s1 25901,n1(CC(N2C(CC(=O)NCc3ncc[nH]3)CC2)=O)ccc2ccccc12 25902,N1(C(Cc2cc(C)ncc2)=O)CC(CNC(=O)C(F)=CC2CC2)C(C)(C)C1 25903,c1(-c2nnc(C(O)CC(C)NCCC(F)(F)Cl)o2)ccc(SC)cc1 25904,Cc1nc(O)nc2ccc(C(=O)NCC3(NC(C4CC5CC5C4)=O)CCC3)cc12 25905,c1(OC)ccc(N2CCCCC2)cc1N1CCOC1=O.N12CCOC(C1)C2=O 25906,Cc1nnc(Cn2cc(C3CN(C(C4COC(=O)O4)=O)C3)nn2)o1 25907,CC(Cc1cccs1)N=c1[nH]c(N(C)Cc2cccnc2O)nc2c1SCC2 25908,Cc1cccc(C(=O)NC2CC(O)CN(C(=O)CN3CCC(C)(C)CC3)C2)c1C 25909,N1(C(c2n(C)ccn2)=O)CC2(CC(NC(C3(C(F)(F)F)CC=CC3)=O)CO2)C1 25910,c1(C(N2C(C)CCC(NC(Cc3c(C)nc(S)s3)=O)C2)=O)cc2c(ccn2C)[nH]1 25911,c1(N2CCCC(NCc3c(C)noc3)(CO)C2)nc(C2CC2)nc2ccccc12 25912,c1(C(=O)NC2CCC(C(=O)NC(c3cn[nH]c3)C)C2)ccccc1C1CC1 25913,C(CC(C)(C)C)(C(=O)NCCC1CCCN1C(c1cc(C)[nH]c1C)=O)OC 25914,c1(OC(N2CCC(C(=O)O)C2)=O)ccccc1OCC1CCCO1 25915,C(C(C)(F)C(C)(C)F)NC(CCCNC(c1n(CC)c(O)nc1)=O)=O 25916,C1(CC=C)(NC(c2cocn2)=O)CC2CCC(C1)N2C(C1CC(=O)N1)=O 25917,N1(Cc2ccc(C#C)s2)CCCN(C(c2ccnc(C(C)(C)C)c2)=O)CC1 25918,N(C1CN(C(c2cncn2C2CC2)=O)Cc2ccccc21)C(CSCC(C)C)=O 25919,C(=O)(C(C(C)(C)C)NC(C1CN2CCN1CC2)=O)N(C)Cc1cocn1 25920,C(C(C)(C)C(=O)N1CC(O)(CNC(c2nnn(C)c2C(F)F)=O)C1)SC 25921,c1(OC)cncc(C=CC(=O)NC2(CN(C(=O)CN3CCCC3C)C)CC2)c1 25922,Cc1cc(C(=O)NC2CCCC2NC(c2ccnc(O)c2)=O)nc(O)n1 25923,c1(C(=O)NCC(C)(C)NC(=O)C(F)F)ccc(OC(F)(F)F)nc1.c1(O)ccccc1 25924,c1(CN2CCC(F)(C(=O)NCCCC)C2)cc(C(C)=O)ccc1OCC 25925,c1(C(N2CC(C(=O)Nc3cc(Br)cc(Br)c3)C(O)CC2)=O)cccc2c1CCC2 25926,CCC(CC(=O)NCC(C)CN(C(=O)Cc1ccn(C)n1)C)C(F)F 25927,C12CCCN(C1)C(C)C(=O)N2.C(C1CCCC1)=C(C)C(=O)Nc1cnn(C(C)C)c1 25928,C(C1=CCN(C(C2CCC(F)CC2)=O)CC1)NC(C(C)C1CCCO1)=O 25929,C(=O)(CCCCCCCCC1CC1)NCC(CC)NC(=O)Cc1cc(CC)no1 25930,c1(OC)cc(OC)c2c(c1)CCN(C(=O)CC1CCCC(C)C1)C2 25931,c1(C(N(CCNC(C2N(CCCC)CCCC2)=O)CCOC)=O)ncc(N)cc1Cl 25932,CCCCCCCCCCCCN(C(=O)CC1CCN1C(=O)OC(C)(C)C)C 25933,c1(C(N(C2C(C)CCC2)CCc2ccccc2)=O)cn2c(n1)CCCC2 25934,CC(C)S(=O)(=O)CC(=O)NCCC1CN(C(C2(C)CCOC2)=O)CC1C 25935,c1(CC(=O)NC2CN(C(C(F)=CCC)=O)C2)ccc2c(c1)CCOC2 25936,C1(CNC(Cc2nc(C(C)C)sc2)=O)CN(C(=O)C=CS(C)=O)CC(C)(C)O1 25937,c1(C(=O)NCCC(=O)NCCNc2nnco2)cccc(=O)o1 25938,C1(C(N2C(CN(C(c3c(COC)cco3)=O)C)COCC2)=O)CC2(C1)OCCO2 25939,c1(C(N2CCC(N(C(=O)CCc3cccnc3C)CC)C2)=O)cc(C)ccc1N 25940,C12(CNC(C3N(CC)CC3)=O)CCC(NC(=O)C(n3cc(Cl)cn3)C)(CO1)C2 25941,C1(C(=O)NOCC(F)(F)F)C2CC3C(C2NC(C2CCCOC2)=O)C13 25942,c1(C(N2C(C)C(NC(=O)C(N)=O)CCC2)=O)cc2c(nc1O)CCC(C(C)C)C2 25943,CCC(C)(C(=O)N1CCC(C)N(C(c2cc(N)c(F)cc2F)=O)CC1)C(F)F 25944,C(=O)(CS(=O)(=O)CC(=O)NCC1CCN1C(=O)Cn1nc(C)nc1C)OC 25945,C(CN=C(NCC1CCCC(C)C1)NC(C)C)c1c(C)nccn1 25946,CC1(C)CN(C(=O)C=Cc2cncs2)CC(CNC(=O)C(F)(F)CC2CC2)O1 25947,N1(C(CC2(C)CCOCC2)=O)CC2CC(NC(=O)CCN3CCOCC3)C(C2)C1 25948,Cn1cnc2c1CN(C(=O)Cn1cc(CNC(c3cc(O)nc(O)n3)=O)nn1)CC2 25949,Cc1nc[nH]c1CC(=O)NCCC1CCC1NC(=O)Cc1csc(NC(N)=O)n1 25950,C(=O)(C(=O)N=c1cc(C)o[nH]1)NCC1C(F)(F)CCN(C(CSCCC)=O)C1 25951,c1(C(=O)NCCC(CCC)C)cc(C(N)=O)cc([N+](=O)[O-])c1 25952,Cc1nn2ccccc2c1C(=O)NC(CNC(C1(N(C)C)CC1)=O)CC(F)(F)F 25953,N1(C(c2cc(OC)no2)=O)CC(NC(=O)Cn2cnc(C#N)n2)C2CCCC2C1 25954,C(=O)(C(CNC(=O)COC(C)C)CC1CCCC1)N(C(C#C)C)C1CC1 25955,N1(C(c2[nH]cc(C(C)=O)c2)=O)CC(NC(c2csc(CO)n2)=O)CC1(C)C 25956,c1(OC)ccccc1C(CNC(=O)Cc1ccc(F)cc1)NC(=O)CO 25957,C12(NC(=O)CC3(CO)CC3)CCCC1N(C(=O)COCC1CCC1)CCC2 25958,Cc1nc(NCCNC(=O)CC2NC(=O)NC2=O)c(C)c(Cl)n1 25959,C1(C(C)(C)O)(CNC(c2ccnn2CC(F)F)=O)CN(C(c2ccccc2)=O)C1 25960,c1(C(=O)Nc2c(N(C)C)nccc2)cc(N)ccc1S(C)(=O)=O 25961,c1(CCC(=O)NC2(C)CC(NC(CC3C(C)OCC3)=O)C2)ccc(C#N)cc1 25962,c1(C(C(N2CCC(CN(C(c3c(CC)ccs3)=O)CC)C2)=O)F)ccc(F)cc1 25963,C1(C(N(CCCNC(C2CC(F)(CO)C2)=O)C)=O)CCCCC1C1CC1 25964,c1(NC(=O)OC(C)(C)C)coc(CCC(COC)C(=O)NC(=O)N)n1.C(C)(C)C 25965,C1(C(N(CC(=C)C)CC)=O)CCN(C(c2cnn(C)c2Cl)=O)C1(C)C 25966,CC(C)S(=O)(=O)C1CCN(C(CCCCCl)c2nnnn2CC2CCCO2)CC1 25967,C1(CCNC(C2CCN2C2CCCC2)=O)CSCCN1C(C1CCC(F)(F)C1)=O 25968,C1(NC(C2(C#C)CCN(C(c3cc(CC)nn3C)=O)C2)=O)CC2C(O)C(O)CC12 25969,c1(C(N2C(CNC(C3COC4(CCC4)C3)=O)COCC2)=O)coc2c1COC2 25970,c1(C(C(=O)NCC(C)(C)OCCNC(Cc2ccc(C)s2)=O)C)cccc(F)c1 25971,N1(C(=O)C=Cc2ccc[nH]2)CCC2(CCN(C(c3ccc4c(c3)CCC4)=O)C2)C1 25972,N1(C(c2scc(CNC(C3C(OC(C)=O)C3)=O)c2)=O)CCCC2CC12 25973,N1(C(c2c(OC)cccn2)=O)CCC2CN(C(c3ccnc(C)c3N)=O)C(C)C12 25974,C(C)(C(=O)NOC(C)C(=O)OC)NC(c1c(CCC)[nH]cc1)=O 25975,C=CCCCCCCCC(=O)NC1CC1NC(=O)CCSc1nccn1C 25976,C1(C)(C(=O)NC2C(NC(C(C)N3CCCC3)=O)CC2)CCCN(C)C1 25977,C1(NC(C(C(C)C)N2CCCC2)=O)CN(C(=O)C=CBr)CC1C1CC1 25978,C(=O)(C(C)(C)C(F)F)NC(C(C(C)C)Nc1ncc(F)cn1)C 25979,c1(NCCC2CCN(C(N(C)C)=O)C2)cc(=NCc2ccc(O)nc2)[nH]cn1 25980,C1(C#N)(C(N2CCC(C)(C(=O)NC3CC3c3ccsc3)C2)=O)CC(F)(F)C1 25981,c1(C(C)=O)cnn(C)c1.C1(NC(=O)N)CCCC1.C1CCN(C)C(=O)CNC(=O)O1.C=N 25982,c1(C(C(=O)NCSc2ccccc2)N(CCC(N)=O)CC)ccc2cnn(C)c2c1 25983,C12(C(N3CCCCC3c3ccc(C(F)(F)F)nn3)=O)CC(CO)(C1)OC21COC1 25984,N1(C(C(C)(C)C)=O)CC2(C1)SCCC2N=c1[nH]ccnc1C(F)(F)F 25985,c1(C(=O)NCCC(C)N(C(C2C(C=C)C2)=O)C)cc(F)cc2nn[nH]c12 25986,C(C1=NOC2CN(C(=O)CC3CC3)CC12)NC(c1cc(CC)c(C)cc1)=O 25987,C=CC(CC(=O)NCC(C)(C)OCCNC(=O)Cn1cncn1)c1ccco1 25988,N1(C(C(CSC)C)=O)CCC(NC(=O)COc2ccc(F)cc2F)C12CCC2 25989,c1(C(C(C)(C)C)SC)nc(-c2cncnc2)nn1-c1ccccc1 25990,C1(NC(c2cnc(CC)o2)=O)CCCN(C(C2(c3ccno3)CC2)=O)CC1F 25991,Cc1nc(NC(C2CCCN2C(c2ccncc2O)=O)=O)cnc1Cl 25992,C1(C(CNC(c2c(C)onc2)=O)(C)O)CCN(C(=O)C(C)OCC(F)(F)F)CC1 25993,N1(C(C(CCNC(C(CC)NC(C)=O)=O)O)=O)CC(O)CC12CCOC2 25994,N1(C(CC2(C)CCOC2)=O)CC2CC1CC2CC(=O)NCC1CCCOC1 25995,C1(NC(COC)C(=O)OC)CN(C(=O)OC(C)(C)C)CC2(CC2)C1 25996,O=C(N=c1ccn(CC(=O)NCCCC(F)(F)F)[nH]1)C(O)CN1CCCCC1 25997,N1(C(c2ccc(CC)[nH]2)=O)CC(NC(=O)CCS(N)(=O)=O)CC12CCOCC2 25998,c1(C(=O)NCCCC(C)(C)NC(=O)CC2CCOCC2)ccc2nonc2c1 25999,c1(N(C)CC2CC2(F)F)nc(N2CCC=C(F)C2)c2c(n1)CCCC2 26000,C(=O)(CC(CC1CC1)NC(=O)C(C)OCC1CC1)N1C(C=C)CC1 26001,C(=O)(C(O)CCCNC(C1CC2CC2C1)=O)N(CC)Cc1ccccn1 26002,C(CN=c1[nH]c(=NC2CC2C(C)(C)C)c2ccccc2[nH]1)c1c(C)nc(C)s1 26003,N1(C(=O)NC2C(C(C)(C)C)C2)CC=C(CO)CC1.c12c[nH]nc1C2 26004,C1(NC(C(CC)NC(C)=O)=O)CN(C(c2cc[nH]c(=NC)c2)=O)CC1N=[N+]=[N-] 26005,c1(OCc2c(-c3n(CC(C)C)ncc3)cnn2C)ccc(Cl)cc1C(N)=O 26006,CN1CCCCC(C(N2CCCC(NC(c3cccnc3N)=O)C2)=O)C1=O 26007,CCCC(CC(C)C)C(=O)NOC(CC(C)C)C(N1CCC(C)(C2CC2)C1)=O 26008,CCC(C)C(=O)NNC(=O)c1nn(C)cc1-c1ccc(C(F)(F)F)c(C)c1 26009,N1(C(C2C(CC)OCC2)=O)CC(OC)C(NC(=O)CC23CCCC2C3)C1 26010,c1(CC(C(=O)N(CCCN(C)C(c2ocnc2C2CC2)=O)C)O)ccccc1Cl 26011,N1(C(=O)CC2CC3(CCC3)CO2)CC2CC1CCC2NC(=O)C(F)(F)C(F)F 26012,C=CC1CCCN1C(C1C(NC(=O)CSC(C)(C)C)CC1)=O 26013,c1(C(N(C(C)CNC(=O)CC(C)N(C)C)C)=O)ccc2c(c1)COC2=O 26014,N1(CCN(C)C(c2ccc(NCC3(O)CCCCC3)cc2)=O)CC2C(CO)C2C1 26015,c1(NCCC(C)NC(=O)C(C)S(N)(=O)=O)cc(C(F)(F)F)ncc1[N+](=O)[O-] 26016,c1(C(=O)NC2CN(C(C(C(=O)N(C)C)(C)C)=O)C3C2C3)cc2c(Cl)nccc2s1 26017,Cc1cccnc1C(N1CC(NC(c2csc(CSC3CCC3)n2)=O)C1)=O 26018,c1(SCCOC(C2CC(C)N(C(C(C)(C)C)=O)CC2)=O)ccccc1[N+](=O)[O-] 26019,C(=O)(C(CC(C)C)ONC(C1CC2C=CC1CC2)=O)NCCC(CC)O 26020,[N-]=[N+]=NC1CCCCC1NC(=O)C(c1ccco1)NC(C1CC(F)(F)C1)=O 26021,CCCCCC(O)CC(=O)NCC1CC(NC(=O)C2=CCCC2(C)C)C1 26022,C1(C(=O)NC2C(SC)C2)(CCO)CN(C(=O)COCCCN=[N+]=[N-])C1 26023,c1(C(C(=O)NC2C(NC(C(c3ccc(Cl)cc3)C)=O)C2)(C)C)ccc(O)cc1 26024,c1(N(CC(C)C(C)(C)C)C)nc(N2CCCC(C)(F)C2)nc2ccc(Cl)cc12 26025,C1(C(N2CC(CCCCC)C2)=O)CCCC(NC(C2(F)CC=CCC2)=O)CC1 26026,c1(CC)ccc(F)cc1C(=O)NCC12CC1CN(C(C1(CC)CC1)=O)C2 26027,CN1CC2CCC(C1)N2c1nc(C(=O)NCc2c(F)cc(Cl)cc2Cl)cnc1N 26028,CC1=C(C(=O)N2CCC(NC(c3cnn(CC(F)F)n3)=O)C(C)(C)C2)CCCO1 26029,N1(C(Cn2c(C)cc(C)n2)=O)CCOC2CN(C(=O)CN3CCCC3)CC12 26030,c1(C(=O)NC(CC)(C)CNC(C2(CCF)CC2)=O)cc(Br)ccc1F 26031,c1(C(=O)NCCN(C(CCC#C)=O)CCc2ccccc2)[nH]c(COC)nc1C 26032,C(=O)(CC(C)(C)CC)N1CC(NC(C2CC(C(F)F)(OC)C2)=O)C1.c1(C)ccccc1 26033,c1(C(=O)NCC(CC(C)C)N2CCOCC2)ncc(S(=O)(=O)N(C)C)s1 26034,N1(C(c2c(Cl)ncc(C)c2)=O)CCCC(NC(C2CC(C)(F)C2)=O)CC1 26035,C1(n2cccn2)(CNC(C(C)N2CCC2)=O)CCN(C(=O)C(F)=CCCF)CC1 26036,Cc1cc(C(=O)NC(C)CNC(c2ccncn2)=O)sn1 26037,N1(C(c2cc(C(=O)OCC)cc(Br)c2)C(=O)NC)CCOCC12CCC2 26038,c1(NC(C2(F)CN(C(c3ccc(C)c(O)c3)=O)C2)=O)c(Br)cccc1[N+](=O)[O-] 26039,N1(c2ccnc(C(C)(C)C)n2)CCN(C(c2cc(Cl)cnc2O)=O)C(C#N)C1 26040,c1(C(=O)OC)cc(C(N2CCCC(C)C2CNC(C)=O)=O)cc(Br)c1 26041,N1(C(c2cncc(C)c2Cl)=O)CCCC(C2CC2NC(C2(N(C)C)CC2)=O)C1 26042,N1(C(CN2C(=O)CCC2)=O)C2CN(c3ncccn3)CC12 26043,N1(C(c2cn(CCNC(c3cc(C#N)[nH]c3)=O)nn2)=O)CC(O)C(C2CC2)C1 26044,N1(C(CCC#C)=O)CC2(CCCCN(C(=O)C(C)C3CCCO3)C2)C1 26045,N1(C(C(C)=C2CCC2)=O)CCCCC(NC(=O)C(CN(C)C)C(C)C)C1 26046,Cc1cnc(C=CC(=O)NC2COCC2NC(=O)CC2COCC2O)[nH]1 26047,c1(OC)cc(C)ccc1C(=O)NCCCC1CCN(C(=O)CC=CC(C)(C)C)C1 26048,N1(C(CC2C(OC)CC2)=O)CCN(C(c2cocn2)=O)C(c2cn[nH]c2)C1 26049,C1(CNC(c2n(CC)ccn2)=O)CCC2(CN(C(c3csc(Cl)n3)=O)C2)O1 26050,C(=O)(C1CCc2c[nH]nc21)NC1(C(=O)NC(C2CCCCC2)C)CSC1 26051,N1(C(CCC#CC)=O)CCCC(CC(=O)NC(C2CCOC2)CO)CC1 26052,c1(C(C(=O)NCC2N(C(C)=O)CCCC2)=O)cc(S(N)(=O)=O)cn1C 26053,Cc1[nH]nc(C(=O)NCC2CCCN(C(C3CC3C)=O)C2)c1C 26054,C1(NC(CC(CC)N(C(=O)CC(C)C(F)(F)F)C)=O)CCCC(C2CC2)C1 26055,c1(C(=O)NCCCCN(C)C(C2CC2c2cccs2)=O)c[nH]nc1C(C)(F)F 26056,N1(C(Cc2cnc(C)o2)=O)CCCC2(NC(=O)CSc3nccn3C)CC2C1 26057,c1(OCC)nc(C(N2CC(CN(C)C(c3ccc(CO)o3)=O)C2)=O)co1 26058,N1(C(Cn2c(N)cc(C)n2)=O)CCCC(N(C)C(c2ccccc2O)=O)CC1 26059,c1(C(C)C(=O)NCC2(CNC(=O)CC3CC(F)C3)CC2)ccc(F)c(Cl)c1 26060,c1(-c2ccc(CC)cc2C)ccc2oc(C(=O)NC(CC)C(C)O)cc2c1 26061,c1(C(=O)NCC(CC)NC(C2(CF)CCC2)=O)nocc1C(C)(C)C 26062,c1(NC(c2c(OC)cncc2)C)ccc(S(=O)(=O)NCC2C3CCCOC23)cn1 26063,c1(CC)[nH]nc(C(=O)NC(CN(C(=O)C(C)(F)F)C)CC)c1Cl 26064,N1(C(c2c(C)occ2)=O)CCN(C(c2csnc2Cl)=O)CC1CF 26065,C1(CNC(C2N(C=O)CCC2)=O)CCCN(C(c2cnc(C(F)F)nc2)=O)CC1 26066,c1(C(=O)NC(C(C(C)C)C)CNC(=O)C2=CCOCC2)c(F)ccc2occc12 26067,O=S(=O)(c1ccc(N2CC3CC3(CO)C2)cc1Br)NCc1cn2ccccc2n1 26068,CC(C)(C#CC(=O)NCC1CC1[N+](=O)[O-])CNC(=O)CN1CC(=O)NC1=O 26069,C1(CCC)CN(C(=O)CN2CC(C)(OC)C2)CCN1C(=O)C(O)CSC 26070,c1(C(N2CC(C(=O)NCc3cc(C)on3)OCC2)=O)cc(Cl)cnc1Cl 26071,C#CCC(C)(C(=O)N1CCC(CN(C)C)C1(C)C)NC(c1ccc(F)c(F)c1)=O 26072,C(=O)(C1=COCCO1)NC1C(CNC(c2cc(C(C)=O)cn2C)=O)C1 26073,N1(C(=O)NC2CCC(SCC)C2)CCC(COC)CC1 26074,C1(c2nnnn2C2CCCCC2)(NC(CCCC)(C)C)CCOCC1OC 26075,c1(CNC(C(CC)F)=O)c(F)cccc1[N+](=O)[O-] 26076,C1(C(N2C(CC)CCC2)=O)CC(C)(C)CN1C(=O)CCc1cscn1 26077,c1(N2CCCC(c3scc(C)n3)C2)ccc(Cl)cc1[N+](=O)[O-] 26078,C1(OCC)COCCC1NC(C1CCCOCC1)(c1nnnn1C1CCCC1)C 26079,c1(C(=O)NC2C(NC(CSC(C)(C)C)=O)CS(=O)(=O)C2)ccc2nncn2c1 26080,N1(C(C2CC(N(C(C(C)NC(CC)=O)=O)C)C2)=O)CCC(CO)C1(C)C 26081,C1(CN(C)C(c2ccc(F)s2)=O)CCN(C(C2(O)CCC2)=O)C1 26082,S(=O)(=O)(c1ccc2[nH]c(=NCc3ccsc3)ccc2c1)NCCCCN(C)C 26083,C(=O)(CP(C)(C)=O)NCC(CN(C(=O)C(C)O)CC)(C)C 26084,CCCCCCC(CC)C(=O)N(C1CCN(c2nccn3nnnc23)C1)CCC 26085,C(N=c1[nH]c(=NC(CCO)c2ccccc2F)[nH]c2c1SCC2)C1(C)CC1(F)F 26086,C1(CN(CCOC)C(c2ccc(C)o2)c2nnnn2C2(C)CC2)CCC(F)(F)CC1 26087,N1(C(c2cnc(C3CC3)nc2O)=O)CCC2C(CCCN2C(c2cnco2)=O)C1 26088,C(=O)(C1CCCc2nccn21)N(C)CC1OCCN(C(CC=C)=O)C1 26089,CCS(=O)CC(=O)NCCCOCCNC(=O)C(c1ncc(Cl)n1C)(F)F 26090,CCC(C)C(C)(O)CNC(C1CC(C)CN(C(=O)Cc2ccc[nH]2)C1)=O 26091,c1(SC)nc(=NCC2(OCc3ccccc3)CC3(CC(C(=O)O)C3)C2)cc(Cl)[nH]1 26092,CCCCCCCCC(=O)NC(C)CN(C(=O)Cn1cc(F)ccc1=O)CC 26093,C1(NC(C(=O)NC(C)C)=O)CCC(F)(CNC(c2cscc2Br)=O)C1 26094,C1(C(=O)NC2CC3(CN(C(c4c(C)noc4C)=O)C3)C2)CCCC1S(C)(=O)=O 26095,C1(CNC(C(C)C(C)(C)C)=O)N(C(c2cc(Cl)cc(F)c2N)=O)CCC1(C)C 26096,c1(OCCC(=O)NCCC2CCCN(C(=O)Cc3ccsn3)C2)ccc(Cl)cc1 26097,C1(C(=O)NCC2N(C(CC3CN(C)C3)=O)CC(F)C2)CC1C1CCCC1 26098,N1(C(c2cncc(C)c2C)=O)CC2CC(NC(=O)C(C)(C)CC(C)C)CC2C1 26099,N1(C(C(C)Cc2ccncc2)=O)CCCCC1CNC(=O)C(O)CC1CCCC1 26100,C(=O)(CC1=NN(C)C(=O)C1)NCC=CCNC(c1cc(OC)n(C)n1)=O 26101,N1(CC)CCC(n2nc(-c3cncc(F)c3)nc2COC)CC1 26102,C1(N(C(COC(C)=O)=O)C)CCCC(NC(=O)Cc2cnn(C)c2C)C1 26103,C1(CNC(C2CCN(CC(C)C)C2)=O)CC(C(=O)N(CCC#N)C(C)C)=NO1 26104,C1(CC(=O)NC2CC2NC(c2cncc(C(F)F)c2)=O)CN2CCN1CC2 26105,C1(NC(C23CC(OC)C2C3)=O)CC2CC(NC(c3cc(C(C)(C)C)no3)=O)C1C2 26106,[N-]=[N+]=NC1(C(=O)NCC(O)CF)CCN(C(=O)CC2CCOC2=O)C1 26107,S(=O)(=O)(CCC(F)(F)F)NC(C1CN(C(C2CC2(F)F)=O)CC1O)=O 26108,c1(C(COC(=O)CCN2Cc3ccccc3C2=O)=O)c(I)cc(F)c(Br)c1F 26109,C(CC(C)C=O)OC.C(CC(C)(C)OC)OC(CO)C 26110,C12(CC=C)CCC(C1)CNCC(C)(C1CC1)NC(=O)C2.c1(C(=O)OC)nc[nH]n1 26111,N1(C(CC2(C)CCN2C(=O)CCC2CC(F)(F)C2)=O)CCOC(C)(CO)C1 26112,C1(C(=O)NCc2cn(CC#C)nc2)C2CCC(C2)C1NC(c1ccc(CO)o1)=O 26113,N1(C(c2cc(C(N)=O)oc2)=O)CC2CC(NC(c3cc4scnc4[nH]3)=O)C1C2 26114,N1(C(CC2(NC(c3c(CC)noc3)=O)CCCCC2)=O)CCNC(=O)C1CC 26115,C1(NC(COC2C(C)CCCC2)=O)CCN(C(=O)CS(C)(=O)=O)CC1O 26116,C1(NC(C(CC)C)=O)CCC2(CC1)CN(C(c1cscc1Cl)=O)CCO2 26117,C(CC(C)NC(=O)CC1CSC1)N(C(=O)CCC1CCCO1)CC 26118,C(c1cc(F)c(F)c(F)c1)=CC(=O)NC(C)C(C)NC(c1ccc(Cl)cn1)=O 26119,c1(C(N(CCCNC(=O)CN2CCOCC2=O)C(C)C)=O)cc2ccsc2n1C 26120,c1(C(C)N(C2CS(=O)(=O)C2)C(=O)C2CC2)cccc(F)c1 26121,CC(N=[N+]=[N-])C(=O)N(CCC(=O)NC1CCN(C)C1=O)C1CC1 26122,C1(NC(c2c(C)nc(CCC)s2)=O)CC2(CCN(C(=O)CSCC#N)C2)C1 26123,Cc1cccc(C(=O)NCC2(CNC(=O)C=CC3CCC3)CCCC2)c1[N+](=O)[O-] 26124,N1(C(C2N(C(C)=O)CC(O)C2)=O)CCN(C(=O)C(F)(F)C(C)O)CC1C1CC1 26125,c1(C(=O)NC2CCN(C(c3nc(C)oc3)=O)C2C2CC2)ccc2c(c1)CCCC2 26126,C1(NC(C2CC(=C)C2)=O)CCCCC1CNC(=O)CCC1(C)CC1 26127,Cc1ccc(CC(=O)NC(CNC(C2CC(n3ccnc3)C2)=O)C2CC2)cc1C 26128,c1(C(C(=O)NC(C(=O)OC)C)N(C)Cc2cscc2C)cccc(OC(F)F)c1 26129,C1(C(=O)OC)CC(NC(=O)COc2ccccc2)CN(C(=O)C(C)OC)C1 26130,CCC(C)CCC(=O)NCCOC1CN(C(=O)CCCc2ccc(C)s2)C1 26131,c1(C(N2C(CCNC(C3CCO3)=O)CCC2)=O)csc2ccc(F)cc12 26132,N1(C(c2c[nH]c(=NC)s2)=O)CC(NC(=O)C(Br)=C(C)C)CC(C)(C)C1 26133,c1(C(=O)NCC2C3N(C(C4CC(OC)C4)=O)C(CC3)C2)c(Cl)c([N+](=O)[O-])nn1C 26134,CCC(CCC(=O)N(CC(C1CCC1)OC)C)NC(c1ccc(F)c(O)c1)=O 26135,C1(C)(CNC(C2C(CNC(c3cc(COC)no3)=O)C2)=O)CNC(=O)O1 26136,c1(CC(=O)N(C)CCNC(C2(P(C)(C)=O)CC2)=O)ccc2c[nH]nc2c1 26137,c1(SC)c(C(=O)NC(C2CCOC2)CNC(=O)CN2CCCC2=O)cccc1F 26138,c1(CCNc2c(C)cc(C)n(C)c2=O)cccc2oc(C)nc12 26139,CCCCCC(=O)NCC(C1(O)CN(C(c2ncn(C)n2)=O)C1)(C)C 26140,c1(N2CCC(Oc3c(OCC(=C)C)cccc3)C2)nc(Cl)c(C#N)s1 26141,C1(NC(C(C)OC)=O)CCN(C(c2ccc(=O)n(C)c2)=O)C1(C)C 26142,C1(N(C(CC2CN(C(C(C)n3cccn3)=O)C2)=O)C)CCN(C2CC2)C1 26143,C1(C(=O)OCC)CCN(C(C2(CNC(C3CCCO3)=O)CC2)=O)C1 26144,c1(CNC(=NCC)NCC23COCC2C3(F)F)ccc(OC(C)(C)C)nc1OC 26145,C12(CC(=O)NCC3(CC(=O)NCC4(CO)C(C=C)C4)CC3)CCCN1CCC2 26146,C1(C)(CNC(c2ccc(C(C)C)cc2)=O)CCC(NC(C2CCC3CC23)=O)CC1 26147,c1(CCCC(=O)NCCC(C)NC(C2COCCO2)=O)ccc(F)c(F)c1 26148,CC1CCN(C(C2(N=[N+]=[N-])CCN(C(C3SCCS3)=O)C2)=O)CC1O 26149,C(C1CN(C(c2coc(CO)c2)=O)CC1C(=O)NOCCCOC)=CC 26150,CCCCC(CC)C(=O)NC1CN(C(c2cccc(C(N)=O)n2)=O)CC12CC2 26151,C1(C)(NC(CC(=C)C)=O)CCN(c2cc(Oc3ccccc3)ncn2)CC1 26152,C(=O)(CS(=O)(=O)C1CC1)NCC1N(C(C(C2CCOCC2)OCC)=O)CC=C1 26153,c1(OC)ccc(C(=O)N(CCC(C)NC(C2(C)CC2(C)C)=O)C)cc1S(N)(=O)=O 26154,N1(C(C2CC(C#C)(O)C2)=O)CC2(C1)C(NC(C1CCC(=O)N1C)=O)CCS2(=O)=O 26155,Cc1nc2c(NC(N3CCC(c4cc(F)ccc4F)CC3)=O)cccn2c1C 26156,N1(C(C(C(C)C)SC)=O)CC(C2CCCCN(C(=O)C(F)C(C)C(F)(F)F)C2)C1 26157,CON1CCC(C(N2CCCC2CC(=O)NC(C)CN(C)C(C)C)=O)CC1 26158,C1(CN(C)C(C2CN(C)C2)=O)C=CC(NC(=O)CC(Cl)Cl)C1 26159,c1(OC)cc2cc(c1)CNc1nc(oc1-c1ccncc1)CO2.c1cn[nH]c1 26160,CC1CCC(CNC(=O)COCC2CCCO2)CN1C(=O)C=Cc1nccs1 26161,Cc1sc(Cl)c(C(N2CCCC(C)(NC(=O)CCNC(C3CCC3)=O)C2)=O)c1C 26162,N1(C(CCc2cc(C)c(Cl)cc2)=O)CCN(CCOC(C)C)CC(C)(F)C1 26163,C1(CC(N2CC(c3ncc[nH]3)C2)=O)CN(C(=O)C=CC2CCC2)CC12CC2 26164,C(=O)(CC1=NNC(=O)C1)NC1C(CC)CN(C(c2ccn(CCC(C)C)n2)=O)C1 26165,c1(C(N2CC(NC(C)=O)CC(C)(C)C2)=O)nnn2cc(C)nc(O)c12 26166,N=c1ncc(C(=O)NCC2(CNC(=O)CCF)CCC2)c[nH]1 26167,C(=O)(C1=NOC2(CCC2)C1)N1CCC(C)(C(=O)NC(Cn2ncc(C)c2)C)C1 26168,N1(C(C(CC)C(F)(F)F)=O)CC2(C=C(C(=O)NCC3CCSC3)CO2)C1 26169,Cc1cc(C)n(CC(=O)NCC2CCN(C(C3CCO3)=O)C2)n1 26170,C(C#C)(C(C)OCC)NC(CCN(C(=O)C(C)SC)CC#C)=O 26171,c1(OC)cc(C(=O)NC2CN(C(C34CC(C)(C3)C4)=O)CC2F)sc1Br 26172,N1(C(C=CC=CC)=O)CC(O)(C2(CNC(c3ccc(=NC)[nH]c3)=O)CC2)C1 26173,Cc1nccc(C(=O)NC(C)CCCCNC(C2C3CCCCC23)=O)n1 26174,N1(C(C2C(C=C)C2)=O)CC(CNC(=O)C(=O)N(C)C)(COC)C1 26175,c1(N2CC(OC)(CNC(C)=O)C2)ccnc(NC(=O)CC(C)C2CCCCC2)n1 26176,S(=O)(=O)(c1cnccc1N1CC(CN(C)C)C1)NCC1CCC(C)C1 26177,c1(C(=O)NCC(C)N(C(=O)COc2ccc(F)cn2)C)cnc(Cl)cn1 26178,C(Cc1ccco1)(C(=O)C(=O)CCc1nc(O)n[nH]1)NC(C=CC(CC)C)=O.N 26179,c1(C(=O)NC2C(C3CCN(C(C(CC)(C)C)=O)C3)C2)ccc2nccc(C)c2c1 26180,c1(CC(N2C3C(NC(C4C(CC)C4)=O)C(CC3)C2)=O)cc(Cl)ccc1Br 26181,C1(NC(c2c(OC)cnc(F)c2)=O)CC2CN(C(=O)CN3CSCC3=O)CC2C1 26182,C(CC(C(=O)N1CCC(O)(C(C)C)C1)NC(c1cccc[n+]1[O-])=O)OC 26183,c1(C(=O)NC(CC)CN(C)C(c2nonc2N)=O)cccc(C)c1N 26184,C1(CCC)CN(C(=O)Cc2csc(Cl)n2)CCN1C(=O)C(C)OCC 26185,N=c1[nH]c(CCC(=O)NCCOCCCNC(c2ccsn2)=O)cs1 26186,Cc1cc(CCNC(=O)CCn2cc(CC(C)O)nn2)ccn1 26187,C1(C(=O)NCC2N(CC)CC2)C=CCN(C(=O)CN2CC(=O)NC2=O)C1 26188,CCCC(C(=O)NC(C)C(=O)NCC(C)(CC)CC)NC(N)=O 26189,N1(C(C(=O)Nc2ccn3cnc(C)c3c2)=O)CCc2ccc(N(C)C)cc2C1 26190,n1(CC(=O)NC2CN(C(CC=C(C)C)=O)CC2C2CC2)ccc2ccc(F)cc12 26191,c1(CCC(=O)NCC2C(CNC(C3(C)CCC(=O)N3)=O)C2)cc(F)cc(F)c1 26192,N1(C(C(c2ccccc2)C)=O)CC(NC(=O)CCC2CCCN(C)C2)C(C)C1 26193,C1(CCNC(C(C)(C)SC)=O)CN(C(=O)Cc2nnc(O)s2)CC(C)O1 26194,c1(NCC(=O)NC(C2CC=CCC2)=O)ccccn1.CN1CCNC1=O 26195,CC(CC(N)=O)C(=O)NC1CC(CNC(c2cc(C3CCOCC3)nn2C)=O)C1 26196,N1(C(c2n(CC#C)ccc2)=O)CC2CCC2(CC(=O)N(CC)CC)C1 26197,c1(CC(=O)NCC2(NC(c3cccc(F)c3O)=O)COC2)nc2ncccn2n1 26198,N1(C(C2(C#C)CCC2)=O)CC(C(=O)NCC2CC(OC3CC3)C2)OC(C)C1 26199,Cc1cc2c(cc1C)C(C(=O)N1CCCC1CNC(c1cnc(N)s1)=O)CO2 26200,N1(C(C=C(C)c2ccco2)=O)CCN(C(=O)CCOCC2CCCO2)CC1CF 26201,Cc1cccc(C)c1CCC(=O)NC1CC12CC(NC(=O)CC13CCCC1C3)C2 26202,CCC(C)C(O)C(=O)NC1CCN(CCNC(=O)C(F)(F)C2CCCC2)CC1 26203,C1(C)(CNC(C2CC(C)N2C(=O)C#CC(C)(C)O)=O)CC2CCC1C2 26204,CC(C)C(CN(C)C)C(=O)N1CCOCC(NC(=O)CCCN=[N+]=[N-])C1 26205,c1(C(N2CC3C(CNC(C(C)=CC)=O)(C3)C2)=O)cccc2cccc(O)c12 26206,c1(C(N2CCC(c3cccc(C#N)c3)C2)=O)c(F)ccc2c1OCO2 26207,c1(NC(c2ccc(CC)o2)c2nnnn2CC2CCCO2)ccccc1OC 26208,Cn1cc(C(=O)NC2(c3nn[nH]n3)CC2)c2c(c1=O)CCCC2 26209,C(=O)CC(O)CC(C)(C)C.C(=O)(CC(C(C)CC)CNC)N1CCC(C#C)(O)C1 26210,c1(C(=O)NC(CCCNC(CSCC#C)=O)C)ccc(Cl)c(Cl)c1C 26211,C1(NC(C2CC(=C)C2)=O)CCC(F)(CNC(=O)CSCc2cccs2)C1 26212,CC(C)C(F)(F)CC(=O)N1CCCC(N(C(=O)C(c2ccc(Cl)cc2)C)C)C1 26213,c1(OC)cc(C=CC(N2CCCC2CCNC(c2cocc2C)=O)=O)ccc1N 26214,Cc1cc(C(=O)NC2CCN(C(=O)CN3CSCC3=O)CC2F)c2[nH]cnc2c1 26215,C1(NC(=O)COC(c2ccsc2)=O)C#CCCCCC1.C12CCN(CC1)C2=O 26216,C1(C(=O)NCC2(F)CN(C(c3ccc(COC)s3)=O)C2)CCCCCCC1 26217,c1(-n2c(CN3CCC(O)(C(C)C)C3)ccc2)cn(C)c2ccccc12 26218,N1(C(C(CC)(C)O)=O)CCC2(CCCC(CNC(C3(C(C)C)CCC3)=O)O2)CC1 26219,c1(NC(C2CCCN(C(CCC3(C#N)CCC3)=O)CC2)=O)cncc([N+](=O)[O-])c1 26220,C1(NC(CN(C)CC)=O)CCC2(CCN(C(=O)CCn3nc(C)c(C)c3C)C2)C1 26221,c1(C(N2CC(NC(c3ccc4sncc4c3)=O)C2)=O)cnn2cc(Br)cnc12 26222,N1(C(c2n(CCC)ncc2)=O)CC2C(CNC(c3cnoc3)=O)C2C1 26223,c1(C(=O)NC(C2N(C(Cn3ncc(C)c3)=O)CCC2)C)cc(C)c(C(F)F)cn1 26224,C1(NC(c2c(CC)cccc2)=O)CN(C(=O)C(O)Cn2cncn2)CC12CCC2 26225,C1(C(F)(F)CNC(=O)Nc2ccc(OC(F)F)cc2)(OC)CCCCC1 26226,C=CCC(CC=C)C(=O)NCCCCC(CO)NC(=O)CSC(C)(C)C 26227,Cn1nnc2cc(C(=O)NC3CN(C(c4ccon4)=O)CC3C3CC3)ccc12 26228,C1(NC(C=CCC2(NC(C3CC(CCOC)C3)=O)CCC2)=O)CCCOC1 26229,c1(OCC)ccc(C(C(=O)NCCC2(C)CC2)N(c2cccc(Cl)c2)C)nn1 26230,c1(C(=O)NC(C)CNC(=O)C(C)Sc2ccccc2)ncc2ccccc2c1N 26231,c1(CC)nn(C)c(NCc2ccc(Br)c(C)n2)c1[N+](=O)[O-] 26232,C(=O)(C1=COCCO1)NCC(C1CCC1)NC(C1(C(=O)OC)CCCO1)=O 26233,N1(C(c2cnn(CC(F)F)c2)C(=O)NC(CC)C)CC(CC(=O)OC)C(O)C1 26234,C1(CCN(C(c2n(CC#C)ccc2)=O)C)CCCCN1C(=O)COCCOC 26235,c1(C(N2CCN(C(C(C)=CC)=O)CC2)=O)cnn2cccnc12 26236,CC1(C)CN(C(=O)C=CC(c2ccccc2F)=O)CC1NC(=O)C=Cc1ncc[nH]1 26237,N1(C(c2ccc(Cl)cc2Br)=O)CCC2(CCN(S(=O)(=O)c3cccc(F)c3)C2)C1 26238,c1(NCC2C(c3c(C)nn(C)c3C)OCC2)cc(F)cc(F)c1CO 26239,c1(NC(N2CC(C(=O)OC(C)(C)C)(CC3CC[Si](C)(C)C3)C2)=O)cnn2ccsc12 26240,C(=O)(CCC(F)F)NC(C1(O)CN(C(c2cc(N3CCCC3)ncn2)=O)C1)C 26241,Cc1nc(=N)[nH]cc1C(N1CCC(N(C(=O)C(C)O)C)C1)=O 26242,c1(C(C(=O)NC2CCC(NC(C3C(C)(C(F)F)C3)=O)C2)O)cccc(Cl)c1 26243,C1(CNC(C(c2scc(C)n2)C)=O)CCN(C(c2cnn(C(C)C)c2)=O)C(C)C1 26244,c1(CNc2cnc(-c3c(OC)cccc3)s2)ccc(Cl)c(Cl)c1 26245,Cc1cc(N(C)C)cc(C)c1CC(N1CCC(=CCNC(=O)CC(C)F)CC1)=O 26246,N1(C(CN(c2ccccc2)C(C)=O)=O)CC2(CC(NC(C3CC(C)(C)C3)=O)C2)C1 26247,N1(C(C(C=C)(C)O)=O)CC(C2CCCN(C(=O)C(c3ccccc3)F)C2)C1 26248,C1(CNC(C(CCOC)C)=O)CN(C(=O)COc2cccc(CO)c2)CC1(C)C 26249,Cc1ncnc(C)c1C(N1CC(c2ocnc2CNC(c2ccc(Cl)o2)=O)C1)=O 26250,O=C1COc2ccc(SCCC(C3CCCOC3)=O)nc2N1 26251,C1(NC(CC(OCC)OCC)=O)CCN(C(=O)CC2CC(C(F)F)C2)CC1CO 26252,c1(C(N(CCCNC(CC(CCC)C)=O)CC)=O)csc(=NC2CC2)[nH]1 26253,c1(C(C)NC(=O)NCC(C)(C)CNC2CC2)ccc(Cl)cc1F 26254,C(=O)(N1CC(O)CCO1)C1CCCN(C(C(N2CCCCC2)C)=O)CC1 26255,C(C1(C)CCOCC1)=CC(N1CCC(C)(NC(c2c(OC)nsc2)=O)C1)=O 26256,c1(CC)ccc(C(=O)C(=O)NCC(C2CC2)N(C)C(C2(C(F)F)CCCO2)=O)s1 26257,CCC(CC(F)(F)F)C(=O)N1CC2CC(C1)CN(C(c1ccc(OC)cc1)=O)C2 26258,n1(CCC)cc(C(=O)NCCCN(C(=O)CNC(=O)OC)C(C)C)cn1 26259,Cc1sc(C(=O)NC2CCC(CCNC(=O)Cc3ccn(C)n3)C2)cc1Br 26260,N1(C(=O)Cc2ccc(Cl)s2)CC2CC(C1)CN(C(C1CCCC1)=O)C2 26261,c1(C(=O)NCC2N(C(CCc3ccc(SC)o3)=O)CC2)cc(C)ccc1F 26262,C1(SCc2cn(CCC(=O)NCc3ccc(CCO)s3)nn2)CCCCCCC1 26263,N1(C(CN(C)CC)=O)CC2CCCC1C2CNC(=O)C(C)(C)n1cccn1 26264,N1(C(=O)CC=CCNC(=O)CC2(O)CCCOC2)CC2(C1)NC(=O)NC2=O 26265,c12ccc(cc1)ONCCNC(=O)N2.C(=O)(CCCc1nc(C)no1)C(C)=O 26266,c1(C(N2CCC3CCN(C(=O)C(F)(F)CC4CC4)CC23)=O)cc2cc(F)ccc2[nH]1 26267,c1(C(=O)NC2C3(NC(c4nnn(C)c4N)=O)CCC(C2)C3)cccc2[nH]ncc12 26268,CCCCCC(O)CC(=O)N1CC2CC2C1C(=O)NC(C)C(C)F 26269,Cc1cnc(C(N2CCOC(CNC(=O)C=CC(C)C)C2)=O)nc1 26270,c1(CN=C(NCc2cc(C)on2)NC2CC2C)cn(C)c(=O)nc1O 26271,CCC(CC)(CCNC(=O)C=NOC)NC(C1CCC1n1cccn1)=O 26272,c1(C(N2CCCC2c2cn(C3C=CCCC3)nn2)=O)ccc2nnn(O)c2c1 26273,c1(C(N2C(CNC(c3c(C)cco3)=O)CCC2)=O)[nH]c2cc(F)cc(F)c2c1C 26274,C(C1=CCN(C(=O)COCC(F)F)CC1)NC(C1C(C)(C(C)C)C1)=O 26275,C(=O)(CCC(C)SC)NCC(CN(C(CSCC#C)=O)C)(C)C 26276,C1(NC(C2(OC)CC(C(F)F)C2)=O)CC2(C1)CC(NC(=O)CSC(F)F)C2 26277,CCCCC(CC)CC(=O)NC1CN(C)CCN1C(=O)COC1(C)CCCC1 26278,N1(C(C2(CNC(CCC3(C)CC3)=O)CC23CCC3)=O)CCC(C2CCC2)C1 26279,C(=O)(CCC(=O)NCCC)NCCC1(NC(CC=CCC)=O)CCC1 26280,N1(C(C(COC)NC(=O)C(C)OC(C)(C)C)=O)CCCN(C(C)C)CC1 26281,C1(n2cc(C3CCN(C)C3)nn2)C=CCC(C(=O)NC2CC(C)(C)C2)C1 26282,C(C(C)(CNC(c1cnc(CC)[nH]1)=O)OC)NC(C(C)OCC=C)=O 26283,CC(C)C(CCNC(c1ccc(N(C)C)cn1)=O)NC(=O)CCN1CCCCC1 26284,c1(C(N2C(CNC(=O)CC3CCCCC3)C=CC2)=O)ccn2ccnc2n1 26285,N1(C(c2c(C)nc[nH]2)=O)CC(CNC(=O)Cc2cnc(C(F)(F)F)s2)C(C)C1 26286,N1(C(C(C(C)C)C(C)C)=O)CCC2CCN(C(c3ccc4cc[nH]c4c3)=O)CC12 26287,CCCCC(C)C(=O)NCCCC(O)C(=O)NCCCC(=O)NO 26288,N1(C(C2(C#N)CC(=O)C2)=O)CCC2CC(N)CCC2C1.C(=O)(C=CC)CCC1CC1 26289,c1(C(N2CCC(N(C(=O)COc3ccccc3Cl)CC)C2)=O)c(O)cccc1Cl 26290,n1(CCC)ccc(C(=O)CCNC(c2cc(C(=O)OC)[nH]n2)=O)n1.C12CN(C1)C2C 26291,CNS(=O)(=O)NCC(=O)NC1COCC1CNC(=O)C(C)NC(N)=O 26292,C(CC(CC)C(=O)N(C1CN(C(C2(c3cccs3)CC2C)=O)C1)CC)=CCCC 26293,C1(NC(c2n(CC)ccc2)=O)CN(C(=O)C(C)C2CC2)CCC12CCOCC2 26294,C1(F)(C(=O)NCC(CN(C)C(C2CC23CCOC3)=O)(C)C)CCCCCC1 26295,CC1(C)CCN(C(C2CCO2)=O)C1CC(=O)NCCCCCCO 26296,C1(NC(CN(CCC)C(=O)NC(C)(C)C)=O)CC2CCC1CC2C(=O)O 26297,c1(C(N(CCN(C(=O)CCc2ccnc(Br)c2)C)C)=O)ccccc1C#N 26298,C1(C)(C(=O)OCC)CN(C(c2cc(C#N)n(C)c2)C(=O)NCC2(C)CC2)CCO1 26299,c1(C(=O)NCC(CN(C(COCCCC)=O)C)C)ccc(F)c(C(F)(F)F)c1 26300,CCC(C)(C)CC(=O)N1CC2CC(N(C(=O)CCCc3ccc(C)cc3)C)C1C2 26301,C1(CNC(=O)NCC(CC)CC(C)C)CCC2(CCCCC2)O1 26302,Cc1c(NC(C2CN(C(=O)CC(C)O)CCO2)=O)cccc1Br 26303,C1(C(N2CC(CC(=O)NCCCN(OC)C)OCC2)=O)CC2CCCC2C1 26304,C1(C(N2CCC(C)C2CNC(c2ccoc2Br)=O)=O)CCCNS1(=O)=O 26305,Cc1ccc(C)c(C(N2CC(C(C)NC(=O)C(C)Sc3nncn3C)C2)=O)c1 26306,c1(CN(C2CN(S(=O)(=O)CCl)C2)Cc2cn(CC)nn2)ccc(Br)cc1 26307,N=c1[nH]n(CC(N2CCC2CNC(=O)CSC2CCCCO2)=O)cc1Br 26308,Cc1oc(-n2cccc2)c(C#N)c1C(=O)NCC(O)CNC(C1(O)CCSC1)=O 26309,Cc1ccc(N)c(C)c1C(N1CC2CCCC2(NC(C2CCC(O)CC2)=O)C1)=O 26310,C1(SCC)CCCC(N=c2[nH]c(=NCc3ncc(CC4CC4)[nH]3)[nH]c3c2CCCC3)C1 26311,c1(Nc2nc(OC)nc(N3CC4C(N(C)C)C4C3)n2)ccc2ccsc2c1 26312,N1(C(C(CCC)O)=O)CC2(CCN(C(C3CCCC3)=O)CC2)CC1C 26313,Cc1cc(C(N2CCC(C)(C)C2CNC(=O)CCN2CCOC2=O)=O)cc(F)c1 26314,C1(C(N(C2CCCC2)CCNC(c2ccc(CC)o2)=O)=O)CC(C)CC(C)(C)C1 26315,c1(CC(=O)NCC(C2CC2)NC(C(C)OCCC=C)=O)ccc([N+](=O)[O-])c(N)c1 26316,C=CC(C)CC(=O)N(C1CCN(C(c2cc(C)sn2)=O)C1)CC 26317,N1(C(=O)NC(CC)C(c2nnnn2C)NC(C)(C)C)CC2(CO)CC2(C(F)(F)F)C1 26318,CCCCC(O)C(=O)N1CC(NC(=O)CCc2ncccn2)C(n2ccnn2)C1 26319,N1(C(CC2C(NC(c3n(C)nc(O)c3)=O)CCCC2)=O)CCOC2CCCC12 26320,Cc1ccc(F)cc1C(=O)C(=O)NC(C)CN(C)C(C1CC2(CSC2)C1)=O 26321,N1(C(c2n(C)nnc2)=O)CCC(CNC(=O)CNS(N)(=O)=O)C1(C)C 26322,C1(CNC(C=CCCC)=O)CC2CC(C1)N(C(=O)CCc1cccnc1)C2 26323,CC(C)(CCCNC(=O)C(=O)NCC1CC1)NC(=O)Cc1sccc1Br 26324,c1(C(=O)NCC2CCC(NC(C(C(C=C)C)C)=O)CC2)c(O)nnc2c1CCC2 26325,N1(CC)CC(C)CC(C)C1.C1CCCC(=O)N1.C1=CCNC1=O 26326,Nc1c(C(=O)NCCOCCOCCNC(=O)C2=COCC2)ccc(Cl)c1O 26327,c1(C(N2C(CCCO)CCCC2)=O)cnc2ncnc(O)c2c1 26328,C1(OC)CCC(C(=O)NCCN(C(=O)CCc2cccs2)C)C1 26329,c1(CC)cc(C(=O)NCC(O)C(=O)NC(C(=O)OC)C2(C)CC2)no1 26330,C(=O)(CC1COCc2ccccc21)N1CCC(NC(CCSCCOC)=O)C1(C)C 26331,CCCCCCCC(=O)N1CCC(NC(=O)COc2cc(F)cc(F)c2)C12CC2 26332,c1(C(=O)NC2C(NC(c3c(C)onc3C3CC3)=O)COC2)cccc(S(C)=O)c1 26333,c1(C(=O)NCC(CC)(C)NC(=O)C(C)C)cc(F)cc(Br)c1 26334,N1(C(C2C(CC)CCC2)=O)CC2(NC(=O)CC3CC4C=CC3CC4)CCC1CC2 26335,N1(C(CCCc2ncc(C)o2)=O)CCC2(CC1)CN(C(=O)CCF)CC2CO 26336,C1(N(C(COCCNC(C(C2CCCC2)OCC)=O)=O)C)COCCO1 26337,c1(CC)nn[nH]c1C(=O)NCC(O)C(=O)N1CCC(c2cnn[nH]2)C1 26338,CC#CCC(C(=O)NCC(C)(O)CCO)NC(=O)C(C1CC1)SC 26339,C1(c2n(CC=C)nnn2)(Nc2cnn(CC(C)(C)O)c2)CCN(CCOC)C1 26340,C1(CCC)CCCN(C(=O)CC2CCCN2C(c2cnc(Cl)n2C)=O)CC1 26341,c1(CC)ccc(C(N2CCC(N(C)C(C3C(C(F)F)C3(C)C)=O)C2)=O)c(O)c1 26342,c1(C(=O)NCCCCN(C(=O)CC2CCC2)C)cc(=NS(C)(=O)=O)cc[nH]1 26343,c1(CN2CCC(F)(C(=O)NC(C)CN(C)C)C2)ccc2ncccc2c1 26344,C1(NC(C(C=C=C)C)=O)CCC12CN(C(=O)CSCC(N)=O)C2 26345,CC1(CC(=O)NCCC2CCCN2C(c2csc(Cl)c2)=O)CC1(F)Cl 26346,C12(CNC(C(=Cc3ccc(F)cc3)C)=O)CN(C(=O)CC3CCC3)CC1CCO2 26347,C1(NC(CCc2c(C)noc2C)=O)CCN(C(=O)CC2CCSC2)CCC1CO 26348,S(=O)(=O)(c1ccccc1)NCC(=O)N(C(C)CCNC(C1CCC(C)CC1)=O)C 26349,C(=O)(C1CCCn2ccnc21)NC1CC2(C(NC(CC(C(C)C)(F)F)=O)C2)C1 26350,c1(OC)cc(C(=O)NC2CC(CO)N(C(C3CCC3)=O)C2)sc1Cl 26351,C(=O)(C(CC)CCc1ccccc1)N1CCC(CC=C)(NC(=O)C(F)C2CC2)C1 26352,c1(C(N2C(CNC(C3(CCC=C)CC3)=O)CCCC2)=O)cccc2ncc(C)n12 26353,Cc1ocnc1C(=O)N(C1CC1)CC1CCCN1C(=O)Cc1cc(C2CC2)no1 26354,c1(C(=O)NCCOC(C)(C)CNC(C2(C3CC3)CCC2)=O)nc(N(C)C)nc(=N)[nH]1 26355,c1(OC)cc(F)c(C(=O)NC(C)CN(C)C(C2CC(F)(CF)C2)=O)c(F)c1 26356,c1(C(=O)NC23CC(c4ccccc4)(C2)C3)cccnc1N1CCOCC1 26357,CC(C)C(F)(CNC(=O)CCC(C)(F)F)C(=O)N1CCOC(C2(C)CC2)C1 26358,c1(CC)nc(C(=O)NC2CCC(NC(=O)COCc3cc(C)on3)C2)co1 26359,C#Cc1ccc(CC(N2CCN(C(c3cccnn3)=O)C(CO)C2)=O)cc1 26360,N1(CCOC(=O)NCc2onc(C)n2)CCCC(C)C1 26361,C1(C(N(CCCC)CCOC)=O)C2CC2CN1C(c1[nH]ccc1CC)=O 26362,Cc1csc2ncc(C(=O)NC(C)(CNC(C3(Cl)CC3(C)C)=O)C3CC3)c(=O)n12 26363,c1(NC2CCC(NC(Cc3ccc(SC)cc3)=O)C2)ncnc2[nH]cc(C)c12 26364,N12CCCC1C1CCCN1Cc1oc(C)c(c1)C2=O.C(C)(C)(C)SCS(C)(=O)=O 26365,C1(C(=O)OC)CC(C)N1C(C1(NC(c2cnc(C(C)C)o2)=O)CC1)=O 26366,c1(C(=O)NCC(C)NC(=O)C2CCCn3cnnc32)ccc2c(c1)C(=O)CCN2 26367,c1(CC)cc(C(N2CCOCC2CCNC(=O)CC2C=CCCC2)=O)cc(O)n1 26368,c1(SC)ccccc1C(=O)NCC(O)CNC(=O)C(C)=O 26369,C1(NC(C(C)(C)SC)=O)CN(C(c2cncc(C(C)(F)F)c2)=O)CC1C(F)F 26370,C1(CC)CCN(C(C2CCC2C(N)=O)=O)C1C(=O)NCCCC1(C)CC1 26371,c1(C(=O)NC2C(C(=O)NCC(COC)C)CCC2)ccc2ccccc2c1 26372,C(C(O)CC(=O)NC)NC(CN(CCC=C)C(c1c(C)coc1CC)=O)=O 26373,C1(C(N2CCC(N(C(=O)C(O)C3CC3)C)CC2)=O)OCC2CCCC12 26374,C1(OCCNC(c2coc(O)n2)=O)CCN(C(C2(C(F)(F)F)CCC2)=O)CC1 26375,c1(C(=O)NCCC2CCC(NC(c3cc(OC)n(C)n3)=O)C2)cn2ccsc2n1 26376,C(=O)(C(C)(C)CC(=O)NCc1nc(CNC(=O)CCc2csnn2)cs1)OCC 26377,C(=O)(C(CCS(C)=O)N(C)C)NC1CCN(C(CCCOC)=O)C1(C)C 26378,C12(NC(CSCC#C)=O)CC3CC(C1)CC(NC(c1nnn(CC)c1C)=O)(C3)C2 26379,C1(NC(C(CC=C)C)=O)CCN(c2ncc(Br)cn2)CC1C 26380,c1(OCCC)ccc(C(=O)NC2(CNC(C3SCCCS3)=O)CC2)cc1N 26381,c1(CC(=O)NCCC2CN(C(=O)COC3COC3)CCO2)c[nH]c2cnccc12 26382,c1(C(c2n(C)nnn2)NCc2cnoc2C(C)(C)C)nn(C)cc1I 26383,c1(OC)c(C)cc(NC(c2n[nH]cc2NC(=O)C(C)(C)CCl)=O)cc1C 26384,Cc1nn(Cc2c(C)noc2CC2CNC2)c(C)c1-c1cn(CCN(C)C)nn1 26385,C1(C(=O)NCC(C)(O)CNC(=O)Cc2csc(Cl)c2)CCOCC12CCC2 26386,C(CCS(=O)(=O)NNCC(=O)NC1(NC(=O)C=CCN(C)CC)CCCC1)OC 26387,c1(-c2cn(CCC(=O)NC(C(=O)N(CC)CC)C)nn2)cccc(N)c1C#N 26388,C1(OC)CCCC1CNC(c1cn(CCNC(C2CNC(=O)N2)=O)nn1)=O 26389,c1(OC)c(C(=O)NC2CCC2NC(C23CC(F)(C2)C3)=O)cc([N+](=O)[O-])cc1Cl 26390,C(CCCC(C)(C)C)NC(C1CC=CC(NC(C(CC=CC)C)=O)C1)=O 26391,C1(CSC)CCCCN(C(=O)C(N2CCSCC2C)=O)C1 26392,CC1CC(NC(=O)C=Cc2ccc(Br)cc2)CN(C(=O)C(C)NC(N)=O)C1 26393,c1(NC(c2ccc(Br)c(Cl)c2)c2n(CCSC)nnn2)ccc(Br)c(C)c1 26394,C1(C(=O)NC(c2ccncc2)C)CN(C(=O)CN2CCC(F)CC2)C2(CCC2)C1 26395,c1(NC(C)=O)ncc(S(=O)(=O)N2CCCC2c2cc(F)cc(Br)c2)s1 26396,CCC(F)(F)C(=O)NCC(F)CNC(c1nc(Cl)sc1C)=O 26397,N(C(=NCC1CCN(c2ccc(F)c(Cl)c2)C1)NCC(F)F)C1CC(C#C)C1 26398,C=CCCCC(C(=O)NCc1cn(C2CC2)cn1)NC(=O)CC1(COC)CC1 26399,C=CCCCC(=O)NCC1(CN(C)C(C2CCC(C)CC2)=O)CC1 26400,c1(C(=O)NCC(C)CNC(=O)CC(C)(C)O)ccc(F)c2ncccc12 26401,C(=O)(CS(=O)(=O)CC(=O)N(C)CC1CCCN1C(=O)C(C)CC(C)C)OC 26402,c1(OC)cccc(CC(O)C(=O)NCC2CN(C(C3CCC(=O)N3)=O)C2)c1 26403,c1(CC)cc(C(N2CCCC2c2ccc(F)cc2)C(=O)NC(C)(C)C)ccc1Br 26404,N1(C(c2cnn(C)c2C2CC2)=O)CCC(NC(C2(C)CC=CCO2)=O)CC(O)C1 26405,C1(C)(CC(=O)OC)CN(CC(=O)NC2OCCC2n2cccn2)CCO1 26406,C1(CNC(C#CC(C)C)=O)C(C2CC2)CCN1C(=O)C=Cc1ccc(Cl)s1 26407,N1(C(C2(CC)CCCC2)=O)CC(NC(C2CN(C(C)=O)C2)=O)CC1(C)C 26408,N1(C(CC(=O)NC)=O)CCC2C1CCCN2C(c1ccc([N+](=O)[O-])c(C)c1)=O 26409,C1(C(c2nnnn2C(C)(C)CC)NCC(=O)NCCC)CCSC1(C)C 26410,CCCCCC(O)C(=O)NCC1CC(C(C)C)CCN1C(c1coc(C)n1)=O 26411,N1(C(c2cc(OC)nn2C)=O)CC2CC(O)C1C2NC(=O)CC(C(F)(F)F)OC 26412,c1(C(=O)NCC2CCC(Cn3cc(C=CC)nn3)CC2)cc(F)ccc1Cl 26413,C1(C)(C(N(CC(C(=O)NC)C)C)=O)CCN(C(=O)CCOCC(F)F)C1 26414,C12(NC(c3ccc(CC)o3)=O)CN(C(c3cc4c(s3)CCC4)=O)C(COC)(C1)C2 26415,C(C#N)(C(=O)C(O)c1ccccn1)c1ccc(C)cc1.c12cn(nn1)C1COC21 26416,c1(-c2scc(C(=O)NC3CN(C(C4CC(F)C4)=O)C3)n2)cccc(Cl)c1 26417,CC(C)C(F)(F)CC(=O)NC(C)(CNC(c1cc2c(s1)CCC2=O)=O)C1CC1 26418,c1(CNC(C(CC)C)=O)ccc2c(c1)CCN(C(C1(C)CCN(C(C)=O)C1)=O)C2 26419,N1(C(C)=O)CC2COCCC2(NC(c2cccc([N+](=O)[O-])c2Br)=O)C1 26420,C1(C(=O)NC(CNC(C(CC)C2CCC(=O)N2)=O)C)CCC(OC)CC1 26421,c1(CC)cncc(NC(=O)C(C2CCN(Cc3csc(Br)n3)CC2)C)c1 26422,c1(N2CCN(C(=O)NC)CC2)nc(=NC2CCCSCC2)[nH]c2c1COC2 26423,N1(C(C2(C(=O)NC)CCC2)=O)CCC2(NC(c3ccc(N)c(N)n3)=O)CC2C1 26424,c1(C(CNC(c2c(C)cncc2)=O)NC(c2ncccc2N)=O)cc(F)cc(Cl)c1 26425,C1(C(N2CC(NC(=O)Cc3cnc[nH]3)C(F)C2)=O)CCC(C)(C)CC1 26426,n1(C(C(=O)NC2CC(NC(C3C(C(=O)OC)CC3)=O)C2)C)cc2c(n1)CCCC2 26427,c1(C(N(C(C)C)CCN(C)C(C2OCC2(C)C)=O)=O)cnc2sccc2c1 26428,C#CC1CC2CCC1N(C(=O)CC1(OC)CN(C(c3cnn(C)c3CC)=O)C1)C2 26429,CC1(C)OC2(CNC(=O)CS(C)(=O)=O)CC1(NC(c1cc(C3CCC3)[nH]n1)=O)C2 26430,C1(C(=O)NCC2CC(SC)C2)C(C)CCN1C(C1(CC2CC2)CCC1)=O 26431,C1(C)(CNC(c2nnc(C)s2)=O)CN(C(=O)CCOC2CC2)CCO1 26432,C1(NC(C(C)c2ccco2)=O)(CNC(=O)Cc2nc(=N)[nH][nH]2)CCCCCC1 26433,C1(C(=O)NCC2CC(O)CN2C(c2cn(C)c(C)n2)=O)(COC)CCOCC1 26434,N1(c2c(N(C3CCCC3)C(=O)OC(C)(C)C)nccn2)CC(C(=O)O)C2(CC2)C1 26435,C12(COCC)CC(C(N3CCC(C)(CNC(=O)C=C(C)C)C3)=O)(CO1)C2 26436,c1(C(=O)Nc2cccc(C(C)C)c2)cc(Cl)ncc1NC(c1cnn(C)c1Cl)=O 26437,C1(NC(c2c(C)snn2)=O)C(CNC(c2cc(C#N)n(C)n2)=O)CCC12CCC2 26438,C1(NC(C(C)OCC=C)=O)(CNC(C2OCCC2C(C)C)=O)CCCC1 26439,CC1CC(NC(=O)NCCOC(=O)CO)CCS1(=O)=O 26440,C(=O)(CCCC(F)F)N(c1ccc(C)cc1)CCCN1CCCC1 26441,C1(F)(CNC(c2cnsc2)=O)CC(NC(C2CC2(F)F)=O)C1 26442,C1(CC(=O)NCC(CO)NC(CSC)=O)CCCOCC1 26443,C=C(C)CCCC(=O)NCC=CCNC(=O)C(C)c1cncs1 26444,c1(Cn2cc(CCOCCO)nn2)ccncc1CO.C1(NC(=O)N)CCCCC1 26445,CC1CCN(CC(=O)NCCN(C(=O)CC2CCSCC2)CC2CC2)C1 26446,C(CCCCCF)N(C(=O)C(n1cc(CCCS(N)(=O)=O)nn1)C)C(C)C 26447,c1(CN(C(=O)C(F)CC2CC2)CC(C)(C)O)cc(C2CC2)ncn1 26448,c1(C(N2CCC(C(C)NC(=O)C(c3ccccc3)O)C2)=O)cncc(N=[N+]=[N-])c1 26449,CCC(C)(CC)C(=O)NC.C12CC(=NO1)CCC2=O.N1(C(CSC)=O)CCC(C)CC1 26450,N1(CC)CCCCC1C(=O)N(C)CC1CCCCN1C(C1(O)CCCCC1)=O 26451,CC(O)CCCCCC(=O)N1CCC(CCNC(c2cccc(N)c2O)=O)C1 26452,c1(C(C)(C)C(=O)NCC2CC(NC(c3ccoc3Cl)=O)C2)cccc(Cl)c1F 26453,c1(C(=O)NCCC2N(C(C3=CCCC3C)=O)CCSC2)n[nH]c2ccc(F)cc12 26454,N1(Cc2cccc(OCC#C)c2)CCC(O)(C2C(C(=O)O)C2)CC1 26455,C1(C(=O)OC)CN(C(=O)CN(C)C(=O)C2CC2)CC1(C)C 26456,C1(CNC(Cn2c(C)ccn2)=O)CN(C(=O)CC2C=CCC2)CC1(C)C 26457,c1(-c2cn(C(C)C(=O)N(C)C)nn2)ccc(N)cc1.C1CCCC1N1CCOCC1 26458,c1(C(=O)NC(C2(O)CCN(C(=O)CCc3ccccc3O)C2)C)cnccc1Cl 26459,C(=O)(C1SCc2cccnc21)NC1(CN(C(C2CCN(CC(C)C)C2)=O)C)CC1 26460,c1(C(C(N2CCCN(c3ccccc3C#N)CC2)C)=O)ccc2c(c1)CCC2 26461,c1(OC)cccc(F)c1C(N1CCCC1CC(=O)NC(CC(=O)O)C(=O)O)=O 26462,c1(OCC(=O)Nc2nc(C(C)C)nc(C(C)(C)C)c2)c(Cl)cc(Cl)cc1Cl 26463,CCC(CC)CCC(=O)N1CCC(NC(c2cncc(F)c2Cl)=O)C(F)C1 26464,C1(NC(C(=O)NCCOC)=O)CCC(CCNC(=O)CC2CCOC2)C1 26465,c1(OC)cc(CNCC(C(=O)O)OC)cc(I)c1OC 26466,C1(NC(Cc2c(C)nn(C)c2)=O)CCS(=O)(=O)C12CN(C(=O)C(O)C1CCC1)C2 26467,c1(OCC)cc(C=CC(c2ccn(C)c2)=O)ccc1OCC(N)=O.C1CCCCC1 26468,c1(CC)cc(C(N2CC(CC(F)C(=O)NC(c3cc[nH]n3)C)C2)=O)ccn1 26469,C1(NC(C2CC(C)(CC)C2)=O)CCCC2CN(C(=O)C=Cc3ccccc3)CC12 26470,c1(CC(=O)NC2CC(NC(C3CC(Cl)(Cl)C3)=O)C2)cnc2ncccn12 26471,c1(NC2CCN(C(=O)OC(C)(C)C)C2c2ccccc2)c(F)cc(C#N)cc1F 26472,c1(C(N(CC(C)NC(C2CCCSC2)=O)CC)=O)cc(SC)ccc1Cl 26473,C1(CNC(CSCCC)=O)(CNC(=O)CC(F)F)CCCCC1 26474,CCCCC(CNC(=O)Cc1ccn(-c2ccc(F)cc2)n1)NC(=O)CC(C)O 26475,Cc1cccc(Nc2cn(CC3N(C(=O)NC4CC4)CC(O)C3)cn2)c1 26476,N1(C(Cc2n(C)ccn2)=O)CCC(NC(c2ccnc(O)c2)=O)C(CO)C1 26477,c1(N2CCC3(C)C(C)(C2)C3(F)F)nc(=NCc2ccccc2I)[nH]c2ccsc12 26478,c1(N2CCCC(CNC(C3(C=C)CCOCC3)=O)CC2)ncccc1[N+](=O)[O-] 26479,c1(C(C)=O)ncc(C(=O)NC2CCC2C(=O)NCCc2cccnc2)s1 26480,C(=O)(C(C(=O)N1CCC(CN(C)C(c2cncn2C(C)C)=O)C1)OC)OC 26481,C1(CC=C)(NC(c2snnc2CCC)=O)CCCN(C(c2ccnc(F)c2)=O)C1 26482,c1(CNC2N(C(=O)OC(C)(C)C)CCCC2(C)C)c(Br)ccc2c1CCC2=O 26483,C1(NC(C(c2ccccn2)C)=O)CN(C(c2cccc(Cl)c2)=O)C2CCCCC12 26484,C(CCNC(=O)C(Cl)=CCl)(C(C)C(C)C)NC(C(CC)(C)O)=O 26485,c1(C(c2n(CC)nnn2)NC2CCC3(CC3)C2)sc(Br)c(C)c1C 26486,Cn1nc(C(=O)NCCCNC(C2(Cc3cccnc3)CC2)=O)ccc1=O 26487,C(CN=c1cc(C)nc(N2CCOC3(CCSC3)C2)[nH]1)(c1ccc(F)cc1)SC 26488,C1(C(=O)NC23C(CN(C(CC4(C)CCC4)=O)C2)C3)CC2CCCC(C1)C2 26489,c1(C(=O)NCC(CNC(c2ncc(C)c(C)c2)=O)O)ccn2ccccc12 26490,C1(C(=O)NCCOCCNC(Cc2ccc(C(C)=O)cc2)=O)CC2C(C1)C2(C)C 26491,S(=O)(=O)(c1ccc(NC(c2ncc(Br)cc2C)C)c(C#N)c1)NC(CC=C)CC 26492,c1(OC)nccc(C(=O)NC2CCCN(C(=O)C(C)(C)Br)CC2)c1Cl 26493,C(=O)(CCCC(=O)OC)N(C1CCN(C(C(C(C)C)OCC)=O)CC1)CCO 26494,c1(CC)nc(N2CC3CC(NC(=O)C(C)C)CC3C2)c(C)c(Cl)n1 26495,C#CC1CCCN(C(C2(CNC(=O)C=Cc3ccoc3)CCC2)=O)C1 26496,c1(OC)cc(F)ccc1C(N1CC(C)(C)CC1CNC(=O)CCCC1CC1C)=O 26497,c1(C(N2CCC(C(=O)NC3C(C4C(C)C4)C3)CC2C)=O)cccc2[nH]ccc12 26498,Cc1ccnc2nc(C(=O)NC3CN(C(=O)C(C)S(N)(=O)=O)CC4(CC4)C3)nn12 26499,Cc1ccc(C(=O)NC(C)CCCNC(c2coc(CO)c2)=O)cc1S(N)(=O)=O 26500,C(=O)(CC(C(F)(F)F)n1ccnc1)N1CC(NC(c2c(C)noc2)=O)C(O)C1 26501,N1(C(CC(CC)C)=O)CCC(CNC(=O)C=Cc2ccc(Cl)s2)C12CC2 26502,N1(C(C(COC)OC)=O)CC(C(=O)N(CCCC(C)(F)F)C)CCC1C 26503,C(=O)(C#CC1(C)COC1)NC1CCCC(CNC(CCc2cc(C)nn2C)=O)C1 26504,c1(C(=O)NCC2CC(C(=O)NC(c3nncs3)C)C2)cccc(C#N)c1 26505,c1(C(N2CC(C(C)NC(C(COC)(C)O)=O)OCC2)=O)cncc2[nH]ccc12 26506,CC(C)CC(C)CC(=O)NCc1nccn1C.C12CCC(CC1)CC(=O)C(=O)N2 26507,C(=O)(C1=CCCOCC1)NC(CC)(CC)CCNC(=O)CCc1cncc(F)c1 26508,CCC(C)C(C(=O)N1CCC(n2cc(Cn3cncn3)nn2)C(O)C1)N(C)C 26509,N1(C(CCn2cc(C(C)=O)nn2)=O)CCCCC1CNC(=O)C(C)CCN(C)C 26510,C1(N(C(=O)CO)CC)CCCN(C(C2C=CCC2)=O)C1 26511,C1(C(=O)NC2C(C)N(C(c3ccn(CCF)n3)=O)CC2)CC2(COC(=O)N2)C1 26512,N1(CC(=O)NCc2scc(CC)n2)CCN(C(c2cnc(Br)s2)=O)CC1 26513,c1(C(N2C(CCCNC(C3CC=C(C)CC3)=O)CCC2)=O)ncn2ccccc12 26514,C(C(C)(C)C(=O)NC(C1CCN(C(c2ccc(C#N)s2)=O)C1)C)SC 26515,C1(CNC(=O)C=C2CCCC2)CCCC1NC(=O)CCC1CC1(Cl)Cl 26516,c1(C(=O)O)cc(NC(Cn2cc(-c3ccc(OC)c(SC)c3)nn2)=O)c(C)cc1C 26517,C1(CNC(C(C(C)C)C)=O)CCN(C(=O)CCC2(C)CC2)CC1(F)F 26518,CCC(C(=O)NC(C)(CNC(c1cc(C2CCCCC2)[nH]n1)=O)CO)C(C)C 26519,N1(C(C(=O)NCCC)CC2CC(F)(F)C2)CCC(C2CCCCC2)CC1 26520,c1(C(=O)NCC2(F)CC(NC(C(CC)(C)O)=O)C2)cccc(F)c1Cl 26521,C1(NC(=O)COC(=O)CO)CCN(CCNC(=O)Cc2cocn2)CC1 26522,c1(C2C(C(N(CCCNC(C(COCC)C)=O)C)=O)C2)cccc(S(C)(=O)=O)c1 26523,CC1CC(C)N(C(=O)CCc2nc(=N)[nH][nH]2)CCN1C(=O)COCC1CCCC1 26524,N1(C(c2cn(C)cn2)C(=O)NCCC2(C)CC2)CCC(CO)C1c1ccccc1 26525,CC1CC(NC(c2cnn(CCO)c2N)=O)CCN1C(C1CC(=O)N1)=O 26526,c1(C(=O)NC2CC3(C(NC(=O)CC(F)(F)F)C3)C2)cc2c(nn1)CCC2 26527,n1(CC)cnc2[nH]c(=NC3CC3CC)nc(N3CCCC(OC)C3)c12 26528,C1(CC(N2CCC(NC(=O)CCCC3CC3)CC2)=O)CC(O)C12CCC2 26529,c1(C(=O)NC(CC)CN(C(=O)C=C(C)N)C)cccc(NC(N)=O)c1 26530,C1(C(=O)NCc2onc(COC)n2)CC(NC(C2OCCC2(C)C)=O)C(O)C1 26531,c1(OC)ncc(Cl)c(C(N2CC(N(C)C(c3ccccn3)=O)C(O)C2)=O)c1Cl 26532,c1(OC)ccc2c(c1)C(C(=O)N1CCC(NC(=O)COC3CCC3)C(O)C1)CC2 26533,C1(CNC(c2nnc(O)nc2O)=O)CN(C(=O)C2=CC(O)CCC2)CC12CCC2 26534,C#CC1(CNC(C2(NC(c3ncc(F)cc3F)=O)CCSC2)=O)CCOCC1 26535,c1(OC)ccc(F)cc1CCC(N1CCCC1CNC(c1cc(O)nn1C)=O)=O 26536,C1(C(=O)NCC(C)C#N)CCCC(NC(=O)CC(C)(C)C)CC1 26537,c1(N2CCC(N(C(C(OC)OCC)=O)C)C2)nc(C)nc2ccccc12 26538,c1(C(=O)NCC2CCCN(C(c3cc(CCOC)on3)=O)C2)cccc(F)c1N 26539,C1(NC(c2cnn(C)n2)=O)C=CCC(C(=O)N(C2COCC2O)C2CC2)C1 26540,C=CCC(CNC(C1(C2CC2)CC1)=O)NC(=O)Cc1c[nH]nc1O 26541,N1(CC#C)CCC(C(=O)NCC(C(C)(C)C)NC(=O)C=CC2CCCN2C)CC1 26542,C1(C(=O)NCCCCCN(C(=O)CC2(O)CCOCC2)C)C2CCCCCC12 26543,CCCC(C#N)C(=O)NCC1(O)CCCN(C(c2c(C)cnn2C)=O)C1 26544,C(=O)(CCC(C)(C)C(=O)N(CCNC(C1CCCCC1F)=O)C1CC1)OC 26545,N1(C(C2CC(=C)C2)=O)CCN(C2CCC(NC(=O)Cc3ncccc3C)C2)CC1 26546,c1(C(=O)NC2CCCN(CCC3CCCC3)C2)cc2ccccn2n1 26547,N1(C(c2c(C)nc(NC(c3c(C)nc(C)o3)=O)s2)=O)CCc2ccc(Br)cc2C1 26548,c1(C(N(C2CN(C(C3C(CC)CCCC3)=O)C2)C)=O)cc2c(C)ccc(F)c2[nH]1 26549,C(c1ccccc1OC)=CC(=O)NCC(C1CC1)NC(Cn1ncc(CC)c1)=O 26550,N1(C(C(CSC)C)=O)CC(C(=O)NCC2(CO)CC(C)C2)CC1(C)C 26551,N#Cc1c(Cl)cc(-c2cn(C3CN(C(=O)C=CC4CC4)C3)nn2)cc1Cl 26552,CC1(CCNC(C2C(F)(F)C23CC3)=O)CCN(C(=O)C=CCn2cncn2)C1 26553,N1(Cc2cccc(C)c2)CCC(C)C(NC(c2cc(C3CC3)nn2C)=O)C1 26554,C1(NC(COCC=C)=O)CCCC(NC(c2cccc(CCN(C)C)c2)=O)C1 26555,CCC(C)(C#N)C(=O)N(C)CCNC(=O)CNC(c1ccccc1NC)=O 26556,c1(OC)ncc(C(N2CC(NS(=O)(=O)C(F)(F)F)CC(F)C2)=O)cc1Br 26557,c1(C(N2CC(=C(CNC(=O)CN3CCCC3)F)C2)=O)cccc([N+](=O)[O-])c1 26558,N=c1nc[nH]n1CC(N1CC(CC(F)C(=O)NCC2CCCCC2)C1)=O 26559,N1(C(n2c(Cc3cc(C)cc(C)n3)cc(OC)c2)=O)CC(C)N(C)CC1C 26560,N1(C(c2c(C)nn(C(C)C)c2)=O)CCN(C(=O)CN2CSCCSC2)CCC1C 26561,N1(CCC)CC(C(=O)NC(C2CCN(C(=O)Cn3cncc3C)CC2)C)CC1=O 26562,N1(C(c2c(C)noc2)=O)CC2CCC1C(CNC(c1ccccc1CC#N)=O)C2 26563,c1(C(=O)NCC2N(C(C(CCOC)(C)C)=O)CCCC2)cccc2ccc(O)nc12 26564,C1(CC=C)(NC(c2ccc(F)o2)=O)CCN(C(C2OCC2(C)C)=O)CC1 26565,S(=O)(=O)(CC(=O)NCC1(F)CC(NC(c2cccn2CC)=O)C1)NCC 26566,CCC(CCCC(=O)N1CC2(C1)CC2(F)F)NC(C1(O)CCSC1)=O 26567,c1(C(=O)NCc2n(C)ncc2)csc(=NCc2c(Br)cnn2C)[nH]1 26568,c1(C(N(CC(CC)NC(C2CCC(C)CC2)=O)CC)=O)cn(C)nc1Cl 26569,C1(CNC(=NCCOC)NCc2ccsc2Br)CCC2(CCC2)CO1 26570,C(=O)(C#CC(C)(C)C)NC1(CC(=O)NCc2nnn(CC)n2)CCCCC1 26571,CCS(=O)c1ccccc1C(N1CCN(C(=O)CP(C)(C)=O)C(C2CCC2)C1)=O 26572,C1(c2cn(CCCOC)nn2)C(C)CCN1C(c1ccc(C(C)=O)s1)=O 26573,C(c1ccccc1)=[SH]CC(=O)NCCC1CC(NC(CCc2nc(=N)[nH][nH]2)=O)C1 26574,c1(OC)ccc(S(=O)(=O)N2CCOC(C)(C(=O)O)C2)cc1-c1ccc(C)cc1C 26575,CCCCCC(F)C(=O)N(CC(N1CCc2nn[nH]c2C1)=O)CCOC 26576,C1(C(C2CCCC(n3cccc3)C2)=O)CCCN(C(=O)C(C)C2CC2)CC1.CC(=O)N 26577,c1(NC(CSC(C)(C)C)=O)ccc(C(F)(F)Cl)cc1 26578,N1(C(CCCOC(C)(C)C)=O)CC2(C=C(C(=O)N3CC(F)CC3CO)CO2)C1 26579,C1(CN(C(=O)CC2CC(F)C2)C2CC2)CCN(C(=O)CC2(O)CCC2)CC1 26580,C1(O)(CC(=O)NC(C(=O)NCC2C(C)(C)C2)C2(C)CC2)CCOC1 26581,c1(OCC)ccc(N)c(C(=O)N(C(=O)CCCC2CC2C)C2CC2)c1 26582,C1(C)(C(N(CCNC(=O)Cc2ccn(CC(C)C)n2)CC)=O)CC(C#N)C1 26583,N1(c2snc(C(C)C)n2)CC(C)CN(C(c2ccc(S(N)(=O)=O)o2)=O)CC1C 26584,c1(CN(C2CCCN(C(c3cc(OC)ccn3)=O)C2)C(C)=O)cc(C)c(C)cn1 26585,c1(C(N(CC(C)NC(C2(SC)CCCCC2)=O)CC)=O)cc2cc(C)ccc2[nH]1 26586,C(=O)(CC1=CCOCC1)N1C(CNC(C(C)(c2cccs2)OC)=O)CCC1 26587,C(=O)(C(C)S(=O)(=O)C(C)C)NC1(CNC(C2(OC)CCCCCC2)=O)CC1 26588,c1(C(=O)NC(C2CCCN2C(=O)C=C2CCCC2)C)scc2c1CCCC2 26589,C1(CNC(CCC)=O)CCC12CCN(C(=O)COc1ccc(Cl)cc1C)CC2 26590,C(=O)(C(CN(S(C)(=O)=O)C)c1ccccc1)N(CCN(CC)CC)CC 26591,c1(N2CCOCC(CO)C2)c(Cl)cnn2cccc2c1=O 26592,c1(NC(c2scc(-c3c(F)ncc(C)c3)n2)=O)cc(Br)c(F)cc1C 26593,N1(C(CCC(C)C)=O)CCN(C(c2cc3n(n2)CCNC3=O)=O)C2COCC12 26594,c1(C(=O)NCC(C(C)C)NC(c2c(CC)scc2)=O)n[nH]c2c1COC2 26595,N1(C(CCc2c(C)noc2)=O)CCC2(C1)CN(C(C1CCCS1(=O)=O)=O)C2 26596,N1(C(C(CC)C)=O)CCC2CN(C(=O)C3=C(C)OCC3)CC2CC1 26597,C(=O)(C1CCc2ccccc21)N1CCC(N2CCN(C(C=CC)=O)CC2=O)C1 26598,C(=O)(C(F)(F)C(C)(C)O)N(C(C)CCC=Cc1ccccc1)C 26599,C1(F)(CNC(C(=O)N(C)C)=O)COCCN(C(C2COCC2(C)C)=O)C1 26600,C#CCC(C)(CC)C(=O)NCCN(C(c1cnc(C2CCC2)o1)=O)C(C)C 26601,C#CCC(C)(CC)C(=O)N1CC=C(C(=O)N2CCC(N(C)C)C2C)C1 26602,Cc1c(O)ccc(C(=O)NC2(C3CN(C(=O)CC(C)C(C)C)C3)CC2)c1C 26603,c1(C(=O)NCC23N(C(C4C(C)(C)CCC4)=O)C(CC2)CC3)ccsc1S(C)(=O)=O 26604,c1(C(=O)NCC(CC=C)NC(=O)CN2CC(C)(C)C2)ccn(C)c1CC 26605,c1(C(N2C(C(=O)O)C=CCC2)=O)cccc2nc(O)ccc12 26606,CC1(C)CCN(C(c2cncnc2)=O)CC1NC(c1cc(-c2ccns2)on1)=O 26607,c1(C(N2CCC(N(C(=O)CCCCC#N)C)CC2)=O)cc2ccncc2cc1F 26608,c1(-c2nc(OCC)oc2)nc(OCc2cccc(F)c2)nn1-c1ncnn1C 26609,c1(C(C)C)cncc(C(=O)N(C(C)CN(C(=O)C(C)C#N)C)C)c1 26610,C1(CNC(=O)Cc2ccsn2)CCCC(NC(c2ccsc2C(F)F)=O)C1 26611,N1(C(C(CC=CC)C)=O)CC(C)(C)C(NC(C2CCNC(=O)C2)=O)C(C)(C)C1 26612,C1(C(=O)OCC)CN(C(=O)C(=O)NC(c2nc[nH]n2)CC)CCC1(C)C 26613,c1(OC)cc(C(=O)NCCN(C(=O)CC2(O)CCCC2)C)cc(Br)c1OC 26614,C12(C(=O)NC(CCSC)CO)CCC(c3cccc(C(F)(F)F)c3)(C1)C2 26615,C(C(=O)Nn1cnnc1)(C(C)CC)NC(c1cc(=NC)[nH]cc1)=O 26616,C(=O)(CCC(C(C)C)NC(c1ocnc1C(C)C)=O)NCC(C1CC1)OC 26617,C1(N(C(CCC)=O)CCO)CCN(C(=O)CCNC(C2CCOC2CC)=O)C1 26618,N1(C(C(C=C)O)=O)C2CCC1C(F)C(NC(=O)C(c1cccc(C)c1)C)C2 26619,N1(C(c2c(C)n(C)nc2)=O)CCC2(CCCN2C(=O)CCCc2cccs2)C1 26620,CC(C)CC(C(=O)NC(CNC(c1cnn(CCO)c1)=O)C(C)C)NC(N)=O 26621,C1(C)(CC)CC(C(N2CCC(OCCNC(c3sc(C)nc3C)=O)C2)=O)CCO1 26622,c1(C(=O)NC(CC)CN(C(=O)C(C(C)C)SCC)C)ccc2nc(C)oc2c1 26623,S(=O)(=O)(c1ccc(Br)cc1N(C)Cc1cccc(Cl)c1)NCC1OCC(C)C1 26624,N1(C(CCC(=O)NCC)=O)CC(NC(C2CC=CC2)=O)CC(F)C1 26625,c1(C(=O)NC(C)CCNC(C2(CF)CC2)=O)cn(C)cc1C(F)(F)F 26626,C12(C(N3C(CNC(c4c(C)n[nH]c4C)=O)CC3)=O)CCC(CC1)C(C)O2 26627,N1(C(Cn2ccc(C)n2)=O)CC(NC(c2ccc(-c3ccco3)s2)=O)C2(CC2)C1 26628,c1(C(=O)NCC(CC)NC(=O)C(O)CC2CC2)cc(F)n(C)n1 26629,N1(C(C(CCC)N(C)C)=O)CC2CC(C(=O)N(C(C)C(C)(C)C)C)C(C2)C1 26630,C(C1=CCN(C(=O)C2=CCCOC2)CC1)NC(C(c1ccc(CC)cc1)C)=O 26631,N1(C(C(CC(N)=O)NC(C2C(C(=O)OC)CC2)=O)=O)CC2CN(C)CC2C1 26632,c1(C(N(CC(O)CNC(=O)CN2CCNC(=O)C2)C)=O)cc2nc[nH]c2cc1F 26633,N1(C(CN(c2ccc(N)c(F)n2)C)=O)C2CCC1CC(N1CCOCC1)C2 26634,C(CC(C)CC(=O)O)(C(F)(F)F)NC(=O)Nc1nccc(-n2c(C)ncc2)c1 26635,c1(C(N2CCC3CCC(C2)N3C(C23CC(F)(C2)C3)=O)=O)cnn2c1CC(F)(F)C2 26636,CCC(CC(C)C)C(=O)N1CC(C(=O)NCc2ccccn2)C2(CC2)C1 26637,Cc1ccc(Br)c(CC(=O)NCC23CC2CN(C(c2csc(=N)[nH]2)=O)C3)c1 26638,C1(CNC(c2c(C)nco2)=O)CN(C(C2CC2c2sccc2C)=O)CC12CCC2 26639,c1(NC(C(=O)NCCCCSC)=O)ccc(Br)cc1SC 26640,C1(C2(O)CN(C(=O)CC3CNC(=O)O3)C2)(CNC(=O)CCc2cnco2)CC1 26641,CN1CCCC(C)(C(N2CC(N(C)C(C3CCCN3N=O)=O)C(C)(C)C2)=O)C1 26642,C1(NC(C(C)=CC=C)=O)CC(CC(=O)N(C)CCc2cnc[nH]2)C1(C)C 26643,c1(CC)[nH]c(C(=O)NCC(C)(CO)NC(c2cc(C)nn2C)=O)nc1Cl 26644,c1(NC(C2(F)CN(C(CCOCC)=O)C2)=O)ccccc1N(C)C 26645,C1(CCNC(C(=O)NC(c2n(C)nnc2)C2CCCC2)=O)CCC(C)(C)CO1 26646,c1(OCC)cccnc1-c1nc(C2(COC(C)(C)C)CCC2)no1 26647,c1(C(N(C2CCC(NC(CC(=O)NCC#C)=O)C2)C)=O)noc2ccc(Cl)cc12 26648,Cc1cnc2n1CC(C(N1CC(NC(C3SCCCS3)=O)C3(CC3)C1)=O)CC2 26649,N1(C(=O)CC2CCCSC2)Cc2n[nH]cc2C1C(=O)N1CC2CCCC2C1 26650,c1(C(N2C(C)CN(C(=O)Cc3cnc[nH]3)C(C)C2)=O)ncn2c1CCCCC2 26651,c1(OC)ccc(C=CC(=O)NC2CC(C)N(C(c3ccc[n+]([O-])c3)=O)C2)c(C)c1 26652,c1(OC)cc(C)c(C(N2CC3CC3(CNC(C3(C)CC4CC4C3)=O)C2)=O)cn1 26653,N1(CN(CCC(=O)N(CC=C)CCO)CCO)CCCCC1=O 26654,c1(CC(=O)NC(C(=O)OC)C2C(NC(=O)OC(C)(C)C)C2)ccc(F)cc1 26655,C1(NC(c2cncc(C)c2Cl)=O)CCN(C(=O)CCOC2CC2)CC1(C)C 26656,Cc1nn(C)cc1C(=O)N(CCCNC(=O)C(C)Sc1ccc(Cl)cc1)CCO 26657,CC(C(=O)NCC1(C(=O)OCC2CC2)CC1)C(=O)CC12CC(C1)C2.NC 26658,c1(NC(CC2CCCN(C(C(CCCC)O)=O)C2)=O)c(I)cc([N+](=O)[O-])cc1I 26659,N1(C(C2(CO)CN(C(c3cnn(C)c3C3CC3)=O)C2)=O)CC2(CNC(=O)C2)C1 26660,C1(C(N(C)CC2N(C(CCc3cc(OC)no3)=O)CCC2)=O)CC(C)OC(C)C1 26661,N1(C(c2c(F)ccc(C)c2O)=O)C2CCC1CC(F)(CNC(C1CC13CC3)=O)C2 26662,C1(C(=O)NC(CNC(c2c(C)scn2)=O)(C)C)CCCC(F)C1 26663,N1(C(CNC(COC)=O)=O)CCC(c2n[nH]c(CNC(=O)C=CC3CC3)n2)CC1 26664,C(=O)(C(O)CC(C)(C)C)NC1(C)CCN(c2snc(C(C)(C)OC)n2)C1 26665,C1(NC(COC)=O)CCN(C(=O)CCSCC(=O)NC(C)=O)CC1C(C)C 26666,N1(C(C(C2CC2)NC(c2cc(C)c(C)nc2)=O)=O)CC2(C1)CN(C)CCO2 26667,c1(C(=O)NC23CCCC(NC(CC=CC)=O)(C2)C3)ccc(Cl)c(F)c1N 26668,c1(N2CCCC(CN(C(C3(OC)CCCOC3)=O)C)C2)cccc(F)c1[N+](=O)[O-] 26669,C1(C(=O)NCC2(OCC)CCC2)(CNC(C23COC(C2)C(O)C3)=O)CC12CCC2 26670,c1(C(=O)OC)cc(CN2CC(C(=O)NCc3ccncc3Cl)(N(C)C)C2)nn1C 26671,N1(C(c2cc(C)c(Br)s2)=O)C2CCC(C2)C1C(=O)NCc1nccs1 26672,c1(C(=O)NCCN(C(=O)Cc2cc(Cl)ccc2F)C)cncc([N+](=O)[O-])c1 26673,N1(CC(N2C(CN(C(CCC)=O)CC)CCC2)=O)C(=O)CCC1=O 26674,C(=O)(C1OCCc2ccccc21)NCC#CCNC(CC(C)OC)=O 26675,C=Cc1ccc(C(=O)NC(C)CC2CN(C(=O)C(C)(C)C#N)C2)cc1 26676,C1(NC(C(COC)C)=O)CN(C(C2CC(S(C)(=O)=O)C2)=O)CC12CCC2 26677,Cc1cc(C(N2CC(NC(=O)C(=O)NCC(F)F)C2)=O)c(C)cn1 26678,C1(C(=O)NCCSC(C)C)CN(C(=O)CCCSc2ccccc2)CCO1 26679,C#CCC(CC(=O)N1CCCC1C(C)CC)NC(c1cc(O)ccc1F)=O 26680,N1(C(CCCC(C)C)=O)CC2(CCN(C(=O)C(c3ccccn3)C)C2)C1 26681,c1(C(N2CCC(OC(=O)N(C)C)C2)C(=O)NC)ccc(F)cc1Cl 26682,C12(NC(c3ccc4scnc4c3)=O)CCN(C(c3cccc(=O)o3)=O)CCC1C2 26683,C1(c2onc(C)n2)CCCCN1C(C1CC(C(=O)N(C)C)C1)=O.c1(S)cccs1 26684,CCCS(=O)(=O)C(C)C(=O)N(C)CCN(C(=O)Cn1ncc(O)nc1=O)C 26685,CC1CC2(CC2)CN1C(C1OCCC1CNC(=O)Cc1cccnc1O)=O 26686,S(=O)(=O)(c1cccnc1Cl)NC(C1CCCCN1Cc1ccc(Br)cc1Cl)=O 26687,N1(C(C(CCC)(C)C)=O)CCC2(CC1)CC(CNC(=O)CC(C)CC)C2 26688,C1(C(N(CC(C)CNC(=O)Cc2nc[nH]n2)C)=O)CCC(O)CN1C 26689,C=CCCCC(C(=O)N1CC(OC(C)C)C1)NC(C1CC1CC(C)(C)C)=O 26690,CC(C)(C)CC(O)C(=O)NCC(c1cccc(O)c1)C(=O)O 26691,c1(C(C)NC(=O)NNC(=O)c2nccn2C)nc2ccccc2o1 26692,N1(C(c2c(CC)ccs2)=O)CCOCC1CNC(=O)C(C)Oc1ccc(F)cc1 26693,c1(C(N2CC3N(C(CCCCSC)=O)C(CC3)C2)=O)n[nH]c2c1CC(F)(F)CC2 26694,C(CN=c1cc[nH]cc1S(=O)(=O)N1CCC(C)(CO)C1)N(C)N(C)C 26695,C(CC(=O)NC1(CCC(=O)NCCc2cn[nH]c2)CCC1)=CC=C 26696,c1(C(=O)NC(C)CCNC(C2COCCN2C)=O)cccc2nc(O)[nH]c12 26697,c1(C(=O)NC2(C)CCN(C(C(C(C)(C)O)F)=O)C2)cc(O)c2ccoc2c1 26698,c1(C(c2n(C(C(=O)OC)C)nnn2)NCCCO)ccc(OC(F)F)cc1 26699,C1(C(=O)NCCC=CCCC)CN(C(=O)CCc2cnoc2)CC1CCOC 26700,N1(C(C2C(C)(CC)C2)=O)CC2CC3CC2C1C3NC(c1ccccc1OC)=O 26701,C1(NC(C2C(C)=CCS2)=O)CCN(C(=O)CCc2ncnn2C)CC1O 26702,c1(C(C)OCC)nc(-c2cccc(Cl)n2)nn1CC 26703,C(C(F)(F)C(=O)O)N(C(=O)C(c1ccc(F)cc1)CN)C 26704,C1(C(N(C2(C(=O)NC3(CCO)CCOC3)CC2)C)=O)CCCCC1(F)F 26705,C(CCCCC(=O)NCC(CC)NC(=O)CC1CN(C)C1)OCC 26706,c1(CN2CC3C(NC(Cc4c(C)n[nH]c4C)=O)C3C2)cc(O)cc2ccccc12 26707,Cc1cccc(C(N2CC(CNC(=O)Cc3ccc(F)cc3)C3CC23)=O)n1 26708,C=CCCCC(C(=O)NC1CC(C2CCC2)C1)NC(=O)CCCC#N 26709,Cc1cnccc1C(=O)NC(C)C(CO)NC(=O)C(c1ccc(Cl)cc1)(C)C 26710,c1(CCNC(=O)NC(c2ccccc2Cl)C)c[nH]c2ccc(O)cc12 26711,Cn1cnc2c(N3CC(O)(CCNC(=O)CN4CCCCS4(=O)=O)C3)ncnc12 26712,CCC(CCOC)C(=O)N1CC(OC)C(C(=O)NCCCCN(C)C(C)C)C1 26713,C1(COC)(CNC(c2cnncc2C)=O)CCCN1C(=O)C(C)CC1CC1 26714,N1(c2ncc(C(=O)OCC)nc2)CCN(C(=O)CN(C2CC2)CC)C(C)C1 26715,CC1(C)CN(C(C2CCCCS2(=O)=O)=O)CCC1NC(c1cc(F)cnc1Cl)=O 26716,c1(CC(=O)NCC(CC)NC(=O)CCCN=[N+]=[N-])ccc(S(=O)(=O)C(C)C)cc1 26717,N1(C(CC2(C=C)CCC2)=O)CCC(CN(C(=O)C(C)C(C)O)C)CC1 26718,Cn1cc(CCNC(=O)C(C2(O)CCC2)NC(C2CCCC2)=O)nn1 26719,C(=O)(C1=CCCCC1C)NC(CC(=O)NCCC=CCCC)C(C)C 26720,c1(SC)cc(C(=O)NCC(C)(C)CNC(c2cscc2SC)=O)n(C)n1 26721,C1(NC(C(CC=C)C)=O)CN(C(c2cccc(F)c2NC)=O)Cc2ccnn2C1 26722,N1(C(c2cc(COC)sc2)=O)CCCCC1C(C)NC(c1ccc(C)n1C)=O 26723,N1(C(C(CC)(C)OC)=O)CCC2(CCCC2CN=c2cccc([N+](=O)[O-])[nH]2)CC1 26724,C1(NC(CC(CN(C)C)O)=O)CCN(C(c2cc(F)ccc2Cl)=O)C12CC2 26725,C(=O)(C1Cc2ccc(Cl)cc21)NCC(C(C)(C)C)NC(=O)CCc1cc[nH]n1 26726,C=CCC(C)C(=O)N1CCOC(CNC(=O)CC(C)C2CCCCC2)C1 26727,c1(C(C(=O)NCCNC(CC(C)CN(C)C)=O)O)ccc(Cl)c(Br)c1 26728,c1(C(=O)NCC(CNC(c2ccn(CC(C)C)n2)=O)F)cccc2c1CCOC2 26729,c1(C(N2CC(C(C)NC(=O)CC(O)C3CC3)OCC2)=O)cc(Cl)ccc1N 26730,C(C(C)(C)CC(=O)N1CCC(NC(c2ncccc2O)=O)C1)OC(C)=O 26731,C1(CNC(C2CC23CCCC3)=O)CC2(CC2)CN1C(=O)C1=CSCS1 26732,N1(CC)C(=O)CCC1CC(=O)NC1CN(C(C2(c3n[nH]cc3C)CC2)=O)CC1O 26733,C(=O)(CCCC(=O)NC(C)C)NCC12CC(NC(C3N(C(C)C)CCC3)=O)(C1)C2 26734,N1(C(c2cccc3sccc23)=O)Cc2ccc(Br)cc2CC12CCC2 26735,c1(C(N(C2CCN(C(=O)COc3cccnc3)C2)CC)=O)ccc2cccnn12 26736,c1(C(N2CC(NC(C3C(C)(C)CC3)=O)CC3(C2)CC3)=O)[nH]c2ccccc2c1Cl 26737,CC(C(C)CO)NCc1ncoc1C1CNC1 26738,c1(CC(C(N2CCC(CNC(C3CC(CCO)C3)=O)C2)=O)O)cc(Cl)cc(Cl)c1 26739,C(=O)(C1=CCCCC1C)NC1CC2C(NC(C(C)N(C(C)=O)C)=O)C2C1 26740,c1(C(N(CCNC(=O)Cc2sc(O)nc2O)CC)=O)c[nH]c(C)c(Br)c1=O 26741,C1(NC(CCNC(=O)CO)=O)CCC2(CC1)CCN(C(C1CCC1)=O)C2 26742,Cc1snnc1C(=O)NC1CC1NC(=O)CC1CCOC1=O 26743,N1(C(C2N(C(C(C)NC(C)=O)=O)C3(CC2)CC3)=O)CC2(CCCCC2)C1 26744,c1(C(=O)NC(C(=O)N(C(C=C)C2CC2)C)CC2CCC2)cc(C)oc1C 26745,c1(CNC(CC)=O)ccc(CC(C)NC(=O)CC=CC(C)(C)C)cc1 26746,c1(C(=O)NC2CN(C(Cn3nnc(C)n3)=O)C(C)CC2)cnn2ccc(O)nc12 26747,N1(C(C(COC)N(C)C)=O)CC(CNC(=O)Cc2c(C)n[nH]c2C)C(C)C1 26748,c1(NC(C2C(NCc3ccc(OCCC)cc3)C2)=O)c(Cl)cc(Br)c(C)c1Cl 26749,c1(CC(=O)NCCCN(C(=O)CNS(C)(=O)=O)C(C)C)nccc2ccccc12 26750,C1(NC(C2CCCN2C(c2ncccn2)=O)=O)CCOC12CCCC2 26751,c1(CCSCC(=O)NC(CCNC(C=C(COC)C)=O)C)ccccc1 26752,C(CC(C)(C)C#N)(c1n(CC(=O)OC)nnn1)NCCC(=O)NC(C)C 26753,COn1cnc(C)c1C(=O)NC1CC(=O)N(C2CN(C(C3CC3C#N)=O)C2)C1 26754,n1(CC)ncc(Cl)c1C(=O)NCC(O)CN(C)C(C1CC1C(C)(C)C)=O 26755,N1(C(CSCCC(C)C)=O)CCCCCCC1C(=O)N(C)CC1CC1C 26756,c1(OC)cc(Br)c(NC(C2CC2C(=O)NCC(C)(C)C(N)=O)=O)cc1C 26757,C(=O)(C(C(C)(C)C)N1CCNC1=O)N1C(C)C(NC(c2cc(N)ccn2)=O)CC1 26758,n1(CC)nnc2c1C(C(=O)NCCc1cccc(F)c1)CN(C(=O)C(O)CCl)C2 26759,c1(C(N(C2CC2NC(=O)CN2CCCCC2)C)=O)cc(Cl)cc(Cl)c1Br 26760,O=S(=O)(c1ccc(NCCCC2CCC2)cc1Br)NC1CC2OCCCC12 26761,Cn1nc(O)cc1NC(C1CC1NCc1cscn1)=O 26762,CC1CN(C(=O)CCc2cccc(C#N)c2)C(C)CN1C(=O)CCc1nc[nH]n1 26763,c1(CC(N2C(CNC(C(C)CC(C)(F)F)=O)CC2)=O)cc(F)cc2c1OCOC2 26764,C(=O)(CC(C)CF)N1CCC(N(C(c2c[nH]c(=N)s2)=O)CC)C1 26765,N1(C(C(C)N(C(c2c(CC)c[nH]n2)=O)C2CC2)=O)CC2(C1)OC(=O)NC2C 26766,C=CCC(C)(C)CNC(c1conc1C(C)NC(c1cnccc1OCC)=O)=O 26767,CN=c1cc(C(=O)NC(C)(C)C(C)NC(=O)C(CN(C)C)C(C)C)cc[nH]1 26768,CC(CC(=O)N1CCN(C(C2CC2(C)Br)=O)CC12CCC2)CC(C)(C)C 26769,C1(C(=O)NCC(=O)OCC=C)CC12CC(NC(c1ccoc1)=O)C2 26770,N1(C(Cc2c(C)scc2)=O)CC2COCC2(C(=O)NCC(C)CN(C)C)C1 26771,Cc1cc(C(=O)NCCOCCC(=O)N2CCC2CN=[N+]=[N-])nc(O)c1 26772,c1(-c2c(OC)ccnc2)ccc(F)c(CN2CCCC(CC(=O)OC)C2)c1 26773,Cc1nc(O)nc(C)c1C(=O)NC1CCCC1CNC(c1ccc(N)c(Cl)n1)=O 26774,CC1CN(C(c2cc(O)nc(O)c2)=O)CCC1NC(=O)CCc1ccc(N)cc1 26775,C(=O)(CCC(=O)NCC1OCCC1C(=O)NC1(C)CC1(C)C)NCCC 26776,CC1CN(C(=O)Cc2c(F)cccc2Cl)CCC1NC(C1(CF)CCOCC1)=O 26777,C1(F)(C(=O)NCC(C(C)C)NC(=O)Cn2cnc(C(N)=O)n2)C2CCCC12 26778,N1(CCN2CC(CC)C(C)C2)CCCC(NC(=O)OC(C)(C)C)C1 26779,c1(C(N2CCC(OCCCC)CC2)=O)cc(CN=[N+]=[N-])cc(N=[N+]=[N-])c1 26780,N1(C(C=C(C)Cl)=O)CCCC(NC(C2CC(=O)N(c3ccccc3Br)C2)=O)C1 26781,C=C(Cl)CCC(=O)NC1CCN(C(c2cncc(N(C)C)n2)=O)C1 26782,N1(C(C(C)C=Cc2ccccc2)=O)CC2CCC1C(NC(=O)C(C)(F)F)C2 26783,N1(C(c2cc(Br)c(O)cc2F)=O)CCC2(CC1)CC(NCc1cnco1)C2 26784,c1(C(N(CC(CN(C(C(=O)N(C)C)=O)C)O)C)=O)ccnc2c1CCO2 26785,C(=O)(C(CC(C)C)C(C)C)NC(C1CCN(c2nc(COC)nc(C)c2)CC1)C 26786,c1(C(=O)NCC2(O)CN(C(=O)CCc3cn[nH]c3)C2)csc2cccc(F)c12 26787,c1(C(=O)NCC2(C(C)(C)O)CN(C(=O)CC3CCCC3(F)F)C2)cccc(=O)n1C 26788,c1(C(N2C(CNC(CC(C(=C)C)O)=O)CCCC2)=O)cn2nc(OC)ccc2n1 26789,CC1CC(C(=O)NCc2ccnc(OCC(F)F)c2)=NO1.C12CCN(CC1)C2=O 26790,N1(C(c2c(C)nc(C(F)(F)F)o2)=O)CCC2C(C1)CN2C(=O)Cn1nnc(=O)[nH]1 26791,C1(CC)CC(C(=O)NC2(CNC(c3ccc(=NC)[nH]c3)=O)CCCC2)CC(=O)N1 26792,C(=O)(C(C)(CC)CO)N(C)Cc1ccc(CNC(=O)Nc2ccco2)cc1 26793,c1(C(=O)NC(CCNC(C2(C)CC(=C)C2)=O)C(C)C)cc2ccccc2[nH]c1=N 26794,CCC1=NOC(CC(=O)NCC2C=CCN2C(c2csc(C)c2)=O)C1 26795,Cc1ncc(CNC(=O)C(F)CC2CN(C(=O)C(c3ccnn3C)O)C2)[nH]1 26796,N1(C(c2c(CC#N)ccs2)=O)Cc2nccn2CC(NC(C2CN(C(N)=O)C2)=O)C1 26797,c1(C(C(=O)NCC(CNC(COC(CC)(C)C)=O)C)C)cccc(F)c1 26798,c1(CC(=O)NCCCC(C)NC(C2OCCCO2)=O)c(Cl)cccc1Br 26799,O=C(CN=c1cc[nH]cc1)NCC1CC1NC(c1ccc(F)c(C(F)(F)F)c1)=O 26800,N1(C(COCC)=O)CCN(C(C23CCC(CO2)C3)=O)CC1C1CC1 26801,S(=O)(=O)(c1cc(C(=O)O)c(C)c(C)c1)NCC(CC(=O)OCC)N 26802,c1(NC(C(C2CCN(C(c3cccc(C)c3)=O)CC2)C)=O)cc(Br)c(Cl)cc1F 26803,C1(CC(=O)NC2(CCNC(C=CC(=O)OCC)=O)CCC2)CCOC1(C)C 26804,C(=O)(C(C#N)C(C)(C)C)NCC(C(C)C)(F)C(=O)NCC1(C)CCCC1N(C)C 26805,c1(C(N2CC3CCN(C(CN(CCC#C)C)=O)C3C2)=O)oc2ccccc2c1C 26806,CCC(C)(CC1CCCCC1)C(=O)N1CCN(C(=O)C(F)F)CC1 26807,c1(C(=O)NCC2C(NC(c3ccc(-c4ccccc4)[nH]3)=O)C2)ccccc1F 26808,N1(C(C(C#C)(C)C)=O)CCC2CCN(C(C3CNC(=O)C3)=O)C2C1 26809,C=CC(C)(O)CCCC(C)C(=O)N1CCCN(C(c2cc(Br)cn2C)=O)CC1 26810,C(=O)(C1=C(C#N)CCC1)N1CC(C(=O)NC2CCN(C(C)=O)C2)(CC)C1 26811,c1(C(CC(=O)OC)N(C2CCCC2NCc2cncc(Cl)c2)C)ccc(F)c(F)c1 26812,c1(C(N(C(CNC(=O)CSCC(F)(F)F)C2CC2)C)=O)cccc2c1COC2 26813,C1(CNC(CCCn2cc(CN(C)C3CC3)nn2)=O)CCSC(C)C1 26814,C(c1cccnc1)=CC(N1C(C(C)NC(C2CC=CCC2)=O)CCC1)=O 26815,C(CCC(C)(F)F)N(C(=O)CN(C(=O)CC1CC2CC2C1)C1CCC1)C 26816,C12(CNC(=O)CCn3ccnn3)CC1CN(C(c1nccnc1C(F)(F)F)=O)C2 26817,C(CN=c1[nH]c2c(c(=NCCCc3ncc[nH]3)[nH]1)COC2)c1n[nH]c(=N)o1 26818,O=C(Nn1ccnn1)C1C(c2ccccc2O)C1(F)F 26819,C(=O)(C(CC(C)C)CC(C)C)NC1CC(C)(NC(c2scc(OC)c2)=O)C1 26820,C=CCC(Cc1ccccc1)C(=O)NC(CNC(=O)CCC=C(C)C)CO 26821,C(CC(=O)N1CC2CC1C2CNC(C1CN(C)C(=O)N1)=O)(C(F)(F)F)OC 26822,Cc1ccc(C(=O)CCC(=O)N(C)CC2CN(C(c3cnccn3)=O)C2)cc1 26823,Cc1onc(C(=O)NC2CCN(C(c3cnn(CC(F)F)c3C)=O)C2)c1[N+](=O)[O-] 26824,Cc1cc(C(=O)NCC2CN(C(=O)Cc3ccco3)CCC2C)cc(C)c1O 26825,C#CCCCC(=O)N1CCN(C2CN(Cc3cnc(Cl)nc3)C2)CC1 26826,C(=O)(C(F)(F)C(O)C(C)C)NC1C(NC(Cc2ccc(OC)c(F)c2)=O)C1 26827,c1(C(N2C3(CNC(CCCC)=O)CCC(CC3)C2)=O)ccc(Cl)c2occc12 26828,N1(C(c2ccc(OCC=C)cc2)=O)CC(C(C)C(=O)O)OCC1C 26829,N1(C(c2c(C)ccnc2)=O)CCC(NC(=O)C(F)(F)c2csc(Cl)c2)C(O)C1 26830,c1(NC(CC(COC)NC(c2cc(C)ccc2I)=O)=O)c(C)cccc1C 26831,C1(C)(C(=O)NCCC(C)NC(c2nccn2-c2ccccc2)=O)COC(=O)OC1 26832,c1(NC(=O)CC2CCSCC2)cccc(NC(C23CCCC2CC3)=O)c1 26833,C(C1=NOC2CN(C(c3cc(C#N)c[nH]3)=O)CC12)NC(CSC(C)C)=O 26834,N1(C(C(C2CC2)OCC)=O)CC(CNC(=O)CSCCOC)C2(CC2)C1 26835,C(CC(=O)NC1CCC1CNC(C1CC1C(C)(C)C)=O)(OC)OCC1CC1 26836,CCC(C)C(C(=O)NCCN(C(=O)C(c1ccc(C(F)(F)F)cc1)(C)C)CC)N(C)C 26837,N1(C(CCCCOCC)=O)CC2(C1)C(NC(=O)C(F)F)CCS2(=O)=O 26838,Cc1cccc(C(C)C)c1C(N1CCC(CNC(=O)CC2C=CCC2)C1)=O 26839,CCC(C(=O)NC(CNC(=O)C(C)C(=O)N1CCOCC1)(CC)CC)C(C)C 26840,CCC(C)(C#N)C(=O)NCCCOCCNC(=O)CC1CCCC(C(F)(F)F)C1 26841,C1(C(=O)NCC(c2ccccc2)NC(=O)Cc2ccoc2)CCCCO1 26842,N1(C(=O)CC2C=CCC2)CCN(C(=O)Cc2ccon2)C(c2ccccc2Cl)C1 26843,Cc1cc2cc(C(=O)NCC(C)CNC(C34CC(CF)(CO3)C4)=O)c(Cl)cc2[nH]1 26844,C1(C(=O)NCC2N(C(CC3ON=C(C)C3)=O)CCCC2)(CO)CC2CCC1CC2 26845,N1(CCC)CC(NC(=O)C(CNC(=O)CN2C(=O)CCC2=O)N(C)C)CC1=O 26846,c1(C(N2CCN(C(=O)C=Cc3ccc[nH]3)CC2C(F)F)=O)cc2n(n1)CCCC2 26847,C1(C(=O)NCCCN(C(c2coc(CO)c2)=O)CC)CC(C(F)(F)F)CO1 26848,C1(NC(c2sc(C)c(Br)c2)=O)CN(C(c2ncccn2)=O)CCC1F 26849,N1(C(C(CC)NC(N)=O)=O)CCCCC(N(C)C(c2ccncc2)=O)C1 26850,C(C(CC(F)(F)F)NC(C1CC1F)=O)NC(COc1c(OCC)cccc1)=O 26851,C1(CC)CNC(C(N2CCC(c3noc(C4CCC4)n3)CC2)=O)CO1 26852,C1(CCN(C2CCCN(C(=O)C(=O)NC(C)C)C2)C(CCC)=O)CC2CCC1N2C 26853,c1(CN)ccc(Cl)c(NC(C2CCC23CCC3)=O)c1 26854,N1(C(C(C)CC2CCC2)=O)CC2(CCCN(C(=O)C=CC3(C)CCOCC3)C2)C1 26855,c1(OCC(=O)NCC2(F)CCN(C(C3CC=CCC3)=O)C2)ccc(F)nc1 26856,c1(OC)ccc(CC(=O)NC2(C)CN(C(=O)C(C)C3CCCO3)C2)cc1F 26857,c1(NC(c2cc(-c3cc(C)cc(F)c3F)ncc2)=O)ccc2ncnc(O)c2c1 26858,C#Cc1ccc(C(=O)NC(C)(C)CNC(=O)Cc2cccn2C)o1 26859,c1(C(N2CCC(CN(C(c3nc(CC)oc3C)=O)C)CC2)=O)cc(C)nc(O)n1 26860,C1(C(=O)Nc2c(C)ncnc2)CC2CCC1N2C(C1CCC1C#N)=O 26861,N1(C(C(C=C)O)=O)CCC(C(C)(C)CNC(=O)C(n2ccc(C)n2)C)CC1 26862,S(=O)(=O)(c1cc(C(=O)NC2CC3(C2)CN(C(C24CC(C)(C2)C4)=O)C3)co1)NC 26863,Cc1cc(C(N2CCC(C)(NC(=O)CC3CCC(C)(C)O3)C2)=O)ccc1Cl 26864,c1(C(=O)NC2CC(NC(C3CC4CC(O)C(C3)C4)=O)C2)cc2cc(Cl)cnc2o1 26865,CCC(C)(COC)C(=O)N1CCOC(CNC(=O)Cc2cc(C(F)(F)F)co2)C1 26866,C(C(=O)NOCC(N1CCC(C(C)(C)C)C1)=O)=CC 26867,C1(C)(COC)CC(NC(c2ccc(N)cc2Cl)=O)CN1C(=O)C=C1CC1 26868,c1(N(CCCC)C)nc(N2CCC(CCCC)C2)c2c(n1)CCOC2 26869,N1(C(c2cc(C)cnc2OC)C(=O)NCC=C)CCc2n[nH]cc2C1 26870,N1(c2c3ncn(CC4CCC(C)C4)c3ncn2)CC=C(c2ccc(Br)cc2)CC1 26871,CC1CN(CCNCC(c2ccc(OC(F)(F)F)cc2)C(F)(F)F)CC(C)O1 26872,C1(OC)(CNC(=O)CCC2CCC(C)O2)CN(C(=O)Cc2n[nH]c(C)n2)C1 26873,c1(CC)ncccc1C(=O)N(C(C)CNC(=O)CC1CCC(C)CO1)C 26874,c1(OC)cc2c(s1)CS(=O)(=NC(=O)c1cn(C3CCCNC3)nn1)C2 26875,c1(OC)cccc(OCC(=O)NC)c1.c1(C(C(=O)NC(C2CC2)=O)C)ccccc1 26876,Cc1cc(F)ccc1C(F)(F)C(=O)NCC1(C(F)F)CCN(C(=O)CC(C)C)C1 26877,CC1CCN(N2CCC(N)C2)CC1.C(=O)(CS(=O)(=O)N1CCN(C)CC1)NCC=O 26878,N1(C(CC(C=C)CC)=O)CCCCC2C1CCCN2C(=O)CC1(C)CCCC1 26879,C1(NC(C2CC2c2ccsc2)=O)CN(C(c2nocc2Cl)=O)CC1C1CC1 26880,Cc1cc(C(=O)N(CCCNC(c2cnn(C3CC3)c2)=O)C)cn1C(C)C 26881,CC1CN(C(c2ccn(C)c2)=O)CC1NC(C1(C(F)F)CCC1)=O 26882,CCCC(C(=O)NCc1c(OC)nsc1OC)N(CCN(C)C)C(C)C 26883,N1(S(Cc2c(C)nns2)(=O)=O)CC(=O)NC(C)C1 26884,c1(C(N2CC3C(C(=O)NCc4ncc(C)cc4)(C3)C2)=O)c(Cl)ccc(Br)c1F 26885,c1(C(N2CC(CNC(C3(CCC=C)CC3)=O)C(C)C2)=O)ccc(N)c(Cl)n1 26886,C(=O)(C1=C(C)CCCC1(C)C)N1CC(N(C(C(c2ccccc2Cl)OC)=O)C)C1 26887,Cc1ccc(C=CC(N2CCCC(C(C)NC(=O)CC(F)(F)F)C2)=O)nc1 26888,Cc1c(C(N2CC=CCC2C(=O)NOC2CCCC2)=O)nnn1C 26889,c1(CC)nccnc1C(=O)NC(C)CC(C)NC(C1CCCS1(=O)=O)=O 26890,C1(CC)CN(C(c2ccnn2C2CCC2)=O)CCC1NC(=O)CC(C)(F)F 26891,N1(C(c2ncc(C)o2)C(=O)NC2CC(F)(F)C2)CC2(C)COCC2(C)C1 26892,c1(C(=O)NCC2N(C(c3c(C)occ3)=O)CCC2)ccc2c(c1)NC(=O)C2(C)C 26893,C#Cc1cc(F)c(C(=O)N(C2CCC(NC(c3csc(C#N)c3)=O)C2)C)cc1F 26894,CCC(CC)(CC)C(=O)N1CCC(OCCCNC(=O)CC2CCC2(C)C)CC1 26895,c1(CNC(C2ON=C(CC)C2)=O)nn(C)c2c1CN(C(=O)C=C(C)C(F)F)CC2 26896,C1(NC(c2nc(C(C)(C)C)oc2)=O)CCC2(CC1)CC(O)C2 26897,Cn1cc2cc(C(=O)NC3C=CC(CNC(=O)Cc4ccco4)C3)ccc2n1 26898,C(CCC(C(=O)N(C)Cc1nncn1C)NC(c1csnc1Cl)=O)OC 26899,c1(C(=O)OC)ccccc1CC(=O)NC1CCCC1Cn1cc(C(C)(C)SC)nn1 26900,Cc1ccc(C(=O)NCCC(O)CNC(C2CC(O)C2)=O)c(N)n1 26901,c1(C(=O)NCC2C(CNC(C(C)NC(COC)=O)=O)C2(F)F)nc(O)sc1C 26902,N1(C(c2c(C)c(O)ccc2)=O)CC2CCN(C(=O)CCc3cccnc3)C2C1C 26903,C(CCCC(=O)NC(CCF)C(=O)NCCOC(=O)C1CC1)OCC 26904,N1(CCC)CCC(C(N2CC(OC)CC2CNC(=O)Cc2cc[nH]n2)=O)CC1 26905,C1(CC(N2CCC(NC(C)=O)C2)=O)CCN(C(=O)Cc2cnnn2C)CC1 26906,c1(C(N2CCCC(NC(C3(CO)CCCO3)=O)C(F)C2)=O)cccc2cncn12 26907,N1(C(C(c2cccnc2)N(C(C(C)C)=O)C2CC2)=O)CC(O)(C2CCC2)C1 26908,c1(OCCC(=O)NCCC(C)NC(C2C(F)(F)C23CC3)=O)cccc(F)c1 26909,c12cc(n[nH]1)C(=O)NC2.N1(C(C(C)C2CCC2)=O)CCCC1c1ncc[nH]1 26910,Cc1nc(C=CC(=O)NCC(C2CC2)NC(=O)CC2(C(F)(F)F)CCC2)cs1 26911,C1(C)(C(N(CC(C)NC(c2csc(-c3cccs3)n2)=O)C)=O)C(C)(C)C1(C)C 26912,C1(C(=O)NCCC#CCC)CCN(C(C2CN(C(C)C)C2)=O)C12CC2 26913,C1(C)(C(C(=O)NC)N(C2(CF)CC2)C)CCN1C(=O)OC(C)(C)C 26914,C1(CC)(CO)CCN(C(C2CCCSC2)C(=O)Nc2cccc(Cl)c2C)CC1 26915,N1(C(c2cnc(SC)s2)=O)CC2CN(C(c3ccc(C)nc3)=O)C2C1 26916,C1(NC(C(CC2CC2)NC(C)=O)=O)CCCC1(C)NC(C1CC1CC(C)C)=O 26917,C1(C(=O)Nc2ccc(OC)nn2)(Nc2ccccc2)CCCC2(CC2)C1 26918,C1(NC(C(CC)=CC)=O)CCS(=O)(=O)C12CN(C(=O)COCCN(C)C)C2 26919,N1(C(C2(C(=O)OCC)CCC2)=O)CCC(NC(=O)CC2(C)CC2)C(O)C1 26920,CCCCCCCC(=O)NC(CC)CCC(=O)N(C)CC1CCOCC1 26921,C1(C(N2CCC(CCC(=O)NC(c3nccs3)CC)C2)=O)CCCC1C1CC1 26922,CC(C)S(=O)c1ccc(C(=O)NCCC2(O)CN(C(C3CCCCC3)=O)C2)cc1 26923,N1(C(C(C)N(C(C)=O)C)=O)CCC12CN(C(=O)C(C)(C)NS(C)(=O)=O)C2 26924,O=C1Cc2cc(-c3nc(C(=O)Nc4ncc(Br)nc4Br)cs3)cnc2N1 26925,C1(NC(CCCC)=O)CCN(C(c2ccc(C#N)s2)=O)CC1C 26926,C1(NC(C2CC(CC)(CC)C2)=O)(CC(=O)CN2CCC(O)CC2)CCCCC1C 26927,C1(C(=O)NCC(C)O)CCN(C(c2cc[nH]c(=N)c2)=O)C1(C)C 26928,c1(C(=O)NC2CC(C)(C)N(C(C3CNC(=O)N3)=O)C2)cccc2nc(CO)[nH]c12 26929,N1(C(CC2C(C)CCC2)=O)CCCC(C)(CNC(c2scnc2C(C)(C)C)=O)C1 26930,c1(C(N(C(CCNC(C=CC(CC)C)=O)C)C)=O)cccnc1N1CCCC1 26931,N1(C(C2C(NC(C(n3c(C)ncc3)C)=O)CC=CC2)=O)CC(F)(F)CC1CO 26932,c1(CN(C)C)cc(C(=O)NC2CC2CNC(=O)C2=COCCO2)ccc1F 26933,N1(C(c2c(C)nc(Cl)cc2)=O)CC2CCC1CN2C(c1ccc(CO)cn1)=O 26934,C1(NC(=O)CCN2CCCC2)CN(C(c2cnc(O)o2)=O)C2(CCOC2)C1 26935,N1(C(CCC=C)=O)CC2(NC(c3ccnc(C(c4ccccc4)=O)c3)=O)CC1C2 26936,C1(C(N(C(C)CNC(=O)C=CCO)C)=O)CC2CC2C1 26937,n1(CCc2onc(-c3ccc4ccn(C)c4c3)n2)cnc2ccccc2c1=O 26938,c1(N2CCC(NC(C(C=C)(C)C)=O)C(F)C2)ncnc2c1CCO2 26939,C1(C(=O)OC)(C(=O)NCC(O)CN(C)C(c2cc(O)ncn2)=O)CCCCO1 26940,C(=O)(C(C)(C)CS(C)(=O)=O)NC1CC(C)CN(C(=O)C=Cc2ccn(C)c2)C1 26941,C(N(C)N1CCC(C)(CC(C)C)CC1)c1cccc(OCCOC)c1 26942,N1(C(CCC2CCC(=O)N2)=O)CCCC(F)(C(=O)NC2CN(CC(F)F)C2)C1 26943,N(C1c2ccccc2CC12CC2)C(c1ccc(SC(F)(F)F)cc1)C(=O)OC 26944,NS(=O)(=O)c1ccc(C(N2CCC(CCNC(C3CC3c3ccsc3)=O)C2)=O)o1 26945,c1(C(=O)NCC(CCNC(CCCC(C)=O)=O)(C)C)cc2c([nH]1)CCCC2 26946,c1(C(C(=O)NC2CC(F)(F)C2)N(CC(=O)NCCC)C)nc(Cl)cc(Cl)c1C 26947,c1(OCC)ncccc1C(=O)NC1CCC(NC(=O)C(C)(O)c2cscn2)CC1 26948,N1(C(C2=NOC(C)C2C)=O)CCC2CC(NC(=O)CC3(O)CCOC3)CCC2C1 26949,N1(C(COC(CC)C)=O)CCC(CNC(=O)Cc2cnsc2)C(CC)C1 26950,c1(OC)cc(Br)c2c(c1)CCN(C(=O)C(=O)N(CCC1(OC)CCOCC1)CC)C2 26951,N1(C(c2cccc(SCC#C)c2)=O)CCC2(CCCN2C(=O)C(C2CC2)OC)C1 26952,N1(C(C2(CCCC)CC2)=O)CC(NC2CC(CC(=O)OC)C2)C(SC)C1 26953,CCCC(C)(CC)C(=O)NC1CN(C(c2cc(C3(C)CC3)n[nH]2)=O)CC1F 26954,Cc1cc(N)c(C(=O)NC2CC(N(C(=O)C(C)CC(C)(C)C)C)C2)cc1C 26955,C(=O)(CC(C)(C)C(F)F)NC1C(NC(c2cc(OC)nc(OC)c2)=O)CCCC1 26956,N1(C(c2[nH]cc(C#N)c2)=O)CCC(CCNC(=O)CC2OCCCO2)C(F)(F)C1 26957,S(=O)(=O)(c1ccc(Br)cc1F)NC(C(=O)NC)Cc1cnc[nH]1 26958,C1(N(C(C2C(OCC)C2C)=O)CCOC)CCN(C(=O)COC)CC1 26959,C=C1CCC(C(=O)NCC2(CNC(=O)C(O)CC)CC2)CC1 26960,c1(C(=O)OCC)ccccc1C(N1CCCC1CC(=O)NCC1CCCCO1)=O 26961,CCCCCCC(CC)NC(C1CCCCCN1C(c1n[nH]c(C)c1O)=O)=O 26962,N1(C(C2N(C)CC(C)(C)C2)=O)CC=C(CC(=O)NCC23CCCC2C3)CC1 26963,N1(C(CC(CC)C2CC2)=O)CCC2C(C1)CN2C(c1csc(Br)n1)=O 26964,C(C1=NOC2OCCC12)NCC(C(=O)N(c1ccccc1)C(C)C)C 26965,CC1CCC(=CC(=O)N(C(C)(C(=O)NCc2cscn2)C2CC2)C)CC1 26966,CCC(CC(=O)NC(C)CN(C)C(C1CCN(C)C(=O)C1)=O)C(C)C 26967,C1(NC(C#CC2(C)CCCO2)=O)C2CCCN(C(=O)C#CC(C)(C)C)C2C1(C)C 26968,c1(NC(=O)NCCCC2CC(C)NC2)ccc(N2CCCCC2)cc1 26969,N1(c2nnc(C(=O)OC)n2CC)CCC2CN(C(c3ccccc3)CCC)C2C1 26970,N1(C(CN2CCN(C(CC=C)C(=O)OC)CC2=O)=O)CCn2c(C)nnc2C1 26971,C1(C)(C(C)C)CCCN1C(=O)CCC1CCCN1C(=O)Cc1cscn1 26972,C1(CN2CCCC(NC(C3(CC(=O)OC)CC3)=O)(CO)C2)CCC2(CCC2)CO1 26973,C(=O)(C1CSc2ccccc21)N1C(C)CN(CCC2CCCC2)CC1 26974,C(=O)(C(Cc1cn[nH]c1)NC(=O)Cc1cnns1)NCCC(C)SC 26975,C(C)(C(N)CC(=O)N1CCCC1C(=O)Nc1cccs1)SC 26976,N1(C(CCN(C)CC)=O)CC2(CCC(NC(c3ccnn3C(C)C)=O)CC2)C1 26977,N1(C(C(=O)NCCNC(COCCC)=O)CC(C)C)C(=O)c2ccccc2C1=O 26978,c1(C(=O)NCC2N(C(CCCOC)=O)CC2)ccc(CNC(C)=O)cn1 26979,C(=O)(C1=NOC2COC12)N(CC(CC)NC(=O)CN1CCC(F)(F)C1)C 26980,CC(C)(O)CC(=O)N1CCC(N(C)C(C2C(c3ccccc3)C2(F)F)=O)CC1 26981,CC1(C)CC(C#N)(CNC(=O)C(CC2CCC2)NC(C2CCCCC(=O)C2)=O)C1 26982,CS(=O)(=O)c1ccc(C(=O)NC2CCN(C(=O)C(F)C3CCC3)CC2)cc1 26983,C1(CNC(c2scc(C)c2)=O)CN(C(=O)CC2CCCC23CC3)CCO1 26984,c1(CC(N2CCN(C(c3ccnc(C)n3)=O)C(CO)C2)=O)coc2ccccc12 26985,c1(C(N(CC(C)(C)CNC(=O)CCn2ccnc2)CC)=O)cc(OC)ccc1C 26986,CC1(C)CC(NC2=NCC(C)(C(F)(F)F)N2)(c2nnnn2C)CNC1=O 26987,C(=O)(C1=C(Cl)CCC1)NC(COCC)C(=O)NC1CC1(C)C(F)F 26988,c1(OCC)ncc(C(=O)NC(C)(C)CCCNC(=O)Cc2ccno2)cc1Cl 26989,N1(C(C2(C(=O)OCC)CC2CO)=O)CCc2cc(NC(=O)C3CC3)ccc2C1.CC 26990,c1(C(N2CC(N(C(CC(C=C)(C)C)=O)C)C(O)C2)=O)ccc(C)c(Br)c1N 26991,c1(C(=O)NCCN2CCC(NC(C(C(C)O)C)=O)CC2)cc2n(c1)CCCC2 26992,c1(NC(C2OCCN(C)C2)=O)cc2c(cnn2C)nc1C(F)F 26993,c1(C(=O)NC(C2CCOC2)CNC=O)cccc(OCCF)c1.C1(CF)CC(CF)C1 26994,N1(C(C(C)NC(N)=O)=O)CCCC(C)(NC(C2CCC(=O)NC2)=O)C1 26995,N1(C(CCNC(CCCCOCC)=O)=O)CC2CCC2(CO)C1 26996,n1(CC(=O)NCC(C)CNC(c2cc(COC(C)(C)C)on2)=O)cc(Br)cn1 26997,c1(CC(=O)NC2CCCC(NC(C(C=C)O)=O)C2)cc(F)ccc1Cl 26998,N1(C(c2c(C)cco2)=O)CC2CCC1C1CN(C(c3occc3F)=O)CC21 26999,c1(CC(=O)NCC(O)CNC(C23CCC(C2)C3)=O)cccc(Cl)c1 27000,C1(C(=O)NC(C#C)CC2CCCC2)C(CC)CCN1C(c1csc(CC)n1)=O 27001,N1(C(c2cccc(F)n2)=O)CCCC(C2CCN(c3ncnc(Cl)c3F)C2)C1 27002,N1(C(CCCOc2ccc(CC)cc2)=O)CCC(C2(CO)CC2)CC1 27003,C1(SC)CCC(C(=O)N(C)CC2(NC(c3ccsn3)=O)CC2)C1 27004,Cn1ccc(=O)cc1C(N1CCOC(C(=O)Nc2nccc(Cl)c2Cl)C1)=O 27005,C1(NC(C(CCC)OCC)=O)CCCN(C(=O)Cc2cnoc2)CC1 27006,N1(C(c2nc(C(C)C)sc2)=O)CCCC(N(C(=O)CC2CCC(=O)N2)CCF)C1 27007,C1(N2c3cccc(c3)CCC2=O)CCNCCC1C.c1(OC)nccnc1C 27008,c1(C(=O)NCC(CC)NC(=O)COCC2CCOC2)ccnc2c(Br)cccc12 27009,C1(NC(c2cncc(C)n2)=O)COC2(CCN(Cc3cnn(C4CC4)c3)CC2)C1 27010,C1(C2CC2)(C(=O)NC2CCC(NC(CCC(=O)OC)=O)C2)CCOCC1 27011,C(=O)(C1CCc2nccn21)NC(C12CC1CCC2(F)F)=O.C12C3CN(CC13)C2 27012,c1(OCC)cncc(N2CCCC2Cc2ccc(C)cc2)n1 27013,c1(C(=O)NC(C2CN(Cc3ncncc3Cl)C2)C)ccc2scnc2c1 27014,c1(C(N2CCC(C(=O)NCCCCC(=O)NC)C2)=O)cc(C)nc(C)c1 27015,C(=O)(C(C)C(=O)OCCC(C)C)NC(CN(C(COC)=O)C)C 27016,c1(C(=O)NC(C(CO)NC(c2c(C)nc(CC)s2)=O)C)c(F)c(F)cc(F)c1F 27017,c1(C(=O)NCC2CCC(NC(c3cnc(C(C)=O)s3)=O)C2)nnn(C)c1C 27018,N(C(=NCC1(O)CCSC1)NC1CCCCC1)CCN(C(CC)C)CC 27019,N1(C(Cn2ncc(C)c2)=O)CC(C)(CNC(C2CC2C2CC2)=O)CC1(C)C 27020,C1(C(=O)NCC2(CNC(CN(S(CC)(=O)=O)C)=O)CCC2)OC(C)(C)OC1(C)C 27021,c1(C(=O)NCCCCC(C)NC(CSCC=C)=O)ccc2n[nH]cc2n1 27022,C(=O)(C1=CSCCO1)NC1CC(C)N(C(=O)Cc2n[nH]cc2Br)C1 27023,C(=O)(C(=O)CC(C)CC)N.c1(C(=O)NCCC=CCCC)ncoc1C 27024,Cc1c(C(N2CC3C(CNC(=O)C4=COCC4)C3C2)=O)cnn1C(C)C(C)C 27025,N1(S(CC)(=O)=O)CCCC1C(=O)NCC(c1ccccc1)NC(=O)C1=CCC1 27026,N1(C(C2(CC(C)C)CC2)=O)C2CCC1CC(NC(C1(C#N)CCOCC1)=O)C2 27027,CC1CCC(CNC(C23CC(C2)C(C)(C)O3)=O)N(C(=O)CSCCC(F)(F)F)C1 27028,N(C(=NCCc1ccc(Br)o1)NC1CN(C2CCC2)C1)C(CC)C 27029,CC1C2CCC(C2)C1C(=O)NCC1CCC(CC(=O)NCCc2nc[nH]n2)CC1 27030,N=c1nc(O)c(CC(=O)NCCCOCCNC(=O)C(F)=C2CCC2)c[nH]1 27031,CCCS(=O)(=O)C(C)C(=O)NCCCOCCNC(=O)CSc1nccn1C 27032,C1(NC(c2c(C)cns2)=O)CC2CC1CN(C(=O)C(C1CCCCCC1)O)C2 27033,CCC(F)C(=O)N(CCCN(C)C(C1CC=CC1)=O)C 27034,c1(CC(C(=O)N(CCN(C(C)C)C(C2C=CC=CC=C2)=O)C)C)cccc(F)c1 27035,N1(C(C(c2cccc(F)c2)C)=O)CC(CNC(c2n[nH]c(O)n2)=O)C(C)C1 27036,N1(C(C(F)=CCC)=O)CCCN(C(c2cnc(OC)nc2C(F)F)=O)CC1CO 27037,C(=O)(C1=CC2(CCN(C(C34C=CC(CC3)C4)=O)C2)C1)N(CC(F)Cl)C 27038,C1(CNC(c2scc(C)c2)=O)N(C(=O)CC2CC(C)(C)C(=O)N2)CCC1(C)C 27039,N1(CCN(C(CCC(C)C)=O)C=O)CCn2ccnc2C1.C(C(C)(C)S(C)(=O)=O)N 27040,C=CCCC(C(=O)NCC(CC)C(C)(F)F)NC(C1CCC1COC)=O 27041,c1(C(=O)NCC(C)NC(=O)CN(C)CCO)cc(Cl)c2n[nH]cc2c1 27042,Cc1cc(C(=O)NC2CS(=O)(=O)CC2NC(=O)CCF)c(Br)cn1 27043,c1(NC(=O)C=CC2CC2)cccc(C(F)(F)F)c1.c12nc(cs1)CC(=O)NC2=O 27044,C1(CNC(C(C)n2ccnc2)=O)CCC(N(C(=O)CC2CCCC(=O)N2)C)CC1 27045,c1(C(=O)OCC)ccc(-c2cn(C(C)CNC(C3CC4(CC4)CO3)=O)nn2)cc1 27046,C1(CCC)CN(C(c2ccc(C(O)CF)cc2)=O)CCN1C(C1CC1OC)=O 27047,c1(C(=O)NC(CC)CN(C(=O)CC2CCOC2)C)ccnn1C(F)F 27048,C(C)(CCCC(=O)NCc1c[nH]nc1C1CC1)NC(COCCC=C)=O 27049,C1(C(=O)NC2CON(CC)C2=O)CN(C(c2ccc(C)nc2O)=O)CC1(F)F 27050,N1(C(c2cc(CC)on2)=O)CC2CCC2(CCNC(=O)CSCCC(F)(F)F)C1 27051,c1(CCC)onc(C)c1C(=O)NCC1(C)CCN(C(C2(C#N)CCCO2)=O)C1 27052,C=CC1(C(=O)NC2CN(C)CCC2O)CCN(C(=O)C2=NOC(C)C2)CC1 27053,C1(CC)CN(C(c2cccc(C)c2)C(=O)NC)CC(=O)N1 27054,CC1CC(C)CC2(C1)NC(=O)N(CC(=O)N(C1CCOC3(CCCC3)C1)C)C2=O 27055,Cn1cc(C(=O)NCC2CCCC(NC(=O)CC3(C4CC4)CC3)C2)ccc1=O 27056,c1(C(=O)NC2C3CCN(C(Cc4nc(=N)[nH][nH]4)=O)CC32)cccc2c[nH]nc12 27057,CN=c1[nH]c(=NCCSc2c[nH]c(=N)s2)[nH]c(=NC2CC3CCC2C3)[nH]1 27058,c1(CC)ccc(C)cc1C(N1CC(Cn2cc(-c3c[nH]nc3C(C)C)nn2)C1)=O 27059,N1(Cc2c(=N)cc[nH]c2)CCCC(C(N2CC3CC(C3)C2)=O)CC1 27060,Cc1cccn2ncc(C(=O)NCCC3(O)CN(C(C4CNC(=O)N4C)=O)C3)c12 27061,C1(C(=O)NCC2CC(NC(CCOC)=O)C2)CC2CC(O)C(C1)C2 27062,N1(C(CCC#CC)=O)CC(NC(c2ncccc2O)=O)CC2(CC2)C1 27063,C1(CC(=O)NC(CCCNC(C=CC(CC)=CC)=O)C)CCC2CC2C1 27064,CN1CC(F)CC1C(=O)NCC1CCC(NC(C2CC2CC(C)(C)C)=O)C1 27065,C1(C)(CC)CCCN(C(=O)NC2CC(C#N)CC(C)(C)C2)CC1 27066,C1(CCNC(C2C(OCC)C2)=O)CCCN1C(=O)CSC(F)F 27067,c1(C(=O)NCC2CC(NC(c3c(C(C)C)ocn3)=O)C2)ccc2c(c1)CCC=C2 27068,C1(CNC(C2CCC(C)(C)CC2)=O)CCC(C)(C)CN1C(C1CC1(C)C)=O 27069,C1(CC(=O)N(CC(C)(C)CNC(=O)CCc2ncnn2C)C)CCCCC(=O)N1 27070,c1(C(=O)NC2CCCN(C(c3sccc3Cl)=O)C2)nnn2c1COCC2 27071,C(=O)(C1=NOCC1)NCC1(O)CC(NC(C(CC)Sc2ccccc2C)=O)C1 27072,C(C(CC(C)C)C(=O)NCCNC(N)=O)NC(CC(C=C)(C)O)=O 27073,c1(CCC(=O)NC(CCCNC(c2c(CC)c[nH]c2)=O)C)ccccc1[N+](=O)[O-] 27074,C1(C(N2CC(C(C)NC(=O)CCc3cnoc3)C2)=O)CCc2nncn2C1 27075,C1(N(C)C)(C(N2CCC(CCNC(=O)C(O)C3CCC3)C2)=O)CCOCC1 27076,c1(OC)cc(C(N2CCC2(C)C(=O)Nc2cc(C)c(F)c(C)c2)=O)cc(O)c1O 27077,C(=O)(C(C1CCC1)NC(=O)COC1CCC1)N(CCCCO)C 27078,Cn1nc(Br)c2c(NC3COC4(CCC(C)(C)C4)C3)ncnc12 27079,N1(C(C(CC)(C)C)=O)CC(C)CN(C(c2sc(N(C)C)nc2C)=O)C(C)C1 27080,C12(CNC(C(CC3CC3)NC(=O)CC34CCCC3C4)=O)CCC(CC1)O2 27081,Cc1ccc(-c2cn(C3CN(C(=O)CN4CCOC(C)(C)C4)C3)nn2)c(F)c1 27082,N1(C(C(C=C)OC)=O)CC2(C=C(C(=O)N3CC(O)(COC)C3)CO2)C1 27083,N1(C(C(C(=O)NC)(C)C)=O)CC(C(=O)N(C)CCc2nccs2)CCC1(C)C 27084,C(=O)(CC(CC)C(C)(C)C)NCC1(COC)CCCN1C(c1csc(Br)c1)=O 27085,C(CC(C)(C)C(=O)N(C(C(C)C)C1CC1)CC(=O)NCc1cnns1)OC 27086,S(=O)(=O)(c1cc(F)cc(F)c1)N1C2CC(N(CCC(O)CO)C)C(C2)C1 27087,C(=O)(CC1OB(O)c2ccccc21)N1C(C)CN(C(C2CC(=O)N2)=O)CC(C)C1 27088,C(C1c2ccccc2CC1C)NC(N1CCC(c2ccc(C)cc2)C1)=O 27089,c1(OC)cc(C(C(=O)OC)C2CN(C(C)=O)C2)c(F)c(F)c1F 27090,C1(CC2CC2)CC(O)CN1C(=O)CCCn1cc(C(N2C(CC)CCC2)=O)nn1 27091,n1(CC(=O)NCC2COCCN(C(=O)CSC3CC3)C2)nc2c(n1)CCCC2 27092,C1(CC(=O)NCc2c(C)n(C)nn2)CC(C)(C)CN1C(=O)CC(F)(F)F 27093,c1(OC)nc(Cl)ncc1Nc1ccnc(OC2CCCC(C)C2)c1 27094,c1(C(N2CC(CC(C)NC(=O)Cn3c(O)nnc3O)C2)=O)n[nH]cc1[N+](=O)[O-] 27095,CC1(NC(=O)CNc2ncccn2)CC(NS(C)(=O)=O)C1 27096,N1(C(C(C)(C)O)=O)CCN(Cc2sc(Br)nc2Br)CC1c1ccccc1 27097,C1(C(N2CC(OCCC(=O)NCC3CC34CCC4)C2)=O)CC(F)(F)C1 27098,N1(C(c2n[nH]c(C)c2O)=O)CCC2CN(C(=O)CCc3nc(C(C)C)no3)C2C1 27099,Cn1c(=O)n(C)c2cc(C(=O)NNC(C3CC4(CCC(N(C)C)CC4)C3)=O)ccc12 27100,C(CN=c1cc[nH]cc1S(=O)(=O)N1CCC2CC12)c1c(SCC)cccn1 27101,c1(OCCCCC(=O)NC(CC)C)ccc([N+](=O)[O-])cc1.c12csc(n1)CN2 27102,c1(C(=O)NC2CCCC(CC)C2)cc(Br)cnc1NC(=O)OC(C)(C)C 27103,N1(C(C2C(C)C2)=O)CCOCCC1C(=O)Nc1cnc(C(C)C)nc1 27104,CCC(F)(F)CC(=O)N1CCC(C)C(NC(=O)Cn2cnc(Br)c2)C1 27105,C(CNC(=O)Cn1cc(N)cn1)(C(C)(C)C)NC(C1(CC=C)CCC1)=O 27106,c1(C(N(C2CCCCN(C(C3CC3C(N)=O)=O)C2)C)=O)cc2cn[nH]c2cn1 27107,C1(NC(C2(CC=C)CC2)=O)CCN(C(c2cc(C)cc(Cl)n2)=O)CCC1CO 27108,C1(CNC(C2(CCCC)CCCC2)=O)CCN(C(=O)CCc2nncs2)CC1O 27109,N1(C(COCCOC)=O)CCN(C(c2cn(C3CCOC3)nn2)=O)C(C2CC2)C1 27110,C(CNC(C1CC1c1cccc(Cl)c1)=O)(C(C)(C)C)NC(C12CC(C)C1C2)=O 27111,C1(CN(C(C(CCC)OC)=O)C)CN(C(=O)CSCCOC)CC1(C)C 27112,N1(C(Cn2cc(CS(CC)(=O)=O)nn2)=O)CCCC(C(C)C)(NCC(=O)OC)C1 27113,C1(C(N2CC(O)(CCC)C2)=O)CCN(C(=O)CCN=[N+]=[N-])C(C)(C)C1 27114,N1(CC(=C)Cl)CCCC(C2CCN(C(C3CC34CCOC4)=O)CC2)C1 27115,N1(C(CCn2c(C)ncc2)=O)CC2CC(NC(C3CCC4(CCC4)O3)=O)C(C2)C1 27116,N1(C(c2cn(CC)nn2)=O)CCOC(CCCNC(=O)C(C)COC)C1 27117,Cc1ccc(CC(=O)NC2CCCC(CNC(=O)CC(F)(F)F)C2)cc1O 27118,c1(N2CCC(C)(NC(CC3CC(OC)C3(C)C)=O)C2)snc(C)c1C#N 27119,C(CC(C)(C)C)(C(=O)NC1CCC1NC(c1ccc(F)c(CC=C(C)C)c1)=O)OC 27120,O=C1CCN(CC(=O)NCCNC(=O)CC2CC=CCC2)CC1 27121,C(=O)(C(C)C(O)CC)NC(CC=C)C(=O)Nc1ccc(CO)cc1O 27122,C(C(C)C(=O)NOCC1CCOCC1)N(C(C(COC)(C)OC)=O)C 27123,CC(=O)CCCC(=O)NCCN(C1CCCCC1)C(C1CCCC1P(C)(C)=O)=O 27124,N1(C(c2ccn3c2CCCC3)=O)CC2CCCC(O)C2C1 27125,N1(C(C=CC)=O)CCC(O)(NC(N2C(C(=O)NC(C)(C)C3CC3)CCC2)=O)C1 27126,c1(C(N2CC(O)(CNC(C3CC(C)OC3)=O)C2)=O)cc2cc(Cl)ccc2o1 27127,c1(C(N(C)CC2CCCN(C(C(C(C)O)(F)F)=O)C2)=O)c(F)cc(F)c(F)c1F 27128,c1(C(=O)NC(CCNC(C2C(=C)CC2)=O)C(C)C)cc(N(C)C)ccc1N 27129,C(=O)(C1=CC2(CCOC2)C1)N(CC(=O)NCCCC1CCC1)CC1CCC1 27130,c1(C(N2C(CCCNC(c3ccno3)=O)CCC2)=O)cnc(C(F)(F)F)cn1 27131,Cc1c(C(=O)N(CC(C)NC(=O)CC2CCN(C)C2)C)nn2c1CCCC2 27132,N1(C(C2C(C)C2)=O)CC(NC(=O)C2=CCOC2)CC12CCC2 27133,n1(CC(=O)NCC2CC2CNC(C2CCC(CCO)CC2)=O)ccc(O)nc1=O 27134,N1(C(c2c(C)cc(C)s2)=O)CCC(CO)C(NC(=O)Cc2cccnc2C)C1 27135,C1(CC(=O)NCCN(C)C(c2ccnc3ncnn23)=O)CCCCCC1(F)F 27136,c1(C(N(C2CCCN(C(c3cc[n+]([O-])cc3)=O)CC2)C)=O)cccn(C)c1=O 27137,c1(OC)cccc(C(=O)NCC2CC(NC(=O)CCCC(N)=O)C2)c1O 27138,N1(C(CC(CC)C)=O)CCC(CNC(=O)C#CC2(C(F)(F)F)CC2)C12CC2 27139,C1(NC(c2c[nH]nc2CNC(c2cccc[n+]2[O-])=O)=O)CC1C1CCC1 27140,CCC(C(=O)NCC12CC(NC(=O)C(F)OC(F)(F)F)(C1)C2)n1ccnc1 27141,c1(NCCCCNC(N)=O)cc(OC(F)(F)F)cc(Br)n1 27142,Cc1cc(C)c(C(=O)NCC2C3CN(C(=O)CCN(C)C)CC23)c(C)c1Br 27143,Cc1ccc(C(=O)NCCC(O)CNC(C2C3CCCCCC23)=O)c(O)c1C 27144,c1(CC)nc(NC2CN(C(=O)CC3CCCC34CC4)CC2(C)C)c(C#N)cc1C 27145,C1(CC(N2CC(NC(c3cccc[n+]3[O-])=O)(CO)C2)=O)CCCC2(CC2)C1 27146,C1(NC(CCSCCC)=O)CC2CCC1CC2NC(c1csc2nccn12)=O 27147,c1(C(=O)OCC)oc2cccnc2c1NC(C1(CSc2cccc(F)c2)CC1)=O 27148,N1(CC)CC2(CCCN2C(C23CC2CN(C(c2ccsc2C)=O)C3)=O)C1 27149,C1(C(N2C(C(=O)OC)CC2)=O)CCCN1C(c1ccc(Cl)o1)=O 27150,c1(C(N2CC(NC(C3CCOC3)=O)CC(C)C2)=O)ccc2ccn(C)c2c1 27151,C1(F)(C(=O)NCCc2onc(C)n2)CCCN(C(=O)C=C2CCC2)C1 27152,Cc1c(O)ccc(C(N2CCCC(CN(C)C(C3(C(C)C)CCC3)=O)C2)=O)c1C 27153,C1(NC(CCc2cc(C)on2)=O)CC2CCC(C1)N2C(C1COC(=O)O1)=O 27154,C(=O)(C1=CCCCO1)NC1CN(CC2(C(=O)NC3CC3)CCCO2)C1 27155,C(=O)(CC1OCc2ccccc21)NCCNC(=O)C(F)CC1CCC1 27156,C1(C(N2CC3=C(CN(C(CCCC(=O)OC)=O)C3)C2)=O)C2Cc3c(Cl)cccc3C12 27157,C1(C)(C(NOCC2CC(=C)C2)=O)CN(C(=O)C(F)F)C(C)(C)C1 27158,CC1CN(C(=O)Cc2cccc(F)c2)CCC1C(=O)NC1CC(=O)N(O)C1 27159,CC1CC(N(C)C(C2CSCCN2C(=O)CCN2CCOCC2)=O)CC(C)C1 27160,N1(C(C(CNC(c2c(C)scc2)=O)(F)C(C)C)=O)CCN2CC(F)CC2C1 27161,c1(C(N(C2CN(C(C3CC(CF)C3)=O)CC2F)C)=O)cnc2c(C#N)cnn2c1 27162,CC1(C)CC(NC(=O)CSC(F)(F)F)CN(C(C2CC(F)(F)C2)=O)C1 27163,Cc1cccc(CCNC(C2CC2c2ccccc2-c2cncn2C)=O)n1 27164,c1(CN2CC3(C(C(=O)NCC(=O)N(C)C)C3)C2)cc(Br)c(F)cc1Cl 27165,C1(C(=O)NCC2CCCN(C(C3OCCN(C)C3)=O)C2)CCC(=O)N(C)C1 27166,c1(C(=O)NCCCCCNC(CC(CC)C2CC2)=O)cc2ccccc2n1CC 27167,C(C(O)C(=O)NC1CN(C(=O)CNC(=O)CC(C)C)C1)OC 27168,c1(CCC)nnc(S)n1CC(=O)NC1(C(C)NC(c2cnc(O)n2CC)=O)CC1 27169,C1(NC(C2CCCN(C(C)=O)C2)=O)CCCC12CN(C(c1ccn(C)c1C)=O)C2 27170,C(CC(C(=O)NCC(=C)Br)NC(=O)COCC(C)C)=CC 27171,N1(C(c2cc(C(C)=O)c(C)o2)=O)CCC2CN(C(C3CC(N(C)C)C3)=O)CCC12 27172,N1(C(C(CCOC)(C)C)=O)CCCC(C2CN(C(C3(S(C)(=O)=O)CCC3)=O)C2)C1 27173,c1(C(=O)NCC(C(=O)N(C(C=C)C)C)(C)CC)cn2ccccc2n1 27174,C12(CC(=O)NCC#CCOC)CCC1CN(C(c1csc(C)c1)=O)C2 27175,c1(C(N(CCOCCNC(CC(CCCC)O)=O)C)=O)cccc2c1OCC2C 27176,C1(C(N(CCCNC(c2ccc(Cl)c(N)c2)=O)C)=O)C2CCCCCCC12 27177,CCCCCC(O)C(=O)NCC1CN(C(C2COCCN2C)=O)C1 27178,N1(C(C(CCNC(CCCOCCC)=O)O)=O)CCCCC(C)(F)C1 27179,c1(C(=O)NCCCN2CCC(NC(c3cc[nH]n3)=O)C2)cc(F)cc([N+](=O)[O-])c1 27180,C12(CNC(c3c(OC)c[nH]n3)=O)CCC1CCN2C(c1cnc(O)s1)=O 27181,C1(CNC(c2c(CC)ocn2)=O)CN(C(=O)Cc2ccc(F)cc2F)CCC1C 27182,CC1C(NC(=O)COCCCF)CCN1C(=O)CCCCN1CCOCC1 27183,CCC(CN(C1CC(OC)(OC)C1)CCCOC)CCC1CCCC1 27184,N1(C(Cc2nc(C)oc2)=O)CC(C2CCCCN(C(=O)Cc3ccns3)C2)C1 27185,C(C)(C)(CC(C)NC(C1(NC(=O)C=Cc2cc[nH]n2)CSC1)=O)OC 27186,c1(C(=O)NC(C)CN(C)C(C2(C)CCCO2)=O)ccc(-c2ccccc2)nc1O 27187,c1(CNC(C2(C)C(C)(C)C2)=O)nnc2n1CCN(C(c1ccc(Cl)c(N)c1)=O)C2 27188,Cc1sc(C(=O)NCC23CC2CN(C(=O)CN(C)C(C)C)C3)nc1O 27189,c1(C(=O)NC2CC2CNC(C2CCCOCC2)=O)ccc2c(c1)CCCCS2 27190,C1(NC(=O)OC(C)(C)C)CCCOC1c1cn(-c2ncccc2Br)nn1 27191,N1(C(CC=C=C)=O)CCCC(NC(c2coc(Cl)n2)=O)CCC1 27192,Cc1cc(O)cc2c1CN(C(C1CCCN1C(=O)CCc1ccncc1)=O)CC2 27193,c1(CCC(=O)N(C)CCNC(=O)CCc2ncccn2)nc2cc(Cl)ccc2s1 27194,n1(CCC)cc(C(=O)NC2CC(N(C(=O)Cc3cccn3C)C)C2)c(C)n1 27195,C1(C#N)(CC)CCN(C(=O)CCNC(c2cc(C3CC3)[nH]n2)=O)CC1 27196,c1(C(=O)O)cccc2c1CN(N1CCC(Br)CC1)CC2 27197,CC(C(CO)NC(c1cnc(C2CC2)[nH]1)=O)NC(=O)C(c1cccn1C)=O 27198,c1(C(c2n(C3CC(C(=O)OC)C3)nnn2)NC2CCC2CF)sc(C)c(Br)c1C 27199,Cc1ccc(C(N2CC=CC(NC(c3cccn3C)=O)C2)=O)c(F)c1F 27200,c1(CC)cc(O)ccc1NC(=O)C(C)(C)C(C)NC(c1ncn(CC)n1)=O 27201,c1(CC(=O)NC(CC=C)CNC(=O)Cc2cccc(Cl)c2)ccc(C)cc1Cl 27202,c1(C(=O)NC2CCN(C(c3c(SC)ccs3)=O)C2)cc2c(cn1)OCCC2 27203,C1(NC(c2cn(CC(N)=O)nn2)=O)(CO)CCCN(C(=O)CCn2cnnn2)C1 27204,CCC(CC)C(C)C(=O)NCCCC(C)(C)NC(=O)CCC1CCC(C)O1 27205,N1(Cc2c(C)c(C#N)[nH]c2)CCC(F)(F)C(C(=O)NC(c2ccccc2)C2CC2)C1 27206,c1(C(=O)NC2(C)CC(NC(C3(C)N(C)CC(O)C3)=O)C2)cc(F)c(Cl)cc1F 27207,N1(C(C(C(CC)C)OC)=O)CCCCCC(NC(c2cc(C)c(F)c(C)c2)=O)C1 27208,c1(C(=O)NC2C(NC(C(C)O)=O)C2)ccc2c(c1)N(C)C(=O)CC2 27209,Cn1cc(S(N)(=O)=O)cc1C(N1CC(NC(=O)CCCN=[N+]=[N-])CC(C)(C)C1)=O 27210,N(C(=NCC1=CCCOC1)NCc1ccc2c(c1)CCC2)CCSC 27211,C1(C)(CNC(c2c(C)nco2)=O)CCN(C(=O)CSCc2cccnc2)CC1 27212,C(C(C(C)C(C)C)NC(=O)COCCCF)NC(c1c(CCC)nsc1N)=O 27213,C1(COC)(NC(C2CC2C(N)=O)=O)CCN(C(C2CN(C(N)=O)C2)=O)CC1 27214,C(=O)(CC(=O)N(CC(=O)N(C1CC1(C)C)C)C1CC1)NCC 27215,c1(CCC2C(=O)CCCN(C(=O)NC3CCC4CC34)C2)ccccc1 27216,C(C(CC(C)C)C(=O)NCCCc1ccccc1)NC(c1cnn(C=C)c1N)=O 27217,CCC(CC(=O)N1CC(F)(CNC(C2CN(C)CCO2)=O)C1)CC(C)C 27218,CCC(C)(C)CCCC(=O)NCCC(C)(C)NC(C1CCCC(=O)N1)=O 27219,O=C1CN(C(C2CC23CC3(F)F)=O)C(C(=O)NCCCc2cncnc2)CN1 27220,Cc1cc(C)c(C(=O)NCC(C)C(=O)NCCc2nccs2)s1 27221,C1(CCNC(=O)C(C)c2ccsc2)(OC)CN(C(=O)CC2CC(=O)C2)C1 27222,C1(CNC(CSCC=C)=O)CCCN(C(=O)C(C)Cn2ccc(C)n2)C1 27223,C(=O)(C#CC(C)(C)C)N(C1CCN(C(c2ccccc2-n2cccn2)=O)C1)C 27224,c1(C(N(CC(F)(F)F)CC#C)=O)cn(C2CCCNC2)nn1 27225,C1(C(N2CC(C(C)NC(c3ccon3)=O)OCC2)=O)CN(C)CC(C)O1 27226,Cc1ncc(C(=O)NCC2CC(F)CN2C(=O)CC2CCOC2=O)n1C(F)F 27227,c1(N2CCC(OCC)C(C)C2)nc(=NCc2cc[nH]n2)[nH]c2c(C)nn(C)c12 27228,CCCCC(F)(F)C(=O)NCCC1CCCN1C(=O)CCC1CNC(=O)N1 27229,C(CC(C)C(=O)N1CC(c2ocnc2CNC(c2sccc2C)=O)C1)OC 27230,c1(N2CC3C(CC)(C3)C2)nc(=NCC2(C)NC(=O)NC2=O)[nH]c2c(F)cc(F)cc12 27231,C1(c2onc(Cc3n(C)ccn3)n2)CC12CCSCC2 27232,c1(CC)cc(CC)nc(N2CCC(C)(NC(=O)C(N3CCOCC3)C)CC2)n1 27233,N1(C(COCCCC)=O)CC2CCC(CNC(C3CC3(C)CC)=O)(C2)C1 27234,C(C(CO)C(C)CC)NC(C1C(CCC)CN(C(=O)C(C)(C)N(C)C)C1)=O 27235,C1(C(C)CNC(=O)CC2CCCN2C)CCN(C(=O)Cc2cc(Cl)n(C)n2)CC1 27236,C12(Cn3cc(CCC(=O)NCCC(COC)(C)O)nn3)CCCC1C2(F)F 27237,C1(NC(c2nc3c(s2)CCC3)=O)CCN(c2nnc(C(F)(F)F)s2)CC1O 27238,c1(C(=O)NCC(CCCC)NC(c2ccc[nH]2)=O)cnc(O)c2ncccc12 27239,CCCCC(CNC(=O)CCCc1ccccc1)NC(=O)CC1CCC12CCC2 27240,c1(NCC2CCN(C(C3CCOC3)=O)C2)ncnc(Cl)c1[N+](=O)[O-] 27241,N1(C(C(C)(C)O)=O)CCCC(CC(N2CCC(CN(C)C)CC2)=O)CC1 27242,Cc1nn(-c2ccncc2)cc1C(=O)N(CCCNC(=O)C(C)(C)CF)C 27243,C(=O)(CCC(=O)N(C(C)CNC(=O)CCCCN1CCCCC1)C)NC 27244,CCCCCC(C)CC(=O)NCc1cc(C(=O)N(c2cccc(C)c2C)C)cs1 27245,C(=O)(CC(CC)CC(C)C)NC(CCC(=O)NCCC(=O)OC(C)C)C(C)C 27246,N1(C(C2CC(NC(c3c(C)cc(F)cc3C)=O)C2)=O)CCc2nc(Cl)ccc2C1 27247,c1(C(N(CCCNC(=O)C=CS(C)=O)CC)=O)cc2ccncc2c(O)n1 27248,c1(C(C)=O)ccc(C(N2CCN(C(c3c[nH]c(Br)c3)=O)C(C)C2)=O)cc1F 27249,CCC(CCC(=O)NCC(O)Cn1cccn1)NC(c1nc(CC)oc1C)=O 27250,C1(NC(C(C)c2ccco2)=O)CN(C(=O)C=CC2(C)COC2)CC1C1CC1 27251,N1(C(CCC(C)(C)C)=O)CCOCC(C)(CNC(C2CNC(=O)C2)=O)C1 27252,Cc1cnc(CC(=O)NC2CCN(C(c3cnc(Cl)s3)=O)C2)o1 27253,C12(NC(CC(CC)SC)=O)CCCCC1CN(C(=O)CCCS(N)(=O)=O)C2 27254,N1(C(C(C)n2cncn2)=O)CC2CC2(C(=O)NOCCF)C1 27255,CC(c1ccccc1)=CC(=O)NC(CC(=O)N1CCC(C)C1)C(F)F 27256,c1(C(=O)NC2CC(F)(CNC(CC3C(C)C3)=O)C2)cccc(F)c1C#N 27257,C1(C(N(C(C)(C)C(=O)NC2CSC2)C)=O)CC1(F)Cl 27258,c1(C(C(=O)NCC2CCN(C(=O)C=Cc3nccs3)C2)O)cc(Cl)cc(Cl)c1 27259,C1(NC(c2c(C)ncnc2)=O)(CO)CCCN(C(c2ccccc2Br)=O)C1 27260,C=CCCCCCC(=O)N1CCCC(C(C)NC(=O)C2CC2)C1 27261,c1(C(=O)OC)cc2c(s1)CCOC2CNCC1CCCCC(O)C1 27262,C1(SC)CN(C(C2(OC(C)C)CCCCC2)=O)CC1NC(=O)C=C(C)C 27263,C(=O)(C1=NOC(C)C1C)N1CC2C(CC(N3CCC(SCC)CC3)=O)(CC2)C1 27264,N1(C(CCC(C)(F)F)=O)CCc2sc(CNC(=O)C=C3CCCCC3)nc2C1 27265,C1(C(=O)NCCC2N(C(C3CN(C(N)=O)C3)=O)CCOC2)CS(=O)(=O)CC12CC2 27266,c1(C(=O)NC2CC3(C2)CC3C(N2CCC3(C2)CC3(F)F)=O)cccc2ccnn12 27267,N1(C(C(CC(F)F)NC(=O)C(C2CC2)C2CC2)=O)CCN2C(=O)OCC2C1 27268,C#Cc1cncc(CN2CCN(C(=O)CN3CCCCC3)C(CC)C2)c1 27269,N1(C(CCOCC#C)=O)CCC(C)C(NC(c2ccc(NC(C)=O)cc2C)=O)C1 27270,c1(CC)ccc(C(=O)OC(C(c2ccc(C(C)=O)cc2)=O)C(C)C)cc1[N+](=O)[O-] 27271,c1(NC(CC(=O)NC(C)C)C)nc(N2CCCNC(=O)CC2)nc2sccc12 27272,CC(C)CCCC(C)CNC(C1CC(C)CN(C(c2cncc(F)c2)=O)C1)=O 27273,CCCCC(C)(F)C(=O)NCC1CCC1NC(=O)C1=CCCCO1 27274,c1(-c2c(C)n[nH]c2)ccc(CNC(C2CCC2)=O)c(F)c1 27275,c1(C(=O)NC2C(C)(C)C(CC(=O)NCc3cc(Cl)ccn3)C2)cncc2[nH]ccc12 27276,C(=O)(C(F)(F)C1(n2cncn2)CC1)NC(C1CC12CC2)CNC(C)=O 27277,N1(C(C(COC)C)=O)CCCC(O)(CNC(c2ccc(C(F)(F)F)cc2Cl)=O)C1 27278,C(=O)(C(C)C(C)(C)O)NC1CCCN(C(CCSc2c(OC)cccc2)=O)C1 27279,c1(C(=O)NCCCC2N(C(CC(C)SC)=O)CCCC2)cccc2nncn12 27280,c1(C(=O)NCc2cccc(CN(C(=O)CCF)C)c2)n[nH]cc1[N+](=O)[O-] 27281,C1(NC(c2csc(C)c2C2CC2)=O)CCCC12CN(C(=O)Cn1ccnc1C)C2 27282,C(=O)(CC(C)(C)C#N)N.c1(CC(=O)OC)ccoc1C(=O)NC1(CNC(C)=O)CC1 27283,c1(C(CNC(CC2CC(=O)C2)=O)NC(c2cnccn2)=O)ccccc1 27284,C1(CNC(CCC=CC)=O)CN(C(=O)C(C)Cc2ccncc2)CC2(CCC2)O1 27285,N1(C(C(CSC)O)=O)CCCC12CCC(NC(=O)CN(C)C1CC1)CC2 27286,C(CC(F)F)(C(=O)NCc1ccccc1F)NC(CC1C(C)(C)COC1)=O 27287,N1(C(C(=O)NC(C2N(C(CSCC)=O)CCC2)(C)C)C)C(C)CCC1C 27288,CC(C(CO)NC(=O)CCc1cncn1C)NC(c1cc(C2CCC2)[nH]n1)=O 27289,c1(CC(=O)N(C(c2ccccc2)CCC)C)ccc2c(c1)CNC2=O 27290,C1(NC(C(CSC)C)=O)CCSC12CN(C(=O)CCc1ccc(O)c(F)c1)C2 27291,CCCCCC(CC)C(=O)NC1CC(NC(c2ccc(Br)cc2C)=O)C1 27292,c1(C(N2C(C)(C(=O)Nc3cccc(OC)c3)CCC2)=O)cc(Cl)cnc1Cl 27293,C(=O)(C(CN=[N+]=[N-])NC(=O)C(C)NC(=O)N(C)C)NC(c1cnsc1)C 27294,C1(C(=O)NC(CC)CC(=O)NC(COC)C(=O)OC)CCC2(CCC2)CC1 27295,c1(OC)ccc(C(=O)NC2CC2NC(c2cc(C)cc(F)c2)=O)cc1C(C)C 27296,CC1(CNC(=O)CN2CC=CC2)CC(NC(c2ncsc2Br)=O)C1 27297,Cc1noc(CC(C)C)c1C(=O)NCC(C1(O)CCN(C(=O)COC(C)C)C1)C 27298,c1(C(=O)NC(C(C)NC(c2cc(N)cnc2Cl)=O)C)ccc(Cl)c2ccccc12 27299,C12(C(=O)OC)CCCC1CCN2C(=O)Cn1cnc([N+](=O)[O-])c1 27300,C1(C(C)NC(=O)C(c2c[nH]nc2C(F)(F)F)C)CCN(C(=O)C=CCF)CC1 27301,CC1CN(C(=O)C2=CCCCC2)CC(CCNC(=O)C(c2ccn(C)n2)C)O1 27302,c1(C(=O)NC2CC2NC(c2noc3c2CCCC3)=O)ccc2cccnc2c1 27303,C(CCCCCO)C=O.N1(C(CCN(CCCO)C)=O)CCCC1C(C)(C)C 27304,c1(NC)ccc(C(N2CCC(SC)C2C(N2CC(OC(=N)O)C2)=O)=O)cc1 27305,C(=O)(CCCCC(=O)N1CC(CNC(=O)CC2(C)CC2(F)Cl)OC(C)(C)C1)NC 27306,CC1(F)CCC(C(N2CCC(CNC(=O)C(F)(F)c3cncs3)C2)=O)CC1 27307,CC(C)C(CC(=O)NCC(C)CNC(c1cnc(C2CCC2)s1)=O)C(C)C 27308,CC#CCCCC(=O)N1CC(C(=O)NC(CCC(C)(C)C)C(=O)OC)C(F)(F)C1 27309,c1(CNC(C(C)O)=O)ccc2c(c1)CCN(C(c1coc(SC)c1)=O)C2 27310,C1(C)(CNC(C2(C)C(C)CCC2)=O)CCCN(C(c2ccc(F)s2)=O)C1 27311,C1(C(=O)NC(C2CN(Cc3ccc(Cl)cc3)CCO2)C)CCc2nncn2C1 27312,CCCCC(C)CCC(=O)N1CCC1CNC(C1(CCCC)CCCC1)=O 27313,c1(OC)cccnc1C(=O)NC1(C)CC(NC(=O)CCC2CCCO2)C1 27314,c1(CCC)c(C(=O)NC2CC(NC(=O)CC3(O)CCCC3)C2)cnn1CCO 27315,Cc1ccc(C(=O)NC2CC(CNC(=O)CS(C)(=O)=O)C(O)C2)c2c1CCCN2 27316,C(C)(C)(CC=CC(=O)NC1CC(SC)C1)NC(CCOC)=O 27317,C(=O)(C1=COCCC1)N(CCCNC(=O)CCC(=O)Nc1ccccc1F)CC 27318,C(=O)(CC(C(F)F)NC(C1CCCC1F)=O)N(CCC(N)=O)C 27319,c1(C(=O)OCC(CCOC)(C)C)cc(O)nc(C(F)F)n1 27320,C1(CC)CN(C(=O)Cn2cc(C(C)O)nn2)CCC1NC(c1cc(C)oc1C)=O 27321,Cc1ncnc(C)c1OCC(=O)N(CC(C)CNC(C12CC(CCO1)C2)=O)C 27322,c1(NCC2(C(=O)Nc3c(F)cccc3Cl)CCCC2)ncnc2ccccc12 27323,c1(NC(C)=O)cccc(C(N2CC(O)(C(C)NC(C3CC34CCCC4)=O)C2)=O)n1 27324,Cc1cc(C)c(C(=O)NC(C)(C)CCCNC(C2CCCC(F)C2)=O)[nH]1 27325,CCCC(C)(C)C(=O)N1CCC(C)(CC(N2CC(N3CCC(C)C3)C2)=O)C1 27326,C1(C(=O)NCc2ccc(F)nc2F)CC12CCN(C(c1cc(O)ccn1)=O)C2 27327,C#Cc1cccc(CNC(=O)C=CC(C)NC(=O)C(C)(C)C(N)=O)c1 27328,C#Cc1cn(C)nc1C(=O)NCc1cc(C(N2CC(O)CC2CC)=O)on1 27329,C(=O)(CCC(=O)c1ccncc1)N1CC(OCCNC(C2CCNC2=O)=O)C1 27330,C1(C(=O)NCCNC(c2c(OCC)oc(C)n2)=O)CC1C1CC(F)(F)C1 27331,c1(SCCC(=O)NC2CC(C)(NC(C(CCN(C)C)O)=O)C2)cc(F)ccc1F 27332,C(CC#C)(CC(=O)NC1(c2cn(-c3ccc(F)cc3)nn2)CCOCC1)NC 27333,C(=O)(CC(O)CC(C)C)N(C(C(=O)NC(C#C)C)C1CC1)C 27334,Cc1ccccc1OCCCC(=O)NC(C)Cc1nccs1 27335,Cc1cc(C)c(C(=O)NC2(CNC(c3cnc(C(F)(F)F)nc3)=O)CCOC2)o1 27336,c1(OC)ncccc1-c1cnccc1C(=O)NC1CCN(S(=O)(=O)CC2CC2)CC1 27337,c1(C(=O)NCC#CCC(=O)NCCC(COC)O)ccc2c(c1)CCC2 27338,C1(C(N2CC(COC)(NC(=O)C=C(C)C3CC3)C2)=O)CCCC(O)C1 27339,c1(C(=O)NC2C(NC(C(COC)O)=O)CCCC2)cnc2sccn12 27340,N1(CC#CC)CCN(C(=O)C(c2ccoc2)NC(=O)C(N2CCOC2=O)C)CC1 27341,CC(C)C(C(=O)Nc1cncc(C#N)c1)C(C)NC(C1CC(O)C1)=O 27342,C1(C(=O)NC2CC3CC(NC(C4=CC(C)(C)C4)=O)CC32)COc2ccccc2O1 27343,C(=O)(C(C)CC(N)=O)N1CCC(C(=O)NCc2c(OC)n(C)nc2)(CF)C1 27344,C(=O)(C(C)CONC(C1CC(NC(=O)CC2CNC(=O)O2)C1)=O)OC 27345,N1(C(Cc2ncn(C)c2)=O)CCOC(C(=O)NC2CC3CC4C(C3)C24)CC1 27346,C1(CC(N2CCC(CC=C)C2)=O)CN(C(c2cc(O)n(C)n2)=O)CC1C 27347,Cc1c(C(=O)NCC(C(C)C)NC(=O)C(C)Cc2ccco2)cnn1CCO 27348,CC(C)CCC(F)C(=O)N1CCC2(CC2C(N2CC3(CCOC3=O)C2)=O)C1 27349,c1(C(N(CC(C)(C)CNC(C2(CC)CCCC2)=O)CC)=O)cc(C)cc(O)c1 27350,c1(CC(=O)NCCCC(C)NC(=O)CC2CCN(C)C2)ccc(N)cn1 27351,N1(C(c2cn(CC=C)nc2)=O)CC(NC(c2onc(CC)c2C)=O)CC1CC 27352,C=CC(C)C(C)C(=O)NCCCN(C)C(c1cncc(C#N)c1)=O 27353,C1(C)(CC)COCCC1NC(c1c[nH]nc1CNC(=O)C(O)CC1CCCC1)=O 27354,CC1(NC(=O)Cn2cnnn2)CC(C(=O)NCC2(c3cnoc3)CC2)C1 27355,Cc1cccc2nc(NC(=O)COc3cccc(Br)n3)[nH]c12 27356,c1(CNC2CCCC(C(=O)Nc3cnoc3)C2)cnc(Cl)nc1Cl 27357,c1(OC)ccc2ccccc2c1CNC12CC(NC(C3CC3C)=O)(C1)C2 27358,C1(C)(CNC(c2ccc(C#C)cn2)=O)CC(F)(F)CN1C(C1COC(=O)N1C)=O 27359,c1(OC)ncccc1C1CCN(C(=O)NC2CCCC2NS(=O)(=O)C2CC2)C1 27360,C1(N(C)C(c2ccc(C(F)F)nc2)=O)CCN(C(C2(C3CC3)CCCO2)=O)CC1 27361,S(=O)(=O)(c1cc(F)c(F)cc1F)N1CCC(CC(N2CCCC(F)C2)=O)C1 27362,N1(C(CCC=C)=O)CCC(C(=O)NC2CCC(C3CC3)C2)C(C)(C)C1 27363,C(C)(C)(CN=c1nc(C)c(Br)c[nH]1)NC(c1c(CCC)[nH]cc1)=O 27364,N#Cc1ccc(S(N)(=O)=O)c(N2CC3CC2C2OCCOC32)c1 27365,C1(O)(CNC(CC2(COC)CC2)=O)CCCN(C(C2(N(C)C)CCC2)=O)C1 27366,n1(C(C(=O)NCC2(C(=O)NC(COC(C)C)(C)C)CC2)C)cnc(C#N)n1 27367,C(C1CCCCCC1)=CC(N1C(CNC(c2c(C)noc2C(F)F)=O)CCC1)=O 27368,C1(O)(CCNC(CCCN(C)C)=O)CCCN(C(=O)CC2CCC(C)(C)CO2)C1 27369,Cn1nc(CC(=O)NCCC2(O)CCN(C(=O)COC3CCCC3)C2)cc1Cl 27370,N1(C(C2(COC)CN(C(C3CC(F)(CF)C3)=O)C2)=O)CCSC(C)(C)C1 27371,CC1CN(C(c2ccc(C#N)cc2)C(=O)NCc2cccs2)C2COCC2O1 27372,c1(C(C(=O)NCC2(CCNC(CCSC(C)C)=O)CC2)O)cccc(F)c1 27373,CC1(C)COC(C(=O)NC2CCC(CC(N3CCOCC3CO)=O)C2)C1 27374,C1(NC(C(C)CC2CCCCC2)=O)CCN(CCCN(C)C)CC1C 27375,c1(C(=O)NCC(CO)NC(c2cc(Cl)cnc2O)=O)ccc2c(c1O)CCC2 27376,C(CC(C)C(=O)NCCN(C(c1ncoc1Br)=O)C(C)C)=CCC 27377,CC(C)C(CC(=O)Nc1cnn(C)c1C#N)NC(C1C2CCC(C2)C1C)=O 27378,N1(C(C2CC(SC)C2)=O)CCN(C(c2ccnn2C2CCOCC2)=O)CC1 27379,N1(C(CC2CCC(=O)N2)=O)CC2(CCCN(C(C3CN(C4CCC4)C3)=O)C2)C1 27380,N1(C(COC2(C)CCC2)=O)CCOC(C(C)(C)NC(c2ccc(C(N)=O)[nH]2)=O)C1 27381,C1(C)(C(N(C2CN(C(=O)Cn3cc(C(F)(F)F)nn3)C2)C)=O)CCC2CC2C1 27382,C1(NC(C2CCC(N(C)C)C2)=O)CCN(C(=O)C(F)(F)C(F)(F)F)CC12CCC2 27383,c1(CC(=O)NC2CC(F)(CNC(c3cn[nH]c3)=O)C2)cccc2ccccc12 27384,Cn1nc(C(=O)NC(Cc2ccccc2)C(C)(C)C)c2c1CNCC2 27385,C(=O)(C1CCCn2cnnc21)NC1C2(CC(NC(CCN(CC)CC)=O)C2)C1 27386,C(=O)(C(O)C(C)(C)CC)NCCCOCCC(NOCCC(=C)C)=O 27387,C(N=c1cc(CNCCCC2C=CCC2)nc[nH]1)c1cccc(N(C)C)n1 27388,CC(C(=O)NC1COCCN(C(C2CN3CCN2CC3)=O)C1)S(C)(=O)=O 27389,C(CC(=O)NC(c1ccccc1C)C)(C(F)(F)F)NC(CC(C=C)C)=O 27390,CC1(C(=O)NCC2(NC(=O)CCNC(=O)CC3CCCCC3)CC2)CNC(=O)C1 27391,C1(CC=C)(C(=O)NCC(COC)NC(C2CCCN2CC)=O)CCCCC1 27392,c1(C(N2C(C(C)NC(CC(CC)SC)=O)CCC2)=O)ccc(OC)c2ccsc12 27393,c1(C(N2CC(COC)(NC(C3CCCC(C)C3)=O)C2)=O)ccc(C)cc1F 27394,C1(CC(=O)NCC(CC)NC(Cn2ncc(CC)c2)=O)CCC(F)(F)CC1 27395,N1(C(CC2CC(CC)C2)=O)CC2CC1CCC2NCc1ccccc1 27396,c1(OC)ccc(O)cc1C(=O)NCC(C)CNC(=O)CC(C)F 27397,c1(NCC(C2CCCC2)NC(c2ccn(C)n2)=O)ncc2c(ncn2C)n1 27398,c1(N2CCN(C)C(CNC(c3cccc(C(F)F)n3)=O)C2)ncc(C#N)cc1F 27399,c1(SC)ccsc1C(=O)N(CC(=O)N(C1CCSC1)C)CC1CC1 27400,c1(C(=O)NCCN(C(c2cc(C(F)F)ccn2)=O)CC)ccc(Cl)cc1 27401,c1(C(N2CC(CC(=O)Nc3c(Cl)n[nH]c3C3CC3)OCC2)=O)cnn2ccccc12 27402,C1(CNC(C(C)NC(C2CCC2)=O)=O)COCCN1C(=O)CCN1CCCC1=O 27403,C(=O)(C#CC1CCCC1)N1CCN(C)C(C(N2CCC(F)(CF)C2)=O)C1 27404,C1(c2cccc(C)c2)CCCN(C(=NCCCC2CC2)NCCF)C1 27405,N1(C(c2[nH]cc(CC(C)C)c2)=O)CC2CCCC2(CNC(=O)CCCC#N)C1 27406,Cc1[nH]c(C)c(C(=O)N(C)CC2CN(C(c3cc(Cl)ccn3)=O)CCO2)c1C 27407,c1(OC)ccc(C(C)C(=O)NC2CC(C)(NC(C3CCCC3(C)C)=O)C2)cc1F 27408,C1(NC(C(CC)SC)=O)CC1C1CCCN(C(=O)C(=O)C(F)(F)F)C1 27409,C(=O)(C(C)CCCC(C)=O)NCCn1cc(C(=O)NCC(C(F)(F)F)OC)nn1 27410,N1(C(CNC(CNC(c2ccc(C)cc2)=O)=O)=O)CCC2C(C(N)=O)C2C1 27411,Cc1cc(C(N2CCCC2CNC(c2cc(=O)cc(Cl)[nH]2)=O)=O)cc(F)c1C 27412,c1(C(=O)NCCCN(C(c2nc(Cl)cs2)=O)CC)ccnc(C(C)(F)F)c1 27413,CC1(CF)CN(C(C2(C3CCCN3C(c3cnn[nH]3)=O)CC2)=O)C1 27414,C(CCC(C(=O)NCCC1CC1C)NC(c1cn(C)cn1)=O)OC 27415,N1(C(C(C(=O)NC)(C)C)=O)CC2CCN(C(C3CC(N(C)C)C3)=O)C(C2)C1 27416,c1(C(C(=O)N(CC(C)NC(C(CC#C)C2CC2)=O)C)(C)C)ccc(F)c(Cl)c1 27417,CCCCCCC(C)(CC)C(=O)NCC(CCCC)NC(c1ccc(O)nn1)=O 27418,S(=O)(=O)(c1ccc(N2CCn3ncc(Cl)c3C2)nc1)NC1C(C)C1C 27419,Cc1ccc(C(N2CCSCC2C(N2CCC(OCC(C)C)C2)=O)=O)nc1O 27420,C(=O)(CCCS(C)(=O)=O)N(C)CC1(CNC(=O)CCCC2CCCC(=O)N2)CC1 27421,C1(NC(CNC(C(CC)C)=O)=O)CCN(C(=O)C(C)COC(C)=O)C1(C)C 27422,c1(C(N2CCOCC(C(=O)NCCC(=O)N(C)C3CC3)C2)=O)cccc2ccoc12 27423,C1(CC(=O)N(CC(O)CNC(=O)C=Cc2cccs2)C)CCC(F)(F)CC1 27424,c1(NC(C(=O)NC(c2c(C)cccc2C)C)=O)ccc2c(c1)CCC2 27425,c1(C(N2CC(N3CCN(C(c4cnc(C)s4)=O)CC3)C2)=O)ncc(F)cc1C 27426,C1(NC(CN(C(C)C)C)=O)(CNC(c2ccn(C3CCCCC3)n2)=O)CCOC1 27427,CCCCC(CC)C(=O)NCC1CC(C(=O)NC2CCOC2C(C)C)C1 27428,c1(-c2cncc(C(=O)Nc3nccc(OC)n3)n2)ccc(Br)cc1[N+](=O)[O-] 27429,CC1(C)OCCC1C(=O)NCCn1ccc(C(N2CCC3CC23)=O)c1 27430,C1(NC(C=CC)=O)CC=C(C(=O)NCc2cnc(CC)[nH]2)C1 27431,C(=O)(CC(C)(C)C(=O)N(CCCN(C(=O)C(C)CN(C)C)CCO)C)OC 27432,c1(OC)cc(Br)cc(I)c1NC(N1CCC(C(c2ccccc2)CO)CC1)=O 27433,C(CCCC)(CN=c1[nH]c(Cl)ncc1[N+](=O)[O-])NC(C(CCC)OCC)=O 27434,c1(C(c2n(CCCC)nnn2)NC2CC(OC(C)C)C2)cccc(Br)c1 27435,C1(NC(C(C)=NOCC#N)=O)CC(C(=O)NCc2cn(C(C)C)nn2)C12CCC2 27436,c1(C(=O)NC(CCNC(CN(C(C)C)C)=O)C)ccc2c(=O)ccoc2c1 27437,C(=O)(C(C)CC(C)C)N1CCC(C)(CC(=O)NCCNC(=O)OCC)C1 27438,Cc1c(NC(c2oc(CNC(=O)CC3CCC(C)C3)nc2C)=O)cnn1C(C)C 27439,c1(C(C(F)F)NC(c2cn(C(COC)C)nn2)=O)ccc(F)cc1F 27440,C(=O)(CN=c1cc[nH]cc1)NCC(CNC(=O)CCC(=O)c1ccccn1)F 27441,C1(C(=O)OC)(CCNC(C)=O)CCCN1C(c1ncn(C(C)C)n1)=O 27442,N1(C(c2c(-c3c(=O)cc(OC)n(SC)n3)cccc2)=O)CCn2cncc2C1 27443,c1(N2CC(O)(C(C)NC(=O)CCc3ccncn3)C2)nc2c(F)cccc2o1 27444,C1(NC(c2c(CCC)nco2)=O)CN(C(C2CC(F)(F)C2(C)C)=O)CC1N=[N+]=[N-] 27445,Cc1cc(Cl)c(C(N2CCN(C(=O)CS(C)(=O)=O)CC2C)=O)c(Cl)c1 27446,C1(CC(=O)NCC(C(C)C)OC)CCN(C(=O)CC2CCCC2)CC1 27447,c1(OCC(N2CC(CCN=c3[nH]nco3)(CC)C2)=O)ccc(C)cc1Br 27448,C1(CNC(c2cn(C)nc2)=O)CCCCCN1C(C1CC1c1ccsc1)=O 27449,c1(CNC(C=CCC2(NC(c3n(C)ncn3)=O)CCC2)=O)cc(=O)cc[nH]1 27450,CC1(C)CN(C(C2(Br)C3CNCC23)=O)CCC1O 27451,c1(C(N2CC3C(NC(C4C(CCC)C4)=O)(CC3)C2)=O)cc(S(C)(=O)=O)co1 27452,N1(CC(CCC)(C)C)CCC(O)C(C(=O)NCc2cccc(OC)n2)C1 27453,CCC(C)(CC)C(=O)NCCNC(C1CN(C(C23CCC(C2)OC3C)=O)C1)=O 27454,c1(C(=O)NC(CCOC)CNC(=O)CSCc2ccc(Cl)s2)cc(=O)n(C)o1 27455,CC(C)C(CNC(=O)COCc1ccccc1)NC(=O)CCc1cc(Cl)no1 27456,c1(OC)cc(C(N2CCC(CNC(c3ccc(CF)cc3)=O)C2)=O)cc(F)n1 27457,C(=O)(C1=C(Cl)CCCC1)NC(C(=O)N(CC)CC1CCOC1)CO 27458,C1(C(=O)NCCC2CCCN2C)(COC)C=CCN1C(=O)CC1COCCOC1 27459,CCC(CC(=O)NC1CCC(NC(c2cc(F)cc(Cl)c2)=O)CC1)C(C)(C)C 27460,N(C1COc2cc(Br)cnc21)C(CC1CCN(C(=O)OC(C)(C)C)C1)=O 27461,CCCC(C(=O)NC(C(=O)NOCCN1CCCC1=O)C1(O)CCC1)C(C)C 27462,Nc1c(C(=O)NC2CC(NC(C3(F)CCC3)=O)C2)cc(Cl)cc1F 27463,c1(C(C(F)(F)F)NC(C2CCSCC2)=O)cccc(Br)c1 27464,C#Cc1cc(C(=O)N(C)CCNC(=O)Cc2ncn(C)c2C)cc(C(F)(F)F)c1 27465,C12(CNC(CC(=O)OC)(C)C)CCC(CF)(C1)OC2 27466,N1(C(c2cc(C(C)C)nn2C)=O)CCN(C(=O)CCOCC2CC2)CC1C(C)C 27467,c1(NCCCC(C)O)[nH]c(=NC(CC2CC2)c2ccccc2Cl)nc2sccc12 27468,C1(N(C(c2c(OC)csc2)=O)C)CCCC2CN(C(C3CCN(C)C3=O)=O)CC12 27469,C1(C(=O)NCc2cc(C3CC3)on2)(COC)CN(C(=O)CCc2cn[nH]c2)C1 27470,c1(C(=O)NCC(CNC(=O)CC2(O)CCOC2)O)ccc2ccccc2n1 27471,C1(CNC(CC(C)OC)=O)CC2(CCC2)CN1C(C1CN(CC(F)(F)F)C1)=O 27472,C1(C(=O)NCCOCCN(C(C2C(C)C2C)=O)C)C(F)(F)C12CCC2 27473,c1(C(=O)NCCC2N(C(CC(C)C(F)F)=O)CCCC2)c([N+](=O)[O-])cnn1C 27474,CC1CCC(C)(C(=O)NCCSCC(=O)NCc2nnc(O)n2C)C1 27475,C1(C(=O)NC2COCCN(C(=O)Cc3ccoc3)C2)CC2(C1)CC(F)(F)C2 27476,CC1(C)CN(C(c2ncccn2)=O)CCN1Cc1cc(OC(F)(F)F)cc(Br)c1 27477,c1(C(=O)NC)ccc(C(=O)NC2CN(C(C3COCCO3)=O)CCC2F)cc1F 27478,C1(C(=O)NOCc2cnc(Cl)s2)CC2(CC2)CN1C(C1CCC(NC(C)=O)O1)=O 27479,C1(NC(=O)C(CO)c2ccccc2)CCCCN(C(C2(CF)CCOCC2)=O)C1 27480,CCC(CC(=O)NC(C)CC1CCN(C(=O)C(C)(C)OC(C)C)CC1)C(F)F 27481,C#CC(C)(C)C(=O)NCCCC1CN(C(c2ccc(CC(N)=O)cc2)=O)CCO1 27482,c1(C(N2CC(CCC(=O)N3CC(OCCF)C3)OCC2)=O)cccc2[nH]ccc12 27483,c1(OC)cc(NC(C2(CNC(C3(C)C=CCCC3)=O)CC(OC)C2)=O)cc(F)c1 27484,c1(C(=O)NC(CNC(C(C2CC2)SC)=O)CO)cc(C(F)(F)F)cc(Cl)c1 27485,c1(C(N2CC(O)(C(C)NC(CC(C)C(F)F)=O)C2)=O)cnc2c(c1)NC(=O)CO2 27486,c1(C2C(NC(=O)NC3CC(OCCCCC)C3)C2)c[nH]c2cc(F)ccc12 27487,Cc1cc(C(=O)NC2CCC(C(=O)NCC34CCC(C3)C4)C2)c(C)o1 27488,Cc1nc2c(o1)CCN(C(C1CCCN1C(C1(C#N)CCCOC1)=O)=O)C2 27489,C1(C(N2CCCC(C)(CC)C2)=O)CCCCCCN1C(c1cncc(OC)n1)=O 27490,C(=O)(CCCC(F)(F)F)NCC(CC)(C)NC(C1(C)CCC(O)CC1)=O 27491,CC(CC(=O)NCCN(CCCN(C)C)C(=O)CC1CCC2CC12)C(F)(F)F 27492,C1(CNC(C(Cc2c(C)nc[nH]2)O)=O)CCCC2(CN(C(c3csnn3)=O)C2)O1 27493,C1(COC)CN(C(=O)CC2(C(F)(F)F)CCC2)CCN1C(=O)CC1OCCO1 27494,c1(NC(Cc2cccc(C)n2)=O)cnc(Cl)cc1C(=O)N(CCCCCO)C(C)C 27495,CC1CC(CNC(=O)C(C)(CO)NC(=O)CCC2CCCO2)=NO1 27496,C1(CCC(=O)NC23CC(NC(C4CC4(F)Cl)=O)(C2)C3)CCCCC1 27497,c1(C(N2CCC(NC(c3cccc(OC)c3)=O)(CO)C2)=O)scc2c1OCCO2 27498,C1(NC(Cn2c(C)ccc2C)=O)CC(C(N2CC(CC(C)C)C2)=O)C12CCC2 27499,N1(C(C(C2CC2)SC)=O)CCN(C(=O)C(C(C)(C)C)c2cccc(C)c2)CC1C 27500,N1(C(C2C(CCC)CN(C(=O)C(C)C(O)C(C)C)C2)=O)CCc2oc(C)nc2C1 27501,C12(NC(=O)CC=C(Cl)Cl)CCC(CC1)N(C(=O)CCCOc1cccc(F)c1)C2 27502,N1(C(CSCC)=O)CCCC2CN(C(c3nccc(C)c3F)=O)CC12 27503,C(=O)(CCCCN=[N+]=[N-])N1CCCC(C(N(C(C)C)Cc2nn[nH]n2)=O)C1 27504,C(=O)(C(O)CC(=O)OC(C)(C)CN1CCCC1=O)N1CC(NC(C(CCC)C)=O)C1 27505,N1(C(C2C(C)CCCC2)=O)CCCCC(CNC(c2cccc(F)c2N)=O)C1 27506,Cc1cccc(F)c1CC(=O)NC1CC2(C1)CC(NC(=O)C(C)c1ccsn1)C2 27507,Cc1nc(C(=O)NCC(C)(O)CNC(=O)Cc2nc(=N)[nH][nH]2)c(C)n1C1CC1 27508,CC(CC(C)(C)C)C(=O)N1CC2CCCC2(NC(C2CCC(N(C)C)CC2)=O)C1 27509,N1(C(C2(COC)CCCC2)=O)CC(NC(c2cscc2OC)=O)CC(O)C1 27510,C(=O)(C(C)(C)CCCF)N1CCCC(N(C(C(c2ccc(C)cc2)C)=O)C)C1 27511,C(C(C(=O)OC)NC(=O)CC(C)NC(=O)CCN1CCOC1=O)OC 27512,C(CCCCC(=O)NCC(c1ccc(F)cc1)NC(c1ccc(CC)s1)=O)=CC 27513,CC(C)CC(C(=O)NC1(C(O)CO)CC1)NC(c1nnc(O)nc1O)=O 27514,Cc1nn2cccnc2c1C(=O)NCC12CC1CN(C(C1CCS(=O)CC1)=O)C2 27515,c1(C(C)C)c(NC(=O)OC(C)(C)C)cccc1Br.C12CC1C(=O)NC2 27516,C(=O)(CCCCC(C)CC)NCCCC(CCC)NC(c1c2c(nn1C)CCC2)=O 27517,C1(NC(C(COC)O)=O)CCC(C)(C)CC1CNC(C1(OC)CCSCC1)=O 27518,Cc1cc(S(N)(=O)=O)cnc1Nc1cc(Br)cc([N+](=O)[O-])c1 27519,c1(C(N2CCC(NC(C(C(CC)O)(F)F)=O)C(O)C2)=O)cc(S(N)(=O)=O)oc1C 27520,C1(NC(CC2(CSC)CC2)=O)COCCN1CC(F)F.C12C=CC(C1)CNC2=O 27521,Cc1cnc(Cl)cc1NC(C1CCCN(C(c2cccnc2C)=O)C1)=O 27522,c1(OC)ccc(F)c(-c2cncc(NC(C3(O)CCCCC3)=O)c2)c1F 27523,N1(C(C2C(C#C)C2)=O)CCN(C(=O)CSCc2ccccn2)CC(C)(C)C1 27524,c1(OC(C)(C)C(=O)NC2CC(CNC(=O)C3=NOCC3)C2)cccc(N)c1 27525,c1(C(=O)NC2CC(NC(=O)Cc3ccns3)C(O)C2)cccc2nc[nH]c12 27526,c1(C(N(C)CC2CCCN(C(C(C3CCC3)OCC)=O)C2)=O)ncnc(O)c1F 27527,N1(C(c2c(C)nc(C(C)C)o2)=O)CC2CC1CN2C(=O)C(c1cccc(O)c1)C 27528,c1(N(C)CC)nc(NCC2(C(F)F)CC(F)(F)C2)nc2ccsc12 27529,c1(CN(c2nc(OC)ncc2F)C(CC)(C)C)cccc2ncccc12 27530,C(=O)(CN=c1cc[nH]cc1)N(C)CCN(C(=O)CC1CCCCO1)C 27531,c1(OC)ccc(C(=O)N(CC(C)N(C(=O)Cc2ccoc2C)C)C)nc1 27532,C1(C(=O)NCC(C)S(C)(=O)=O)C(C)OCCN1C(=O)CC1CCOC1(C)C 27533,Cc1nc(NCC2CN(C(C3C=CCC3)=O)CCC2C)ncc1Br 27534,N1(C(COCCCOC)=O)CCCC(NC(c2cc(CN=[N+]=[N-])on2)=O)C1C 27535,C(=O)(C(F)C(C)CNC(=O)Cc1cc[nH]c1)Nc1cn(CCOC)nc1 27536,CC1CN(C(c2ccc(-c3ccncc3)s2)=O)CC(C)C1NC(c1cc[nH]c1)=O 27537,C1(c2ccc(OC)cc2)NC(=O)N(CCC(C)Sc2ccccc2)C1=O 27538,Cn1c(C(=O)NC2(CNC(=O)CS(N)(=O)=O)CC(F)(F)C2)cc2sccc12 27539,c1(C(N(CC)CC2CCC(C)CC2)=O)c(-c2ccnc(O)c2)cncc1F 27540,C(CC(C)CCO)NC(C1CC(C)(NC(CCCOCC=C)=O)C1)=O 27541,C1(C(N2CC(CC(=O)NC3CC(CO)C3)(OC)C2)=O)CCCCC1O 27542,N1(C(C(CCC2CC2)NC(COCC(=C)C)=O)=O)CCC2CCN(C)CC12 27543,c1(NC(C(=O)OC)(C)CC2CCC2)nc2ccc(OC)cc2cc1C#N 27544,C1(C(=O)Nc2c(C)n(C)nc2)CC(F)CN(C(C2CCCCN2C)=O)C1 27545,c1(C(N(C)CC2(O)CN(C(c3c(C)nc[nH]3)=O)C2)=O)[nH]c(C)c(S(N)(=O)=O)c1C 27546,C1(N(C(C(C)CO)=O)C)CC2CCC(C1)N2C(=O)CC1=NNC(=O)C1 27547,C12(NC(=O)C3=CCCOC3)CCN(C(c3ccnc4c3CCC4)=O)CCC1C2 27548,Cc1c(Br)ccc(F)c1CNC(=O)NCC1=CCCCC1 27549,c1(C(N2CCC(C)(O)C2)=O)cc(-c2ccco2)cc2[nH]ncc12 27550,C1(C(=O)NCC(CN(C)C(C2(F)CCCCC2)=O)(C)C)CC2C=CC1C2 27551,N1(C(C2(O)CCCC(C)(C)C2)=O)CC2CCCC(CNC(=O)CS(N)(=O)=O)C2C1 27552,c1(CNC(C(CC#C)C)=O)nc(CNC(c2ncc(Cl)cc2O)=O)cc(O)n1 27553,C(=O)(C(C(C)CC1CCCC1)N1CCC(F)(C(=O)OC)C1)NCC=C 27554,n1(C(C)C)ccnc1NC(c1ncc(C2CC2)s1)c1nnnn1C(C)(C)C 27555,c1(-c2nc(COC)nn2-c2cc(O)nc3c2cnn3C)ccc(=O)n2c1CCC2 27556,CC(C)C(CCN(C)C(C1CCCC(=O)N1)=O)NC(=O)CC1CCCCCC1 27557,c1(OC(C)CNC(C2(C)CC=CC2)=O)cccc(N)c1 27558,CC(F)(C(=O)NC1CCC(NC(c2cnn(CCO)c2)=O)CC1)C(F)(F)F 27559,C1(C(N(C)CC2N(C(c3cc(C)ncc3)=O)CCC2)=O)CCC2CC(C)CN2C1 27560,N1(C(CC2COCC(C)O2)=O)CCCC(O)(CN(C(=O)C(C)(C)CC2CC2)C)C1 27561,S(=O)(=O)(c1ccc([N+](=O)[O-])cc1OC)N1CC(C(=O)NCCC=C)C(F)(F)CC1 27562,N1(C(C(C)NC(=O)N(C)CCS(C)(=O)=O)=O)CCc2ccsc2C1 27563,N1(C(C=CC(=O)OCC)=O)CCC2(COC(CNC(c3ncccc3F)=O)C2)C1 27564,C1(O)(C(N(CCCN(C(=O)C=CC(N2CCOCC2)=O)C)C)=O)CC(F)(F)C1 27565,N1(C(CSCC(=O)OC)=O)C(C(=O)NCc2conc2C(C)C)CC2CCCC12 27566,c1(C(N)CO)ccc(C(=O)NCC(c2cccs2)=O)cc1 27567,C12(C(=O)OC)CC(NCc3ccccc3)C1C2.C1CO1 27568,N1(C(CN(C)C2CC2)=O)CCN(C(c2ccccc2OCC#N)=O)CC12CC2 27569,c1(C(=O)NCc2cccnc2Br)n[nH]c2cc(C3=CCCCC3)ccc12 27570,C(C(=O)NCC1CCCN1C(c1occ(C)c1C)=O)(C(C)C)N(CC)CC 27571,Cc1cccc(CC(=O)NC2CCC(NC(C3CSCN3C(C)C)=O)C2)c1F 27572,Cc1nocc1C(=O)NC(CNC(=O)C(C)c1ccco1)C1CC1 27573,N1(C(CCSc2n(C)cnn2)=O)CCCC(CCNC(=O)C(=O)NCC2CC2)C1 27574,N1(C(c2ccc(N(C)CC)cc2)=O)C2CCC1C(NC(C1(C)COCCO1)=O)C2 27575,S(=O)(=O)(c1ccc(CCC(=O)O)cc1)N1CCC(C)CC1CN 27576,CCCCC(F)C(=O)N1CCCCC(C(=O)NCCc2ccc(C)c(C)c2)C1 27577,N1(C(C(=O)NCCC2CCCCC2(F)F)=O)CCc2ccc(Cl)c(F)c2C1 27578,N1(C(C=CC=CC)=O)CC2CCCC2C1C(=O)N(CCC(C)C)C 27579,C1(NC(C(n2ncc(C)c2)C)=O)CCC(C)(NC(c2ccc(Cl)nc2N)=O)CC1 27580,C=CCCC(F)(F)C(=O)NC(CC=C)C(=O)NC(c1nccn1C)C 27581,c1(C(N2CC(CNC(c3cc(OC)n[nH]3)=O)C(O)C2)=O)c(C)nn(C)c1F 27582,CC1CCC(CC(=O)Nc2nn(C)cc2Br)CC1C 27583,N1(C(CNC(=O)OC)=O)CC(CNC(=O)CC(C)C(F)F)C(F)(CO)C1 27584,C(=O)(C(O)CC(C)(C)C)NCC1OCC(C(N2CC(C)N(CCO)CC2)=O)C1 27585,C1(CNC(c2ccc(SCC)nc2)=O)CC12CCN(C(C1CCOCC1)=O)CC2 27586,CCC(C)C(O)C(C)C(=O)NC1(C(=O)NOCCc2ccccc2)CCC1 27587,C(C)(C(C(=O)N(C)CC1CCCC1)C(C)C)NC(c1snc(C)c1N)=O 27588,Cn1nccc1C(N1CC(c2ocnc2CNC(c2cnoc2)=O)C1)=O 27589,C1(CC)CC(C(=O)N(C)CCNC(=O)C(F)OC(F)(F)F)CC(=O)N1 27590,NS(=O)(=O)c1csc(C(N2CCC3C(NC(=O)CCCn4cncn4)CC23)=O)c1 27591,c12cc(C)c(o1)C(=O)NC2.CCC(C)C(=O)NCC(CO)N(C)C 27592,c1(C(=O)OCC)cc(C(C(=O)NCc2ccco2)N(C(C)C)CC2CC2)on1 27593,N1(C(C(CCC)OC)=O)CCN(C(c2cnc(O)o2)=O)CC(CO)C1 27594,C1(CNC(C2C(C(C)O)C2)=O)CCC(NC(=O)C(CO)N(C)C)C1 27595,c1(CC(N2CCC(NC(COC(CC)C)=O)C2)=O)ccc(F)cc1 27596,c1(OC)ccc(NC(C2(CCNC(=O)C=CC(F)(F)F)CCC2)=O)c(F)c1 27597,C1(CC)CCN(C(=O)CCS)C1CNC(CC(N)=O)=O.c1(CCN)scnc1C 27598,N1(C(c2cccnc2NCC2CC2)=O)CCN(Cc2ncccc2Cl)CC12CC2 27599,c1(C(N2CC(CCC)C(C(=O)NC3CCSC3)C2)=O)ccc(=O)n(C)n1 27600,c1(SCC(=O)N(C(CCNC(C(C)OCC=C)=O)C)C)cccc(F)c1 27601,c1(C(=O)NCCC2N(C(C3CC=C(C)CC3)=O)CCOC2)cc(C)c(C)cc1C 27602,CCCC(C(=O)N1CCOCC1CN(C)C(C1CS(=O)(=O)C1)=O)N(C)C 27603,CC1CC(C(=O)NC(C2CCCC2)CNC(=O)C(C)CC(N)=O)=NO1 27604,N1(C(COCC)=O)CC(C)CN(C(c2cccc([N+](=O)[O-])c2O)=O)C(C)C1 27605,c1(C(=O)NC2CN(C(CCc3cccc(C)c3)=O)CC2CO)[nH]c(C)c(C)c1C 27606,C(=O)(C1=CCCCO1)NCC(N(C(=O)Cn1ccc(C(F)(F)F)n1)C)C1CC1 27607,Cc1cccc(CNC(=O)CC2CCN2C(=O)CSC(C)(C)C)c1F 27608,CC1CCN(C(c2cncc(O)c2)=O)CC1CNC(C1CCCC1)=O 27609,C(C(C(=O)N(C(C)C(C)(C)C)C)C(C)(C)C)NC(c1n(C=C)ncc1)=O 27610,C(=O)(C1=COCCC1)NCCC1(NC(=O)Cc2ccccc2F)CC(O)C1 27611,CC1CN(C(c2nnn(C)c2N)=O)CCN1C(c1cccc(CN(C)C)c1)=O 27612,C(=O)(C1CCc2c(Cl)cccc21)NCC(C)NC(=O)C1c2c[nH]nc2CCC1C 27613,C#Cc1cc(C(=O)NCC2(O)CC(NC(=O)CC3CCC3(F)F)C2)ccc1C 27614,N1(C(c2cc(C)sn2)=O)CCC(CCNC(C2C(F)(F)C23CC3)=O)C(F)(F)CC1 27615,N1(C(c2nc(CCC)oc2)=O)CC2(CCN2C(C2C(C#N)C2(C)C)=O)C1 27616,c1(C(=O)NC2CCCN(c3cc(C)[nH]n3)C2=O)ccc2[nH]c3c(c2c1)CCCC3 27617,C(=O)(C(F)CCC(C)C)N1CCC(NC(C=CCC=C)=O)CC1C1CC1 27618,c1(C(C(=O)NCC(=C)C)N(C2CC3(CCC3)C2)CCC)nc(C)c(C)s1 27619,N1(C(C(CCC)C#N)=O)CCCC(C)(C)C1C(=O)NCC1CC(C(C)C)C1 27620,C1(C(=O)OC(c2ccccc2OCC)CC)CC(=O)N(C2CCN(C)CC2)C1 27621,N#CCCCC(=O)NC1CCC(CNC(C2(c3ccccc3)CCCC2)=O)C1 27622,Cc1cc(C)n(CCN(C(C2CN(C(=O)OC(C)(C)C)CCO2)=O)C(C)C)n1 27623,c1(C(N(CCNC(C2(CCCC)CCC2)=O)CCOC)=O)ccc2oncc2c1 27624,C12(CNC(c3cc(C)ncc3)=O)CCC(CNC(c3cscc3C)=O)(CC1)CO2 27625,N1(C(C2CC2C2CC2)=O)CC2C3CCC(C2C1)N(C(C12CC(F)(C1)C2)=O)C3 27626,c1(CNC(CCC=CC)=O)nc(CNC(=O)C(C)=C2CCCC2)cc(O)n1 27627,c1(OC)cc(Br)cnc1C(N1CCCC1c1ccn(C)c1)=O 27628,N1(C(c2cc(C)c(C#N)cc2)=O)CCC2CN(C(=O)CCS(N)(=O)=O)CCC2C1 27629,c1(CC)c(NC(C2CCN(CCC)C2)=O)noc1CC.C1CCNC(=O)CO1.CC 27630,C1(C(=O)NC2C(OC)CN(C(C3CC(O)C3)=O)C2)CC2(C1)CC(F)(F)C2 27631,c1(C(=O)NCC2CN(C(C(C)NC(COC)=O)=O)CC2C)cc(N)c(C)cc1C 27632,c1(C(OC)OCC)ccc(C(=O)NCCCNC(C2CC2(C)C)=O)c(O)n1 27633,C12(C(=O)NCC(c3ccsc3)C)CCC(CC1NC(=O)CC1(O)CCCOC1)C2 27634,N(C1CCCn2ccnc21)C(C1CCN(C(c2cc(CC)ncc2)=O)C1)=O 27635,C1(NC(c2cc(C#N)[nH]c2)=O)CC2CCC1(NC(=O)Cn1cc(Cl)cn1)C2 27636,CC(C)CC(CNC(=NCc1ccsc1C(F)(F)F)NCc1cncnc1)OC 27637,CCCC(O)C(=O)N1CC(CNC(=O)C(C)OCCC(C)C)C1 27638,C1(C)(COC)CC(NC(=O)CCC(C)(C)F)CN1C(=O)C=C(Cl)Cl 27639,c1(C(N2CCC(NC(c3c(CC)noc3)=O)C2CC)=O)cc(S(N)(=O)=O)co1 27640,c1(NCCC(C)(C)C2CC2)[nH]c(=NCC2CCCSCC2)nc2scnc12 27641,N1(C(=O)NC(c2c(C)cccc2)C)CCCCC1(C(=O)O)N(C)C 27642,C(=O)(CC(C(F)F)NC(=O)C(C)(C)CCSC)NCC1CCCC(CC)C1 27643,C1(C(N2C3C(CN)C(CC3)CC2)=O)CCC12CCNCC2 27644,Cc1ccc(Cl)cc1C(=O)NC1COCCC1NC(c1cnn(C)c1F)=O 27645,C12(NC(CCCCCN(C)C)=O)CCCC1N(C(C1CCC(=O)C1)=O)CC2 27646,Cc1nn(C)c(C)c1C(=O)NCC(C1(O)CCN(C(=O)C2=NOCC2)C1)C 27647,N12CC(=O)NC(C1)C(=O)NCC(C)(OC)C2=O.C(=O)(CCC(C)C)NC 27648,N1(C(C(C(C)C)SC)=O)Cc2ccnn2CC(NC(=O)Cc2cc(C)cs2)C1 27649,Cc1c(C)c(C)c(C(=O)NC2CCN(Cc3cn(C(C)(C)C)nn3)C2)c(C)c1C 27650,C1(CCNC(CC2(CC)CC2)=O)CC(C(=O)N(CCF)CC)C1 27651,C1(NC(CCSC)=O)CS(=O)(=O)N(C)C12CCN(C(=O)C1=CCCC1C)CC2 27652,CC1CN(C(c2nccc(C(F)F)n2)=O)CCN1C(C1CCCC(F)(F)C1)=O 27653,C1(N(C(=O)CSSC(F)F)CC)CCN(C(C2CC2c2ccccc2)=O)C1 27654,C1(C(=O)NC2C(F)CCN(C(c3c(CC)noc3)=O)C2)C2CCC1(C)C2(C)C 27655,N1(C(C=NOC)=O)CCOC(C(C)NC(c2csc(C(F)F)n2)=O)C1 27656,c1(NS(NCC)(=O)=O)ccc(C(=O)NC2CCC2NC(=O)CNC(N)=O)cc1 27657,c1(C(=O)NCC2(NC(C=CCC)=O)CCC2)cc(O)nc2ccc(F)cc12 27658,c12ccc(cc1)OC(C(=O)O)CNC2=O.C1(OCCO)CCOCC1 27659,c1(C(N(C(=O)CN2CCCC2C2CCOCC2O)C)=O)c(O)cccc1Br 27660,C1(NC(=O)CCc2cccs2)CC2CCC1C(NC(c1ccsn1)=O)C2 27661,C1(SC(c2ccc(OC(C)C)cn2)c2nnnn2CC2CC2)CC2C=CC1CC2 27662,N1(C(N=c2c(C)c(Cc3ccccc3)[nH][nH]2)=O)CCC12CCOC(C)(C)C2 27663,Cc1nn(CC(N2CC(N(C)C(C3CC4(CCC4)CO3)=O)C2)=O)c2ncccc12 27664,N1(C(C(=O)NCCOC)=O)CC(NC(C2CC23CC(F)(F)C3)=O)CC(C)(C)C1 27665,C(C(Cl)C(C)(F)F)NC(CCN(C(c1c(C)n[nH]c1)=O)C(C)C)=O 27666,N1(C(=O)CN2CCC(F)C2)CCC2C(CCN2C(=O)CCc2cnc(O)[nH]2)C1 27667,C1(CNC(Cn2ccc(C)n2)=O)CC(NC(c2cn(C(F)F)cn2)=O)CC1O 27668,C12(NC(c3cc(C)c(F)cc3)=O)CCCC1N(C(c1cc(O)nn1C)=O)CCC2 27669,N1(C(C(C)C2CCC2)=O)CC(N(C(=O)COC2CN(CC3CC3)C2)C)CC1(C)C 27670,CC(C)CC(CCO)CN=c1cc(NCC2CCC(F)(F)C2)nc[nH]1 27671,N1(C(c2cc(C)n(C)n2)C(=O)NCC)CC(OC)CC(OC(C)(C)C)C1 27672,N1(C(C(C)CF)=O)CC(C2CCN(C(=O)C(C3CC3)C3CC3)CC2)C1 27673,C(=O)(CC(C)CCC(=O)NC(C)(C)CCNC(c1nn(C)cc1Cl)=O)OC 27674,c1(C(N(CC(CC)NC(C(CC=CC)C)=O)CC)=O)ccc2nc(C)nn2c1 27675,c1(CC)cc(C(N2CCC(CCNC(C3CCOC3C(F)(F)F)=O)C2)=O)nn1C 27676,c1(C(N2CCC3(NC(=O)C(F)=CC4CC4)C(C2)C3)=O)ccc2nnc(S)n2c1 27677,C(=O)(C#CC1CCOCC1)N1CCC(C=C)(C(=O)N(CCCC(O)CO)C)C1 27678,c1(C(N2C3CN(Cc4cccc(C(N)=O)c4)CC32)=O)cc(O)ccc1I 27679,C1(C(N(CC(C)C)CC)=O)CC(=O)N(C(c2ccc(Cl)s2)=O)C1 27680,c1(N(C(C(CC)(C)C)C)CC(O)COC)ccc(CC(C)C)c([N+](=O)[O-])c1 27681,n1(CC(=O)NC(CCNC(CC(C=C)CC)=O)C)ccc(=O)n(C)c1=O 27682,N1(C(c2cc(OC)n[nH]2)=O)CC(C(=O)NC23CC(F)(C2)C3)C2(CCC2)C1 27683,N1(C(C2(SCC)CC2)=O)CCC(C2CCN(C(C3(C)CCC(C)C3)=O)C2)CC1 27684,Cc1ccc(N(C2COC2)C(c2ccn(Cc3ccccc3)n2)=O)cn1 27685,c1(C(=O)NC23C(CN(C(CC(CCC)(C)C)=O)C2)C3)cnc2[nH]c(O)nc2c1 27686,N1(C(CC)=O)CCOCC(CNC(=O)CC2CCCN2C(C)=O)C1 27687,c1(OC)cc(OC)c(NCC2CCCC(CCN)C2)c(OC)c1 27688,C(CCNC(c1cccc(F)c1)=O)(C(F)(F)F)OC(C)C(=O)NC(C)(C)C 27689,C1(CCC=C)CCCN(C(c2ccc(OC)cc2)C(=O)Nc2cnn(C)c2)C1 27690,C(=O)(C1COc2ccc(F)cc21)N1CC2(CCN(C(C(CC=C)CC)=O)C2)C1 27691,N1(CC(=O)N(C(CNC(C(c2cccnc2)C)=O)C)C)CCC(N(C)C)CC1 27692,C1(CNC(CCC=C)=O)COCCN(C(C2C3CCCOC23)=O)C1 27693,Cc1cnc2n1CCN(C(=O)C(c1ccco1)NC(c1coc(C3CC3)n1)=O)C2 27694,C(=O)(C(CC)C(C)C)NC1(CNC(c2c(CC)cc[nH]2)=O)CCCC1 27695,C1(CC(=O)N(C(CC(C)C)C)C2CC2)CCN(C(C2CCCC(C#N)C2)=O)C1(C)C 27696,c1(OC)ccc(C(=O)NC2(C)CCCN(C(C3(CCN(C)C)CC3)=O)C2)cc1Cl 27697,N1(C(C(F)OC)=O)CCN(C(=O)C2=CCCC2)C(C)C1 27698,N1(C(C2CC3C=CC2C3)=O)CCC2(CCC2)C(NC(C2(C3CCC3)CC2)=O)C1 27699,N1(C(CC2N(C(COC(CC)C)=O)CC(F)C2)=O)CCC2C(O)CC12 27700,c1(C(=O)NCC2CCC(C(N3CC4(CCOC4)C3)=O)CC2)nccc2cc[nH]c12 27701,c1(C(N2C(CCCNC(CC)=O)CCC2)=O)c[nH]c2cccc(Cl)c12 27702,C12(NC(c3ccc(CC)nc3)=O)CCCC(CN(C(=O)C(Cl)=CCl)C1)C2 27703,CC(C)(C)CC(=O)N(CC(N1CCSCC1C1CC1)=O)CCO 27704,C(=O)(C(C)S(C)(=O)=O)N1CC(C(C)NC(=O)C=Cc2cc(C(N)=O)co2)C1 27705,c1(C(=O)NC2CC(N(C(=O)CC3CCCO3)C)C2)cnc2c(c1)CCOC2 27706,C(=O)(C(C)CC(C)(C)C)NCc1ccc(CN(C(c2onc(C)c2C)=O)C)cc1 27707,c1(C(=O)NC2(CNC(c3c(SC)scc3)=O)CCOC2)cncc(F)c1Cl 27708,C1(O)(CN(C)C(c2cnnn2C)=O)CCN(C(=O)CC2CCCN2C)C1 27709,N1(c2ncnc3n[nH]c(C)c32)CCC2CC(CNC(=O)C=C(Cl)Cl)CCC2C1 27710,Cc1cncc(CC(=O)NC2(CC(=O)NC3CCSCC3)CCCCC2)c1 27711,c1(C(N2CC(NC(C#CC(C)C)=O)C(C(F)F)C2)=O)cccc2c1COC2 27712,C1(C(=O)NC2CCCC(CC(=O)NCC3C(C)(C)COC3)C2)CCC2(CCC2)C1 27713,C(=O)(CC1=CCOCC1)N(CCCC(=O)NC1CCNC1=O)C 27714,C(CC)(C(=O)NCCC1(NC(=O)C=Cc2nc[nH]n2)CCC1)OCC 27715,C1(C(=O)NCC2(CCNC(CNC(C(CC)C)=O)=O)CC2)CCC(=O)NC1C 27716,N1(C(C(C)C(F)F)=O)CCCCC(C(=O)NC23CCN(CC2)C3)C1 27717,CC1CN(C(=O)CC2CCC(=O)NC2=O)CCN1C(C1(NC(N)=O)CC1)=O 27718,C(CC(C)C(=O)NC(CCC1CCC1)C(=O)N(CCCOC)C)=CCC 27719,c1(C(=O)NC2CN(C(C(C)c3cncs3)=O)CC23CC3)cnn2cnnc2c1 27720,c1(C(=O)NC(C(C)NC(C2CNC(=O)C2)=O)CO)cnc2nccn2c1 27721,c1(C(=O)NCCn2cc(-c3c(C(=O)OC)ccc(F)c3)nn2)cc(F)c(O)c(Cl)c1 27722,C12(NC(C3Cc4ccc(F)cc4C3)=O)COCCC1CN(C(c1ccsc1)=O)C2 27723,CC1(NC(C2CC3(C2)CC3F)=O)CCN(C(=O)C(c2ccccc2)C2CC2)CC1 27724,c1(C(N2C3C(C(N4CCN(C)CC4)=O)C(C3)C2)=O)ccc2[nH][nH]c(=N)c2c1 27725,c1(OC)ccc(C(=O)NCCC(O)CNC(C2(C)CCOC2)=O)cc1S(C)(=O)=O 27726,C1(NC(c2noc(CC)c2C)=O)CN(C(c2c(C)noc2N)=O)CC1S(C)(=O)=O 27727,C(=O)(C1CSc2ccccc21)N1CCC(C(C)NC(c2ccnnc2Cl)=O)C1 27728,Cc1cc(NC(C2CCCN(C(=O)CCCF)CC2)=O)cc(Cl)c1 27729,c1(C(N2C(C(=O)NCCSCCC=C)CCC2)=O)cccc(=O)o1 27730,N1(C(c2cc(C)c(F)c(C)c2)=O)Cc2[nH][nH]c(=NC(=O)C3CC4CCC3O4)c2C1 27731,N1(C(C(c2cccnc2)NC(C(COC)OC)=O)=O)CC(C2CCCCC2)C1 27732,C1(CNC(C(C(C)C)n2cnnc2)=O)CC2COCC2N1C(=O)CO 27733,c1(CNC(C2CCCN(C(=O)C(C)=O)C2)=O)ccc(OC(C)=O)cc1 27734,Cc1c(C(N2CCC(NC(c3nccn3C)=O)C2)=O)oc2cc(Cl)ccc12 27735,C1(C(=O)NCc2cc(C(=O)NCC(C)C3CC3)no2)(CC)CCCCC1 27736,c1(C(=O)NCC2CC2(F)F)cc2n(n1)CC1(CC1)C2 27737,C1(N(C(COC)=O)C)CCCN(C(C2CCCS2(=O)=O)=O)CC1 27738,c1(C(=O)NC2CN(C(C3(C)CC3(F)Cl)=O)C2)cccc(NC(N)=O)c1 27739,C1(CC(C)NC(c2cccnn2)=O)CCN(C(C2CNC(=O)C2)=O)CC1 27740,C(C)(C)(C=CC(=O)NC(C1CC1C(=O)NCCCn1cnnn1)C)SC 27741,C1(C(=O)NC2CC3CN(C(C=CC(=O)NC4CC4)=O)C2C3)CCn2nncc2C1 27742,C=C(CNC(C1(C)C=CCN1C(=O)C(CCC)OC)=O)C1CCOCC1 27743,C1(C(=O)OCC)(NC(=O)NC2CC2(c2ccc(Br)cc2)C)CCOCC1 27744,N1(C(C(=O)N(C2CCCCN(C(CCOCC)=O)C2)C)C)CCc2ccccc21 27745,c1(C(C2C(Cl)(Cl)C2)NCCOCC2CCCC2)nnnn1CC1CCOCC1 27746,C1(C(N(CC#C)CCOC)=O)(NC(=O)Cc2ccccn2)CC1(C)C 27747,N1(C(c2n(C(C)C)ccc2)=O)CCN(C(C2CC3CCCCC23)=O)C(CO)C1 27748,C1(C(N(CCN2CC=CC2)CC)=O)CSCCN1C(=O)C=CCN1CCC1 27749,c1(C(=O)NCCN(CCC)Cc2scnc2Cl)cn(CCC)nn1 27750,N1(C(C(CCC)(C)CCC)=O)CCC2(CC1)CC(NC(C1CC(C)C1)=O)CCO2 27751,C(=O)(C(CC=C)CC(C)C)NC(CC#C)CC(=O)NC1COCC1SC 27752,CC1(C)CC(CNC(=O)C=Cc2nccs2)N(C(=O)CCc2cnn[nH]2)C1 27753,C1(NC(C2=NOC(C)C2)=O)CC1C1CCCN(C(C23CC(C2)C3)=O)C1 27754,N1(C(CNC(CC)=O)=O)CC(C)CN(C(c2cccc(=O)o2)=O)C(C)C1 27755,N1(C(=O)CCC2CCOC2)CC2CC1CN2C(C1C2(CC2)C12CC2)=O 27756,c1(C(N2CCC(N(C(C(CC=C)C)=O)C)C2)=O)c(C)ccc2ncccc12 27757,C1(C(C(=O)OC(c2cc(CCN(CC)CC)nnc2C)=O)O)CCS(=O)(=O)CC1 27758,c1(C(N2CC3CC(NC(c4c(O)cc(C)nn4)=O)C3C2)=O)ccc(C#N)nc1C 27759,C1(C(N(CCCN(C(=O)CN2CC(C)(C)C2)C)C)=O)CCC(C#N)C1 27760,N1(C(c2c(OC)c(F)ccc2)=O)CCC2CN(C(=O)CCCN(C)C)CC12 27761,c1(OC)ccc(C(=O)Nc2ncoc2-c2cccs2)c([N+](=O)[O-])c1 27762,C1(C2CCN(C(=O)CS(=O)(=O)NCC)CC2)(NC(C(C)SCCCC)=O)CC1 27763,C(=O)(C1=C(CC)OCCC1)NC(C(=O)NCCCCCCCC)CC(F)F 27764,c1(OCC)cc(F)c(F)cc1C(=O)NC1CC(NCc2c(F)ccc(C)c2Cl)C1 27765,N1(C(C(C(=O)OC)OC)=O)CC(F)(F)CC1CCNC(C1CCCN1C(C)C)=O 27766,C#CC1CN(C(=O)CC2C(CC)C2(F)F)CCN1C(c1cc(Cl)cs1)=O 27767,C1(NC(C(C)OCC)=O)CCN(C(c2cc3cccnc3s2)=O)C12CCC2 27768,C(=O)(C(C)(C)C(C)O)Nc1cccc(-c2cn(C(C)C(=O)O)nn2)c1 27769,C(=O)(C(C(C)NC(c1cccn1C)=O)C(C)C)Nc1c(C)noc1 27770,c1(CNC(C2CNCCN2Cc2ccc(Br)c(Cl)n2)=O)ccc(O)c(O)c1O 27771,CN1C(=O)NC2(CCC(C(=O)OCc3ccsc3[N+](=O)[O-])CC2)C1=O 27772,C(=O)(C(CC)CC(F)(F)F)NCc1cccc(CN(C(CCC(=C)C)=O)C)c1 27773,c1(C(CNC(=O)CCOC2CCC2)NC(C2(CCOC)CC2)=O)ccc(C)cc1 27774,c1(CCN2CCN(c3scc(CCOC)n3)CC2)nc(SC)sc1C#N 27775,CC1CC(F)(F)CCN1C(=O)CC1CCC(NC(=O)C(C2CCC2)C2CCC2)C1 27776,c1(NC(c2c(C)cccn2)C2CC2)ncc(S(=O)(=O)N(C)CC2CC2C)cc1Cl 27777,CC1(C)CC(=O)c2cc(C(N3C4CCC3CSC4)=O)c(=O)oc2C1 27778,Cc1nccc(Cl)c1C(N1CC(NC(=O)CC(C)c2ccccc2)C1)=O 27779,C1(C(=O)NCC2CC2Cl)(CNC(=O)CC2CC3CC3C2)CC12CCC2 27780,Cc1[nH]c2ccccc2c1CC(=O)NCC1(O)CCN(C(=O)COC(F)F)CC1 27781,c1(C(=O)OC)c(F)cc(CNCCCc2cncnc2)cc1F 27782,c1(SCCNC(C)=O)nc(-c2ccoc2)nn1C1CCOC1(C)C 27783,C1(CSCC(=O)NC(C)CC2CN(C(C3CC(F)C3)=O)C2)CCCCO1 27784,c1cc(OC)cc(C)n1.c12ccccc1C(=O)N1CC(C1)NC(=O)C21CC1.CC 27785,C1(CNC(CSCC#C)=O)CCC(NC(=O)C(O)COCc2ccccc2)C1 27786,Cc1[nH]nc(CO)c1C(=O)NC1CC(C#N)C1.N1(C(N)=O)CCC(C(C)C=O)C1 27787,c1(CC)nn(C)c(CC(=O)NCCCC(C)NC(=O)C(C)C(F)(F)F)c1Cl 27788,Cc1cc(NC(=O)C(=O)NCC2CCSC(C)C2)cc(C(N)=O)c1 27789,n1(CC=C)c(N2CCCC2c2ccccc2)nnc1CS(=O)(=O)CC1CC1 27790,Cc1c(C(N2CCC(N(C(=O)Cc3cnoc3)C)C2)=O)oc2c(C)cccc12 27791,CON1CCC(C(=O)NC2CCC(C)N(C(=O)CCc3ccc(Cl)s3)C2)CC1 27792,CCCC(C)C(=O)NC1CC(C)(NC(=O)CCc2ccccn2)C1 27793,C1(O)(C(=O)NCC2(O)CN(C(CCc3cnc(C)o3)=O)C2)CCCC(C)CC1 27794,c1(SCC)ccc(C(=O)NC(CO)C(C)NC(=O)CC2CC(SC)C2)cc1 27795,C1(C(N2CCC(NC(CCOC)=O)C2)=O)CCc2nc(C)ncc2C1 27796,C(=O)(C(=O)C(C)(C)C)N1CC(C(=O)NC(CC(C)C)c2ccccc2)C(F)C1 27797,C1(O)(CN(C)C(c2cnns2)=O)CN(C(=O)CCN2CCC2)C1 27798,C1(C(=O)NC2CCC(NC(C(OC)OC)=O)CC2)CC(F)(F)CCC1(C)C 27799,N1(C(C(COCC)C)=O)CC(CC(=O)NCCn2cc(C)cn2)CC1(C)C 27800,c1(C(N(C2CCN(C(C(COC)(C)OC)=O)C2)CCO)=O)cncc(F)c1Cl 27801,c1(C(N2CC(CC)N(C(=O)CCn3ccc(C)n3)CC2)=O)ccnc2ccsc12 27802,c1(C(N2CCCC(Cn3cc(C(C)(C)N(C)C)nn3)C2)=O)cncc(F)c1Cl 27803,c1(CCCC(=O)NC23C(CN(C(CC(=C)C)=O)C2)C3)csc2ccccc12 27804,c1(C(=O)NC(C(C)(C)NC(CC2CC(OCC)C2)=O)C)ccc(Cl)nc1 27805,Cc1cc(Cl)c(-c2cccc(NC(=O)C(C(C)C)N3CCCC3)c2)cc1F 27806,Cc1cc(C(C)(C)C(=O)NCCOCCCNC(=O)C=CC(C)C)cs1 27807,C(=O)(C#CC1CC1)N(CC(C)O)CCNC(C1CCCN1Cc1ccccn1)=O 27808,c1(OC)cnc(C(=O)NCCNC(c2sccc2-n2cccc2)=O)c(OC)n1 27809,c1(-c2cn(CC(CNC(c3ccc(CCC)[nH]3)=O)OC)nn2)c(F)cccc1F 27810,C#CCCC(C(=O)NC12CC(COC)(C1)C2)NC(=O)C=CC(=O)N(C)C 27811,C(CC(=O)NC(c1ncccc1C)C)(C(F)F)NC(C(C)(CC1CCC1)OC)=O 27812,c1(C(=O)NC2CN(C(c3c(OC)nc(C)cc3)=O)CC2F)cc(C)c(Cl)cc1C 27813,O=C1NC(C(=O)NCC23CC2CN(C(=O)CN2CCCCC2=O)C3)CCO1 27814,CC(C)C#CC(=O)N(CC(C)NC(c1cnn(C)c1C1CC1)=O)C 27815,CC1(C)CN(C(c2ccc(-n3cc(Cl)cn3)cc2)C(=O)NC2CCC2)CC1O 27816,C(CN=c1ccnc(NCC2CC23CCC3)[nH]1)(C(F)(F)F)OC(C)(C)C 27817,OC1CCCCC(CNC(c2nnnn2-c2ccccc2)CC2CC2)C1 27818,N1(C(c2cn(CC)nc2)=O)CCCCC1C(C)ONC(C1CS(=O)(=O)C1)=O 27819,C1(C2CCN(C(=O)CSc3ccc4c(c3)NC(=O)C4)CC2)(NC(C)=O)CCC1 27820,N1(C(COCCOCC#C)=O)CCCC1C(=O)NC1(C#C)CC1 27821,CC1CCC(C)(C(N2CC3(CO)CC2(C(=O)N(C2CCOC2)CCO)C3)=O)CC1 27822,c1(C(N(CCCNC(=O)CCc2csnn2)CC)=O)cncc(OC)n1 27823,CC1(C)C(C(=O)NCC(C)(F)CNC(C2COCCO2)=O)CC1(F)F 27824,CC1=NC(C)(CNC(c2coc(C(C)NC(c3cnc(C)o3)=O)n2)=O)CS1 27825,C(=O)(CC(C(F)(F)F)c1ccc(Cl)cc1)N(C)CC1OCCC1(C)C 27826,C(=O)(C(CC(=O)OC)N(C)C)N(C1CCN(C(C(CCOC)C)=O)CC1)CCO 27827,c1(C(=O)NCC(c2ccccc2)N)nnsc1-c1ccccc1 27828,C1(NC(c2c(CC)c[nH]c2)=O)CN(C(=O)Cc2csc(Cl)c2)CCC12CCC2 27829,C1(C(=O)NC2C3CN(C(C(C#C)(C)C)=O)CC2C3)CCC(S(N)(=O)=O)CC1 27830,n1(CC=C)cc(CNC(=O)C(F)CC2CN(C(=O)CSC(C)C)C2)nn1 27831,CCC(C)C(C(=O)NCc1cc(C)ncn1)NC(C1C2CCC(F)C12)=O 27832,c1(SC)ncc(C#N)c(N2CCN(c3ccnc(Br)n3)C3CC23)n1 27833,c1(C(=O)NC(C(=O)OC)C(O)C(C)C)cccc2c1NCC2C(F)(F)F 27834,N1(C(c2n(CC)ncn2)=O)CCCN(C(c2cc(C#N)oc2C)=O)CC1CO 27835,c1(C(N2CCC(N(C)C(C3CCCC3)=O)CC2)=O)cc(O)nc2ccccc12 27836,C(F)(C(=O)NN1CCCC1C(=O)NC(C1CCCOC1)(C)C)=C(C)C 27837,CCC(C)CCCCC(=O)NC(c1cn(-c2cc(OC)ccc2C)nn1)(C)C 27838,S(=O)(=O)(c1ccc(C(C)C)cc1)NC(C(=O)NC1C(OC)C(C)(C)OC1)C 27839,N1(CC)CCC1C(=O)NC1(CC(=O)NC2(c3cc[nH]n3)CC2)CC1 27840,c1(C(=O)NC(C2N(C(C(C)=C3CCCC3)=O)CCC2)C)cn2c(n1)C(C)CCC2 27841,C1(NC(=O)CC2CC3CC3C2)CN(C(=O)Cn2nccn2)C2(CCC2)C1 27842,C=CCC(C)C(=O)N(CC(C)CNC(C1CN(C)CC1c1cccnc1)=O)C 27843,C1(C(=O)NC2CC(C)(NC(c3ccc(CC)o3)=O)C2)CCOC1(C)C 27844,c1(OC)ccc2c(=NC(C)CN(C)C)[nH]c(=NC3CCCN(C)C3C)[nH]c2c1 27845,C(CNC(=O)C(C)N1CCCC1)(CCNC(c1cnc(C)s1)=O)OC 27846,Cc1nc2c([nH]1)CC(C(N1CCC3CN(C(=O)C(=O)NC4CC4)C3C1)=O)CC2 27847,Nc1cc(C(=O)NCC2CC(NC(C3CC34CC(O)C4)=O)C2)cc(F)c1 27848,CCS(=O)(=O)CC(=O)N1CC(C(N2C3CCCC2CC3)=O)CC1(C)C 27849,c1(C(=O)NCCOCCN(C(=O)Cc2ccoc2)C)c(Cl)ccc(F)c1N 27850,C1(C(N2CCC(O)(CNC(Cc3cnc(C)o3)=O)C2)=O)CC(C)(C)CN1C 27851,Cc1ccc(N(C(c2ccc(C(c3cc(Br)ccn3)=O)cc2)=O)CC2CC2)cc1 27852,C1(CNC(c2cn(CC)nc2)=O)C2CN(CC=CCc3cncc(Cl)n3)CC12 27853,CCC(CC(=O)N1C2CCC1CC(CNC(=O)CCCS(N)(=O)=O)C2)C(C)C 27854,N1(C(c2ccc(OC(C)(C)C)cc2)=O)CC2(CC(N3CCCOCC3)CS2)C1 27855,N1(C(C(CC)(C)C)=O)CCC2(CC1)CC2CNC(=O)Cc1ccsc1C 27856,CC(CS(C)=O)C(=O)NCCCCN1CCCN(C(=O)CC(C)(C)F)CC1 27857,c1(C(=O)NCCCCCCN(C(C(C)OCCCC)=O)C)cccc(C)c1N 27858,C1(C)(CNC(c2cnc(C(C)C)[nH]2)=O)CCCN1C(C1CCN(C)C1C)=O 27859,N1(C(c2ccc(CNC(C(CCC=C)(C)C)=O)cn2)=O)CCc2c(O)noc2C1 27860,Cc1ccc(O)cc1C(=O)NC(CNC(=O)CSc1ccccc1O)CO 27861,C(CC(C)(C)C(=O)NCC1(F)CN(C(C2CCC(C)CC2)=O)C1)SC 27862,C(C(=O)NCCc1c[nH]nc1O)(C(C)(C)O)NC(c1c(CC)n(C)cc1)=O 27863,C1(C(N(c2c(C)csc2)C)=O)CC12CC2(F)F 27864,C1(OC)CC(CNC(c2ncc(F)cn2)=O)N(C(c2cnc(C(C)(C)C)o2)=O)C1 27865,c1(C(=O)NC2CCCN(CC3CCOC(C(Cl)Cl)C3)CC2)c(F)ccc(O)c1F 27866,C1(NC(Cc2onc(C(C)C)n2)=O)CC12CCN(C(=O)C(O)c1ccsc1)CC2 27867,N1(C(=O)NCCOC(CC)(C)C)Cc2cccc(C(=O)NCC(=O)OC)c2C1 27868,C(CC(C)C(=O)N(CC(C)NC(=O)C(c1cnn(C)c1)=O)CC)=CCC 27869,Cc1nc(Sc2ccc(F)cc2)oc1C(=O)NCC1C=CCN1C(C1CC1F)=O 27870,S(=O)(=O)(c1ccc(OC)c(SC)c1OC)N(C(c1ccccc1)C)CC 27871,N1(C(c2ccn(COC)n2)=O)CCC(C)C(NC(=O)C(C)(O)C2CC2)C1 27872,C1(N(C(CCOCCC)=O)C)CN(C(=O)Cn2c(C)c(C)sc2=O)CC1(C)C 27873,C1(OC(CCNC(N)=O)=O)CCNC(=O)C1.C1(=O)CC2(CC2)O1 27874,C1(N(C(c2cc(C(N)=O)no2)=O)CC)CCCN(C(C2CC3CC2CC3O)=O)CC1 27875,c1(CC)ccc(S(C)(=O)=O)cc1C(=O)NC1C2CC3CN(C(=O)C4CC4)C1C3C2 27876,c1(OCC(=O)NC(C2CCCN2C(=O)COc2ccon2)C)cc(F)cc(F)c1 27877,C1(OC)(NC2CCC(n3cc(CCC(C)(C)CO)nn3)CC2)CC(C)(C)C1 27878,c1(NC(=O)CN2CC(Oc3cccc(F)c3)C2)ccc2c(c1F)OCCO2 27879,c1(N2CC(CNC(=O)CN3CC(=O)NC3=O)OCC2)ncnc2scc(Br)c12 27880,N1(C(C2CCCCCC2)C(=O)NC(CC)C)CCC2(CCCCC2)CC1 27881,C(=O)(CCCCN1CCCC1)N(C1CN(C(=O)CCc2cncc(O)c2)C1)C 27882,c1(C(N(C2CN(C(c3cccn3C)=O)CC2F)C)=O)ccc2cc(F)ccc2n1 27883,N1(C(C2C(CC)OCC2)=O)CC2(CC(C(=O)NC(COC)C3(C)CC3)C2)C1 27884,C1(CC=C)(C(=O)OC)CCCN1C(=O)CCCC1CC(CC(=O)O)C1 27885,c1(NCC2CCC(NC(c3c(CCC)nco3)=O)C2)ncccc1C#N 27886,C1(C(=O)NCC(CC)NC(CSCCC)=O)CC2(C1)CC1(CCC1)C2 27887,Cc1nnc2n1CC(C(N1CCOC(c3ccc(Cl)cc3)C1)=O)CC2 27888,c1(C(=O)NCCC2(OC)CN(C(C3CCCC3C)=O)C2)c(C)nn(C(C)C)c1C 27889,C1(NC(C2(CC#C)CCCC2)=O)CCN(C(=O)C(C)(F)C(F)(F)F)CC(O)C1 27890,C1(NC(CCc2cnc(C)s2)=O)CCN(CCC2CCOC2)CC1(C)C 27891,c1(C(=O)NC2(c3cccc(F)c3)CCN(C(C(C=C)O)=O)C2)ccc(N)c(Cl)n1 27892,C1(F)(CNC(c2c(CCC)nco2)=O)CCC(NC(=O)C=Cc2cscn2)C1 27893,C1(O)(CNC(C2(OC)CCCCC2)=O)CCCN(C(c2cnc(C3CC3)s2)=O)C1 27894,c1(C(=O)NCCCN(C(c2[nH]nnc2-c2ccsc2)=O)CC)cocc1C 27895,c1(SCC)nccnc1C(N1CC(OC)CC1CCNC(C1CC(C)(C)C1)=O)=O 27896,O=C1CCc2ccc(C(=O)NC34CC(CNCc5cncc(Br)c5)(C3)C4)nc2N1 27897,c1(NC(C2C(NC(C(CC)C)=O)CCCC2)=O)ccnc(CO)c1C 27898,C(C(=O)N1CC(N2CCOC2=O)C1)(C(C)(C)C)NC(Cc1c(C)ccnc1)=O 27899,C1(CC(=O)NC(C)C(C)NC(=O)Cc2ccoc2)C2CC3CC(C2)CC1C3 27900,N1(Cc2c(C#N)c(Br)ccc2)CCC2(CC1)CCN2C(c1cc[n+]([O-])cc1)=O 27901,c1(CCC)[nH]nc(C(=O)NCC2CCN(C(C3CC3C)=O)C2(C)C)c1[N+](=O)[O-] 27902,N1(C(C2=CC(C)(C)C2)=O)CC2CCC(C(=O)NCC(c3ccsc3)O)(C2)C1 27903,C=CCCCC(=O)NCC1CN(C(=O)CCN(C(CC)CC)C)CCO1 27904,N#Cc1cc(CNC(C2CC2NC(c2ccncc2Cl)=O)=O)cc(F)c1 27905,N1(C(C2(C#C)CN(C(c3cn(CC)cn3)=O)C2)=O)CCOC(CC)CC1 27906,O=C(O)CCCn1cc(C2(O)CN(C(c3nn[nH]c3C(F)(F)F)=O)C2)nn1 27907,N1(CCNC(CN(C(Cn2c(C)ncc2)=O)CC2CC2)=O)CCC(F)(F)CC1 27908,C1(N(C(=O)CSc2nc[nH]n2)C)CCCC(NC(=O)Cc2ccc(Cl)cn2)C1 27909,C1(C(=O)NC(CC(C)NC(C(C)S(N)(=O)=O)=O)C)CN(C)CCN(C)C1 27910,N1(C(C2CCC(CCC(=O)OC)O2)=O)CCN(C(c2ccc(C)cc2)=O)C(C)C1 27911,C1(NC=O)CC(CC(N2CC(Cn3cc(CCC4CCCO4)nn3)C2)=O)CCO1 27912,C1(CNC(CC2(OCC)CCCC2)=O)CCN(C(=O)Cn2ncnn2)C12CC2 27913,Cc1ccc(F)c(C(=O)NCC2CC(C(=O)NCC(c3cnn(C)c3)C)=NO2)n1 27914,C1(C(N(CCCN(C)C)C)=O)CCC(n2cc(CCN3CCSCC3)nn2)CC1 27915,N1(CCN(C(=O)OC(C)(C)C)CC2CCCC2)CC(CO)Cc2c(Cl)cccc21 27916,N#Cc1ccc(CCC2CCN(C(=O)ON3CCCC3)CC2)cc1 27917,c1(N(S(C)(=O)=O)CCCNC(=O)C#CC2(C)COC2)nc2ccccc2[nH]c1=O 27918,CC1(C)CCN(C(c2cc(C3CC3)nn2CC(F)F)C(=O)NCC2CCCO2)C1 27919,Cc1ccc(C(F)CC(CC(=O)NC(C)C(C)C)c2ccccc2)cc1C 27920,C1(CCC(=O)N(CCOC)CCNC(=O)CCNC(C)=O)CCCCN1C 27921,C1(NC(Cc2c(C(C)C)con2)=O)C2CC(NC(C3(C)CCSCC3)=O)CC12 27922,Oc1nc(-n2cc(-c3ccccc3Br)nn2)nc2c1COCC2 27923,N1(C(c2nc(COC)oc2)=O)CCN(C(=O)CN2CCC(CC(=O)OC)CC2)CC1 27924,C#CCCCCC(=O)NCC12CC1CN(C(c1ccc(C)cc1)=O)C2 27925,c1(C(C)C)ccc(C(=O)NC2CCCN(C(=O)C#CC3CC3)C2C)c(F)c1 27926,CC(C)(C)C(C#N)C(=O)NCCC(N1CCCCC1CC(N)=O)=O 27927,C1(C)(COC)CC(NC(c2n[nH]c3c2COC3)=O)CN1C(c1cc(Cl)cn1C)=O 27928,C(=O)(C(C(C)(C)O)NC(=O)C(C)n1cccc1)NC(c1ncc(C)cn1)C 27929,C1(C(=O)NC)CC2CCC(C1)N2C(=O)C(F)=C(C)C.N12CCCC1CNCC2=O 27930,c1(C(N2CCC(C(C)(C)NC(C3OCCCO3)=O)C2)=O)cn2c(n1)CCC2 27931,C(=O)(C(C(C)(C)C)NC(=O)C1=NOCC1)NC(c1ncc(C)s1)C 27932,c1(C(N(CC(C)O)CCNC(c2cccc[n+]2[O-])=O)=O)cnc2ncccc2c1 27933,C(=O)(C1CCc2snnc21)N1C2CN(C(CN(S(C)(=O)=O)C)=O)CC1CC2 27934,O=C1CCCC(C(N2CCC(C(F)CNC(C3CC3(F)F)=O)CC2)=O)O1 27935,Cc1ccc(CC(=O)NC(C)CCCNC(C2C=CCC2)=O)c(C)c1 27936,CCCCCCNC(=O)C(Cc1cnc[nH]1)NC(=O)CSc1cn[nH]c1 27937,c1(C(N2CCC(C3CC3NC(=O)C(F)(F)C3CCCC3)C2)=O)ccc2ncnn2n1 27938,N1(C(c2c(OCC)nccc2)=O)C2CCC1CN(C(c1noc(C)n1)=O)C2 27939,Cc1cnc(Cl)c(C(N2CCC(CC(C)NC(c3ccc(F)nc3)=O)CC2)=O)c1 27940,c1(C(=O)NCCN(C(C(=C(C)C2CC2)F)=O)CC(C)O)ccc(N)c([N+](=O)[O-])c1 27941,C(N=c1[nH]c(C)c(C(=O)NC(CCO)C(C)C)s1)c1c(F)ccc(OC)c1 27942,Cc1cc(NC(=O)C(=O)N(C)Cc2ccnc(Cl)c2)cnc1C 27943,c1(C(=O)NC(c2cn(CC3CCCCC3)nn2)CCC)csc(C)c1Br 27944,C1(CC#C)(C(=O)NCC2CN(C(C3CC(CF)C3)=O)C2)CCC1 27945,Cc1ccc(C(=O)NCC2CN(C(c3nncn3C)=O)CC2C)c2ccccc12 27946,c1(C(C)=O)ccc(OCC(N2CCC(C)C2CNC(c2ccon2)=O)=O)cc1 27947,N1(C(CCn2ncn(C)c2=O)=O)CC2CC(NC(c3cnccc3Cl)=O)C2C1 27948,C1(NC(CCC=CC)=O)CC2CC(NC(c3cc(OC)cnc3F)=O)CC2C1 27949,N1(C(C(C2CCCC2)SC)=O)CC(F)(NC(=O)COc2ccncc2)C1 27950,c1(C(N2CC(COC)(CNC(=O)C(C)(Cl)Cl)C2)=O)ccnc(S(N)(=O)=O)c1 27951,C12(CNC(c3c(CC)cccc3)=O)CN(C(=O)CN=S(C)(C)=O)CC1CCO2 27952,CC1CN(C(=O)C(N)=O)CC2(CCN(C(=O)CC34CCCCC3C4(F)F)C2)O1 27953,N1(C(C(C(C)C)C2CCC2)=O)CCC2(C=C(C(=O)NC34CCN(CC3)C4)C2)C1 27954,C1(CN(CCC(CC)C)CCOC)COc2ccccc2O1 27955,c1(NC2(CCC)CCN(C(=O)C(C)(CC)OC)CC2)cccc(CO)c1[N+](=O)[O-] 27956,Cc1ccc(C)n1CC(=O)NCC(C)N(C)C(C1CCCS1(=O)=O)=O 27957,C1(NC(c2ccc(C#C)o2)=O)CCN(C(c2ccc(SC(F)(F)F)s2)=O)CC1C 27958,N1(C(C(CSC2CCC(C)O2)(C)C)=O)CCOC2(C1)CN(C(=O)CS(N)(=O)=O)C2 27959,C1(C(=O)NCCc2cn(CC(=O)O)nn2)COc2ccc(F)cc2C1 27960,Cc1nnc(N2CCC(C(=O)O)C(C(=O)CCc3cc4ncccn4n3)C2)c(C#N)c1C 27961,N12CCC3C1CCN3C(=O)CC2C.c1(C(=O)NCCN(C)C)ccc(=O)oc1 27962,C1(NC(c2nc(CCC)sc2)=O)CC2CCC1N(C(=O)C(CC)NC(N)=O)C2 27963,N1(C(c2nncn2C)C(=O)NC(c2ccccc2)C)CC2CCC(C1)C(=O)N2 27964,c1(CC(=O)NCC(C2CC(F)(F)C2)NC(CCC)=O)c(C(F)(F)F)coc1C 27965,c1(C(N2CC(O)(CN(C(CCc3scc(C)n3)=O)C)C2)=O)ccc(C#N)c(C)c1 27966,C1(NC(CC2(OC)CN(C(=O)CC3CC3C3CC3)C2)=O)CCOC(C)(C)C1 27967,c1(CC(=O)NC(CNC(C(CCC)(C)O)=O)(C)C)ccc(S(C)=O)cc1 27968,C1(NC(C(CC)C)=O)CCCCC12CCN(C(c1cc3n(n1)CCCN3)=O)C2 27969,N1(C(C=C(CC)C)=O)CC2C(CNC(=O)CNC(N3CCOCC3)=O)C2C1 27970,N1(C(C)CCN(C)C)CCC(C(=O)NCc2cc(C3CC3)no2)C1 27971,C1(CCCOC(C)=O)(Cc2cn(CCNC)nn2)CCOCC1 27972,N1(C(c2ccc(CC)cc2C)=O)CC(C)N(C(c2cnc(S)n2C)=O)CC1C 27973,C1(NC(CC(C)n2ccnc2)=O)C2CC3CN(C(=O)Cc4cnsc4)C1C3C2 27974,Cc1oc([N+](=O)[O-])cc1C(=O)NCC1(C(F)F)CCN(C(=O)C#CC2CC2)C1 27975,c1(CCC(=O)NCC(CO)NC(C=C(CC)C)=O)ccc2ccccc2n1 27976,Cc1occc1C(=O)NC1CCC1C(=O)NCCNC(=O)N(C)C 27977,N1(C(c2n(C)ncn2)=O)CC(NC(c2ccc(Br)nc2Br)=O)C(C#N)C1 27978,CC(C)(CCC(=O)NC1CCCC(O)CC1)NC(=O)CCCC1CC1 27979,CC1CCN(C(=O)CCNC(C2CC3CC4C(C3)C24)=O)C(CO)C1 27980,C1(C(=O)NC2CCC(CCNC(C3(C#N)CC3)=O)C2)CCS(=O)(=O)CC1 27981,c1(C(N(CCC(C)NC(C2CCCC2(C)C)=O)C)=O)cnc(N)c(Br)c1 27982,O=C(C(O)C(F)(F)F)N1CCN(CC2CN(C(C3(C(F)F)CCCO3)=O)C2)CC1 27983,N1(C(C(CCOC)NC(=O)C2=NOCC2)=O)CCCC(F)CC1 27984,c1(COC)cc(C(=O)OC(CCOCCOC(C)C(=O)OC)C(C)C)ncc1F 27985,C1(CC#C)(C(=O)NCc2ccc(Cl)cn2)CCN(C(=O)CCSC)C1 27986,c1(C(=O)NC(c2ccc(F)cc2)C)cccc(C(=O)NCC(CNC(C)=O)F)c1 27987,c1(SC)nc2ncnc(NCC3(F)CCN(C(=O)C(C)C4CCCO4)CC3)c2s1 27988,C1(CNC(CCCOCCOC)=O)CC(CC)CCN1C(=O)COC1CCOC1 27989,c1(OC)ccc(OC)c(C=CC(=O)N(C(C)CNC(c2cc(OC)n[nH]2)=O)C)c1 27990,Cc1ccc(C(=O)NC2CCOCC2NC(=O)CCc2ccoc2)cc1N 27991,C1(NC(Cc2cc(OC)no2)=O)CCCCC1(C)NC(c1c[nH]c(=NC)s1)=O 27992,c1(NC(CN2CCC(OC)C2)=O)ccc2c(c1)CN(C1CCC(=O)NC1=O)C2=O 27993,N1(C(C=CC2COC(C)(C)O2)=O)CCN(C(=O)CSC(F)F)CC(C)(F)C1 27994,C1(CC2CN(C(C(=O)NCC(C3CCCS3(=O)=O)(C)C)=O)C2)CC2COCC2C1 27995,CCCS(=O)(=O)C(C)C(=O)N(C(C)CCNC(c1cc2sccc2n1C)=O)C 27996,N(C1CCc2c(Br)cccc21)c1cc(NC(CC(C)(C)OC)C)nc(C(C)C)n1 27997,c12ccc(c(C)c1)[nH]c2=O.C(C(F)(F)C(C)C)NC(C(CC)CO)=O 27998,c1(C(N(C(CNC(CCC(=C)C)=O)C)CC)=O)cc(OC)c(OC(C)C)c(Cl)c1 27999,c1(CCn2c(CNCCC(C)CO)nnn2)ccc(Cl)c(F)c1 28000,N1(C(c2c(CC)sc(=N)[nH]2)=O)CCCOC(CNC(=O)C2=C(Cl)CC2)C1 28001,CN1C(CNC(=NCC2CCC(O)CC2)NC2CCS(=O)(=O)C2)CCS1(=O)=O 28002,c1(N(c2n(C3CCC(C(N)=O)C3)nnn2)C2CCOC2)ccc(F)cc1Cl 28003,N1(C(C(OC)OC)=O)CC(CNC(c2c(F)cncc2Br)=O)C2(CC2)C1 28004,CN1c2ccc(C(=O)NCCCNC(c3coc(Cl)c3)=O)cc2C(C)(C)S1(=O)=O 28005,C1(NC(CC2C(CC)C2)=O)CCN(C(=O)CC2COCC(C)O2)C1C1CC1 28006,N1(C(CSCC(N)=O)=O)CC2(CCC2NC(=O)C=CCF)C1 28007,c1(CNC(c2ncc(C)cn2)COC)ccc(OC)cc1Cl 28008,c1(C(=O)NC(C2CC2c2ccoc2)=O)cc(C)cc(C#N)c1.C1C(C)CN1CC 28009,CN=c1[nH]cc(C(=O)N(C2CCN(C(=O)CCc3ccncn3)C2)C)s1 28010,c1(C(=O)NC(C)CCNC(=O)CCOC2COC2)[nH]c(=N)sc1C(F)(F)F 28011,N1(C(CC2(C=C)CCCCC2)=O)CC2(C1)CN(C(=O)C(C)NC(=O)NC)CCO2 28012,c1(CCNC(C2(CCCC)CC2)=O)ccc(CN(CCCCC(=O)NC)C)cc1 28013,c1(CNC(c2cnc(-c3cc(F)ncc3O)cn2)=O)ccc2nc(O)[nH]c2c1 28014,C(=O)(CC1=CCN(C)CC1)NCC(C#C)OC.O1NC(=O)C2CC2C1C 28015,c1(C(N2CCN(C(CSCCCC)=O)CC2C(C)C)=O)cccc2cncn12 28016,CC1C(NC(=O)CNC(C2CCCC2)=O)CCN1C(C1C(C)C1C)=O 28017,N1(C(c2nc(N(C)C)oc2)=O)CCC2(CCN(C(=O)Cn3cc(CO)nn3)C2)C1 28018,C1(CNC(c2c(CC)n(C3CCCC3)nc2)=O)CC2(CC2)CN1C(C1CC1C)=O 28019,N1(C(c2c(O)ccc(C#N)c2)=O)CCC2(CCCC2NC(C2CC(=O)N2)=O)CC1 28020,c1(CC)cc(NC(=O)C(C)(C)C2CCN(C(=O)C(C)C(F)(F)F)C2)ccc1C 28021,c1(OC)ccc(C)nc1C(N1CC(OC)C(NC(=O)COc2ccccc2)C1)=O 28022,C(=O)(C(C(C)(C)C)n1ccnn1)N(CC(CC)NC(c1csc(=NC)[nH]1)=O)C 28023,Cc1[nH]nc2c1CCC(C(=O)NC1CCCN(S(=O)(=O)c3ccc(Br)cc3)C1)C2 28024,C1(O)(C(C)NC(C(CC)OC)=O)CCN(C(=O)Cc2ccccc2SC)C1 28025,c1(OC)ccccc1C(N1CCN(Cc2cn(CC3C(C)C3(F)F)nn2)CC1)=O 28026,C1(OC)CC(CNC(=O)C(=O)NCCC(N)=O)N(C(=O)Cc2ccon2)C1 28027,c1(C(N(CCOC)CCNC(=O)Cn2cncn2)=O)cc(S(N)(=O)=O)sc1C 28028,N1(Cc2ccc(C#N)s2)CCCC2C1CCN2C(c1ccc2c(c1)CC(=O)N2)=O 28029,C1(OC)CN(C(=O)Cc2nccn2C)CC1NC(C1CCOCC1)=O 28030,CCCCS(=O)(=O)NC(CC(CN(C(=O)C(=Cc1cccnc1)F)C)CC)=O 28031,C(=O)(N1CCCCCO1)c1c(CNC(C2C=CCS2)=O)ocn1 28032,c1(OC)ccc(C(N2CCOC(C)(CNC(=O)C(F)(F)C3CC3)C2)=O)cc1F 28033,S(=O)(=O)(c1[nH]c(=NCCCCCN(C)C)ccc1Br)N1C(C)c2cccnc2CC1 28034,Cc1cn2ccc(C(=O)NCC3CCCC3NC(c3sccc3F)=O)cc2n1 28035,N1(C(C(C)(C)N2CCCC2)=O)CCOCC(C(=O)NCc2conc2Br)C1 28036,Cc1ccc(NC(C2CCCOC2)(c2nnnn2CCC2CC2)C)cc1C 28037,C=CC1CN(C(=O)CC(CC)N(C(=O)CCCCCC)C)CCO1 28038,CCC(C)(C)CCCC(=O)NC(C)Cn1cc(CCc2ccccc2)nn1 28039,Cc1cc(Br)c2cc(C(=O)Nc3cc(Cl)ccc3I)[nH]c2c1 28040,C1(CC)CCCCCN1C(c1cc(OCCCn2cc(CO)nn2)ccc1C)=O 28041,c1(C(=O)NCC(CNC(c2c(N)nc(Cl)cc2)=O)CO)ccc2nonc2c1 28042,CCC(C)C(O)C(C)C(=O)N(C)CC1CCCN1C(C12CCCN(CC1)C2)=O 28043,C1(C(N2CCCC(NC(c3cn(C)nn3)=O)C2)=O)CCC=CCCC1 28044,C1(CCC(=O)NCC(CC)(C)NC(c2cc(Cl)ccn2)=O)NC(=O)NC1=O 28045,CC1CN(C(=O)C2=CCSC2)CC2(CCN(C(c3cc(Cl)ccn3)=O)C2)O1 28046,C(CN=c1nn[nH]n1Cc1ccccc1)N(C1CC2CC2C1)CC 28047,C1(CC(N2C(CN(C(C(C)C#N)=O)C)CCC2)=O)COC(C)(C)CO1 28048,N1(C(CCC(CC)CC)=O)CC(C2CCCCN(C(C3CCSC3)=O)C2)C1 28049,c1(C(N2CCC(NC(C(C(C)C)OC)=O)C(CO)C2)=O)cc2ncccc2[nH]1 28050,C12(NC(COC3(C)CCC3)=O)CC(CNC(c3ccc(=O)oc3)=O)(C1)OC2(C)C 28051,C12(CNC(c3[nH]c(CC)c(Cl)n3)=O)CCC(C1)N(C(C1CCC(OC)CC1)=O)C2 28052,C1(C(=O)NC(C(=O)OC)CN2CCCC2)CCNC2(CC2)C1 28053,N1(C(c2c(CC)noc2C)=O)CCC(CNC(=O)CCc2cnc[nH]2)C(C)C1 28054,C12(C(N(C(CN(C(CNC(CCC)=O)=O)C)C)C)=O)CC1COC2(C)C 28055,C1(C(=O)OCC2(F)CCN(C(=O)OC(C)(C)C)C2)CCCS(=O)(=O)C1 28056,C1(COCC)CCCN(C(C2(C)CCN2C(c2ccnc(F)c2)=O)=O)C1 28057,C(C(CC(=O)NC1CC(CCO)C1)OC)NC(C(C)=C(CC)C)=O 28058,C(C[Si](C)(C)C)NC(CN(CC#C)C(c1cc(Cl)cs1)=O)=O 28059,C(CC(N)=O)(C(=O)NCc1cnc(O)c(F)c1)NC(C1C(C(=O)OCC)C1)=O 28060,c1(C(=O)NC2C(NC(C3(CC#C)CCC3)=O)C2)cc(C(F)(F)F)cnc1O 28061,N1(C(c2cnc(COC)s2)=O)CCC2(NC(=O)CSS(C)(=O)=O)CCCC12 28062,N1(C(CCC(=O)N(C)C)=O)CCC(C2CCN(C(c3ccc(F)cc3Cl)=O)C2)C1 28063,c1(CCC(=O)NC2C(NC(Cc3c(C)scc3)=O)COC2)cccc(C(N)=O)c1 28064,c1(C(=O)OC)cc(F)ncc1C(N(c1n(CC)nc(C)c1)C1CC2CNC1C2)=O 28065,N1(C(C)=O)CCC(NC(C2(OC3(CCCNC(=O)CC(F)F)CC3)CCC2)=O)C1 28066,c1(NC(C2(C)N(C(c3cncc(OC)c3)=O)CC2)=O)ccc2ncc(Br)cc2c1 28067,C1(NC(c2c(O)cc(C)nn2)=O)CCN(C(=O)CSC2CC2)CCC1(F)F 28068,N1(C(Cc2n(C)cnn2)=O)CCC(CNC(C2CC(n3cnnc3)C2)=O)C12CC2 28069,C1(C(N2CCC(C3(C)N=N3)CC2)=O)CN(C(c2ccccc2Cl)=O)CC1(F)F 28070,CCCCCCC(C)(c1nnnn1CCCF)NCC=C1CCSCC1 28071,C=CC(C)(O)CC(=O)NCC1CCCCN(C(c2nc(OC)cc(OC)n2)=O)C1 28072,c1(NCC2CN(C(C3C(OC)CCC3)=O)C(C)C2)nnc(C)c(C)c1C#N 28073,C=C(C)C(C)(C)C(=O)Nc1ccnc(CN(C(=O)CSC)C)c1 28074,N1(C(c2cccc(C)c2F)=O)CCC2(C1)CN(c1ccnc(C3CC3)n1)CCO2 28075,c1(CN=C(NC2CC(SC)C2)NC2CCS(=O)(=O)C2)ccc2c(c1)OCCCO2 28076,N1(C(=O)C(F)(F)F)Cc2cccc(F)c2C1.N12CCC(C3CC13)NC2=O 28077,N1(C(CSc2[nH]c(=N)sc2)=O)CC2CCCC(NC(=O)COCC3CCOC3)C2C1 28078,N1(C(C=C(C)C(F)F)=O)CCC(F)(C(N2CCCC2C2(C)CC2)=O)CC1 28079,C#CCCCC(C(=O)Nc1ccc2c(c1)OCO2)N1CCC1(C)CCO 28080,c1(NC2(c3c(OC)ccc(Br)c3)CC2)ccnc2c(I)cccc12 28081,Cc1c(C(=O)NC2CN(C(c3ccc(N)cc3)=O)C2)cnn1-c1ccc(O)nn1 28082,c1(OC)c(CC(=O)NC(C)CCNC(C2CCC(=O)N2)=O)cccc1C#N 28083,CC1CN(C(c2cnn3c2SCC3)=O)CC(C)N(C(c2cncs2)=O)C1 28084,C(=O)(C(F)C(C)CNC(c1ccc(C)o1)=O)N(C(CC)C(=O)OC)C 28085,N1(C(C2CC2F)=O)CCC2(CC1)CN(C(c1c(F)cccc1Cl)=O)CCC2O 28086,c1(C(=O)NC(C(C(C)C)NC(Cc2c(C)ocn2)=O)C)ccsc1S(C)(=O)=O 28087,N1(c2c(C#N)cnc(C)n2)Cc2ccc(NC(=O)C(c3ccccc3)O)cc2C1 28088,Cc1ccc(N)c(C)c1C(=O)NC1CCC1NC(=O)CC(C)n1cccn1 28089,CCC(CC(=O)N(CC(C)C(=O)NC(C)CC1CC1)C)CC(C)C 28090,C1(NC(C=C2CCN(C(C3(COC)COC3)=O)CC2)=O)CC(=O)N(C)C1=O 28091,C1(CNC(C(CCCC)C)(C)c2nnnn2CC(F)F)Cc2ccccc2CO1 28092,c1(C(=O)NCC2CC(NC(c3cc(F)cc(Cl)c3)=O)C2)n[nH]cc1[N+](=O)[O-] 28093,N1(C(c2c(C)ncc(N)c2)=O)CC(NC(C2(C)CCCCC2)=O)CC(C)(C)C1 28094,CON1CC(C(=O)NCCN(C2CCCCC2)C(=O)C=Cc2ccoc2)CC1=O 28095,C(=O)(C1=CC2C=CC1C2)N1CCCC(C(=O)NC(c2nncs2)C)CC1 28096,C12(CNC(C(C)=CC)=O)CCCCC1CN(C(c1ccc(C(F)(F)F)o1)=O)C2 28097,C(CCN(C)C)(C(=O)NCC(C)NC(Cn1ncc(CC)c1)=O)NC(C)=O 28098,C#Cc1cccc(CNC(C2(CCNC(=O)C(c3cnccn3)C)CCC2)=O)c1 28099,N1(C(c2cnco2)=O)CC2CCN(C(c3ccc(-n4cnnn4)cc3)=O)C(C2)C1 28100,CC1(C)CC1(C#N)C(N1CC2C(NC(=O)Cc3cn[nH]c3)C2C1)=O 28101,c1(C(=O)NCC2C(C)CN(C(c3nnc(C(C)(C)C)s3)=O)C2)cc(C#N)cn1C 28102,c1(C(=O)NC2C(C)(C)CCN(C(C3(C)COC3)=O)C2)cc2nn[nH]c2cc1F 28103,C(=O)(C1=CCCC(C)(C)C1)N(C1CCN(C(C2(S(C)(=O)=O)CCCC2)=O)C1)C 28104,CC(C)(C)C(CNC(C12CCCC1C2)=O)NC(C1CCC(=C2CCC2)CC1)=O 28105,N1(C(c2cnn(C)n2)=O)CCCC(C2CCCCN2C(=O)CNC(=O)C2CC2)C1 28106,c1(C(C)(C)C)ccc(C(=O)NC2CCCC2C(=O)NCc2ccc(O)cn2)cn1 28107,CN(S(=O)(=O)N1CC(O)C(O)C1)CC(c1ccccc1)O 28108,Cc1csc2nc(C(=O)NC(C)CNC(=O)C(=O)N(C)C)cn12 28109,C12(CCNC(=NC)NC3CCC3)CCC(F)(CN(C(=O)OC(C)(C)C)C1)C2 28110,C(=O)(C(O)CCC1CCC1)NCC1(C(=O)NC(C)CN(C)C)CC1 28111,C1(CC=C)(NC(C2C3CCC(F)C23)=O)CCN(C(c2cc(C(C)=O)cs2)=O)C1 28112,N12CCC3(CC3C1)c1cn(nn1)C1(CC1)C2=O.Cn1ccc(C2CC2SC)n1 28113,C(=O)(CS(=O)(=O)CC(F)(F)F)NCCC1(O)CCN(C(C(CC)(C)O)=O)C1 28114,c1(C(N(CC(C)NC(C2CCCO2)=O)C)=O)ccc(N)c(C(F)(F)F)c1 28115,C1(C(N2C(C3(NC(C4CC(SC)C4)=O)CC3)CCCC2)=O)CCCC(=O)N1C 28116,n1(CCC)ccc(C(=O)NC2(c3ccccc3)CC(NC(=O)C=C(Cl)Cl)C2)n1 28117,c1(C(=O)NCCSC(C(=O)NC2CCN(C(C)C)C2)C)ccc(O)nn1 28118,c1(C(=O)NCC2(F)CN(C(Cc3nc(C)sc3)=O)C2)ccc2c(n1)CCC(C)C2 28119,Cn1ncc2ccnc(C(=O)NCC=CCNC(=O)C(O)P(C)(C)=O)c12 28120,c1(NC(C2N(Cc3c(C)c(O)ccc3)CCOC2)=O)cnn2ccc(Cl)nc12 28121,Cc1nc(O)sc1C(=O)NC(C)(CSC)C(=O)N(C)C.C1CCN(C(N)=O)CC1 28122,N1(C(C(=O)N(C)C)=O)CCCC2(CNC(c3sccc3Br)=O)CCCC12 28123,CC(CC(=O)NC1CN(C(c2nc(Cl)c(=O)[nH]c2N)=O)CC(C)(C)C1)C(C)(C)C 28124,C(=O)(C(CCC1CC1)NC(=O)C(C)NC(=O)CC)NC(CC=C)C1CC1 28125,C1(NC(c2cscc2Br)=O)CN(C(c2cncnc2)=O)CC1(F)F 28126,c1(C(=O)NC2(CN(C)C)CC2)ccccc1CC(=O)Nc1cc(OCC)n[nH]1 28127,c1(NC(CC(C)NC(c2c(COC)cco2)=O)C)ncc(Cl)c(C)c1C#N 28128,c1(C(N2CC3(CCN3C(N3CCC(n4cncn4)C3)=O)C2)=O)cc(F)cc(F)c1 28129,N1(C(C2=CC(C)CC2)=O)CCC2(CC1)CCN(C(c1c[nH]nc1C1CC1)=O)CC2 28130,c1(C(N2CC(C)C(NC(c3cscc3S(C)(=O)=O)=O)C2)=O)ccn2ccnc2c1 28131,C(c1csc2ccccc12)=CC(=O)OC1CCCCN(CC)C1=O 28132,c1(CCNC(C2COCCN(c3ncc(C)cn3)C2)=O)cccc2c1OCCO2 28133,CC(C)CCCCCC(=O)NCCC1(NC(=O)Cn2nnc(=O)[nH]2)CCC1 28134,c1(CC(=O)NCC(C)NC(c2c[nH]nc2-c2ccccc2)=O)cc(F)cc(F)c1 28135,c1(CNC(N2CC(c3ccn(C)n3)OCC2)=O)ccc(I)c(Br)c1 28136,C1(OC)CC(NC(=O)CN(CC(C)C)C(=O)Cc2cccnc2)C1(C)C 28137,C1(CC(=O)NC)CN(C(=O)C(O)CC(F)F)CCN1C(c1nc(C)sc1C)=O 28138,N1(C(c2c(C)nc(CNC(C3C(C)(C)C3(F)F)=O)o2)=O)Cc2n[nH]cc2C1CO 28139,C1(C(N2CC(NC(C3C(=C)C3C(=O)OC)=O)C2)=O)CC(c2ccc(C)cc2)=NO1 28140,N1(C(c2cccc(C)c2F)=O)CCC2CN(C(=O)Cc3cnn(C(F)F)c3)C2C1 28141,Cc1c(C(N2CCC(CCNC(C3CC(=O)N(CC4CC4)C3)=O)C2)=O)ncn1C 28142,N1(C(CS(N)(=O)=O)=O)CCOCC(NC(=O)C(O)Cc2ccccc2)C1 28143,Cc1nc(Cl)ccc1CC(=O)NC1CN(C(c2ccc(O)c(N)c2)=O)CC1C 28144,Cc1ccc(CNC(N2CCC(NC(C34CC(CO3)C4)=O)C2)=O)cc1 28145,c1(OC)ccc(C(N2CC(O)CC2C(=O)NCc2ccc(Br)c(Br)c2)=O)cc1I 28146,C1(C(=O)NCCNC(CC2(C)CCCCC2)=O)CCOC(=O)CC1 28147,c12ccc(nc1)N(CCO)C2.Cc1noc(C(C)OC(C)(C)C)n1 28148,C12(CC(N3CCC(n4cnnn4)C3)=O)CCC1CN(C(C1CCCO1)=O)C2 28149,C1(NC(=O)Cn2cccc2)CCCN(C(c2cc(Cl)sc2Cl)=O)CC1 28150,C1(SCC(=O)NC(C(N2CC(NC(C)=O)C2)=O)C2(C)CC2)CCCCO1 28151,c1(CC(N2CCC(NC(C3C(C)C3)=O)C2C2CC2)=O)ccc2oc(O)nc2c1 28152,N1(C(c2c(C)cncc2C)=O)CCC2C(CCCN2C(=O)C(F)CC(C)C)C1 28153,c1(C(=O)Nc2cnc(CCCC)nc2)ccc(Cl)c(O)c1 28154,C1(NC(C2CC(=O)NCC2)=O)C2CC(O)C1N(C(=O)C=CSc1nc[nH]n1)C2 28155,CC1CCCCC1(CNC(=O)Cc1sc(O)nc1O)NC(=O)CC1CC(F)(F)C1 28156,N1(C(c2nc(OCC)sn2)=O)CCC(C2(NC(c3ccnnc3)=O)CC2)CC1 28157,CCCCCS(=O)(=O)CC(=O)N1CCC(NC(c2cc(OC)c(O)c(N)c2)=O)C1 28158,C1(NC(c2c(CCC)nns2)=O)CC(C)N(C(=O)C(C2CC2)SC)C1 28159,N1(C(C2(CNC(=O)C(C)S(N)(=O)=O)CC(=C)C2)=O)CCC(C2(C)CC2)C1 28160,c1(C(N(CC(C)O)CCNC(c2cncc(C=C)c2)=O)=O)cnc2scc(C)n12 28161,S(=O)(=O)(c1c[nH]ccc1=NCc1csnn1)N1C(C(CCC)C)CCC1 28162,N1(C(c2ccc(CC)o2)=O)CCC(CNC(c2cccc(C)c2C)=O)C1(C)C 28163,c1(C(N2CCN(C(Cc3nc(C)sc3)=O)C3C2C3)=O)cnc2cc(Cl)ccn12 28164,c1(CC(N2CC(OC)C(NC(=O)C(C)S(N)(=O)=O)C2)=O)ccc2c(c1)NC(=O)C2 28165,N1(C(C(CC)SC)=O)CCC2(CC1)CCN(C(=O)C=C(C)c1ccco1)CC2C 28166,CC1=C(C(=O)NC23CCN(C(=O)CC(C)(C)C)CC2C3)CCC1 28167,N1(C(c2c(CC)csc2)=O)CCC(CNC(=O)Cn2nc(C)oc2=O)C(C)C1 28168,C(=O)(CC1OCCc2ccsc21)N1CC(NC(CCCCC(C)C)=O)CC1(C)C 28169,c1(C(N(CC(=O)NCC2(C)CCCC2O)C2CCC2)=O)cc2cc[nH]c2cn1 28170,C(=O)(CCCCCN(C(C1CCC1C)=O)C1CC1)N(CC(C)C)CC 28171,C(C)(C)(CC(F)C(=O)NCCc1cccnc1)NC(c1scc(C)c1)=O 28172,c1(C(N2CCCC(NC(C(C)n3cccc3)=O)C2)=O)ccc2c(c1)COC2 28173,C(CC(=O)N1CC(CC(C)(C)C)C1)N(C(=O)CN1CCCC1)CC#C 28174,C(C(C)(C(C)C)NC(=O)C=CC(=O)N(C)C)NC(c1scc(C(=O)OC)c1)=O 28175,C1(NC(c2n(C(C)(C)C)ncc2)=O)CCC(C)(CNC(=O)Cc2cnoc2)C1 28176,c1(C(=O)NC(C)CC(C)NC(c2cc(CC3CC3)on2)=O)ccc(=O)n(CF)n1 28177,CC1CCC(C)(NC(c2cn(C3C4C(=O)OCC34Br)nn2)=O)C1 28178,c1(CN2CC(NC(c3ccc(=O)oc3)=O)C(F)(F)C2)ccc2c(c1)CCO2 28179,C1(COC)(NC(=O)CCCCn2cc(-c3ccc(F)nc3)nn2)CCS(=O)(=O)C1 28180,C1(OCCNC(c2cnsn2)=O)CCN(C(c2ccnn2CC(F)(F)F)=O)C1 28181,CC1CCCCC1C(=O)NC(C)(C)C=CC(=O)NCC(F)Cl 28182,c1(C(N)=O)ccc(CC(N2CCOCC2CNC(=O)CCC2CCCO2)=O)cc1 28183,C1(c2cccc(C)c2)CCCC2(CN(C(c3ccc([N+](=O)[O-])s3)=O)C2)O1 28184,Cc1c(C(=O)NCC2CN(C(=O)C(F)C3CCC3)CCCO2)nn(C)c1N 28185,Cc1cccc2c(C(N3CCC4(NC(=O)C(C)NC(N)=O)CCCC34)=O)coc12 28186,N1(C(C2C(CC)CCO2)=O)CCCC1(C)CNC(C1(c2ncco2)CCC1)=O 28187,N1(C(C(C(C)C)SC)=O)CCN(C(=O)Cn2ccccc2=O)CC12CC2 28188,Cc1cccc(C(=O)NCC(F)CNC(c2cnc(CC(C)C)[nH]2)=O)c1C 28189,c1(C(=O)NC2CCNC2=O)cc2c(s1)CCN(C(c1cc(Cl)ccc1Cl)=O)C2 28190,C(=O)(C(F)(F)CO)NCC1(F)CC(NC(c2c(C)csc2)=O)C1 28191,c1(C(=O)NCC)ccc(N(C)C(C)=O)cc1C.n12cc(nn1)CNC(=O)C2 28192,CC1(C)CC(CNC(=O)CCCNC(N)=O)CN(C(C2(F)CC2)=O)C1 28193,N1(C(C(C)=C2CCC2)=O)CC2CCCCC2(CNC(=O)C(F)=C2CCC2)C1 28194,C#Cc1ccc(C(=O)NC2CCCC2CNC(=O)CCc2ccc(O)cc2)cn1 28195,CP(C)(=O)C(O)C(=O)NCCOCCOCCNC(=O)Cc1cnccn1 28196,C#CC1CN(C(C2CCC2C#N)=O)CCN1C(c1cnc2[nH]nnc2c1)=O 28197,C(=O)(CCCCCCNC(=O)C(C)(CO)NC(C)=O)N(CC(C)N(C(C)=O)C)C 28198,N1(C(C(F)=CC)=O)CC(CN(C(=O)CN2CCCC2)CCC)CCC1=O 28199,c1(OC)ccc(C(=O)NC2CCC2CNC(c2[nH]ncc2C#N)=O)c(C)c1 28200,C#CCC(C)(C(=O)NCC(C)S(N)(=O)=O)NC(c1cccnc1NC)=O 28201,Cc1c(F)ccc(CN2CCC(F)(C(=O)NC(c3cccnc3)C)C2)c1Cl 28202,CCCC(CCC)C(=O)NCCN(C1CCCCC1)C(C1CC1COC)=O 28203,c1(C(=O)NCC(CO)NC(c2cc(SC)oc2)=O)ccc([N+](=O)[O-])s1 28204,n1(CCC(N2CCC(CNC(c3ccc(CCC)[nH]3)=O)C2)=O)ccc(O)nc1=O 28205,CCCC(C(=O)OC)C(=O)N1CCC(C)(C)C1CNC(=O)CCc1cnc(O)[nH]1 28206,C1(Cl)(C(N(C(C)CNC(=O)COC2CCC2)CC)=O)CC1 28207,C(=O)(CCN=c1[nH]ccs1)NCC1CC(OC)CN1C(c1c[nH]nc1C)=O 28208,c1(N2CC(C)(CNC(C(CC)OC)=O)OCC2)ncnc2sc(C(F)(F)F)nc12 28209,C(=O)(C1=NOC(C)(C)C1)N1CC(C(=O)NCC(COC)C(C)C)C(F)C1 28210,N1(C(c2cnn(CC(F)F)n2)=O)CCN(C(c2cscc2Cl)=O)CC1 28211,c1(C(=O)NCC2(C(N)=O)CC2)cc(CCNC(=O)C(F)C2CCCC2)on1 28212,C(=O)(C(C)(C)C(F)F)N1CCCC(CCNC(C2C(C)(C)C2(F)F)=O)C1 28213,N1(C(c2ccc(C)cc2)=O)CCC(C2CC2)C1CNC(c1ncccc1Cl)=O 28214,N1(C(c2c(CC)ncs2)=O)CCCC(C(C)NC(c2c(C)nnn2C)=O)C1 28215,C(CCCCCNC(=O)C(Br)=C(C)C)N(C(c1c(CC)cco1)=O)C 28216,c1(C(=O)NCC#CCNC(=O)C=CC2CCCO2)cc2ccccn2n1 28217,c1(C(=O)NC(C)(CNC(=O)CCS(N)(=O)=O)CO)ccc2c(c1)CCC2(F)F 28218,S(=O)(=O)(c1ccc2c(c1)C(=O)C(=O)N2)Nc1c(C)n(CC)c2c1cc(OCC)cc2 28219,C1(C(=O)NC2CCCC(NC(=O)CSCC(F)(F)F)C2)(CC)CCC(O)CC1 28220,c1(C(=O)NCC2C(NC(C3C(C)C3)=O)CC2)cnn2c(-c3cccs3)ccnc12 28221,C[Si](C)(C)CCCNC(=O)NCCCCN1CCC1 28222,Cc1ccccc1CC(C)C(=O)NCCC1(NC(=O)CCSCC(N)=O)CC1 28223,CS(=O)(=NC(=O)CC1CCCCS1(=O)=O)c1ccccc1 28224,c1(C(N(C)CC2CCCN(C(CCC3CCC(C)O3)=O)C2)=O)c[nH]cc(F)c1=O 28225,C12(NC(CC(CC)C(C)C)=O)CCCC(CN(C(c3cccn3C)=O)C1)C2 28226,N1(C(CCC(C)(C)F)=O)CC2CCC(C1)N2C(C1(C)CSC1)=O 28227,c1(NCC(=O)NC(N(CCCOC)C)=O)cccc(C(N)=O)c1 28228,Cc1nnc2n1CCN(C(=O)NCc1ccc(C3CCC3)nc1)C2 28229,N1(C(C2CC(C(C)C)OCC2)=O)C2CCCC1CN(C(c1cccc(O)n1)=O)C2 28230,C1(NC(c2c(OC)scc2)=O)CC2CC(NC(=O)C(C)(O)C3CCC3)C1C2 28231,c1(C(=O)NCC2C(CNC(Cc3c(C)occ3)=O)C2)c(N(C)C)cccc1Cl 28232,CCC(CCCC(=O)NC1(C(=O)NC2(CO)CC2)CCC1)NC(N)=O 28233,N1(C(C(CNC(CCCNC(C)=O)=O)C(C)C)=O)CC2CC(O)CC1C2 28234,CCC(CC(=O)N1CCC(C(C)O)CC1)NC(=O)C(=CC1CCCC1)C 28235,NS(=O)(=O)CCC(=O)N1CC(Cn2cc(CCC3CCCCO3)nn2)C1 28236,Cc1nc(C(C)C)ccc1CNC(=O)C=CC(C)NC(C1CC1(C)C)=O 28237,N1(C(C2(CCOC)CC2)=O)CCC2C(C1)CN2C(=O)CC1(C(F)(F)F)CC1 28238,C#CC1CN(C(=O)CC(CC)N(C(=O)C(C)CC(C)C)C)CCN1C 28239,N1(C(=O)Cc2ccccc2Cl)CCCC(F)(CN=c2[nH]nc(C3CC3)s2)C1 28240,Cc1ccc(CN2C(C(=O)NCC3CCC(O)CC3)CC3CC23)c(Cl)c1Cl 28241,C1(C(N2CCC(OCCNC(C(COC)(C)C)=O)C2)=O)CCc2nccn2C1 28242,N(C1CC(C)n2ncnc21)C(N1C(C)(Oc2cncc(C)n2)CCC1)=O 28243,C1(CNC(C2CN3CCC2CC3)=O)CCN(C(=O)Cc2c[nH]nc2O)C12CC2 28244,C(=O)(C1Cc2ccc(Cl)cc21)N1C2CCN(C(C(=O)NCC3CC3)=O)CC1CC2 28245,C1(CC(=O)NCC(N2CCN(C(c3ncccc3F)=O)CC2)C)CC2(CCC2)C1 28246,C1(C(C(=O)NCc2ccco2)N(CC(C)C)Cc2ccccc2)CCOC(C)C1 28247,N1(C(CNC(CNC(c2cc(C)sc2N)=O)=O)=O)CC2CCCCC2C1C 28248,C(=O)(C(C)(C)C(F)(F)F)NC1CCC(CNC(CCC(=O)OC)=O)CC1 28249,CCCCCCCC(=O)N1CC(C(=O)NCc2ccc(Cl)cc2Cl)C1 28250,C1(N(C)C)CCCCC1C(=O)NC1CC(C)(NC(=O)CCC2CC2(C)C)C1 28251,C1(NC(CCCCOCCC=C)=O)CC2C1CCN2C(=O)CC(CC)C1CCC1 28252,N1(C(c2ccc(C)cn2)=O)CCC2(CC1)CC2(CO)CNC(C1(Cl)CC1)=O 28253,N1(C(C(CC)C#N)=O)CCCC(C(=O)NC2COCC2CO)CC1 28254,N1(c2nnc(CC(C)C)n2CC(C)C(C)C)CC2C3CCC(CC3)C2C1 28255,Cc1ccccc1CC(N1CCCC(CCNC(c2cncn2C(C)C)=O)C1)=O 28256,c1(OCC#C)cncc(CN2CCC(SC)CC2)n1 28257,C(CC(C)(C)CC(=O)NCC1CC(C)CCN1C(c1cccs1)=O)OC 28258,c1(C(=O)NC2(CC=C)CCN(C(=O)CSCCC(C)C)C2)cnc(C)c(C)c1 28259,CC1C2CCC(C2)C1C(N1CCC(C)(CC(N2CCC2C2CCCC2)=O)C1)=O 28260,N1(C(C=C(C)C)=O)CCC2CCC12CNC(=O)Cn1cc(Br)ccc1=O 28261,c1(-n2c(C3CCC(C(C)OC)CC3)nc(CCCCCC)n2)cc(C)ccc1C 28262,c1(C(=O)NC(CC=C)CNC(=O)CCCC2CCCCC2)ccc(C(C)C)cn1 28263,c1(C(=O)OC)cncc(C(=O)NC23CC(NC(C4CCCNC4=O)=O)(C2)C3)c1 28264,C(C(C(=O)N1CCCC(CN=[N+]=[N-])C1)C(C)C)NC(c1nc(CC)oc1C)=O 28265,C(C(CC1CCCC1)C(=O)NC1CCC(C)CC1)NC(COC(C)=O)=O 28266,CC(C)(C)COCC(=O)NC(C(=O)NCC(C)(O)C1CC1)c1cccs1.C(C)(C)C 28267,N1(C(c2c(OC)cccc2F)=O)CCC(C2CCN(C(=O)C(C)(C)C(C)C)C2)C1 28268,CCC(C(=O)OC)C(=O)NC1(CNC(c2cccc(SC(F)(F)F)c2)=O)CCC1 28269,c1(C(=O)NCc2cn(CCNC(C3C(=C)CC3)=O)nn2)cnnc(C)c1 28270,c1(CNC(c2cccc(O)c2OC)CC)cc(F)c(N2CCOCC2)c(F)c1 28271,N1(CC(=O)NC(c2cn(C)nn2)C(=O)NCC(=C)Br)CCOC1=O 28272,C1(NC(C(C)C2CCC2)=O)CN(C(c2cncn(C)c2=O)=O)CC12CC2 28273,C1(NC(CCC(C)c2ccccc2)=O)CC=C(C(=O)N2CCSCC2)C1 28274,c1(NCCCCC=C)nc(N2CC(C)OC3(CCCC3)C2)nc2c(C)nn(C)c12 28275,N1(C(C2CCC(=O)OCC2)=O)CCN(C(c2ccc(F)s2)=O)C2CCC12 28276,C(=O)(C(F)CC(C)(C)NC(c1ccc(O)cc1)=O)N1CC(C#C)C(O)C1 28277,N1(C(C2C3CN(C(c4cc(OCC)c(Br)cc4)=O)C2C3)=O)CCC(C)C(F)(F)C1 28278,N1(C(c2c(CNC(c3cc(C(C)C)[nH]n3)=O)occ2)=O)CC2(CSC2)C1 28279,N1(C(C(C)CS(C)(=O)=O)=O)CCN(C(C2(C)CCN(C)C2=O)=O)CC(C)(C)C1 28280,N1(C(C(=O)NCCOCCOCC)C2CC2(Br)Br)CC(C)(C)C1c1ccccc1 28281,C1(C(=O)NCCCN(C(C=C2CCC(C)C2)=O)C2CC2)(CO)CC(C)(C)C1 28282,C=CCC(CC(F)F)NC(=O)C(CCC1CC1)NC(c1ccn(C)c1C)=O 28283,C1(CC(=O)NCCCCCNC(C(C(C)C)F)=O)CC2(CCOCC2)CO1 28284,C1(NC(C(c2ccc(Cl)nc2)(C)C)=O)CN(C(C2CC(C)(C)C2)=O)CC(F)(F)C1 28285,CCS(=O)CC(=O)NCC(C)NC(c1cccnc1OCCOCC1CC1)=O 28286,n1(CCC(N2C(CC(=O)NC)COCC2)=O)ccc2ccccc2c1=O 28287,CC1=C(C(=O)N2CCCCCC(CNC(=O)CNc3ccccc3Cl)C2)CCO1 28288,O(N(C(=O)CN=c1[nH]c(=NC)[nH]c(=NC(C)C2CCC2OC)[nH]1)c1cccnc1)CC 28289,c1(C(N(C)CC2CCCN2C(c2coc(Cl)c2)=O)=O)ccc(F)c(O)c1 28290,c1(C(=O)NCCCC(C)NC(C2(CCF)CCC2)=O)cc2cccnc2nc1O 28291,c1(C(=O)NC2CCCC23CN(C(=O)Cc2cccs2)C3)ccc2nccnc2n1 28292,C1(C)(C(N2CC=CC(NC(C(CCC)=CCC)=O)C2)=O)CCS(=O)(=O)CC1 28293,C(=O)(C(C)(C)CCC(=O)OCC)N(C(C1CCCN(C(C2CC(=C)C2)=O)C1)C)CC 28294,C1(C(N(C2CC(CO)C2)C)=O)CCOC1C(=O)NC1CCCC1F 28295,C1(COCC)CCCN(C(=O)C(Cn2cccn2)NC(c2ccc(C#N)o2)=O)C1 28296,C(=O)(Nn1nnc2c1CCCC2)C1C2(CC(NC(C(C)(C)OCC)=O)C2)C1 28297,C(=O)(C1=CC2(CCN(C(=O)Cn3c(O)nnc3O)C2)C1)NCc1cc(C)oc1 28298,c1(NC(C2C(NC(C3(c4ccncc4)CC3)=O)C2)=O)cccc(Br)c1 28299,c1(C(=O)NCCC(CNC(C2COCC2(C)C)=O)OC)cc2nccnc2[nH]1 28300,C(=O)(C(CCCc1ccc(Cl)cc1)N1CCC(C)(OC(C)=O)C1)NCCCSC 28301,C(CCC(C)(C)C(=O)Nn1nnc(C)c1C)NC(C(CC#C)O)=O 28302,N1(C(CC2C(C(C)C)OCCC2)=O)CCN(C2CC2)CC(O)C1 28303,CCC(C)C(O)C(C)C(=O)N1CCCC(CCNC(c2cscn2)=O)CC1 28304,N1(C(C2C(OCC)C2)=O)CCCC(C)(C)C1CNC(c1cnn(CC(F)F)n1)=O 28305,C1(NC(C(CC=CC)C)=O)C2CCC1CN(C(=O)CC1(O)CCCOC1)C2 28306,N1(C(C2C(NC(c3c(CC)ccs3)=O)C2(C)C)=O)CCC(O)(C(F)F)C1 28307,c1(CNCC(=C)Cl)csc(C2OCCO2)c1 28308,C1(C(N(C)Cc2c(C)ncs2)=O)CCN(C(c2cncc(C#N)c2)=O)C(C)(C)C1 28309,c1(C(N2C(CC)C(NC(c3ccccn3)=O)CC2)=O)ccc(OC)c(Cl)c1F 28310,CC1(CNC(C2(CF)CCOCC2)=O)COCCN(C(C2CN(C(N)=O)C2)=O)C1 28311,C1(C(=O)NCCC(C)N(C)C(c2ccc(C3CC3)o2)=O)C2CC(F)(F)CC12 28312,Cn1nnc(N2CCCC2C(C)(C)NC(=O)C(F)OC(F)(F)F)n1 28313,Cc1nc(N2CCCC(NC(c3cc(C)c(F)cc3C)=O)C2)c2c(n1)CCC2 28314,CCC(C#N)(CC)C(=O)NC1CCC(NC(=O)CCOc2ccccc2F)C1 28315,c1(C(=O)NC(CN(C(CC2(COC)CC2)=O)CC)CO)ccc(F)c(C(N)=O)c1 28316,N1(CC)CCCCCC1.C12CCN(CC1)C(=O)Cn1ncnc1C(C)NC2=O 28317,c1(CC)cc(CC)cc(S(=O)(=O)N2CC(C(=O)OC)OCC2C)c1 28318,C=CCC(C)(C)C(=O)NCC1(O)CC(NC(c2nnn(C)n2)=O)C1 28319,C1(CNC(C2(CC)CC2(F)F)=O)CCCN(C(C2(C(C)(C)C)CCC2)=O)C1 28320,C1(C(=O)NC(C2CCN(C(=O)C(n3cc(Cl)cn3)C)CC2)C)CCCCC(=O)C1 28321,N1(C(C(CCC)(C)O)=O)CC(C)(C)OC2(C1)CN(C(=O)C(C)C(O)CC)C2 28322,N1(C(C=C(CCN(C)C)Cl)=O)CCC2(CCN(C(c3ncccc3N)=O)C2)C1 28323,C1(C(N2CCN(C(c3ccc(C(C)=O)nn3)=O)CC2)=O)CCc2ncncc2C1 28324,c1(C(=O)NCCN(C)C(C2CCC(N(C)C)C2)=O)ccc(CCC(N)=O)cc1 28325,c1(C(=O)NC(C)CNC(c2cc(C(N)=O)co2)=O)c(Br)ncn1C 28326,C(=O)(C1=CCCCCC1)NC(CCO)C(F)F.C12CCCN(C1)C(=O)C2C 28327,c1(C(=O)NC23CCN(C(c4ccc(C)c(O)c4)=O)CC2C3)nccn2cnnc12 28328,C1(C(N2CCN(C(c3cnc(Cl)s3)=O)C3C2C3)=O)CCc2ccccc2CC1 28329,c1(NCC)ccc(Nc2cn(C)nc2C(=O)OC)cc1OC 28330,N1(C(C2(CC)CCCC2)=O)CCN(C(=O)C(C)Sc2ccoc2)CC1 28331,N1(C(c2c(C)cnnc2)=O)C2CCC1C1CC1(NC(C1CCCCN1N=O)=O)C2 28332,c1(OC)cc(C(=O)NCC2(F)CN(C(c3cc(O)cs3)=O)C2)c(F)cc1F 28333,C(CCC(=O)NC(C1CN(C(c2occc2Br)=O)C1)C)N(C(C)=O)C 28334,Cc1nc(C)c(C(=O)NCCCN2CCC(NC(=O)CS(N)(=O)=O)CC2)[nH]1 28335,Cc1ccc2c(C(N3CC(NC(C4(N(C)C)CCC4)=O)CC3C)=O)csc2c1 28336,C1(C(=O)NCCC2CC(NC(c3nc(CC)sc3)=O)C2)CN2CCN1CC2C 28337,Cc1ncnc(C)c1CNC1CCCN(CC(C)(C)C)C1=O 28338,N1(C(C(C)=C(C)C)=O)CCN(C(c2cc(C#N)ccc2C)=O)C2CCC12 28339,C1(OC)CC2(C1)CC(C(=O)NC1CCN(C(c3cnn(CC4CC4)c3)=O)C1)C2 28340,C1(N(C)C)(C(=O)NCC2C=CC(NC(c3cccnc3S)=O)C2)CCCCC1 28341,N1(C(c2cn(CCC(C)C)nn2)=O)CCC(NC(=O)CCC(C)(C)O)C(C)C1 28342,N1(C(CNC(C)=O)=O)CCCC(N(C)C(C2COCC(=O)N2C(C)C)=O)CC1 28343,C1(C(=O)NCC2CC(F)CN2C(c2cc(Br)c[nH]2)=O)CCCC12CCC2 28344,c1(C(c2cn(CC3CC3)nn2)NC(C23CC(C)(C2)C3)=O)ccc(F)cc1 28345,c1(C(=O)NC2C3(NC(Cc4c(C)non4)=O)CCC(C2)C3)cc(N)c(C)cc1Cl 28346,c1(C(N2CC(NC(CN(CCC)C)=O)C(F)(F)C2)=O)cc(C)c(C)cc1C 28347,c1(NCC(CC)N(C)C)ccc(S(=O)(=O)NCC(N2CCOCC2)C)cc1Br 28348,c1(OC)ncnc(N(C2CNCCOC2)C(c2cc(SC)oc2C)=O)c1C 28349,C(=O)(CS(=O)(=O)Cc1cccs1)NC1(CN(C(C(C)n2cnnn2)=O)C)CC1 28350,c1(C(=O)NC(C2CCOC2)C#C)oc(CNC(=O)OC(C)(C)C)cc1C 28351,N1(C(C2CCC(C)CC2)=O)CC2CC(C1)N2C(=O)CS(=O)(=O)N(C)C 28352,c1(C(N2C(C(C)NC(C(=O)NC(C)C)=O)CCC2)=O)cc2ccsc2n1C 28353,C1(C(=O)NCCC2CN(C(C3(C)CC4CC4C3)=O)C2)CCC2(CCCO2)CC1 28354,n1(C(C)C(=O)O)cc(-c2noc(C3CC34CC4)n2)c(O)nc1=O 28355,CC1CC2(CC(C(=O)NCC(O)C(=O)NC)C2)C1.C12(CC=CC1)C(=O)N2 28356,C1(CC(=O)NCC(CNC(C2(OC)CCCC2)=O)O)CCCCC1(C)C 28357,C1(N(C(C(CSC)C)=O)C)CN(C(c2c(O)cccc2F)=O)CC12CC2 28358,CCC(c1ccc(C)cc1)=CC(N1CCN(C(=O)COCCF)CC1C(C)C)=O 28359,c1(CC)ccc(NC(C2CN(C(C3CCCC(=O)C3)=O)CC2N(C)C)=O)c(F)c1 28360,N1(C(=O)NC2CC(OC)C2)CC(O)(Cc2nccs2)C1 28361,C1(NC(c2cn(CCC)nc2)=O)CCCCCC1NC(=O)C(F)(F)c1cncs1 28362,C(=O)(CC(F)(F)C(F)F)NC(C1CCCC1)CNC(Cc1c(C)nc(C)s1)=O 28363,c1(CC(=O)NCCC2CC(NC(c3c(CC)c[nH]n3)=O)C2)cccnc1OC 28364,C(=O)(C(CC(C)(C)C)NC(c1ccc(O)cn1)=O)NC(CC#C)C(N)=O 28365,c1(OC)cc(C(N2CCC(CNC(=O)C(F)=C3CCC3)C2(C)C)=O)oc(=O)c1 28366,N1(C(c2ccc(C)c(Cl)c2)=O)CCC2(CC1)CC2NC(C1(C)CCSCC1)=O 28367,C1(CNC(C(CCC)OCC)=O)CN(C)CCN1c1cnc(C#N)cn1 28368,C1(NC(C(C(C)(F)F)(C)C)=O)CCC2CN(C(C3(C(F)F)CC3)=O)CC2C1 28369,N1(c2cc(C)nc(C)n2)CCC(NC(C2CCC3CCCCN23)=O)C(C)(C)C1 28370,CC1COCCC1NC(C1CC12CC(NC(C1(c3cc[nH]n3)CC1)=O)C2)=O 28371,N1(CC(=O)N(C(C)CCO)C)CCN(C(c2ccc[nH]2)=O)CC1 28372,c1(CC(=O)NCCCN(C(C=CC(C)C)=O)CCO)cscc1OC(F)F 28373,c1(OC)ccccc1OCC(=O)N(C(C)CN(C(=O)C1=CCSC1)C)C 28374,C1(NC(C(C)NC(C)=O)=O)COCCC1C(=O)N(C1CC(C)(C)C1)C 28375,N1(C(C2C(C)CC2)=O)CCOC(CC(=O)N(C2CCCCC2)CCO)C1 28376,N1(C(C=C2CCN(C)C2)=O)CCC2CN(C(C3CC(N4CCOCC4)C3)=O)CC12 28377,Cc1cc(C(=O)NCC2C3CCC(C3)N2C(c2cnc(Cl)cn2)=O)cc(F)c1 28378,N1(CCCC2C(C)C2)CC2(CO)CC2(CO)C1 28379,c1(CNCCOCCOC)cnc2cc(Br)ccn12 28380,c1(NC(C2C3(CC(NC(c4ccn(CC)c4C)=O)C3)C2)=O)cccc2occc12 28381,C1(CC(N2CCC(OCC#C)C2)=O)C2CC(C2)N1C(c1cc(C)oc1C)=O 28382,Cc1cc(C(N2C3CCC2C(C(N2CC(C(C)(C)C)C2)=O)C3)=O)cc(O)c1 28383,c1(NC(C2(C)CCN(Cc3cccc(C=O)c3Br)CC2)=O)csc2nccnc12 28384,N1(C(CC(C)C2CC2)=O)CCC2(C(=O)NCCCP(C)(C)=O)CCCC12 28385,c1(NC(CNC(=O)NC2C(c3ccccc3)CCC(=O)C2)=O)nnc2ccccn12 28386,C1(NC(C2CCN(C(c3c(C)cc(CC)o3)=O)O2)=O)C(=O)NCCC1C 28387,C#CCC(C(=O)NOCC=CC)NC(=O)Cc1cn(C)cn1 28388,c1(OC)ccc(NC(=O)NCCc2ccc(C(C)C)c(F)c2)cc1C 28389,c1(C2C(C)C2)csc(NC(=O)OC(C)(C)C)n1.c1(N2C(=O)NCC2)cn[nH]c1 28390,C1(NC(C2CN(CC)C(=O)C2)=O)CN(C(=O)CSCC(C)C)CC2(CC2)C1 28391,c1(C(=O)NCCC(C)N(C)C(c2cccnn2)=O)csc2ccc(F)cc12 28392,c1(C(=O)OC)ccc2c(c1)CCC2NC(=O)Nn1cc(-c2nnccc2C)nn1 28393,C(C1=NOC2CN(C(=O)C#CC3CCOCC3)CC12)NC(c1c(C)scc1)=O 28394,c1(C(=O)NCC2(O)CCN(C(C3(C#N)CC3)=O)C2)ccc2ncnn2c1 28395,C1(C)(NC(CNC(CNC(c2cnc(C(C)C)o2)=O)=O)=O)CCCC1(C)C 28396,CCCCC(C)CCC(=O)NC1CC(CCC(=O)NC2COCC2CO)C1 28397,N1(C(c2cc(C)sc2C)=O)CC(C)OC2(CCN(C(C3CC3C(C)C)=O)CC2)C1 28398,c1(N2CCC(C=C)C2)nc(=NCCc2cccnc2C)[nH]c2c1cnn2C 28399,C(=O)(C1CCCc2c1ncn2C)NCC(C)(CO)NC(Cc1cc(C)on1)=O 28400,N12CCC(C1C)NC(=O)C1CCN1Cc1ccc(o1)C2=O.C(C)(C)(C)SC 28401,c1(C(=O)NCC2(SCC(=O)NCc3cn[nH]c3)CCCC2)cc2n(n1)CCCO2 28402,c1(OC)cc(C(=O)NCC2C=CC(NC(c3cc(=O)n(C)cn3)=O)C2)c(F)cn1 28403,C1(C(=O)NC2C(NC(C3CC(C)(C)OCC3)=O)CC2)CC2(C1)CC1(CC1)C2 28404,C1(NC(C2ON=C(C)C2)=O)CC2(C(=O)NCC3(C4CC4)CCC3)COC1C2 28405,C1(C(=O)NCCN(C(c2ncc(N)nc2C)=O)CC)CCC2CC2CC1 28406,N1(C(CC2CCC(C)CO2)=O)CCC(C)(CNC(C2C3CC4C(C3)C24)=O)CC1 28407,N1(C(C2C(NC(=O)C3CC3)COCC2)=O)CCC(F)(F)C(O)C1 28408,CCCCC(C)(F)C(=O)NCC(C)(C)NC(c1cc(OC)c(N)cc1F)=O 28409,c1(NC(CC2N(C(c3n(C)ccc3)=O)CCC2)=O)ccc(C(C)(C)C)cc1 28410,C1(CN(C2CCN(C(c3ccc(-c4ccco4)s3)=O)C2)C2CC2)CCCOCC1 28411,N1(C(Cn2c(C)ncc2)=O)CCC2(CCN(C(=O)C(S)C(C)C)C2)C1 28412,C12(CCS(=O)(=O)CC1)C(=O)N2.c1(CC(C(=O)NCC2CCC2)N)ccc(Cl)cc1Cl 28413,n1(CC)cnc2c(NCC3CC3(F)F)[nH]c(=NCC3(C)CCC(F)(F)CC3)nc12 28414,c1(N(C)C)cc(CNC(=O)C(c2ccc(-c3nn[nH]n3)cc2)O)cc(F)c1 28415,c1(C(N(CC(C)(C)CNC(c2ccc(C(F)F)o2)=O)CC)=O)cnnc(C)c1 28416,C#CCCCCCCC(=O)NCC(C)C(F)C(=O)N1CC(NC(C)=O)C1 28417,C1(NC(C=CC)=O)CN(C(c2ccc(C(=O)OC)cn2)=O)C2CC12 28418,C(COCC)(CCCC)NC(CONC(CN(C1CC1)CC)=O)=O 28419,C1(CNC(COC)=O)CCCC2CN(C(c3cnc(CC(C)C)s3)=O)CC12 28420,C(=O)(C1=C(Cl)CCC(C)C1)N(CCN(C(CC(C)P(C)(C)=O)=O)C)C 28421,C(=O)(CS(=O)(=O)CC(C)C)NCC1C(C=C)CN(C(=O)C(C)(CO)NC(C)=O)C1 28422,Cc1ccccc1-n1cc(C(N2CC(NC(C3CC3C(F)F)=O)C2)=O)nn1 28423,CCN=C(NCCC(=O)NC)N1CCC(O)CC(C)(C)C1 28424,N1(C(C23C(CN(Cc4cccc(N(C)C)c4)C2)C3)=O)CC2CCCC2C1 28425,c1(CC(=O)N(CCC(C)NC(=O)CCCCN(C)C2CC2)C)ccc2c(c1)CCO2 28426,C1(NCc2c3ccncc3no2)CCCC1C1CCCC1 28427,c1(C(=O)NCC2C(NC(CCCOCC)=O)COC2)ccc(-n2cnnn2)cc1 28428,N1(C(c2c(C)n(C)nc2)=O)CCCC2(CCN(C(c3cc(N)cc(O)c3)=O)C2)C1 28429,C1(NC(c2n(CC)ncc2)=O)CC2CN(C(c3cccc4c[nH]nc34)=O)CC2C1 28430,C1(CC(=O)NCCOC2CN(C(C3C(C(C)O)C3)=O)C2)CCCCC1C 28431,C1(OC)CC(C(=O)NCC(C2CCCCC2)NC(C)=O)N(C(=O)C(C)C(C)O)C1 28432,c1(CC2(CC(=O)NCCNC(=O)CNC(=O)C3CC3)CC2)ccccc1 28433,N1(C(C(C)CC2CC2)=O)CC2CCC1C(NC(=O)CN1CCS(=O)(=O)CC1)C2 28434,C1(NC(CCCSC)=O)CS(=O)(=O)C2CN(C(C3CC4CC3CO4)=O)CC12 28435,C(=O)(C(CO)C(C)(C)C)N1CC(C)C1C(=O)NCc1nnnn1C1CC1 28436,c1(CC)nc(N2CC3C(CNC(C4(CC(C)C)COC4)=O)C3C2)cc(C#N)n1 28437,C1(N(C(C(C)c2cccs2)=O)C)CN(C(C2CC(=O)C23CCC3)=O)CCC1O 28438,CCCC(O)C(CO)NC(=O)C(CCC1CCC1)NC(C1CCCN1C=O)=O 28439,CC1=CCCN(C(C2CC(=O)CN2C(C2CC(O)C(F)C2)=O)=O)C1 28440,N1(C(C(COC(C)C)NC(C)=O)=O)CCC(C(=O)NC2(C(C)C)CCC2)C(O)C1 28441,c1(C(=O)NCCCN(C(C2CCC2(F)F)=O)CC)cc(F)cc(F)c1OC 28442,N1(CCC2(C(=O)N)CC2)CCCC1.C1(C(=O)NC(C)COC)(COCC)CC1 28443,c1(C(=O)NCC(C2CCCC2)NC(c2cnn(C)c2Cl)=O)c(F)cc(Cl)cc1F 28444,N1(C(CCC=C)=O)CCN(C(=O)CNC(=O)C=Cc2ccco2)CC1CC(F)F 28445,O=C1NC(C(N2CCC3CN(C(=O)CN4CCOCC4)C3C2)=O)C2CCCOC12 28446,C1(NC(C2(CNC(=O)CC3CCSCC3)CC2)=O)CCN2CCCCC12 28447,CCCC(CC)C(=O)NCC1(F)CCCN(C(c2cc(O)ccc2Br)=O)C1 28448,N1(C(CCOC)=O)CCC(C(C)(C)C)(CNC(=O)C(C)Oc2ccccc2F)C1 28449,N1(CC(=O)NC(C2CCN(C(C3CCCC34CCC4)=O)C2)C)C(=O)NC(C)(C)C1=O 28450,N1(CCNC(C(C)CC2CC2)=O)CCC(NC(C2CCOC2(C)C)=O)CC1 28451,Cc1nn(C)c(C)c1C1OCCC1n1cc(CS(=O)(=O)CC(C)C(=O)O)nn1 28452,c1(C(C(=O)N(C2CCOC2)CCc2cc[nH]n2)Nc2cccs2)ccc(Br)cc1 28453,C(C(C)(C)CN=C(NCC1CCCO1)NC1CC(c2ccccc2C)C1)OC 28454,C(C)(C(C)C=O)N(C)C.c1(CNC(CSCCOC)=O)noc(C)n1 28455,C1(COC)CC(CNC(=O)C(C)Cc2ccnn2C)N(C(c2cccn2C)=O)C1 28456,Cc1ccc(CC(=O)NC2CC(CCNC(c3ccc(C(F)(F)F)[nH]3)=O)C2)o1 28457,c1(C(=O)NCC(C)CNC(=O)CNC(C2CCCC2)=O)coc(Br)c1 28458,CC(C)CC(C(=O)NC(CC1CC1)C(=O)N(C)Cc1cnn[nH]1)C(N)=O 28459,C12(CNC(CC(CCCC)CC)=O)CC3CC(CC(C3)C1NC(=O)CC#N)C2 28460,CCCC(C)(CC)C(=O)NC(C)CCNC(=O)C1=CSCS1 28461,c1(CNC(c2n(CC=C)nnn2)c2cnn(C)c2)cc2c(s1)CCCC2 28462,C12(CNC(C3CCN3C(C3(COC)CCCCO3)=O)=O)CCC(CC1)OC2 28463,C(CC(=O)NC1CCN(C(=O)C(F)(F)c2csc(Cl)c2)C1)(C(F)(F)F)OC 28464,C1(CC)(CC)CC(C(N2CC(N(C(=O)C(C3CCCOC3)OC)C)C2)=O)C1 28465,C1(NC(c2c(OC)ccs2)=O)CN(C(C2(C)CCNC2=O)=O)CCC12CCC2 28466,CCCC(C)(CC)C(=O)N1CC(CC(N2CCCC2CCO)=O)(OC)C1 28467,C(C)(C)(CN=c1[nH]c2ccccc2o1)NC(C(C(CC)C)O)=O 28468,c1(C(CNC(C2(C(C)(F)F)CC2)=O)NC(C2C(COC)C2)=O)ccc(C#N)cc1 28469,c1(C(=O)NC2CCC(NC(C(CSC)O)=O)CC2)ccnc2[nH]c(C(F)F)nc12 28470,Cc1cncc2cc(C(=O)NC3CCCC3NC(C3CC(=O)NC3(C)C)=O)sc12 28471,N1(C(CN(C)CC)=O)CCC2(C=C(C(=O)NCC3CC(C(=O)OC)C3)C2)C1 28472,CCCC(CNC(C1CCCC1O)=O)C(=O)NCCC1CC1C 28473,N1(C(c2c(C)n(C)nc2)=O)CCC(C2CC(NC(C3(C)CCCS3)=O)C2)CC1 28474,CC1CC(CCNC(=O)CCOC2CCCC2)CCN1C(=O)CC(Cl)Cl 28475,Cc1cc(C(=O)NCC2(C(=O)NCCN3CCCCC3)CC=CC2)ncc1F 28476,CC(C)CC(F)(F)C(=O)NCC1CC(C)CCN1C(C1CCC(CCO)CC1)=O 28477,C1(NC(C(CCCCC)O)=O)CCN(C(c2ncc(C)cc2C)=O)CC12CCC2 28478,C1(CNC(c2ccoc2)=O)OCCC1C(=O)NC(C1CCOC1)C1CC1 28479,CC1CCC(CNC(=O)CCOCC(F)F)CN1C(c1ccc([N+](=O)[O-])[nH]1)=O 28480,c1(OC)ccnc2c(NC(=O)Cc3csc(=NCc4cocn4)[nH]3)cccc12 28481,C(=O)(C(C)(O)C(C)(O)C(=O)Nc1csc(Br)n1)OC 28482,N1(C(C(C=C=C)C)=O)CCN(C(=O)Cn2nc(C)c(Cl)c2C)CC1C(F)F 28483,CC(C)C(F)C(=O)NC1CCC(CNC(c2cc(Cl)ccn2)=O)C1 28484,Cc1ccc(N)c(C(=O)NCC2CCCN2C(=O)C(C2CC2)N(C)C)c1 28485,C(CNC(=O)Cn1cc(C)cn1)(CC(=O)NCCn1nncc1C)OC 28486,N1(C(C2N(CCCC)CCCC2)=O)CCN(C(c2ccc(O)nc2)=O)CCC1C 28487,c1(OCC(=O)NC)cc(CN2CCC(CF)CC2)ccn1 28488,N1(C(C2(OCCNC(C=CC=C(C)C)=O)CCC2)=O)CCC12CCCC2 28489,N1(C(=O)OC(C)(C)C)CCCC(C(N2CCC(NC(=O)C3CC3)C2)=O)CC1 28490,c1(C(N(CCC2CCN(C(C(CCC)(F)F)=O)CC2)C)=O)[nH]cc2c1CCCC2 28491,Cc1cccc(C(O)C(=O)NC2CC2NC(=O)CCC2(C)CC2)c1 28492,C1(C(N2CCC(CN(C)C)C2)=O)CN(C(C2COCC2(C)C)=O)CC1(F)F 28493,C(=O)(C(C)(C)C(C)O)N(CCCNC(c1ccnn1CC(F)(F)F)=O)CC 28494,CCC(CCC(=O)NC1C=CCN(C(=O)CCc2ccc(C)s2)C1)OC 28495,Cc1csc(=O)n1CC(=O)NCC1CC(C)N(C(=O)C=CC(C)(C)C)C1 28496,CCC(C)CC(=O)C(=O)N1CCC2(CC(C(N3CCOC(C)C3C)=O)C2)C1 28497,c1(OCC(=O)N(C)CCOCCCNC(C2CCC(F)C2)=O)ccc(Br)cn1 28498,C1(CCCC)(C(=O)OC)CCCN(C(=O)C(c2ccccc2OCC)OC)C1 28499,Cc1n[nH]cc1S(=O)(=O)NC(c1cn(C(F)F)ccc1=O)=O 28500,n1(CC)nnc2cc(C(=O)N(CC(O)CNC(=O)C(=O)NCC(F)F)C)ccc12 28501,C1(CC)CN(C(c2ccc([N+](=O)[O-])s2)=O)CCN1C(C1CCN(C)CC1)=O 28502,C(=O)(C1=CCCOC1)N(CC(C1CCCC1)C1CC1)C(C)C.C1=C(C)NC1=O 28503,C=CCCC(F)(F)C(=O)NCCCC1CN(C(c2cnn(C(F)F)c2)=O)CCO1 28504,c1(C(=O)NCC2C(NC(c3c(OCC)cccn3)=O)C2)cc2cc(O)ccc2[nH]1 28505,c1(C(N(C2CCN(C(=O)CSC3CC3)C2)CC#C)=O)cc(Cl)n(C)n1 28506,N1(c2nc(CC)nc(Cl)c2CC)CC(NC(=O)C(O)C(C)C)C2(CCOCC2)C1 28507,C1(C(N2CCC(c3cccc(F)c3)CC2)=O)CC2CC2N1C(C1CC1F)=O 28508,c1(SC)ccc(CC(=O)NC2CCCC(NC(=O)Cc3ccc(Cl)cn3)C2)cc1 28509,C1(O)(CN(C)C(C2(C)CCSCC2)=O)CCCN(C(C2CC23CC3)=O)C1 28510,c1(C(N(C(CN(C(C(CC=C)CC)=O)C)C)C)=O)cccn2nccc12 28511,C1(C(C(=O)NCCC(C)N(C(=O)CC2(C)CC2)C)OCC)CC(F)(F)C1 28512,C(CC(=O)OCC1CCCN(C(=O)CN2CC3CC3C2)C1)(C(N)=O)N(C)C 28513,c1(N2CCCCC(SC)C2)nc(=NCC2SCCS2)nc(N2CCOCC2)[nH]1 28514,c1(CN2C3C(C(N4CC(C(=O)OC)C(O)CC4)=O)C(C3)C2)cc(O)c(Br)cc1O 28515,c1(NC(C2(CNCc3c(C)cccc3)CC2)=O)cccc2nscc12 28516,C(=O)(CC(F)(F)F)NC1(CNC(COCCC)=O)CCOC1.C1(=O)C(O)CN1 28517,c1(C(=O)NC(C2CCN(C(c3ccnc(C(F)(F)F)n3)=O)C2)C)cncc(N)c1 28518,c1(OC)cc(C(=O)NC(CNC(C2CC(=C3CC3)C2)=O)C2CC2)c2occc2c1 28519,C(=O)(CC(O)c1ccccc1)NCC(C)N(C)C(C1(C)CCCC1)=O 28520,CCC(C)(C)CCCC(=O)NC1(CCNC(c2ccc(CF)cc2)=O)CCCC1 28521,c1(C(N2C3C(NC(CSCC#C)=O)CC(C3)C2)=O)cccc2nccnc12 28522,c1(C(=O)NCc2ccsc2C(N2CCC2C2CCC2)=O)n[nH]cc1[N+](=O)[O-] 28523,C(=O)(C(F)(F)F)NCC(=O)N(CCCN(C(C(C)OC1COC1)=O)C)C 28524,CCC(C(=O)NCC1CN(C(c2ccc(C)c(CO)c2)=O)CC1(F)F)C(C)C 28525,c1(NC(C)=O)c(C(N2CCC(NC(=O)CCC3CC(C)C3)C2C)=O)cccc1C 28526,C#CC1CN(C(=O)C(C)=CCC)CCN1C(=O)CCc1ccccc1C 28527,CN1CCC(C(=O)N2CC(CO)(NC(=O)C3=CCCC3(C)C)C2)c2ccccc21 28528,c1(C(=O)NC2C3CN(C(C4(SC)CC4)=O)CC32)ccc(F)c(C(C)C)c1 28529,C1(N2CCOCC2)(CNC(=O)Nc2nc(N(C(C)=O)CC)sc2)CCN(C)CC1 28530,c1(C(=O)Nc2c(C)csc2)cc2cccnc2s1 28531,C1(C(N2CC(C)(CO)C2)=O)CCCCN1C(C)=O.O(C=CC(=O)NC(C)C)CC 28532,N1(C(CCC=C(C)C)=O)CCOC2(C1)CN(C(=O)C(C)SCc1ccccc1)C2 28533,CC1CCC(C)(C(N2CC3(CC(NC(C4CN(C5CCOC5)C4)=O)C3)C2)=O)CC1 28534,Cc1ccnc(O)c1C(=O)NCCC1CC(N)C1 28535,n1(CC(N2C(C(NOCC(CC)C)=O)CSC2)=O)nc(C)cc1C 28536,S(=O)(=O)(c1ccc(C)c(C)c1)NCCNC(CCC)CC(F)(F)F 28537,C1(NC(c2c(CC)occ2)=O)C2CC3C1C3C2C(N1CCCC1CN=[N+]=[N-])=O 28538,CC1CN(C(c2sccc2CNC(c2cc[nH]n2)=O)=O)CC1O 28539,Cc1ccc(O)c(CC(N2CCN(C(c3nc(O)sc3C)=O)C(C)C2)=O)c1 28540,CC1CCCCCN1C(=O)CCOCCN(C)C(c1cncn(C)c1=O)=O 28541,N1(C(c2ccc(C(C)C)cn2)=O)CCCC(C)(NC(=O)CC2(O)CCCOC2)C1 28542,c1(C(=O)NCC2(CNC(C(c3cncnc3)C)=O)CCC2)ncc(Cl)cc1F 28543,C1(C(N(C)CCNC(C2CCC(C(F)(F)F)CC2)=O)=O)CCc2nnc(O)n2C1 28544,C1(NC(CSC(C)C)=O)CC2CN(C(=O)CN3CC(=O)NC3=O)CC2C1 28545,C1(C)(NC(CC2OCCN(C(C3CCN(C)CC3)=O)C2)=O)CCC(C)(C)C1 28546,CCC(CCCO)NC(=O)C(CO)NC(=O)CC(C)=C(C)C 28547,c1(CC(=O)NC(CC2CN(C(c3cc(C)oc3)=O)C2)C)cnc(Cl)cc1C 28548,C1(O)(CC(=O)N(C(C)CNC(=O)C(c2ccc(Cl)s2)C)C)CCCCCC1 28549,CC1=C(C(=O)N2C3CCC(C3)C2C(N2CC(C(C)(C)O)C2)=O)CCC1 28550,c1(C(=O)NC2CC(C)(C)N(C(C3COCCO3)=O)C2)cc(F)cc2nn[nH]c12 28551,C1(NC(c2nnc(C)s2)=O)C2CC1CN(C(C1CC1C1CCCC1)=O)C2 28552,C(=O)(C(C)(C)CS(N)(=O)=O)NC1(CCNC(C2(C)CC2c2ccccc2)=O)CC1 28553,C1(O)(CCNC(C2CCS2(=O)=O)=O)CN(C(c2ncoc2Br)=O)C1 28554,c1(C(=O)NCCN(CCOC)C(C2CCOC2C)=O)cc(C)ncc1C 28555,CC1(C(=O)N2CCC(C(C)(C)NC(c3cn[nH]c3)=O)C2)COc2ccccc21 28556,C(=O)(CCS(=O)(=O)CC(C)C)N1CC(NC(Cc2cc(C)on2)=O)C(CO)CC1 28557,c1(C(=O)NC(CC=C)CNC(c2cnc(C(F)F)nc2)=O)cc2n(n1)CCC2 28558,CC(Cc1cccn1C)N=c1ccnc(NC2CCC(=O)NC2)[nH]1 28559,N1(C(C(=O)C2CC2)=O)CCC(O)C2(CCN(Cc3ccn4ccnc4c3)CC2)C1 28560,c1(C(=O)NC2CC(NC(c3ccn(C(C)C)n3)=O)C2)ccc(=O)n(C2CC2)c1 28561,CC(=NO)C1CC(C(N2CC(NC(=O)CSCc3ncc[nH]3)C2)=O)C1(C)C 28562,Cc1cccnc1C(=O)NC(C1CCOC1)CNC(c1cncc(C(F)F)c1)=O 28563,C1(C(N(CC#C)C)=O)(SC2CCCC2)CCOCC1.c12cn(nn1)CC(=O)NC2 28564,Cn1nc(C(=O)NC2CC(CNC(C3(C#N)CCCO3)=O)C2)cc1Br 28565,c1(-n2cc(CN3CCN(N(C(C)C)C)CC3)nn2)ccc(Cl)c(C(=O)O)c1 28566,c1(SCC(=O)NC(COC)(C)C)ccccn1.C1CC(=O)N1 28567,C1(C(N(CCCCCC)CCNC(=O)C(O)CCCC)=O)CCn2nccc2C1 28568,c1(C(N2CCC(CN(C)C(C3C(OC)COC3)=O)C2)=O)ccncc1N(C)C(C)C 28569,c1(OCC)ccc(F)c(CN2CCN(CC(=O)OC(C)(C)C)C(=O)C2)c1Br 28570,C12CC(COC)CN1C2=O.n1(C(CCC)C2CCCC2)cc(-c2cc[nH]n2)nn1 28571,c1(C(=O)NCC(C)=CC(N2CC(C)CCC2C)=O)cccc2cc[nH]c12 28572,C(CC(=O)N1CC(C)(NC(=O)CC23CCC(C)(C2)OC3)C1)(C(C)C)OCC 28573,c1(-n2ccc(C)n2)ccccc1C(=O)NCC(F)CNC(C1CCOCC1)=O 28574,C1(C(=O)NCC2C(NC(c3cc(C(F)(F)F)ccn3)=O)CC2)CC2(CCCC2)C1 28575,N1(C(C(CC)NC(N)=O)=O)CC(F)(F)CC1C(=O)Nc1nc(C)ccc1C 28576,c1(C(N(CCN(C)CC2CCC(C)(C)CC2)C)=O)occ2c1CCC2 28577,N1(C(C2C(CCC)C2)=O)CC(NC(=O)C=C2CCCCC2(C)C)C2CCCC12 28578,c1(C(=O)NC2(CNC(C3C(C)(C)COCC3)=O)CCOC2)ccc2cc[nH]c2n1 28579,O=C1CC(NC(C2CCCC2NC(c2ccco2)=O)=O)C(=O)N1 28580,C(C(=O)N(CC(C)(O)C1CC1)C)(C(C)OC)NC(CC1(CSC)CC1)=O 28581,CC1(CC(=O)Nc2ccn(C3CC3)n2)CCN(C(=O)CCCn2cccn2)C1 28582,c1(OC)snc(C)c1NC(=O)NCC1CCN(C(C2CCCN2C)=O)C1 28583,C1(CC)CCC(C(=O)N(C2(C(N3CC(C(F)(F)F)C3)=O)CC2)C)CC1 28584,C1(CNC(COCC(=O)NC)=O)CN(C(=O)CCc2ccc(NC)cc2)CCO1 28585,c1(NC(C(C(=O)OC)OC)=O)ccc(NC(=O)CCCSC(C)(C)C)c(C)c1 28586,C1(C(=O)OC(C)(C)C)CCC(C(=O)O)CC1.n12cc(nn1)CNC1CC2C1 28587,n1(C2(N3CCOCC3)CC2)ncc2cc(-c3ccc(C=O)cn3)cnc12.CC(C)C 28588,CCC(CCC(=O)N(C)CC1CCCN(C(C2CC(N(C)C)C2)=O)C1)OC 28589,C#CCCCCC(=O)N1CCC(OCCCNC(C2CCCS(=O)(=O)C2)=O)CC1 28590,N1(C(c2cnc(COC)s2)=O)CCCCC1CNC(c1cc(C(C)(C)C)[nH]n1)=O 28591,Cc1cn2cc(C(=O)N(C3CCN(C(=O)C4=COCCC4)C3)C)sc2n1 28592,C1(C(=O)NC(C=C)CO)CCCCN1C(c1cncn1C1CC1)=O 28593,c1(C(=O)NCC(CN(C(C(C)N(C(C)=O)C)=O)C)(C)C)cccc(CS(C)=O)c1 28594,C1(CC(=O)OCC)CN(C(CC2CC2)C(=O)NCCCF)CC(C)O1 28595,CC1(C)CC1(C(=O)NCCC(F)(F)F)NC(=O)CC1CCCSC1 28596,Cc1cnc2cc(C(N3C4CCC3CC(CNC(=O)COC(C)C)C4)=O)ccn12 28597,c1(C(=O)Nc2ccccc2Cl)c[nH]c2cc(-c3ccc(CNC4CC4)cc3)cnc12 28598,C(=O)(CC(C(F)F)C(C)(C)C)NCCCN(C(c1cccc(OC)c1)C)CC 28599,c1(C(=O)NC(C2CCCN(C(COCC(=O)NC)=O)C2)C)c[nH]c(=N)nc1C 28600,C1(C(=O)NC2(C(N)=O)CC2)(CNC(C2C(OC)CCC2)=O)CC12CCC2 28601,C1(C(=O)NC(C)(C)CNC(c2[nH]ccc2-c2ccccc2)=O)CCC2(CCC2)O1 28602,C(C)(C(=O)NC(C1CCC1)CO)N(C(=O)C=CCO)CC 28603,c1(C(N2C(CNC(c3c(C)c(Cl)ccn3)=O)CCCC2)=O)ccc(N)c(Cl)c1O 28604,c1(C(=O)NC2CCCC23CN(C(=O)CC(F)F)C3)ccnc2ccc(Cl)cc12 28605,C(=O)(CC(CC)CC(F)(F)F)NCC1N(C(CC(=C)C)=O)CCCCCC1 28606,N1(C(CN(C(c2ccco2)=O)Cc2ccccc2)=O)CCCC2(CCC2O)C1 28607,n1(CC)nccc1C(C(=O)NC1CCCC1)N(C1CCOCC1)C 28608,c1(C(=O)NC2CC3(C(NC(CCCC4C(C)C4)=O)C3)C2)cccc2c1C(=O)NC2 28609,Cc1cc2[nH]c(C(=O)NC34CCC(CC3NC(c3cc[nH]c3)=O)C4)cc2s1 28610,C1(NC(C(CCCC)O)=O)CC2CC(NC(C3(S(N)(=O)=O)CC3)=O)CC2C1 28611,c1(OCC)nc(C(N)=O)ccc1NC(c1cccc(-c2cccc(NC)c2)n1)C 28612,C12(CC(=O)NCC3C(CNC(CCCCCSC)=O)C3)CCC(CC1)C2(C)C 28613,N1(C(CC)C)CCc2cc(NCCN(CC)CC3(C)CCC34CCC4)ccc21 28614,N1(C(c2c(C)ccc(C)c2)=O)CC2CCC(C1)C2NC(=O)C(O)C(C)C 28615,c1(C(=O)NC2C(C)CN(C(=O)C=Cc3cocn3)C2)nnn2c1CCCC2 28616,CC1CN(Cc2ccc(N3CCOCC3)cc2Cl)CC(C)N1C 28617,C1(C(N2CCCN(C(c3cc(O)cc(=O)o3)=O)CC2)=O)(OC)CCC(C)CC1 28618,C(=O)(C(C)(F)C(=O)OC)N(C1CCN(C(C(CC#C)C)=O)CC1)CC#C 28619,Cc1ccc2c(c1)CC(C(=O)NCC(C)N(C(=O)CCSc1nccn1C)C)O2 28620,N1(c2nnc(CCC(CC(C)C)C)n2CC2CCOC2)CC2C(=O)NC(=O)C2C1 28621,Cc1sc(C(N2CCC(N(C(=O)C(CSC)NC(=O)C(F)(F)F)C)C2)=O)c(C)c1C 28622,N1(C(C(CC)=CCCC)=O)CCOC(C)C1C(=O)NCCOCCCF 28623,C(=O)(CCCCC(=O)NC(C(=O)NCCOC(=N)O)C1(O)CCC1)OC 28624,C=C(C)CCCC(=O)N(CC(=O)NC1CC1CC)C 28625,N1(C(Cc2c(C)nn(C)c2)=O)CCC2(CC1)CC2NC(=O)C(F)C(C)(F)F 28626,N1(C(c2nccc(CC)c2)=O)CCC2(CO)CN(C(=O)CS(C)(=O)=O)CC2C1 28627,CCC(CC(=O)NC(C)(C)C(C)CC(=O)N1CCCC1C1CC1)C(F)F 28628,c1(C(=O)NC(CCCC)CNC(=O)CNS(=O)(=O)NC)coc2c1C(=O)NCC2 28629,N1(C(CCC#C)=O)CCN(C(=O)C(C)(CC)CO)CC1c1ccccc1OC 28630,C1(NC(N(CCOC)CC=Cc2ccccc2)=O)CCOC2(CCC2)C1 28631,C(C)(CNC(c1nnsc1C)=O)(CC(C)C)NC(CCCC)=O 28632,Cc1c(C(=O)NC(C)CCCNC(=O)C(C#N)C2CC2)nnn1C(C)C 28633,c1(NC(=O)N(C2CCCC2)CCCC)ccc(C2CC2)cc1Cl 28634,c1(C(=O)NC(C)(Cc2ccncc2)C(=O)O)ccc([N+](=O)[O-])cn1 28635,C1(C(=O)NCC2C(COC)C2)CN(CF)CC12CCC2.C1(C=O)CC(CO)(CO)C1 28636,N1(C(=O)NC2CC(c3ccc(Br)cc3)C2)CCC12CC1CCC2C1 28637,C1(C)(C(N2CCC(NC(CCC(CC)OC)=O)CC2)=O)CC2CCC(C1)S2(=O)=O 28638,c1(C(=O)NCC2(NC(CC(=O)NCC#C)=O)CC2)ccc2c(c1)C(=O)CCC2 28639,C(=O)(CCCC(=O)OC(C)(C)C)NC1CCCC(NC(c2c(C)coc2)=O)C1 28640,N1(C(C(C2CCCO2)SC)=O)CCCC(CO)(CNC(C2(CO)CC2)=O)C1 28641,C1(NC(C(C)C)=O)CS(=O)(=O)C12CCN(C(c1cnn3ccnc(N)c13)=O)CC2 28642,c1(C(=O)NC2CC(OC)CN(C(c3c(Cl)n[nH]c3C)=O)C2)c(C)cc(C)nc1O 28643,c1(-c2ccc(CN(C)C)cc2)ccc2c(CNC(=O)C3CC3)cnn2c1.C1CCO1 28644,c1(C(C(=O)NCCCC)NC(C2CCN2C(C)(C)C)=O)cccnc1 28645,C(=O)(CC(F)(F)C(F)F)NC1(C(N(CCC(C)(C)C)C)=O)CC(CO)C1 28646,C1(NC(C(CCC)O)=O)CCN(C(c2ccc(NS(C)(=O)=O)c(C)c2)=O)C12CC2 28647,c1(NC(C(=O)N(CC(=O)NC2CCS(=O)(=O)C2)CC2CC2)=O)ccc(O)cc1 28648,CCCCC(CC)C(=O)NCC(O)CC(N1CCC2(CSC2)C1)=O 28649,C1(C)(CNC(c2c(C)sc(Br)c2)=O)CCCN(C(=O)CC2CCC2)C1 28650,N1(CCC)C(=O)CCC1C(=O)NCC(C)(C)CN(C(=O)Cn1nc(C)nc1C)C 28651,c1(C(C)C)cc(C(=O)NCC2CCCC2NC(=O)CC2CCOC2)ccc1O 28652,Cc1c(NC(N2CCOC(CC(N3CCCC(C)CC3)=O)C2)=O)cccc1Br 28653,CC1CN(C(c2ccn(C)c(=O)c2)=O)C(C)CN1C(C1CCNC1=O)=O 28654,C1(CN(C)C(c2scnc2C(F)(F)F)=O)CCCN(C(c2ncccc2C)=O)C1 28655,C1(CC)(NC(=O)C(F)F)CCN(C(=O)C(C)(C)C)CC1 28656,c1(NC(C2CN(C(C3NC(=O)CC3C)=O)CCO2)C)ccc([N+](=O)[O-])cn1 28657,CCC(CC)CC(F)C(=O)N1CSCC1C(=O)NC1(c2cc[nH]n2)CC1 28658,c1(N2CC3C(CNC(C4C(OCC)C4)=O)C3C2)ncnc(C)c1F 28659,c1(C(=O)NC(CC)CNC(C2(C)CC(C)=NO2)=O)sc2cncn2c1C 28660,c1(C(=O)NC2CCN(C(C(CC)n3ccnc3)=O)C23CC3)cccc2[nH]ncc12 28661,c1(C(C(C)C)OC(C(c2ccccc2Cl)OC)=O)cc(Cl)ccc1F 28662,CC1(C)C2CCC(NC(=O)NC(C3CCCCC3)Cc3ccccc3)C1C2 28663,C(=O)(C1=CCC2CCC1N2C(=O)COC)N(C(CC)COC)C 28664,n1(CC(=O)N(CC(C)NC(C2CCCCC2O)=O)CC)nc(C)c([N+](=O)[O-])c1C 28665,C1(NC(c2c(OCC=C)cccn2)=O)CN(C(c2cc[nH]c2C)=O)CC2(CC2)C1 28666,N1(C(Cc2c(C)scc2)=O)CCC(C)(O)C1C(=O)NCCc1nnc(O)o1 28667,c1(C(=O)NCC(C)CN(C(=O)C(C)Oc2ccc(Cl)cc2)C)cccc(CO)n1 28668,CC(C)CCC(F)C(=O)NCC1CC2CCCC2N1C(=O)C=C(Cl)Cl 28669,N1(C(C=CC(C)(C)C)=O)CCCC(C2CCN(c3nc4ccccc4o3)C2)C1 28670,C1(NC(CSCC=C)=O)CC(NC(C2CC(c3cccc(Cl)c3)C2)=O)CC1O 28671,C1(C(=O)OC)CC(F)(F)CN1C(c1cc(C)c(C)s1)C(=O)NC(C)C 28672,C1(CNC(C(CC)(C)C)=O)C2CCCC1N(C(c1cc(C#N)no1)=O)C2 28673,C1(NC(CC(CC=C)(C)C)=O)CC2(CCC(CNC(C3C4COCC34)=O)CC2)C1 28674,n1(CC)cc(C#N)cc1C(N1CCCC1C1CCCCCC1)C(=O)NC(C)(C)C 28675,CCCC(C)(CC)C(=O)N(C)CCC1CCCCN1C(c1cnn(CCO)c1)=O 28676,N1(C(C(C)OCC2CC2)=O)CC(CNC(C2(C)CCN(C)C2)=O)CC(C)C1 28677,C(=O)(C(O)CC(C)(C)C)NCC(CC(C)C)NC(C1CCCC(F)C1)=O 28678,c1(C(N(C2CCN(C(c3cnsn3)=O)C2)CCC)=O)cc(Cl)cc(Cl)c1F 28679,c1(OC)nccc2c(C(N3CC4C(NC(c5cc(C)oc5C)=O)C4C3)=O)c[nH]c12 28680,N1(C(CC(n2ccc(C)n2)C)=O)CCCCC(NC(c2n[nH]c(C)c2F)=O)C1 28681,C12(C(N(C(=O)NC(C(C)C)C3CC3)C)C3CC3)CC3CC(CC(C3)C1)C2 28682,c1(C(C(=O)NC(CNC(Cc2cc(C(C)C)no2)=O)C)O)ccccc1F 28683,CC1(CC(N2CC(CO)(NC(c3coc(O)n3)=O)C2)=O)CCS(=O)(=O)N1 28684,C(C1CCCN1C)=CC(=O)N(CC)Cc1ccccn1.C1=CC(=O)NC1(C)C 28685,CC(C)(C(=O)N1CCC(NC(=O)Cn2nnc(=O)[nH]2)C1)C1CCCCO1 28686,C12(NC(C3CC(=C)C3)=O)CCC(CNC(=O)C(C)OCCOC)(C1)OC2 28687,c1(C(N2C(CNC(C3(C)CC(C#N)C3)=O)CC2)=O)ccc2c(Br)cncc2c1 28688,c1(C(=O)NCCCC2N(C(CSCCOC)=O)CCCC2)cccn2nncc12 28689,N1(C(C=CCCC)=O)CCCC(C(=O)NCc2conc2C)CC1 28690,c1(C(=O)NC2CN(C(c3cc(Cl)cnc3O)=O)CC2F)ccc2nonc2c1 28691,C1(NC(=O)Cc2nc(C3CC3)cs2)CN(C(c2cc(Cl)ns2)=O)CC12CCC2 28692,C(=O)(CCCC(C)(C)C#N)N1CCN(C(CSc2c(C)cccc2)=O)CC1CF 28693,c1(C(=O)NC(CC)CNC(=O)CC2CCC(=O)N2)cc(C)c(F)cc1O 28694,Cc1ccc(C(=O)NC(C(C)NC(=O)C(C)C)C(C)C)c(=O)n1C 28695,c1(-c2c(C(=O)NCCN(C(c3c(CC)csc3)=O)CC)c[nH]n2)ccccc1F 28696,c1(C(=O)NCC2CCC(NC(Cc3scc(C)c3)=O)C2)cc2nccnc2cc1C 28697,c1(OC)ccccc1C(=O)NCC1CCC1NC(C1(C)CC=CCC1)=O 28698,c1(NC(COC)=O)ccc(F)cc1S(=O)(=O)N1CCCC1.C12CCN1C(=O)NC2 28699,c1(CCN(C(c2ccc(Cl)cc2)CCSC)CC)nnc2n1CCC2 28700,c1(C(C(=O)NCc2ccc(OCC(F)F)cc2)N(C)C)cc(F)c(F)c(Cl)c1F 28701,c1(OC)ccc(CO)c(NC(C2(C(=O)N(c3ccccc3)C)CC2)=O)c1 28702,C1(NC(C)=O)CC2CCCCCC12.[nH]1ccc(C)n1.C1CC(=O)N1C(C)(C)C 28703,C1(SC)COCCN1C(=O)CC1C2CN(C(=O)C=C3CCOCC3)CC12 28704,N1(C(C(F)=CC)=O)CC(NC(C2(c3ccccc3)CC(C)C2)=O)C(SC)C1 28705,c1(NC(=O)NC2C(CC)CC2)ccc(C(C)O)cc1 28706,c1(C(=O)NCCN(C(C2CCC2C(F)(F)F)=O)CC)cc2cccnc2cc1F 28707,c1(C(N(CC(C)NC(=O)C=CCOCCO)CC)=O)c(F)cc(OC)cc1F 28708,c12cccnc1CONC2=O.C1(CC(=O)NC2(C)CC2)CC(O)C1(C)C 28709,CC1CCC(C(=O)NC2(CNC(c3cncc(C(N)=O)c3)=O)CCOC2)CC1 28710,C1(C(F)(F)F)(OC)CC(NC(=O)NC2CS(=O)(=O)C2)C1 28711,Cc1csc(=O)n1CN(C(Cc1ccc(NC2CCC3CC23)cc1)=O)C 28712,C12CN(C(=O)C3=COCC3)CCN1C2.c1(CCCOCCOC)ccccc1 28713,N1(C(c2c(CC)cccn2)=O)CCN(CC2CCC(=O)N2)C(CC)C1 28714,CC(C)CCC(=O)NC(c1ccccc1F)CNC(c1ccco1)=O 28715,N1(C(C(c2ccccc2)NC=O)=O)CCC2CCC12 28716,Cc1cc(O)c(C(=O)NCC2(O)CCN(C(=O)CN3CCC(C)CC3)CC2)nn1 28717,CCC(CCC(=O)NCC1(C)CC1(C)C)NC(=O)CCN(C)CCO 28718,C1(CC(=O)N(C2CCCN(C(=O)Cc3conc3C)C2)CC)CCCOCC1 28719,C1(N(C)C)CC2(CCC(CNC(C3CCC4CCCCN4C3)=O)CC2)C1 28720,N1(C(CCc2ccc(C)nc2)=O)CCC(C)C(NC(c2ncc(F)cc2C)=O)C1 28721,c1(CN2CCC(C(=O)NCCc3c(C)ncs3)C2)csc2ccccc12 28722,N1(C(CN2CC(C)(OC)C2)=O)CCN(C(C2(CO)CC2)=O)CC2(CC2)C1 28723,n1(CC)nc(C(C)C)cc1C(=O)N(CC(C)NC(c1cc(C)c(Cl)s1)=O)C 28724,c1(C(N2CCC2CN(C(C(C)(C)C)=O)CCO)=O)ncccc1F.N12CCC(C1)C2=O 28725,CCCC(F)C(=O)NC(CCOC)C(=O)NCC1(CCO)CN(C)C1.N(C)C 28726,Cc1nnc(O)c(C(=O)NCC2CCCN2C(=O)CCCN=[N+]=[N-])c1C 28727,N1(C(C(C=CC)O)=O)CCC(CO)(CNC(C2(OC)CCC(C)(C)C2)=O)CC1 28728,C=CCCCC(=O)NCCOCCNC(c1cnc(SC)n1C)=O 28729,c1(CCC(N2C(C3(O)CN(C(=O)C=CBr)C3)CCC2)=O)cnc2n1CCCC2 28730,C1(NC(C(C)Oc2ccc(OC)cc2)=O)CCCCCN(C(=O)CN2CC=CC2)C1 28731,c1(C(N2CCC(NC(C(CC)NC(N)=O)=O)(CF)C2)=O)ccn2nccc2n1 28732,C(=O)(C(O)C(C)(C)C)NC(C)CC1CCN(C(c2cc(C(C)(C)C)no2)=O)CC1 28733,C#CCS(=O)(=O)CCNC(C1(C)CC(C(=O)OC)C1)=O 28734,C(=O)(C(=O)C(C)(C)C)NCC1(OC)CCN(C(=O)CCn2ccccc2=O)C1 28735,C1(CNC(C2C(C)N(C)CC2)=O)CN(C(c2cc(C(F)(F)F)ns2)=O)CC1(C)C 28736,c1(NC(C2CC(NC(CNC(CCC)=O)=O)C2(C)C)=O)n[nH]c2ccccc12 28737,c1(C(N(C2CCCC2n2cc(-c3ccccn3)nn2)C)=O)nn(C)cc1I 28738,C(=O)(C(O)(C(C)C)C(F)(F)F)NC1CN(C(c2c(C)nc(O)[nH]2)=O)C(C)(C)C1 28739,CCC(CNC(=O)C(=O)Nc1ccn(C)c(=O)c1)CC(F)(F)F 28740,N1(C(c2ccn(CCC)n2)=O)CC(C)(CNC(=O)CS(=O)CC)CC1(C)C 28741,c1(NC2(c3ccccc3)CC2)ccc2[nH]nc(Cl)c2c1.C12CCCCN1C2 28742,N1(C(COCCNC(CC)=O)=O)CC2CC(O)C1C2NC(=O)CN1CCCCC1 28743,N1(C(C2N(C)CCC2)=O)CCCC2(CCN(C(c3cscc3Cl)=O)C2)C1 28744,C(=O)(C1=CCCCO1)NC1C(C)(C)C(CC(=O)Nc2ccc(CO)nc2)C1 28745,c1(C(=O)NC2C(NC(C3(C(=O)OCC)CC3)=O)C2)occc1C 28746,N1(C(C(C)Sc2ccccc2F)=O)CCCC(C(=O)NC2C3CCC(F)C23)(CC)C1 28747,C(=O)(CCC(C)(F)F)N1C(C(N2CCC(OC(C)=O)C2)=O)COCC1 28748,C1(CCC)(CO)CCN(C(=O)Cc2nc(CNC(c3cnn[nH]3)=O)cs2)CC1 28749,c1(OCC)ccc(OCC(=O)N(CC(C)NC(=O)C(C)=C(C)C)C)cc1 28750,C(=O)(C(CC(C)C)N(C)C(c1cc(C(N)=O)[nH]n1)=O)NCc1[nH]nc(CC)n1 28751,N1(C(=O)NC2CCN(S(=O)(=O)C3CCOCC3)CC2)CCc2ccc(F)cc2C1 28752,C(C(C(=O)NC1CC1)N(CC(=O)OC)CC#N)(c1ccccc1)OCC 28753,C(=O)(CC(C)C(C)(C)C)NC1CC=C(C(=O)NC2CCN(CCOC)CC2)C1 28754,Cc1nc2ncc(C(N3CC4C(NC(C5CC(C)(C)CO5)=O)C4C3)=O)cc2o1 28755,C12CC(O)C1NC2=O.O=C1CC(CC(=O)NCCC(=O)N2CCCC2)C1 28756,c1(C(N2CCCCC(NC(=O)C=CC3CCOCC3)C2)=O)csc2ccccc12 28757,N1(C(CC2CC(C)C2)=O)CCC(C)(NC(c2cccc(N3CCOC3=O)c2)=O)C1 28758,CC(C)CS(=O)(=O)CC(=O)N1CC(O)CC1CNC(c1ccccc1)=O 28759,C(=O)(CCC(N(C)C)C1CC1)NC(C1CCN(C(=O)C(C)(C)Br)CC1)C 28760,CC1(C)CC(CC(N2CC(NC(c3ccc(Cl)o3)=O)C(C)(C)C2)=O)CCO1 28761,N1(C(CCn2cc(-c3c(C(=O)OC)cnnc3)nn2)=O)Cc2nccc(Cl)c2C1 28762,c1(C(=O)NCCN(CCC)C(c2cccc(CF)c2)=O)nn(C)c2c1CCC2 28763,N1(C(CSSC)=O)CCN(c2cc(CNC(=O)CCC(F)F)ccn2)CC1 28764,n1(CCCNC(=O)C(O)Cc2cnc[nH]2)cc2ccccc2n1 28765,c1(OC)ccc(C)c(C(=O)NC2(CCNC(=O)C(C)S(C)(=O)=O)CC2)n1 28766,C12(CNC(C=CC(C)(C)C)=O)CN(C(=O)C=CSc3nc[nH]n3)CC(F)(C1)C2 28767,CC(=O)CCN=C(NCc1cc(Br)ccc1O)NC1CC(C)(C)C1 28768,C1(C(N(CCCNC(C2CCN(C)C2)=O)CC)=O)CC12CC(C)(C)C2 28769,C1(NC(C(CSC)OC)=O)CCN(C(=O)CC2(C#N)CC2)C1(C)C 28770,N1(C(CCN(CCC(C)C)C(c2c(C)nc(O)cc2)=O)=O)CC(C)C12CCOCC2 28771,c1(C(C(C2CCN(C(=O)Nc3c(C)n[nH]c3)C2)F)=O)ccc(C(F)(F)F)cc1 28772,N1(C(c2c(OC)nccc2)C(=O)Nc2ccc(F)cc2)CCCC(C)(O)CC1 28773,CC(Cl)(Cl)C(=O)NCC(C1CCOC1)NC(=O)C=Cc1cc[nH]n1 28774,C1(CNC(C(COCC)C)=O)CN(C(=O)Cc2cccnc2Cl)CC1O 28775,c1(CC)nc(C)c(C(=O)NC2CCC2NC(c2cn(CC(N)=O)nn2)=O)s1 28776,CCCC(C(=O)NCc1nc(C(N2CCC23CCCSC3)=O)co1)C(C)C 28777,c1(C(N2CC(NC(c3cc(C)cc(F)c3)=O)C(C)C2)=O)cc(C#N)ccc1C 28778,c1(CN(CC=C)C)cc(C)c(-c2ccccc2OC)s1 28779,c1(C(=O)OC)ccc(C(=O)NCCCC(C)NC(=O)CC2CCCC2)cn1 28780,C1(NC(CSCC#C)=O)C(CNC(c2cc3ccncc3s2)=O)CCC12CCC2 28781,c1(OCC)ccc(Cl)c(C(=O)NC23CC(C2)N(C(=O)C(C)COC)C3)n1 28782,N1(C(CC=CC(C)(C)C)=O)CC(NC(c2cc(C3CC3)no2)=O)CC(O)C1 28783,C1(C2CCC2)(C(=O)NCC2N(C(=O)Cc3ccccc3F)CC2)CC1(F)F 28784,c1(C(=O)CNC(C2CCC3NCCC3C2)=O)ccc2c(c1)CCOC2 28785,C1(CC)CCN(C(C2C(C)C2C)=O)C(C(=O)NC(C2CC3(CCC3)C2)C)C1 28786,C1(c2nnnn2C(C)(C)C)(NC(C2(CC=C)CCCC2)=O)CCCC2CC12 28787,C(=O)(C(F)C(C)CNC(c1cc(C)cc(O)c1)=O)NC(COC)(C)C 28788,CCC(CCC(=O)NC(C)C(C)F)NC(C1C2(CC2)C12CC2)=O 28789,Cc1cc(F)cc(C)c1C(=O)NCC(C)CNC(C1CN2CCN1C(C)C2)=O 28790,C=CCCCCCN(C(=O)CC1CCCN1C(=O)C(O)C1CCC1)C 28791,C(CCCCC(=O)N(CCCCN(C)C(C1CCCN(C(C)C)C1)=O)C)OC 28792,C1(NC(CCS(C)=O)=O)CCC2(CCN(C(C3(CCOCCO)CC3)=O)C2)C1 28793,C1(C(=O)NCC(=O)OC(C)C)CC2(CCN1C(=O)C(C)N=[N+]=[N-])CC2 28794,C1(O)(CC(=O)NC2(CF)CCN(C(c3c(C(C)C)ocn3)=O)C2)COC(C)(C)C1 28795,O=C(C1=CCCO1)N(C1CCCC1)CCCNC(=O)C(F)(F)c1ccccc1 28796,N1(C(C(C2CCC2)OCC)=O)CC(C)(C)CC1C(=O)NCC1(C)CNC(=O)O1 28797,N1(C(CCc2n(C)ccn2)=O)C(CNC(=O)CO)CC2CCCC12 28798,c1(C(C(=O)NC2CN(C(C3C(OCC)C3)=O)C2)C)cccc(Cl)c1 28799,C1(NC(C(C)=C(C)C)=O)CCC(N(C)C(c2cc(-c3ccccc3)[nH]n2)=O)CC1 28800,c1(NC(C2C(NC(C3CN(C)C3)=O)CCC2)=O)cc(C(F)F)cnc1Br 28801,C(=O)(CCCCCNC(N)=O)N(CC(CNC(CN(C(C)=O)C)=O)O)C 28802,c1(-c2c(OC)ccc(C(C)C)c2)cncc2sc(C(=O)Nc3conc3C)cc12 28803,c1(O)c(C(=O)CC)cccc1Br.C1(CNCC)CN(C(C2(C(N)=O)CC2)=O)C1 28804,C1(NCC=O)CCC(O)CN1CC(c1sccc1C#N)=O.CCCCSCC 28805,C(=O)(N=c1[nH]nc(-c2ccc(F)cc2)s1)NC1CN(CC)C1 28806,C(CCC(C(=O)Nc1ccc(C)nc1C)NC(c1ccc(O)nn1)=O)OC 28807,C12(NC(C(C)Sc3ncccn3)=O)CCCCCC1N(C(=O)CC(C)(F)F)CC2 28808,N1(c2nnc(C#N)s2)CCC2(NC(c3ncc(Cl)s3)=O)CCCC12 28809,Cc1cc(C(N2CC3CC(CNC(c4cnco4)=O)C3C2)=O)n2nccc2n1 28810,c1(N2CCC(CNC(=O)NC)CC2)nc(Cl)c(C)nc1C#N 28811,N1(C(C2CC(C)CN2c2nccc(-c3ccccc3)n2)=O)CC2CCCCC2C1 28812,C1(C(=O)NCCCOCCCNC(COCCOC)=O)(CF)CC=CCC1 28813,C(C(=O)NCC1CCC(F)(F)C1)(C(C)CC)NC(C=CCCC)=O 28814,C1(N(C2CC3CNC2C3)C(=O)NC2(c3ccc(Cl)cc3)CC2)CC12CCOCC2 28815,N1(C(CC=CC)=O)CCC2CCCC12CNC(=O)CCc1ccc(CC)cc1 28816,C1(C(N2CCC(N(C(C3(c4cc[nH]n4)CCC3)=O)CC)C2)=O)CC(C)(C)CN1C 28817,C1(NC(C(C)N(CCC)C(c2cc(O)cs2)=O)=O)CCC2CCC12 28818,N1(C(C2CC(SC)C2)=O)CCC2CN(C(c3cnc4ccccn34)=O)C2C1 28819,c1(C(=O)NCCC2CC(NC(C3CCC3)=O)C2)cnoc1-c1ccccc1 28820,c1(C(=O)NC2(CN(C)C(C3CC(C(F)(F)F)CO3)=O)CC2)ccnc2c1ccn2C 28821,c1(C(C)NC(=O)CC(Cc2cccs2)Nc2cn[nH]c2)cccc(F)c1I 28822,C1(CC=C)(NC(=O)CS(=O)(=O)CCO)CC2CCC(C1)N2C(=O)C(C)CF 28823,C1(OCC)CC(NC(C2CC23CCC(F)(F)CC3)=O)C12CCCCC2 28824,C(=O)(C1=CC2(CCOCC2)C1)NCC(C)(C)CNC(C1CC1c1ccccc1)=O 28825,N1(C(=O)Nc2c(C(=O)OC)cc(OC)cc2)CCN(C)CC(C)C1 28826,N1(C(CC(=O)N(C)C)=O)CC(CNC(=O)C(=Cc2c[nH]cn2)F)CC12CCC2 28827,C1(O)(CNC(c2c(CC)c[nH]n2)=O)CCCN(C(C2CC(O)(CC)C2)=O)C1 28828,CCCCC(C(=O)N1CCC2CCC12CNC(C12CC(C)(CCO1)C2)=O)N(C)C 28829,c1(C(=O)NC2C3(CC(NC(CCC(=O)NC)=O)C3)C2)oc2ccccc2c1Cl 28830,c1(OC)nn(C)cc1C(N1CC(CNC(=O)Cn2nc(C)oc2=O)CC1C)=O 28831,C#CCC(C(=O)N1CCCC(CN(C)C(c2cnn(C3CCCC3)c2)=O)C1)C1CC1 28832,C12(C(=O)NC3C(C)(NC(C4C(CC)CCO4)=O)CCC3)CC=CCN1CCC2 28833,N#Cc1cccc(-c2cn(CCCCNC(=O)Cc3nc[nH]n3)nn2)c1 28834,C1(CC(=O)NC(CCCNC(c2c(CC)nco2)=O)C)CCC(F)(F)CC1 28835,C(=O)(CC(CC)C(C)(C)C)N1CCC(CNC(C(C(CC)C)C)=O)CC1 28836,C(=O)(C1CCCc2nn(C)cc21)NCC(C)NC(=O)CCc1c(F)cccc1Cl 28837,C1(F)(C(N2CCN(CCCCCNC(C=CCC)=O)CC2)=O)C2CCCCC12 28838,Cc1cc(C(=O)NC2CN(C(=O)C(=O)N(C)CC3(N(C)C)CC3)C2)cc(OC)n1 28839,c1(C(C(=O)N(C(C)C2CC2)CC2(C(=O)N(C)C)CC2)C)cn(C)c2ccccc12 28840,N1(C(C(C)OC2CCCC2)=O)CCC(C(N2CC3CCC(C2)N3C)=O)C12CCC2 28841,Cc1ccnnc1C(=O)NCCCOCCN(C(=O)C#CC(=O)N(C)C)C 28842,N1(C(C(C2CC2)NC(CC=C(C)C)=O)=O)CC2(CCCCC2)C1 28843,C(CNC(c1ncsc1C(F)(F)F)=O)(C(C)C)NC(C1CC(C(=O)OC)C1)=O 28844,C1(C(=O)Nc2cc(CCC)n[nH]2)COCC1(C)C 28845,CC1CCN(C(c2ccc(Cl)cc2N)=O)CC1NC(=O)CSc1ccccc1 28846,C=CC1(NC(=O)NCCN(C)CCOC)CCC1 28847,C12(CNC(CCCC=C)=O)CCC(CN(C(=O)C=CC=Cc3ccccc3)C1)C2 28848,N1(C2CCN(CC(=C)F)CC2)CCN(C(c2ccc(O)cc2)=O)C(=O)C1 28849,C=CCC(CC)C(=O)NCC1CN(C)CCN1C(=O)CCCC(N)=O 28850,N1(C(CCCCC=CC)=O)CCC2(CCN(C(C3CCOC(C)C3)=O)CC2)C1 28851,C(CC(=O)Nc1cnn(CCO)c1)(C(C)CC)NC(c1cc(SC)oc1)=O 28852,N1(C(c2cn(C)nc2)=O)CC2CC(NC(C3CC4(CCCO4)C3)=O)C1C2 28853,Cc1nccc(C(=O)NC2C3CN(C(c4c(Cl)noc4C)=O)CC23)c1O 28854,C#CCC(C(=O)NCC)NC(C12CC1CCN2C(c1cc(C2CC2)on1)=O)=O 28855,CC1=NOC(=O)C1CC(=O)NCC1(CNC(C2(O)CC(F)(F)C2)=O)CC1 28856,N1(C(C(C2CCCO2)NC(c2cc(CC)n(C)n2)=O)=O)CC2CC1CN2CC 28857,C(=O)(C#CC1CCOCC1)N(C(C(N1CC(C)C1)C)=O)CCC1CCCCC1 28858,c1(C(N2CC(C(C)NC(c3ccc[nH]3)=O)C2)C(N)=O)ccc(Br)cc1 28859,N1(C(C(N2CCCC(O)C2)C)=O)C2CCCC1CN(C(c1ccno1)=O)C2 28860,C1(NC(Cn2c(=N)nc[nH]2)=O)CN(C(=O)CC2CC(F)C2)CC1c1ccccc1F 28861,c1(C(N(C2CCCC2)CCNC(=O)CC2CC(F)C2)=O)ccc(CO)cc1 28862,N1(C(c2ncc(Br)cc2C)C(=O)NCCCSCC)CCC2(CO)CCCC12 28863,c1(NC(c2n(CCC)nnn2)c2ccc(Cl)s2)ccc(-c2nnco2)cc1OC 28864,Cc1cccc(C(=O)NCCN(C(=O)C2=CCCC2C)C2CCCCC2)c1N 28865,c1(C(=O)NC(C#C)C2CC2)cccc(CNC(C2CC3(CC3)CO2)=O)n1 28866,N1(C(c2cc(COC)sc2)=O)CCC(N(C(=O)Cc2cc(C)no2)C)C(C)C1 28867,C1(C(=O)NC(C2(CNC(C3COCCOC3)=O)CC2)C)CCC=CCC1 28868,C=C(C)CC(C(=O)N1CC(OCCF)C1)NC(=O)Cc1nocc1C 28869,C(=O)(CC(CC)C1CCC1)NC1N(C(C(=O)NCCOCCCC)=O)CC1 28870,C1(C(N2CCCC(c3nncs3)C2)=O)CC2CCCCC2O1 28871,CN1CCC(O)(CNC(c2cc(CNC(C3(C)CC3(C)C)=O)cs2)=O)C1 28872,N1(C(CC2(C)CCCC2)=O)CCC(C)(C)C(NC(C2COCCO2)=O)C1 28873,C1(C)CN(NC(CCn2c(C)ccc2C)=O)CCCO1.C1(CN)CC[Si](C)(C)C1 28874,C(N=c1[nH]c(=NCC2=CCOCC2)[nH]c2c1CCC2)c1ccc(OC)cc1 28875,c1(C(=O)NC2C(CNC(C3N(CC)CCC3)=O)C2)sc(Br)c(C)c1C 28876,Cc1cnc(NCC2(C)CCN(C(=O)CCC(C)(C)C)C2)c([N+](=O)[O-])c1 28877,c1(C(C)NC(C2COCCN2C(c2cc(Cl)ncn2)=O)=O)ccc(Cl)cc1Cl 28878,C1(N(C(=O)Cc2cn(C)cn2)CC)CCCN(C(c2cnn(C)c2Cl)=O)C1 28879,N1(CCOC)CC(NC(=O)NCC(Cl)Cl)C(C)C1 28880,c1(OC)ccc(C(=O)NC(C)CC2CN(C(=O)CCCc3ncco3)C2)nc1 28881,C1(CNC(COCCOC)=O)CC(C)N(C(C2CCC(F)(F)C2)=O)C1 28882,C1(C(=O)NC2C(CNC(CCCC(N)=O)=O)C2)C2C3CC4C1C1C2CC3C41 28883,c1(SCC)ccccc1CC(=O)NCC1CCN(C(=O)CC2CC3(CC3)C2)CC1 28884,CC1(C)CCC(C(N2CCOCC2CCNC(C2COCCN2C=O)=O)=O)CC1 28885,C(=O)(CCCC(C)(C)C)N(CCC(=O)NCCC(O)C(C)C)CC=C 28886,N1(C(c2nc(CC(C)C)sc2)=O)CC2CC(NC(=O)CCN3CCCC3=O)C2C1 28887,N1(C(C2(C#N)CCCO2)=O)CCCC2(C1)CN(C(c1ccc3cnnn3c1)=O)C2 28888,C(=O)(CCC(C)(F)F)NCC(CNC(c1cccc(OCCOC)c1)=O)OC 28889,CCC(C(=O)NCC1(OC)CN(C(=O)CC(C)F)C1)N(C)C 28890,Cc1sc(NC(=O)C(C)(C)C)c(NC(=O)CCCN(C)C)c1C.C12CC1NC2=O 28891,c1(-c2cn(CC(CNC(=O)C(c3cncnc3)C)OC)nn2)cc(C)ccn1 28892,C=Cc1ccc(C(=O)NC2CCC(CNC(c3ccc(CC)s3)=O)C2)cc1 28893,CN1CCCC(F)(C(=O)NC(C)CCN(C(=O)CCCc2cccnc2)C)C1 28894,c1(-c2ccc(C(C)(C)C)[nH]2)nc(Cc2cccc(F)c2)nn1CC(F)F 28895,Cc1cc(C(=O)NCCCN(CCCCNC(C2CC=CCO2)=O)C)sc1C 28896,C1(N(C(CS(=O)(=O)NC)=O)C)CN(C(C2CC(F)(F)C2)=O)CCC1O 28897,C1(C(=O)NC2(CC=C)CCN(C(c3ccnn3CC)=O)C2)CC(C2CCCC2)C1 28898,c1(CC)nccn1C(C)CC(=O)N(C)CC1(NC(=O)CCc2ccccn2)CC1 28899,c1(C(=O)NC2(C(C=CC(N3CC(CC(C#C)C)C3)=O)OC)CCC2)ccc(F)s1 28900,c1(C(N(CCCN(C)C(C2CSCCS2)=O)C)=O)ccc(-n2cccn2)nc1 28901,N1(C(Cc2cncc(OC)c2)=O)CCC(NC(=O)CCc2nc[nH]n2)C(O)C1 28902,C1(n2ncc(C(N(C3CCCN(C(=O)C(C)(F)F)C3)CC)=O)c2)CCC(C)CC1 28903,c1(CC)ccc(C(C)=CC(=O)NC2CCN(C(C3COC(C)(C)CO3)=O)C2)cc1 28904,C(=O)(C1=CCCN(C(C2CCC3CC23)=O)C1)NC1(C(C)C)CC1 28905,CCC(CC(C)CO)NC(c1cnc(OC(F)(F)F)cc1)c1nnnn1C(C)C 28906,C=C(Cl)C(C)(C)C(=O)N1CC(O)(CCNC(C2CC23CC(C(F)(F)F)C3)=O)C1 28907,O=C(C1=CCS(=O)(=O)C1)N1CCC2(C1)CN(C(c1cc(F)cc(F)c1)=O)C2 28908,C1(NC(C(n2cc(Cl)cn2)C)=O)CCCN(CCOc2ccccn2)CC1 28909,Cc1ccc(F)c(C(N2CC(NC(c3cc(Cl)ncc3Br)=O)C(F)C2)=O)c1 28910,C(CCS(C)=O)(C(=O)N1CCC(CCNC(c2ccc(Cl)c(F)c2)=O)C1)N(C)C 28911,C(=O)(C1=CCC(C)CC1)NC1C(SC)CN(C(C23CCCC2C3(F)F)=O)C1 28912,C(=O)(CCCCC(=O)Oc1ccc(Br)c(C)c1)C1CC(OC)C1(C)C 28913,C1(COC)(NC(c2ccccn2)=O)CCN(C(c2ccc(C(N)=O)[nH]2)=O)CC1 28914,c1(SCCC(=O)NC2CC(NC(CCN(CCC)C)=O)C2)ncnc2[nH]cnc12 28915,C1(NC(C2CC(OCC)C2)=O)CCC2(CCN(C(C3(C)CC(C)(C)C3)=O)C2)C1 28916,C1(CNC(CCc2c(C)noc2Cl)=O)CC(O)CCN1C(=O)Cc1cncn1C 28917,N1(C(c2c(C)nn(CC(F)F)c2)=O)CCN(C(C2C3CCC(=O)C23)=O)CC1C 28918,CC(CNC(=O)C(C)NC(c1cc(=N)[nH][nH]1)=O)CCCO 28919,C1(CC(=O)NCc2c(C)nccc2)C2CCCC2N1C(=O)C(C#N)C(C)C 28920,c1(CN)ncc(CCNC(=O)C(=O)N2CC(O)C2)s1 28921,C(c1cccc(F)c1Cl)=CC(=O)NCCC1(CNC(CCN(C)CCO)=O)CC1 28922,c1(C(=O)NCCCN(C(C(C2CCC2)OC)=O)C2CCOC2)ccccc1 28923,c1(C(N2CC(c3c(CNC(c4ccon4)=O)nco3)C2)=O)cccc(C(F)F)n1 28924,C1(CC(=O)NCc2c(C(N(CC(F)Cl)C)=O)c[nH]n2)CC2(CCC2)CO1 28925,c1(C(Nn2c(SC)nnc2-c2cc(C)cc(C)c2)=O)cc2c(cc1Br)CCC2 28926,CC1CN(C(=O)CCC(=O)c2cccc(F)c2)CC1NC(C1CC1C)=O 28927,c1(NC(=O)CCNCc2ccc(Cl)o2)ccc(Cl)cc1F 28928,CC(C)CC(CCO)NC(C1OCCC1CNC(c1ccn(C2CC2)n1)=O)=O 28929,c1(C(=O)OC)cc(C)cnc1NCC1CCCN1OC(C1CC(=O)N(OC)C1)=O 28930,Nc1cc(C(=O)NC2CC3(C2)CN(C(C2CC24CCC4)=O)C3)c(F)c(F)c1F 28931,c1(SCC)cccc(C(=O)N(CCCNC(=O)CCSC)CCO)n1 28932,N1(CCSC)C(=O)NC(c2csc(C#N)c2)C2=C1CN(c1ccc(Cl)cc1)C2=O 28933,S(=O)(=O)(c1ccc(N2CCCCC(OC3CCCC3)C2)cc1Br)NC1(C)CSC1 28934,C#Cc1ccc(Cl)c(C(=O)NC2CCCC(NC(c3cnsc3C)=O)C2)c1 28935,c1(OC)ccccc1C(C)NCCN(C)C.N1CCN(C(=O)C=CC=O)CC1C 28936,C1(CNC(C2CCC(C)C2)=O)CCCN(Cc2nnn(C)n2)C1 28937,c1(NCc2c(-c3c(F)cccc3)nccc2)cccc2c(Br)cccc12 28938,C1(OC)(OC)CCOCC1NC(C1CCCN(C(c2cc(Cl)c(C)cn2)=O)C1)=O 28939,C(N=c1[nH]c(=NCC2CN(C3CCC3)C2)[nH]c2ccsc12)c1c(C)cccc1Cl 28940,c1(NCCSNC(C(C)(C)C2CC2)=O)cccc(-n2cc(C3CC3CO)nn2)c1 28941,N1(C(Cc2c(OC)nccc2)=O)CC2CC(NC(C3CCC3C(F)F)=O)CC1C2 28942,C(=O)(C1CCCc2nncn21)N1CC2CN(C(CN(C)C3CC3)=O)C2CC1 28943,N1(C(C2N(C)CCC2)=O)CCN(C(=O)C(O)C2CC2)C(CO)C1 28944,c1(C(C)C)ccc(-n2nc(COc3ccccc3)nc2C2CC2F)cc1 28945,c1(C(=O)NCC2N(C(C(CCC)(C)C)=O)CCC2)cc(OC)c(N)c([N+](=O)[O-])c1 28946,C(N=c1nc2scnc2c(N2CCOCC(F)(F)C2)[nH]1)c1n(C)nnn1 28947,C1(C(=O)NCC2(C)CCCO2)(NC(C(CC2CCC2)OC)=O)CCCCC1 28948,c1(NC(=O)NCCc2c(SCC)cccc2)c(C)nn(C)c1-n1ccc(C)n1 28949,c1(C(N2C(C)CC(CNC(=O)CC3CCOCC3)C2)=O)cncc(C#N)c1 28950,c1(C(N2CCC(NC(C(CCC)OCC)=O)C2(C)C)=O)cc(F)cc(Cl)c1N 28951,c1(C(=O)NCC2(F)CN(C(=O)C=C3CCC3)C2)cc2cccc(Br)n2c1 28952,c1(C(=O)NCC(CC)NC(=O)CCc2scnc2C)cccc(C#CC2CC2)c1 28953,C(c1nc2cc(Br)cnc2s1)=C(C)C(C)C 28954,CC1(CNC(c2ccc(CNC(c3cccc(F)c3F)=O)o2)=O)CCCCC1O 28955,c1(CC(N2C(CNC(C3(C)CCOC3)=O)CCCC2)=O)ccccc1[N+](=O)[O-] 28956,C(=O)(C1=C(Cl)CCOC1)N1CCC(C(N2CC(CC)NC(=O)C2)=O)C1 28957,C(CN=c1nc(N2CCS(=O)C(C)(C)CC2)c2c([nH]1)CCS2)SCC 28958,N1(C(c2ccc(CNC(CC(C)SC)=O)o2)=O)CCCC2OCCC12 28959,c1(C(=O)NC(CNC(C2OCC(C)OC2)=O)C)cn2cccnc2n1 28960,N1(C(C(C)Oc2ccccc2)=O)CC2CC2(NC(c2ccn(C3CCC3)n2)=O)C1 28961,c1(CC)ccc(F)c(C(N2CC3CCOC3(CNC(=O)C(=O)N(C)C)C2)=O)c1F 28962,n1(CCC(N2C(CNC(C(C)OC)=O)CCC2)=O)ccc2ccccc12 28963,C1(C(=O)NC2CN(C(C=C(C)C(C)C)=O)C3C2C3)(CF)CCC(F)(F)CC1 28964,CCCCC(C)CCC(=O)N1CCC1CNC(c1sccc1CC#N)=O 28965,C(=O)(C1=C(C)OCCS1)NCC(CCOC)NC(=O)CC1CCC(C)(C)O1 28966,N1(C(c2ccc(SC(F)F)cc2)=O)CC2CN(C(C3CC3(F)F)=O)CC2C1 28967,N1(C(C2=CC(C)(CC)C2)=O)CC2CC(C1)CN(C(c1cc(Br)c[nH]1)=O)C2 28968,c1(OCC)ccc(C(=O)NCCN(C(=O)C2CC2)C2CC2)c(Cl)c1 28969,N#CC1CCN(C(C2CN(C(=O)CC3CCCOCC3)CC2F)=O)CC1 28970,c1(C(c2n(CCCOC)nnn2)NCCS(C)=O)ccc2ccn(C)c2c1 28971,c1(C(N2CC3C(CN(C(C4CC(C)C4)=O)C)C3C2)=O)ccnc2ncn(C)c12 28972,C(=O)(C1=CCOCC1)NCC(COC)NC(=O)CC1CCN(C)C1=O 28973,CN1N=C(C(=O)Nc2cccnc2C(N2CCCC(NC(N)=O)C2)=O)CCC1=O 28974,c1(C(N2C(CCNC(CS(CC)=O)=O)CSCC2)=O)csc2ncnc(O)c12 28975,c1(SCC)ccc(CN2CCN(C(C)C(=O)Nc3cn[nH]c3)CC2)cc1 28976,c1(OC)nc(C)ccc1C(=O)NCC1(C)CN(C(c2c[nH]nc2F)=O)CCO1 28977,c1(C(N(CC(CNC(C(CC)C(C)C)=O)O)C)=O)cc2c(C)ccc(F)c2[nH]1 28978,c1(SCCC)cccc(C(=O)NCC(C)(C)NC(C2CCOC2=O)=O)c1 28979,CC1CC2CN(C(=O)C(CO)C(F)(F)F)CC2N1C(=O)CCC(=O)C1CC1 28980,c1(CCOC)cc(C(N2CC(O)(C(C)(C)CNC(=O)CC(C)=C(C)C)C2)=O)no1 28981,Cc1noc(C)c1C(C)CC(=O)NCC1(CCNC(C2(C)CNC(=O)C2)=O)CC1 28982,n1(CC)nc(C(N2CCN(C(c3cnc(OC)s3)=O)CC2)=O)c(Br)n1 28983,c1(C(=O)NC2C(SC)CN(C(C3CCCC3(C)C)=O)C2)cc2c(cn1)OCCC2 28984,Cc1cc(C)n(CC(=O)NCCCCNC(=O)CC2CC(C)(C)CO2)n1 28985,c1(OC)cc(C(N2CCC(F)(C(=O)Nc3cccnc3)C2)=O)cnc1OC 28986,c1(C(=O)NCCC2(CNC(C(C)OCC=C)=O)CC2)scnc1C(F)(F)F 28987,CCCC(C)(C)CC(=O)NC1CN(C(=O)Cn2c(C)c(C)sc2=O)C2(CCC2)C1 28988,Cn1cccc(C(=O)NCC2C3CN(C(C4(CCF)CC4)=O)CC23)c1=O 28989,C1(NC(CSS(C)(=O)=O)=O)CCN(C(=O)CCN2CCCC2=O)CC1C(N)=O 28990,c1(COCC)nc(Cl)cc(=NC(C)CCNC(c2cc(C)sc2C)=O)[nH]1 28991,C1(NC(=O)Cc2cccc(Cl)c2)CN(C(=O)C(F)C2CC2)CC2(CCOCC2)C1 28992,C1(C2CCN(C(C3COC(=O)N3)=O)C2)(NC(CC2(C)CC2)=O)CC1 28993,C12(C(=O)NC(CNC(C(CC)Oc3ccccc3)=O)C)CCN(CC1)S(=O)(=O)C2 28994,c1(C(=O)NCC(CN(C(C(CCC)OC)=O)C)O)cc2c(=O)cc[nH]c2s1 28995,N1(C(=O)CCNCc2ccccc2)CCCOCC1c1ccccc1 28996,C1(CC(=O)N(C(CNC(c2n(C(C)C)ccn2)=O)C)C)COCC(C)(C)O1 28997,c1(CNC(C(COC)C)=O)ccccc1CNC(C)=O 28998,C(C(C(=O)N1OC2CCC1C2)NC(c1cccnc1NC)=O)SCC 28999,C1(CC)CCN(C(c2ccc(O)cc2)=O)C1C(=O)Nc1cnsc1 29000,N1(C(C(c2cncnc2)C)=O)CCCC1C(C)(C)CNC(=O)CC1C=CCCC1 29001,C1(NC(COCC=C)=O)CCN(C(c2ccc(OC)cc2N)=O)CC1F 29002,c1(C(=O)NC2CC(F)(CNC(CC3(NC(C)=O)CC3)=O)C2)c(F)cncc1Br 29003,C(=O)(CCCSC(C)(C)C)NCCC1(NC(COC(CC)(C)C)=O)CCC1 29004,Cc1[nH]c(C)c(C(=O)NCCCNC(c2cccc(N(C)C)c2)=O)c1C 29005,c1(C(C)=O)cccc(-c2cc(-c3nccn3CC3(C)CCCCC3)n[nH]2)c1 29006,c1(C(=O)NCC2(O)CCN(C(C3(CC4CC4)CC3)=O)C2)csc2ccc(F)cc12 29007,C1(NC(C(CSC)OC)=O)CC(C(=O)N2CC=CC2(C)CO)=CC1O 29008,c1(C(N2CC(OC)C(NC(=O)C=Cc3cnc[nH]3)C2)=O)sc([N+](=O)[O-])cc1Cl 29009,CC1CCN(C(=O)C=Cc2ccccc2)CC1NC(=O)CC1CC(=O)NC1=O 29010,C1(NC(c2c(CC)nccn2)=O)C(C)CN(C(=O)C2=C(C)CCCC2)CC1C 29011,C1(NC(CN(CC(=O)NC(C)C)C)=O)CCN(C(C2CCS(=O)(=O)N2)=O)CC1 29012,N1(C(C(=O)NCCNC(C)=O)=O)CCN(C(=O)C2=CCCOC2)CC1C 29013,c1(NCC=C(C)C)ccc(C)c(NC(=O)Cn2nccc2N)c1 29014,C1(C(N(CC(C)NC(c2cnc(O)s2)=O)CC)=O)CCC(NC(C)=O)CC1 29015,c1(CCC)ncc(C(=O)NC(C)C(C)(C)NC(C2CC(OC(F)(F)F)C2)=O)s1 29016,CCCCC(O)C(=O)NCC(CC1CC1)C(=O)NC12CCC(CC1)C2 29017,C1(NC(C(F)=C(C)C)=O)CCCCCN(C(C2CN3CCCN2CC3)=O)C1 29018,c1(CC(=O)NC2CC(C)(NC(c3ccno3)=O)C2)ccc(Br)cn1 29019,c1(CC)ccccc1N(C)C.c12nnc(o1)C(=O)N(C)C2 29020,C(CC(C(=O)NC(C(C)(C)O)C1CC1)NC(=O)CCc1ccc(C)o1)=CC 29021,N1(C(C=C(C)C)=O)CCC(C(=O)NCCc2ccnc(O)c2)(CF)C1 29022,Cc1sc(-c2cc[nH]n2)nc1CC(=O)N(CCCC1CCC1)CC1CCCC1 29023,C1(C(=O)NCC#CCNC(c2c(C)occ2)=O)C2CCC1(c1cccs1)C2 29024,C1(CC)CN(C)C(=O)CN1C(=O)CC1(C)CCN1C(C1CCCC(O)C1)=O 29025,N1(C(=O)NC(c2cncc(OC)c2)C)C2COCC1CC(F)C2 29026,C(=O)(C1COc2ccccc21)NCC1(C)CCN(C(c2cc(F)ccc2N)=O)C1 29027,C1(C(N(C2(CC(=O)NC3(COC)CCOC3)CC2)C)=O)CCCC(=O)C1 29028,C1(NC(c2ncc(OC)c(Br)c2)=O)CCCCNC12CCC2 29029,CCCCC(=O)C(=O)NCCCN(C)C(C1CCCC1c1nnc(S)n1C)=O 29030,C=CC(F)(F)C(=O)NCC(CC(=O)N1CCC(CC=CC)CC1)OC 29031,c1(N(C)CC2CCCN(C(C(=Cc3ccco3)C)=O)C2)nc2c(C)cccc2o1 29032,C12(NC(C3CC(CCC)C3)=O)CC(CO)(C1)OC21CN(C(=O)C(C)(C)C(=C)C)C1 29033,C1(CC(=O)NCC=CCNC(C(N(C)C)C2CC2)=O)OCCCO1 29034,c1(NC(CN(C(C2N(CC)CCC2)=O)C)(C)C)nc2cc(Cl)cc(Cl)c2o1 29035,c1(C(=O)NC(C2C(C(=O)NC(C=C)CO)C2)C)nc(=N)cc[nH]1 29036,c1(CC)nc(Cl)nc(N2CCCCC(CNC(C3(CO)CCCO3)=O)C2)c1C#N 29037,C12(C(=O)NC(CCCNC(C3CCN(C(=O)NC)C3)=O)C)C=CC(CC1)C2 29038,C1(NC(C2CC(C#C)(O)C2)=O)CCCC(C(=O)N(C)Cc2occc2C)CC1 29039,CC(C)(F)CCC(=O)NC1CC2(C1)CN(C(=O)CC(=O)NCC(F)(F)F)C2 29040,c1(N(C(c2nccn2C)C)CC)nnc(C2CC2C)n1CC 29041,CCCCC(O)CCC(=O)NC1CC(C)N(C(=O)Cc2cnn(C)c2C)C1 29042,Cc1noc(Cl)c1CC(=O)NC1(C)CCN(C(=O)CCCn2cnc(C#N)n2)C1 29043,c1(C(N2C(C)CC(NC(c3nccn3C)=O)C2)=O)ccccc1S(=O)(=O)C(F)F 29044,C1(NC(C2N(C(C)C)C(=O)CC2)=O)CCCCN(C(=O)C(F)C2CCC2)C1 29045,Cc1cccc(C(N2CCCC2C(=O)NCCCCN2CCCC2)=O)c1Cl 29046,CCCC(CCCNC(=O)C(c1ccc(Br)cc1)O)NC(C1OCCO1)=O 29047,CC1(C(=O)NCc2nocc2C(=O)NC2CC(c3ncc[nH]3)C2)COCCO1 29048,C(=O)(C1=C(Cl)CCC1)NC(CCCCNC(C(CC)(C)C)=O)C 29049,n1(CC(=O)NC(C2CC(NC(C(C)OCC)=O)C2)C)nccc1C 29050,CC(CC(=O)N1CCC(C)(C2CC2)C1)C(C)(C)NC(C1CCC(=O)O1)=O 29051,C1(CNC(c2nc(CC)oc2)=O)CN(C(=O)Cc2ccc(C)o2)CCC1(F)F 29052,CC1CC=C(C(=O)NCc2cncc(C(=O)N(C)Cc3cc[nH]n3)c2)CC1 29053,C(=O)(CC(C)(C)C(=O)NC(C)C(C)NC(=O)C=Cc1cncc(OC)c1)OC 29054,C(CCCCC(=O)NC1CC(CNC(=O)CC2CC(F)C2)C12CCC2)SC 29055,c1(C(C)=O)ccc(CC(=O)NC2CC(C)(NC(C3(C4CCCO4)CC3)=O)C2)cc1 29056,N1(C(=O)OC(C)(C)C)CCC2(C1)CN(N1CCc3nc(Cl)ccc3C1)C2 29057,c1(OC)cc(F)c(NC(=O)NC2CCNCC(C)(C)C2)cc1[N+](=O)[O-] 29058,c1(OC)c(CN2CCCCC2CNC(c2ncccc2O)=O)cccc1Br 29059,C1(CC(=O)NCC2(F)CC(NC(C(C#N)C3CC3)=O)C2)NC(=O)NC1=O 29060,C1(C(=O)NC(C(=O)N(C(CC)CO)C)C)(CF)CC(=O)C1 29061,N1(C(C(c2ccccc2)NC(c2n[nH]cc2Br)=O)=O)CC(C(=O)O)C2(CC2)C1 29062,c1(C(=O)NCCN(CC)Cc2cnn(C(C)C)c2)cc(N)c(Cl)c(O)n1 29063,C(CN=C(NCC(N1CC=CC1)=O)N1CCS(=O)(=O)CC1)N(C(C)=O)CC 29064,c1(C(=O)NC(C2CCN(C(CSCCC)=O)C2)C)cc2c(C)ccc(F)c2o1 29065,C(c1ccco1)=C(C)C(N1CCC(CNC(=O)C(F)=C2CCCC2)C1)=O 29066,CCC(C)(O)C(=O)N1CC(C(C)NC(C2(O)CCC2)=O)C1 29067,N1(C(CC2CN(C)C2)=O)CC(C)(C)OCC1CNC(C1CN2CCC1CC2)=O 29068,C1(C)(CNC(c2c(C)cco2)=O)CCCN1c1nnc(CC(F)(F)F)s1 29069,C(=O)(C#CC1CCOCC1)N1C(C)CC(CC(=O)NCCN2CCOCC2=O)C1 29070,C1(NC(CSCC=C)=O)CC2CC1CN(C(=O)COC1CCOCC1)C2 29071,CC1CN(C(=O)C=Cc2cncc(F)c2)CC1(C)CNC(c1ncncc1F)=O 29072,N1(C(C)=O)CCCC2(C1)CN(C(c1cc3ccc(C)cn3n1)=O)CCO2 29073,Cc1cc(C(=O)N(CCNC(c2cccc(CO)n2)=O)CCOCCO)sc1C 29074,CC1(C)CC2(CC(C(N3CCC(CNC(=O)CCS(N)(=O)=O)C3(C)C)=O)C2)C1 29075,CCCCC(O)CC(=O)N1CC2C(C(=O)NCC(=O)NC(C)C)C2C1 29076,N1(C(c2ccc(COC)o2)=O)CCCCC(CNC(=O)C(CBr)=CC2CC2)C1 29077,C1(C#N)(C(N2CCC(CC(C)NC(C3COCCO3)=O)CC2)=O)CCOCC1 29078,C(=O)(C(C)C(F)(F)F)NCCCC1(NC(Cn2c(CCC)nnc2S)=O)CC1 29079,C1(C(N2CCC(CNC(C3CC4CCC3CC4)=O)C2)=O)CCC2CCC1O2 29080,C(c1cccc([N+](=O)[O-])c1)=CC(=O)NCCC(C)NC(c1ccc(Cl)c(Cl)c1)=O 29081,c1(OC)ccc(NC(C2CCCN2C(C2CCC2)=O)=O)cn1 29082,Cc1c(CC(N2CCCCC2c2cn(-c3cccc(N)c3)nn2)=O)nc(Br)n1C 29083,C#CC1(O)CC(C(=O)NC(c2cnn(C)c2)C(=O)NC2CC(C)(CO)C2)C1 29084,C1(CCC(=O)NCCOCCCNC(CC(C)O)=O)CCC(=O)NC1 29085,Cn1nc(C(=O)NC2CCN(C(C34CC(C)(C3)C4)=O)C2)cc1Br 29086,C1(CNC(C2(Cc3ccccc3)CCOC2)=O)NCC12CCC2 29087,N1(C(c2c(C)occ2)=O)CCC(NC(=O)Cc2sc(O)nc2O)CC1C1CC1 29088,c1(SC)ccc(C(N2CC(C)(NC(C3CC4CC4C3)=O)C2)=O)cc1Br 29089,c1(C(=O)NCCOC2CN(C(C(CCCC)O)=O)C2)ccc(Cl)c(S(N)(=O)=O)c1 29090,n1(CC(=O)N(CC(C(=O)OC)N(C)C)CC)c(C)nc2ccc(Cl)cc2c1=O 29091,c1(CC)ccccc1C(CNC(C1CC1CC)=O)NC(=O)C=C(C)c1ccco1 29092,Cc1nccc(C(N2CC(CNC(=O)CNC3CCCCC3C)C(C)C2)=O)n1 29093,C1(O)(CNC(C(CC2CC2)NC(C(CC=C)C)=O)=O)CCN(C)CC1 29094,c1(C(N2CC3CCN(C(CC(C)C(F)(F)F)=O)C3C2)=O)cnn(C)c1S(N)(=O)=O 29095,C1(CC)(CN2CCCC(c3nccs3)C2)CNC(=O)O1 29096,C1(C)(CC)CC(NC(c2cc(N)c(F)cn2)=O)CN1C(C1CC(=C2CC2)C1)=O 29097,N1(c2nc(=NCCS(C)(=O)=O)[nH]cc2)CCOCC12CCS(=O)(=O)C2 29098,N1(CC(N2CC(C(C)NC(C(CCC)C)=O)C2)=O)C(=O)NC2(CCCC2)C1=O 29099,C1(NC(c2n(C=C)ncc2)=O)CC2CC1CN(C(=O)Cc1cccnc1Cl)C2 29100,N1(C(c2c(C)nccn2)=O)CCN(C(=O)CN2CCCNC2=O)C2(CC2)C1 29101,O=S(=O)(c1cc2sc(=NCCCCO)[nH]c2cc1Cl)NC1C2CCC(F)(F)C12 29102,N1(CC)CCC(CNc2cn(C3CCCC3)nn2)CC1 29103,Cc1cc(S(N)(=O)=O)oc1C(=O)NCC1CCN1C(=O)C(F)CC1CCC1 29104,c1(C(C)OC(=O)C(C)Sc2ccccc2)cccc(OC(F)(F)F)c1 29105,C1(C(=O)NC(C(CC)C)CO)CCN(C(=O)C2=CCCCC2)CC1C 29106,C(=O)(C(CC(C)C)NC)N1C(CNC(=O)C=Cc2cnccc2C)CC(OC)C1 29107,CC1=C(C(=O)N2CC(NC(c3cc(Cl)cn3C)=O)CC2(C)C)CCCC1 29108,c1(N2CCC(CC(=O)Nc3c(SCC)nccn3)C2)ncc2c(Br)cccc2n1 29109,c1(CC)cc(F)ccc1C(=O)NCC1CC1NC(c1nn(CC)cc1Cl)=O 29110,O=C(CCCCF)NCC1CCN(C(=O)CCc2ccsc2)C1 29111,Cc1noc(Cl)c1CC(=O)NC1CCCCC1NC(C1(F)CC=CCC1)=O 29112,c1(C(=O)NCC(C(C)C)NC(=O)CCN(CC(F)(F)F)C)ccc(F)cc1F 29113,Cc1ccn(C)c1C(=O)NCCC1CN(C(C2CC2C(C)(F)F)=O)CCO1 29114,C1(C)(CNC(C(CC)F)=O)COCCN(C(c2ccc(CO)cc2)=O)C1 29115,c1(C(=O)OCC(COC)C(C)C)sc2ncn(CCC(C)C)c(=O)c2c1C 29116,c1(OC)ncnc(C(=O)NCC2(O)CN(C(=O)Cc3ccc(C#N)cc3)C2)c1F 29117,N1(C(CCC=C=C)=O)CCN(C(=O)C(C)(C)COC)CC1C(C)C 29118,c1(C(=O)NC2CC(CNC(c3c(OC)csc3)=O)C2(C)C)ccc(CO)c(Cl)c1 29119,Clc1ccc2c(c1)CCC2NC(c1cnc2sccn12)c1nnnn1CC1CC1 29120,O=C1CCCC2C(C(N3CCCC3Cc3cn(C4CCCC4)nn3)=O)C12 29121,CN1CCCCC1CC(N1CCC(N(C(=O)CC2CNC(=O)C2)CCO)C1)=O 29122,c1(C(N2CC(N(C(CC)=O)C)C2)=O)ccc(C23CCC(C2)OC3)cc1 29123,Cc1nc(S)sc1CC(N1CCC(F)(CNC(c2cncc(F)c2)=O)C1)=O 29124,C1(N(C)CC)CN(C(c2ccc(C3CCC3)cn2)C(=O)NC)CC12CCC2 29125,C1(NC(c2cc(C(C)C)on2)=O)CCCCC1CNC(=O)C(C)CN(C)C 29126,Cn1ccc2cc(-c3nc(-c4ccncc4)nn3CCc3ccccn3)ccc12 29127,c1(C(C)NC(=O)C(=O)NCC(c2cccc(Cl)c2Cl)N)scc2c1OCCO2 29128,c1(C(N2CCCCC(NC(C(CCC)(C)O)=O)C2)=O)c(F)cc(F)cc1F 29129,c1(NC(CN(CCN(C(CCc2cnc(C)s2)=O)C)C)=O)ccccc1C 29130,C12CCCCN1C(=O)c1ccsc1C(=O)N1CCCC1CC2.c1(CC)ccoc1 29131,N1(C(c2c(CC)c[nH]c2)=O)CCOC(CNC(=O)C(C)(CO)OC)C1 29132,CCCCC(C)(F)C(=O)N(CC(C)NC(c1cc(N(C)C)ccn1)=O)C 29133,N1(C(c2c(C)con2)=O)CCC2C(C1)CN2C(C1CCCCC1(F)F)=O 29134,C12CCCCN1C2=O.C1(N(CC)CC)CCN(c2ncc(CNS(C)(=O)=O)s2)C1 29135,N1(C(Cc2c[nH]c(=N)s2)=O)CCCCC1C1(NC(C2CC(=O)N(C3CC3)C2)=O)CC1 29136,C(C(F)(F)C(=O)NCC1(CNC(=O)Cc2cccc(C(C)C)c2)CCC1)OC 29137,c1(C(N2CCC(CNC(C3(C)CC3(F)F)=O)C2)=O)cc2nc(F)ccc2o1 29138,C=CCCC(C(=O)NCCCCC(C)(F)F)NC(=O)CCS(N)(=O)=O 29139,O(C1CCCc2ccc(Br)cc21)C(c1cc(F)c(OCC)c(F)c1)=O 29140,C=C(Cl)CCC(=O)N1CC=CC1C(=O)NCCC1CCCCO1 29141,C(=O)(C1=C(Cl)CCC1)N1C(CCNC(CSCC#C)=O)CCC1 29142,N1(C(c2ccc(OC)c(O)c2)=O)CC2CCC1CN2C(=O)Cc1cc(Cl)cs1 29143,c1(CC(=O)NC2(c3cccs3)C(C)C2)csc(-c2cccnc2)n1 29144,C1(CC(=O)NC(C2CCN(C(=O)C(F)CC3CCOC3)CC2)(C)C)SC(=N)NC1=O 29145,C1(NC(c2c(SC)cn(C)n2)=O)C2COCC1CN(C(C1CCCO1)=O)C2 29146,c1(C(=O)NC(CCNC(C2N(CC)C(=O)CC2)=O)(C)C)ccc2c(c1O)CCC2 29147,C1(CNC(C(C)C2CCCC2)=O)CCCCN1C(=O)C(c1csc(=N)[nH]1)=O 29148,CC(C)C(C(=O)NC1CC(CNC(c2nocc2Cl)=O)C1)N(C)C 29149,n1(CC)nc(C)cc1C(=O)N(C)CC1CCCC1NC(C1(C)CC1C)=O 29150,c1(CCC(=O)N(CC(C)N(C(CCOC)=O)C)C)ccc(Br)cc1 29151,c1(C(N2CC(NC(CC(c3ccccc3F)C)=O)C2)=O)cc2c(s1)CCCCC2 29152,c1(CN2C(C)CCC2C(N2CCC(CN(C)C)C(O)C2)=O)cc(Cl)c(Cl)c(Cl)c1 29153,C1(NC(C2(CNC(C3C(CC(C)C)C3)=O)CCCC2)=O)CCN(C)CC1C 29154,c1(C(=O)NCC(F)CNC(C2CC2F)=O)cc2sc(Br)cc2[nH]1 29155,Cn1c(C(=O)NC2CN(C(=O)CNC(=O)C(C)(C)C)C3CC23)cccc1=O 29156,Cc1nc(O)[nH]c1C(=O)N(C)CC1(O)CCN(C(=O)C(C)Cc2ccnn2C)C1 29157,N1(C(C(C)N(CC)CC)=O)CC2CC(C(N3CC(C(CC)CC)C3)=O)(C2)C1 29158,C1(C(N2CCN(C(=O)Cc3cccnc3)CC2)=O)CC12CCCOC2 29159,c1(C(N2CCC(C(=O)OC)CC2(C)C)=O)cccc2c1CCCC2 29160,C(c1ccc(Cl)cc1F)=CC(=O)NC1CCC(CNC(c2n(CC)ncn2)=O)C1 29161,C(C)(CCC(=O)NCC(c1ccc(OC)cc1)NC(=O)CCOC)OC 29162,c1(C(=O)NCC(CC)NC(C2CC23CCOCC3)=O)ccc(C)c(C(=O)OC)c1 29163,c1(CC(C)NCc2ccc(N3CCC(O)C3)cc2)ccc(SC2CC2)cc1 29164,c1(C(=O)NCC(C)NC(c2nocc2Cl)=O)cncc2c1CCC2 29165,c1(Oc2c(Oc3ccccc3)ccc(C)c2)cc(=NCCS(N)(=O)=O)[nH]c(C)n1 29166,c1(C(N2CC(C(C)NC(CC(COC)C)=O)C2)=O)ccc2c(c1)CCO2 29167,N1(CCC(=O)NC(C2CCCN(C(=O)CCF)C2)C)CCCCC1=O 29168,c1(OC)ccc(C(=O)NCCCCCCNC(C2CCCCN2C)=O)nc1N 29169,Cc1cccc2c1ccn2CC(=O)NC(C)CNC(C1CC(=O)NC(C)C1)=O 29170,C1(CCNC(C2C(CC)C2)=O)COCCN1C(c1ccncc1Cl)=O 29171,Cc1nccn1CCC(N1CCCC1CNC(=O)C=CCO)=O 29172,N1(C(C2C(CC)CCCN2C(=O)Cc2ccnn2C)=O)CC(S(C)(=O)=O)C1 29173,C1(NC(C2(NC(CSCCCC)=O)CCC(C)(C)C2)=O)CC(C2CCCC2)C1 29174,CC1(C(=O)O)CCCNC1.c1(C)cc(-c2ccccc2)n[nH]1 29175,N(C(=NCCS(=O)(=O)C(C)(C)C)NCC1(CF)CC(F)(F)C1)CC1N(C)CCC1 29176,CC1(C)CCC2(CN(c3cc(Cl)ccc3[N+](=O)[O-])CCO2)C1 29177,c1(NC(C2COC(CNC(C3(O)CC(CF)C3)=O)C2)=O)cnc(F)nc1 29178,N1(C(C(C)=CC2CC2)=O)CCCC2CN(C(=O)Cc3cncc(C#N)c3)CCC12 29179,c1(CN(C(c2ncc(Cl)n2C)C(=O)NCCCC)C)noc2ccccc12 29180,C#CCCCC(C)C(=O)NC1CC1NC(=O)CC1CCOCC1 29181,c1(CC(=O)N(CC(C)(C)CO)C(CN(CC)CC)C)cccnc1 29182,c1(CC(=O)NC(C)C(C)N(C)C)csc2ccccc12.c12nc(cs1)CC(=O)N2 29183,Cc1cc2c(C(=O)NC(C)CC(C)NC(c3cnc(O)nc3O)=O)cccc2o1 29184,c1(C(N2C(C(=O)NCCc3c(C)nn(C)c3)CC2)=O)cc(C#N)cn1C 29185,Cc1ccc2c(c1)CC(C(N1CCCCC13CN(C(C1CC1[N+](=O)[O-])=O)C3)=O)S2 29186,C12(CNC(=O)CC3OCCO3)CCCC1CCN2C(=O)Cc1cnc[nH]1 29187,C=CCCCC(=O)NCC(C)(C1CCC1)NC(C1(c2ccccc2)CC1(F)F)=O 29188,C1(NC(C=C(CC)CC)=O)CC12CCN(C(=O)CC1CCCC(C3CC3)O1)CC2 29189,C=Cc1ccc(C(N2CC(O)CC2CC(=O)NCc2ccc(Cl)c(F)c2)=O)cc1 29190,CCCCN=C(NCC(c1ccnn1C)O)NC1CCN(C(=O)CCOC)CC1 29191,c1(C(=O)NCCCCC2CCCN(C(=O)CO)C2)cc(Cl)c2c(c1)OCCCO2 29192,CC(C)CCC(C(=O)NCC1(O)CSC1)NC(=O)C(O)C(C)(C)C 29193,c1(C(c2nn[nH]n2)NC(N2CCc3ncncc3C2)=O)cncc2ccccc12 29194,C#CCC(C(=O)NCC(O)COCC)NC(=O)C(C)NC=O 29195,c1(OCC(=O)OC2CC3CNCC23)ccc(N2CCOC2=O)cc1 29196,N1(C(C=Cc2cn(C)nn2)=O)C2CCC(C2)C1C(=O)NCc1ncn(C)n1 29197,c1(C(N2C3CCC2C(NC(=O)C(F)(F)C(F)(F)F)C3)=O)ccc2nsnc2c1 29198,N1(C(CC2CCC(CC)CC2)=O)CC2CCC1CN2C(c1cc(CO)n(C)n1)=O 29199,N1(C(CNC(=O)NC)=O)CCC(NC(C23CCCC2CCC3)=O)C(C(N)=O)C1 29200,CC(C)(CCC(=O)NCC1CC2CC2N1C(c1nccc2cc[nH]c12)=O)[N+](=O)[O-] 29201,C=C=CC(C)C(=O)N1CC(CC(=O)NCCN2CCCCC2C)C(C)C1 29202,c1(C(=O)NCC(=C)CCNc2cc(=O)n(C)cn2)ccc2c(c1)COCC2 29203,N1(C(C(C)NC(CC)=O)=O)CCC(C(N2CCCC(CC3CC3)C2)=O)C12CCC2 29204,CCS(=O)(=O)c1ccc(F)c(C(=O)N(CCC(C)NC(=O)Cc2ccco2)C)c1 29205,C12(NC(CC#N)=O)CCC(CC1)N(C(=O)Cn1cnc([N+](=O)[O-])n1)C2 29206,C#CCC(C)(C(=O)N(C1CC(COC)C1)C)NC(C1CC(=O)CS1)=O 29207,C1(NC(CCN(CC#C)C(C2CC3(C2)CC32CC2)=O)=O)CCCCCC1(C)C 29208,C(C(C)(O)CCC)NC(C(C)(C)NC(Cc1cnc[nH]1)C(=O)CCN=[N+]=[N-])=O 29209,N1(C(C2C(OC)CC2)=O)CC2C(C(=O)NOCCN3CCCC3)C2C1 29210,c1(C(=O)OC)cc(C(=O)NC(C)CNC(C2(C)CCN(C)C2)=O)cc(C)c1 29211,N1(C(C2C(=C)C2)=O)CCCC1C(C)NC(=O)CCc1nc(-c2ccoc2)no1 29212,c1(C(N2C(C)(CNC(=O)C3=C(Cl)CC3)CCC2)=O)cc(=O)n2ccccc2n1 29213,N1(C(c2cnc(C(C)OC)s2)=O)CCCC(N(C)C(c2c(C)nsc2C)=O)CC1 29214,N1(C(CC(C)(F)F)=O)CC2CC(NC(C3(c4cccs4)CC3)=O)CC2C1 29215,N1(C(CC2CC(C)(C)OCC2)=O)CCC2(CCCN2C(=O)C(O)C2CCC2)C1 29216,c1(C(N2C3(CNC(C4CNC(=O)N4)=O)CC(C2)C3)=O)cn2cc[nH]c(=O)c2n1 29217,S(=O)(=O)(c1c[nH]ccc1=NC1CC2CCCCC12)NCCC#N 29218,C=C(C)CC(C(=O)NCCCCNC(c1ccsc1)=O)NC(C)=O 29219,C1(C)(C(N2CCC(NC(c3ccn(C)c3)=O)C(CO)C2)=O)CC(C2CC2)=NO1 29220,Cc1cccc(Cn2cc(C3CC(NC(C4(CO)CC5CCC4C5)=O)C3)nn2)c1I 29221,Cn1cc(-c2nc(C(N3CC(O)(CCNC(C4CCOC4)=O)C3)=O)co2)cn1 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29240,N1(C(C2CCCN(C(=O)OC)C2)=O)CC2(CCC2NC(=O)C(F)=C(C)C2CC2)C1 29241,C1(CNC(CC(CC)C)=O)CN(C(=O)C(F)(F)c2ccccn2)CCC1C 29242,C(=O)(C(CCc1ccccc1)CC(C)C)N1C(CNC(C(C=C)(C)O)=O)CCCC1 29243,c1(C(N2CC(C#C)C2)=O)sc2ccccc2c1COC 29244,C1(C(N2C(CCNC(C(=Cc3cn[nH]c3)C)=O)CCC2)=O)CCCC2CCCN12 29245,CCN=c1cc(-c2nc(CC3C=CS(=O)(=O)C3)n(CCC(C)(C)C)n2)cc[nH]1 29246,c1(NC(N2CCC3CC(NC(C4CC4(Cl)Cl)=O)C3C2)=O)cccc2ccccc12 29247,C1(NC(=O)Nc2cc(OC)c(C(=O)OC)c(Br)c2)CCC(P(C)(C)=O)C1 29248,C1(O)(CC(=O)NC(C2CCCCC2)CC)CN(C(=O)Cc2nocc2C)C1 29249,c1(C(C)=O)cc(S(=O)(=O)N2CC3CC4CCCN4C3C2)c(F)cc1I 29250,CC1CC(C)N(C(c2cccc(NC(N)=O)c2)=O)CCN1C(=O)C=C1CCCC1 29251,C1(O)(C(C)NC(=O)C(C)P(C)(C)=O)CCN(C(c2cc(CN(C)C)c[nH]2)=O)CC1 29252,N1(C(CCN(C(=O)CN2CC=CC2)CC=C)=O)CC2CCC2(C)C1 29253,N1(C(C#CC(=O)N(C)C)=O)CC2CC(NC(c3cc(CN(C)C)on3)=O)C2C1 29254,N1(C(C(COC)C)=O)Cc2cccn2CC(C(=O)NCc2cncc(F)c2)C1 29255,C1(C)(OCC)CC(NC(=O)Cc2csc(N3CCCCC3)n2)C1(C)C 29256,Cc1ncc(Br)c(N2CCC2C(=O)Nc2ncc(Br)cc2I)n1 29257,CC1CC(=O)NC(C(=O)N(C(C)CNC(c2ccc(CO)cn2)=O)C)C1 29258,C1(NC(CCC#CC)=O)CC(O)CN(C(=O)CCC2CC2(F)F)C1 29259,c1(C(=O)NCCC(C)NC(C2N(C(C)=O)CC(O)C2)=O)ccc(=O)n(C)c1 29260,C(=O)(C1=CCCOC1)NCC1CCC(NC(c2ccc(OC)s2)=O)CC1 29261,c12cccc(n1)NCC2.c1(C(CCCOC)(C)OC)nnnn1C(C)C 29262,c1(CNC(=O)NCC2(C)N=C(C)SC2)cc(C)c(F)cc1Br 29263,c1(C(=O)NCC2CCN(C(C3(C)C(C)(C)C3)=O)C2)ccc(-c2ncnn2N)cc1 29264,N1(C(C(CC)=CCCC)=O)CC2CC(C1)N(C(=O)CCCc1ncco1)C2 29265,N1(C(CC=C)=O)CCCCC1CCC(N1CCC(CCC)(CO)C1)=O 29266,C#Cc1ccc(C(N2CCN(C(C3CCC4CC34)=O)CC2CC(=O)NC)=O)nc1 29267,C(=O)(C(C)CCC(C)(C)C)NC1C2CN(C(c3cc(C)c(O)c(C)c3)=O)CC21 29268,C1(NC(C(C2CCOCC2)OC)=O)CCC(C)N(CC(=O)NC(=O)C(F)(F)F)C1 29269,C12(SC)CC(C(=O)N(C(C(=O)NC3C=CCCC3)C3CC3)C)(C1)C2 29270,c1(C(=O)NCC(CC)NC(=O)C(F)(CC)C(=O)OC)ccnc2nc(C)nn12 29271,c1(N(C(c2csnc2C2CC2)=O)C(N(C)CCN2CCCC2)=O)cc(CO)[nH]n1 29272,CCCC(C(=O)OC)N(CC1CCC(c2ccccc2)C1)Cc1ccc(F)cc1 29273,N1(c2nnc(-c3nn(C)c(Br)c3)n2CCC#N)CC(N=[N+]=[N-])CCC1(C)C 29274,c1(C(=O)NC2C(NC(CN(C(C(C)C)=O)C)=O)CC2)cc(CO)ccc1O 29275,c1(CC)cc(Cl)ccc1Oc1ccccc1.n12cc(nn1)C(C)NC(=O)C2 29276,C1(CNC(c2c(Cl)cn(CCC)n2)=O)CN(C(c2ncc(CC)s2)=O)CCN1C 29277,C(=O)(C(O)CSC)NCCOCC(=O)NCC(=C)Cl 29278,C1(=O)CCCCC(=O)N1.CCCC(C(=O)NCC(C)(C)OCC)NC(N)=O 29279,C12(NC(C(C)OCCC(C)C)=O)COC(C1)C(NC(c1cccc(CO)c1)=O)C2 29280,C1(C(=O)NC(c2nc(C(C)(C)C)no2)CC)CCC(=O)NC1 29281,C1(C(=O)NCC(CO)NC(C2(C#N)CCCC2)=O)(COC)CC=CCC1 29282,C1(NC(=O)CN2CCCCC2)CN(C(=O)C=CC2CCCO2)Cc2nccn2C1 29283,N1(CC(=O)N(C)CC2CCCCN2C(=O)C=CCF)CCCCC(O)C1=O 29284,c1(OC)ncccc1CC(=O)NCC1C2CC1N(C(=O)CN1CCCC1C)C2 29285,N1(C(C2N(C(c3c(CC)nn(C)c3)=O)CCCC2)=O)CCC(O)CC1C1CC1 29286,CC1CCc2[nH]nc(C(=O)NCCC3CCCN3C(=O)C(C)c3cccs3)c2C1 29287,N1(C(Cc2ccc(C(=O)OC)cc2)=O)CC2CCC(CC(=O)O)CC2C1 29288,C(=O)(C(C)N=c1cc[nH]cc1)NCCN(C(COCCCC#C)=O)CC(C)O 29289,c1(OCC(=O)NCC(C(C)C)NC(c2cc(Cl)cn2C)=O)nc(O)nc(O)n1 29290,c1(N2CCC(=CCC)C2)nc(NCC2COCCN2C)c2ncn(C(C)C)c2n1 29291,C1(C(=O)O)CCCC2(CCN(Cc3c(F)cccc3Cl)C2)O1 29292,C1(C(=O)NCCc2nccs2)C2CC3C(C2NC(C2C4COCC24)=O)C13 29293,C(=O)(CCCC(=O)N(CCCCN(C(=O)Cc1ccno1)C)C)OCCC(C)C 29294,Cc1cccc(C2(C(=O)NC3CCCC(CNC(c4cocc4C)=O)C3)CC2)c1 29295,C(=O)(C1=C(CCCOC(C)(C)C)NC(=O)NC1C)OCC.C1C(CO)CN1 29296,c1(C(=O)NC2C(NC(c3[nH]c(=N)sc3)=O)C2)cnc2cccnn12 29297,C1(C(=O)NCCN(C(C(C)OC)=O)Cc2ccccc2)CC2CCC1CC2 29298,c1(C(=O)NC2CCC(NC(CC=C(C)C)=O)CC2)[nH]nc([N+](=O)[O-])c1Cl 29299,N1(C(c2c(C)nns2)=O)C2CCC1CN(C(c1cccc(C(F)F)n1)=O)C2 29300,C1(OCC)CN(C(C2(COC)CCC2)=O)CC1CNC(=O)Cc1nc[nH]n1 29301,c1(C(N2CCCC2C2CCOC2)C(=O)N(C(CC)(C)C)CC)ccc(C)c(C)n1 29302,C(=O)(CCCC(F)(F)Br)NC1CCC(N(C)C(c2cc(C#N)on2)=O)C1 29303,C(C#Cc1cc(Cl)cnc1F)NC(N1CCC(O)(C(C)O)CC1)=O 29304,C1(NC(C(C)OC2COC2)=O)CCC2CN(C(c3ccnn3C)=O)CCC2C1.C 29305,N1(C(C2CCC(C)O2)=O)CC2CCCC1(CNC(c1ccc3c(c1)CCO3)=O)C2 29306,c1(C(=O)NCCCN(C(CCC=CC)=O)CCO)cnc(N2CCOCC2)nc1 29307,c1(C(C)=O)cc(NC(C2CC2C(=O)Nc2ccc(Br)c(F)c2O)=O)cc(C#N)c1 29308,N1(C(CC2(C#N)CCCC2)=O)CCOCC(NC(C2CC3CCCCC23)=O)C1 29309,CC1(C)C2CN(C(C3CC3F)=O)C(C(N3CCCC(O)C3)=O)C12 29310,C#CC1(C(N2CC3(CC(=C)C3)C2)=O)CCN(C(=O)C(CC)C(=O)OC)C1 29311,CCCC(C)CC(C(=O)OC(C)(C)C)N1CCCC1(CC)CC 29312,C1(NC(CC(COC)C)=O)(CO)CCCN(C(=O)CCc2conc2C)C1 29313,c1(C(=O)NCC(C)(C)NC(C2CCCS2)=O)cn(CCN2CCOCC2)nn1 29314,N(C1CC(F)(F)c2cc(Br)ccc21)C(N1CCC(O)(c2cccc(F)c2)C1)=O 29315,c1(SCC(=O)NCC(C)(CO)NC(=O)CCCCCC2CC2)c(F)cccc1F 29316,CCCC(CCNC(=O)C#CCNC(c1c[nH]nc1C(C)C)=O)C1CC1 29317,C1(CC)CCN(C(=O)CCN2CCC2)C1C(=O)Nc1ccnc(C(N)=O)c1 29318,S(=O)(=O)(c1ccc(F)cn1)NC(C=Cc1ccc(OCC)c(OCC)c1)=O 29319,C1(C(=O)NCC(=O)NC)CSCN1C(=O)CCc1ccncn1 29320,c1(C(C(=O)N(CC(=O)NCC2(CN(C)C)CC2)C)O)ccnn1C 29321,c1(C(N2CCC(CCNC(C(C)=CC)=O)CC2C)=O)cccc2c1ccn2C 29322,C1(N2C(=O)C2)CCCN(C(c2cnc(N(CC(C)C)C3CCC3)[nH]2)=O)C1.COCC 29323,n1(C(C)(C)C)ncc(C(=O)NCCN(C2CCCC2)C(=O)COCP(C)(C)=O)c1Cl 29324,C1(C(=O)NCCN(c2ccc(C)cc2)C(=O)C(=O)NCC#N)CCCC(C(C)=O)C1.O 29325,C1(C(=O)NCCC(C)N(C(=O)CCc2ccn(C)c2)C)(C(F)F)CC(=O)C1 29326,CC1CN(C(C)C(=O)NC(C)(C)C)CCC1NC(C1CCC2(CC1)N=N2)=O 29327,c1(CC)ccc(C(=O)NCC2(C)CCCN(C(c3csnn3)=O)C2)c(O)c1 29328,C1(CCC)(NC(=O)COCC(F)F)CCCN(C(=O)CCCn2cncn2)C1 29329,N1(C(c2c(CNC(C(C3CCC3)OCC)=O)n[nH]c2)=O)CCOCC(O)C1 29330,C1(NC(CC(=C2CCCC2)NC(C(C)=CCO)=O)=O)CC2CC1CC2CO 29331,O=S(=O)(c1cnc(N2CCC(F)(CO)C2)c(Cl)c1)NC1CCC2(CC1)CC(O)C2 29332,Cc1c(NC(C2(F)CN(Cc3ccc(Br)s3)C2)=O)cccc1F 29333,c1(CN(C(c2snc(C)n2)C(=O)Nc2ccccc2)C)ccnc(Cl)c1 29334,c1(COC)ccc(CSC)cc1.C1(C)CC(=O)N1.C123CC(C1)(C2)C(=O)N3 29335,N1(C(C(c2ccccc2F)C)=O)CCCC(CO)(NC(c2cccn2C)=O)C1 29336,CC(C)(O)C(F)C(=O)NCCC1CC(F)CN1C(=O)C1CC1 29337,C(C(C(C)(C)C)NC(=O)CCc1nc(C(C)OC)no1)NC(C1C(CC)C1)=O 29338,c1(C2CCN(C(c3sccc3I)=O)C2)ccc(Cl)nc1 29339,c1(SC)nccc(=NC(=O)c2cc3ccc(-c4cnn(C)c4SC)nc3[nH]2)[nH]1 29340,N1(C(C(C)(CO)NC(=O)CC2C=CCCC2)=O)CCOC2(CCC2)CC1 29341,c1(NC(C2CN(S(CC)(=O)=O)C2)=O)cc(-c2ccco2)nn1C 29342,CC1CCN(C(=O)C(F)F)C(C(N2CCCC(C)(O)C2)=O)C1 29343,C1(CNC(COC(C)C)=O)CCN(C(=O)C(C)(C)CC2CCOCC2)CC1C 29344,N1(C(C(C=C)(C)O)=O)CCc2nc(CNC(C3CC(C)CC(C)(C)C3)=O)sc2C1 29345,c1(CC)nn(C)cc1C(N1CCCC(NC(c2cc(C(=O)OC)c[nH]2)=O)C1)=O 29346,CCCCCC(O)C(=O)NC1CC2(C1)CC(NC(=O)CC1CC=CCC1)C2 29347,C(CN=c1ccc(N2CCc3ncncc3C2)n[nH]1)N(C(C)C1CC1)CC 29348,N1(C(CC(C)F)=O)CCN(C(=O)CCc2cccnc2)C(C2CC2)C1 29349,N1(C(=O)COC2CCCC2O)CC2CCCC(C1)N2C(C1CC(F)(F)C1)=O 29350,C(C(CC1CCCC1)C(=O)Nc1ccc(SC)cc1)NC(CC(=O)NCC#C)=O 29351,c1(C(=O)NC(CCCNC(C(Cn2ccc(C)n2)C)=O)(C)C)cnc(N)c(N)c1 29352,c1(C(N2CCN(C(CNC(C(C#C)(C)C)=O)=O)CC2)=O)ccnc2c1nnn2C 29353,CC(C)C(C(C)NC(=O)C(c1ccccc1F)O)NC(c1csnn1)=O 29354,C(N=c1cc(CC2CC2)nc[nH]1)C1CC(NC(C2CC(C)OC2=O)=O)C1 29355,N1(C(c2c(C)c(Br)n(C)n2)=O)CCCC(C2CN(C(=O)CN(C)C(C)C)C2)C1 29356,c1(C(N2CCN(C(c3c(C)nn(C(C)C)c3)=O)C3C2C3)=O)ccc(P(C)(C)=O)o1 29357,c1(CN2CCC3(C(C(=O)NCCc4ccc(F)nc4)C3)C2)cc(Cl)cc(Cl)c1O 29358,c1(CCC(=O)N(C(C)CNC(COC2(C#C)COC2)=O)C2CC2)cccnc1F 29359,C1(CN(C(=O)Cc2cn(C)cn2)C)CCN(C(c2csc(C#N)c2)=O)CC1 29360,C(=O)(CCCCCNC(N)=O)NC(C)CCCCNC(C12CCC(C1)OC2)=O 29361,C1(CC)CC(C(=O)NCCc2ccsc2)CCN1C(c1csc(C)n1)=O 29362,C12(C(N3CC(C4N(C(=O)COCCCF)CCC4)(O)C3)=O)CCC(CC1)C2 29363,N1(C(C(C)=CC)=O)CCN(C(c2nn[nH]c2C(F)(F)F)=O)C2(CCC2)C1 29364,N1(C(CCS(C)=O)=O)CCC2(CC1)CN(C(c1csnc1Br)=O)C2 29365,C1(CNC(C2CC(C(N(CC(C)O)C(C)C)=O)C2)=O)CCCCC(C)(C)C1 29366,Cc1nn(C)c(Cl)c1C(=O)NC1CCCC(NC(c2cc(C(F)F)[nH]n2)=O)CC1 29367,C1(NC(c2ccnc(C)n2)=O)CCCCCN(C(c2ccc(C3CC3)cc2)=O)C1 29368,c1(C(N(C(C)C)Cc2nc(C(F)(F)F)cs2)=O)ccc(F)cc1 29369,c1(C(=O)NCCC2N(C(C(CC=C)C)=O)CCC2)ccc(C)c(OC)c1 29370,C1(NC(C2(C)CCN(C(C(CC)C#N)=O)C2)=O)CC2(C1)CC(C)(C)C2 29371,C(=O)(C1=CCCN(C(C2CC2C(C)(C)C)=O)C1)NC1CN(C)CC1(F)F 29372,C1(NC(N(CC(O)COCc2ccccc2)C)=O)CC12CCCCCC2 29373,N1(C(c2ccc(CO)s2)=O)CC2CC1(C(N1CCC(c3ccon3)C1)=O)C2 29374,C(C(CCC(F)(F)F)NC(c1cnn(C)c1F)=O)OC 29375,C(=O)(C1=NOC(C)(C)C1)NC12CC(NC(Cc3c(C)nc(Cl)cc3)=O)(C1)C2 29376,C(CC(CC)C(=O)NCC1CN(C(=O)CN2CCN(C)C(=O)C2)CC1(C)C)=CC 29377,C1(NC(COCCC(C)C)=O)CCCC1C(=O)N(C)CCC1CN(C)C1 29378,C1(C(N2C(C)(C(=O)OCC)CC2)=O)CCn2c(Br)cnc2C1 29379,c1(N2CC(N(C)C(c3cnn4c3CCCC4)=O)C2)ncnc2cc(I)sc12 29380,C(=O)(C1CCCc2nc[nH]c21)NC(C)(CNC(c1snc(O)c1Cl)=O)C1CC1 29381,CC(C)C(C(F)F)NC(C1CCN(c2cccc(F)c2)CC1)=O 29382,c1(C(N2CCC(C(C)NC(CCSC)=O)CC2)=O)c(C)nn(C(C)C)c1C 29383,N1(C(CC=CCC)=O)CCOC(CNC(c2sc(-c3ncccn3)nc2C)=O)C1 29384,C(=O)(C1=C(C#N)CCC1)N(C1CCCC(NC(=O)C=CC2CC2)C1)C 29385,CCC(CC)(C(=O)NCCC1CN(C(C2(COC)CC2)=O)CC(C)O1)OC 29386,C12(C(=O)NCC#CC(=O)N3CCC(C(F)(F)F)C3)CCCC1CCC2 29387,CC1CN(C(=O)CCCC(=O)N2CCN(C)CC2)CC(C)N1.C1CCN1 29388,C(=O)(CN=c1cc[nH]cc1)NC1CC(NC(c2cc(CC)no2)=O)C12CCC2 29389,C(=O)(CCC(C)(C)C)N1CC(NC(C(CC)C)=O)C(C)C1 29390,C1(C(N2CC(O)(C(CNC(C(C=CC)O)=O)(C)C)C2)=O)COc2ccccc2O1 29391,c1(OC)cc(C(=O)NC2CCCCC2NC(c2ncccc2N)=O)cc(F)c1F 29392,Cc1nc(C)c(C(=O)NCC2CCN(C(=O)C(C)(C)C3CCCCO3)CC2)[nH]1 29393,c1(C(=O)NCC2(C)CN(Cc3cc(F)ccc3Cl)C2)cc(F)ccc1C#N 29394,c1(CC(=O)NC2(CCNC(CCCSC)=O)CC2)ccc(O)c(F)c1 29395,C1(NC(C2CC(CC)(CC)C2)=O)CC2CC1CN(C(=O)CCC1CCC(C)O1)C2 29396,C1(C(=O)NCC2(O)CCCCC2)Cc2nnsc2S1 29397,C12(CNC(c3cc(CC)nn3C)=O)CN(C(=O)C=CC3CC3)CC1CCO2 29398,C1(NC(C2CCOCC2)=O)CS(=O)(=O)C2CN(C(c3ncccc3Cl)=O)CC12 29399,C1(CC)CCN(C(C2CSC2)=O)C1CNC(c1ccc(NC(C)=O)nc1)=O 29400,c1(C(=O)NCC(C)=CC(=O)NCCc2ccccc2C)cc(F)ccc1O 29401,C1(F)(CNC(C2CCN(C(C)=O)C2)=O)CCCN(C(=O)Cn2c(O)nnc2O)C1 29402,N1(C(c2nn[nH]c2Cl)=O)CCN(C(=O)C=CBr)C2CCCCC2C1 29403,C1(CNC(COCCCCC)=O)CC(CO)CO1.C12CC(C1)CNC2=O 29404,O=CN1CCCN(C(=O)CC2CC=CCC2)CC1 29405,C#CC1(O)CCN(C(=O)C(CC(=C)C)NC(c2ccccc2C#N)=O)C1 29406,N1(C(C2(C(=O)NCc3c(COC)nccc3)CC2)=O)CCc2nc(Cl)ccc2C1 29407,c1(C(N2CCC(NC(C(CCC)OC)=O)C2)=O)coc2cc(OC)ccc12 29408,Cc1occc1C(=O)NCC(O)CCNC(=O)CC1(O)CCOC1 29409,CN1C(=O)CCC1CC(N1CCCCC1C(C)(C)CNC(c1csc(Cl)n1)=O)=O 29410,c1(NC(C2C3CN(Cc4ccc(OCC)c(Cl)c4)C2C3)=O)cc(Br)c(Cl)cc1F 29411,O=C(C=C1CCN(CC23CCN(CC2)C3)CC1)N=c1[nH]oc2ncccc12 29412,C1(C)(CNC(C23CC(CC)(C2)C3)=O)CCN(C(=O)CCCCc2ccccc2)C1 29413,c1(C(=O)NC(C(C)(C)C)CNC(=O)Cn2cnc(=N)[nH]2)ccc(S(C)(=O)=O)s1 29414,C1(C(=O)NC(c2ccc(F)cc2Cl)Cc2n(C)ccc2)CCN2CCOCC12 29415,C(=O)(C(CO)C(C)(C)C)NC(CNC(c1ccc(C#C)o1)=O)CC(C)C 29416,C1(CNC(c2c(CC)onc2)=O)CN(C)CCN1C(=O)Cc1ccn(C)c1 29417,CC(C)CCC(=O)NC(C(=O)NCCc1cccc(Cl)n1)C(C)C 29418,c1(C(=O)OC)cc(Br)c(C(=O)O)cc1NC(C1CC1c1ccccc1Cl)=O 29419,C1(CNC(c2c(CC)cccn2)=O)CCN(C(C2CC(C)(C)C2)=O)CC1C 29420,c1(C(=O)NCCOc2ccc(C#N)cc2)c(Br)cc(F)c(F)c1F 29421,c1(C(=O)NCC(C)NC(c2ccc(-c3cscn3)cc2)=O)cc2n(n1)CCOC2 29422,N1(Cc2cccc(SCC)c2)C(=O)CCN(CC2CCCc3sccc32)C1=O 29423,O=S(=O)(c1cc(Br)c(F)cc1F)NCC1CCN(Cc2cncnc2)C1 29424,C(=O)(C(C)CCCC(C)C)N1CC(CCNC(=O)C(C)C2CCOC2)(OC)C1 29425,CONC(=O)C(=O)NCCC1CN(C(=O)CC=C(Cl)Cl)CC1C 29426,C(=O)(C(C)(C)CCC#N)NC(CC)CNC(=O)C(C)Oc1ccc(F)cc1 29427,C1(O)(C(C)C)CCCN(C(=O)CC(O)CNC(C2COCOC2)=O)C1 29428,Cc1coc2ccc(C(=O)NC3CCC3NC(C3CC3C#N)=O)cc12 29429,CCC(CC(=O)N1CCOCC1CNC(=O)C=Cc1nccn1CC)C(F)F 29430,CC(C)(C)C1=NOC(C(=O)NCC2CCN2C(=O)C=C2CCCCC2)C1 29431,C1(N(C(=O)CC2(OC)CN(C(=O)OC(C)(C)C)C2)CC(C)O)(OC)CCNC1=O 29432,C(CC(=O)N1CC(NC(C2(Cl)CC2(F)F)=O)C1)(CC(C)C)NC(=O)OC(C)(C)C 29433,N1(C(c2c(C)nns2)=O)CC2CC(C1)N(C(C1CCN(CCO)C(=O)C1)=O)C2 29434,Cc1cc(C(=O)N(C)C)c[nH]c1=NCc1ccc2c[nH]nc2c1 29435,C1(COC)(NC(c2cc(C(C)C)nn2C)=O)CCN(C(C2(F)CCCC2)=O)C1 29436,c1(NC)ccc(C(=O)C(=O)NCCCCC(C)NC(c2ccc(F)o2)=O)cc1 29437,C(C(F)(C(=O)NCC1CC2CCC(C1)C2)C(C)C)NC(CCC(CC)=O)=O 29438,C=CCCCC(C(=O)NCC(O)COCC1CC1)NC(=O)Cc1ccc(C)nc1 29439,c1(CC)cc(C(N2CCC(N(C(=O)CC3CCCC(O)C3)C)C2)=O)c(C)o1 29440,C(=O)(C1(C)CCn2c(C)nnc21)N1CC(O)(CNC(C(CC)O)=O)C1 29441,C(=O)(C1CCCn2ncnc21)N1C2CN(C(c3nccc(OC)c3C)=O)C(C2)C1 29442,c1(OC)cc(C)c(C(=O)NCC2CC(O)CN2C(C2CCC(=O)N2C)=O)c(C)c1 29443,N1(C(c2[nH]cc(CC)c2)=O)CCN(C(c2sc(C(C)(C)C)nc2C)=O)CC1C 29444,C1(C(=O)NCCCC(C)NC(C=Cc2c(C)cccn2)=O)CCc2ccnn2C1 29445,C1(C(=O)NCCN(C(c2cc(Br)cs2)=O)CC)CCc2nnc(O)cc2C1 29446,Cc1nc(NC(C2C3CN(C(=O)CNC(N)=O)CC23)=O)nc(C)c1Br 29447,C(=O)(C(O)Cc1cnn(C)c1)N(CCCNC(C(c1ccc(Cl)s1)C)=O)CCO 29448,C1(CNCc2ccc(N(C)C)cc2)CCCCN(C(C2COCCO2)=O)C1 29449,c1(C(N(C(CN(C(C(OC)OC)=O)C)C)C)=O)cccc2c(C)c(C)[nH]c12 29450,N12CC(C3CC3C1)C2=O.C(=O)(CCCOC(C)C)NCCCOCCCOC 29451,c1(CCC(N2CCC(N(C(C=NOC)=O)C)C2)=O)ccc([N+](=O)[O-])cc1 29452,N1(C(C23C4C5C6(C)C4C2C6C53)=O)CCC2CN(C(C3CCC34CCC4)=O)CC12 29453,c1(C(COC)N(C)C(c2nnsc2C)=O)ccc(Cl)cc1 29454,c1(OC)c(F)ccc(C(=O)NC2CC(O)CN(C(c3cc(C)c(C)[nH]3)=O)C2)c1F 29455,CC(CCCNC(c1ncoc1C1CCC1)=O)NC(=O)C(N1CCOCC1)C 29456,c1(C(=O)OCC)nc(C(N2CCC(O)(CNC(=O)CC(C)COC)C2)=O)c(C)s1 29457,O(NC(=O)C(CNC(C1(CO)COC1)=O)C(C)(C)C)CC(C(C)(C)C)O 29458,C1(CF)CC1N=c1[nH]c(N2CCCC(c3cccnc3)C2)nc2c1CCC2 29459,NS(=O)(=O)C1(c2cn(CCC(=O)OC(C)(C)C)nn2)CC1.C12COC(=O)N1CC2 29460,c1(CC(=O)N(CCC(=O)NC2CN(C(C)C)C2)CC=C)csnc1C 29461,C#CCC(C(=O)N(CC(C)NC(C1(C(C)(C)O)CC1)=O)C)NC(=O)OC(C)(C)C 29462,C1(F)(CNC(C2CC(OC)C2)=O)CCN(C(c2coc(C3CC3)n2)=O)C1 29463,c1(C(N(CC(C)NC(CC(CC(=O)OC)C)=O)CC)=O)c[nH]c2cccc(F)c12 29464,c1(NC(c2c(O)cn(-c3ccc(OC)cc3)n2)=O)c(Cl)cc(Br)cc1Cl 29465,c1(C(F)(F)F)cc2ccccc2c(=NCC2CCCOCC2)[nH]1 29466,C(=O)(CC1=NN(C)C(=O)C1)N1CCC(C)CC1CNC(C1CNC(=O)O1)=O 29467,C(CC(C(C)(C)C)NC(c1c[nH]c(=N)s1)=O)N(C(C(CSC)OC)=O)C 29468,C1(N(C)C(c2cc(C(C)(C)C)ccn2)=O)CN(C(C2CCNC2=O)=O)CC1(C)C 29469,N1(C(c2ccc(OC)cc2)=O)CC(C)(C(=O)NCC(C)C(C)(C)C)CC1(C)C 29470,C1(NC(CNC(CC)=O)=O)CN(C(=O)CS(N)(=O)=O)CCC1C 29471,C(C(COC)CC(=O)NCC1C(C)CCN1C(=O)CN1CC(C)C1)OC 29472,c1(N2CCCN(CC)CC2)ccc(C(F)(F)F)cc1S(=O)(=O)NC(C)CCCO 29473,Cc1nc(Br)c(Cl)cc1NC(=O)NC(c1ccn(C(C)C)n1)C 29474,N1(C(CN(C)C(C2CCOC2(C)C)=O)=O)CCC2CCN(C)C2C1 29475,C1(C(N2CC(NC(CC=CC=C)=O)(CO)C2)=O)CCCC2(CCC2)O1 29476,C(=O)(CC(C)(C)CC(=O)NCC1CCCN1C(C1CC2(CCC2)C1)=O)OCC 29477,C(CC(C)C)(C(=O)NCC(CC1CC1)C(=O)NC1COCCOC1)OC 29478,CN=c1nc(C(=O)NCC2(CNC(=O)CC(C)P(C)(C)=O)CCCC2)cc(C)[nH]1 29479,C1(CNC(C(CC(C)C)C)=O)CC2CCC(C1)N2C(=O)CCc1nncn1C 29480,C=CCCC(C(=O)NOCC(C)(C)C)NC(=O)CNC(=O)CCCN=[N+]=[N-] 29481,c1(C(=O)NCCC2CC(NC(c3nnc(C)s3)=O)C2)ccc(-n2cccc2)nc1 29482,C1(COC)CC(CNC(=O)CCc2ccc(F)cc2)N(C(=O)CC(C)F)C1 29483,C(N=c1[nH]c(=NCC2CCCC23CCC3)[nH]c2c1CSC2)C1CCC(SC)CC1 29484,c1(-c2n(CCCC)nc(-c3ccoc3)n2)cc2ccsc2s1 29485,c1(CC)ccc(C(=O)NC2COCC2NC(=O)CCc2nnc(O)nc2O)cc1N 29486,N1(C(=O)Cc2ccc(Br)cn2)CC2CCC(C1)C2NCc1c(F)cccc1Cl 29487,N1(C(CCC(C)O)=O)CCC2(CC1)CN(C(c1ns[nH]c1=O)=O)CCO2 29488,c1(C(n2cc(CC3CCCN3C(=O)CC(Cl)Cl)nn2)CC)cccnc1 29489,c1(C(N2CCC(NC(CS(CC)=O)=O)C2C)=O)ccc(Br)cc1OC 29490,N1(C(=O)NC2CCC(F)(F)C2O)CCOc2cccc(CO)c2C1 29491,C1(O)(CC(N2CC(O)(CN(C)C(c3ccc(NC=O)cc3)=O)C2)=O)CCCCC1 29492,N1(C(c2cc(C)no2)=O)CC(NC(=O)Cc2ccc(O)c(F)c2)CC1(C)C 29493,C1(CNC(C2(N(C)C)CC2)=O)COCCN1C(c1ccc(Br)s1)=O 29494,C(C(COC)C(=O)NC(Cc1ccco1)C(=O)NCCC1CC1C)OC 29495,C(C)(CO)(C(=O)N1CC(C)(C)C1C(C)C)NC(c1c(OC)ccs1)=O 29496,N1(C(c2c(C)snc2)=O)CC(C)C(NC(c2ccoc2)=O)C(C)C1 29497,c1(C(=O)NC2(C)CCN(C(c3cc(C)sc3)=O)C2)cc(C)c(F)c(S(C)(=O)=O)c1 29498,C1(C(N(C(C#C)C2CCC2)C)=O)CCCC1CNC(=O)C(O)C1CCC1 29499,CC(C)(C)CCCC(=O)N1CC2(CC(NC(=O)C=CC3CC4(CCC4)C3)CO2)C1 29500,c1(SCC#C)cccc(C(=O)NCC2CC(NC(C3CN(C(N)=O)C3)=O)C2)c1 29501,c1(NC(CN(C(c2ccc(C)s2)C(=O)NCC2CCC2)C)=O)ccc(Cl)cc1F 29502,Cc1ncc(F)c(=NCC2(C)CCN(C(=O)CC3CCC(C)C(C)C3)C2)[nH]1 29503,N(C(=NCC(C)Oc1ccccc1F)NC1CCOCC1)Cc1cnc(C)o1 29504,C1(C(N2CCC(CNC(C(CCC)c3ccccc3)=O)C2)=O)CCC(F)(F)CC1 29505,c1(CC(=O)NC(C)CCNC(=O)CC2(C)OCCO2)ccc(C#N)nc1 29506,C=CCN=C(NCc1nnn(C)c1C(F)F)NCC(CO)CC=C 29507,Cc1ccccc1CC(C)C(=O)NCC(C(C)C)NC(=O)CN(C(=O)C(C)C)C 29508,C1(CNC(C2(N(C)C)CCCC2)=O)C2CC1N(C(C1CCS(=O)CC1)=O)C2 29509,C(c1ccc(C)c(Cl)c1)=CC(=O)N(CCCNC(CSc1ccc(C)cc1)=O)C 29510,c1(N(CC(=O)NCCCNC(C(C2CC2)SC)=O)C)c(C)nc(O)nc1O 29511,C12COCCC1NC(=O)CONC2=O.C1CSCCO1.NC=O 29512,N1(C(c2c(OC)n(C)nc2)=O)CC2CC(NC(C3CCS(=O)(=O)CC3)=O)C(C2)C1 29513,c1(CC(=O)NCC2CCN(C(c3ccoc3Br)=O)C2)c[nH]c2cnccc12 29514,S(=O)(=O)(c1ccc(NC2CC(C3CC3)C2)c(Br)c1)NC1(CC(C)C)CC1 29515,N1(CC)CCC(N(C)C(c2ccc(Cn3cccn3)cc2)=O)C1C1CC1 29516,C1(CNC(C2(SC)CC(O)C2)=O)CCN(C(=O)CCC2CC2(F)F)CC1 29517,n1(C(C)C)ccc(=NC(=O)C2(CNC(=O)CN3CCCCCC3)CCCCC2)[nH]1 29518,Cc1cnc(N2CCSCC2C)c(S(=O)(=O)N2CCOC(C3CCCC3)C2)c1 29519,C1(C)(C(=O)NC(c2ccccc2C)COC)CCCN(C(=O)C(O)C2CCCC2)C1 29520,C(=O)(C1=CCC(NC(c2ccc(C#N)n2C)=O)C1)NC1C(C=C)COC1 29521,C1(C(=O)OC)(C(C)C)CCN(C(=O)OC(C)C)C1C(=O)OC(C)(C)C 29522,C1(CC(=O)N(C2CCCC2)CCNC(C2CN(C(=O)NC)C2)=O)CC(F)(F)C1 29523,Cc1coc(-c2ccccc2)c1C(=O)NC1CC(CNC(C2CC2CF)=O)C1 29524,C(=O)(CCS(N)(=O)=O)N1CC(C(C(=O)NC2C(C)C2(C)C)O)C1 29525,N1(C(C(CC=C)CC)=O)CCC2(CCCN2C(=O)CCCOC(C)C)C1 29526,CCCCC(CNC(C1CCCCO1)=O)NC(c1ccc(OC(C)CC)cc1)=O 29527,c1(OC)ccc2c(c1)NC(=O)C2CC(=O)NC1CCN(C(C2CC(=C3CC3)C2)=O)C1 29528,CC1(C)CN(C(=O)CC2CC(=O)NC2=O)CC1NC(=O)Cc1ccc(O)cn1 29529,C1(CNC(C(C(C)C)CN(C)C)=O)CN(C(c2ccsc2Cl)=O)CCC12CCC2 29530,C1(C(N2CCC(NC(c3c(OC)oc(C)n3)=O)C2)=O)CC(c2cnn(C)c2)=NO1 29531,C1(NC(C2(CCOC)CCCC2)=O)CC(C)N(C(c2ncncc2Cl)=O)C1 29532,C1(C(=O)NCC=C)CC(O)CN1C(c1ccc(-c2ccc(C(F)(F)F)cc2)o1)=O 29533,C(=O)(C1=CS(=O)CCC1)N1CCC(CCN)CC1.C(=O)(CC(C)(C)C)NC(C)C(=O)N 29534,N1(C(=O)COC2(NC(=O)COC3CC=CC3)CCC2)CCSC2CCCCC12 29535,C=C1CC2(C1)CC(C(=O)NCC(CC)NC(=O)C=Cc1cncc(O)c1)C2 29536,C(=O)(CCCN(C(c1cc(Cl)c[nH]1)=O)CC)NC1CN(C(CC)=O)C1 29537,N1(C(C(C)(C)Nc2ccccc2)=O)CCN(C(C2CC(F)(F)C2)=O)CC(O)C1 29538,N1(C(COC)=O)CCC2(CCC2)C(NC(c2csc(S(N)(=O)=O)c2)=O)C1 29539,N1(C(C)=O)CC2CC1CN2C(=O)CN(C1CNC(=O)C1)CC1CCC1 29540,CC(CC(=O)N1CCCC1CN(C(=O)C(C)(C)c1ccns1)C)P(C)(C)=O 29541,N1(C(C2C(=C)CC2)=O)CCC2(CCC2)C(CNC(c2ccc(N)cn2)=O)C1 29542,O=S(=O)(c1ccc2c(c1)CCCO2)NCC1CC(O)C12CCC2 29543,CCC(C)C(C(=O)NCCOCC(=O)NCc1cnc(C)o1)OC 29544,N1(C(c2cnc(C3CCCO3)s2)C(=O)NCCCOC)CCCCC(SCC)C1 29545,c1(C(N2CC3C(N(C)C(C4CCS(=O)(=O)N4)=O)C3C2)=O)cnn(C)c1C#N 29546,N1(C(C2(CC)CC2(F)F)=O)CCCC(N(C(=O)CC2(OC)CCOCC2)C)CC1 29547,Cc1noc(CCC(=O)NCC2CCN(Cc3nc(CC4CC4)no3)C2)n1 29548,N1(C(C2CCC(=C)CC2)=O)CCCC2(CCSCC2)C1 29549,C1(C(=O)NCCC2CCC(NC(c3nc(C)sc3)=O)C2)CCS(=O)(=O)N1 29550,CC1(NC(C2CCC(NC(C3CCCC3F)=O)CC2)=O)CC(F)(F)C1 29551,c1(C(=O)NCC2CCN(C(c3cc(C(C)=O)oc3)=O)C2)cnn(C)c1C 29552,c1(C(=O)NCC(C)NC(c2c(CC)nco2)=O)ccc(OCC(C)C)cc1 29553,c1(C(=O)NCC2C(NC(CC=C(C)C)=O)COC2)cnn2c1C(C)CCC2 29554,c1(C(=O)NC2CC(O)(CNC(CC3CCN(C)C3)=O)C2)cccc(C(F)F)c1Cl 29555,c1(OC)ccc(C(C)=CC(N2CC(OC)CC(NC(C3(O)CCC3)=O)C2)=O)cc1 29556,c1(C(=O)NCCCC(C)NC(CC(=O)NCC)=O)c(C)[nH][nH]c1=N 29557,Cc1ccncc1C=CC(=O)NCC(CC(C)C)NC(c1ccnc(C)c1Cl)=O 29558,C12(NC(CCC#C)=O)CCOCC1CN(C(c1cc3sccc3cn1)=O)C2 29559,c1(N2CC(CCOC)OCC2)nc(NC(c2cccc(F)c2)C)c2ncsc2n1 29560,S(=O)(=O)(CC(C)c1ccccc1)NC(C(C(C)c1ccc(F)cc1)C)=O 29561,c1(C(N2C3(C(N4CCN(CC)CC4)=O)CC3CC2)=O)cc(C)n(C)c1C 29562,C1(C)(CNC(Cc2n(C)nnc2)=O)COCCN(C(C2CCC3CCC2O3)=O)C1 29563,N1(C(C(CNC(CN(C(C(C)C)=O)C)=O)CC2CC2)=O)CCC(O)C(C)(C)C1 29564,Cc1cccc(C)c1CNC(C1CCCN1C(c1cnc(Cl)c(I)c1)=O)=O 29565,C12(CC(N3CCC(N4CC(C)(C)C4=O)CC3)=O)CCC(CC1)OC2 29566,CC1(OCC(=O)NC2(C)CC(F)C2)CN(C(C2(OCCC(O)CO)CCC2)=O)C1 29567,C1(NC(=O)CC2CC=CCC2)CN(C(C2(CC(F)F)CC2)=O)CC12CCC2 29568,C1(C(N(C)CC2(CNC(c3ccn(CCOC)n3)=O)CC2)=O)CC2CC1CO2 29569,CC1CCCCC1(C)CN1CC(n2cc(CCCC3CC(C)(C)OC3=O)nn2)C1 29570,N1(C(c2c(OC)nc(Cl)cc2)=O)CC2CCC1CN2C(c1ccc(CO)cn1)=O 29571,c1(C(N(C2CCCC(NC(=O)CNc3nccs3)C2)C)=O)ccc(O)nn1 29572,C(CCS(N)(=O)=O)NC(C=C(C)CNC(C1CC1(Cl)Cl)=O)=O 29573,C1(OC)(OC)CC(NC(=O)NC2(C(=O)OC(C)(C)C)CC2C)C1 29574,N1(C(c2c(C)cncn2)=O)CCC2(CCC(NC(c3sccc3C)=O)C2)C1 29575,Cc1c[nH]c(CC(N)=O)c1C(=O)NCC1CCC(O)CC1 29576,N1(C(C2(CC)CC2)=O)CCC2(CC1)CCN(c1ncnc3c(C)cccc13)CC2 29577,c1(C(N2C(C)CC(CNC(CCc3cc(C)no3)=O)C2)=O)ccc(N)c(O)c1 29578,C1(C(N2C(C(=O)NCCC3CCCCC3)C=CCC2)=O)CC2CCC(C1)C2 29579,c1(C2(C3CC(OC)C34CC4)CC2)cccc(SC(Cc2cn(C3CC3)nn2)=O)n1 29580,C#CC1CN(C(c2ccc(F)c(OC)c2)C(=O)NC(C)(C)C)CCO1 29581,C1(C(=O)NCC(C)CC2CCCC2)CCCN(C(c2ccc(C(F)F)o2)=O)C1 29582,N1(C(CC=CC=C)=O)CC2CC1CC2NC(=O)C(C)(C)C1CC1 29583,C1(c2scc(C)n2)CCCN(C(C(C)(C(C)C)c2nnnn2CC(F)F)=O)C1 29584,C1(C2(O)CCN(C(C3CCCO3)=O)CC2)(NC(c2[nH]cc(C(C)(C)C)c2)=O)CC1 29585,C#CCCC(C(=O)N1CC(CO)C2(CC2)C1)NC(=O)C(CSC)OC 29586,Cc1ccc(C(O)C(=O)NC2CC(NC(c3cnc(O)n3C)=O)C2)cc1 29587,Cc1nn(CC(N2CC3CCC3(NC(=O)COC3CC3(F)F)C2)=O)c(C)c1Br 29588,CC(C)CC(CNC=O)CC(=O)NC1CC1NC(c1ccc(CCO)cc1)=O 29589,C(=O)(CCCCN1CCCCC1)NCC1(NC(C2CC(OC(C)(C)C)C2)=O)CC1 29590,CCCC(CC(=O)NC1CC(CSC)C1)NC(c1ccc(CO)nc1)=O 29591,C1(C(=O)NC2CC(CCNC(c3c(C#C)cnn3C)=O)C2)CC2(COC(=O)N2)C1 29592,CCS(=O)(=O)CC(=O)NCC(C)(C)NC(C1CCC(C)(CC)C1)=O 29593,CC1CC(CCNC(c2ccoc2)=O)CCN1C(c1ccc(C(N)=O)[nH]1)=O 29594,N1(C(C(C(CC)C)OC)=O)CCCN(C(=O)CCc2cc(C)n(C)n2)CC1CO 29595,C1(CC)(NC(c2cccc(F)c2F)=O)CCN(C(=O)CN2CC(=O)NC2=O)CC1 29596,c1(C(=O)NC2CCC(CNC(=O)Cc3nc[nH]n3)C2)ccc2c(c1F)CCC2 29597,C1(CCNC2(c3n(C4CCC4)nnn3)CCSC2)CC2CCC1O2 29598,c1(OC)ccc(N(C)C(c2ccn(C)c(=O)c2)=O)cc1F 29599,C1(C(=O)NC2(CN(C)C(c3nccn3C)=O)CC2)C2CCC1(c1ccccc1)C2 29600,Cc1ccc2c(c1)C(NCCCC(N)=O)C(C)C2 29601,C1(CCCNC(=O)COc2ccsc2Cl)CCN(C(=O)C(F)CC2CCC2)CC1 29602,N1(C(C(CC=CC)NC(=O)C(C)CC(C)C)=O)CC2(C1)CC(C)(C)C2 29603,N1(C(C(C)CN(C)C(C2CCCOCC2)=O)=O)CCc2sccc2C1 29604,N1(C(c2cccc(C)n2)=O)CCC(NC(C2C3CCC(=O)C23)=O)C(C)C1 29605,N1(C(C(C(C)(C)C)SC)=O)CCC2(CC1)CCN(C(C13CC(C1)C(C)O3)=O)C2 29606,c1(NC(c2n(CCOC)nnn2)C(C)OC)cccc(NS(C)(=O)=O)c1.C(C)(C)(C)N 29607,C(C(CC(C)C)NC(C1(C(F)F)CCOCC1)=O)NC(C1(COC)CC1(F)F)=O 29608,c1(N2C(CC)CCCCC2)ccc2c(n1)CCCC2=O 29609,Cc1sc(O)nc1C(=O)N(CCNC(=O)C#CC(C)C)C1CC1 29610,N1(C(c2c(C)cc[nH]2)=O)CCC(NC(c2ccc(C(=O)N(C)C)cc2)=O)C1(C)C 29611,CC(CC(C)(C)C)C(=O)C1C(=O)C2(CNCC(C(=O)N)N(C)C)C(C1)C2C 29612,N1(C(CC(CC)O)=O)CCC2(CC1)CC2NC(=O)CSc1nnc(C)n1C1CC1 29613,C(=O)(C1=CS(=O)(=O)CCC1)NCC1(C2CC2)CCN(C(c2cnn(C)n2)=O)C1 29614,O(NC(=O)C(Cn1cccn1)NC(=O)Cc1ccn(C(C)C)n1)CCN(C)C 29615,CC1CC1N=c1nc2c(cnn2C)c(N(C)CCSc2ccc(F)cc2)[nH]1 29616,c1(C(N2CCN(C(=O)NC)CC2)=O)cccc(P(C)(C)=O)c1 29617,Cc1ccc(O)cc1C(=O)N(CC(C)CNC(c1ccc(F)o1)=O)C 29618,C1(C(N(C)CC2(CNC(C3CCCN(CC)C3)=O)CC2)=O)CN2CCN1CC2C 29619,Cc1cccc(OCCCC(=O)NCCCCCNC(c2cc(C)[nH]n2)=O)c1 29620,C(CC(N)=O)(C(=O)N1C(CO)CC1C)NC(C1CC(=C)C1)=O 29621,c1(C(=O)NCC(C)N(C(=O)COCc2cccc(O)c2)C)cccnc1C1CC1 29622,n1(CC)nnc(C(=O)NCCCCC(=O)NCC2(F)CCN(C)C2)c1C 29623,C12(C(N3C(CNC(C=CC(CC)=CC)=O)CC3)=O)CCOC1CCOC2 29624,N1(C(CCOCCCOC)=O)CCCCC(CNC(c2ccc(C(C)=O)o2)=O)C1 29625,c1(C(=O)NC(C(C)NC(C2CCCN(C3CC3)C2)=O)CO)cnc2[nH]ncc2c1 29626,c1(CC(=O)NCCC2(NC(=O)CC3CCCCO3)CCC2)cccc(F)c1 29627,C1(CNC(=O)CCC2CC2)CC2(CCC2)CN1c1nc2ccccc2o1 29628,Cc1cncc(CCNc2oc(CNC(c3cnn(C(F)F)c3)=O)nc2C)n1 29629,C(=O)(C(C)(O)C(C)C)CCC.C(CCC(=O)NCC)N(C(=O)CN1CCNC1=O)CCC 29630,C1(NC(c2n(C)ncc2)=O)CC2CCC1(NC(c1cc(C(N)=O)co1)=O)C2 29631,N1(C(C2CC(C(C)=O)C2(C)C)=O)CC2CCC(CNC(=O)Cc3cnoc3)(C2)C1 29632,C1(NC(c2cc(C)no2)=O)CC12CCN(C(=O)Cc1nc(=N)[nH][nH]1)C2 29633,S(=O)(=O)(c1cc(Cl)ccc1Cl)NCC1(F)CCCN(C(C(CC)O)=O)C1 29634,c1(OC)ccc(CC(C)C(=O)NC(C)CCNC(=O)Cc2sccc2C)cc1F 29635,C1(NC(C2CN(CC)C(=O)C2)=O)CC2CCC(C1C)N2C(c1cc(C)c(C)o1)=O 29636,C(C)(C)(CC(F)C(=O)NN(CC(C)C)C)NC(C(COC)COC)=O 29637,C(CC1=CCN(C(C2(C)CCCO2)=O)CC1)NC(C(C(C)C)n1cc(C)nc1)=O 29638,c1(C(=O)NCC2CCCC(NC(=O)CCn3cnnn3)C2)cncc(Cl)c1Cl 29639,N1(CCCS(C)(=N)=O)CC2C3CCC(C2C1)N(Cc1ccccc1)C3 29640,c1(OCC)cccc(CCC(=O)NC(C)C(C(C)C)NC(c2cncnc2)=O)c1 29641,N1(C(C2C(CC(=O)OC)CCCN2)=O)CCCC(c2ccccc2)C1C 29642,C(=O)(C1CCCn2nccc21)N1CCC(Cc2cn(C(C)CO)nn2)CC1 29643,Cc1cc2c(cc1C)C(N(C(c1cc(F)cc(C)c1N)=O)C1CC1)CCCO2 29644,N1(C(c2cc(OCC)n[nH]2)=O)CCC(C(=O)Nc2cccc(Cl)c2)C12CC2 29645,n1(CC(N2CC(C(C(=O)NC3CC(C(C)(C)C)C3)O)C2)=O)cnc(C#N)n1 29646,c1(C(N2CC(CCNC(c3cc(C)c(N)cn3)=O)C2)=O)ccc2c(n1)OCCO2 29647,C(CC(Cc1ccccc1)NC(C1CCC1)=O)NC(c1cnnn1C1CC1)=O 29648,c1(C(N2CC(CCNC(C3CC=C(C)CC3)=O)C(C)C2)=O)cccc2nc[nH]c12 29649,C1(NC(C(F)OC)=O)CN(C(=O)CSCC(F)(F)F)CC2(CC2)C1 29650,C1(C(=O)NCC(CCC)CCO)CC2CC1CN(C(=O)C(C)(C#N)CC)C2 29651,C(=O)(C(CCC(C)C)NC(c1cnn(C)c1Cl)=O)N(C(CCSC)C)C 29652,c1(C(N2CCCN(C(Cc3onc(CC)n3)=O)CC2)=O)cccc2c(N)cccc12 29653,C(c1ccc2ccccc2n1)=CC(=O)N(C)CC1CCN(C(C(C)O)=O)C1 29654,C#CCCCCCC(=O)N1CC2(CC(C(=O)NC3CC(=O)N(C)C3)CO2)C1 29655,c1(C(=O)NC2C(NC(C(C)NC(C)=O)=O)CCC2)cc(CN(C)C)ccn1 29656,Cc1nnc2cnc(C(=O)NC3CC(CNC(c4ccc(Cl)[nH]4)=O)C3)cn12 29657,c1(OC)ccc(S(=O)(=O)N2CCCC(c3ccccc3)C2)cc1.C12CC1C(=O)N2 29658,C1(C(=O)NC2C(C(=O)NC(c3c(C)nns3)C)CC2)CCC(C)CC1 29659,c1(CC)conc1CC(=O)N(C(C)CC(=O)NC1COCC1CN(C)C)C 29660,C(=O)(C(CC1CCC1)NC(c1cc(F)c[nH]1)=O)N(C)CCOCC1CC1 29661,n1(CC(=O)N(CCCCCCNC(C2N(CC)CC2)=O)C)cc(C)c(O)nc1=O 29662,C1(NC(=O)Nc2cc(NC(C)=O)c(OCC)cc2)CN(C(C)=O)C2CCCC12 29663,C(=O)(CCCCC(N)=O)NC(CCCNC(C1CC(C)CC(C)C1)=O)(C)C 29664,c1(CNC(C(C)C#N)=O)cccc(CNC(=O)CC(C2CC2)C2CC2)c1 29665,C1(C2CC2)(NC(C2CCC(NC(Cc3c(C)ccs3)=O)C2)=O)CCCC1 29666,CC1(C)CN(C(=O)Cc2ccccc2CO)CC1NC(=O)CSc1nncs1 29667,Clc1ccccc1Cn1nnnc1N1CCN(CCSc2ccccc2)CC1 29668,C(=O)(CCN=[N+]=[N-])NC1(CCC(=O)NC(c2ncc[nH]2)C)CCCC1 29669,C1(NC(c2nc(C)oc2C)=O)CCN(C(=O)C(F)C(C)C)CC1CO 29670,C1(CNC(c2cc(O)ccc2I)=O)CCN(Cc2c(F)cncc2F)CC1(F)F 29671,c1(C(N(CC(C)C)CC(=O)NCC2CC(=C3CCC3)C2)=O)ncccc1N 29672,N1(C(C(C2CC2)NC(C2CC3CC(=O)C2C3)=O)=O)CC2CC=CCC2C1 29673,CC(CC(=O)NCC1CC12CC2(F)F)C(C)(C)NC(=O)C=C1CCOCC1 29674,C(=O)(C(C)(C)C(F)(F)F)NCCN(C1CCCC1)C(c1c(C)n(C)nc1)=O 29675,CCC(CCC(=O)NOC1CCC1)NC(=O)Cn1ccc(C)n1 29676,Cc1nn(C)c(C(=O)NCC2CN(C(=O)COC(F)F)CCCO2)c1Cl 29677,S(=O)(=O)(c1ccc(Br)cc1NCc1cn2ccsc2n1)N(CCC)CC1CC1 29678,C=CC1OCCC1C(N1CCN(CC2(NC(=O)Cn3ccnc3C)CC2)CC1)=O 29679,c1(C(=O)NCC)ccc(C(c2nnnn2CCSC)NCCc2nncs2)o1 29680,C1(CC2CCCN(CCCn3cc(-c4ccn(C)n4)nn3)C2)COC2(CCC2)C1 29681,c1(C(=O)NCC2N(C(C3=C(C)OCC3)=O)CCOC2)ccc([N+](=O)[O-])c(F)c1 29682,C1(NC(c2nn(CC)c(C3CC3)c2)=O)CCN(C(=O)C(=O)NCC2CCC2)C(C)C1 29683,C=CCC(C(=O)NC1CCCN(C(c2snnc2CC)=O)C1)OC 29684,C(=O)(C(C)(C)C(F)F)N(C)CC1CN(C(C(C)SC)=O)C1 29685,CCC(C)(CNC(C1CC(F)(F)C1)=O)NC(c1snnc1C1CC1)=O 29686,c1(CNC(C2CC(NC(COCCOC)=O)C2(C)C)=O)ccc(O)c(C)c1 29687,c1(C(C)=O)ccc(C(N2CCCC(C)C2)=O)cc1F.C1(=O)C(=O)NCCN1CC 29688,c1(C(=O)NCCCNC(C=CCOC)=O)ccc(S(=O)(=O)CCN(C)C)cc1 29689,C1(COC)CN(C(c2ccc[nH]2)=O)CCN1C(=O)CCc1ccc(O)c(F)c1 29690,N1(C(C2CC(SC)C2)=O)CC2CC(NC(=O)CC3(O)CCCC3)CC(C2)C1 29691,c1(-c2cn(C3CCN(Cc4c(Cl)c[nH]n4)CC3)c(-c3ccccc3)n2)cccc2c1OCO2 29692,c1(OC)ccc(OC(F)(F)F)cc1CN1CCCC1CCC(N1CCCC(C)C1)=O 29693,c1(Nc2c(C)cns2)sc(C)cc1Br 29694,Cc1cc2ccc(C(N3CCC(NC(c4[nH]c(O)nc4C)=O)CC3C)=O)cn2c1 29695,N1(C(C2N=C(C)SC2)=O)CCOCC(CNC(=O)Cc2cccc(N)c2)C1 29696,C1(C(=O)NC(C(N2C(C(=O)NC)C=CC2)=O)CC2CCCC2)C2CCC(F)C12 29697,C(=O)(C(F)CC1CC1)N(CC(C)NC(=O)Cn1ncnn1)CC.O=CC1CC1 29698,c1(C(=O)NC(C(C)NC(c2c(C)cc(F)cn2)=O)CO)cnc2c(c1)COCC2 29699,C1(C(=O)NCCOCCCNC(=O)Cn2cccc2)CC(=O)N(c2cn[nH]c2)C1 29700,c1(C(=O)NCC2(C(N)=O)CN(C(C3(OC)CCC(C)C3)=O)C2)ncc(C)cc1C 29701,c1(CN2CCN(c3cc(C)c(F)cn3)CC2)cc(C(F)(F)F)cc(S(C)(=O)=O)c1 29702,C1(C)(C(=O)NCC2CCN(C(CCCCOC)=O)C2)CC(=O)N(C)C1 29703,c1(C(=O)NCCC2N(C(CNC(C(CC)C)=O)=O)CCC2)nc(C)ccc1F 29704,c1(C(N(C)CCn2cc(CCN3CCSCC3)nn2)=O)snc(Cl)c1Cl 29705,CCCCC(O)C(=O)NCC1C(C)CCN1C(c1cc(Br)n[nH]1)=O 29706,C(=O)(C(C(C)C)NC=O)N(CCCN(C(c1nc(C(C)=O)sc1)=O)C)C 29707,C1(O)(CNC(c2c(C(C)C)occ2)=O)CCCN(C(C2(S(C)(=O)=O)CC2)=O)C1 29708,C(=O)(C(C(C)c1ccccc1)N1CCC2CCC12)NCCCC(=O)OC 29709,CC(C)C(F)(CNC(C1CCCCCN1C)=O)C(=O)NCC1CCC1(F)F 29710,C#CCCC(O)C(=O)NCCOCCNC(C1(C)CCCNC1=O)=O 29711,Cc1cc(C)n(C(C)CC(=O)NC23CC2CN(C(c2sc(F)cc2C)=O)C3)n1 29712,C1(CNC(c2cnn(CC)c2C)=O)CN(C(=O)C(N2CCOCC2)C)CCC1C 29713,N1(C(=O)N(C(c2cnn(C)c2)C(C)C)C)CCOC(C)(C2CC2)C1 29714,c1(-n2c(CC(C=C)C)nc(C3CCCCC3)n2)ccnc2ccccc12 29715,C1(NC(CCC(=O)OC(C)(C)C)=O)CC2CC1CN2C(c1cnc(C(N)=O)s1)=O 29716,CC(O)C(C(=O)NCC1(CO)CC1)NC(C1CC(F)(F)C1)=O 29717,c1(-c2nc(CC)nn2-c2cccc(NC(C)=O)c2)cnn2ccc(O)nc12 29718,N1(C(C2CCn3nccc3C2)=O)CCCC2(CCN(C(C34CC(F)(C3)C4)=O)C2)C1 29719,C=CC1(CC(N2CCC(NC(c3cscc3C)=O)C(CC)C2)=O)CCOCC1 29720,C1(C(=O)NCC2CCCN2c2ncnc3ccccc23)COc2ccccc2O1 29721,CCCCCCC(=O)NCC(C)(C)CN(C)C(C1CCCSC1C)=O 29722,c1(NCC23N(C(=O)OC)CC(C2)OC3)nc2ccccc2nc1C 29723,c1(C(=O)NCCCC2N(C(C(CCCC)O)=O)CCC2)c(C)nc2sc(C)cn12 29724,C(CCC(C)C(=O)NCC12CC(CO1)N(C(=O)CCc1nc(O)n[nH]1)C2)OC 29725,c1(C(=O)NCCNC(C(c2cccc(C)c2)(F)F)=O)ccnc(C)c1C 29726,C1(CNC(CC(C)n2ccnc2)=O)C(C)CCCN1C(=O)CC1(O)CCCOC1 29727,c1(NC(C2CSCCN2C(c2ccc(Br)s2)=O)=O)cccc(O)c1F 29728,c1(CC(N2CCC(N(C(CC3N(C(C)=O)CCC3)=O)C)C2)=O)ccc(C#N)nc1 29729,N1(C(C2(CC)CC2)=O)CCCC2CN(C(=O)C(=O)Nc3ccc(C)cc3)CC12 29730,C(C(CC1CC1)C(=O)NC(C)COC)NC(C(C1CC1)OC)=O 29731,n1(CCCO)nc(-c2ccc(Br)cc2)nc1Cn1nnnc1-c1ccsc1 29732,c1(C(=O)NCC23C(CN(C(C=C(C)C)=O)C2)C3)cc(F)ccc1S(C)(=O)=O 29733,c1(-c2nnc(N3CCCC(C(F)(F)F)(OC)C3)n2C)ccc2c(O)ncnc2c1 29734,CCC(C#N)(CC)C(=O)NCC(O)CNC(C1(OC)CC1)=O 29735,C(=O)(CCCCCCNC(C1CCOC1(C)C)=O)NCC(C(C)O)C 29736,c1(C(=O)NCC(CC)NC(C2(O)CCCCC2)=O)cn(C)nc1C(C)(F)F 29737,N1(C(C2CC(NC(CCC3(C#N)CCC3)=O)C23CCC3)=O)CCOC2COCC12 29738,C1(COC)(CNC(c2csc(C)c2N)=O)CCN(C(=O)C(C)c2ccsc2)CC1 29739,N1(C(C(C)C2CCOC2)=O)CC2(CC(CNC(c3ccnc(Cl)n3)=O)C2)C1 29740,C1(NC(c2c(C(C)(C)C)nc[nH]2)=O)CC2(C1)CC(NC(c1ccc(O)nn1)=O)C2 29741,c1(C(=O)NC2C(NC(C3(C=C)CC3)=O)CCCC2)cc(C)nc(O)c1 29742,N1(C(c2coc(C3CCCC3)n2)=O)CC2C(NC(C3(CF)CC(F)(F)C3)=O)C2C1 29743,C(N=c1cc(CC2CC2)nc[nH]1)C1(NC(CC(C(C)C)O)=O)CCCC1 29744,c1(CNC(C(=O)N(C)Cc2ccc(C#N)cc2)=O)sccc1S(C)(=O)=O 29745,c1(OC)ccnc(C(=O)NCC2CCCCN(C(c3csnc3C)=O)C2)c1F 29746,c1(C(=O)NCC(C)CNC(c2cc3nc[nH]c3cn2)=O)cncc2sccc12 29747,C1(C(N2C(C=C)CC2)=O)(NC(=O)CCOC(C)=O)CCCC1C 29748,CN1CCN(C(=O)CCC2NC(=O)NC2=O)C(CNC(=O)CCc2cnoc2)C1 29749,c1(NC2CCC(C(=O)O)C2)ncc2cccnc2n1.C12(CCCC1)C(=O)N2 29750,N(C(=NCCSc1cccc(OC)c1)N1CCCC2(CC2)C1)C(CC)C 29751,C1(NC(C(n2ncc(C)c2)C)=O)CC(CNC(=O)C=Cc2cnc[nH]2)CC1O 29752,C(=O)(CC(C(=C)C)OCC)NC1(CC=C)CCCCC1.N12CCC(=CCC1=O)CC2 29753,c1(C(=O)OC)ccc(CC(=O)Nc2cccc(CNc3cnc(C)nc3)c2)cn1 29754,C1(C)(C(N2C(C(C)NC(C(c3cccc(C)c3)C)=O)CCC2)=O)C(C)(C)C1(C)C 29755,C1(NC(C=C(C)C(C)C)=O)C2CC1N(C(=O)CC(c1ccccc1)NC(N)=O)C2 29756,C(N=c1[nH]c(N(C)Cc2ccc(Br)o2)nc2c1SCC2)c1c(C)csc1 29757,CCCC(C#N)C(=O)NCC1(F)CC(NC(=O)C(c2cncn2C)O)C1 29758,C(=O)(CC(F)(F)CC)NC(CCC)C(=O)NCCCSCCO 29759,N1(C(c2cc(COC)no2)=O)C(C(=O)NCc2snnc2C)CCC12CC2 29760,c1(OC)n[nH]c(C(=O)N(C)CCNC(c2sc(C)cc2Br)=O)c1Cl 29761,N1(C(CC2N(C)CCC2)=O)CCC(C2CCCN(C(c3ccc(Cl)o3)=O)C2)CC1 29762,N1(C(c2c(C)nc(C)o2)=O)CC2CCC(C1)N2C(c1cc(I)c(O)cc1O)=O 29763,C1(C(N2CCC(NC(c3cnn(C)c3Cl)=O)C2)=O)Cc2ccccc2CO1 29764,c1(CNc2ccc(C(N3CCC(NC(C)=O)CC3)=O)cn2)cc2ccccc2[nH]1 29765,CCC(C)C(C(=O)NCCc1cc(C)on1)NC(=O)CC(C)n1cccc1 29766,CC(C)CCCCCCC(=O)NCC(C)CN(C)C(c1ccncc1N)=O 29767,c1(C(N(C2CCN(C(C(=CC3CCCC3)C)=O)C2)C)=O)nc(Cl)c(Cl)s1 29768,C1(NC(COC(c2nccn2C)C)=O)CC(F)CN(C(c2cncc(F)c2Cl)=O)C1 29769,CCCCC(=O)C(=O)NCC=CC(N1CC(S(C)=O)C1)=O 29770,C1(C(=O)NCCc2ccn(C)n2)CCC2(CCC2)N1 29771,N1(C(COCCC=C)=O)CC(NC(c2cc(C)n(C(C)C)c2C)=O)CC1(C)CC 29772,C(=O)(CS(=O)(=O)C(C)(C)C)NC12CC(NC(C(CC)N(C)C)=O)(C1)C2 29773,CCCC(CC)C(=O)N1CCC(CNC(c2csc(CC)n2)=O)C12CC2 29774,C(=O)(CCC(F)(F)C(=O)N1CCCCC1CNC(C1(C)CNC(=O)C1)=O)OCC 29775,N1(C(c2nc(CCC)sc2)=O)CCC(NC(=O)CS(=O)(=O)C2CC2)C12CCCC2 29776,CC(C)C(C(=O)N(C)CCOCCCO)C(C)NC(=O)CC1(C#N)CC1 29777,C(=O)(CC(O)CC(C)(C)C)N1CCC(CCNC(Cc2cncc(C)c2)=O)C1 29778,c1(C(=O)NC2CN(C(C=CCOC)=O)C2)cccc2ccc(Br)nc12 29779,C(CO)(CCF)NC(C(C)N(C(=O)C=C1CCC1)C1CC1)=O 29780,Cc1cccc2c1c(NC(=O)CC1CN(Cc3ccc(F)cc3)C1)cn2C 29781,c1(C(C)CNC(=O)CN2CC2CNC(C2(C)CC2Br)=O)ccccc1 29782,Cc1oc(C#N)cc1C(=O)NCC1(C)CCN(C(C2CCCC(C)CC2)=O)CC1 29783,CCC(CC(=O)N1CCOCC1Cc1cnn(C)c1)C(C)(C)C 29784,CC1(C)OCCC1CC(=O)NC1CCCC1NC(c1ncccc1O)=O 29785,N1(C(c2c(C)n(C)cc2)=O)CCCCC(NC(c2ccc(CO)s2)=O)C1 29786,Cc1ccc(O)nc1CNC(C1CCCN(CC2CCSC2)C1)=O 29787,N1(c2cc(=NC)[nH]c(Cl)n2)CCC2(CC1)COC(CNC(=O)CN1CCOCC1)C2 29788,N1(C(CC(=O)OCC)=O)CCC(NC(=O)Cn2ncnn2)CC(C)(C)C1 29789,N1(C(c2c(C)nn(C(C)(C)C)c2)=O)CC2CCC1C2NC(=O)COC(C)C 29790,C1(C(=O)NC2CN(C(c3c(C)onc3)=O)CC2(C)C)Cc2ccccc2S1 29791,C(C1=NOC2CCCC12)NC(C(=O)N(C(COc1ccc(C)cc1)C)C)=O 29792,C=C(C)C1CN(C(=O)CN(C)C(C2CCN2CC)=O)CCO1 29793,c1(C(=O)NC(CCCCNC(COCCC=C)=O)C)ccnc(Cl)c1OC 29794,CCCC(CC)C(=O)NCC1CCC1NC(=O)COCC1CCCC1 29795,C12(C(=O)NCC(CC)(C)OC)CC(CN1C(=O)CCOCC(C)(C)C)C2 29796,C(=O)(CC(C)P(C)(C)=O)NCCCN(C(CSCC(=O)OC)=O)C(C)C 29797,C(=O)(C1=CCCN(C(C2CCC=CCC2)=O)C1)NCCc1n(C)nnc1 29798,C1(C(C)C)CCCN(C(C2C=CCN2C(c2scnc2Cl)=O)=O)CC1 29799,N1(C(C(c2ccc(C)cc2)F)=O)CC2=C(C1)CN(C(=O)CCc1cnc(C)o1)C2 29800,C12(CNC(C3(NC(C(C)C)=O)CC=CC3)=O)CCC(CN(C(=O)C3=NOCC3)C1)C2 29801,CCCC(C)(CCC)C(=O)NCCSC1COCCN1C(C=O)C(C)C.OC 29802,C(N=c1nc(O)c(Br)c[nH]1)C1CCC(NC(c2ccc3nncn3c2)=O)C1 29803,c1(C(N2C(CNC(C3CC(=O)N3)=O)CC(C)(C)C2)=O)cnc(O)c2ncccc12 29804,Cc1nc2ccnn2c(C)c1C(N1CCN(C(c2cnc(O)n2C)=O)C(C)C1)=O 29805,Cn1cnc(C(C(=O)NCCC(O)C2CCC2)NC(C2CC(F)(F)C2)=O)c1 29806,Cc1ccc(C(N2CC(NC(=O)Cn3nnc(-c4cccs4)n3)C2)=O)cc1CO 29807,N1(C(c2cc(SC)oc2)=O)CCN(CC(C)NC(=O)CCCCN(C)C)CC1 29808,C1(CNC(CNC(c2c(C)occ2)=O)=O)CN(C(=O)CCCCF)CCC1C 29809,c1(C(N2C(C)CC(NC(C3CC4(C3)CC(O)C4)=O)C2)=O)cn2cc[nH]c(=O)c2n1 29810,C1(n2c(C(c3n(C)cc(Br)n3)NCc3ccccn3)nnn2)CCC(F)(F)CC1 29811,C1(c2nnn[nH]2)(Cc2nc(C3CCOCC3)no2)CCOCC1.Cn1cnnc1SN 29812,c1(C(N(CCC(=O)NC2CC3CCC2CC3)CCO)=O)ccc2cc[nH]c2c1 29813,CC1OC2(C(=O)NCCC(C)(C)NC(c3cnn(C)c3Br)=O)CCC1C2 29814,N1(C(C#CC2(OCC)COC2)=O)CCN(C(C2Cc3ccccc3O2)=O)CCC1C 29815,C1(C(=O)NCC2C(NC(C(C3CCCC3)OC)=O)C2)C2CCC3C(C2)CC13 29816,Cc1c(Br)c(C(N2CCC(CNC(=O)C(C)N(C)C)C23CC3)=O)nn1C 29817,C1(C(=O)NCC2CCC(NC(Cn3c(C)c(Cl)cn3)=O)C2)CCC2(CCC2)CC1 29818,C(=O)(C1=CC2C=CC(C1)C2)NCc1occ(C(N(C2CC(C)C2)C)=O)n1 29819,C1(CC(=O)NC(C(C)C)CNC(=O)CCN2CCCC2=O)CCCS(=O)(=O)C1 29820,c1(C(=O)NCCCCNC(CSCCOC)=O)cc(C)ccc1C1CC1 29821,c1(SCC)cccnc1C(=O)NCC(C)CNC(=O)C(=Cc1ccccc1)C#N 29822,Cc1ccc(C(N2CCCCC2CC(=O)Nc2ccnc(F)c2F)=O)c(I)c1 29823,N1(C(Cc2cccc(CC)c2)=O)CCC(NC(C2CC(=O)N(C)C2)=O)C(O)C1 29824,C(=O)(CC(C)(C)C#N)N1CCCC(C(C)NC(CCC(=C)C)=O)C1 29825,C1(CNC(C=Cc2c(C)nn(C)c2Cl)=O)CCC2(CC1)OCCO2 29826,n1(CC)nccc1C(=O)NC(C1CCCN1C(c1cc(CCO)on1)=O)C 29827,C12(NC(c3ccc(C)nc3)=O)COCCC1CN(C(=O)CC1CC(F)(F)C1)C2 29828,C12(C(=O)NCCc3cncc(C)n3)CC(CN(C(C3(C)CCOC3)=O)C1)C2 29829,CC(CC(=O)N1CCC1CNC(=O)CCn1cnccc1=O)C(C)(C)C 29830,C(=O)(C1OCCn2ccnc21)N1CCC(CNC(c2n(C(C)C)ccn2)=O)CC1 29831,c1(OC)ccc(C2CCN(C(=O)NC(C)C(C)(C3CC3)OC)CC2)cc1 29832,N1(CC)CC(NC(=O)C(CCF)NC(=O)C=CC(F)(F)F)C(C)C1 29833,N(C(=NCCCCl)N1CCC(C)(F)C1)Cc1ncc(CC)s1.c1(O)ccccc1 29834,CC1(C)CCN(C(c2nnsc2C(F)F)=O)CC1NC(c1ccc(C(N)=O)o1)=O 29835,C1(CNC(C2CCC(O)C2)=O)CC(O)CN1C(C1CCN1Cc1ccccc1)=O 29836,c1(OC)c(C(=O)NC(C2CCCN2C(=O)CC2(OC)CCCC2)C)ccnc1F 29837,C1(C)(C(=O)NCC(CNC(CCOc2c(C)cccc2)=O)C)CCS(=O)(=O)CC1 29838,c1(C(=O)NC(CC(C)C)CNC(=O)C(F)=CCCF)cc(Cl)ccc1C(C)C 29839,C(CCC)(C(=O)NC1CCN(C2CN(C(=O)C=Cc3cccs3)C2)CC1)=CCC 29840,Cc1cc(N(CCO)C(=O)Nc2ccccc2Br)ccc1C(C)C 29841,C1(C2CC2)(C(=O)OCCCCCl)CCN(C(=O)Nc2ccn(C)n2)C1 29842,C1(C2CCN(C(=O)C(F)C(C)C)CC2)(NC(c2ccnc(OC)n2)=O)CCC1 29843,C1(NC(=O)Cn2cc(C3CCC3)nn2)CN(C(C2CCC2)=O)C2(CCCC2)C1 29844,N1(C(c2cnc(C(C)=O)s2)=O)CC2(CC(NC(C3COCCC3(F)F)=O)C2)C1 29845,C#CC1CCC(C(=O)NCC2CN(C(c3ccc(C(=O)OC)c(F)c3)=O)C2)CC1 29846,C1(CC(=O)N(C2CCN(C(CCc3onc(C)n3)=O)C2)C)CC(C)(C)CO1 29847,c1(C(=O)NCCC(C)NC(=O)C=Cc2ccc(F)cc2)cc2c(Cl)cccc2[nH]1 29848,N1(C(C(CCC)NC(N)=O)=O)Cc2[nH]nc(C(=O)N(CCC(=O)N(C)C)C)c2C1 29849,c1(CC(=O)N(C2CCN(C(=O)C3=COCC3)C2)CC)cc(C)ccc1F 29850,Cc1cc(N(CC(C)O)C(=O)CNC(=O)OCCC(C)C)c[nH]1 29851,CC1CC(c2ccccc2)(C(N2CC(F)(CNC(=O)C(C)CO)C2)=O)C1 29852,C(=O)(C(CC=C)CC(C)C)NC(C(=O)NCC(=O)OCC#C)CCF 29853,c1(CCC)[nH]nc(C(=O)NCC2CN(C(C3CCN(C(C)=O)C3)=O)C2)c1[N+](=O)[O-] 29854,CC1CCCN(C(=O)CC2CCCC2C)C1CNC(c1cnc(C#N)s1)=O 29855,N1(C(C(=C(C)C2CC2)F)=O)CCC2(CC1)CC2NC(c1ccc(CO)c(Cl)c1)=O 29856,C1(N(C(C2C3COCC23)=O)CC)CCCN(C(=O)Cc2ccoc2C)CC1 29857,c1(CNC(=O)NC(C2CCCOC2)C#C)ccc(C)o1 29858,C1(C(=O)NCc2c(C(N3CCC(C(CC)CC)C3)=O)occ2)CCS(=O)CC1 29859,N1(C(C(c2cccnc2)C)=O)CCC(N(C(=O)C=CCF)C)CC1 29860,c1(C(N2C(C(C)NC(=O)CCc3cncnc3)CCC2)=O)c[nH]c2ncccc12 29861,Cc1cc(=NC2CCC(=O)N(C)C2)[nH]c(N2CCC(c3ncc[nH]3)C2)n1 29862,C1(C(=O)NC(CCNC(CC(CC)OC)=O)(C)C)CC12CCS(=O)(=O)CC2 29863,C1(C(=O)NC)C=CC(NC(=O)Cc2nnnn2C2CCC2)C1.c1(C)ccon1 29864,CC1CS(=O)CCN1N1CCc2c(ncn2C2CCOCC2)C1.CCC 29865,N1(C(C2COCC(C)N2)=O)CCOC(C#N)C1 29866,C(CCCC(=O)N1CCCC1(C)CNC(C1C(C(F)F)C1(C)C)=O)OCC 29867,C1(NCc2c(C)c[nH]n2)CCC(NC(c2ccc(CO)cc2)=O)CC1 29868,C1(NC(C2N(C(c3c(C)oc(CO)c3)=O)CCC=C2)=O)(CO)CC2CCCC12 29869,c1(CNC(C2(COC)CC2(F)F)=O)oc2c(c1C)C(=O)CCC2 29870,C1(CC(=O)NC(C)CN(C)C(c2ncoc2-c2ccccc2)=O)CCCCN1C 29871,c1(C(=O)NCCC(C)NC(Cc2ccn(CC)n2)=O)cc(C(C)=O)c(C)nc1C 29872,C12(C(N(CCNC(C(CN(C)C)O)=O)C3CC3)=O)C3CCC(CC13)C2(F)F 29873,CC1CCC(CNC(c2cnc(N(C)C)cn2)=O)CN1C(=O)C=CC1CC1 29874,C1(N(C(C(CC#C)O)=O)C)CCCCN(C(c2cnn(C(F)F)c2)=O)C1 29875,C(CC(C)(C)C)(C(=O)N1CC(CNC(=O)C=C(C)Cl)C2(CC2)C1)OC 29876,C1(CCOC)(OC)CCN(C(=O)OC(C)(C)C)CC1.c1(C(=O)NC)ncno1 29877,Cc1ocnc1CC(=O)NCCC1(C(=O)NC2(C3CCCO3)CC2)CCCC1 29878,c1(C(N(CC(C)NC(=O)CC2(CO)CC2)CC)=O)ccc(C(F)F)cn1 29879,C#Cc1cccc(C(N2CCC(CN(C)C(C3CC(=O)NC3(C)C)=O)C2)=O)c1F 29880,Cc1noc2nc(C(=O)NCC3(Cn4cc(CN)nn4)CCC3)ccc12 29881,N1(C(c2nc(Br)nn2C)C(=O)NCC=C)CCCC(O)(C(F)F)C1 29882,c1(CN2CCC(CC(N3CCC(N4CCCC4)C3)=O)CC2)cccc2nonc12 29883,CCCC(CC(C)C)C(=O)NC1CC(NC(=O)CCCC(F)(F)F)CC1O 29884,C(=O)(CCCC(=O)C1CC1)N1CCC(C(C)NC(C(C)O)=O)C1 29885,N1(C(C(CC=C)C)=O)CCC2C(C1)CN2C(C12CC(c3ccccc3)(C1)C2)=O 29886,CCCCCC(C)CC(=O)NC1C2CCC1N(C(=O)C1=NNC(=O)CC1)C2 29887,Cc1noc(N)c1C(=O)NCC(C)C(N1CCOC(C2CC2)C1)=O 29888,C(=O)(C(O)CC(N)=O)N1C(C2CCN(C(CCCC3(C)COC3)=O)CC2)CCC1 29889,C(=O)(C(CC)C(=O)NC(C)Cn1cccn1)OCC 29890,CC1CN(C(=O)CCn2ncn(C)c2=O)CC1CNC(=O)CSCC#N 29891,Cc1cc2ccc(C(=O)NCC3(O)CCN(C(=O)Cc4ccoc4)CC3)cc2o1 29892,N1(C(c2c(C)snn2)=O)CCC(CCCNC(C2(P(C)(C)=O)CC2)=O)CC1 29893,N1(C(c2c(C)ccnn2)=O)CCC2CCN(C(c3cc4n(n3)CC(F)C4)=O)CC12 29894,c1(C(=O)NCC(C)(C)NC(c2c(COC)ncs2)=O)cccc2c(C)cccc12 29895,c1(C(=O)NCC2(OCC)CCS(=O)(=O)C2)nccn2cccc12 29896,C1(NC(CCCC(C)C)=O)CC(NC(c2csc(=N)[nH]2)=O)C12CCOCC2 29897,C1(NC(CC2CCC(NC(CCC(=O)N(C)C)=O)CC2)=O)CCN2CCC1C2 29898,C1(C2CC2)(CNC(COCCCC)=O)CCN(C(c2cnn3c2OCCC3)=O)C1 29899,C=C(C(=O)OCC=CC)C(C)(C)C.c12ccc(cc1)CCC(=O)N2 29900,CC1(C)CNC(=O)CN1c1ccn(-c2ccccc2)n1.C(F)F 29901,Cc1ccc(-n2nc(-c3ccncc3)nc2CC2CCN(C)C2)cc1Cl 29902,O(S(=O)(=O)CCC(CC1CC1)N1CCCCC2(CCC2)C1)NC(=O)OC(C)(C)C 29903,c1(C(=O)NC(C)C(N)c2ccco2)nccc2ccn(C)c12 29904,C(=O)(C(C(C)C)NC(=O)C1CC1)NCC(C(C)C)NC(c1n(CC)nnc1)=O 29905,C(CCNC(c1ccc(CC(C)C)s1)=O)(C(C)C)NC(C1(CC#C)CCCO1)=O 29906,c1(OC)cc(CC(N2CC(O)(CCNC(c3cnc(C(F)F)s3)=O)C2)=O)on1 29907,N1(CC(CCCC)CC)CCC(=O)N(Cc2cnn(Cc3ccccc3)c2C)C1=O 29908,c1(C(C(=O)NCCCN(C(CCC(=C)Br)=O)CCO)O)ccc(C#N)cc1 29909,C1(C(N(CCCNC(CS(=O)(=O)NCC)=O)CCO)=O)CCCC2(CCOC2)O1 29910,c1(C(c2n(CCCSCC)nnn2)NCC2CC(CC)C2)ccc(NC)cc1 29911,C(=O)(CC1=CCN(C(c2cccnc2O)=O)CC1)N(CC(C1CC1)OC)C 29912,C(=O)(C1c2c[nH]nc2CN1C(=O)C(Cl)Cl)N1C(C)COCCC1 29913,C1(C#N)(C(=O)OC)CCN(C(=O)CSC2CCOC2=O)C1 29914,CCC(CC(=O)NC1CCC(NC(=O)Cc2ccc(C#N)cc2F)CC1)C(F)F 29915,C(=O)(CC(O)CNC(C1CC1C(F)(F)F)=O)N(CC(CC)CC)C1CC1 29916,c1(OC)ccc(F)cc1C(=O)C(=O)NCC(C1CC(OC(C)(C)C)C1)=O 29917,c1(NC(C2CCCCC2)=O)ccc2ncoc2c1.C1(NC(C2CC(C)C2)=O)CC1C 29918,C(=O)(C(F)CC1CC1)N(C(C)CN(C(=O)CCOC1CC1)C)C 29919,Cc1cnc(C(=O)NC2CCCCC2CNc2nccc(CC#N)n2)cn1 29920,C1(C)(CNC(C2CC(C)C2)=O)CN(C(=O)CNC(c2ccc(F)c(F)c2)=O)CC1C 29921,C(CC1=CCN(C(=O)Cc2cn[nH]c2)CC1)N(C)C(C1CCCN1S(C)(=O)=O)=O 29922,N1(C(Cc2c(C)non2)=O)CCCC(CCNC(C2CCN(C)C2)=O)C1 29923,Cc1c(C(=O)NC(C(=O)N(CC(C2CCCC2)O)C)C(C)O)[nH]ccc1=O 29924,c1(N2CCC(Nc3c(C)n[nH]c3C)CC2)ncnc2c1nnn2C1CC1 29925,c1(CC)ccc(F)c(C(=O)NCC(O)CNC(c2c[nH]c(=N)o2)=O)c1 29926,C1(CN(C)C(c2[nH]nnc2C2CC2)=O)C=CC(NC(=O)CC2CCCC2)C1 29927,c1(N(CCOC)CCNC(=O)Cn2cnc([N+](=O)[O-])c2)ncnc2scc(C)c12 29928,C(C(CNC(C1SCCS1)=O)S(C)(=O)=O)NC(CCNC(=O)NC)=O 29929,c1(OC)cc2cc(C(N3CCOC(CNC(=O)C(O)CF)C3)=O)[nH]c2cc1OC 29930,N1(C(C(C)=C(CC)C)=O)CCCN(C(C2CC3CCC(C2)C3O)=O)C(C)C1 29931,CCCC(C)(CC)C(=O)NCCCCC(=O)NC1(CO)CC2CC1C2 29932,c1(C(=O)Nc2ccc(OC(C)C)cc2Cl)cccc2oc(O)nc12 29933,c1(CN(C2CNC(=O)C23CCC3)C=O)c(F)c(F)c(Cl)c(F)c1F 29934,c1(OC)ccc(F)cc1C(=O)NCCCCCCNC(=O)C(F)C(C)C 29935,c1(C(N2CCC(NC(C3(OC)CCC(C)(C)C3)=O)C2)=O)cccc2c1CC(=O)N2 29936,C12(C(=O)NC(CC=C)C)CC(C)(CN1C(c1c[nH]c(=N)c(C)c1)=O)C2 29937,C1(OC)(CNC(c2cccc(-c3csc(C)n3)c2)=O)CCN(C(C2CC2C)=O)C1 29938,S(=O)(=O)(c1ccc(C#N)cc1)NCC(=O)Nc1c(NC(C(F)=C(C)C)=O)cccc1 29939,CC(=O)CCN=C(NCc1cccc(C(C)C)n1)N1CCN(c2cccs2)CC1 29940,c1(CC(CNC(N(CC)Cc2cccnc2O)=O)CO)ccc(Br)c(F)c1 29941,c1(C(=O)NCC2(OC)CN(C(C3(CC=C)CCCC3)=O)C2)ccc(F)cc1N 29942,OCCC(N=c1[nH]c(=NCCc2cccc(Cl)c2F)c2ccccc2[nH]1)C1CC1 29943,C(C)(CCCCNC(=O)Cc1cnn(C)c1)NC(C1(NC(C)C)CC1)=O 29944,C(=O)(CN1C(=O)CCc2ccccc21)NC(CN(C(=O)CSC)CC)C 29945,Cc1nc(C(c2nnnn2-c2ccccc2)NCCC2(SC)CC2)sc1C 29946,c1(OC)ccc(Cl)c(C(N2CC(NC(c3cc(O)ncn3)=O)CC(O)C2)=O)n1 29947,N1(C(C(CNC(C(C)SCC)=O)CC(C)C)=O)CCc2c(C#N)cccc21 29948,C1(C(C(=O)NC2(CN(C(C3(COC)CC=CC3)=O)C)CC2)C)CCC(C)(O)CC1 29949,N1(C(c2c(OC)nn(C)c2)=O)CCC2(NC(=O)CCc3cnn[nH]3)CC2C1 29950,n1(CC)cc(CC(=O)NCC(O)CNC(C2(C)CCCO2)=O)cn1 29951,c1(C(=O)NC2C(C)C2)cn(CC(=O)NCC(=O)NCc2c[nH]nc2C2CC2)cn1 29952,C1(O)(C(=O)NC(C(=O)OCC)C)CCN(C(=O)C(=O)NCCOC)C1 29953,C(=O)(CCCCC(N)=O)N1CCCC(CCNC(C(CN(C)C)O)=O)C1 29954,c1(C(N2C3CCC(NC(C(CCC)OC)=O)(C3)C2)=O)cnc2ccc(C#N)cn12 29955,c1(NCCCCOCC)[nH]c(=NCc2ccc3ccsc3c2)nc2scnc12 29956,Cn1cnc2c(N3CC(CNC(c4cn(CCN(C)C)nn4)=O)C3)ncnc12 29957,C(CCCC(C)(C)C(=O)NNC(=O)CC(C)(C)C)NC(CC)CC(=O)OC 29958,N1(C(C2N(C(C3C(C(=O)OCC)C3)=O)C(C)C2)=O)CC(C)CCC12CC2 29959,N1(C(=O)C=CCF)CC(NC(=O)CSN2CCCC2)CC1CSc1cccnc1 29960,c1(C(=O)NCC(C(C)C)NC(=O)C(C)(C)c2ccccc2)nn(C)cc1Cl 29961,c1(C(N(C2CN(C(C(CC)OC)=O)CC2O)C)=O)cc(F)cnc1O 29962,c1(C(C)(C)C)cncc(C(=O)NCC(=O)NCCOCC(F)F)c1 29963,N1(C(C2(C)CCN(Cc3c[nH]ccc3=N)C2)=O)CCc2ccc(C#N)cc2C1 29964,C(C(C(=O)NCC1CCCO1)N(C)Cc1cocn1)(C1CCCC1)OC 29965,C(c1ccccc1)=CC(=O)N(CC(CNC(c1cc(SC)oc1)=O)O)C 29966,Cc1cc(C(=O)NCCC2CCN(C(C3C(C)C3C)=O)C2)cc(N)c1O 29967,C1(NC(C2C(NC(C(C)C3(O)CCC3)=O)COC2)=O)CC(C)(C)C12CCC2 29968,c1(C(N(CCCNC(C2(C(C)C)CCC2)=O)CCO)=O)ncccc1Br 29969,c1(C(=O)NCC2(F)CCC(CNC(C3C(C)C3)=O)C2)n[nH]c2c1CS(=O)(=O)CC2 29970,CCC(C(C)(C)O)NC(C12CC(NC(C3CC4(CC4)CO3)=O)(C1)C2)=O 29971,N1(C(C2C(CCC)C2)=O)CCC(C(=O)NC2C=CCCC2CO)CC1(C)C 29972,c1(C(C(=O)NCC(C)N(C(=O)C(O)P(C)(C)=O)C)=O)cc(Cl)cc(Cl)c1 29973,c1(N(C(COC)C2CC2)C)cccc(S(=O)(=O)NCC(C)S(C)=O)n1 29974,CC(C)CCC(O)C(=O)NC1CCC(CC(=O)NCC(O)CNC(N)=O)CC1 29975,C(=O)(CCC(C)(C)NC(c1ccccc1CC=C)=O)N1C(CCC=C)CCC1 29976,c1(CC)cc(C(N2CCC3(NC(c4coc(CO)c4)=O)CC3C2)=O)cn(C)c1=O 29977,C(CCCCNC(c1cc(C2CCOC2)[nH]n1)=O)N(C(C(C)C1CCC1)=O)C 29978,C(CCCC(=O)NC(COC)CC(=O)NC(C)Cc1nc[nH]n1)OCC 29979,c1(C(=O)NCCN(C2CCCC2)C(c2c(COC)cc[nH]2)=O)ccn(C)c(=O)c1 29980,CCCCC(O)C(=O)N1CC(NCc2ccc(Br)nc2)C2(CC2)C1 29981,CC1C(C(=O)NCCNC(C2(c3cc[nH]c3)CC2)=O)CCN1C(=O)OC(C)(C)C 29982,C1(F)(CNC(C2C(C(=O)OC)CC2)=O)CCC(NC(=O)CN2CCCC2=O)C1 29983,C1(C(N(CCOCC=C)C)=O)CC(NC(=O)CCCNC(C)=O)CCO1 29984,N1(C(Cc2ccc(C)o2)=O)CC(CNC(c2cnc(C(C)(C)C)o2)=O)CCC1C 29985,C(c1cc(F)c(F)c(F)c1)=CC(=O)N(C)CC1N(C(CC(=O)OC)=O)CCOC1 29986,c1(OCC)ncccc1C(=O)NCCOCCNC(=O)C(CC)c1ccccc1 29987,O=C1CN(CCC2CC=CCC2)CC2(CO)COCCN12 29988,Cn1ccc(C2CC2C(=O)NCC2CCN2C(=O)CNc2ccccc2)n1 29989,C1(CNC(CNC(=O)NC)=O)CC2(CCC2)CN1c1cc(Cl)nc(COC)n1 29990,c1(C(N(CC(CNC(C2(CC#C)CCCC2)=O)C)C)=O)[nH]nc2ncccc12 29991,c1(C(N2CCC(CC(=O)NC3CCS(=O)(=O)C3)C2)=O)cc(F)ccc1Br 29992,N1(C(C(CCC)N(C)C)=O)CCN(C(C2(C)CCCOC2)=O)CC1C 29993,C1(CNC2(CC(N)=O)CCC2)CC1(Br)Br 29994,CC(O)CCCCCC(=O)N1CC(CNC(c2ccon2)=O)C2(CC2)C1 29995,CCN=c1[nH]cc(C(N2CCC2CO)=O)s1.C1(=O)CC(C)N1 29996,C(=O)(C1=CCCC1)NCC(CO)NC(c1cc(CC)on1)=O 29997,c1(C(N2CCN(C(c3coc(CO)c3)=O)C(CCO)C2)=O)cc2cnccc2o1 29998,C1(C(=O)NCCC(C)N(C(c2ccc(C)o2)=O)C)CC=CCC1C 29999,c1(C(=O)NC2C3(CN(C(CSCC(=O)OC)=O)C3)CC2)cnc2snc(C)c2c1 30000,c1(OC)cc(C)c(F)cc1S(=O)(=O)N1CCc2ccc(CSC)cc2C1 30001,C1(C)(CNC(CN(CCC#C)C)=O)CCCC1NC(c1cnsc1)=O 30002,CC(C)(C)CCC(=O)NC12CCC(NC(C3CCC(C)(C)CC3)=O)(CC1)C2 30003,N1(C(C(CCNC(=O)CCc2nc[nH]n2)OC)=O)CCC2(CCOC2)CC1 30004,N1(C(C(=O)NCC(=C)C)CC(C)C)CC(C)CC2CCCCC12 30005,c1(C(N(C)CC2N(C(CC(=C)C)=O)CCC2)=O)cc2c(cc1C)OCO2 30006,n1(CC)nc(C)c(C(N2CCCN(C(=O)Cc3cc(C)ccc3C)CC2)=O)c1C 30007,c1(CNC(=O)NCC2CC2C2(O)CN3CCC2CC3)cc2cccn2c(O)n1 30008,C1(C(=O)NC2CC(CNC(=O)CC3CSCCS3)C2)(OC)CC(C)C1 30009,C(CNC(=O)Cn1cnccc1=O)(C(C)(C)C)NC(CN(S(C)(=O)=O)C)=O 30010,c1(CO)cc2cc(O)ccc2[nH]1.C12CCCCN(C1)C(=O)c1ccc(o1)C(=O)N2 30011,C1(CC(=O)N(C)CCOCCCNC(=O)CC2COC(=O)C2)OCCC1(C)C 30012,N1(C(CCCc2n(C)cnn2)=O)CC2CC1C2NC(=O)C(C1CCOCC1)O 30013,Cc1ccc2nc(C)c(C)c(C(=O)NS(=O)(=O)CC3CNCCO3)c2c1 30014,N1(CC=C)CCc2nc(C(=O)NCC3(CCOCC)CCCC3)cn2CC1 30015,CC(=O)n1cc(CN2CC3(CC3C(=O)NCC(C)(C)F)C2)c2cccnc12 30016,CN1CC(C)(C)CC1C(N1CCC(CC(=O)NCCCN2CCCC2)C1)=O 30017,CCC(N=c1[nH]c2c(c(=NC(C)c3ncc(C)s3)[nH]1)COC2)C1CCCC1 30018,Cn1cc(CN2CCC(C)(C(=O)Nc3cccc4[nH]ncc34)C2)c2ccccc12 30019,CCC(CC)C(F)C(=O)NCC(O)CCNC(c1ccc(F)c(C)c1)=O 30020,n1(CC(=O)N(C2CC2)CC2N(C(C(C)C(C)O)=O)CCC2)ccc(=O)n(C)c1=O 30021,CCC(CC)CCC(=O)NCCC1(O)CCN(C(=O)CCNC(=O)C=CCl)CC1 30022,c1(C(c2nnnn2C(C)(C)C)Nc2c(CC)nc(C)cc2)ccc2c(c1)CCC2 30023,c1(OC)ccc(F)c(CN2CCCC(NCc3ccc(F)cc3C#N)C2)c1Br 30024,CCCCC(O)C(C)C(=O)N1CCCC1CC(=O)NC1(C)CC(C)(C)OC1=O 30025,C(=O)(C#CC1CCCOC1)N1CCC(NC(C2CCC(CC)O2)=O)C(C)C1 30026,c1(CCC(N2CCC(NC(C(C)OCCC#C)=O)C2)=O)c(C)nc(O)nc1C 30027,C12(C(=O)NCC3CCC=CCC3)CCCC1N(C(c1sccc1F)=O)CC2 30028,Cc1ccc(C(=O)NC(C(=O)NOC2CC3CCC2C3)c2cccnc2)nc1C 30029,N#Cc1ccc(C(c2nnnn2C2CCC2)NCC2(n3ccnn3)CC2)cn1 30030,C1(OC)CC2CC1CN(C(C1CC(O)CN1C(C)=O)=O)C2 30031,c1(CC)ccnc(C(C(=O)NCC2CC2)N(C)CC2(C#N)CCC2)c1 30032,c1(SCCNC(CC)=O)nccc(=NCCOCc2ccc(OC)cc2)[nH]1 30033,C(C(C)C(C)C(=O)N1CC(CCCCNC(c2nnc(O)nc2O)=O)C1)OC 30034,c1(C(=O)NCC23N(C(c4cn(COC)nc4)=O)CC(C2)C3)ccsc1S(C)(=O)=O 30035,CC(CC(=O)N1CCN(C(c2cnn(CC3CC3)c2)=O)C(CCO)C1)C(F)F 30036,N1(C(C(C)OCC=C)=O)C2CCC(C2)C1CC(=O)N(c1cncc(F)c1)CC(C)C 30037,C1(CC)(NC(=O)CC2(n3cccn3)CC2)CCCC1.C12C=CCN1C2=O 30038,C1(C(=O)NC(C(C)O)CO)COC2(C1)CN(C(=O)COCCOCCO)C2 30039,Cc1cc(C(=O)N(C)CCN(C)C(c2cc(C3CC3)n(C)n2)=O)sc1Cl 30040,C1(NC(C(CCC)C)=O)CN(C(=O)C2=CCC(C)(C)CC2)CC2(CCC2)C1 30041,N1(C(C(C)NC(N2CCNC(c3ccccc3F)C2)=O)=O)CCc2ccccc21 30042,C1(=O)CC(O)CN1.c1(C(=O)NCCCNC(C)=O)nc(Cl)cs1 30043,N=c1nc[nH]c(=NCCOC2CCN(C(=O)C=C3CCC3)CC2)[nH]1 30044,N1(C(c2cnc(C(C)C)nc2)=O)CC(O)C(O)C1CNC(=O)C(C)CC1CCC1 30045,n1(CC)cc(CC(=O)NC2CCCC2CNC(=O)N(C)C)cn1 30046,c1(C(=O)NCC(C)(C2CCC2)NC(CSC(C)(C)C)=O)ccnc2ccncc12 30047,c1(CC)ccc(F)cc1C(N1CCCC(CN(c2ccncn2)C)C1)=O 30048,c1(C(=O)NCC(n2cc(-c3c(COC)nns3)nn2)C)cc2n(n1)CCCO2 30049,O=S(=O)(c1sccc1I)N1CCCC(Oc2cccc(Cl)c2)C1 30050,Cc1nc(=N)[nH]cc1C(=O)N(CCNC(C1CCN(C(C)C)CC1)=O)C 30051,C(CC(CNC(=O)C(CO)N(C)C)NC(=O)C=CCCC(F)(F)F)OC 30052,N1(C(CCOCCOCCN)=O)CCC(c2nncs2)C1 30053,c1(C(=O)NC(CNC(C2CC2c2ccncc2)=O)CO)cc(Br)c(Cl)s1 30054,C(=O)(CCCCCc1cn(CC(C)NC(=O)CN2CCC(C)CC2)nn1)OC 30055,CCC(C)C(=O)C(=O)N1CC(C)C(C)(C(N2CC(C)C(C)C2C)=O)C1 30056,N1(C(C(CO)NC(C2N(CCC)CCC2)=O)=O)CCC2(CCN(C)C2)C1 30057,C12(C(=O)NC(c3ccc(F)cc3)CC)CC1CN(c1ccnc(NC)n1)C2 30058,c1(C(N2C(C)CC(CNC(c3ccc(F)nc3)=O)C2)=O)ccc(F)c(N)c1 30059,c1(C(=O)NC2CC(NC(CCn3ccc(C)n3)=O)C2)cn2ccc(Br)cc2n1 30060,N12CCC3(CC1)CC3C2=O.N1(Cc2c[nH]c(=N)o2)CCC(CCCO)CC1 30061,C=CC(C)(CC)NC(c1cc(CNC(c2cocn2)=O)[nH]n1)=O 30062,N1(C(C)CNC(c2cc(C(N)=O)c[nH]2)=O)CCN(C(=O)CN2CCOC2=O)CC1 30063,CC1C(c2ccco2)N1.C1(C(N(CC(F)F)C(=O)OC(C)(C)C)=O)CCC1 30064,CC1CN(C(c2cc[n+]([O-])cc2)=O)CC(C)C1NC(c1nnc2ccccn12)=O 30065,Cc1nncc(C(N2CCC(C)(C)C2C(=O)NC2CCCC2C#N)=O)c1C 30066,N(C(=NCCC1CCCO1)NCC(C)(C)C)CCOc1cccc(C)c1 30067,c1(CC(N2CCN(C(CCC(=O)OC)=O)CC2CO)=O)ccc2ccccc2c1 30068,Cc1nc(C(F)(F)CNC(=O)NCCc2ccoc2)n[nH]1 30069,C(=O)(CCCS(N)(=O)=O)NCCCN(C(C(C)NC(COC)=O)=O)CCO 30070,C1(NC(CN(C)C)=O)CN(C(c2cn(C)c(O)n2)=O)CC2(CC2)C1 30071,c1(C(=O)NCC2(O)CCN(C(CCCCC)=O)C2)cc(OC)c(O)c(N)c1 30072,C(C)(CCC(=O)NC1CN(C(=O)CC(F)(F)F)CC1CO)OCC 30073,c1(C(C)NC(c2cccc(CNC(=O)CCC3CCC3)n2)=O)ccc(O)cc1 30074,C1(NC(C(N2C(=O)CCC2=O)C)=O)CCCN(C(=O)Cn2[nH]cnc2=N)CC1 30075,Cc1ccncc1CC(N1CC2C(CNC(C3(CO)CCCO3)=O)C2C1)=O 30076,Cc1cnc(C(N2CC(CCNC(=O)C(c3ccc(F)c(F)c3)O)C2)=O)cc1Cl 30077,CC1CC(=O)NC(C(=O)NCC(C)(CO)NC(c2ccc(F)c(C3CC3)c2)=O)C1 30078,CCCC(O)(CCC)CC(C=O)N1CCC1(C)C(=O)OCC.C(C)(C)N 30079,C1(OC)CC2CC(C(=O)NCCCN(C(=O)Cc3csnc3C)CCO)CC12 30080,N1(C(CN(C)C)=O)CCC2(C=Cc3ccccc32)CC1.C12CCC(C1)C(=O)N2 30081,N1(C(c2cc(C)ncc2)=O)CCC2CCN(C(=O)C(CN(C)C)N(C)C)CC12 30082,n1(CC)ccc(=NC(=O)C2CC(CNC(=O)C(C#N)C(C)C)C2)[nH]1 30083,C(CC(C(=O)N1CCC1CN=[N+]=[N-])NC(c1csc(C)n1)=O)OC 30084,C(=O)(C(CC(C)C)NC(C1CN(C)C1)=O)NCC(CC)NC(=O)Cc1cccs1 30085,c1(CCC)onc(C)c1C(=O)NCCCN(C(=O)C=CC(CC)=CC)C 30086,c1(C(N2CC(OCCCCC)C2)=O)cc(CNC(C2COCC(C)O2)=O)nn1C 30087,C(=O)(C(C)(C)CN1CCOCC1)NC(C1CCOC1)CNC(C=C(C)Cl)=O 30088,C(C(O)C(=O)N(CC(C)C(=O)NCC1CSCCO1)C)SC 30089,C(C(=O)NC(CO)C(C)NC(C1(CCF)CCC1)=O)(C(C)C)SCC 30090,S(=O)(=O)(c1cccc(C(=O)N=c2cc[nH]cc2Cl)c1)NC(COC)COC 30091,N1(c2ccnc(C)n2)CC23CCCCC2(CN(C(C2(CC4CC4)CC2)=O)C3)C1 30092,N#CC1CCCC(C(N2CCN(C(=O)CCCN3CCCC3)CC2CCO)=O)C1 30093,c1(C(N(CC(CNC(Cc2cc(C)nn2C)=O)(C)C)C)=O)cc2n(c1)CCOC2 30094,C=C1CCN(C(=O)CC2(N(C)CC)CCC2)C(C(N2CCC(C)(CCO)C2)=O)C1 30095,c1(CCNC(C(CC)N(C)C(c2cc(C3CC3)no2)=O)=O)noc(=O)n1C 30096,C1(CC(=O)NCCC2(NC(C(C(C)C)C)=O)CCCC2)COC(C)(C)CO1 30097,c1(C(=O)NCCC2(O)CCN(C(=O)C3=CCSC3)CC2)cc2c(nn1)CCC2 30098,C1(CNC(C2(C)CC2)=O)(CNC(C2CCCC2Cc2ccccc2)=O)CCOC1 30099,C(=O)(C(C)S(=O)(=O)C(C)C)N1CCC(C(CNC(C(COC)(F)F)=O)F)CC1 30100,CCC(C)C(=O)C(=O)N(C)CC1(O)CCCN(C(c2sccc2CO)=O)C1 30101,Cc1cc(F)c(CC(N2CCC(C)C(CNC(C3(O)CC3)=O)C2)=O)cc1F 30102,N1(C(CC(C)CN(C)C)=O)CCCC(CC(=O)NCCN2CC3CC3C2)CC1 30103,C1(C(N2C(CCCNC(COCCC#C)=O)CCCC2)=O)CCOCC1(C)C 30104,N1(C(Cc2c(C)nc(SC(F)F)s2)=O)CC(C2CCCCN(C(=O)C=CCF)C2)C1 30105,C(C1=NOC2OCCC12)OC(C1CCC=CC1O)=O 30106,C1(C(=O)NC(CC#C)CCOC)CCN(C(=O)c2csc(C)c2)O1 30107,N1(C(C(C2CCCC2)OC)C(=O)NC(C)C)CCC(O)(CCO)CC1 30108,N1(C(C(C)OC)=O)CCCCC(NC(c2cnoc2C)=O)C1 30109,C1(OCC)CCCC1NC(=O)C(c1ccnn1C)C 30110,CCCC(CC(=O)N(C)CCN(C)CCOC)OC1CC1n1cc(NC(=O)C)nn1 30111,C(=O)(CCC(=O)N1CCOC(C2CN(C(c3coc(C)c3)=O)C2)C1)OC 30112,c1(C(N2CCC(F)(CNC(c3nc(C)oc3C)=O)C2)=O)cc([N+](=O)[O-])ccc1N 30113,N1(C(C(C=C)(C)CC)=O)CCCN(C(c2cc[nH]c3nccc2-3)=O)C(C(C)C)C1 30114,C1(C(N2C3CN(C(c4ccc(C)nc4)=O)C(C3)CC2)=O)CCc2ncccc2C1 30115,Cc1ccc2nc(C3CC3)cc(C(N3CCCC3CNC(=O)C(F)F)=O)c2c1 30116,N1(C(c2cccnc2S)=O)CCC2(CCCN2C(c2ccc[n+]([O-])c2)=O)C1 30117,c1(C(N(CCCNC(c2ccc(C(C)=O)n2C)=O)CC)=O)c(C)nn(CCO)c1C 30118,C1(C(=O)Nc2nccs2)CN(Cc2ccc(Br)cc2Br)CCC1O 30119,N1(C(C2C(NC(CCCN=[N+]=[N-])=O)C=CCC2)=O)CCC12CCCCC2 30120,c1(C(N2CC3CSCC(C3)C2)C(=O)NCc2ccco2)cc2c(Br)cccc2s1 30121,N1(C(CCC(C)N(C)C)=O)CCC2(CCC2)C(CNC(C2CCC(C)(C)C2)=O)C1 30122,c1(C(N2C(CNC(c3c(COC)scc3)=O)CC2)=O)nnn2c1CCCC2 30123,Cc1cccc(N2CCC(NC(=O)NC3OCCC3CN)C2=O)c1 30124,C(=O)(CCCCCN(C)C)N(CC(CC)NC(=O)CSc1n[nH]c(C)n1)C 30125,C1(N(C(COCC)=O)C)CCC(NC(c2[nH]ccc2CC)=O)CC1 30126,Cc1cc(C(N2CC3CCC2C(NC(C2CCC2)=O)C3)=O)c(N)c(F)c1 30127,C(CC(=O)NCCc1ncn(C)n1)(C(C)CC)NC(CC(C=C)CC)=O 30128,CC(C)CC(C)C(=O)N(CC(O)CNC(=O)CCOc1ccc(C(C)C)cc1)C 30129,c1(C(N2CC(NC(C34CCN(CC3)CC4)=O)C2)=O)ccc([N+](=O)[O-])[nH]1 30130,c1(C(=O)NCC2C(NC(CN(CCC#C)C)=O)C2)ncccc1OC 30131,C(CC1=CCN(C(c2ccc(C)c(C#N)c2)=O)CC1)NC(C=CCOC)=O 30132,N1(C(N2CC(C(=O)OCC(=O)N(C)C)CC(C)C2)=O)CCc2ccccc21 30133,N1(C(C(C)=CC2CC2)=O)CC(NC(C2CCCO2)=O)C(N=[N+]=[N-])C1 30134,C#CCCCC(=O)NC(Cc1ccoc1)C(N1CC2C=CC2C1)=O 30135,C1(NC(CCC=C=C)=O)CC=C(C(=O)N2CCC(OC(C)=O)C2)C1 30136,Cc1cccc(F)c1C(=O)NC1CCC(NC(C2CC23CC3)=O)CC1 30137,N1(C(C(C)(C)c2cccs2)=O)CCCC(O)(CNC(c2ccc(C(F)F)o2)=O)C1 30138,CCC(CC(=O)NO)C(=O)c1ccc(O)cc1C 30139,N1(C(CCOCCOC)=O)CCC2(CC1)CC(=O)N2.C(CCO)(C1CC1)SC 30140,n1(CC(N2C(C)CC(CNC(=O)CC3CS(=O)(=O)C3)C2)=O)nnc2c1CCCC2 30141,c1(C(=O)Nc2ccc(C#N)cc2)cnc2c(-c3ccc(CO)nc3)cccc2c1 30142,CCCCC(CC)C(=O)NCC(C)(F)CNC(c1ccn(CC)c1C)=O 30143,c1(C(N2CC(NC(c3ccccn3)=O)C3C2C3)=O)ccc2cnccc2n1 30144,C1(C)(NC(CCCN(C)C)=O)CCN(C(=O)C2=CCCC2)CC1 30145,N1(CC)CCCCC1C(=O)NCCC1(NC(c2cnn(CC(F)(F)F)c2)=O)CC1 30146,N1(C(=O)OC(C)(C)C)C2CCC1CC(CNC1CCC(O)CC1)C2 30147,C(=O)(C(C)(C)CCSC)N1CC(CCCC(=O)N(C2CC(OCC)C2)C)C1 30148,c1(C(N2C(CNC(C(C)(C)F)=O)C3CCC2C3)=O)cnn2c(Cl)cccc12 30149,c1(-c2n(C)cnc2)ccc2oc(C(=O)Nc3cc(O)ccc3Br)cc2c1 30150,c1(C(=O)OCC)cnc(NCCC2CN(C(C3CC4(C)CC3CO4)=O)C2)nc1C 30151,C(C(=O)NCC(F)F)(C(C)CC(C)C)N(C(COC)C)Cc1cccc(Cl)c1 30152,c1(C(=O)NCC(CC)NC(=O)C(CC)Nc2nc(C)cs2)cccc(=O)o1 30153,Cc1c(C(N2CC(NC(=O)C=CC(C)C)C(F)C2)=O)cc(Br)cc1F 30154,CC(F)(F)C(C)(C)CNC(C1(NC(=O)COCC2CCCO2)CSC1)=O 30155,N1(CC)CCCC1CC(=O)N(CC(O)CNC(c1cscn1)=O)C 30156,Cc1cc(C(=O)NC2CC23CCN(C(=O)OC(C)(C)C)CC3)nc2nccn12 30157,CN1CCOC(C(=O)NCC2(F)CCC(NC(C3(c4cc[nH]n4)CC3)=O)C2)C1=O 30158,c1(OC)ccc2c(C(N3CCC(N(c4c([N+](=O)[O-])cnn4C)C)C3)=O)cnn2c1 30159,C1(C(=O)OC)CCCC(C(N2CCCCC2CN(C)C(c2cocn2)=O)=O)C1 30160,N1(CC(=O)NC(C2CC(NC(C(C)SC)=O)C2)C)OC(C)(C)CC1=O 30161,C#CC(CC(C)C)NC(=O)C(CC1CCOCC1)NC(=O)CCCF 30162,C1(NC(c2cc(O)nc(O)n2)=O)COC2(CCN(C(c3cccnc3Cl)=O)C2)C1 30163,CC1CN(C(=O)CC(C)(C)CCC2OCCO2)CCC(c2nn[nH]n2)O1 30164,c1(SC)ncc(C#N)c(N2CC3C(C2)N3C(C2CC2C)=O)n1 30165,c1(C(N2CCC(NC(c3cc(=N)[nH]cc3)=O)(CO)C2)=O)ccc(C(F)F)cc1F 30166,Cc1ccnc(CNc2ccsc2C(=O)Nc2nccnc2C(F)(F)F)c1 30167,C1(C2(C(=O)NC(C3CCOCC3)C#C)CC2)CCCN1C(=O)CSC 30168,c1(SCC)cc(C(=O)N(c2cccc(CN(C)C)c2)C(C)=O)c2sccc2n1 30169,N1(C(CCN(C(C(C=C)C)=O)CCCO)=O)CC=CCC1CC 30170,N1(C(c2cc(C(=O)O)nn2-c2ccncn2)=O)Cc2cccc3c2C(CCC3)C1 30171,n1(CC)ncc(C(=O)NCC2CCN2C(c2ccc(C)s2)=O)c1C 30172,CCC(CNC(C1(n2ccnn2)CC1)=O)NC(=O)Cc1cnc[nH]1 30173,c1(CC)cc(C(=O)NCCN(C(=O)CSCC2CCCCO2)CCOC)on1 30174,C(CCCCC(=O)N(C1CCN(C(=O)CC2CCCCC2(F)F)C1)CC)=CCCC 30175,c1(C(=O)NCCN2CCC(C(F)C(=O)O)C2)cc(Br)ccc1F 30176,Cc1ccc(OCC(=O)NC(C)CCNC(c2cn(C)cn2)=O)cc1C 30177,c1(OC)c(C(=O)NCC2CN(C(=O)CCN3CCCCC3)CC2C)csc1Cl 30178,c1(N2C(CN(C(C3CC(C)SCC3)=O)C)COCC2)c(Cl)cccc1[N+](=O)[O-] 30179,N1(C(N(CC)CC)=O)CCN(C(=O)C2=CCCN(S(C)(=O)=O)C2)CC2CCCCC12 30180,S(=O)(=O)(CCC(=O)NCC1CC(O)CN1C(c1cccc(=O)n1C)=O)N(C)C 30181,c1(C(=O)NC(CC)CNC(=O)CN2CCN(C)CC2)cnc2ccccn12 30182,N1(C(c2c(C)oc(C(C)C)n2)=O)C2CCC1CC(N(C(=O)C(C)CC1CC1)C)C2 30183,C1(C(N(CC(C)NC(C23CCCC(C)(C2)OC3)=O)C)=O)CNC(=O)CC12CCC2 30184,C=CC1OCCCC1C(=O)NCC1(NC(c2[nH]cnc2C#N)=O)CCOC1 30185,N1(C(=O)NC2CC3N(C)C(CCC3)C2)CCn2cccc2C1c1ccccc1 30186,C12(C(N(C(CNC(CC(C=C)C)=O)C)CC)=O)C3CC(CC13)C2(F)F 30187,C1(C(C)O)CCN(C(=O)N(c2cc(Br)n(C)n2)C2CC2)CC1 30188,N1(C(CCNS(CC)(=O)=O)=O)CCCC(C)(CNC(C2(O)COC2)=O)C1 30189,CCC(C)CCC(=O)N1CCC(F)(NC(=O)COc2ccccc2)CC1 30190,CC1CCN(C(=O)CCc2cnn(C)n2)CC1N(C)C(C1COC(C)(C)CO1)=O 30191,O(NC(=O)C(C)(C)C#N)CC(=O)NC(C#C)C(C)C 30192,Cc1cccn2cc(C(N3CC(CNC(C4COC(C)C4)=O)CC3C)=O)nc12 30193,C1(CC(=O)NCc2cc[nH]c2C(=O)NCC2CC23CC3)CCCC12CC2 30194,c1(C(N2C(C(=O)Nc3cc(Cl)ccc3CO)CC(C)C2)=O)cc(F)c(Cl)cc1O 30195,c1(CC(=O)NC2(C)CN(c3nccc(C)n3)C2)c(C)cc(C)nc1O 30196,c1(CC)nn(C)c(CC)c1C(=O)OCC(c1ocnc1C1CC1)=O 30197,c1(C(=O)NC(C(CC)C)C(N2CCC3(CC(CO)C3)C2)=O)ccn2nccc2c1 30198,c1(C(=O)NCC(C)(C2CC2)NC(C(C)OCCCC)=O)cc(O)cc(C#N)c1 30199,C1(CNC(C2(C)CCC(=O)C2)=O)CC(C(=O)NC2(CC(N)=O)CC2)=NO1 30200,N1(C(CCNC(C)=O)=O)CCC(CCNC(c2ocnc2C2CC2)=O)C1 30201,CCC(CC)C(C)C(=O)NCCC1(C(=O)NOCCCN(C)C)CC1 30202,C1(C(=O)NC(C2CCN(C(C3(n4ccnn4)CC3)=O)C2)C)CCCCC(F)(F)C1 30203,CCC(C(=O)N1CCCC(NC(c2nc(Br)sc2C)=O)C1)C(C)(F)F 30204,N1(C(C(C)CC(C)(C)C)=O)CCC(O)(C2(NC(C3CCC(F)(F)C3)=O)CC2)CC1 30205,C1(C2CC2)(C(=O)NCC(C2CN(C(=O)Cc3nccn3C)C2)C)CCC1 30206,c1(C(N)=O)ncn(CC(=O)NCC2CCC(NC(C3CC4CC4C3)=O)C2)n1 30207,N1(CCCC(=O)NCC(C)N(C(=O)CC=CC(C)(C)C)C)C(=O)NC(C)(C)C1=O 30208,c1(C(N2CCCN(C(C34CCC(OC)C3C4)=O)CC2)=O)ccc2c(c1)CCCS2 30209,C1(C)(N)CCN(C(C)=O)C1.C(CCC=O)OC.C1(C(C)C)CNC(=O)N1 30210,c1(OC)ccc2sc(CNC(C)C(=O)Nc3ccc(C)c(C)c3)c(C)c2c1 30211,Cc1cn(C)nc1C(=O)N(CCC(C)NC(C1CCCN1S(C)(=O)=O)=O)C 30212,c1(NCC(CC)(C)C(C)O)nc2ccccc2nc1NCCN1CC2CC2C1 30213,CC1C(NC(=O)COC2CCOC2)CCN1C(=O)C=CC1CCC1 30214,N1(C(c2cc(C)c(O)cc2)=O)CCC2(CC1)CC(N1CCCC(C)(F)CC1)C2 30215,C=C(C)C(C)(C)C(=O)N(CC(O)CN(C(=O)C(C)C#N)C)C 30216,S(=O)(=O)(c1ccccc1F)NC(C1C(NC(c2cccc(F)n2)=O)C2CCC1C2)=O 30217,c1(C(N(CC(=O)NCCC(=C)C)C)=O)ccn(C)n1 30218,CC1CN(C(=O)C(C)Cc2ccncc2)CCCN1C(C1CN2CCC1CC2)=O 30219,CC1OCCC1C(=O)NCC1CCOC1C(=O)NCCc1cnnn1C 30220,C1(CNC(=O)NC)CCN(C(=O)Cn2ccnc2C(C)C)CC1 30221,C(C(C)(C)C(=O)N1CCCCC1Cn1cc(C2(O)CCC2)nn1)OC 30222,Cc1sc(=O)n(CC(N2CCCC2CCNC(c2cc(Cl)c(Cl)n2C)=O)=O)c1C 30223,C(C)(CO)(C(=O)NCCc1cnn(C)c1)NC(C(C)O)=O 30224,C=C(Cl)CC(C(=O)N=c1cc(C)n(CCO)[nH]1)NC(=O)C1=CC2(CCOC2)C1 30225,C(=O)(C1=NOC2(CCOC2)C1)N(CCNC(C1(c2c(C)c[nH]n2)CC1)=O)C1CC1 30226,CC1C(=O)N(CC(=O)NCCCN(C)C(c2nc(=N)cc[nH]2)=O)C(=O)C1C 30227,C1(C(=O)NCCC2CCN(C(C(C)n3cncn3)=O)CC2)CC(F)(F)C12CCC2 30228,C(C(=O)N=c1ccn(CC(C)C)[nH]1)NC(C1CN(C)CCO1)CC 30229,N1(C(CCC(C)OC)=O)CCC2(CCC(NC(=O)CCc3ccoc3)C2)C1 30230,C1(C(C)(C)C)CCC(C(=O)NC23CC(NC(C4(C5CCCO5)CC4)=O)(C2)C3)CC1 30231,C1(CNC(C=CCC)=O)CC(CNC(=O)CCOC2CCC2)CO1 30232,C(=O)(C1CCCc2scnc21)NC.C1(C)(CO)CNC(=O)C1.C(=O)(CO)NC 30233,C1(C(=O)NC2(C)CCN(C(=O)CCc3cccc(Cl)c3)C2)CCCC1S(C)(=O)=O 30234,c1(C(N(C)C)=O)cc(NC(=O)NCC2CCC(F)C2)ccc1F 30235,C(CCC(C)C)(C(=O)N1CCC(C)=C(C)C1)NC(C=CCCC)=O 30236,C1(CC(=O)NC2(CNC(=O)CC3CCCCC3)CCOC2)CCCS1(=O)=O 30237,C(=O)(C(F)C(C)CNC(=O)C(=C1CCCCC1)F)N(C(C)C(=O)OC)CC 30238,c1(C(=O)NC2CCN(C(C(CNC(C)=O)(C)C)=O)C2)n[nH]c2ccc(F)cc12 30239,N1(C(CCN(C(C)=O)C)=O)CCOC2CN(C(C3CCC(O)CC3)=O)CC12 30240,c1(C(=O)NCCC2(C(=O)NC(c3ccncn3)C)CCC2)ncccc1N 30241,N1(CCC)CC(C(=O)NCCCCCNC(=O)COCC(C)(C)C)CC1=O 30242,S(=O)(=O)(c1ccc(C#N)c(N2CCC3CC23)c1)N1CCCC(=C)C1 30243,c1(C(=O)NCC2(F)CC(CNC(C3C(OC)CCC3)=O)C2)ncc(C)cc1F 30244,C1(NC(c2ccc(OC)nc2C)=O)COC2CN(C(=O)CNC(=O)C3CC3)CC12 30245,c1(C(CN2CC(=O)O2)=O)cccc(Cl)c1F.c1(CC)nn[nH]c1C(=O)O 30246,c1(C(=O)NC2CC(NC(Cn3c(C)nnn3)=O)C2)cccc2c1OCC2(C)C 30247,CC(C)CC(C(=O)NC1CC2CC(NC(=O)CSc3nnnn3C)C1C2)C(N)=O 30248,C(=O)(C(C(=O)C1CC1)OC(C)CC)OCC.C1(=O)CCNC(=O)NCCN1C 30249,C1(C(N2CC(C)(NC(=O)CC3CCC4CC4C3)C2)=O)(OC)CCS(=O)(=O)C1 30250,N1(c2nccc(N3CCN(C)C(c4ncc[nH]4)C3)n2)CC2(CNC(=O)N2C)C1 30251,c1(OC)ccc2nc(N3CCC(n4cc(-c5cnc(C)o5)nn4)C3)sc2c1 30252,N1(C(c2ccc(C(C)=O)o2)=O)CC2(CCCN(C(c3ccccc3F)=O)C2)C1 30253,C1(COC)CN(C(=O)Cc2cncc(Br)c2)CCN1C(=O)CC(C)OC 30254,C(C(CC(C)C)C(=O)NC(C)(C)CNC(C1(C)CC1)=O)OC 30255,c1(N2CCCC(=C)C2)ncc(C)cc1S(=O)(=O)N1CCC(OCC)CC1 30256,C(=O)(C1=CC(O)C(NC(=O)CC#N)C1)N(C)Cc1ccn(C)c1 30257,Cc1ccc(C(C(=O)NC2CNC2)N(C2CCC2)C2CCC2)cc1C 30258,N1(C(=O)C=C2CCOCC2)CC2(CO)CC1(C(=O)NCC1(O)CC(CO)C1)C2 30259,N1(C(c2c(C#N)ccs2)=O)CC2CCC2(CNC(=O)CNS(=O)(=O)C2CC2)C1 30260,C1(NC(C2CC(C#C)(O)C2)=O)CS(=O)(=O)CC1NC(=O)C=C1CCN(C)CC1 30261,C1(NC(C2(CC=C)CCOCC2)=O)CC2(C1)CN(C(c1csc(C(F)F)n1)=O)C2 30262,CC(C)CC(O)CC(=O)N1CCC=CC1C(=O)NCC1(C)CC1(F)F 30263,C1(CNC(C2CCOC2)=O)CC2COCC2N1C(=O)CCc1ccc(Cl)nc1 30264,N1(CCC)C(=O)CCC1C(=O)NCCC(C)N(C)C(c1c[nH]c(=N)o1)=O 30265,CC1c2ccc(Br)c(Cl)c2CCN1C(c1c(F)cncc1I)=O 30266,CC1=C(C(=O)NC2CN(C(=O)CC(C)C3CC3)CC23CCC3)C(C)(C)CCC1 30267,C(=O)(CC(CC)C(C)(C)C)N(CCC(=O)NCc1nc(C)c(C)[nH]1)CC=C 30268,C(=O)(C1=CCC(C)CC1)NCC(CC=C)NC(c1ncsc1S(N)(=O)=O)=O 30269,c1(C(N2C(CNC(c3c(CCC)cccc3)=O)CCC2)=O)ccc2cncn2c1 30270,C1(CNC(Cn2c(CCC)ncc2)=O)CC(F)CN1C(c1cnncc1OC)=O 30271,C(=O)(CC(F)(F)C(F)F)N1CC(NC(=O)C=Cc2ccsc2)C(F)C1 30272,c1(-c2cn(C3C(NC(C4C(C(=O)O)C4)=O)COC3)nn2)ccnc(C2CC2)c1 30273,C#CCCCCCC(=O)N1CCC(CNC(C2CCCC2C)=O)C12CC2 30274,c1(CC(=O)N(C(C2CC2C(F)F)=O)C2CC2)cccc(I)c1.C12CN(CCO1)C2 30275,N1(C(c2cc(OC)nn2C)=O)CC(CNC(=O)CCCCC#N)CC1(C)C 30276,c1(C(C)C)nn(C)c(Cl)c1C(=O)NCC1CC(NC(=O)CC2CC(O)C2(C)C)C1 30277,N1(C(c2cc(C)c(C)s2)=O)CCCC(O)(CN(C)C(C2(C)CC(C)(C)C2)=O)C1 30278,c1(CC(=O)NCC(CC=C)NC(c2ncc(C)cc2C)=O)csc2ccccc12 30279,Cc1cccc2c1c(CN1CCC(C#N)(NC(=O)C(C)n3cccn3)C1)cn2C 30280,C1(C(N(CC(=O)NCC2CCCCO2)C2CCC2)=O)(CC)CCCCO1 30281,C1(NC(=O)CC(O)c2ccccc2)CN(C(c2ccsc2C2CC2)=O)CC12CC2 30282,N1(C(CCC2C(C)=NOC2=O)=O)CCCCC(CNC(=O)CC2CC2)C1 30283,C1(C(C)NC(c2c(C)c[nH]n2)=O)CCN(C(c2c[nH]ccc2=O)=O)CC1 30284,C(C(CC(=O)NC1(c2ccsc2)CC1)NC(=O)Cc1csnc1C)OC 30285,CN1CCC2CN(C(C3CC(NC(C4(O)CCC4)=O)C3)=O)CC2C1 30286,N1(C(C2CCC(OC)CC2)=O)C2CC1CN(C(C1(C)CNC(=O)C1)=O)C2 30287,N1(C(C2(SCC(=O)NC(C)C)CC2)=O)CCC(C2=NOCC2)C1.C1C(=O)N1 30288,C1(NC(CCCOC)=O)CC=C(C(=O)NC2(C(C)O)CC2)C1 30289,C1(CC(=O)NC2(C(N3CCC(CCO)CC3)=O)C(C)C2)CCOC1(C)C 30290,n1(CCC)cc(C(=O)N(CCC(=O)N(C2CCCC2C)C)CC)nn1 30291,C1(NC(c2c(N)cncc2)=O)CC(NC(c2cc(C(F)F)cs2)=O)C12CCC2 30292,N1(C(CCC)C)CC(C(=O)NC(C)CNC(C2(C(F)F)CCCC2)=O)CC1=O 30293,CC1C(C)N(C(=O)Cn2ncnn2)CCN1C(c1cc2ncccn2n1)=O 30294,Cc1cccc2cc(C(=O)NC3CCCC3NC(=O)C#CC3CCC3)oc12 30295,N1(C(=O)CC2(n3nccn3)CC2)C2CCC1CC(NC(C1CC(O)C1)=O)C2 30296,c1(C(CC)Sc2cn(-c3ncccn3)nn2)cccc(O)c1 30297,c1(C(=O)NC(CC(C)NC(c2c(C)nncc2)=O)C)ncc(C#N)cc1Cl 30298,CC12COC(C(=O)NC3CCCN(C(C4CC4C4CCCO4)=O)C3)(C1)C2 30299,c1(NC(C(N2C(CC)CC(O)C2)=O)=O)cccc(C(F)(F)F)c1Cl 30300,Cc1cc(C(=O)NC2CC(CNC(c3cccc(Cl)c3C)=O)C2(C)C)cc(O)n1 30301,Cc1cnc(F)cc1C(N1CC(CC(C)NC(=O)C(C)Sc2ccccc2)C1)=O 30302,N1(C(C(C)c2ccco2)=O)CCC(C)(C(N2CCC(CCCO)C2)=O)C1 30303,C1(C(=O)NC(CC#C)C(=O)NCc2nc(C(C)C)n[nH]2)CC2(CCO1)CC2 30304,c1(OC)ccccc1NC(C1C=CC(NC(c2csc(Br)c2)=O)C1)=O 30305,C(=O)(CCC(=O)NN(C)C)NC(C1(CNC(C(CCC)C)=O)CC1)C 30306,C1(CCOC)(NC(C2CC(C3CC3)=NO2)=O)CCN(C(C23CCC2C3)=O)CC1 30307,n1(CCCSCC)nnnc1C(C1C=CCC1)NCCC1(CO)CC1 30308,C1(NC(c2c(CC)nc(C)n2C)=O)CCN(C(=O)Cc2cnoc2)CC1(C)C 30309,N1(C(C(C)C2CCCOC2)C(=O)NCC(F)F)CCc2ccc(F)c(F)c2C1 30310,N1(CC2CC(OC)(OC)C2)CCC(=O)N(CC2CC2C2CCOCC2)C1=O 30311,Cc1ccc(F)cc1C(=O)NC1CCCN(C(=O)C(n2ccc(C(F)(F)F)n2)C)C1 30312,N1(C(COC(=O)NC(C)(C)CC(C)(C)C)=O)CCCc2ccc(S(C)(=O)=O)cc21 30313,C(=O)(C(C)(C)C(C)O)NCc1cccc(CN(C(CC(C)O)=O)C)c1 30314,C(CC1CCOCC1)(C(=O)N1CCCCCO1)NC(C1CN2CCC1C2)=O 30315,CCC(CN(C)C)C(=O)NC(C)CN(C)C(c1cc(Cl)cnn1)=O 30316,CCCCCC(O)CC(=O)NCCC1CCCCN1C(=O)C(CC)SC 30317,C1(NC(C2(c3ccno3)CC2)=O)CC2CC(NC(CCc3ncnc(=N)[nH]3)=O)CC12 30318,C1(CCCCCC)CCN(c2cc(N3CCOC(C4CCCC4)C3)ncn2)CC1 30319,C#CC1(C)CCCN(C(=O)C(CC(=C)Cl)NC(C23CCC(C2)C3)=O)C1 30320,C1(CNC(Cc2[nH]cc(C)c2)=O)COCCN(C(c2csc(CO)n2)=O)C1 30321,C(=O)(C(C)(C)CCSC)NCC1CC(COC)CN1C(=O)CNC(=O)C1CC1 30322,CC(C)N(NC(=O)c1ccccc1OC1CCOC1)C(=O)c1ccc(O)cc1 30323,c1(CC)ccc2c(c1)CN(c1nnc(-c3ncc[nH]3)n1CCC#N)CC2 30324,c12nn(C)cc1C(=O)N2.c1(C(C)=O)ccc(CNC2CCCC2CCO)cc1 30325,Cc1ncc(C(=O)NCCC2CCN(C(=O)C(C)C(C)O)CC2)c(C(C)C)n1 30326,Cc1cccnc1OC1CC(NC(=O)NC2CCC(C)(C)C2)C1 30327,c1(C(N2CCC(C(F)(F)F)C2)=O)ccc(-n2cc(-c3c[nH]nc3F)nn2)cc1 30328,N1(C(c2cnc(CC)s2)=O)CCCCC(NC(=O)C(O)CC2CCOCC2)C1 30329,c1(C(N2CC(NC(CS(CC)=O)=O)C(C)(C)C2)=O)c(O)cc(Cl)cc1F 30330,C1(C(=O)NCCCN(C(C(CN(C)C)O)=O)C)CCCCC1C(N)=O 30331,c1(C(N)=O)cc(C(N2CCC(F)C(NC(C3CCCSC3)=O)C2)=O)ccc1Cl 30332,C(=O)(CCCCC(=O)N(C)CCNC(=O)Cn1cc(Br)c(C)n1)OC 30333,c1(OC)ccc2cccnc2c1C(N1CCC(CNC(=O)C(C)C#N)C1)=O 30334,N1(C(c2c(CC)csc2)=O)C2CCC1CN(C(c1ccn(C(C)C)c(=O)c1)=O)C2 30335,c1(C(=O)OC)cc(Cl)nc(Cl)c1NC(C1(C)CCN1C(c1cscc1C)=O)=O 30336,c1(C(N2CCCC2CCNC(C23C=CC(CC2)C3)=O)=O)ccc2c(c1)COC2=O 30337,c1(OC(=O)CNC(=O)NCC(C2(C)CCN(C)C2=O)=O)ccc2nc(S)oc2c1 30338,N1(c2nnc(C(C3CC3)OC)n2Cc2ccsc2)CCCC(C)(OC)C1 30339,C1(C(=O)NCC2CC3(CC3)CN2C(c2ccc[nH]2)=O)CCC(C2CC2)CC1 30340,C1(c2nnnn2C2CC2)(Nc2n(CC)ncc2)CCCOC1 30341,N1(C(c2cnc(N(C)C)s2)=O)CC2(C1)CN(C(C1CCC(=C3CCC3)CC1)=O)C2 30342,c1(CS(C)=O)cccc(C(=O)NC23CC(C(N)=O)(C2)C3)c1.c12sccc1CN2 30343,C1(C(=O)NC(CC=CC)C(=O)N2CCC(O)(c3cc[nH]n3)C2)CCC(O)CN1C 30344,N1(C(c2c(C(C)(C)C)ocn2)=O)CCC(F)C(NC(C2(F)CC2(C)C)=O)C1 30345,C1(NC(C2C(C)COCC2)=O)CC2CN(C(=O)CN)CC2C1 30346,C1(CNC(C(C)NC(N)=O)=O)CN(C(=O)C(C)C)CCO1 30347,C1(N(C(=O)Cc2nc[nH]n2)CC)CCN(C(=O)Cc2ccsc2C)C1 30348,N1(CC)CCN(C(=O)COCCNC(C2CC(C(C)C)C2)=O)CC1C 30349,N1(C(C(CC)(C)CC)=O)CCC2CC(CNC(c3ccsn3)=O)CCC2C1 30350,C1(CC)CCCCN1C(c1cc(Cl)cs1)C(=O)Nc1ccc(OC(C)C#N)cc1 30351,Cc1ncc([N+](=O)[O-])n1CC(N1CCN(C2CCCC2O)CC1)C 30352,c1(NC)ccc(F)cc1C(N1CCCC1(C)CNC(c1c(C)[nH]c(C)c1C)=O)=O 30353,C1(C(N2CC(C=C)C2)=O)CN(C(=O)CCc2cccs2)CCO1 30354,N1(CC(NNC(c2ccc(OC)cc2OC)=O)=O)C2CCCC1CC(O)C2 30355,c1(CC2N(CC(=O)N(C(c3cccs3)=O)CC)CCC2)cn(C)nc1C 30356,CC1C(C(=O)N2CCCC2CC(=O)NCC2CN3CCC2C3)=NOC1C 30357,N1(C(c2ccc(CC)o2)=O)CCN(C(c2cc(Cl)cn2C)=O)CC1CC(F)(F)F 30358,CC1CN=C2NC(C(=O)N3C4CCC3C(CNC(c3cccnn3)=O)C4)=NN2C1 30359,C(C1=CCN(C(C2CCC(CCO)CC2)=O)CC1)NC(c1cn(C)nn1)=O 30360,Cc1cc(C(=O)NCc2cc(C)c(C(=O)NCCC(F)F)o2)c(C)[nH]1 30361,CC(C)(C(=O)NC1CCCN(C(c2csc(-c3nc[nH]n3)n2)=O)C1)C(F)F 30362,c1(CCC(=O)NCC2(CN(C(CCSC)=O)C)CC2)ccc(Cl)cc1 30363,c12cnc(cn1)C(=O)NCCOC1CCN(C1)C2=O.c1(C(C)C)nsc(N(C)C)n1 30364,C(=O)(C1=CCCSC1)N1C(CNC(C2CCC3(CC3)C2)=O)CCC1 30365,CC1C(C(N2CCN(CC3(NC(C4(C)CCCN4C)=O)CC3)CC2)=O)CCN1C 30366,c1(CC)nc(C(N2CCC(NC(=O)C3=CCCS3)CC2)=O)c(C)o1 30367,C1(C(=O)NCCN(C(CNS(C)(=O)=O)=O)CC2CC2)CC12CCC1(CC1)CC2 30368,c1(C(=O)NCC(CC=C)NC(c2cnn(CCC)c2)=O)ccc2c(c1)COCO2 30369,c1(C(=O)NC(CNC(CCOCC)=O)(C)C2CC2)ccc(C2(C#N)CC2)cc1 30370,c1(C(N2CC(CNC(COC)=O)N(C)CC2)=O)cc2ccccc2n1CC1CC1 30371,c1(Sc2ccccc2)cccc(CC(=O)N(C)CC2ON=C(C)C2)c1 30372,C1(NC(C(CCC)C)=O)CCC12CN(C(=O)CCCCN1CCCCC1)C2 30373,c1(C(=O)NC(CCC(=O)OCC)C(=O)O)cc2ccc(OC(F)F)cc2o1 30374,C(=O)(C(C)Cc1cn(C(C)C(=O)O)nn1)N(C(c1csc(C(=O)N(C)C)n1)C)C 30375,CCC(C)C(C(=O)NC1CCCCC1CC(=O)Nc1ccc(F)nc1)N(C)C 30376,c1(C(N(C2C3CN(C(=O)CC4(C)CC4)CC23)C)=O)ccc(Cl)cc1 30377,C=CCC(C(=O)NCC1(O)CCN(C(c2ncoc2CC)=O)C1)C(C)C 30378,CC(C)(O)C(F)(F)CC=CC(N1CCOCC1CC1CCC1)=O 30379,c1(C(N2CCN(C(C3C(CCN=[N+]=[N-])C3)=O)CC2)=O)cc2c(F)ccc(F)c2s1 30380,c12ccc(nc1C)C(OC(=O)C(=O)N(C(C)C1CC1)C)C2=O.C(C)(C)(C)OC(C)=O.CO 30381,c1(CCC=C)ccc(CN(C)CC2CN(C(CNC(=O)CCCSC)=O)C2)cc1 30382,c1(C(N2CCCN(C(C3CCCCS3)=O)CCC2)=O)cnc2c(c1)CCCO2 30383,N1(C(C(=O)c2ccco2)=O)CCCC(C2CN(Cc3c(F)cc(O)cc3F)C2)C1 30384,CN1CCCCC1CC(=O)NC1CC1C(=O)Nc1ccccn1 30385,c1(C(N2C(C(N(C3CCC3)C)=O)CCCC2)=O)cn2ncccc2n1 30386,C1(NC(C2CCCOC2)=O)(CO)CCCN(C(c2cnn[nH]2)=O)C1 30387,C(=O)(CC(C(F)F)C(C)(C)C)NCC1CN(C(C2C3COCC23)=O)CC(C)(C)O1 30388,C1(C(N(C2(CC)CC2)C)=O)CCN(C(=O)Cc2csc(Cl)n2)C1C(C)C 30389,C(=O)(C1=C(C)OCCC1)N1C(CCC)CN(C(=O)Cc2coc(COC)n2)CC1 30390,C1(NC(CCOC(C)C)=O)CC(NC(c2cc(O)cc(F)c2)=O)C12CCOCC2 30391,C1(C(=O)O)(Cc2cn(CCOC)nn2)CCN(C(c2cc(C)oc2C)=O)CC1 30392,C1(CNC(c2nnc(C(C)C)s2)=O)C(C)CCCN1C(c1cc(=O)cc(Cl)[nH]1)=O 30393,c1(C(=O)NCCN(CC)CC2NC(=O)NC2=O)ccc2c(c1)C(C)(C)CO2 30394,C1(C(N2CCC(C)(NC(C(CC)C)=O)C2)=O)C2Cc3ccccc3C12 30395,C1(NC(c2c(C)nc(C)o2)=O)CCC2CN(C(=O)CC3CC4CC4C3)CC2C1 30396,NC(Cc1cccnc1)CC1CCc2ccccc21.N12CCC(CC1)CN1CCC2C1 30397,CC(CC(N)=O)C(=O)N(C1CCN(C(c2cccc(Cl)c2C(F)(F)F)=O)C1)C 30398,c1(NCCC(=O)NC(CN(C(C(CC#C)C2CC2)=O)C)C)ccc(Cl)cc1Cl 30399,O=C(CN=Cc1ccco1)N1C2CN(C(C3CCCS3)=O)CC12 30400,C1(c2[nH]nc(C3CCC(N(C)C)O3)n2)CCN(C(=O)NCc2ccc(I)cn2)CC1 30401,C1(C)(C(N2CCC(N(C(c3c(COC)noc3)=O)CCO)C2)=O)CCC(F)(F)C1 30402,C1(NC(c2cnc(C(F)F)s2)=O)CN(C(=O)C2=CCCC2)CCC1F 30403,C1(OC)CCOCC1NC(=O)C(c1ccc(Br)cc1)(C)N 30404,C1(CCC(C)(C)NC(C2CC2(F)F)=O)CCN(C(=O)COCCF)CC1 30405,C=Cc1ccc(C(=O)NC2CC(C(=O)NC3Cc4ccccc4C3)C2(C)C)cc1 30406,C(=O)(C(F)C1CCOC1)N(C)CCOCCCN(C(=O)CNC=O)C 30407,CC1CN(C)CC1C(=O)NCC1CC(NC(c2ccc(-c3cccs3)s2)=O)C1 30408,c1(C(N(C(C(=O)NC(COC)C)C)C2CC2)=O)coc(OCC)n1 30409,C(=O)(CCCCN=[N+]=[N-])N1CC(C)OC(CCNC(C23C=CC(CC2)C3)=O)C1 30410,CN1CCC(C(=O)N(CCCNC(C2CC2NC(c2ccccc2)=O)=O)CCO)C1 30411,c1(C(=O)NC(C2CN(C(C3CC3(C)C)=O)C2)C)ccc(N(C)C)cn1 30412,C1(CNC(c2cnn(C(C)C)c2N)=O)CCN(C(=O)CC(C)(C)N(C)C)C1(C)C 30413,N1(C(c2ccc(CNC(C3N(C)CC(O)C3)=O)o2)=O)CC(O)CC12CCOC2 30414,C#CCCCC(C)OC(C1CC1c1ccccc1Nc1ccccc1)=O 30415,N1(c2ccnc(NCC3ON=C(C(C)(C)C)C3)n2)CC2C(C1)C(F)(F)C2(F)F 30416,Nc1ccc(C(N2CC(CC(N3CCC3CO)=O)C3(CC3)C2)=O)nc1F 30417,C1(C(NCC)=O)CC(F)CN1C(=O)Cc1ccc(C(C)(C)C)cc1.c1nc[nH]n1 30418,c1(C(=O)NCCCCCNC(=O)CC23CC(C2)C3)cc(O)ncc1Br 30419,Cc1cc(=NCc2n[nH]c3c2CCC3)[nH]c(=NCc2ccc(Br)s2)[nH]1 30420,C=CCC(C(=O)NC(c1ccccc1)C(=O)Nc1ccc(OC)nc1)C(C)C 30421,N1(C(Cc2c(C)n(C)cn2)=O)C(CC(=O)NC23CCC(C2)OC3C)C2CCCC12 30422,c1(C(N2CC(C)C(CNC(=O)CCC3CCCCO3)C2)=O)ccnc2[nH]ncc12 30423,c1(OC)ncnc(C(N2CC3C(CNC(C4(C#N)CCOC4)=O)C3C2)=O)c1F 30424,C1(C(N2CCN(C)CC2)=O)CCC2(CC2)N1C(=O)CCc1nc(Br)n[nH]1 30425,C1(NC(CC(c2ccccc2Cl)C)=O)CCCC12CNC2 30426,N1(C(=O)Cc2ccn3cncc3c2)CCC2CCN(c3ccncn3)CC2C1 30427,c1(N2CCCC(CCNC(c3cc(CC)nn3C)=O)C2)cc(S(C)(=O)=O)ncn1 30428,C(=O)(C(C)(C)CC(F)F)NCC(C(C(C)C)C)NC(c1ccsc1Cl)=O 30429,C1(C#N)(C(N2CCCC(NC(C(C)C3CCCC3)=O)C2C)=O)CC2(CCC2)C1 30430,N1(C(C2C(C)SCCC2)=O)CC(CC(=O)NC(c2ccon2)(C)C)C2(CC2)C1 30431,Cc1cncc(C(=O)NC2CCC(N(C)C(C3(CN(C)C)CC3)=O)CC2)c1C 30432,CCC(CCO)CN=c1nc(N2CCC(CC(F)F)CC2)c2c(ncn2C)[nH]1 30433,CC1(C)CCC(C(N2CC(CF)C2)=O)CN1C(=O)C=Cc1cc[nH]n1 30434,CC(C)C(C)(CN=c1cc(F)nc[nH]1)NC(=O)CCN(C1CCCCC1)C 30435,c1(C(N2C(C(=O)Nc3ccc(C)nc3)C=CCC2)=O)ccc2c(c1)CCCC2 30436,C12(NC(c3cnc4n3CCCC4)=O)CCCCCC1N(c1ccncn1)CC2 30437,c1(C(N(C)CC2N(C(C(CSC)O)=O)CCCC2)=O)[nH]c2ccc(C)cc2c1Cl 30438,N1(C(C2CCC(=O)C2)=O)CCc2ccccc2C(NC(=O)Cc2ccc(Cl)s2)C1 30439,N1(C(c2c(COC)noc2)=O)CC2C(C(F)(F)F)CC2(NC(C2CC2CF)=O)C1 30440,Cc1cc([N+](=O)[O-])ncc1C(=O)NC(C1CCCN1C(=O)C=CC(F)(F)F)(C)C 30441,c1(NC(=O)N(C)C2CC2)cccc(C(N2CCCCC2c2ccco2)=O)c1 30442,c1(-c2nc(C(CC)C)nn2C23CC(C2)C3)ccc(Cl)c(S(C)(=O)=O)c1 30443,c1(OC)cc2cc(C(=O)NC(C)CCS(C)=O)[nH]c2cn1 30444,N1(C(C=CS(C)=O)=O)CCN(C(c2cccc(OC(F)(F)F)c2)=O)CC1C1CC1 30445,c1(CCC)cccc(OC(C2CC2c2cccs2)=O)c1 30446,Cc1nn(-c2ccccc2)c(C)c1C(N1CCCC(NC(=O)CC(F)(F)F)C1)=O 30447,N1(C(CC(C)SC)=O)CC(NC(c2cc(C)cc(F)c2)=O)CC(F)C1 30448,c1(C(N(C(C)CNC(=O)C(F)(F)C(F)F)CC)=O)ccc2c(c1)COC2 30449,C1(CCNC(C2(C(=O)OC)C(=C)CC2)=O)CCCN(C(=O)C(C)(Cl)Cl)CC1 30450,C(=O)(CC(C)CC(C)(C)C)NCCC(=C)CNC(=O)CS(=O)(=O)N1CCCCC1 30451,c1(NCC(=O)NC(C2CCN(C(=O)CC3(C(F)F)CC3)C2)C)cc(F)cc(F)c1 30452,c1(NCc2c(C)cco2)[nH]c(=NCC23CC2CN(C)C3)nc2sccc12 30453,C1(C(=O)NCCN(C(c2c(C)oc(C)c2C)=O)CC2CC2)CCOC2(CCC2)C1 30454,N12CCCC(C1C)C2=O.Cc1ccc(C(=O)NCC(C)C)cc1 30455,c1(C(N(CCNC(CC(CCC)(C)C)=O)CCC)=O)c(F)ccc2nc[nH]c12 30456,C(=O)(C(F)C(F)(F)C(F)(F)F)N1C(C)CCC(NC(C2CC(OC)(OC)C2)=O)C1 30457,c1(C(N2CCC(CC)(NC(c3cnoc3)=O)CC2)=O)ccc2c(c1)nc(O)n2C 30458,C1(CC(=O)N(CC(CN(C)Cc2sccc2Br)O)C)CC(C)(C)CO1 30459,CCC(C)(CNC(C1(CC)CCN(C(=O)CSC)C1)=O)CO 30460,C1(NC(C=CSC)=O)CC2CCC1C(NC(=O)C1=C(Cl)CCC1)C2 30461,CC(O)(C(=O)NC(Cn1ccnn1)C(=O)NCCc1cnco1)C1CCC1 30462,C(=O)(CC(C)C(F)(F)F)NCC1=CCCN(C(C2=CCCC2C)=O)C1 30463,C1(C(C)(C)O)(CNC(C2CCC(=O)C2)=O)CN(C(=O)CCc2ccoc2)C1 30464,C(C(CC(F)(F)F)NC(=O)CC(CN(C)C)CC)NC(c1cc(OCC)n[nH]1)=O 30465,C1(C(C)(C)CNC(C2COC(=O)N2)=O)CCN(C(C2CCC23CCC3)=O)CC1 30466,CC(C)(CC(=O)NC1CN(C(C2CCn3ncnc3C2)=O)CC1C(F)F)C(F)F 30467,C(=O)(C1CCCc2nccn21)NCC(C)NC(=O)Cc1nc2ncccn2n1 30468,C1(NC(C2CC(n3ccnn3)C2)=O)CCC(NC(C2CCS(=O)(=O)N2)=O)CC1 30469,S(=O)(=O)(c1cc(C)c(Cl)cc1F)N1CCCC(C(C)NC(c2c(C)csc2)=O)C1 30470,Cc1cc(=NCC2(NCc3ccccc3)CC2)[nH]c(C2(CO)CC2)n1 30471,C(=O)(CCCCCCSC)NC(c1ccccc1OC(c1ccccc1)C)CC 30472,c1(C(N2CC3C(CNC(=O)C=CC4CC4)C3C2)=O)ccc(F)c(F)c1 30473,Cn1ncc(C(=O)NCCNC(C2COC(C)(C)C2)=O)c1C#N 30474,CC1CC(C(N2CCCC(CN=[N+]=[N-])C2)=O)CN(C(=O)CCNC(=O)CO)C1 30475,c1(C(N2CCC(C(C)NC(C(CC=C)(F)F)=O)C2)=O)[nH]c2c(Cl)cccc2c1C 30476,C1(C(=O)NC(CC)(C)C)CC2CC2N1Cc1ccncc1-c1ccns1 30477,N1(C(c2ccnc(C)n2)=O)CC2C3CCC(C2C1)N(C(C1(N(C)C)CCC1)=O)C3 30478,CC1CCC(C)N1CC(N1CCC(Cn2cc(-c3ccc(O)cc3)nn2)CC1)=O 30479,C1(C(N2CCC(C(=O)NCc3c(C(C)C)cccc3)C2)=O)CC(O)C(F)C1 30480,c1(C(CC(=O)NCC(C)NC(=O)CC2CCN(C)C2=O)C)ccc(Cl)cc1 30481,C(CS(=O)c1ccc(C)cc1)NC(CCCOC)(C)c1nnnn1C(C)C 30482,N1(C(C2(C(N)=O)CC2)=O)CCC(CCNC(N2CSCC2=O)=O)CC1 30483,c1(C(=O)NCC2N(C(CC=C)=O)CC=C2)ccc(C2CC2)c(C)c1 30484,C1(CNC(C(C)OCC)=O)(CNC(C2CC(F)C2)=O)CC12CCC2 30485,c1(C(N2CCN(C(CCOCC)=O)C(CCO)C2)=O)oc2ccccc2c1CC 30486,C(=O)(C(C)(CC)C(N)=O)N(CCOCCN(C(CCC(=O)NCC)=O)C)C 30487,c1(-c2scc(C(=O)Nc3cc(C)[nH]n3)n2)cncc(N2CCCC2)c1 30488,c1(CN2CCCC(CC(=O)Nc3c(C(N)=O)nccn3)C2)ccc2c(c1)CCO2 30489,c1(C(=O)NCC2(C(C)NC(C3=CCCC3C)=O)CC2)ccc(F)cc1[N+](=O)[O-] 30490,C1(CN(C(CCN(C(c2nccn2CC)=O)CC)=O)C)CCOC1C 30491,c1(C(N2CC(O)CC(NC(CC=CC=C)=O)C2)=O)nc2ccccc2nc1C 30492,CC(C)(C(=O)NC(Cc1ccccc1)CCNC(C1CC1F)=O)c1ccccc1 30493,C(C(C(=O)NCCN1CC=CCC1)NC(c1ccn(C(F)F)n1)=O)OC 30494,N1(CC(C)(C)NC(C(CC)OC2CCCCC2)=O)CCN(C(C2CC2C)=O)CC1 30495,C1(C)(C(=O)NC2C(N(C(CCOCCC)=O)C)CCCC2)CCCCCCC1 30496,C(C1CCCCCC1)=CC(=O)NCCCC(C)NC(C1CC(C(C)C)C1)=O 30497,N1(C(c2ccsn2)=O)CCC(NC(C2(C(F)F)CCOCC2)=O)C(F)C1 30498,C(C)(CCCC(=O)NC1CCC(C)CC1)NC(c1c(OC)n[nH]c1)=O 30499,c1(NCCCC(=O)NC(C(C)NC(=O)NCCC#C)C(C)C)scc2c1OCCO2 30500,C(=O)(CC(C)CC(=O)NC1(C2CN(C(C3(OC)CCOC3)=O)C2)CC1)OC 30501,C(C(N=c1[nH]nc(C#N)s1)C(C)C(C)C)NC(c1c(F)cc(OC)cc1F)=O 30502,C12(CNC(=O)Cc3ccccc3)CCC1CN(C(=O)CCc1ccccc1O)C2 30503,N1(C(Cn2c(C)cnc2)=O)CCOC2CCN(C(=O)CNC(=O)CC(C)C)CC12 30504,N1(C(C=CCNC(C(C)c2cc[nH]n2)=O)=O)CCCC(C)C1CCO 30505,C(=O)(C(C)CC(F)F)NC(C(=O)NCCc1cnc(C)[nH]1)CO 30506,CC1CCN(CC2CCCC(=O)N2)CC1NC(c1ccsc1-n1cnnn1)=O 30507,C12(C(=O)NCC(CNC(c3nc(OCC)oc3)=O)(C)F)CCCCC1C2 30508,CC1CCC(CNC(=O)Cc2cncnc2)CN1C(=O)C(=O)NCCC(N)=O 30509,c1(NC(C2(NC(CN(C)C(=O)C3CC3)=O)CC2(C)C)=O)ccc2ccoc2c1 30510,C(C(C(=O)NC1COCC1NC(=O)C(C)(C)c1cccnc1)N(C)C)OC 30511,N1(C(Cc2cn(CC)nn2)=O)CC(F)CC1CN(C(=O)CCc1csc(=N)[nH]1)C 30512,N1(c2cc(OC)ncn2)CCC(F)(F)C(CNC(C2(S(N)(=O)=O)CC2)=O)C1 30513,CC1CCN(C(=O)NCc2cccc(-n3cnnn3)c2)CC12CCC2 30514,CC1(C)CCN1CC(=O)NC1CCCC1NC(C1(c2cccnc2)CCCC1)=O 30515,C(CC(C(C)C)NC(=O)CCNC(C)=O)NC(C1CC(C(F)F)(OC)C1)=O 30516,c1(CC(=O)NC(C(C)NC(COCCCCC)=O)CO)ccc(C2CC2)cc1 30517,c1(CCC(=O)NCC(CC)NC(c2cc(C(C)C)oc2C)=O)ccc(O)cc1 30518,C1(CNC(CCSCCCC)=O)C=CC(NC(C2OCCC2C)=O)C1 30519,Cc1cnn2ccc(C(=O)NCCCC(C)(C)NC(C3CCC(F)CC3)=O)nc12 30520,CC1CN(C(=O)CN2CCCCCC2)CCCN1C(C1CCCC(C#N)C1)=O 30521,C1(OC)CCCCC1C(=O)NCc1cccc(CNC(=O)COC2CCOC2)c1 30522,C1(CNC(c2c(OCC#C)nccc2)=O)CN(C(c2cnn[nH]2)=O)CC(C)(C)O1 30523,N1(C(CSCCC(C)C)=O)CC2(CCC2)CC1CNC(c1nn[nH]c1C(C)C)=O 30524,c1(C(N(CC(C)NC(=O)C(C)n2ccnc2)CC)=O)ccc(Cl)c(C)c1 30525,O(C1CCCc2ccccc21)CC(=O)NC1CCN(C(c2cnc(C)o2)=O)C1C 30526,C1(CCCNC(CNS(NC)(=O)=O)=O)CN(C(=O)CC2CSC2)CCO1 30527,C1(C(=O)NCC2CCCN2C(C2C=CC=CC=C2)=O)CC2CCC(C1)S2 30528,N1(C(c2ccc(CNC(C(CC)CN(C)C)=O)nc2)=O)CC(O)CC1(C)C 30529,c1(C(=O)NCC(N(C(CC(CCC)C)=O)C)C2CC2)cnc2scc(C)n2c1=O 30530,N1(C(COCC)=O)CC(OC)CC(NC(c2ccc(CC(C)C)cc2)=O)C1 30531,C(C(C(=O)NCCc1cn[nH]c1)C(C)C)NC(C1CC(CCC)C1)=O 30532,CC1CN(C(=O)CNc2ncccn2)C(C)CN1C(=O)C=Cc1cncnc1O 30533,c1(C(=O)NCC2CC3COCC3N2C(=O)C(F)(F)CO)n[nH]c2ccc(Cl)cc12 30534,Cc1cnnc(O)c1C(=O)N(CCCCCNC(=O)CC(=O)NCC1CC1)C 30535,c1(C(=O)NC(CC)CN(C)C(c2cn(C)cn2)=O)cc(OC)n(C)n1 30536,C(=O)(C1=NOC2(CCC2)C1)N1CC(CCNC(=O)C2=CCC(C(F)(F)F)OC2)C1 30537,N1(C(CSC)=O)CCN(C(=O)C(CC(C)C)OC(C)=O)CC12CCC2 30538,CC1(C)CCC(C(=O)NCC2(C)CCCN(C(c3ocnc3C(F)F)=O)C2)OC1 30539,c1(CNC(CC2CCC(NC(C3CN(C(C)=O)C3)=O)C2)=O)ncccc1Cl 30540,c1(OCC(=O)NCC2CCN(C(C(CSC)C)=O)C2)cccc([N+](=O)[O-])c1 30541,Cc1cc(C(N2CCCC(CC(=O)NC3CN(C)CCC3O)CC2)=O)cnc1O 30542,Cn1c(O)nc2cccc(C(=O)NCC(C)(CO)NC(C3OCCCO3)=O)c12 30543,c1(NCCN2C(=O)CCCC2)nccc(=NCC2(CF)CC(F)(F)C2)[nH]1 30544,C12(C(N3CC(NC(C4(OC)CCC4)=O)C3)=O)CCOC1CS(=O)(=O)C2 30545,c1(CC(=O)NCC2(OC)CN(C(=O)CC(O)C3CC3)C2)c(F)cccc1Cl 30546,c1(OC)ccc(C2CCN(Cc3ccccc3F)CC2)c(F)c1F 30547,C(=O)(C(F)C(C)CNC(=O)Cc1ccsn1)NCC(C)OCCO 30548,c1(C(N(C2CC(C(=O)NC3CC3(F)F)C2)C)=O)ccccc1S(C)(=O)=O 30549,C=CCC(C(=O)NC(C)CCN(C)C(c1cnn(C)c1OC)=O)C(C)C 30550,c1(OC)ccc(C(N2CCC(CN(C)C(C3(CO)CCCO3)=O)C2)=O)c(F)n1 30551,C1(NC(COCCSC)=O)CC12CCN(C(c1csc3cncn13)=O)CC2 30552,N1(C(C(CC#C)NC(C2CC(COC)C2)=O)=O)CCCC(C)(N(C)C)C1 30553,C1(C(N(CC(CC)OC)C)=O)CCC(C)(C)N(C(=O)CC2(O)CCCCC2)C1 30554,c1(C(=O)NCC2(C)N(C(=O)CS(N)(=O)=O)CC(OC)C2)cc2cnn(C)c2s1 30555,N1(C(C2CCN(C(CC)=O)CC2)=O)CCC(CNC(C2CC(OC)C2)=O)C(O)C1 30556,N1(C(=O)CCF)CCCC(C2CCCN(C(c3ccc4nncn4c3)=O)C2)C1 30557,C(CCCCCNC(c1cccc(C2CCOC2)c1)=O)NC(C(=O)NC1CC1)=O 30558,Cc1[nH]nc(C(=O)NCCCOCCCNC(=O)CCc2ccnn2C)c1Cl 30559,N1(C(c2c(C)c(Br)cnc2)=O)CCCN(C(=O)C(C(C)O)N(C)C)CC1C 30560,C1(NC(C2(NC(C(C)C(C)(C)C)=O)CCN(C)C2)=O)CC2(CCCCC2)C1 30561,n1(C(C(=O)N(CCNC(c2c(C)ccnn2)=O)C2CC2)C)cnc2ccccc12 30562,CC1=C(C(=O)N2C3CCC(C3)C2C(N2CCCCC2(CO)CO)=O)CCC1 30563,c1(C(N(C2CCN(C(C3CCCOC3C)=O)C2)CC)=O)cc(C(C)(C)C)nn1C 30564,c1(C(CNC(C(C)OCCN(C(=O)C(=C2CCCCC2)F)C)=O)O)cnn(C)c1 30565,n1(C(C)C)cnnc1SCC(N1CCCC1C1CCN(C(c2cnc[nH]2)=O)C1)=O 30566,C1(NC(Cc2cnc(C)s2)=O)CC2CC1CN(C(C1(Br)CC1)=O)C2 30567,C1(CNC(C2(SCC)CC2)=O)CCN(C(=O)Cc2cccc(C)c2)C12CCC2 30568,C1(NC(C2CN(C)C(=O)C2)=O)CC12CCN(C(c1conc1C(C)(C)C)=O)CC2 30569,CCC(=O)CCC(=O)NC(C)CCNC(c1cocc1C(N)=O)=O 30570,N1(C(C(C)SCCCC)=O)CC(C2CC2)(C(=O)NCc2csc(C)c2C)C1 30571,C1(NC(C=NOC)=O)CCC2(CCN(C(=O)CCc3ncc(F)cn3)C2)C1 30572,c1(COC)cncc(CNC(=O)C(C)CNC(=O)C(c2cnn(C)c2)O)c1 30573,N1(C(C(N2CCSCC2)C)=O)CCc2ccccc2C1CNC(=O)CSC(F)F 30574,c1(CC#N)ccc(NC(C2CCN(Cc3cccc(Br)n3)C2)=O)cc1 30575,C1(NC(C2CCN(C)C2)=O)CCC12CN(C(=O)C=CSc1nnc[nH]1)C2 30576,N1(C(C(CCC)NC(C)=O)=O)CC2CCC(NC(=O)CSC(F)(F)F)C2C1 30577,Cc1sc2ncnc(N(CCCNC(C3COC(C)C3)=O)C)c2c1C 30578,N1(C(C(CCC)CNC(c2nccnc2C)=O)=O)Cc2nncn2C(C)C1 30579,N1(C(CCC(=O)NC)=O)CC(NC(C2(C(F)F)CCCCC2)=O)CCC1C 30580,Cc1cccc(C)c1NC(C1CCC(CN)CC1)=O.c12nc(no1)SC2C1CC1 30581,CCC(F)(F)C(=O)N1CCC(C(C)CNC(=O)CCC2CC(F)(F)C2)CC1 30582,N1(c2nc(NC(c3ncc[nH]3)C)c3c(n2)scc3)CCOC2(CCSC2)CC1 30583,N1(C(C2C3N(C(c4cc(C)c(O)nn4)=O)C(CC3)C2)=O)CC2CCC1C(CO)C2 30584,S(=O)(=O)(c1ccc(C(F)(F)F)nc1)NC(C(c1ccccc1)NCC)C 30585,N1(C(c2c(OC)csc2)=O)CC(CNC(C2CC(=C3CCC3)C2)=O)C(O)C1 30586,c1(CNC(COCCOC)=O)cccc2c1CN(C(=O)CCN=c1[nH]ccs1)C2 30587,c1(CC)cc(C)n(CC(=O)NC(C2CCCCN2C(=O)CCC(=O)NC)C)c1C 30588,C(=O)(C#CC1CCOCC1)N1CC(CCCCNC(c2n(CC)c(O)nc2)=O)C1 30589,C(=O)(CCC(=O)C(C)(C)C)N1CCC(C)C1CNC(=O)C(c1ccccn1)O 30590,CCC(C(=O)NCC(C)CNC(c1ccsn1)=O)C(C)O 30591,CC(=O)C(C)(C)CC(=O)N(C)CCN(C1CCN(S(=O)(=O)C(F)(F)F)C1)C 30592,C(=O)(C(C)(F)C(F)(F)F)NC(C1CCN(C(C2(C(=O)NC)CC2)=O)CC1)C 30593,S(=O)(=O)(c1cccc(C(=O)NC23CC(NC(=O)C4=CCC4)(C2)C3)c1)NC 30594,Cc1cc(CCNC(=O)CN(C(=O)CC2CC(C)C2)C(C)C)nn1C 30595,c1(CC(=O)NCC(CC)NC(C(CCC)NC(N)=O)=O)cc(Cl)cc2c1OCC2 30596,Cn1[nH]nnc1=NC1CC2CN(C(=O)C3=CCC(C)CC3)CC2C1 30597,N1(C(C(C(C)(C)C)O)=O)CC2(C(=O)NCCn3ccnc3)CCC1CC2 30598,C1(C(=O)NCC2CC(CN=[N+]=[N-])C2)C2CCN(C(C3(CO)CC=CC3)=O)CC12 30599,c1(C(=O)NCC(c2ccccc2Cl)N(C)C)cccc(NC(C2CCCO2)C)c1 30600,C1(NC(c2n[nH]c(C)c2C)=O)CC2CC(NC(=O)CCn3cccc3)CC2C1 30601,Cc1nc(C(C)C)ccc1C(=O)N(C)CC1(O)CN(C(=O)COc2ccon2)C1 30602,c1(C(=O)NCC(C)N(C)C(c2cnco2)=O)c(F)ccc(N)c1Br 30603,CCC(F)(F)CC(=O)NOCCCC(=O)NCc1sc(C)cc1C 30604,N1(CCCNC(c2cscn2)=O)CCN(C(c2cnn[nH]2)=O)CC1 30605,c1(CC)cc(C)c(C(=O)NC2(C(=O)NCCN3CC4CC4C3)CC2)o1 30606,N1(C(COCC(C)C)=O)CCC(CCCNC(=O)C(F)(F)c2csc(Cl)c2)CC1 30607,C1(F)(CNC(C=C(C)C(C)C)=O)COCCN(C(=O)CC2(CS(C)(=O)=O)CC2)C1 30608,S(=O)(=O)(c1ccc(Br)cc1NCc1cc(Br)cs1)NCC1CCN(CCOC)C1 30609,Cc1cncc(NC(=O)Cc2ccc(O)nc2)c1 30610,C(=O)(CCCCN(C(=O)C(C)(C)C1(O)CCC1)C)NCC(C)CCO 30611,S(=O)(=O)(c1ccc(=NCCCC(F)(F)F)[nH]c1)N(C1CC(C)OCC1)C 30612,c1(C(N2CCCC(NC(C3(COC)CCC3)=O)C2)=O)ccc(C)cc1C 30613,CC(C)C(C(=O)N1CCC(C(CO)NC(C2CC2C(F)F)=O)CC1)NC=O 30614,C1(C(=O)OCC(N2CCCC(N3CCOCC3)C2)=O)CC2(C1)CC(O)C2 30615,c1(NC)ncccc1C(=O)NC1CN(C(c2cn(C(C)C)cn2)=O)CC1O 30616,N1(Cc2cccc(CNC(C)=O)c2)CCC2CCC12CO 30617,c1(C(=O)NCC2C(NC(c3cnc(OCC)nc3)=O)C2)c(F)ccc2nc[nH]c12 30618,C(=O)(C(F)CCC(C)C)N(C1CCN(C(CCC(C)(C)OC)=O)C1)C 30619,N1(C(c2nc(CS(C)(=O)=O)oc2)=O)CCN(C(c2cncc(O)c2)=O)C2(CC2)C1 30620,c1(C(N2C(CNC(C3(C)CC(C)(C)C3)=O)CC(F)C2)=O)ccc(C#N)cc1 30621,Cc1c(C(=O)NC2C=CCCC2C(=O)NCC(C)(C)OC(C)C)nnn1C 30622,c1(C(=O)NCC2CCN(C(C(C)(CO)OC)=O)C2)cc(Cl)c(F)cc1N 30623,CCCCC(=O)C(=O)NCC1CN(C(C2CC23CCOCC3)=O)CCO1 30624,c1(CC(=O)N(C(c2ccccc2)CNC(=O)Cn2nccn2)C)nnc(O)s1 30625,c1(-c2ccc(CC)cc2)ccc2[nH]cc(CC(=O)NCCc3cccs3)c2c1 30626,C1(NC(c2ccccc2)=O)CCN(C(C(=O)N(C(c2ccco2)=O)C2CC2)C2CC2)C1 30627,C=CC1(C(=O)NC(C)CCc2cn[nH]c2)CCN(C(c2ccn(C)c2)=O)C1 30628,c1(C(=O)NC(CC)(CNC(=O)C(Cc2ccsc2)NC=O)CC)ccc(N)cc1Cl 30629,N1(C(C2CC(SC)C2)=O)CC(NC(c2ccccc2SC(F)F)=O)C(F)C1 30630,O(NC(=O)C(CCF)NC(=O)CC12CCCC1C2)C(CC)CC 30631,c1(C(N(C(C)C)CCNC(=O)C(C)CO)=O)ccc2nncn2c1 30632,Cc1nc(C)c(C(=O)NCC2(C(F)F)CCN(C(=O)C(c3ccccc3)F)C2)[nH]1 30633,N1(C(CSC(C)=O)=O)CCCN(CC(=O)Nc2ccc(Cl)cc2)CC1C 30634,c1(C(C(=O)NCC2(CN(C(C(CC)N(C)C)=O)C)CC2)O)cc(F)c(F)c(F)c1 30635,c1(C(N(C(CN(C(C(C)OCC)=O)C)C)C)=O)ccc(CO)nc1 30636,C(=O)(CC(O)CC(C)(C)C)N1C2C(N(C(CCCCCCC)=O)C)CC(C2)C1 30637,C1(C(=O)NCCOCCN(C(=O)C(F)CC2CC2)C)CC2CSCC(C1)C2 30638,C1(NC(C2(C(C)C)COC2)=O)CN(C(=O)CC2OCCC2(C)C)C2(CCC2)C1 30639,C(C(C)(CO)NC(=O)CCCNS(C)(=O)=O)NC(C1C(COC)C1)=O 30640,C1(C(N(CCC(C(C)C)NC(=O)C(C)c2ccco2)C)=O)CN2CCCN1CC2 30641,Cc1cc(C(=O)NC2C(C(=O)NC3CCCC(O)C3)C2(C)C)n(C(F)F)n1 30642,C#Cc1ccc(C(=O)N(CC(O)COC)C)c(C)c1.c12ccc(s1)C(=O)NC2 30643,Cc1c(-c2nc(-c3cccnc3)nn2C(c2ccncc2)C)cnn1C(C)C 30644,C12(c3cc(Nc4c(C(=O)NC5CC5)cccn4)n[nH]3)CC3CC(CC(C3)C1)C2 30645,N1(C(C(C(CC)O)C)=O)CCN(C(c2cc(C)ccc2OCC)=O)C2(CC2)C1 30646,CC1CN(C(C2CCC3(CCC3)OC2)=O)CCCN1C(=O)CC1CC(C2CC2)C1 30647,C12(C(N(CC#CC)CC#C)=O)CC1CCN2C(C1CCCS1)=O 30648,n1(CCS(CC)(=O)=O)c(=NCCc2sc(N(C)C)nc2C)[nH]c2cc(Cl)ccc12 30649,C1(C(C)CO)CCN(C(=O)C(c2ccnn2C)NC(=O)CCN(C)C)CC1 30650,N1(CCC(N2CCC(C)(C)SCC2)=O)C(=O)C2CC=CCC2C1=O 30651,COn1cnc(C)c1C(=O)NCC1CC1NC(c1cc(C)ccc1C1CC1)=O 30652,C1(CCNC(c2ccc(Cl)s2)=O)CCN(C(=O)COc2cccc(O)c2)CC1 30653,C(C(=O)NCC(CO)OCC)(C1CCCC1)NC(COC)=O 30654,c1(C(=O)NCCCCNC(c2ccnc(C)n2)=O)cccc2c1COC2 30655,c1(C(=O)NCCN(C(=O)C(F)CC2CCC2)CC)ncncc1Cl 30656,CC1Cc2ccccc2N1C(C1CC2CCCC2N1)=O 30657,N1(C(C(CC)NC(N)=O)=O)CCN(C(c2n[nH]c(O)n2)=O)CC1c1cnn(C)c1 30658,n1(CC)cc(CN2CCC(CC(N3CCCC(CN(C)C)C3)=O)C2)c(C)n1 30659,c1(CC2CN(S(C)(=O)=O)C2)nc(-c2ccccc2)nn1-c1cnn(C)c1 30660,c1(OC)ccc2nc(C)c(C(=O)NCC3CCC3NC(=O)Cc3ccsn3)n2n1 30661,C1(NC(c2c(COC)cccc2)=O)CN(C(=O)Cc2ncccc2C)CCC1C 30662,C1(NC(C(c2cccs2)NC(c2cc(C)sc2C)=O)=O)CN2CCC1(C)CC2 30663,Cc1cnc(C(=O)NC2CCN(C(=O)C(=CC3CCCCC3)F)C2(C)C)cc1C 30664,Cc1ncc(C(=O)NC2(C)CCCN(C(c3c[nH]c(Br)c3)=O)C2)c(=N)[nH]1 30665,c1(C(=O)NC(C2CCCCN2C(=O)COc2cccnc2)C)cccc(N)c1O 30666,N1(C(Cc2nc(C)[nH]n2)=O)CCCC12CCN(Cc1nnnn1C1CC1)CC2 30667,C(=O)(CC(CCC)NC(C1CCCC(=O)N1C)=O)Nc1ccc(OCC=C)cc1 30668,C1(C)(C2CCCN(C(C(=O)NCCCOC)c3cccs3)C2)NC(=O)NC1=O 30669,C1(NC(=NCCSC)NCCc2cccc(O)c2)CCOC2(CCSC2)C1 30670,N1(C(c2ccn(C(C)C)n2)=O)CCC=C(C(=O)N2CC3CCC2C3)C1 30671,n1(CC)ncc(CNC(N2CC(CC(=O)OC)C2)=O)c1C 30672,c1(C(N2CCCCC(NC(C(CCC)C#N)=O)C2)=O)noc2ncccc12 30673,c1(-c2onc(-c3cnc(-c4cccc(F)c4)o3)n2)cc2c[nH]nc2s1 30674,N1(CCN(C)C(C2CN3CCCN2CC3)=O)CCc2ccccc2C1 30675,C1(C(=O)O)C=CCN(Cc2ccc(N3CCCC3)nn2)C1 30676,c1(C(C(=O)N2CC(N(C(Cc3cnc(C)[nH]3)=O)C)C2)(F)F)cccc(F)c1F 30677,CC1CN(C(=O)CC2CCC2)C(C)C1C.C(=O)(C(C)N(C1CCC1)C)OC(C)=O 30678,c1(C(N2CCCC2)=O)ccc(Cl)c(S(=O)(=O)N2C3CCCC2CC(O)C3)c1 30679,C1(C(N)=O)C2CC3CC(C2)CC1(C(NC1CCCc2occc21)=O)C3 30680,C1(OC)(CNC(C2(C)CCCCCC2)=O)CCN(C(c2[nH]c(O)nc2C)=O)CC1 30681,CC1(C#CC(=O)N2CCC3C(C2)CN3C(c2nccc(C(F)(F)F)n2)=O)COC1 30682,C1(CC)CCCC2CN(C(c3ccc(C)o3)C(=O)N(C)Cc3ccccc3)CC12 30683,C1(NC(=O)CC2CCOC2)CCCCN(C(=O)Cc2c(O)ncnc2O)C1 30684,C1(C(=O)NCCOCCCNC(=O)Cc2ccco2)CS(=O)(=O)CC12CCC2 30685,C(C)(CC(=O)N1CCC(NC(C2CCCCC2)=O)C12CCC2)(C(F)F)N(C)C 30686,c1(CN2C(CNC(C3CC3C3CC3)=O)COCC2)cccc(CO)c1 30687,c1(-c2sc(C(N(Cc3c(C#C)cccc3)CC)=O)c(C)n2)ccc(F)c(C#N)c1 30688,c1(C(N2C(C(C)C)CN(C(=O)C(F)(F)CF)CC2)=O)ccc2c(n1)OCCO2 30689,C#Cc1cn(C)nc1C(=O)NC1CCCC(C(=O)NC(c2ccns2)C)C1 30690,C1(C(F)(F)F)(OC)CCCN(C(=NCc2ccc(C)cc2C)NC(C)C)C1 30691,C(=O)(C1=CCC(NC(C2(C)CCOC2)=O)C1)N(CC#CC)CC#C 30692,CCC(O)(C(=O)NCC1CC2CC2N1C(C1OCCO1)=O)c1ccccc1 30693,C1(NC(c2cc(C)no2)=O)CCC2CN(C(c3cncc(C(C)C)c3)=O)CC2C1 30694,CC1CCCCN1CC(N1CCC(CCC(=O)NCCC(O)C2CCC2)CC1)=O 30695,c1(C(N2CCC(C(C)NC(CCCSC)=O)C2)=O)sc(C)cc1Cl 30696,C1(SCC)CCC(NC(c2c[nH]nc2-c2ccccc2Cl)=O)CC1 30697,c1(CCNC2CC(CSC)C2)nc(O)c2c(C)c(C)sc2n1 30698,N1(C(CCOCCOC)=O)CCC(CC(=O)NCC2CCC2C)C1 30699,c1(C(N2C(C)CCN(C(c3c(C(C)=O)ccs3)=O)CC2)=O)cc(C)c2[nH]cnc2c1 30700,c1(C(=O)NC2CCN(C(c3c(C)ncn3O)=O)CC2)cnc(C2CC2)[nH]c1=N 30701,c1(SC)ccc(NC(c2cc(-c3ccc(NC(C)=O)nc3)[nH]n2)=O)cc1 30702,N1(C(c2c(C(C)C)ccc(C)c2)=O)CC2CC(NC(c3cc(Cl)c[nH]3)=O)CC1C2 30703,N1(C(CNC(CC(C)O)=O)C)CCN(C(C2CCN(S(C)(=O)=O)CC2)=O)CC1 30704,C12(NC(c3c(OC)ncnc3C)=O)CC(CNC(=O)CCC3CC3)(C1)OC2(C)C 30705,C1(C(=O)NC2CCN(CC)C2)CCC(CNC(C2C3COCC23)=O)CC1 30706,C1(OC)(OC)CC(C)(C(=O)NC(C)CNC(=O)C=CCO)C1.C(C(C)(C)C)OC 30707,c1(C(=O)NC2(C3N(C(c4nncc(OC)c4)=O)CCC3)CC2)c(Cl)cccc1Cl 30708,c1(SC)cc(C(=O)NC(C)(CNC(=O)CCc2ccccc2)C2CCC2)c(C)o1 30709,c1(CCCC(=O)N(C2CCN(C(CC=C(C)C)=O)C2)C)ccccc1Cl 30710,CCC(CC(C)C)C(=O)N1CCC(NC(C2CCCO2)=O)C(OC)C1 30711,c1(C(=O)NCCCC2N(C(CCCCOCC)=O)CCC2)c(Cl)cncc1Cl 30712,Cc1cc(NC(c2cc(CNC(c3cc(CO)ccn3)=O)on2)=O)c(=O)n(C)c1 30713,N1(C(C(CCCC)O)=O)CC(CNC(=O)C(=C2CCCCC2)F)OC2(CCC2)C1 30714,N1(C(CCc2onc(CC)n2)=O)CCC(O)(CN(C(=O)C(C)CC2CCC2)C)C1 30715,c1(NC2CCN(C(C=C)C)CC2)ncc(S(=O)(=O)N2CCCC(C)C2)cc1Cl 30716,CCC(CCOC)C(=O)NCCC1CCCN1C(c1c(NC(C)=O)c[nH]c1C)=O 30717,C1(C(=O)NCc2c(C)nco2)C2CC2CN1C(=O)CC1COCCO1 30718,C(CC#CC(C)(C)C)NC(CC(CC)N(C(=O)CCC1(C#N)CCC1)C)=O 30719,Cc1cc(C(=O)NC2CN(C(C3CCOC(=O)CC3)=O)CC2C)cc2nc[nH]c12 30720,c1(SCC(=O)NCCC2COCCN2C(C2CCCCS2)=O)cccnc1Cl 30721,Cc1cc(Cl)cc(C)c1OCCNC(=O)NCc1ncnc(C(C)(C)C)n1 30722,c1(NCC(C)S(C)=O)ncccc1S(=O)(=O)NCCCc1ncco1 30723,c12nnc(n1Cc1ccc(Br)s1)s2.O=C1CCCN1C1CCCN1C1CC1 30724,Cc1ccc(C(N2CC3(CCC3NC(=O)CC3CC4(CCC4)C3)C2)=O)cc1C#N 30725,CN1CCCC(CNC(C2CSCCN2C(c2ccc(C#N)cn2)=O)=O)C1=O 30726,c1(C(=O)OCc2c(COC)nccc2)cc2ccc(C)cc2o1 30727,C1(C)(CNC(C(C2CCOC2)OC)=O)CCN(C(C23CCN(CC2)CC3)=O)CC1 30728,C1(CC(N2CCN(C3CCN(C(=O)C(F)C4CC4)C3)CC2)=O)CCCCC1(F)F 30729,C(=O)(C(C)CC(F)F)NC1CC(C(C)NC(c2ccn(CCC)n2)=O)C1 30730,CCC(C)C(=O)N(C(CNC(C1CC2CC2C1)=O)C1CC1)C 30731,c1(-c2cccc(CCC(C)=O)c2)ccc(S(=O)(=O)NCC2(O)CC2)cc1 30732,C1(NC(c2n(CC)ccn2)=O)CCCN(Cc2nnc(CCOC)s2)C1 30733,C(=O)(N=c1nc[nH]n2cccc12)C1N(C(Cc2cccc(NC(C)=O)c2)=O)CCC1 30734,C(=O)(C(C)=NOCC#N)NCCC(C)N(C(C(C1CCCC1)OCC)=O)C 30735,CCC1=C(C(=O)NCC2CCN2C(C2CCc3n[nH]c(C)c3C2)=O)CCCO1 30736,C1(NC(c2c(OCC)scc2)=O)CS(=O)(=O)CC1NC(c1c(C)ncn1O)=O 30737,N1(C(C(C)OC(C)(C)C)=O)CC(C2CN(C(=O)CSC3CCCCO3)C2)C1 30738,C1(COC)(NC(=O)C(F)CC2CCCC2)CN(C(=O)Cn2cc(Cl)cn2)C1 30739,CCC(CCC(=O)NCCSCC(=O)NCCc1n[nH]c(C2CC2)n1)OC 30740,Cc1c(O)ccc(C(=O)N(CCCNC(=O)CC(C)CN(C)C)C2CC2)c1C 30741,C1(C)(C(=O)NC2CC(CNC(C(C)OC3CCCC3)=O)C2)CCC(F)(F)CC1 30742,c1(CC(=O)NC(CCCCNC(C2(C)ON=C(C)C2)=O)C)c(C)nc(O)nc1C 30743,c1(OC)cc(CN2CC3(CC(C(=O)Nc4cn(C)cn4)C3)C2)cc(F)c1 30744,C(CCCCCC(=O)NCC(O)C1(Cl)CC1)NC(CC(COC)C)=O 30745,C(CC(=O)NCC1C(C)CCN1C(=O)CSCCN(C)C)(C(F)(F)F)OC 30746,CCCC(CSc1nc(C(F)F)nn1CC(C)(C)C)C(=O)O 30747,O=C(N=c1ccn(Cc2ccc3c(c2)CCO3)[nH]1)C(F)(F)c1ccc(Br)cc1 30748,N1(C(C2C(C)CCC2)=O)CC2(CC2)CC1CNC(=O)Cn1cncn1 30749,CC1(C(=O)NCCOCCNC(C2CCCCNC2=O)=O)CCCNC1=O 30750,C1(CNC(CC(C)n2cccn2)=O)C2CN(C(=O)CCc3nc(=N)[nH][nH]3)CC12 30751,C(=O)(CCCCCCCC=C)NC(CC#C)C(=O)NCCN1CCC(O)C1 30752,c1(CCN)cc(C(N2CC(F)(c3cccnc3)C2)=O)no1 30753,C(=O)(C1=NNC(C(F)(F)F)C1)N1CC(C)(NC(C(C(C)O)C)=O)C1 30754,c1(C(=O)OC)ccc2c(C(=O)NCCOCCOc3ccccc3F)ncn2c1 30755,C(=O)(C1c2ccccc2CN1C(c1cnc(O)c(Cl)c1)=O)NC1CC(=O)NC1 30756,Cc1nc(C(N2CCC(CC(N3CCC(C(C)(C)O)C3)=O)C2)=O)c(C)s1 30757,C1(NC(N(C)C2CC2)=O)CCN(C(=O)C#N)CCC1CO 30758,c1(C(=O)NCC#CC(=O)NCc2onc(COC)n2)cnnc(C)c1C 30759,c1(C(=O)NCC(CNC(CC(CC)CC)=O)OC)ccc(F)c2ccoc12 30760,CCCC(CCCNC(=O)CC(c1ccc(F)cc1)C)NC(C)CC(N)=O 30761,C1(C(N2CC(C)CC(CC)C2)=O)(CC)CCCN(C(=O)CC#N)C1 30762,C1(C(=O)Nc2ccc(OC)c(-c3ccccc3)c2)CCC(C2CC2)CC1 30763,N1(C(=O)NCCN2CCC(C)(C)C2)CCC(CCCc2ccccc2)C(CO)C1 30764,N1(C(C(C(C)C)SCC)=O)CC(NC(c2cnnn2C(C)C)=O)CC1(C)C 30765,c1(C(N2C(C)(C)C(CNC(=O)CCC3CC3(F)F)CC2)=O)cc(F)c(O)c(F)c1 30766,c1(C(=O)NCC2N(C(c3cccc(S(C)=O)c3)=O)CC2)cc2c(s1)CCCCC2 30767,c1(C(=O)NCCC2(NC(C3C(c4cn(C)nc4)C3)=O)CC2)ccnc2ncnn12 30768,C(CC(F)F)(C(=O)NC1CC2(CCCC2)C1)NC(Cc1c(CC)con1)=O 30769,c1(C(=O)NC2CN(C(c3cccc(C(C)C)n3)=O)C2)[nH]nc2cnccc12 30770,c1(OC)cccc(C(C(=O)Nc2cccc(C)c2)NCCc2ccccc2)c1C 30771,c1(NCCC2(O)CN(C(C(CC)SC)=O)C2)ncc(Br)cc1[N+](=O)[O-] 30772,C1(C)(C(=O)NCCCN(C(=O)CC2(C#N)CC2)C)CCC(=O)N1 30773,CC1(C2CC2C(=O)N(CCNC(c2ccc(C(F)(F)F)nc2)=O)C2CC2)COC1 30774,NS(=O)(=O)N1CCCC(C(=O)NC2(C3CN(C(=O)CCC(N)=O)C3)CC2)C1 30775,NS(=O)(=O)c1ccc(O)c(C(=O)NC2CC(NC(c3nn[nH]c3Cl)=O)C2)c1 30776,C1(C(=O)Nc2ccc(CSCC)cc2)CC2(CC2)CN1C(C1CCCC1)=O 30777,C1(C(NOCC)=O)CCN(C(=O)C(C(C)C)C2CCC2)C1C(C)C.C1CC(=O)N1 30778,C(c1cccc(CN2CCC(c3nn[nH]n3)C2)c1)=CC(=O)Nc1c(C(C)C)n[nH]c1 30779,S(=O)(=O)(c1cnccc1N1CCc2c(C)cccc2C1)N1CCC(OCC)CC1 30780,CC1(C)CC=C(C(=O)N2CCC3(CCCN3C(c3ncoc3C3CC3)=O)C2)CC1 30781,C(CC(C)(C)C(=O)NC1(C)CSC1)NC(c1cn(CC)nn1)=O 30782,CCC(C(=O)NC1(C2CCN(C(c3cc(N)cc(O)c3)=O)C2)CC1)C(F)(F)F 30783,N1(CCCNC(C(CC)C)=O)CCN(C(=O)CN2CCC(C)(O)C2)CC1 30784,Cc1[nH]c2ncnc(N3CCC(NC(C4(C)CC=CCC4)=O)C(O)C3)c2c1C 30785,C1(C)(CC)CCCN(C(C2CCC(O)CN2C(=O)CC2CCOC2=O)=O)C1 30786,N(C(=NCCc1ccncc1C)NC1CCS(=O)(=O)C1)C1CC(OC)C1 30787,C(=O)(CS(=O)(=O)C1CCCC1)N(C(C)Cc1cc2ccccc2o1)C 30788,c1(C(N2CCOC(CCNC(C3CC(C(F)F)C3)=O)C2)=O)ccc2nnnn2c1 30789,C1(NC(C=CCCC)=O)CN(C(=O)C(c2cccc(C)c2)(C)C)CC1O 30790,C1(NC(C(CC)OCC)=O)CC(NC(c2csc(C(C)C)n2)=O)C(O)C1 30791,C=CC1(C(=O)O)CCN(C(=O)C(C2CN(C(=O)OC(C)(C)C)CCO2)C)C1 30792,Cn1cc(CC(O)C(=O)NCCCOCCNC(=O)C=Cc2cnc[nH]2)cn1 30793,C1(NC(c2ccn(CCC)n2)=O)CC12CC(NC(c1cc(C3CC3)on1)=O)C2 30794,c1(C(=O)NC(C2CCN(C(=O)C(F)=C3CCC3)CC2)C)ccc(N)cc1[N+](=O)[O-] 30795,C1(C(N2CCC(C(C(=O)NCC3(OC)CCCC3)C)C2)=O)CCCCN1C 30796,C(=O)N=c1nc2ncc(Cl)cn2[nH]1.c1(C(C)(C)C)cnc(C2CCC2)o1 30797,n1(CC)nc(C)c(CC(N2CCCCC2C(C)NC(=O)CC2=CCCC2)=O)c1C 30798,N1(CCC=CCC)CCC2C(CCCN2C(c2cnn(C)c2)=O)C1 30799,Cn1c(=O)oc2c(C(=O)NCC(CNC(c3ccnc(O)c3)=O)CO)cccc12 30800,OCC1CN(c2nccc(N3CCC(F)(CF)C3)n2)Cc2ccccc21 30801,N1(C(C(C)n2cnnn2)=O)CC(CNC(=O)Cc2ccsc2)CC(C)(C)C1 30802,N1(C(C(C)NC(C)=O)=O)CC2(CCN(C(=O)C(F)=C(C)C)CC2)CC1C 30803,c1(C(=O)NC(CNC(c2cc(CC)c(CC)o2)=O)CO)ccn2cncc2c1 30804,N1(C(c2c(C)cns2)=O)CCC(Cn2cc(CNC(=O)C(C)C(C)C)nn2)CC1 30805,c1(NC(C2CCC(OCC(=O)NC)CC2)=O)cccc(F)c1C(F)(F)F 30806,N1(C(c2cc(CCC)on2)=O)CCC(O)(CN(C)C(C2CCN(C)C2C)=O)C1 30807,C1(NC(C(COC)C)=O)COC2(CCN(C(C3CN4CCN3CC4C)=O)C2)C1 30808,N1(C(c2cn(CC(CC)O)nn2)=O)CCC2CCN(C(=O)CN=S(C)(C)=O)C2C1 30809,S(=O)(=O)(C(F)(F)F)NCC1C(NCCC(=O)Nc2cn[nH]c2)COC1 30810,N1(C(CC(C)n2ccnc2)=O)CCC2(CC1)CC2NC(C1(C(C)(F)F)CC1)=O 30811,c1(C(=O)NC2CC(CNC(CCCC)=O)C(O)C2)ccc2oc(=N)[nH]c2c1 30812,C12(NC(c3coc(O)n3)=O)CCCCCC1N(C(c1cc(C3CC3)n[nH]1)=O)CC2 30813,CC#CCCC(=O)N1CCC(C(N2CCC2C(=O)OC)=O)O1 30814,N1(C(=O)CCN(C(c2ccco2)=O)C2CC2)CC2(CCC2O)C1 30815,n1(CC(=C)C)nnnc1C(c1csnc1OC)NCCn1cccn1 30816,CCCCCCC(=O)NC1(CC(N2CCC3CC2C(=O)O3)=O)CCC1 30817,c1(NC(=O)OC(C)C)cc(NC(C)CC#N)ccn1 30818,C(=O)(CCS(N)(=O)=O)NCC(C(C)(C)C)NC(CCC(C)SC)=O 30819,c1(C(CC)N(C(c2cc(C)[nH]n2)C(=O)NC2CCC2)CCC)ccccc1Cl 30820,C(C(=O)NC(C)(CO)C(=O)NC(C)Cc1nn[nH]n1)(C(C)C)SC 30821,C1(CN(C2CCN(C(=O)CN3C(=O)CCC3=O)C2)C)COc2ccccc2O1 30822,C1(C(C#C)NC(=O)N(CCCN(C)C)C)CC(F)(F)C1 30823,S(=O)(=O)(c1cc(F)c(OCC)cc1OC)C1CC(C)(CC)C1 30824,C1(CNC(c2ccoc2Br)=O)CCCCC1NC(C1(C2CCCO2)CCC1)=O 30825,c1(N2CCC(Nc3c(C(=O)OC)c(C)sc3)C2=O)cc2ccccc2o1 30826,Cc1ccn(C)c1C(=O)NCCC1CCCN(C(C2(O)CCCCC2)=O)C1 30827,N1(C(c2ccnnc2C(F)F)=O)CCCS(=O)(=O)CC1c1ccccc1 30828,C(=O)(C(O)C(F)(F)F)NCC(CCC)NC(C1CCCN(C)C1)=O 30829,c1(CN2CCC(CNC(CSCC)=O)C2c2cccnc2)cc(Cl)c(F)c(Cl)c1 30830,c1(OC)ccc2c(c1)C(C(=O)NCC1C(NC(c3ccoc3C3CC3)=O)C1)CC2 30831,C1(C(=O)NCC2(C)CCN(C(C=COCC)=O)C2)CCC12CCOCC2 30832,N1(C(c2cn(CCOC)nc2)=O)CC(NC(c2ccoc2C)=O)C(O)C1 30833,c1(C(N2C(C)C(NC(C3C(C)(C)C3(C)C)=O)CCC2)=O)cc2c(cc1O)OCO2 30834,N1(C(C(C#C)(C)C)=O)CC2CC(NC(=O)CCc3cncc(O)c3)C(C2)C1 30835,c1(C(=O)NC2(C(=O)NCC(C)(C)CN=[N+]=[N-])C(C)CCC2)ccn2nccc2c1 30836,c1(C(=O)NC(CCN(C(c2ccc(SC)o2)=O)C)C(C)C)c(C)ccc(C)c1N 30837,C1(C(=O)NC(C(N2CCC2(C)CCO)=O)C2(C)CC2)CC=CC(O)C1 30838,C12(CNC(=O)C=C(Cl)Cl)CCC(CC1)CN2C(c1cc(C(F)(F)F)cc(O)c1)=O 30839,CC1CCN(C(c2cc(C(F)(F)F)cs2)=O)CCN1c1ncc(I)cn1 30840,Cc1c(F)ccc(C(=O)NC2CCCCC2NC(C2(O)CCCC2)=O)c1Cl 30841,c1(C(=O)NC2CC(C)N(C(=O)C3=CCOCC3)C2)c[nH]c(=N)nc1O 30842,Cc1cnncc1C(N1CCC(NC(C2CC23CCC3)=O)CC1)=O 30843,N1(C(C(C)OCCCCCC)=O)CC(NC(c2ccnnc2C)=O)CC(C)(C)C1 30844,N1(C(c2c(C)coc2C)=O)CC(O)(C2(CNC(=O)Cc3cc[nH]n3)CC2)C1 30845,C1(CNC(C(CN(C)C)(F)F)=O)CC2CCC1N2C(C1(C2CCCO2)CCC1)=O 30846,CCCCCC(O)C(=O)NCC1CN(C(c2cnc(NC)cn2)=O)CC12CCC2 30847,n1(COC)ccc(C(=O)NCCCOCCC(=O)NCCc2noc(C)n2)n1 30848,C1(CNC(C(CC)=CCCC)=O)CN(C(=O)COC)CCN1C 30849,N1(C(CC(C)C(F)F)=O)CCOC2(C1)CN(C(=O)CCOc1ccccc1F)C2 30850,C=CCCC(CO)NC(=O)C(O)C1CN(C(c2cn(C3CC3)nn2)=O)C1 30851,c1(OC(C(=O)N(CC(CNC(C=CCCC)=O)(C)C)C)C)ccc(Cl)cc1 30852,n1(CC)cc(CC(N2CCCCC2CCCNC(=O)CC(C)(C)O)=O)c(C)n1 30853,C(c1ccncc1)=C(C(=O)NC(CCN(C(C(CC)F)=O)C)C)C 30854,c1(C(=O)NCc2ccc(-c3ccc(SC(C)C)cc3)cn2)c(O)ccc(F)c1F 30855,C(=O)(C(CO)NC(c1[nH]ccc1CNC(=O)CC12CCCC1C2)=O)N(C)C 30856,C1(SC(C)C)CCN(C(=NCC2CC3(CCOCC3)C2)NC2CCC2)C1 30857,c1(C(C(C(=O)N(C)CCOc2ccc(C(F)(F)F)cc2)N)=O)ccc(F)cc1F 30858,C1(C(=O)OC2CC3CC3C2)(OCC(=O)OC)CC(C(F)(F)SC)C1 30859,c1(OC)cc(C)c(Br)cc1C(N1CCC2(CC2C(=O)Nc2cc(O)ncn2)C1)=O 30860,N1(C(CC(COC)NC(=O)CCC(=O)N(C)C)=O)CCN(C)CC1CCO 30861,CON(CCC(=O)N1CC(C2CC2)(OCC)C1)C(=O)C1CCC(C)(C)CC1 30862,C(CC(=O)N1CCC(OCC(N)=O)C1)(C(F)(F)F)NC(C1C(C)(C)C1(F)F)=O 30863,N1(C(C2C(CC)CCC2)=O)CCC(CO)(CNC(C2CCC(=O)N2)=O)CC1 30864,c1(C(=O)NC2(CN(C(C3CCN(C(=O)NC)C3)=O)C)CC2)ccn2nccc2n1 30865,C=C1CCN(C(=O)C(C)OCCC)C(C(=O)N(C2CC(C)(C)C2)C)C1 30866,Cc1nc2c(s1)CCCC2C(=O)NCC1(CNC(=O)C(C)SC(F)(F)F)CC1 30867,c1(C(=O)NCC(CC)(C)NC(=O)CC2CCNC(=O)C2)oc(C)cc1C 30868,c1(C(=O)NCC2N(C(C=CC(=O)N(C)C)=O)CCC2)c[nH]c(=O)c2ccncc12 30869,C(CCC1CCC1)(C(=O)NCc1cnn(C)c1O)NC(c1c(C)ocn1)=O 30870,c1(C(=O)NCC(CC)NC(=O)C(C2CCCCC2)F)ccc2nnnn2c1 30871,c1(C(=O)NC2CC(N(C(CCC(=O)NC)=O)C)C2)cc(N)nc(Br)c1 30872,C(C(=O)N(CC)OC)NC(C(CNC(CC1C(CC)C1)=O)C)=O 30873,c1(C(=O)NC2C(NC(CCc3nnc(C)o3)=O)CCC2)cc(N)c(F)cn1 30874,N1(C(C2CNC(=O)N2)=O)CCCC2(CCN(C(c3cnco3)=O)C2)C1 30875,C(=O)(C1CCc2cccc(F)c21)NC(CC)CNC(=O)Cn1ccc(=O)cc1C 30876,C=CC1(C(=O)NC2CCCCC23CC3)CCN(C(=O)Cc2cscn2)C1 30877,CCC(C)CCCCC(=O)NCC(C)CNC(=O)C(n1cc(C)cn1)C 30878,N1(C(c2ccn(CCC)n2)=O)CC2CCC(C1)N2C(c1cnc(C2CC2)s1)=O 30879,c1(C(=O)NC2CCC(CCNC(C(C(C)C)C)=O)C2)nn(C)c(Cl)c1Br 30880,N1(C(C(CC)OC2CCCCC2)=O)CC(OC)CC(NC(=O)COC)C1 30881,C(=O)(C(COC)COC)N1CC(CC=C)(C(=O)NC2CCC(N(C)C)C2)C1 30882,C(=O)(C(CC(C)C)n1ccnc1)NCc1nc(SC)nn1-c1cccc(F)c1 30883,C1(C(C(=O)NCC(CC)NC(C2(C)COCCO2)=O)(C)C)CCCCCC1 30884,c1(C(=O)NCC(CC(C)C)NC(=O)C(c2ccccc2)O)csc([N+](=O)[O-])c1 30885,C1(CNC(C(c2cn(C(CC)C)nn2)(C)C)=O)CCN(C(=O)C(F)Br)CC1 30886,C(C(=O)NCC#CC#CCO)(C(C)(C)O)NC(CCCCSC)=O 30887,N(C(=NCCc1cnc(C)cn1)N1CCC(CS(C)(=O)=O)C1)CC(=C)C 30888,C1(NC(COCCN(C)C)=O)CN(C(C2CCCC23CC3)=O)CC12CCOCC2 30889,N1(C(C2CCCC2C)C(=O)NC(CC)C)CCOc2c(OC)cccc21 30890,C(=O)(C(C)(CC)CC)NC(CNC(Cc1c(SCC)cccc1)=O)CCOC 30891,c1(NC2CCC(C(=O)Nc3cnc(C)c(Cl)c3)CC2)nccc(S(C)(=O)=O)n1 30892,c1(N2CC(C)C(NC(c3cnc4n3CCC4)=O)CC2)ncc([N+](=O)[O-])cc1Cl 30893,c1(NC(CN(C(CCc2n(C)c(S)nn2)=O)CCO)=O)cccc2c1SCCC2 30894,N1(C(c2cc(C(=O)OCC)n[nH]2)=O)CCCC1(C(=O)OC)COCC1CCOCC1 30895,c1(CN(CCOCC)C)ccc(Br)c(Cl)c1.C(=O)NC(C)C.C1C(=O)N1 30896,N1(C(C(CC)c2ccccc2)=O)CCN(C(c2n[nH]c(C)c2O)=O)C2(CCC2)C1 30897,N1(Cc2cnn(C)c2Cl)CCc2cc(NS(=O)(=O)c3cccc(Cl)n3)ccc2C1 30898,CC1CCC(NC(c2c[nH]ccc2=N)=O)CN1C(c1csc(-c2nc[nH]n2)n1)=O 30899,C1(NC(CC(C=C)CCC)=O)CCC2(CCCN(C(=O)CCCC(=O)OC)C2)C1 30900,CC1CN(CC(=O)NCC23COC(C2)C(O)C3)C(C)CC(C)O1 30901,c1(C(N2CCC(CC=C)(NC(=O)C(CC)=CC)C2)=O)c(C)cccc1[N+](=O)[O-] 30902,C(=O)(C1CCCc2nn[nH]c21)N1C(C)CC2CN(C(c3c(C)coc3C)=O)CC21 30903,N1(C(CCCC(C)=O)=O)CC2CCCN(C(=O)CC3(C)OCCO3)C2C1 30904,N1(C(c2c(OC)nsc2)=O)CC(CC(N2CCC2(C)C(C)C)=O)C2(CC2)C1 30905,c1(CC)cc(C(=O)NCCCCCNC(=O)C(CC)n2nccc2C)c(C)nn1 30906,C1(NC(C(C)C)=O)CCN(C)C12CCCN(C(=O)C=CCO)C2.C12CCC1CC2 30907,c1(C(=O)NC2CN(C(c3cc(OC)cc(F)c3)=O)CC2F)cc(Cl)c(F)cc1F 30908,n1(COC)cc(C(=O)NC2CCC(SC)C2)c2ccccc12.C12CN(C1)C2=O 30909,N1(C(C2(CCOCC)CCC2)=O)CC(N(C(=O)C(N)=O)CC)CC(C)C1 30910,N1(C(c2c(CC)nccc2)=O)CC2(CCN(C(C3CCN3CC)=O)CC2)C1 30911,c1(N2CC(C)(CC3CC4(CCOCC4)C3)C2)ncc(C#N)cc1C(F)(F)F 30912,C(=O)(CCN=C(NCc1cccc(SC)c1)N1CC(=O)N(CCCOC)C1)NC 30913,c1(OC)cc(C(=O)NCC2CCCCN2C(c2nccnc2Br)=O)ccc1O 30914,C1(C)(C(=O)NC2(CNC(C(COC)O)=O)CC(OC)C2)CC2(CC2)C1 30915,C(CC(=O)NCC(C)(C1CC1)NC(=O)C=CCO)C1(C)N=N1.C(C)(C)(C)OC=O 30916,Cc1ccc(F)c(NC(=O)Cc2cccc(NC(c3cc(C)cc(Cl)c3)=O)c2)c1 30917,N1(C(CN(C)CC)=O)CCC2C(CCCN2C(c2cc3nc[nH]c3cn2)=O)C1 30918,N1(C(c2c(C)nc(N)cn2)=O)C2CCC1CN(C(c1cncc([N+](=O)[O-])c1)=O)C2 30919,c1(C(=O)NCCC(C)NC(=O)CCc2nc(O)n[nH]2)c(F)ccc(F)c1N 30920,C1(CNC(c2c(C)n[nH]c2C)=O)CN(C(c2cc(CC3CC3)on2)=O)CCCO1 30921,C1(CNC(CC2C(CC)C2)=O)CCCC1NC(c1snnc1C1CC1)=O 30922,N1(C(C(C)(C)C2CCC2)=O)CCC(NC(=O)CC=CC(=O)O)CC1 30923,CCC(CC(=O)NCCC(C)(CC)NC(=O)Cc1ccccc1C)SC 30924,c1(C(N2CC3C(C(=O)NC(C(CO)N(C)CC)C)C3C2)=O)ccc(O)cc1C 30925,c1(SC)cccc(C(=O)NC2CCCN(C(=O)C(C)(C)CC(F)F)C2)c1[N+](=O)[O-] 30926,N1(C(CCOCCOC)=O)CCC2(CC1)CC2(CO)NC(=O)CSc1cccs1 30927,CC1(C)CC(CNC(c2cncc(Cl)n2)=O)N(C(=O)CCC2COC(C)(C)O2)C1 30928,c1(C(=O)NC(C2CCCCN2C(=O)Cc2cocn2)C)nn(C)c2c1COCC2 30929,C(=O)(C(C)(F)C(=O)NC1CC(CNC(c2cc(Cl)cc(Cl)c2)=O)C1)OC 30930,N1(C(CNC=O)=O)CCN(C(C2CCCC23CCC3)=O)C2CCC12 30931,C(C1=CCN(C(=O)CC2CCC3CC3C2)CC1)NC(C(C)n1cccn1)=O 30932,C1(NC(c2ccsc2Cl)=O)CN(C(=O)C(F)=CC2CC2)CC12CCOCC2 30933,N1(C(CSCCCN(C)C)=O)CCN(C(C2(C3CCCCO3)CC2)=O)C2(CC2)C1 30934,C1(C(=O)NCC(N)=O)CC(NC(c2cccc(OCC(=O)O)c2)=O)C12CCC2 30935,c1(C(N2C3(CNC(CC(CC)O)=O)CC(C2)C3)=O)cc2cc(C)cc(C)c2[nH]1 30936,C(CS(=O)(=O)CC(=O)NC1CC1CNC(c1nc(C)c(C)nc1C)=O)OC 30937,c1(CC)cc(C(=O)NC(CC2CCC2)C(=O)NCCCc2cn[nH]c2)nn1C 30938,c1(C(=O)NC2C(NC(C(CC(C)C)NC(C)=O)=O)CCCC2)cc2ncccc2s1 30939,Cc1c(N)c(C(=O)NCC2CCCCN2C(=O)CC(C)c2ccccc2)nn1C 30940,N1(C(c2cc(C)cc(F)c2)=O)CC(C)CN(C(C2COC3COCC23)=O)CC1C 30941,CC1CCCCCC1(c1nnnn1CC(F)F)NC1(c2cccc(F)c2F)CC1 30942,N1(C(C(CC=CC)NC(C2CC2CC(C)(C)C)=O)=O)CCC2(C=CCO2)CC1 30943,C=C(Cl)C(C)(C)C(=O)N1CC(NC(c2cnccc2Cl)=O)C(C(F)(F)F)C1 30944,C12(CC(=O)NCCNC(c3c(CCC)onc3C)=O)CC3CC(CC(C3)C1)C2 30945,Cc1ccc(C(=O)NC(C)(C)CNC(=O)CC2CC(O)C2(C)C)c(F)c1Br 30946,CC1CC(NC(N2CC(CO)C(CO)C2C(F)(F)F)=O)C(=O)N1c1ccccc1 30947,C#CCCCCCC(=O)N1CC2CN(C(C3CC(=O)N(CC(C)C)C3)=O)CCC12 30948,C(=O)(C(C)(CC)CC#C)N1CC(CCNC(CC2(OCC)CCC2)=O)C(C)C1 30949,c1(COC)ncc(C(=O)NC(CCN(C)C)C(=O)NC2CC3(CC3)C2)cn1 30950,c1(C(N(CC=CC(=O)N(C2(COC)CC2)C)C)=O)ccc([N+](=O)[O-])o1 30951,C(C)(C)(C(=O)NCCC(C)(C)NC(=O)C(C)Sc1nnnn1C1CC1)OC(C)=O 30952,c1(C(N2CC(C)C(NC(=O)C(c3ccc(F)c(F)c3)O)C2)=O)nc(Cl)ccc1N 30953,O=C(C1CCCc2nccn21)NCC#CCNC(C12CCC(CC1)C2)=O 30954,c1(C(=O)NC2CCCC(NC(C3CC4(CC4)C3)=O)C2)c[nH]c(=O)c2ccnn12 30955,N1(C(C(CC=C)N(C)C)=O)CCC(C2CC2)C1CNC(=O)Cc1ccc(F)cc1 30956,c1(NC)c(C(=O)NC2CCC2CCNC(=O)C(C)C(C)(F)F)cccc1F 30957,c1(C(N2CC3(CCN(C(C4C(OC)C4)=O)C3)C2)=O)cc2n(n1)CC(C)NC2=O 30958,CC1CN(C(C2C3(CC3)C23CC3)=O)CC2(CCN(C(=O)CC3OCCO3)C2)O1 30959,N1(C(CSCC#C)=O)CCC2(CC1)CN(C(=O)Cc1nonc1C)C2 30960,C12(C(N(C)CC3CCCN(C(=O)C(C)(C)C)C3)=O)CCC(CF)(C1)OC2 30961,N1(C(c2c(C)cccc2O)=O)CCC2(C=C(C(=O)NCCC3(C)CCCO3)C2)C1 30962,CCCC(C)=CC(=O)NC(C(=O)NCC(O)COCC)C1(C)CC1 30963,c1(OC)nc(=NCC(C)(C(C)C)NC(=O)C(=O)Nc2ncc[nH]2)[nH]c2[nH]cnc12 30964,C1(NC(C2(Br)C(C)(C)C2)=O)CCCN(C(c2ccc(F)o2)=O)C1 30965,c1(C(N2CC(CCOC)N(C(=O)C(C)CSC)CC2)=O)cccc2c1OCCO2 30966,Cc1cc(C(=O)NCC(C)NC(=O)COc2cccc(O)c2)ccc1F 30967,C(CCCCCCC)NC(CC(=O)NCCOCCNC(C(C=C)(C)O)=O)=O 30968,c1(SC)ocnc1-c1cn(C(C)CNC(=O)Cc2conc2C)nn1 30969,C(=O)(C(=O)CCC(C)C)NC1CCN(C(C(=O)Nc2c(SC)cc(C)cc2)C)C1 30970,N1(C(c2cc(C(C)(C)C)on2)=O)CC(NC(C2(Cl)CC2)=O)Cc2ccccc21 30971,N1(C(c2ccc(OC)s2)=O)CC(NC(c2ccc(CO)nc2)=O)C(F)C1 30972,c1(CCNC(=O)C(=O)NCC2(F)CC3(CNC3)C2)ccc(Br)cc1Cl 30973,N1(C(C(CC2CC2)OC)=O)CCCCC1C(=O)NC(C)CCCCO 30974,CC1(C)CC(NC(=O)Cc2nc[nH]n2)CN1C(=O)COc1ccsc1 30975,C(c1cc(C(F)(F)F)ccc1Cl)=CC(N1CC(CNC(=O)CCF)OCCC1)=O 30976,C#Cc1cc(C(=O)N(C)CC2(NC(=O)C(F)(CC)C(=O)OC)CC2)ccc1Cl 30977,CC12CCN(C(c3c(O)c(Cl)cc(Cl)c3Cl)=O)CC1C2(F)F 30978,C1(NC(C(C2CCN(C(CC3CC(=C)C3)=O)C2)F)=O)CCCCC1(C)O 30979,n1(CC)nc(C(=O)NC(C)CC(C)NC(=O)C(c2ccc(F)cc2)=O)c(C)n1 30980,C1(C(N(C2CC(C#N)C2)CC(=O)NCCc2c(C)ocn2)=O)CC(=O)NC(C)C1 30981,Cc1cc2[nH]c(=O)c(C(=O)NCC3CN(C(C4CC4(F)F)=O)CC3C)cn2n1 30982,Cn1c(Sc2nnc(-c3ccccc3)n2CCCN)c(C#N)c(=O)n(C)c1=O 30983,N1(C(c2cccc(CCC)c2)=O)CCCC(F)(C(=O)NCc2cnsc2)C1 30984,O(NC(=O)C(F)(CNC(=O)CCC(F)(F)F)C(C)C)CC#C 30985,C(C(=O)N=c1cc(C)o[nH]1)SCC(=O)NCCCC(CO)NC(CCCC=C)=O 30986,N1(C(CC(C)OC)=O)CC(CNC(=O)CCc2cncc(Br)c2)C(C)C1 30987,CCCC(Cc1ccccc1)NCc1ccc(-c2csc(C)n2)s1 30988,C(C(C(=O)N1CC(C)(CSC)C1)C(C)(C)C)NC(C=CC(CC)C)=O 30989,C1(C)(C(N2CCN(CCCNC(c3c(C)ncnc3)=O)CC2)=O)CCCCC1C 30990,CC(C(=O)N(CCNC(c1cnsc1)=O)CC1CC1)NC(c1ccco1)=O 30991,Cc1ccc(S(=O)(=O)N(C)C)c(F)c1.c12cccc(C)c1-c1cnc(nc1)NC2 30992,c1(C2C(NC(=O)NCCc3cc(OC)ncc3)C2)cc(C)cc(Br)c1 30993,CCCC(C)CCCC(=O)NC(C)CCCNC(=O)Cc1csc(COC)n1 30994,S(=O)(=O)(CCC(=O)NC1CCC(CNC(=O)COC2CCCOC2)C1)N(C)C 30995,C1(C)(CC)CC(CC(=O)NCC2C3CN(C(C)C(=O)NCCOC)CC23)=NO1 30996,N1(C(c2c(OC)nn(C)c2)=O)CCCC(NC(c2ccc(O)nn2)=O)CC1 30997,N1(C(c2c(C)nn(C)c2Cl)=O)CC2(CCN(C(=O)CCc3cncc(O)c3)C2)C1 30998,C1(CN(C(=O)Cn2ccccc2=O)C)COCCN1C(=O)C(F)(F)C1(O)CCC1 30999,c1(C(=O)NC(CCCC)CNC(C2COC(=O)N2)=O)ncc(C2CC2)cc1F 31000,O=C(N=c1c(Cl)c[nH]cc1Br)C1CC12CCN(C(c1ccccc1Br)=O)CC2 31001,N1(C(c2nnc(C)o2)C)CCCC(C2CCN(C(=O)C(C)(C)S(C)(=O)=O)CC2)C1 31002,CC(CC(=O)N1CCN(C(=O)CC(O)C2CC2)C(CCO)C1)C(F)(F)F 31003,c1(C(N2CCOC(CCOC)C2)C(=O)NCCC(=O)OCC)cc(C)nc(C)n1 31004,CC1C(NC(=O)Cc2cnoc2)CCCN1C(=O)C(c1cc(F)ccc1F)=O 31005,N1(C(C=CC2C(C)C2(Cl)Cl)=O)CCCN(C(=O)Nc2cccc(=O)n2C)C(C)C1 31006,c1(C(N2C(CN(C(CSCCC(C)C)=O)C)CCC2)=O)ccccc1CC(C)C 31007,C(=O)(CCCC(=O)N1CCC(CNC(c2ncoc2C)=O)C1)OCC 31008,N1(C(C(CC)CC)=O)CCCC(NC(C23CCC(C(F)F)(CC2)C3)=O)CC1 31009,c1(C(=O)NC(CC=C)CNC(c2cc(OC)ccc2O)=O)cnn2cnnc2c1 31010,N12CC(OC)CC(C1)OC1CC(OC)(C1)C2=O.C(=O)(COC(C)(C)C)NC 31011,C12(OC)CCC(C(=O)NC3CCN(C(C4CCCOCC4)=O)C3)(CC1)C2 31012,c1(OC)c(C(N2CC(CO)(NC(c3ccc(=O)oc3)=O)C2)=O)cnn1C 31013,Cc1c(C(=O)NC2(CNC(C3CC4(C3)CC43CC3)=O)CCCCC2)cncc1F 31014,n1(CC)ccc2ccc(NC(=O)C(N3CCC(C(=O)OC)(C(C)C)C3)=O)cc12 31015,n1(CCNC(=O)CNC(C2CCCC2)=O)cc(-c2nccs2)nn1 31016,CN1CCN2CCN(C(C3CCCN(Cc4cncc(O)c4)CC3)=O)CC2C1 31017,N1(C(CCOC(=N)O)=O)CCCC1CC(c1ccco1)O 31018,C(CN=c1ccc(S(=O)(=O)NC(c2nnc(C)s2)C)c[nH]1)SC 31019,CC1(C)CCN(C(=O)CC2CC2(C)C)C(C(=O)Nc2ccc(F)c(O)c2)C1 31020,c1(CC(=O)N(CCCNC(CC2C(CC)C2)=O)CC)ccc(OC)c([N+](=O)[O-])c1 31021,C1(C(N(CCC(=O)NC2CC(=C3CC3)C2)CC)=O)CCSCC1 31022,c1(C(=O)NC(CC=C)CNC(=O)Cc2cscn2)ncccc1C 31023,CC(CC(=O)NC1(C(=O)N(CC(O)C(F)(F)F)C)CSC1)CC(C)(C)C 31024,CC1CN(C(c2cnn(C)c(=O)c2)=O)CC(C)CN1C(C1CC(C)(F)C1)=O 31025,C1(NC(C(C)NC(CC)=O)=O)CC(OC)C(OC)C1.C12(CC1)CCCN2 31026,N1(C(Cn2ncc(C#C)c2)=O)CCCC(COC)(NC(=O)CSCCC#N)C1 31027,C(=O)(C(O)CC(N)=O)NC(C(N1CCCC(N(C)C)C1)=O)(C)CO 31028,C1(NC(C2CN(S(CC)(=O)=O)C2)=O)CCC(C)N(C(=O)Cc2ccns2)C1 31029,C1(CNC(c2n(C(C)(C)C)ncc2)=O)CCCC(NC(C2C3CCCC23)=O)C1 31030,C1(CNC(C(COC)O)=O)CCN(C(C2CC(c3cccc(F)c3)C2)=O)C1(C)C 31031,N1(C(C2C(NCc3ccc(C(=O)OCC)cc3)C2)=O)CCc2cccnc2C1 31032,c1(C(N2CC3C(CNC(c4c(C)nc(C)s4)=O)(C3)C2)=O)ccc(CO)c(F)c1 31033,C(=O)(C1CCc2c(Cl)cccc21)N1CCCC(C)(C)C1CNC(=O)C1=C(Cl)CC1 31034,CC1=NOC(=O)C1CC(N1CCOC(CNC(C2CN(C)CCO2)=O)C1)=O 31035,c1(NC(C)=O)ccc(CC(=O)NCC(N2CCN(c3ncc(C)cn3)CC2)=O)cn1 31036,Cc1ccc2c(C(=O)NC3CC3CNC(=O)CC(C)F)onc2c1 31037,N1(C(=O)CCc2ccon2)CCC2CN(C(=O)CCc3ccc(CO)cc3)C2C1 31038,C(C)(C(=O)NC(C)C(=O)NCC(C)C(C)CC)(C(C)C)OC 31039,N1(C(CNC(C)=O)=O)CCC(C)(C(=O)NCc2cccc(OC(F)F)c2)C1 31040,c1(C(N(C)CC2CCCN(C(=O)CS(C)(=O)=O)C2)=O)cnc2cccnn12 31041,C#CCC(C)(C(=O)NC1CN(C)CC1O)NC(C1CCCCN1C)=O 31042,C1(C)(C(=O)NCC(N(C(Cc2nc(CC)sc2)=O)C)C2CC2)COC(=O)C1 31043,Cc1ccc(N)c(C(N2CCCC2C(C)NC(=O)CCCC2CCCC2)=O)c1 31044,C1(CCC(=O)N(CC=C)CCN(C)C)CN(C(=O)COCCC)CCC1C 31045,n1(CC)ncc(C(=O)NCC(C)N(C)C(c2cccnc2NCC(C)C)=O)c1C 31046,c1(C(=O)NCc2scc(CNC(c3cc(C)ns3)=O)n2)cc(O)nc(C2CC2)n1 31047,CC(C)C(O)C(C)C(=O)NCC1(F)CN(C(c2ncn3c2CCC3)=O)C1 31048,c1(C(N(CC(C)NC(C(C2CC(F)(F)C2)OC)=O)C)=O)coc(C#N)c1 31049,c1(CC(=O)NCC(C)CN(C)C(C2CC2c2ccccc2)=O)c[nH]c(=N)nc1O 31050,c1(C2C(C(F)(F)F)(C(=O)NC3CC3c3nc[nH]n3)C2)ccccc1-c1nn[nH]n1 31051,c1(CCC(=O)NC(CN(C(=O)C(c2ccc(Cl)s2)=O)C)(C)C)ncc(F)cn1 31052,c1(OC)ccc(C(N2CCCC(C)C2CNC(=O)C(F)(F)C(F)F)=O)c(N)c1F 31053,N1(C(Cc2ccc(OC)cc2F)=O)CCN(C(C2(C)CCOC2)=O)CC2(CC2)C1 31054,c1(C(=O)OC)cc(C)[nH]c(=NC(C)CC(C)NC(=O)C(C)N2CCC2)c1[N+](=O)[O-] 31055,c1(CC(=O)NCC(C)NC(C2(CS(C)(=O)=O)CC2)=O)ccc(OC(F)F)c(F)c1 31056,C(=O)(C1CCc2nccn21)N1C(C)(C)CC(NC(C2(c3cccs3)CC2)=O)C1 31057,c1(C(=O)NCC2N(C(CCc3n(C)ccn3)=O)CC(F)C2)ccc2c(c1)CCN2 31058,CC1=C(C(=O)NCC2CC(F)CN2C(c2ccc(F)c(F)c2F)=O)CCS1(=O)=O 31059,CC(CNC(C1CC1(C)C(F)F)=O)C(F)C(=O)NCC1CSC1 31060,C#Cc1ccc(C(=O)NC2(C(N3CCC(CO)C3(C)C)=O)CC(O)C2)nc1 31061,N1(C(c2c(C)nco2)=O)CC(CNC(C2CCn3nncc3C2)=O)C2(CCC2)C1 31062,c1(N2C(C(N3CCCC(C(=O)OC)C3)=O)CC3CC32)ncnc2c(Br)c[nH]c12 31063,C1(C)(C(NOC2CCCN(CC)C2)=O)CC(O)CN1C(=O)CCc1cscn1 31064,C1(CNC(C2C(CCC)C2)=O)(CO)CC12CCN(C(c1cnnn1C)=O)CC2 31065,CC1(C)CC(CC(N2CCOC(CC3CCCCC3)C2)=O)CN1C1CCC1 31066,c1(C(=O)NC2CN(C(C(COC)(C)OC)=O)CC2C)ccc(F)c(C(C)C)c1 31067,[N-]=[N+]=NC1CN(C(c2ccc3cc[nH]c3c2)=O)CC1NC(C1CC2CCC2C1)=O 31068,C1(C)(C(N2CC(N(C(c3c(SC)cn(C)n3)=O)C)C2)=O)CCCS1(=O)=O 31069,N1(C(Cc2nnc(C)o2)=O)CCC(C2CC2)(NC(c2ccc(C)c(F)c2F)=O)C1 31070,N1(C2CN(C(C=CC(=O)N(C)C)=O)C2)CCN(C(C23CCCCC2C3)=O)CC1 31071,C(=O)(CCC(C)(F)F)C(=O)C(O)CN.CC(O)CNCCN(C)C 31072,C(CN=c1[nH]c(=NCCc2cccn2C)[nH]c2cc(C)ccc12)NC(C)=O 31073,C=CC(CC)CC(=O)NCC1CN(C(C2CC3(CCC3)CO2)=O)CCN1C 31074,c1(C(=O)NC(C2CCN(C(C3(F)CC3C)=O)C2)C)ccnc(N2CCCC2)c1 31075,C(C1(C)OCCc2ccccc21)NS(c1c(CC(=O)OC)cc(Br)c(F)c1)(=O)=O 31076,C1(C)(CNC(CCSC)=O)CN(C(c2ccc(OC)c(N)n2)=O)C(C)(C)C1 31077,C1(NC(=O)C2=COCCC2)CCN(c2ncc(Br)cn2)CC12CCC2 31078,N1(C(C(C)c2cccs2)=O)CCCC(CCNC(=O)COc2ccccc2)C1 31079,N1(C(Cc2n(C)cnn2)=O)CC2CC(NC(c3ccn(CCF)n3)=O)CC1C2 31080,N1(C(C2(N(C(c3cccc(NC)c3)=O)C)CC2)=O)CCC(F)(F)C(O)C1 31081,n1(CC)nc(C)cc1C(=O)N(CCCNC(C1(C)CC=CC1)=O)C 31082,Cc1nc(C(=O)NC2C3CN(C(=O)C=CC4CCC4)CC23)c(=O)[nH]c1C 31083,c1(C(=O)NC2C(NC(CC3C(C)OCC3)=O)CCC2)c(N)cccc1F 31084,C1(NC(COCC(=O)NC)=O)CCCC1NC(C1CC(Cl)(Cl)C1)=O 31085,C(=O)(CS(=O)(=O)CC(C)C)N1C2CC(CC(NC(C3C(C)=CCS3)=O)C2)C1 31086,c1(C(=O)NC(CC)(C)CNC(C2(C)CCOCC2)=O)nc2ccccc2cc1C 31087,Cc1cc(C)c(NCC(N2CC(N(C(=O)CCC3CNC(=O)N3)C)C2)=O)c(C)c1 31088,C1(OC)COC2(CCN(CC34C5CCC3C4C5)CC2)C1.c12cccc(c1)O2 31089,c1(C(N2CC(CC=C)(NC(C3CCC(CS)O3)=O)C2)=O)c(Cl)nn(C)c1Cl.SCC 31090,C1(N(C(c2cc(OC)nc(F)c2)=O)C)CC2CCC(C1)N2C(=O)C(O)CC(C)C 31091,N1(C(c2nc(CC)sc2N)=O)CC2(C1)CN(C(=O)CC1CCCS1(=O)=O)C2 31092,C1(NC(C(C)(O)C2CC2)=O)CN(C(C2CCC3(C2)N=N3)=O)CCC12CCC2 31093,CCCCCC(O)CC(=O)N1CCC(NC(c2c(Cl)ccc(F)c2F)=O)C(C)C1 31094,c1(C(C(=O)NCC2(C(=O)NC(c3cccs3)C)CC2)C)ccccc1 31095,C(C(F)(F)CCC(=O)NNC(=O)c1cncs1)n1cc(C(C)N(C)C)nn1 31096,c1(C(N2CC(CNC(CCN(C3CC3)CC)=O)C2)=O)nc(C(C)C)n[nH]1 31097,C12(CNC(C(C)(C)C)=O)CCCCC1CN(C(c1ccc(O)nc1Cl)=O)C2 31098,N1(C(CC=C)=O)CCCCC1CN(C)C(C1(n2cccn2)CCOCC1)=O 31099,C12CN(CC1C)C2=O.c1(C(=O)OC)nc[nH]c1NC(C1CC(=C2CCC2)C1)=O 31100,C1(C(=O)NCCCOCCNC(c2ccc(C(C)C)s2)=O)CN2CCCC1C2 31101,c12ccc(cn1)C(=O)NC2c1n(C)ncc1.C1(COc2ccccc2)CNC(=O)CO1 31102,C1(C(N(CC(CNC(CCCOC)=O)C)C)=O)CC(C(=O)OC(C)(C)C)=NO1 31103,N1(C(CN(CCC#C)C)=O)CCC2(COC(CNC(=O)CC3OCCCO3)C2)C1 31104,c1(CN2CC(CC(=O)NC3CC4(CCC4)C3)OCC2)cc2ccccc2o1 31105,N1(C(C2N(C)CCOC2)=O)CC2(CC(NC(C3(CC(C)(C)O)CCNC3=O)=O)C2)C1 31106,N1(C(C(C)(C)CF)=O)CCC2(CC1)CCN(C(=O)CC1(c3ccon3)CCC1)C2 31107,n1(CC)cc(C(=O)NCC2CC(NC(=O)Cc3ccnn3C)CCO2)c(C)n1 31108,O=C(COCc1ccccc1)N1CCC(S(=O)(=O)Nc2ccccc2)C1 31109,C(=O)(C(C)(C)CC(F)(F)Br)NC1CC(N(C)C(c2cc[nH]n2)=O)C1 31110,C1(C(=O)NC2C(CNC(c3c(C)ncn3C)=O)CCCC2)CCCCN(C)C1=O 31111,N1(C(c2cc(C#N)sc2)=O)CCC(C2CCN(C(=O)CCCCC(F)F)CC2)C1 31112,C(=O)(CC(C)CC(=O)NC(CNC(=O)CCn1cc(C)cn1)CO)OC 31113,N1(C(CCC=C)=O)CC(NC(=O)C(C)N2CCC2)CCC1C 31114,C1(C(=O)NC(CNC(N)=O)C2CC2)(NC(C2(O)CC2)=O)CC1 31115,C(CN=c1[nH]c(Cl)nc2ccccc12)NC(C(C(C)C)NC(C)=O)=O 31116,C(C(C(C)(C)C)NC(C1(C)COC(=O)N1)=O)NC(Cc1cn(C)nc1)=O 31117,c1(C(N(C)CC2CCC(NC(CC3C(OC)CC3)=O)CC2)=O)cc([N+](=O)[O-])c[nH]1 31118,C1(CC)(NC(=O)CN(C)C(N)=O)CCCN(C(=O)C(COC)N(C)C)C1 31119,c1(C(C)C)cncc(C(=O)NCC2CC(NC(=O)CCc3cccn3C)C2)c1 31120,c1(C(N(CC(CC)NC(c2cccnc2)=O)C)=O)c(C)oc(C)c1C 31121,N1(C(c2n(C)nnc2)=O)CCC2(CC1)CC(NC(=O)C(C)(F)F)c1ccccc12 31122,c1(C(N(CC(C)O)CCNC(C2(C)CC=CC2)=O)=O)ccc(-c2cnn[nH]2)cc1 31123,C1(C(=O)NCCS(=O)(=O)NC)CC2CC1CN(C(=O)CCc1cscn1)C2 31124,N1(C(C2CC=CC2)=O)CC2CC(C1)CN(C(C1(CO)CCOC1)=O)C2 31125,c1(C(=O)NC2C3CN(C(c4cc(C)sn4)=O)CC32)cc(=O)n(C)cn1 31126,N1(C(c2csnn2)=O)CC2(C1)CN(C(C1CCCC1C(F)F)=O)CC2CO 31127,C1(NC(C(C=C)(C)C)=O)CCN(C(=O)Cn2cncc2C(=O)OC)CC1C 31128,N1(C(C2(OCC)CCC2)=O)CC2CCC(C1)CC(NC(C13CCC(CC1)C3)=O)C2 31129,c1(C(N(CC(CC)NC(=O)Cc2ccns2)C)=O)c(NC(N)=O)cccc1F 31130,CC(CNC(=O)COC(F)(F)F)CNC(=O)C(F)C1CCCC1 31131,C1(NC(C(C)n2cccn2)=O)COCC1CNC(c1n[nH]cc1Br)=O 31132,N1(C(C2C(c3ccc(-c4cc(SC)[nH]n4)nc3)C2)=O)CC(CO)CC1(C)C 31133,c1(NC(C2CC(NC(C3N(C)CCC3)=O)C(O)C2)=O)ccc2c(c1)CCC2 31134,c1(C(=O)NC(CN(C(C2(COC)CC=CCC2)=O)C)C)ccc2ccccc2c1 31135,C1(NC(CCSCC)=O)CC2CCC1N(C(c1cc(C(N)=O)cs1)=O)C2 31136,O=C(C1=COCCO1)N1CCN(C(c2ccc(-c3ccco3)[nH]2)=O)C(CF)C1 31137,C1(CNC(C(C)=C(CC)C)=O)CCC(C(=O)NCCc2noc(CC)n2)C1 31138,Cc1nc(Cl)nc(N2CC3CN(C(C4CCS(=O)(=O)C4)=O)CC3C2)c1C#N 31139,C(C(C(=O)N(C)CC1CCCN1C(c1ncoc1C)=O)C(C)(C)C)OCC=C 31140,C1(NC(CCN(C(CCC)C)C)=O)CN(C(C2(CSC)COC2)=O)CC1C 31141,CC(C)CC(C)(C)C(=O)NC(C)CCC(=O)NC1(CO)CCCCC1 31142,C1(C(=O)NC(C2CCCC2)COC)CC(=O)CN1C(=O)Cn1nnnc1C 31143,C1(C(N2CC(CNC(Cc3c(OC)nccc3)=O)C2)=O)CCc2ncncc2C1 31144,C1(C2CC2)(C(=O)NCC(CC)(CC)NC(c2cnn(C)c2C)=O)CC=CC1 31145,N1(C(c2cc(OC)c(O)nc2)=O)CC2(CCN(C(c3nc(C)n(C)n3)=O)C2)C1 31146,CCCCCC(O)CC(=O)NC12CC1CN(C(=O)CC(N1CCCCC1=O)C)C2 31147,c1(C(N2CC(CC(N3C(C(=O)NCC)CCC3)=O)C2)=O)ncccc1NC 31148,N1(C(c2c(C)scn2)C(=O)NC(C)(C)C)CCC2(CCOC2=O)C1 31149,C1(SCC(C(=O)NCC(C)C)N(C)C)CCCCN1C(c1ccc(C(F)F)s1)=O 31150,C1(C(N2CCCC2c2ccccc2)=O)(COC)CCCNC1 31151,C1(C(=O)NCCC(CNC(=O)CCOCC(F)F)O)CC(c2ccccn2)=NO1 31152,C(N=c1[nH]c(=NC(C)CCOC)[nH]c2c1CCC2)c1n(CC)ccc1 31153,N1(C(C(COC)(C)O)=O)CCC2(CC2C(=O)NCc2cnn[nH]2)C1 31154,CCCC(CNC(C1CCC(=O)N1C)=O)CCO 31155,c1(CC)c(C(=O)NC(C2CCOC2)CNC(c2cccc(OC)n2)=O)nnn1C 31156,C(=O)(C(O)CC(F)(F)F)N(CCC(=O)NCCCc1cnn(C)c1)CC#C 31157,c1(-c2scc(C(=O)NCC=CCNC(C(CC)SC)=O)n2)cccc(C#N)c1 31158,c1(SCC)cnc(O)c(C(=O)NCCCNC(c2ccncc2)=O)c1 31159,C(CO)(CCCO)NC(CCCCNC(C1(CCC)CC1)=O)=O 31160,c1(C(N2CCC(CC=C)(NC(C3C4CCCC34)=O)C2)=O)ccc2c(c1)CCN2 31161,c1(CC)ccc(C(C)C(=O)N2CC(CCNC(c3cccnc3O)=O)C2)cc1 31162,C1(O)(c2onc(C(C)C)n2)CCN(C(c2cccc(-c3ccccc3)n2)=O)CC1 31163,C1(NC(CCCC#C)=O)CCCC12CCN(C(c1cc(N)nc(Br)c1)=O)C2 31164,c1(C(=O)NCC(CCOC)NC(=O)C(C#N)C(C)(C)C)cc(S(C)(=O)=O)co1 31165,N1(C(COCCCOC)=O)CCCN(C(=O)CN2CCC(C)CC2)CC1C(C)C 31166,CC1(C)C(CC(=O)NC(C2CCCCC2)C(=O)NCc2ccc(O)cc2)C1(C)C 31167,CC1CC(NC(c2nncs2)=O)CCN1C(=O)CCN1CCOCC1 31168,N1(c2ncc(C(=O)OCC)s2)CCC2(CCC2)C(NC(=O)C2=COCCC2)C1 31169,CC(C)C(C)C(CNC(=O)C=CCF)NC(C1(Br)CC1)=O 31170,C(=O)(C(=O)C(F)(F)F)N(CC(C)NC(C1(C)CCCO1)=O)C 31171,N1(C(CC(=O)NCC)=O)CCCCC(C2CN(C(c3coc(COC)n3)=O)C2)C1 31172,N1(C(Cc2c(C)non2)=O)CCC(C2CCCCN2C(=O)COCCF)CC1 31173,Cc1cc(Br)cc(C)c1COC(=O)CCc1cccs1 31174,Cc1c(C(N2CCC(NC(=O)Cn3cncc3C)C(F)C2)=O)c(C(F)F)nn1C 31175,N1(C(c2nnn(C)c2C(F)(F)F)=O)CCCC(NC(c2cnco2)=O)C(F)C1 31176,CCCCCCN(C(=O)CCC=C(C)C)CCCC.C1(=O)C(C)N1 31177,N1(C(C(CC=C)OC)=O)CCOCC12COCCN(C(=O)CCCCC(C)CC)C2 31178,c1(C(N2CC(C)(c3cn(-c4ccc(Cl)nc4)nn3)C2)=O)nccc2cccnc12 31179,C(=O)(CCCCCNC(=O)CC1CC1(C)C)NC(c1nccs1)(C)C 31180,c1(CNC(C(CC)O)=O)ncc(C(=O)NCCC23CC(CCO2)C3)cn1 31181,c1(C(=O)NCC(C)(C)OCCNC(C2CCS(=O)CC2)=O)cc(Cl)n[nH]c1=N 31182,c1(C(N2C(C3CCN(C(C(C=C)O)=O)C3)COCC2)=O)cccc(C)c1C#N 31183,C(=O)(C1=C(C)CCOC1)NCCN(CC(C)O)C(c1cnc(CC)[nH]1)=O 31184,C1(C(=O)N(C2CN(C(=O)C(=CC3CCCC3)C)C2)C)(OC)CCCOC1 31185,CS(=O)(=O)CC(=O)N1CCCC1C1CCCN(C(=O)N(c2ccc(O)cc2)C2CC2)C1 31186,C(=O)(C1=CCC(F)(F)CC1)NCC1(C)CCC(NC(CC(CC)O)=O)CC1 31187,N1(C(c2c(C)scn2)=O)CC2C3CCC(C2C1)N(C(c1cccnc1O)=O)C3 31188,C(CCCC(=O)N1CC(OCC(=O)NCCCC(O)CO)C1)OC 31189,N1(C(COC2CN(C(C)=O)C2)=O)CCC2CN(C(=O)Cn3ccc(C)n3)CC12 31190,c1(C(N2CCC(C(C(N3CC(O)(C(=O)OC)C3)=O)(C)C)C2)=O)cccc(CO)c1 31191,c1(CC)cc(C(N2CCC2C(=O)NOCc2ccco2)=O)ns1 31192,c1(C(=O)NCCC(C)N(C(c2n(CC)ncc2)=O)C)cc2c(Cl)cccc2[nH]1 31193,c1(OC)cc(N)c(F)cc1C(=O)NC1(CN(C)C(c2ccnnc2S)=O)CC1 31194,C#Cc1ccc(C(N2CCC(NC(c3ccc(SC)o3)=O)C2)=O)cc1F 31195,C12CCN(C1)C(C1CC=CCC1)C(=O)NC21N=N1.C1(C(N)=O)CC(F)(F)C1 31196,C1(C(N2CC(C(C(=O)NCC3(c4ccno4)CCC3)O)C2)=O)COCCC1(F)F 31197,c1(CC(=O)NC2CCN(C(c3n(CC)cnn3)=O)C(C)C2)nnc2n1CCCC2 31198,C12(NC(C3CCC4(CCC4)O3)=O)CCCC1N(C(c1cncs1)=O)CCC2 31199,N1(C(C(=O)N(CCNC(C(CC)(F)F)=O)C)CC)CCc2ccccc21 31200,CC1CC(C(=O)NCC2(C(=O)NCC(F)Cl)CC2)=NO1 31201,C1(C(=O)NC(CC)CNC(c2cc(C)co2)=O)CC2(C)CCCN2S1(=O)=O 31202,C(CC(C)(C)CC(=O)NC1CCC(CCNC(C2(C3CCC3)CCC2)=O)C1)OC 31203,c1(OC)ccccc1C(CNC(c1ccsc1)=O)NC(c1cc(C#N)cs1)=O 31204,c1(C(=O)NC(C(=O)NC(C2(OC)CCC2)C)Cc2ccoc2)ccc(F)cn1 31205,c1(C(N(c2cc(I)ccn2)C)=O)cccc(Oc2ccccc2)c1 31206,C1(CC(=O)NCC(C)Oc2cccnc2)CC=CCC1 31207,C1(NC(c2cc(Br)ccc2Cl)=O)CCCN(C(c2ccc(I)c(O)c2)=O)CC1 31208,c1(-c2n(C3(C(=O)N(CC(F)F)CCO)CC34CCC4)ccn2)ccc(F)c(Cl)c1 31209,N1(C(c2ncn(CC)c2)=O)CCC(C)C1CNC(=O)C=Cc1ncco1 31210,c1(C(=O)NC(CC(C)NC(c2cccc(C(C)=O)c2)=O)C)cc(C)c(C)nn1 31211,C1(NC(C2CCC3(CN(S(=O)(=O)CC4CC4)C3)O2)=O)CCc2ccccc2O1 31212,c1(C(CNS(C(C)CCCc2ccc(F)cc2)(=O)=O)=O)cccc(S(C)(=O)=O)c1 31213,CCCCC(C(=O)N1CCN(C(C2CN3CCC2CC3)=O)C(C(F)F)C1)C(C)C 31214,c1(C(N2CCC(C)C(NC(=O)CCF)C2)=O)c(Cl)oc2ccccc12 31215,N1(C(CN(CC(=O)NC(C)CCC=C(C)C)CC=C)=O)CCCCCC1 31216,C1(NC(c2ccc(F)c(C)c2Cl)=O)CCC2C(CCN2C)C1 31217,C(=O)(C(CO)N(C)C)N(CC(=O)NC1(CC(=O)OCC)CC1)C1CC1 31218,C(CCCC(CO)S)NC(CC(Cc1cccc(OC)c1)C)=O.c1(O)nccs1 31219,C1(COC(C2C(C)C(=O)C2)=O)(CF)CCOCC1 31220,C1(c2n(CCC)nnn2)(Nc2cccc([N+](=O)[O-])c2)CC2(COC(C)C2)C1 31221,c1(C(C(=O)NC(CC)CNC(C2CN(C(=O)NC)C2)=O)(C)C)ccc(Cl)c(C)c1F 31222,C1(C(=O)NC2(CC=C)CCCN(C(=O)C(CC)=CC)C2)CC(C(C)=NO)C1(C)C 31223,N1(C(C)=O)CC2CCC(NC(c3ccnc(C(N)=O)c3)=O)(C2)C1 31224,c1(C(N2CC(CNC(CC3CCN(C)C3=O)=O)C2)=O)ccnc2ncnn12 31225,c1(C(=O)NCCN(C(CC(C)O)=O)CC(C)O)cnc2c(c1)NCC2 31226,c1(CC)nc(C)c(C(=O)NC(C)CNC(c2nnsc2SC)=O)o1 31227,c1(C(N2C(CN(C)C(C3CCCO3)=O)CC(F)C2)=O)c(F)ccc(F)c1F 31228,C1(CNC(CN(C)C)=O)CCC(C)(C)CN1C(=O)C=Cc1nc[nH]n1 31229,N1(C(C(CC=C)C(C)(C)C)=O)CCC2C(CCCN2C(c2cc[nH]c2CC)=O)C1 31230,c1(C(N2CC3(C(=O)NC4CCCC4)CC2CO3)=O)ccc2[nH]ccc2n1 31231,C12(C(C)NC(C3CN(C(=O)C4=CSCS4)C3)=O)CC3CC(CC(C3)C1)C2 31232,c1(C(N2CCN(C3CCOC3=O)CC2)C(=O)NCCC#N)cnc2c(c1)COC2 31233,c1(C(N2CCCC(C(=O)Nc3ccc(Cl)cc3CO)C2)=O)cc2ccoc2cn1 31234,c1(OCC)cnc(C(=O)NC2COCC2NC(=O)CCc2cnoc2)c(Cl)c1 31235,CCC(COC)C(=O)N(CCNC(=O)C(c1ccc(Cl)cc1)C)C1CC1 31236,c1(CC)cc(C)c(C(=O)NC23CC(C2)N(C(=O)C(COC)N(C)C)C3)o1 31237,C1(C(N2CC(C(=O)NCC(F)(F)C(N)=O)(CC)C2)=O)CC(O)C(F)C1 31238,C=CC1(c2ccccc2)COCCN1C(c1ccc(Br)s1)c1nnnn1C(C)C 31239,N1(C(c2ccc(N(C)C)cc2)=O)CC(NC(=O)CC2C=NN(C)C2=O)CC(F)C1 31240,C1(C)(CNC(C2C(C)(C)C2)=O)CCN(C(c2cnn(C3CC3(F)F)c2)=O)C1 31241,c1(C(=O)NC2CCC(C)(NC(COC)=O)CC2)ccc2ncccc2c1F 31242,C1(NC(C2C(OC)CCC2)=O)COC2(C1)CN(C(=O)CC1(C)CC1(F)Cl)C2 31243,CCCC(=O)N(CCN(C(=O)Cn1cccc1)CC)CC 31244,C1(CN=[N+]=[N-])CC(C(=O)N(c2ccc(-n3cccn3)cc2)C2CC2)CCO1 31245,Cc1cc(NC(C2(c3ccc(Cl)s3)CC2)C)cc(Br)c1 31246,Cc1ccc(F)c(CN2CC3CC2CN3C(c2cn(C)nc2C)=O)c1Cl 31247,c1(OC)nc(C)ccc1C(=O)NCC(C)(C(C)C)NC(C1C2CCCCCC12)=O 31248,N1(C(c2c(C)snn2)=O)CCN(C(C2(C(C)(C)O)CC2)=O)CC(CO)C1 31249,N1(C(Cc2c(C)cccc2C)=O)CCN(C(c2cncnc2C)=O)CC(CO)C1 31250,c1(C(=O)NCC2CC(NC(COCC)=O)C2)ccccc1SC(C)C 31251,CCCCCCCC(F)C(=O)N1CCOCC12CCCC2 31252,C(=O)(CCN=C(NCC(C1CCCCO1)(C)C)NC1CC(F)C1)N(C)C 31253,CC1(C)CN(C(c2cc(C(=O)NCCc3ccco3)ccc2Cl)=O)CCC1CO 31254,Cc1scc(C(=O)NCC(C)(O)CNC(c2cccn2C2CCCC2)=O)c1N 31255,C(=O)(C(CC(C)C)n1ccnc1)NC(c1ccccc1OCC)C(C)OCC 31256,C(=O)(C(C)(O)C(C)C)N(CCCN(C)C)CCNC(c1ncc(OC)nc1)=O 31257,Cc1oc2cc(C(=O)NC3CN(C(c4nccc5n[nH]cc45)=O)C3)[nH]c2c1C 31258,c1(C(=O)NC(C2CCOC2C)CC)ccc(CNC(c2coc(N(C)C)n2)=O)cc1 31259,C1(CC(=O)NCC(CC)(CC)NC(=O)CC2CCCOCC2)CCCS(=O)(=O)C1 31260,C1(NC(c2n(CC)cc(Cl)c2)=O)CC2CN(C(C3(O)CCC3)=O)CC2C1 31261,CCC(C)(C(=O)NCC1CCN(C(=O)CC2CCCC(C)(C)C2)CC1)C(N)=O 31262,C1(C(N2CCCCC(NC(CCC(=O)NCCC)=O)C2)=O)CC2(CCCC2)CO1 31263,c1(C(=O)NC(C(=O)N(CC(F)F)CCOC)C2CCC2)ccc2c[nH]nc2c1 31264,Cc1nc(N)cnc1C(=O)NC1(C)CC(NC(C2CNC(=O)C2)=O)C1 31265,N1(C(=O)OC(C)(C)C)C(CNC(=O)Cc2nc(=N)[nH][nH]2)CC2COCC12 31266,CCC(C(=O)N1CCC(NC(=O)CN2CCN(C)C(=O)C2)C1C(C)C)C(F)(F)F 31267,c1(C(N2CCC3(CC(C(=O)NC(C=C)C)C3)C2)=O)noc2ccc(Br)cc12 31268,C1(C(=O)Nc2scc(C(=O)NC(CCCC)C)n2)CCCCCC1 31269,C(C)(C(=O)N1CC(C(O)C(=O)NCCn2ccnn2)C1)OCCCC 31270,C(=O)(C(O)CC(N)=O)N1CCC(CCNC(C2(OC)CCCC2)=O)C1 31271,N#Cc1c[nH]c(C(N2CCC(C(N3CCN(c4ccncc4)CC3)=O)CC2)=O)c1 31272,C1(NC(c2nc(CC)sc2)=O)CCCN(C(=O)C=C2CCCCC2(C)C)CC1F 31273,N1(C(c2c(SC)cnn2C)=O)CCc2ncc(C(F)(F)F)cc2C1 31274,c1(C(=O)NC2C3CC(OCC)C(C3)C2)noc2c1CC(F)(F)CC2 31275,CCCC(O)C(=O)N1CC=CC1.C(=O)(CC=C(C)C)NCCOCCOCCN 31276,C1(C(C)(C)C)(CNC(CN(S(CC)(=O)=O)C)=O)CCN(C(=O)C(F)C2CC2)C1 31277,c1(C(=O)Nc2ccn3nccc3c2)cc(Br)c(O)cc1Br 31278,CCC(CCC(=O)NC(C)(C)C(=O)N(C)C)NC(c1cn(CC)nc1C)=O 31279,C1(C(N2CC3C(CNC(CC(C=C)(C)C)=O)(C3)C2)=O)CCC2(CC1)COCCO2 31280,N1(C(c2c(C)cc[nH]2)=O)CCC(C2CCN(C(=O)CC3COC(C)(C)C3)C2)CC1 31281,C1(CNC(CCC(C)C)=O)C2CCC1CN(C(c1cc3ccnn3cn1)=O)C2 31282,c1(OCC(=O)NC2C(NC(c3c(C)cno3)=O)C2)cccc(Br)c1C#N 31283,C(C(C)(C)CC(=O)N1CC(NC(=O)CCc2c(C)noc2C)C(C)C1)OC 31284,c1(CCC)c(C(=O)N(C2CCCN(C(=O)C(F)=C(C)C)C2)C)nnn1CC 31285,c1(N(C(C(C)OCC=C)=O)C)nc(Cl)ncc1OC 31286,CC1(CNC(=O)CC2COCCO2)CCCN1C(c1ccc(NC=O)cc1)=O 31287,Cc1ccc2c(C(=O)NC3CCC4CCN(C(c5cccs5)=O)C3C4)n[nH]c2c1 31288,N1(C(C(C)C)=O)CCCCC1C(C)NC(=O)CCCc1nccs1 31289,C(=O)(C(CC)CC(F)F)NC(CNC(CCCOCCOCC)=O)CC(F)(F)F 31290,N1(C(c2cc(C)oc2C)=O)CC(F)(F)CC1C(=O)N(C1CN2CCC1CC2)C 31291,C1(C(CNC(CN(c2ccccc2)C)=O)=O)CCCN1C(=O)COC1CCC1 31292,C1(C)(C(N(C2CC2)CC2N(C(Cc3c(C)con3)=O)CCC2)=O)CCCCO1 31293,N1(C(C(Br)=C(C)C)=O)CCC(NC(=O)CC2(O)CCOC2)CC1C 31294,C1(CCC)(NC(c2ccnn2C(C)C)=O)CCCN(C(c2n[nH]c(CC)n2)=O)C1 31295,CC1(C)CN(C(c2nc(Cl)cs2)=O)CC1NC(c1c(F)cccc1F)=O 31296,c1(NC(CCCC=C)C)ncc(S(=O)(=O)NCCN(C2CCCC2)C)cc1Cl 31297,c1(CNC(c2c(C)nc(C(C)SC)s2)=O)cc(F)c(F)cc1Br 31298,C(=O)(C#CC1(C)CCCO1)NCC1(CCNC(c2cccc(C)c2)=O)CC1 31299,C1(COCC(=O)OCC)CN(N2CCCCC2C)C1 31300,Cc1cc2ccccc2nc1C(N1CC(CNC(c2ccc(F)c(O)c2)=O)C1)=O 31301,c1(C(=O)NC(CC)(C)CNC(C2CC2C(C)C)=O)sccc1C#N 31302,C(=O)(C1=CCC(C)CC1)NCCOC1CCN(C(c2c(C#C)cn(C)n2)=O)CC1 31303,C1(O)(CNC(C2CCC2)=O)CC2CCC(C1)N2C(c1cc(Br)no1)=O 31304,C(=O)(C1=CCS(=O)(=O)C1)NCC1N(C(CCC(=C)C)=O)C2C(C1)C2 31305,C(C)(Cc1ccc(C(F)(F)F)cc1)(C(=O)O)NC(CC)CNS(C)(=O)=O 31306,N1(CC(=O)OCCCCCF)CCN(C(c2cnco2)=O)CC1 31307,C1(C#N)(C(=O)NC(C)CN(C)C(c2cc(O)nc(O)c2)=O)CC12CCOCC2 31308,N1(C(CC(C)(C)CO)=O)CCN(C(C2C3CN(CC(F)(F)F)CC23)=O)C(C2CC2)C1 31309,C1(CCOC)CN(C(=O)C=CC(C)C)CCC1NC(=O)CCNS(=O)(=O)C(F)F 31310,N1(C(CCCCCC)=O)CC2CC3CC2C1C3NC(C1CN(C(=O)OC)C1)=O 31311,c12c[nH]c(c1)C2=O.C(=O)(C(O)C1CC1)OCCSCc1ccco1 31312,CC1(C)C(NC(=O)C2=NOCC2)CC1CC(=O)NC1CCOCC1F 31313,C1(CCCNC(C2C(C(=O)OC)C2)=O)CCCN1C(C1CCC(=O)C1)=O 31314,C1(C(=O)NCCSCC)C2CC3C(C2NC(C2(C)C(C)(C)C2(C)C)=O)C13 31315,N1(C(C2(COCC)CCOC2)=O)CCCC2(CCc3ccccc3O2)C1 31316,n1(CC)nc(C(=O)NC2CC23CC(NC(=O)CS(=O)(=O)NC(C)(C)C)C3)c(C)n1 31317,C1(NC(c2c(C)n[nH]c2)=O)COC2CN(C(c3ocnc3C)=O)CC12 31318,c1(CCC)ncc(NC(=O)C(C)(C)CN(C(=O)C=CC2CCOC2)C)cn1 31319,c1(CCC)nc(C(N2CC(CO)(NC(c3nc[nH]c3C(F)(F)F)=O)C2)=O)cs1 31320,C#Cc1ccc(C(N2CC3(CC(NC(C4CC(C)C4)=O)C3)C2)=O)nc1 31321,n1(C2C(SC(C3(n4cc(C(=O)OC(C)(C)C)nn4)CCC3)C)C2)cnc(=N)[nH]1 31322,N1(C(C(C)NC(CC)=O)=O)CC(F)(F)CC1CNC(c1cccc(C)n1)=O 31323,C1(CC(=O)NC(C)(C)CC=CC(=O)NCCCN2CCC(O)C2)CC2C=CC1C2 31324,c1(-c2cc(C)[nH]n2)cccc(C(=O)NC(=O)C(O)CNC(=O)OC(C)(C)C)c1.OCC 31325,S(=O)(=O)(c1ccc(Br)cc1NCC1OCC1(C)C)N1CCCC(CCC)C1 31326,c1(SCC)nccnc1C(=O)NCC(C(C)C)NC(C1(CC)CCC1)=O 31327,CC1C(NC(C2CCC2)=O)CC2CCC1N2C(=O)CC1CC(F)(F)C1 31328,C1(C(=O)NCCCCNC(c2c(C)n(C3CCOC3)nn2)=O)CCCS(=O)(=O)C1 31329,c1(C(C)NC(c2ccnnc2)c2nnnn2CC(F)F)cccnc1 31330,c1(C(=O)NCC2(F)CCC(NC(C3CCS(=O)(=O)N3)=O)C2)ccc2nn[nH]c2c1 31331,Cc1ccncc1CCC(=O)NCC1C=CCN1C(c1ccncc1)=O 31332,c1(C(N2C(CCCNC(=O)COCCF)CCC2)=O)ccc2ncc(=O)[nH]c2c1 31333,C1(c2cn(CCCN(C)C(c3cncc(OCCF)c3)=O)nn2)COCC1(C)C 31334,C1(NCc2c(F)cc(Cl)cc2Cl)CCNC12CCOCC2 31335,C(N=C(NCc1ccco1)N1CCn2c(n[nH]c(=O)c2=O)C1)C1N(CC)CC1 31336,C(=O)(CCC(C)OC(c1ccc(C2CCC2(C)C)cc1)=O)OCC 31337,CCCCC(C(=O)N1CC(C)(C#N)C1)NC(=O)CC=CC(C)(C)C 31338,c1(C(N(C(CCNC(c2c(C)cc(C)s2)=O)C)C)=O)ccc(S(=O)(=O)CF)nc1 31339,C1(CNC(C(C)OCCC#C)=O)CC2CN(C(C3(C(F)F)CCCCC3)=O)CC12 31340,c1(C(N2C(C(N(C)CC3CCCO3)=O)COCC2)=O)ccc(O)c(F)c1 31341,CC1SCCC1NC(C1(CCNC(C2CC3(CC3)C2)=O)CCCC1)=O 31342,c1(OC)ccccc1CC(=O)NCCNC(c1cc(O)cs1)=O 31343,C1(CCOC)(NC(=O)Cc2cc(C)cc(F)c2)CCN(C(=O)CC(C)OC)CC1 31344,C1(F)(CNC(C(F)=C(C)C)=O)CCCN(C(=O)CCCC2CCC2)CC1 31345,CCC1=NOC(C(=O)NC2(C(=O)NOCc3ccncc3F)CCC2)C1 31346,C(C)(CCC(=O)NC(CSC)C(=O)NCc1nc(CSC)no1)OC 31347,C1(C(CNC(CC(C)F)=O)(C)C)CCN(C(c2cnn(C)c2C(C)(F)F)=O)CC1 31348,C1(C(=O)NC2CC(C)(NC(C3N(CCC(C)C)CCC3)=O)C2)CCS(=O)(=O)N1 31349,C(CC(=O)NCCC1(C(=O)NC2CC2c2cnc[nH]2)CC1)OCC 31350,N1(C(c2cncc(COC)c2)=O)CC(NC(c2ccncc2OC)=O)CC(O)C1 31351,N1(C(C2C(C)(C)CC(=O)NC2)=O)CC23CCCC2(C1)CN(c1ncc(F)cn1)C3 31352,N1(C(c2c(C)ncc(Br)c2)=O)CC2CCCC(C1)N2C(=O)C(C)(O)C1CC1 31353,C(=O)(C1=CS(=O)CCC1)NC1CC2CC(NC(c3c(C)nc(C4CC4)o3)=O)CC21 31354,Cc1cc(C)c(C#N)c(NCCC2CCCN(C(c3cccnn3)=O)C2)n1 31355,c1(OC)ccc(C=CC(=O)NC2CCN(C(C3(C)CC3(F)F)=O)CC2O)cc1Cl 31356,c1(C(N2CCOCC(NC(C3(C)CCCS3)=O)C2)=O)sc([N+](=O)[O-])cc1Cl 31357,c1(C(=O)OC)cc(C(=O)NC2CN(C(=O)CSCCC(C)C)CC2C)n(C)n1 31358,c1(OC)cnc(F)cc1C(=O)NC1COCC1NC(=O)C=CC1CCCC1 31359,C(=O)(C(C)CC(=O)OC)NC(C(N1CCC(NC(CC)=O)CC1)=O)c1cccs1 31360,N1(C(C2CC(O)(CC#C)C2)=O)CCC2CCN(C(=O)C(CC)(CC)OC)CC12 31361,c1(C(=O)NCC(N2CCN(C(C3(CC4CC4)CC3)=O)CC2)C)nccn2nccc12 31362,c1(COC(c2ccccc2Cl)c2onc(C3CC(C)(C)C3)n2)cc2occc2s1 31363,C1(CSC)CCN(CCNC(=O)CN(CC(C)C)C(c2cnn[nH]2)C)CC1 31364,c1(C(N2CCC(C)(CNC(C(C)(C)SC)=O)C2)=O)nnc2ccccn12 31365,c1(CC(=O)NC(C2(O)CN(C(=O)C=Cc3cccs3)C2)C)sccc1Br 31366,c1(NC(c2c(OC)ccc(C(=O)O)c2)=O)cc2cncn2c(O)n1 31367,N1(C(Cc2c(OC)nccc2)=O)CC2(CCCCN2C(C2OCCOC2C)=O)C1 31368,C12(NC(CC(C)(C)OC)=O)CC(CNC(C3CCC(=O)O3)=O)(C1)OC21CCC1 31369,C1(C(=O)NCc2cc(C(=O)NC3(C(F)(F)CO)CCC3)co2)CCCCC1CO 31370,c1(CC)c(C(N2CCC(CN(C(C3CC3C(=O)NC)=O)CC)C2)=O)ccnc1Cl 31371,C1(C(=O)NCC(CC)NC(=O)CC2CCCO2)(OC)CCS(=O)(=O)C1 31372,N1(Cc2cn(C(C3CCC4(CC4)C3)c3sccc3)nn2)CCCc2ccccc21 31373,c1(CC(=O)NC2C(NC(Cn3c(C)ccn3)=O)COC2)ccc2cccnc2c1 31374,c1(C(=O)OC)nn(C)c(NC(C2CN(C(C3CN(C)C3)=O)CCS2)=O)c1Cl 31375,CCCCN=C(NCC1(CCl)CN(C(=O)OC(C)(C)C)C1)NC1CCS(=O)(=O)C1 31376,N1(C(C2CN(CC)C(=O)C2)=O)CCC2C(C1)CN2C(=O)C=C1CCC1 31377,C1(C(N2CCOC(c3cn[nH]c3)C2)C(=O)NCC(F)F)CCOC2(CCC2)C1 31378,Fc1cc2nc(CN=c3ccnc(-n4cccn4)[nH]3)[nH]c2cc1F 31379,C1(C(=O)NCC(C)(C(C)C)NC(c2c(OC)n(C)nc2)=O)CCN(C)C(=O)C1 31380,N1(C(C2(C)CCSCC2)=O)CCC(F)C(NC(C2(CC3CC3)CCOCC2)=O)C1 31381,C(=O)(C(C)CC(C)C)NC1C(CNC(c2nc(OCC)sn2)=O)CC1 31382,N1(C(c2ccc(NC)c(F)c2)=O)CCC2CCN(C(C3CC=CC3)=O)CC12 31383,c1(C(N2C(C(N3CCC(CN(C)CC)C3)=O)C=CC2)=O)ncccc1Cl 31384,N1(C(=O)NC)CCC(C(=O)NCC(O)CNC(c2sccc2-n2cnnn2)=O)C1 31385,CCC(CCOC)C(=O)N1CC2CC(C1)C2NC(C12CCC1CC2)=O 31386,c1(C(=O)NCC2CCC(C(=O)NC(C=C)CO)C2)cccnc1CC 31387,C(=O)(CC1=CCN(C)CC1)NC1C(C(N(OCCOC)C)=O)CCC1 31388,C1(C(N(C(=O)Nc2cnco2)CC)C)CCCN(C(=O)OC(C)(C)C)C1 31389,Cc1nc(C)c(C(=O)NC(C2CC2C(=O)Nc2ccc(CO)nc2)C)s1 31390,CC(CC1CCCO1)C(=O)N(CCCOCCNC(c1csc(O)n1)=O)C 31391,C1(NC(c2cc(N3CCCCC3)ncn2)=O)CCCC(F)(F)CC1 31392,C1(C(N(CCCNC(C(C)=C2CCC2)=O)C(C)C)=O)CC(C(F)(F)F)(OC)C1 31393,C1(CC)CCN(C(=O)COc2cc(C)on2)C1C(=O)NCC(c1ccsc1)C 31394,C(=O)(C(C)(C)C(F)F)NC1CCC(F)(CNC(c2ccc(CC(C)C)s2)=O)C1 31395,C1(C(=O)NCCN(C(c2cc(C)oc2C)CC)CCC)CC2(CCOCC2)C1 31396,c1(C(N2CC3CC(NC(C(=O)N(C)C)=O)C3C2)=O)ccc2c(c1)CCCCN2 31397,O=C(CCC(F)(F)F)NCC12CC1CN(C(c1cncc(O)c1)=O)C2 31398,CCC(CNC(C1CCOC(C)C1)=O)(CC)NC(c1ccnnc1S)=O 31399,C1(C(C)C)(C(N2CCC(CC(C)NC(c3cccnc3)=O)CC2)=O)CNC(=O)C1 31400,CN1CC(F)CC1C(N1CC(OCCNC(C2CC2[N+](=O)[O-])=O)C1)=O 31401,C1(COC)(CNC(C2C(C)C2C)=O)CCN(C(=O)Cc2cnc(C)[nH]2)CC1 31402,C1(CNC(C(CC)(C)COC)=O)CC2CCC(C1)N2C(=O)C1=NOC(C)(C)C1 31403,C1(O)(CNC(c2c(CC)occ2)=O)CCCN(C(=O)C(C)(C)C2(C)CC2(F)F)C1 31404,C1(C(=O)NC(CC)CNC(C2C3(CC3)C23CC3)=O)CCc2c(ncn2C)C1 31405,C1(NC(CCc2scc(C)n2)=O)CC2CC1N(C(=O)Cc1nnc(S)n1C)C2 31406,c1(CNC2C(NC(=O)OC(C)(C)C)CC=CC2)cc2c(o1)CCCC2 31407,Cc1c(C(=O)NCCCCNC(C2C3CC3C3CC23)=O)cccc1C#N 31408,C1(CNC(=O)NC(c2n[nH]c(C3CC3)n2)C)CC(C(F)(F)F)CO1 31409,C12(COC)CN(C1)C(=O)C=CC(=O)NC2=O.C1(C)(CCC2CC2)CCC1 31410,Cc1sc(Cl)c(C(=O)NCC2CCCN(C(=O)C=CC(C)(C)C)CC2)c1C 31411,C#Cc1ccccc1CC(=O)NC(C)CN(C)C(C1CN(CC)C(=O)N1)=O 31412,N1(C(C(CCC)NC(CC(C=C)CCC)=O)=O)CCC2(CCC(OC)C2)C1 31413,c1(C(=O)NCCCNC(C(C2CCCCC2)N(C)C)=O)cccc(CCO)c1 31414,C(C1CN(C(c2cnc(CC)nc2)=O)CC1C(=O)N(C(C)CO)C)=CC 31415,c1(COC(C)=O)ccc(C(=O)NC(C)(C)CCCNC(=O)CC2CCOCC2)cc1 31416,C(=O)(N=c1cc(-c2cccc(Cl)c2)o[nH]1)NC(C(C)CN1CCCC1=O)=O 31417,c1(CC)ccc(N)c(C(N2CCN(C(c3cnc(C)nc3)=O)C(C3CC3)C2)=O)c1 31418,N1(C(c2c(C)cn(C)n2)=O)CC(C(=O)NCC2CC(C)(O)C2)CCC1C 31419,CC1CCN(C(c2ccncn2)=O)CC1NC(c1c[nH]nc1F)=O 31420,Cc1cc(C(=O)NC2CCC(N(C(=O)COC3CCCCC3)C)C2)cc(N)c1O 31421,C(CC(CC)C(=O)N1CCCC1C(C)(C)NC(=O)CCCC1CCOCC1)=CC 31422,C12(CC(=O)NC3CC(O)(CNC(c4n(C)nc(O)c4)=O)C3)CCCN1CCC2 31423,c1(C(=O)OC)ccccc1C(=O)N(CC(C)N(C(=O)C(C)Cc1ccco1)C)C 31424,N1(C(C(CC#C)NC(C)=O)=O)CC(C2CN(C(c3ccc(N)c(OC)c3)=O)C2)C1 31425,CC(C)(CCC(=O)NCC(=O)NCC(F)(F)F)c1ccccc1 31426,C(=O)(CCCC(C)C)N(CCOCCN(C(COc1c(CC)cccc1)=O)C)C 31427,C(=O)(C(F)CCC(C)C)NC(C(=O)NCCCOCC=C)CC1CC1 31428,CC(O)C(O)CNC(=O)CCC1CCC(NC(C2CCO2)=O)C1 31429,c1(C(N2CCCC(OCC)C2)=O)cccc2c1ccn2CC(C1CC1)OC 31430,C1(C)(CC)C=C(C(=O)NCC(C)N(C)C(c2ncc(Br)cc2C)=O)C1 31431,C(=O)(C=CS(C)=O)NCCNC(C(=O)N(C1C(OC)COC1)C)=O 31432,C1(C)(C(N2CC(CNC(c3ccc(C(C)=O)nc3)=O)C(O)C2)=O)CCCS1(=O)=O 31433,N1(C(C(COC)N(C)C)=O)CC(CNC(=O)CCSC(F)(F)F)CC1(C)C 31434,C(=O)(C1Cc2ccc(F)cc21)NC1(CO)CN(C(CC2(C)CCC2)=O)C1 31435,c1(C(N2CCC(C(=O)NCC(C(C)O)O)C2)=O)ccc(Cl)nc1O 31436,c1(CC)nc2ccccn2c1C(=O)NCC(C)N(C(=O)C(C)C(F)(F)F)C 31437,CC(C)CCCC(=O)N1CCC(C(N2CCC(c3ccncc3)C2)=O)C(O)C1 31438,N1(CC)CCC(C(=O)NC(C)(C)CNC(c2c[nH]nc2C2CCCCC2)=O)C1 31439,CC(C)C(C)(CNC(=O)CN1CC2CCC1C2)NC(=O)CN1C(=O)CNC1=O 31440,c1(CN2C(CNC(c3c(C)cc[nH]3)=O)CCC2)ccc(C(F)(F)F)cc1Br 31441,c1(C(=O)NCCC2CCCN(C(C3C(C)(CC)C3)=O)C2)noc2cc(Cl)ccc12 31442,c1(C(N(CC(C)NC(=O)C(O)CSC)CC)=O)cccc(NC(N)=O)c1 31443,C(C(C(=O)NC1(CNC(=O)C(F)CC)CCCCCC1)C(C)(C)C)OCC=C 31444,C(=O)(CCCC(N)=O)NCC(C1CCN(C(c2cccc(N)c2)=O)CC1)C 31445,CC(C(=O)N1CCC(NC(C2(C)CC(F)(F)C2)=O)C1)S(N)(=O)=O 31446,c1(NC(C2CC(F)CN2C(c2ccnc(Cl)n2)=O)=O)cc(F)c(F)cc1Br 31447,c1(C(N2CCC(C)(NC(=O)Cc3nnc(O)s3)C2)=O)ccc(Cl)c2cccnc12 31448,CC(CCC(=O)NC1C=CCN(C(c2ccc(-c3cccs3)cn2)=O)C1)N(C)C 31449,Cn1nc(C(F)F)cc1S(=O)(=O)NCCc1cccc(Cl)c1 31450,C(C(=O)N(CC(=O)NC1CC1)C)(C1CCOC1)NC(CC1(OC)CC1)=O 31451,C1(CN(C)C(C23COCC2C3)=O)(CNC(=O)CN2CC3CC3C2)CCCC1 31452,C(=O)(CCC(F)(F)F)N1CC(NC(=O)C(C2CC2)C2CC2)C(n2ccnn2)C1 31453,C(=O)(C(C)(C)C(C)(C)O)NC1C=CC(CNC(C(C)c2cc[nH]n2)=O)C1 31454,Cc1nc2ccccc2cc1C(=O)NC1CC2CC1N(C(=O)C(C)(C)C)C2 31455,c1(C(N2C(CN(C(C3CN(C(C)=O)C3)=O)CC)CCC2)=O)nc(OC)c(C)s1 31456,O=C1CCC(CC(=O)NCCCn2cc(-c3ccccc3F)nn2)C(=O)N1 31457,C(=O)(CC1OCCc2ccsc21)NCC1CCN(C(C2C(C)(C)C2(C)C)=O)C1 31458,C1(NC(=O)NCC2(C)COC2)CCOC2(CCOC2)C1 31459,C1(C(=O)NCC2(CC)CCCC2)CCN(C(=O)C(C)(C)C2CCCO2)C(C)(C)C1 31460,c1(C(C(=O)NCC=C)N(C)CC2COCCO2)ccc(OC(C)C)cc1 31461,Cc1[nH]nc(C(N2CC3C(NC(=O)C(C)(C)n4cc(Cl)cn4)C3C2)=O)c1F 31462,C1(COC)(CNC(c2ccc(C(N)=O)o2)=O)CCN(C(=O)C=C(C)Cl)C1 31463,c1(C(C)C)ncc(CNC(C2CCC(CNC(c3csc(F)c3)=O)C2)=O)[nH]1 31464,c1(OCC(=O)N(CC(C)N(C(CS(CC)=O)=O)C)C)ccc(C(C)C)c(C)c1 31465,C#Cc1ccc(C(=O)NCC2(F)CCC(NC(c3cnc(OC)s3)=O)C2)cc1 31466,c1(C(=O)NCC2(C)CCN(C(=O)C3=C(Cl)CCC3)C2)cc(=O)c2ccncc2o1 31467,c1(OC)ncc(CN2CCCC2C(c2ccccn2)O)c(C)c1Br 31468,CC1(C)CN(C(c2cccc3cc[nH]c23)C(=O)NC2CCC2)c2cccc(Cl)c21 31469,N1(C(c2cc(C3(C)CC3)n[nH]2)=O)CCCCC1CN(C(C1CCOC1=O)=O)C1CC1 31470,C1(CNC(C(C)SC(C)C)=O)(NC(=O)COC2CCC2)CCCCC1 31471,N1(C(C2(CSC)CC2)=O)CC(C2(NC(c3cnc(S)n3C)=O)CC2)C1 31472,Cc1cccn2cc(C(=O)NCC3C(O)C(O)CN3C(c3ccsn3)=O)nc12 31473,c1(C(=O)NC2C(NC(c3ccnc(OC)n3)=O)CCC2)ccc(C#N)n1C 31474,N1(C(c2c(-c3c(OCC)cc(F)cc3)c[nH]n2)=O)CCC2(CC1)OCCO2 31475,Cc1nc(C#N)c(NCCC(N2CCN(C(=O)C(C)(C)C(N)=O)C3CC23)=O)o1 31476,C1(C(N2CCC(CNC(C(C)=C(CC)C)=O)C2)=O)CCc2[nH]nc(O)c2C1 31477,N#CC1CCCC(C(=O)NC(Cc2ccco2)C(N2CC(F)CC2CO)=O)C1 31478,c1(C(=O)NC2CC(CNC(C(CC=C)C)=O)C2)ccc(Cl)cc1-c1ccccc1 31479,Cc1ccc(CC(=O)N(CCCNC(=O)C(C)OCCN(C)C)CCO)c(Cl)c1 31480,C1(OC)CCC(C(=O)NCCC2(NC(=O)Cc3csc(CCl)n3)CCC2)C1.C(C)C 31481,O=C1OC2CC(C(=O)NC3CN(C(=O)C4CC4)CC3C3CCCC3)CC2O1 31482,C(C)(CCCCNC(c1ccc(F)cn1)=O)NC(C(N1CCSCC1)C)=O 31483,Cc1ccnnc1C(N1CC(CNC(=O)CNC(C2CCOCC2)=O)C(C)C1)=O 31484,c1(C(C)C)nc(NC2CCc3n[nH]cc3C2)cc(=NC2CC3C(C#N)(C2)C3)[nH]1 31485,N1(C(CC2C(=O)NC(=N)S2)=O)CC(NC(C2CCC3(CCC3)C2)=O)CC(O)C1 31486,c1(OC)cccc(COCC(=O)NC2CCCCC2NC(c2cscn2)=O)c1 31487,CCC(C(=O)NCC(O)CCNC(=O)Cc1csc(C(C)C)n1)NC(C)=O 31488,n1(CC)nc(C(N2CCOC(CN(C(=O)C(C)CCOC)C)C2)=O)cc1C1CC1 31489,C12(NC(c3ccc(C)c(F)c3)=O)CCOCC1CN(C(=O)C(C)SC(F)(F)F)C2 31490,C(=O)(C#CC(C)(C)C)N1CCC(C(C)NC(=O)CN2CCCC2CO)CC1 31491,c1(C(N2CCC(CC(=O)NC(c3cccnc3)CC)C2)=O)ccncc1F 31492,Cc1ccc(F)c(C(=O)NC2CCC2NC(c2cc(N)nc(Cl)c2)=O)c1Cl 31493,c1(C(N2C(C(=O)Nc3ccc(Cl)c(O)c3)CC2)=O)cnc2c(Br)cccc2c1 31494,c1(C(=O)NC2C(C)(CNC(C(CCC#C)O)=O)CCC2)ccc2occc2c1 31495,n1(CCOCC)cc(C(N2CC(NC(c3cc(C4CC4)cs3)=O)C2)=O)nn1 31496,c1(OC)ccc(C)c(N2CCCC2=O)c1.c12nnc(n1CC1CCOC1)C1CC21 31497,c1(C(N(C2CCN(C(c3cncn3C)=O)C2)CC)=O)c2c(nn1C)CCCC2 31498,c1(C(C)=O)cc(CNC(CC2CN(C(C3CCCN3C3CC3)=O)C2)C)ccc1C 31499,C=CC(C)(C)CCNC(=O)C(C)N(C(c1ccnc(CO)c1)=O)C1CC1 31500,C1(CC(=O)NC(C2(O)CCCCC2)C(=O)N(C2CC(F)(F)C2)C)CC2CCC1C2 31501,n1(CC)nc(C(N2CC3(NC(C45CC(C)C4C5)=O)CCC2C3)=O)c2c1CCOC2 31502,c1(C(=O)NCC(CC)(C)NC(=O)C=CC2CCOCC2)cn(C)nc1C 31503,CCC(C)CC(=O)C(=O)N1CC(C(=O)NCCCCCCF)C(F)C1 31504,c1(NCC2C(C(=O)NCCN3CCOCC3=O)CCO2)ncc(CCF)cn1 31505,c1(C(=O)OC)ccc(-c2nc(Br)ccc2C)cc1C 31506,c1(CC)c(C(=O)N(CC(C)NC(=O)C(c2ccc(Cl)s2)=O)C)cnn1CC 31507,N1(C(C(Cc2ccoc2)C2(CC=O)CC2)=O)CC(C)OC2(CCC2)C1.COC 31508,c1(C(N(C(CCN(C(C2(CC#C)CCCO2)=O)CC)C)C)=O)cccc2c[nH]nc12 31509,Cc1cccc(CCC(N2CCN(C(=O)C(O)C(C)(C)C)C(C)C2)=O)c1Br 31510,CN1CCN(C(=O)CC2(O)CCCCC2)C(CNC(c2ccc(C3CC3)o2)=O)C1 31511,C(N=c1[nH]c(=NCc2ccc(F)cc2)[nH]c2cc[nH]c12)c1cc(CC)[nH]n1 31512,CC1CN(C(C2CC(n3ccnc3)C2)=O)CCC1NC(c1ccc(O)nc1)=O 31513,C(=O)(C(F)C(C)CNC(c1cc(O)ccc1C)=O)NC1(c2onc(C)n2)CC1 31514,N1(C(CCCCSC)=O)CC2CCCN(C(=O)CCc3cc(C)[nH]n3)C2C1 31515,C=CCCCCC(C(=O)NCC)N1CCC(OC)C1C1CC1 31516,c1(C(N2CCC(n3cc(CNC(=O)C=CCO)nn3)C2)=O)cc(Cl)c(F)cc1F 31517,C1(CC)(CNC(C2CCCC2CNC(C2CCCOCC2)=O)=O)CCC(=O)N1 31518,C(N=c1[nH]c2ccccc2s1)C1(CNC(=O)Nc2cc(Br)n3ccccc23)CC1 31519,Cc1cc2ccnc(NC3CC(c4cccs4)C3)c2cc1F 31520,C1(C(N2CCC(C3CCCN3C(c3cn(C)nc3C)=O)C2)=O)(OC)CCS(=O)(=O)C1 31521,N1(C(C2C(OCC)C2)=O)CCC2CN(C(c3cc(NC)nc(Cl)c3)=O)CC2CC1 31522,C(=O)(C(F)(CNC(=O)Cn1ccnc1)C(C)C)NC(C#C)C(C)OC 31523,c1(CCc2nc(C=CC(C)C)n(-c3ncnn3C)n2)ccc2c(c1)OC(F)(F)O2 31524,CC(CN=c1[nH]c2ncnc-2c(C(F)(F)F)[nH]1)(C1CC1)NC(=O)CCF 31525,Cc1nn(C)c(CN2CCCC(CCF)C2)c1C(=O)O 31526,N1(CC)CC(NC(=O)C(c2ccccc2)NC(c2csc(Cl)n2)=O)CC1=O 31527,C1(C(N(CC(F)F)C)=O)Cc2nccnc2CN1C(c1ccc(F)cc1CO)=O 31528,CCC(C)C(O)C(C)C(=O)N1CCC(CCC(=O)NCCSCCOC)C1 31529,c1(C(=O)NCC2CCN(C(C3C(C=C)C3)=O)C23CC3)ccnc2[nH]c(C)nc12 31530,C12(NC(N3CCC(c4ccccc4Br)C3)=O)CCC(CC1)NC2=O 31531,C(=O)(CC(F)(F)C(F)F)NC1C(NC(CC(n2c(C)cc(C)n2)C)=O)COC1 31532,C(=O)(C(C(C)(C)C)N(C)C)NC1C(NC(c2cc(CC(C)C)[nH]n2)=O)CC1 31533,C(=O)(C(C)(F)C(=O)NCCCOCCCNC(=O)CC1(C)CCCCC1)OC 31534,c1(SC)noc(C)c1-c1cnc(CN2CCN(C(=O)C#CC(=O)O)CC2)nc1 31535,C(=O)(CCCCc1cnc[nH]1)NCC(CC)NC(=O)C(O)C1CC1 31536,C=CC1CN(C(=O)C(CC(C)C)OC)CC1NC(=O)CCN1CCC(O)CC1 31537,Cc1cccc(C(C)C)c1C(=O)NCC1COCCN1C(C1CCNC(=O)C1)=O 31538,N1(C(c2c(CC=C)cccc2)=O)CC(C)CCC1CNC(=O)CNC(C)=O 31539,c1(C(=O)NC2CN(C(C(c3cscn3)N(C)CC)=O)C2)ccn(C)c(=O)c1O 31540,c1(C(=O)NC2CCC(CCNC(CN(C(C)=O)C)=O)C2)noc2c(F)cccc12 31541,c1(C(C(=O)NCCC2CC2)N(C(C)COC)CCOC)ncn(C)n1 31542,c1(C(=O)NCC(CNC(CN(S(CC)(=O)=O)C)=O)(C)C)ccc(C(C)(F)F)cc1 31543,C1(CC)C=CCCN1C(=O)CCC1(C)CCCN1C(=O)COCCCOC 31544,c1(OC)cc(C(=O)NC2CCCN(C(=O)CC(C)F)C2)c2ccccc2n1 31545,c1(SC)cc(C(N2CC(N(C)C(C3CC(O)CN3C)=O)C(O)C2)=O)n(C)n1 31546,c1(NCCO)ccccc1C(CNC(=O)NCCC(O)c1cccs1)=O 31547,C1(NC(CC(=O)N(C)C)=O)COC2(CCN(C(=O)Cc3ccon3)C2)C1 31548,C(=O)(CC1=CCN(C(c2cnc[nH]c2=N)=O)CC1)NC1(C(=O)OCC)CC1 31549,C1(CC(=O)NC2C(NC(=O)COC3CC(F)(F)C3)CCCC2)CCC(F)(F)CC1 31550,CCCCC(C(=O)N(C)CC1(COC)CCC1)NC(=O)CCCC(C)=O 31551,N1(C(c2c(C)cns2)=O)CC=CC(C(=O)NOCCOC(C)C)C1 31552,C1(CC=C)(NC(=O)C=C)CC2CCC(C1)N2C(C1CSCN1S(C)(=O)=O)=O 31553,C1(C(=O)NCC(C#C)OC)CCN(C(c2n[nH]c(C)c2Cl)=O)C(C)C1 31554,c1(CN=C(NCC(O)C(O)c2ccccc2)NC2CCC2)ccc2c(c1)CCO2 31555,c1(COC)cccc(C(=O)NCC2CCC(F)(CNC(=O)CC3CCCO3)C2)c1 31556,N1(C(C2CN(C(c3c(C)nn(C)c3C)=O)CC(C)C2)=O)CCOC2(CCC2)C1 31557,c1(C(=O)NC2C(CNC(=O)COC(F)F)C2)cc2ccc(Br)cn2n1 31558,c1(COC(C)C(N2CC(O)(CNC(c3cnc(C4CC4)o3)=O)C2)=O)ccccn1 31559,c1(NC(=O)C(N2CCCC2C2COCCC2O)=O)cnc2c(c1)CCC2 31560,N1(C(CCSCC(C)C)=O)CCCC(C)(NC(=O)Cc2ccc(Cl)cc2)C1 31561,Cc1cc(C(=O)Nc2ccc(C(=O)Nc3cc(Br)cnc3F)nc2)ccc1Br 31562,C1(SC)C(NCCCO)C1(C)C.C1C(C)(O)CNC(=O)C(=O)N1c1cccnc1 31563,C=CCCN=C(NCC1(C(=O)OC(C)(C)C)CCC1)NC1CCCC(OC)C1 31564,N1(C(C(c2cnccn2)C)=O)CCc2[nH]nc(CNC(=O)C=CBr)c2C1 31565,c1(C(C)(C)C)ccc(C(=O)NC2(CNC(C3CCCOC3)=O)CCC2)[nH]1 31566,N1(CCCc2cccc(N(C)CC3CCC3)c2)Cc2ccccc2CC1CCO 31567,c1(C(=O)NC2C(NC(c3cscc3F)=O)C2)ccc(-c2ccco2)[nH]1 31568,c1(C(=O)NC2CC3(CC(NC(C4C(C)C4)=O)C3)C2)cc(N)cc2ccccc12 31569,N1(C(CNC(=O)OC)=O)CC2CCN(C(=O)CC3CCCCN3C(C)=O)C2C1 31570,c1(C(N(C)CC2CCCN2C(C2OCC2(C)C)=O)=O)c(C(F)(F)F)cnn1C 31571,CC(CC(C)(C)C)C(=O)N1CCCOC(CNC(C2CC(F)(F)C2)=O)C1 31572,CC1(C)CC(CNC(c2ccco2)=O)CN1C(c1ccccc1CC#N)=O 31573,C1(CN(C)C(=O)NC2CC(CNC)C23CCC3)CCN(C)C1(C)C 31574,c1(OCC)ccccc1C=CC(=O)NC(C)CC(C)NC(=O)CCSCC(C)C 31575,C(=O)(C(F)C(C)C(F)(F)F)N(CCNC(c1nc(C)sc1)=O)C(C)C 31576,c1(C2CC(C(=O)NCCOC3CN(C(C4CCC4C(F)F)=O)C3)C2)ccccc1 31577,C1(C(=O)NC23C(CN(C(C4C=CCC4)=O)C2)C3)CCC(F)(F)CC1 31578,c1(C(C)=O)ccc(C(N2CCCC2C(C)NC(=O)CCC2CC2(F)F)=O)o1 31579,N1(C(c2cnccn2)C(=O)NCCSC)Cc2cc(Cl)c(Cl)cc2C1 31580,c1(C(=O)Nc2scc(CC(N3CCC(C(F)(F)F)C3)=O)n2)nc2ccccn2n1 31581,CC(C)CC(C(=O)NCC1(O)CC(O)C1)N(C)C(C1CCC1C#N)=O 31582,N1(C(CN(C)S(N)(=O)=O)=O)CCn2nc(CNC(C3(F)CCC3)=O)cc2C1 31583,N1(C(N)=O)CCCCC1C(=O)NC1C=CCN(C(C2CCC2)=O)C1 31584,c12cccnc1NC2.Cc1occc1COC(F)F 31585,C(CCC(O)C(=O)NC(C)(C)C(C)O)NC(c1n(C)cc(Cl)c1)=O 31586,C1(C(=O)O)(C)CC=CCC1.c1(COC(C)(C)C)ncc(CN2CCCC2)s1 31587,C1(C(N(CC(C)O)CC)=O)C2CCC(C2)C1NC(=O)CCCn1ccnc1 31588,Cc1c(C(=O)N(C(C)CNC(=O)Cc2cnco2)C)cc(O)cc1N 31589,CC(C)CC(F)C(=O)N(C)Cc1cccc(CNC(=O)C(C(C)(C)C)N(C)C)c1 31590,N1(C(COCC(=C)C)=O)CCC2(CC1)CN(C(C1C3CCC(C3)S1(=O)=O)=O)C2 31591,c1(C(CN2CCC(O)(C(C)C)C2)O)cc(=O)oc2cc(O)c(Cl)c(O)c12 31592,c1(C=O)ccc(-c2cccc(C=O)c2)cc1.N1(N(C)C)CCCC1SCCC#N 31593,c1(C(=O)NCC(CC=C)NC(c2cnn3cnnc3c2)=O)ncc2[nH]ncc2n1 31594,C1(NC(CC=CC=C)=O)CC12CC(NC(C1CCCCN1C(=O)CCC)=O)C2 31595,CC1(F)CC2(CN(C(=O)C(c3cccnc3)NC(C3CC3(Cl)Cl)=O)C2)C1 31596,C(=O)(C(C#N)C(C)(C)C)NCCc1c(C(N2CCC(CC#C)C2)=O)c[nH]n1 31597,C1(C(N(C(C=C)C)C)=O)CCOCC1NC(=O)C(=O)C1CCCC1 31598,Cn1cnc2ccsc2c1=NCC1CCCN1C(c1cc(Cl)c[nH]1)=O 31599,Cc1[nH]nc(C(N2CCC3CCC23CNC(=O)CC(F)(F)F)=O)c1[N+](=O)[O-] 31600,Cc1nc(N(CCCNC(c2cc(C3CC3)nn2C)=O)C)c(C)c(C)n1 31601,N1(C(C(C(=O)OC)C)=O)CCC(CNC(=O)C(=Cc2ccccc2Cl)C)CC1C 31602,c1(CC(=O)OCC(C2CC(O)C2)=O)cccc(NC(c2cnco2)=O)c1 31603,C(C(C)C(=O)N1CC(CC(C)NC(C2CCCC2C(F)(F)F)=O)C1)OC(C)=O 31604,c1(CC)[nH]c(C(=O)NCC2CCCC2NC(=O)C#CC(C)C)c(C)c1C(=O)OC 31605,N1(C(CCCc2cc(C)no2)=O)CCC2(CCCN(C(C3CCC(=O)N3)=O)C2)C1 31606,c1(C(N(CCOC)CCNC(c2cc3sccc3s2)=O)=O)c2ccccc2nn1C 31607,C=C(CNC(=O)C(F)C(C)CNC(=O)C=Cc1ccco1)C1CCOCC1 31608,c1(C(N2CC(NC(CC3N(C)CCC3)=O)C2)=O)ccc2c(O)nc(S)nc2c1 31609,C1(NC(C(C)OCC)=O)CCCCCN(C(=O)CCCC2CCCCC2)C1 31610,c1(-c2cn(CCCOC)nn2)ccnc(F)c1OC.C12CN(CCO1)C(=O)C2 31611,N1(C(C2C(C)=C2)=O)CCC(NC(=O)CN2CCCS2(=O)=O)CC1C 31612,c1(OC)cc(C(N2CCCC2CNC(C2CC(CN(C)C)C2)=O)=O)ccn1 31613,N12CCC3C(CCN3Cc3cc1ncn3)C2.c1(C2(C(=O)OCC)CC2)cccs1 31614,CN1CC2CC1CN2C(=O)CCC(=O)N1CCN(Cc2ccc(O)cc2)CC1 31615,C(=O)(C1OCCn2ccnc21)NC1C(NC(c2cc(CO)on2)=O)C1 31616,N1(C(COCCC=C)=O)CCC(NC(c2nn(CC)cc2Cl)=O)C(F)C1 31617,C1(CNC(C2(C)CC2)=O)CCC2CN(C(=O)Cn3c(F)cccc3=O)CCC2C1 31618,c1(C(=O)NC2(C)CN(C(C3C(C)SCCC3)=O)C2)cc([N+](=O)[O-])n[nH]1 31619,Cc1cnc(F)cc1C(N1CCN(C(=O)CCC[N+](=O)[O-])C(C)C1)=O 31620,C1(C(N(CCCC)C2CCC2)=O)CCC2(CC2)N1C(=O)CN(C)C(C)C 31621,c1(C(N2CCC(NC(C(C)=C(C)C)=O)(CF)C2)=O)cc(C2CC2)nc(Cl)c1 31622,C(=O)(C(C(C)C)NC(=O)CO)N(CCC#C)CC.C1(S)CCCCO1 31623,C(CNC(C1CN(C)C1)=O)(CC(=O)NCC(c1ccccc1)O)OC 31624,C1(C(=O)NC(CNC(CC(CC)C2CCC2)=O)C)CCC2CCCCC2C1 31625,Cc1ccc(F)c(C(=O)N(CCCCN(C)C(C2(C)C=CCCC2)=O)C)c1Cl 31626,N1(C(c2cc(OCC)n[nH]2)=O)CC(C(=O)NCC(C)(C)COC)C(F)(F)C1 31627,c1(C(=O)NC(C2(O)CN(C(CC(C)OC)=O)C2)C)ccnc(C2CC2)n1 31628,C(=O)(C1CCCc2cc(O)ccc21)N(C1CCN(C(C2(C)CCCC2)=O)C1)CC 31629,c1(C(N2CCCCC2)COC)ccc(Br)cc1.c12cn(nn1)CC(=O)N1CC(C1)C2 31630,C12CCCCCN1C(=O)CN1CCN(CC1)N(CC1CCC1)C2=O.CC 31631,C(=O)(CC1=CCCCC1)N1CCC(NC(c2ccc(N3CCOCC3)c(Cl)n2)=O)C1 31632,O=C(C1CCCc2nn[nH]c21)N1CCC(OC2CN(CC(Cl)(Cl)Cl)C2)CC1 31633,C=CC1(C(=O)NCCC2CCOC2)CCN(C(=O)Cc2ccc(C)s2)C1 31634,C12(CC(=O)N(C3CN(C(=O)CN4C(=O)CCC4=O)C3)C)CCC(C)(C1)OC2 31635,C1(O)(C(=O)NCC(C)(C2CCC2)NC(=O)CN2CCC(O)CC2)CCCCCC1 31636,C1(NC(C2NC(=O)OCC2)=O)CCCN(C(c2cnc(S)n2C2CC2)=O)CC1 31637,O=C(CC(O)CNC(C1CCN(C2CC2)C1)=O)NCCc1ccccc1F 31638,C(=O)(C(C)(O)C(F)(F)F)NCC1(C)CCN(C(=O)Cn2ccnn2)CC1 31639,C(C)(CCC(=O)NC1CCCC1COC)NC(c1n(CC)ccn1)=O 31640,N1(C(Cc2cc(C)sc2C)=O)CCCC(CO)(CNC(C2OCCC2(C)C)=O)C1 31641,Cc1ccc(F)c(CC(=O)N(C(C)CNC(=O)CCCC2CC2)C)c1 31642,N1(C(CC2CCC(=O)C2)=O)CCCC2(CCN(C(=O)CN3CCCCC3=O)C2)C1 31643,C(=O)(CC1C(=O)Nc2ccccc21)N1CCC(C(=O)NCC(COC)(C)O)CC1 31644,C1(NC(C(CCOCC)NC(=O)CS(=O)CC)=O)CCCC2(CC1)CC2 31645,c1(C(N2C3CC(N(C(C(CC)O)=O)C)CC2CC3)=O)c2ccccc2nn1C 31646,N1(C(C(F)=CCC)=O)CC(NC(=O)COc2ncccc2Cl)CC(F)C1 31647,C1(NC(C2C(OCC)C2)=O)(NC(=O)C#CC2CC2)CCCCC1 31648,c1(SCCNC(C(C)C(N)c2ccccc2)=O)cn(C)c2cc(Cl)ccc12 31649,N1(C(CC(C=C)(C)O)=O)CC(C2CN(C(=O)CCC3CCC(=O)N3)C2)C1 31650,C1(NC(c2cc(C)nn2C)=O)CCSC12CN(C(c1ccc(N)cc1O)=O)C2 31651,C1(NC(c2c(OC)nn(C)c2)=O)CN(C(c2cn(C3CCC3)nn2)=O)CC1(C)C 31652,C1(N(C(=O)Cc2csc(C(C)OC)n2)CCC)CCN(C(C23CCC2C3)=O)CC1 31653,N(C(=NCCC1CC1)NC(c1ccco1)C)Cc1n(CC)ccc1 31654,c1(CC(=O)NC2(CO)CN(C(CC(CC)C3CCC3)=O)C2)cnc2ncccn12 31655,C1(C(=O)NCC(C)NC(C2(c3cccnc3)CC2)=O)CCc2nnc(O)cc2C1 31656,c1(C(=O)NCC2N(C(C34CC(CC(C)C)(C3)C4)=O)CCC2C)cccc(O)c1Cl 31657,C1(C(N2CC3C(NC(C4C=CCC4)=O)C(C3)C2)=O)COc2ccccc2O1 31658,N1(C(C(CC)NC(N)=O)=O)CCN(C(=O)CCc2ccc(Cl)nc2)CC1CC 31659,N1(CC(=O)N(N(C)C)CC)CCN(C(c2cnn3c2CC3)=O)CC1.NC 31660,CCC(CN(C)C)CC(=O)NCC1C(C(=O)NCCC(C)c2cn[nH]c2)C1(C)C 31661,C1(C(=O)NC2CCC(CNC(=O)CC3(C)CCCO3)CC2)(OCC)CCCCC1 31662,N1(C(C(CC)C#N)=O)CC(C(=O)NCC2(O)CCN(C)C2)CC(C)C1 31663,c1(C(N2CC(C)N(C(c3cccnc3)=O)CC2)=O)cc2c(F)c(Cl)ccc2[nH]1 31664,C1(C(=O)NCC(CC)C)CC(F)CN(C(c2ccc(C(F)(F)F)cc2)=O)C1 31665,C1(CNC(CSSC)=O)CCN(C(=O)C(C)Sc2ccc(N)cc2)C1(C)C 31666,c1(C(=O)NC(C)C(c2ccc(Br)cc2)O)ccc2c(c1)CC(C)(C)O2 31667,c1(C(=O)NC2CCCC(NC(CCC(=C)C)=O)C2)cnc(O)c(OC)c1 31668,c1(-n2c(C(c3n(C=C)ccn3)NC3(COC)CC3)nnn2)ccc2c(c1)OCCO2 31669,N1(C(C23CC(C(=O)OC)(C2)C3)=O)CC(NC(C23CCCN2CCC3)=O)CCC1C 31670,CCC(O)C(C)C(=O)NC1CCCCC1CNC(=O)CCC1CC1(F)F 31671,c1(C(=O)NC(c2ncc(Br)cn2)(C)C)cc(Cl)c(N)c([N+](=O)[O-])c1 31672,c1(C(=O)NCC2N(C(C(C)n3ccnc3)=O)CC=C2)nn(C)c(Cl)c1Cl 31673,N1(C(C2(C)CCCCO2)=O)CCOC2(C1)CN(C(=O)Cn1ccnn1)C2 31674,C1(C(=O)NC(CC(=O)NCC(CN(C)C)O)C2CC2)CC(C)(C)CO1 31675,C(C)(C(=O)N1CC2(C)CC1(C(=O)NC1CC1C1CCCC1)C2)(C(C)C)OC 31676,C1(NC(C2(CN(C(=O)CC3CN4CCN3CC4)C)CC2)=O)CC1C1CCCCC1 31677,Cc1oc(C(C)C)nc1C(=O)NC1CCC(NC(C2CC(C)OC2C)=O)C1 31678,Cn1nc(CNC(=O)C(C)(C)NC(C2CCCCN2C)=O)n(C)c1=O 31679,N1(C(C(C)N2CCC2)=O)CC=CC1CNC(C1(Cc2ccccc2)CCCC1)=O 31680,Cn1cc(CC(=O)NC2COCC2NC(c2cnns2)=O)cn1 31681,CC1CN(C(C2CC23CC(C)(C)C3)=O)CC2(CCN(C(C3CC3(C)C)=O)C2)O1 31682,C(=O)(C(F)C(F)(F)F)NCCC1(CNC(c2cc(F)cc(F)c2)=O)CC1 31683,C12(NC(=O)CSCc3ccccc3)CCCC1N(C(=O)COc1cn[nH]c1)CC2 31684,C(CC1=CCN(C(=O)Cc2cccc(F)c2)CC1)NC(C(=O)NC(C)C)=O 31685,C(CCCC(=O)NC(C)CCC(C)C)NC(CCCOCC=C)=O 31686,c1(OC)c(C(=O)NC2CCN(C(c3cc(C(C)(C)C)[nH]c3C)=O)C2)ncnc1C 31687,c1(C(=O)NCC2CCC(NC(C3(CCCC)CC3)=O)C2)[nH]nc2ncnc(O)c12 31688,C12(Nc3c(C(=O)OCC)cccn3)CCCC1N(C(C1CCCSC1)=O)CC2 31689,N1(C(Cc2n(C)ccn2)=O)CCCC(C2CN(C(c3cc(Cl)ncc3F)=O)C2)C1 31690,Cc1ccc(C(=O)C(=O)NC2CC(NC(=O)C(C(C)C)N3CCN(C)CC3)C2)cc1 31691,C=C(C)C1CC(=O)N(C2CC2)C(C)C(=O)NO1.c1(C(N)=O)c[nH]ccc1=O 31692,c1(C(=O)NCC2CN(C(c3c(C)cc(C)oc3=O)=O)C2)c(C)c(Cl)cc(C)c1N 31693,C1(NC(Cn2ccc(C)n2)=O)CC2CC(NC(c3ccnc(Cl)c3N)=O)C2C1 31694,C(C(=O)NCCCOC(C(CC)C)=O)(C(C)C)SCC 31695,c1(C(C(=O)NCC(CC=C)NC(c2c(C)ncn2O)=O)=O)cc(Cl)ccc1OC 31696,C(=O)(CC(C(F)F)NC(c1ccnc(C)n1)=O)NCCOCCC=C 31697,C1(C(N2CC(C)(OCC(=O)NC(c3nc[nH]n3)C)C2)=O)CC=CCC1C 31698,N1(C(Cc2cnc(C)o2)=O)CC2CC(NC(c3ccc(C(C)(C)C)o3)=O)CC1C2 31699,CC1CCCn2ncc(C(N3CCC(NC(c4cc5ncccn5n4)=O)C3)=O)c21 31700,Cc1cccn2cc(C(=O)NCC3CCN3C(=O)CC(C)CN(C)C)cc12 31701,C12(C(=O)Nc3c(C(=O)OC)ccs3)CC1CN(C(=O)CC1CN(C(C)=O)C1)C2 31702,C1(c2cn(C3CC(F)CC3=O)nn2)CC2(CC2)CN1C(c1cc(SC)c(C)o1)=O 31703,Cc1oc2ccccc2c1C(N1CCCOC(CCNC(=O)C2=CCOC2)C1)=O 31704,N1(C(C(C=CC)O)=O)CCN(CC(=O)NCCC2(C)N=N2)CC1 31705,C(CN=C(NC(C)C1CC1)NC1CC=CCC1)n1ncc(C)c1 31706,N1(C(c2csc(C)n2)C(=O)NC(C(=O)OC)C)CCN(c2ccccc2O)CC1 31707,c1(C(=O)NC(C2CN(C(c3c(Cl)cc(C)s3)=O)C2)C)c(C)nc(C2CC2)nc1O 31708,c1(C(N2CCCC(N(C(c3ccc(C)o3)=O)C)C2)=O)[nH]c(=N)ccc1C 31709,CC1CN(C(C2CC23CC3)=O)CC(C)N(C(=O)C(C)Cc2ccccc2)C1 31710,C1(CNC(=O)C=CC=C(Cl)Cl)CN(C(=O)CC2CC2)CC12CCC2 31711,C1(C(N2CCSCC2)=O)(CC)CCCN1C(=O)Cn1cnnc1O 31712,c1(C(N2C(COC(C)=O)CCCC2)=O)cc(Br)cc(C(F)(F)F)c1N 31713,Cc1c(C(=O)NCCC2(CNC(c3ncccc3Cl)=O)CC2)cccc1F 31714,CC12CCOC(C(=O)NC3(CNC(C4Cc5nccn5C4)=O)CC3)(C1)C2 31715,C1(CC)CN(C(=O)CCN(C(c2ccnn2C(F)F)=O)C(C)C)CC1O 31716,c1(SC)cn(C)nc1NC(=O)NC1C=CCN(C(=O)COC2CCOC2)C1 31717,c1(C(N=C(C(c2n(C)ccn2)N2CCCCC2)N)=O)ccc2nc(O)[nH]c2c1 31718,c1(C(=O)OCC)ccc(C(=O)OC2C(CCC)CN(C(C)=O)C2)c(O)c1 31719,c1(C(=O)OCC)cccc(N(C(CNCc2cc[nH]c2)=O)C2CC2)c1 31720,C(=O)(CC(O)CC(C)(C)C)NCC(CNC(CCCc1ccc(C)c(C)c1)=O)O 31721,c1(C(N(C)Cc2c(CNC(C3C(C)CCO3)=O)cccc2)=O)c(Cl)cncc1Cl 31722,c1(C(=O)NCCOCCCNC(CCCC(CC)C)=O)c(F)ccc2n[nH]cc12 31723,C1(C(=O)NC2C(SC)CN(C(=O)CSC(C)C)C2)CCCCC(F)(F)C1 31724,Cc1cc([N+](=O)[O-])cnc1N1CC2CCN(C(=O)Oc3ccccc3)CC2C1 31725,C1(NC(C(C2CCCC2)NC(C)=O)=O)CCN(C(c2ccc(C(F)F)s2)=O)C1 31726,c1(CC(N2CC(CC=C)(NC(=O)CC3CCC(O)C3)C2)=O)sc(C)cc1C 31727,Cc1cc(C#N)cnc1C(=O)NC1(C)CCCN(C(c2nc(Cl)cs2)=O)C1 31728,C12(C(=O)NC(CNC(c3ccnc(C)c3C)=O)(C)C)CCOC1CCOC2 31729,N1(C(COC2CCN(C(CC3CCCN(C)C3)=O)C2)=O)CC2CC2C2CC12 31730,C1(C(=O)OC)CN(C)CC1NC(=O)NCc1cccc(-c2nc[nH]n2)c1 31731,C1(NC(C2CC(C)NC(=O)C2)=O)CN(C(=O)CC2CC(F)(F)C2)CC12CCCC2 31732,C(=O)(C1(C)c2ccccc2-c2ccccc21)N1CCC(CNC(CCSC)=O)C1 31733,C#CCCCC(=O)NCC1(CNC(C2CC(OC3CCCCC3)C2)=O)CC1 31734,c1(C(N(C2CN(C(C(C)OC)=O)C2)C)=O)c(NC(C)=O)c[nH]c1C 31735,c1(C(N(C2CC(NC(=O)CC3CCC(=O)NC3=O)C2)C)=O)cc(O)cc(C#N)c1 31736,CC1CN(N(Cc2ccc(F)cc2Cl)Cc2ccccc2)CC1F 31737,N1(C(CC2C(CC)C2)=O)CCC(C)C(CC(N2CCCC2CN=[N+]=[N-])=O)C1 31738,CCC(C)C(CC(=O)N1CCCC(F)(F)CC1)NC(=O)CCC(C)(C)N(C)C 31739,CCCC(CC)CC(=O)NC(C1CCN(C(c2cn(C)cc2C)=O)C1)C 31740,C1(CN(C(Cc2c(C)non2)=O)C)CN(C(c2ccc(Cl)c(O)c2)=O)CC12CC2 31741,C(C(C)C)(C(O)C(=O)N1CCOCC1CC(=O)NCCCC1(C)CC1)OC 31742,CCC(CC)C(C)C(=O)N1CC(NC(=O)Cc2cc(F)ccc2OC)CC(F)C1 31743,C1(NC(C(C(=O)OC)OC)=O)CCN(C(C2CCOC2)=O)CC1F 31744,C1(COCC(F)(F)F)C(=O)N1.C1(=O)CCCCCN1.C(C(=O)C1CC1)NC(C)=O 31745,C#Cc1ccc(C(=O)NCC2C3CC2N(C(c2sccc2C(F)F)=O)C3)c(C)c1 31746,CCC(CN(C(=O)Cc1cscn1)C)NC(C1CC1C)=O 31747,Cc1ccc(C(C)NC(C2CNCCN2)=O)cc1Br 31748,N1(C(C(C)CC2CCCCC2)=O)CCC(O)C(NC(=O)C=CC2CC2)C1 31749,C(C(C)(F)CNC(=O)Cc1ccccc1)NC(COCC(C)C)=O 31750,C12(C(N3CCC(CNC(C4N(C(=O)NC)CCC4)=O)C3)=O)CCC(CO1)C2 31751,C1(CC(=O)NCC(=O)NCC)N(C(c2cc(C)[nH]c2C)=O)CCC1(C)C 31752,Cc1cnc(F)cc1NC(=O)NC1(CN(C)C)CCN(C)CC1 31753,c1(C(=O)NC(C2CCOC2)CNC(c2ccc(C)nc2)=O)c[nH]cc(F)c1=O 31754,C(=O)(CC1=NNC(=O)C1)N1C2CN(C(C(COC)NC(C)=O)=O)C(C2)C1 31755,c1(C(N2CC(CC(N3CC(C#N)C3)=O)C3(C2)CC3)=O)c[nH]c2ncccc12 31756,c1(-c2ccc(NC(c3c(C)ccc(F)c3)=O)cc2F)cccc(S(C)(=O)=O)c1 31757,CCC(C(=O)N(CCNC(=O)CC(c1ccc(Cl)cc1)O)C(C)C)C(C)(C)CC 31758,Cc1ncc(N)cc1C(N1CC(C2(NC(=O)Cn3cc(Cl)cn3)CC2)C1)=O 31759,C1(C(N2CC(C)C2CO)=O)N(C(=O)C2=CCCCC2)CCC1(C)C 31760,CCC(CC)CC(=O)N1CCCC(C2CCCN2C(c2c[nH]c(=N)nc2C)=O)C1 31761,Cc1cc(C(=O)NC2CCC(CNC(C3CCCOC3)=O)C2)ccc1O 31762,C1(CC(=O)OC)CCCN(c2ncccc2-c2c(C)noc2C)C1 31763,c1(OC)cccc(NC(C2(O)CCN(C(c3ccc(O)c(F)c3)=O)C2)=O)c1C 31764,N1(C(C23CC(NC(c4c(CCC)nco4)=O)(C2)C3)=O)CCC(O)CC12CC2 31765,CCC(O)CC(=O)N1CC(C)(C(=O)NC2(C(=O)OC(C)(C)C)CCCC2)C1 31766,N1(C(C(=O)N(C)C)=O)CCN(C(=O)CC2CSc3ccccc3O2)CC(C)(C)C1 31767,c1(CCC(N2C3CC(NC(C(c4ccnn4C)C)=O)(C3)C2)=O)cc(F)cc(F)c1 31768,N1(C(C(=O)OCC)=O)CC(F)(F)CC1C(=O)NCc1nn(CC)nc1Br 31769,C1(CCN(C(=O)COC(c2ccccn2)=O)C)CCCCN1C(=O)C(C)(C)C 31770,CCC(CC)C(=O)NCC(=O)NCCC1(C(=O)NCCc2cccs2)CCCC1 31771,N1(C(c2cn(-c3cn(C)nc3)nn2)=O)CCC(NC(c2scnc2Br)=O)CC1 31772,c1(CC)nc(C)c(CNC(=O)C(F)CC2CN(C(c3cc[nH]c3)=O)C2)o1 31773,c1(CC)ccc(CNC(C2CN(C(=O)C3=C(C)OCC3)CCN2C)=O)cc1C 31774,N1(C(C=C(CCC)C)=O)CCC(O)(CN(C)C(c2snnc2COC)=O)CC1 31775,C(=O)(C(F)C(C)(F)F)N(CCCCCCN(C(CCC(=O)N(C)C)=O)C)C 31776,N1(C(c2cc(C)sn2)=O)CC(CCNC(C2CC3C=CC2C3)=O)C(C)C1 31777,C12CC3CN(CC13)C2=O.N1(CC(N2CC(n3cc(C)nn3)C2)=O)CC(=O)NC1=O 31778,C1(CC(=O)N(CCCNC(=O)CCCC2CCOCC2)CC)CCCC(C)C1 31779,C1(NC(c2ccco2)=O)CN(C(C2CCCN2CC2CCCC2)=O)C2(CCC2)C1 31780,c1(OCC)cc(C(=O)N(CC(O)CNC(=O)CCc2cc[nH]n2)C)on1 31781,N1(C(Cc2c(C)non2)=O)CC(C)CN(c2cc(O)ncn2)C(C)C1 31782,C1(NC(C(C)OCC#C)=O)CCN(C(c2cnc(C(C)(C)C)nc2)=O)C1C(C)C 31783,c1(C(=O)NCC2CCN(C(C3CCC(CC)O3)=O)CC2C)csc(=NC2CC2)[nH]1 31784,C1(C(C)C#N)CCN(C(c2cc(CNC(c3nonc3N)=O)[nH]n2)=O)CC1 31785,N1(C(CC(CCSC)O)=O)CCC(C2CC2)(CNC(C2CC(C)=NO2)=O)C1 31786,Cc1ccn(C)c1C(=O)NC1CC(NC(C2(C(C)(F)F)CCOCC2)=O)C1 31787,Cc1cccnc1CN1C(CNC(c2cncc(NS(C)(=O)=O)c2)=O)COCC1 31788,N1(C(c2cc(C3(C)CC3)n[nH]2)=O)CCC2(CCC(NC(C3(CO)CCC3)=O)C2)C1 31789,C(=O)(C1CCc2c(Cl)cccc21)NCC1N(C(c2n(C(C)C)ncc2F)=O)CC1 31790,c1(CNC(=O)NC2(SC3CCCCO3)CCCC2)ccoc1OC(F)(F)F 31791,C1(NC(C2CC(C)OC2C)=O)CC2(C1)CC2N=c1cnc(F)c[nH]1 31792,C1(C(N(CC#N)CC#N)=O)CN(C(c2cccnc2C(N)=O)=O)CCN1 31793,CCCCC(C(=O)NCCCN1CCC1)NC(=O)C(C)n1cncn1 31794,C1(NC(C2CC2CF)=O)CC2CC1N(C(=O)Cn1ccccc1=O)C2 31795,CC1(C(=O)NCC2(F)CCCN(C(=O)Cc3cccnc3)C2)CCCCNC1=O 31796,c1(C(N(C2CCN(C(Cc3nc(C)sc3C)=O)C2)C)=O)cc(Cl)ccc1N 31797,C1(C(N(CCCN(C)C)CCNC(C2(C)COC2)=O)=O)CCCC1S(C)(=O)=O 31798,C1(C(=O)NC(C(=O)NC)C(C)C)CC12CCN(C(=O)C(O)C(F)(F)F)C2 31799,N1(C(CCN)=O)CC2CC(NC(COC)=O)C(C2)C1.c12cccc(c1)O2.OC 31800,CCC(C#N)C(=O)N1CC(NC(c2cccnc2S)=O)C(c2cncn2C)C1 31801,N1(C(CCC=CCC=C)=O)CC(F)(F)CC1C(=O)NCCc1ccc(C)s1 31802,c1(C(N2CC(NC(C3C(OC)C3)=O)C(O)C2)=O)sc2sccc2c1Cl 31803,c1(NC(=O)NCC2CC2Nc2ccc(C(F)F)cn2)ccc(Br)cn1 31804,C(C)(C(CC(=O)NCc1ccc(C#N)s1)NC(C1CCC(C)(C)C1)=O)OC 31805,C(=O)(C(C)(C)C(=O)N(C)C)NC(CNC(C(C)SCCCC)=O)CCOC 31806,n1(CC)cc(C(N2CCN(CCO)C(C)C2)=O)c(=O)c2cc(Br)ccc12 31807,c1(CNC(COC(C)=O)=O)ncccc1C(=O)NC1(C)CCCC1C 31808,c1(C(=O)NC(C)CNC(C2CC2F)=O)ccc(Br)s1 31809,CC(C)CC(F)(F)C(=O)NC1CC2(C1)CC2NC(=O)CN1C(=O)CN(C)C1=O 31810,C(CCCCC(=O)N1CC(NC(=O)CCc2cncc(OC)c2)C1)OC 31811,C1(N(C(c2c(SC)cccc2)=O)C)CCN(C(c2c[nH]c(C#N)c2)=O)CC1C 31812,c1(CC(=O)NCC2CCCCC2NC(c2ccccn2)=O)ccc(O)cc1 31813,CC1CCN(C(c2ccnc(-n3cccc3)c2)=O)C1CNC(=O)C(C)CO 31814,C(CC(C(=O)NC(c1nccnc1C)C)NC(C1CN(C(C)C)C1)=O)OCC 31815,C(CC(=O)NCCCCCNC(C1CCCCO1)=O)(C1CC1)NC(=O)OC(C)(C)C 31816,Cc1ccncc1CC(=O)NCC1(C)CCC(NC(=O)CCc2cccs2)C1 31817,N1(C(=O)CN2CCC(F)CC2)CCC2(CCN(C(=O)C3=CC4C=CC3C4)C2)C1 31818,C1(NC(C2CCC(NC(C)=O)CC2)=O)CN(C(C2CC3CCC2O3)=O)CC2CC12 31819,N1(C(C(C)n2ccnn2)=O)CC(CC(=O)NC2CCCCCC2F)CC1(C)C 31820,c1(OCC)ncc(-c2cnccc2C(=O)NCCN(C)CCN)c(C(C)C)n1 31821,c1(CCC(=O)NC(C2CCCN2C(=O)CN2CCCC2)C)cccnc1Cl 31822,O=S(=O)(C1CCCCC1)NCC1CCCN1.c1(C2CC2)ccccc1 31823,CC(C)CC(O)CC(=O)N1CCCCCC1C(N1CC(N(C)C)C1)=O 31824,c1(C(=O)NC(C)CN(C)C(c2c[nH]cc(Cl)c2=O)=O)cccc2c1oc(=O)n2C 31825,C1(NC(C=CC(=O)OCC)=O)CCCCCC1C(=O)Nc1cc(C)ccc1OC 31826,C(=O)(C1OC(=O)c2ccccc21)N1CCC2(C(NC(c3c(C)occ3)=O)C2)CC1 31827,C1(C(C(N2CC(=C(CNC(C(C3CCOCC3)C)=O)F)C2)=O)F)CCCCCC1 31828,CC(C)CC(C(=O)NOC1CCCC1)OCc1ccncc1 31829,CC(C)C(O)C(=O)NC1(c2ccc(F)cc2)CCN(C(=O)C2=CCOC2)C1 31830,C1(CCCCCNC(CCSC)=O)CCN(C(C2CCC(F)C2)=O)CC1 31831,C(CS(=O)(=O)NC1CC12CCC2)NC(=O)OCCOCC 31832,c1(C(N2CCC(CNC(C(=O)N(C)C)=O)C(F)(F)C2)=O)n[nH]c2ccc(O)cc12 31833,c1(CC)cccc(C(=O)NCc2nnn(C)c2C(=O)NC(CC)CC(C)C)n1 31834,CCC(CCCC(=O)NCCN(C(C)C)CC)NC(c1nc(C)c(C)s1)=O 31835,CC1CNC(=O)CN1C(C1CC12CCN(C(=O)CN1CC3CC3C1)C2)=O 31836,N1(C(C(CC)CCOC)=O)CC2CC(C1)C(CO)C2NC(c1cc(CF)on1)=O 31837,N1(C(C2CC(=C)C2)=O)CCC(C2(NC(=O)Cc3cnccn3)CC2)CC1 31838,Cc1nsc(NC(CNC(=O)C(F)(F)C(C)O)Cc2ccccc2)c1C#N 31839,c1(NC(N2CCN(C(=O)OC(C)C)CC2C)=O)cccc2c1OCCC2CCO 31840,N1(C(Cc2ccc(C)s2)=O)CCC2C(C1)CN2C(=O)Cn1cc([N+](=O)[O-])nc1C 31841,C=C(Cl)C(C)(C)C(=O)NCC1(NC(=O)C(C)OCC(C)C)CCCCCC1 31842,CC(CC(F)(F)F)C(=O)N1CCC(C(=O)NCc2cc(O)ns2)C12CCC2 31843,C1(C(=O)NCC(C)CN(C(=O)CSCc2cccnc2)C)C2COCC12 31844,c1(C(=O)NC(CNC)C(C)(C)C)cc2cccnn2c1 31845,N1(C(C(C(CC)C)N)=O)CCCC12CCCN(C(=O)CCNC(C)C)CC2 31846,C1(CC(N)=O)(NC(=O)CCN2CCC(F)(F)C2)CCCN(C(=O)CC2CCC2)C1 31847,C12(CNC(c3cc(Cl)no3)=O)CCCC1CN(C(C13CCC(CF)(C1)OC3)=O)C2 31848,C1(CSC)CC(C(=O)NC2(CNC(C3(C)CCC3)=O)CC2)C1 31849,CCC(C)(CC(=O)N1CCC(NC(C2CCC3(CC2)CC3)=O)CC1)C(=O)OC 31850,N1(C(CCCCCNC(CN(C(=O)OC)C)=O)=O)CC(C)(CO)CC1(C)C 31851,C(C(F)(C(=O)NCc1ocnc1CC)C(C)C)NC(C(C=C)(C)CC)=O 31852,C(=O)(C(O)CCCNC(=O)CC1(N(C)C)CCC1)NC1C(CCC)C1 31853,C(=O)(C1COc2ccccc21)NCC1CN(C(CCC#CC)=O)C2C(O1)COC2 31854,N1(C(C2C(C)(C)C(NC(=O)Cc3ccns3)C2)=O)CCC2(CC1)CC2C#N 31855,N1(C(C2C(C)OCC2)=O)CCC(C2CC2)(CNC(=O)CC2(O)CCN(C)CC2)C1 31856,C1(C)(C(=O)NC2(CNC(C(COC)(C)C)=O)CCCCCC2)CC(C)OC(C)C1 31857,C1(NC(c2c(C)n(C)cn2)=O)CC(O)CN(C(=O)C(F)C(C)(F)F)C1 31858,CCC(C)C(C)C(=O)NCCCN(C(c1ncc(C)cn1)=O)C1CC1 31859,c1(CC)cc(NC(C2(F)CCCN(C(c3cccc(C#N)c3)=O)C2)=O)ccc1F 31860,C(C1CN(C(=O)C(C)C2CCC2)CC1C(=O)NC(C)C(F)(F)F)=CC 31861,c1(N2CCC(=C)CC2)nc(N2CCCC(C)C(C)C2)c2c(n1)CSC2 31862,C(=O)(C(CCC1CC1)NC(c1c(C)csc1)=O)NC12CCCC1C2 31863,N1(c2nc(C)cc(OCC)n2)Cc2nccn2CC(NC(c2coc(C)c2)=O)C1 31864,Cc1ccc(O)c(NC(c2ccc(OCC(N3CCCC(F)(F)C3)=O)cc2)=O)c1 31865,c1(C(=O)NC(CNC(c2c(C)ccnc2)=O)(C)C(C)C)onc2c1CCCC2 31866,CC(C)(C)C(O)CC1CCN(NC(=O)CCC(=O)c2cccc(C(=O)O)c2)CC1 31867,S(=O)(=O)(c1ccc(Br)cc1NC(C)CCSC)NC(C=C)COC 31868,c1(CC)noc(C)c1C(=O)NC(C)CN(C(C1CC1C1CC1)=O)CC 31869,C(=O)(C=C1SCC(=O)N1C)NCC(=O)OCc1nc(Cl)cc(C)c1Br 31870,Cc1nc2cc(C(=O)NCC3CN(C(C4CCOC4)=O)CC3C)cc(Br)c2o1 31871,Cc1noc(CNC(=O)NC2CCC(C)(C)C2)c1[N+](=O)[O-] 31872,Cc1cc(C(N2CCN(C3COCC3NC(=O)CC3(C)CC3)CC2)=O)oc1C 31873,N1(C(C2C(NC(C3C(C(=O)OC)C=C3)=O)CC2)=O)CC2(CCNC(=O)O2)C1 31874,CCC(C)CC(=O)C(=O)N1CCCC(CCNC(c2cc(O)n(C)n2)=O)C1 31875,N1(C(c2cc(CNC(c3sccc3F)=O)ncc2)=O)CCCC2(COC2)C1 31876,C(=O)(C(C(C)CC)c1ccco1)NCC1(CNC(CCC)=O)CCCC1 31877,C1(NC(c2sc(CCC)c(CC)c2)=O)CCC(C)N(C(=O)Cc2ccc(C)s2)C1 31878,C1(C(C)NC(Cc2c(C)cco2)=O)CCCN(C(=O)CCc2c(C)noc2Cl)C1 31879,N1(C(Cc2c(C#C)cccc2)=O)CCN(C(=O)CCC2CCCCC2)C(C)C1C 31880,CCC(CCCC(=O)NCCCc1nncs1)NC(C1CCC(O)C1)=O 31881,c1(C(=O)NCCCN(C(=O)CC2CCN(C)C2=O)CC)cc(OC)c(Cl)s1 31882,N1(C(C2Cc3ccncc3C2)=O)CC2CCN(C(c3ncccn3)=O)C2C1 31883,CC1(C)COCCC1C(N1CC2CC(NC(c3cnoc3C3CCC3)=O)C2C1)=O 31884,c1(C(N2C(CNC(CCOCC(C)C)=O)CC3(CC3)C2)=O)nsc2ccccc12 31885,c1(CC)ccc(N)c(C(=O)NC(CNC(c2cc(O)n(CC)n2)=O)CCC)c1 31886,n1(CC)nncc1C(=O)NC12CC(CNC(=O)CC3(O)CCCC3)(C1)C2 31887,C1(CC)CCC(NC(=O)C(Cn2ccnn2)NC(=O)C(C2CCOCC2)C)CC1 31888,c1(C(=O)NC2CCC(NC(Cc3c(C)nn(C)c3C)=O)C2)ccc(C#N)nc1O 31889,c1(CN2CCC(N(C)C(c3c(I)ccnc3Cl)=O)C2)cc(F)ccc1[N+](=O)[O-] 31890,c1(NC(C2C(NC(C3C(C)(C)OC(=O)C3)=O)C3CCC2C3)=O)cc[nH]c2nccc1-2 31891,Cc1c(C(N2CC3CCC3(C)C2)=O)sc2ccc(C#N)cc12 31892,n1(C(C)C)ncc(F)c1C(=O)NC1CCCC1CNC(=O)Cc1cnn(C)c1 31893,C1(C(=O)NCCC)CC2CC1CC2O.C1CC(=O)NCC(=O)N1CC#C 31894,N1(C(C2(SCC)CCC2)=O)CCC(N(C(=O)Cc2cccc(CO)c2)CC)CC1 31895,Cc1cnc2n1CCC(C(=O)NCCNC(=O)C1=CCCS1)C2 31896,N1(C(CC2CC(=O)NC2)=O)CC=C(CNC(C23CCCC2C3(F)F)=O)CC1 31897,N1(C(c2ccnc3c2CCC3)=O)CCN(C(C2CCC(O)C2)=O)C2(CCC2)C1 31898,C1(NC(COCCC=C)=O)CC2CCC(C1C)N2C(=O)CC12COC(CF)(C1)C2 31899,c1(NCC2CN(C(C3CCc4nccn4C3)=O)C2)ncc([N+](=O)[O-])cc1F 31900,CC1CCN(C(=O)CN2CCCCCC2)CC1NC(=O)CC1CC=CCC1 31901,CC(CC(C)(C)C)C(F)C(=O)N1CCOC2(C1)CN(C(=O)C(C)(F)C(C)(C)F)C2 31902,c1(C(=O)NCC(C)(CO)NC(C(COC)COC)=O)cnn2ccccc12 31903,C1(OCCCNC(C(C)c2ccco2)=O)CCN(C(c2c[nH]ccc2=O)=O)CC1 31904,CCCC(C)(O)C(=O)NCC(CO)NC(c1ccnc(Cn2cnnc2)c1)=O 31905,N1(C(C2CCC(=O)CC2)=O)CCC2CCCC12C(=O)NOCC1CCOC1 31906,C(=O)(C(C)(C)C(N)=O)N1CCC(CCN(C)Cc2nc(O)n[nH]2)CC1 31907,C1(N(CCCC(=O)NC2(C)CN(C(=O)C3CC3)C2)C)CCCCC1O 31908,N1(C(C2CCOC3(CCSC3)C2)=O)CCC(N=c2nc(-c3ccccc3)[nH]s2)CC1 31909,CC(C)CCCC(C)C(=O)NCCOC1CCN(C(=O)C(C2CCCO2)C)CC1 31910,c1(C(=O)NC23CC2CN(c2ncc4sccc4n2)C3)cc(Br)cc2[nH]ccc12 31911,Cc1ncccc1CC(=O)N(C1CCCCC1)CCNC(C1COC(C)(C)C1)=O 31912,C1(OCC(N2CCN(C3CC(C)OC3=O)CC2)=O)CCC(F)(F)CC1 31913,C(CC(CC)C(=O)N1CCC(CCC(N2CC=C(C)C2)=O)CC1)=CC 31914,C#CC(CC(C)C)NC(=O)CN(C(=O)CSc1cn[nH]c1)CCOC 31915,c1(C(=O)NC2(C(F)F)CC(NC(c3ccc[n+]([O-])c3)=O)C2)cnc2n1CCCC2 31916,c1(C(N2CC3CN(C(c4scc(OC)c4)=O)C3CC2)=O)[nH]cc2c1CCS2(=O)=O 31917,CC(=O)C(C)CC(C)C(=O)N1CC=CC1(C)C(=O)N(C1CC(C)(C)C1)C 31918,N1(C(c2cccc(OC)c2F)=O)CC2(C1)CN(C(=O)C(O)CCN(C)C)CCO2 31919,c1(C(=O)NCCC2(C(NOCC=C)=O)CC2)ccc(C#N)c(C)n1 31920,c1(CCC(N2C(C)C(NC(C3(CO)CC3)=O)CCC2)=O)ccc2c(c1)OCCO2 31921,C1(NC(CCCOCCC)=O)C2CCN(C(=O)C(C(C)C)n3cnnn3)C12 31922,c1(C(=O)NCC2CC(NC(CC(C=C)(C)O)=O)C2)cn2c(C)cccc2n1 31923,N1(C(C(C)OCCC=C)=O)CCCC1C(C)(C)C(=O)NCC(=O)N(C)CCOC 31924,Cc1ccnc(C(=O)NCC(C)(C)CCNC(=O)CN2CCOCC2)c1 31925,N1(C(C(C)NC(C)(C)C)=O)CCC(C(C)CNC(c2scnc2C2CC2)=O)CC1 31926,c1(C(N2CC(n3cc(-c4ccc(C)cn4)nn3)C2)=O)cc(N)ccc1C 31927,N1(c2ncc(C)cn2)CCC(C2CCN(C(=O)Cn3nccn3)CC2)CC1 31928,c1(NC(CC2N(C(C(CC)=O)=O)CCOC2)=O)nc(O)ccc1[N+](=O)[O-] 31929,C1(CCC(=O)N(CCN(C(=O)C(C)c2ncco2)C(C)C)C)CCC(=O)N1 31930,C1(COC)(CNC(=O)C(Cc2ccccc2)NCCC2CCCC2)CCCC1 31931,C(CC(C(=O)NC1(C)CC1)NC(=O)C=CC1CCCN1C)N(C)C 31932,c1(SC)ccc(C(=O)NC(C)CCN(C)C(C2CCOC2C(C)C)=O)o1 31933,N1(C(C2C(C)(C)CC2)=O)CC2CN(C(c3nnc(O)nc3O)=O)CC2(C)C1 31934,CC1CC(CNC(C2(C(F)F)CC2(F)F)=O)=NO1 31935,c1(N2C3(CNC(N4CCC5(CCOC5)C4)=O)CC3CC2)ncnn2ccc(Br)c12 31936,CC(CN(C)C)CCC(=O)N1CC2CC(C1)C2NC(C1CC2CC1CC2O)=O 31937,c1(C(=O)NC2CN(C(c3cc(C)n(C)n3)=O)CC2F)ccc2ccccc2c1O 31938,Cc1nn2c(c1C(N1CCCC(NC(=O)Cc3cccnc3O)C1)=O)CCCC2 31939,C(=O)(C(O)CC1CC1)N1CC(CC(C)NC(=O)Cn2cnnn2)C1 31940,c1(CN(C(=O)Cn2ccnn2)C)ccc(CNC(C2CC(C)(C)C2)=O)cc1 31941,C1(C(=O)OC)COCCC1C1CCN(C(=O)Nc2nccnc2Br)CC1 31942,C(=O)(C(C)S(=O)(=O)C(C)C)N1CCC(NC(=O)Nc2c(C)cc(C(C)C)cc2)C1 31943,Cc1cc(C(=O)NCCOc2ccc(F)c(F)c2)c2ccc(Br)cc2n1 31944,C(=O)(CCCCC1CC1)NC(CNC(C(C=C)OC)=O)(C)C1CC1 31945,c1(C(=O)NC2(CO)CN(C(C(C)SCC)=O)C2)cc(OC)cc2c1OCC2 31946,C(=O)(CC(F)(F)C(F)F)NCC(CC=C)C(=O)N1CC2CC2(C(N)=O)C1 31947,C1(CCNC(C2CC(C)(F)C2)=O)CCN(C(c2ncoc2-c2ccco2)=O)CC1 31948,C(=O)(C(C)CC(F)(F)F)NCCCC(C)NC(C1(n2cccc2)CCCC1)=O 31949,N1(CC=C)C(=O)C(CC(=O)N(C2CC2)CC2CC2)SC1=Nc1cccc(F)c1 31950,C#Cc1cncc(C(N2CCC(NC(c3cc(C(N)=O)[nH]n3)=O)C(CC)C2)=O)c1 31951,C1(C(=O)NCCN(C(=O)C(O)c2cnc[nH]2)C2CC2)CCC(OC(F)(F)F)CC1 31952,C1(CNC(C(c2ccc(Cl)cc2)N(C)C)=O)COCCN(C(=O)CC(F)(F)F)C1 31953,C1(C(N(CCCCCNC(=O)CCCn2ccnc2)C)=O)CC2CCC1C2 31954,C1(NC(CCOC)=O)CCCCC12CCN(c1ncnc3sccc13)CC2 31955,N1(C(CSCCOC)=O)CCC=C(C(=O)NC2(CCCN(C)C)CC2)C1 31956,c1(C(=O)NC(C(C)NC(C(COC)C)=O)CO)c(C)ccc(Cl)c1N 31957,c1(C(C(=O)NCCCCC(C)C)N(C2CC2)CC)ccc(C(C)C)cc1F 31958,C1(CC(=O)NC(CC)CNC(c2cc(Cl)c(Cl)[nH]2)=O)CCCC(F)(F)C1 31959,CCC1=C(C(=O)NC2C(C)CCN(C(c3csc(Cl)n3)=O)C2C)SCCO1 31960,c1(NC(c2ccc(C)o2)=O)cccc(N2CCN(C(=O)CSC(C)=O)CC2)c1 31961,N1(C(C(C)OCCC(C)C)=O)CC(C2CN(C(=O)C(N3CCOCC3)C)C2)C1 31962,CCC(CC(C)C)C(=O)NC(C)CCCNC(=O)CSCCOC 31963,C1(C(N2CC(C(N3CCC(CCOC)C3)=O)(CC)C2)=O)COCC(C)O1 31964,c1(C(=O)NC2C3CN(C(C4C(C)=CCS4)=O)CC2C3)cc2cccc(C)c2o1 31965,c1(C(N(C)Cc2ncc(C)o2)=O)cncc([N+](=O)[O-])c1 31966,C(CCCCNC(=O)CCC1(NC(=O)CC2CC2(C)C)CCC1)N(C)C 31967,CC1(C)CCC(C(=O)NCC2CC2CNC(=O)CC2CC3C=CC2C3)CC1 31968,C=CCN=C(NCC1CCC(C(=O)N(C)C)CC1)N1CCC(C)(OC)C1 31969,C(=O)(C(CCC(C)C)N)NC(C#C)C(C)C(=O)Cn1[nH]cnc1=N 31970,n1(C(C)C)cc(Br)c(C(=O)N(C)CC2COCCN2C(=O)C=CC2CC2)n1 31971,n1(CC)nc(C(=O)N(C(C)CCNC(=O)C(C)CSC(F)(F)F)C)cc1O 31972,Cc1oc(CO)nc1C(=O)NCC(C1CCCN1C(c1cnc(S)[nH]1)=O)(C)C 31973,c1(C(N2CCSCC2CCc2ccccc2)=O)cnc2c[nH]nc2c1 31974,C1(NC(c2ccon2)=O)CCC2CCN(C(=O)C#CC3CCCCO3)C1C2 31975,C(C)(CN=c1cc(C)c(S(=O)(=O)N(C)C(c2nccs2)C2CC2)c[nH]1)SC 31976,C(=O)(C1CCCc2scnc21)NCC1CN(C(CCCCC(=O)NC)=O)CC1C 31977,CCCCCC(C)CC(=O)NC1CCC(N(C(=O)C2=CCC(C)CC2)C)CC1 31978,C(=O)(CC1=CCCC1)NCc1c(CNC(C2C(=O)NCC2)=O)cccc1 31979,C(=O)(CC(C)C(=O)NC1C=CC(CC(=O)N(C2CC2C2CC2)C)C1)OCC 31980,C1(COC)CC2(CCN2C(c2cccc3cn(C)nc23)C(=O)NC(C)C)C1(C)C 31981,C1(CNC(c2ncc(OC)cn2)=O)CC(C(F)(F)F)CCN1C(=O)C(C)O 31982,c1(CC)ccc(C(=O)NCC2(NC(C3CCC(C)C3)=O)CCCCC2)c(C)c1 31983,c1(C(CNC(C2C(C)C2)=O)NC(c2cccc(C3CC3)c2)=O)cccc(Cl)c1 31984,C1(NC(c2cnc(OC)nc2)=O)CC(F)CN(C(C2(O)CCCCC2)=O)C1 31985,C1(CNC(c2c(OC)n(C)nc2C)=O)C(C2CC2)CCN1C(C1CC1(Cl)Cl)=O 31986,CC1CN(C(c2cnncc2O)=O)CC1(C)CNC(=O)C1=CCCC1 31987,c1(CCC(=O)OCCCOCCC(C)C)ccc(F)cc1F 31988,C(=O)(CCC(=O)c1ccc[nH]1)NN(C1CCN(C(COCCSC)=O)C1)C 31989,N1(C(C2CC(c3c(C)n[nH]c3C)C2)=O)CCN(C(C)C)C(C(=O)O)C1 31990,N1(C(c2cnc(C)[nH]2)=O)CC2CCC1C(CNC(c1ccc(F)c(Cl)c1)=O)C2 31991,N1(C(C(C)(CO)OC)=O)CC2(C1)CN(C(C1CCn3nncc3C1)=O)CCO2 31992,C(=O)(C(C)CC(C)C)NCC(CNC(c1cccc(C(=O)OC)n1)=O)(C)O 31993,CN1C(=O)CC(N2CC(CNC(=O)NCCS(C)(=O)=O)C2)C1=O 31994,c1(C(N2CC(O)(CNC(C(=CC3CCCC3)C)=O)C2)=O)ccc2c(c1)CC2 31995,C=CCCCCCC(=O)N1CCCC1(C(=O)NCC1CN2CCC1C2)COC 31996,c1(C(=O)NCC2(F)CC(NC(C3(C)CCOC3)=O)C2)ccc(S(C)(=O)=O)s1 31997,c1(C(N(CCCNC(c2cnn(CC)n2)=O)C)=O)c(OC)c(Cl)cc(O)c1Cl 31998,C(=O)(CCCCCNC(=O)CCCc1cccs1)N1CCC(C)(CCO)C1 31999,N1(C(CCC(C)(F)F)=O)Cc2ccccc2CC1CNC(=O)CCOC1COC1 32000,c1(C(=O)NC2CCCN(C(C3CC3c3ccccc3)=O)C2)ccc(Cl)cc1CO 32001,c1(COCC)ncccc1S(=O)(=O)N(C)Cc1conc1C(C)(C)C 32002,Cc1ccn(CC(C)(O)C(=O)N2CC(NC(=O)C(C)(C)OC3CCCC3)C2)c(=O)c1 32003,CC1CCc2[nH]nc(C(=O)NC34CCCC3CN(C(=O)CCCC(N)=O)C4)c2C1 32004,N1(C(c2c(CC)c[nH]n2)=O)CC=CC(NC(=O)COC)C1 32005,c1(C(N2C3CC(CNC(CC(C)(C)O)=O)C2CC3)=O)ccc2c(n1)CCC2=O 32006,C1(NC(Cc2c(C)cccc2)=O)CC2(C1)CC(NC(=O)CCC1CCCN1C)C2 32007,c1(OC)ccc(F)c(F)c1CN1CCOC(C(=O)Nc2ccc(C#N)cc2O)C1 32008,C1(C(N2CCCC(CCNc3ncc([N+](=O)[O-])cn3)C2)=O)CCC2CCCCN12 32009,c1(C(=O)NCCOc2ccc(C)cc2)ccc(C#N)cc1.C=C1CC2(C1)C(=O)N2 32010,Cc1cc(C(=O)NCCC(C)CCNC(C2(C(F)(F)F)CC2)=O)nn1C(C)(C)C 32011,C(c1ccncc1)=C(C)C(=O)NCCN(C)C(C1CCCCC1C)=O 32012,c1(C(=O)NC(CNC(c2c(OC)cccn2)=O)CO)ncnc2c1ccn2C 32013,C1(CNC(c2c(CC=C)cccc2)=O)CCN(C(C2CC(F)CN2C)=O)C12CC2 32014,N1(C(c2c(C)ocn2)=O)CC2C(CN(C(=O)CC3CC34CC4)C)C2C1 32015,CC1CN(C(C23CSC(C2)C3)=O)CC(C)C1NC(=O)C=Cc1cnn(C)c1 32016,Cc1csc2nc(CC(N3CC(NC(C4CCCN4C4CC4)=O)CC3C)=O)cn12 32017,C1(CN(C)C(C2CC=CCC2)=O)COCCN1C(C1COCCOC1)=O 32018,c1(CC(N2CCCC2c2c(F)cccc2F)=O)ccc2ncccc2c1 32019,c1(CNC(C(CC)NC(=O)C(COC)CC)=O)ccc(OC)cc1 32020,C1(NC(=O)N(Cc2ccc(F)cc2)CC2(F)CCC2)C2CCC(F)C12 32021,c1(CC)cc(C(N2CCCC(O)(CCNC(=O)C(C)(F)F)C2)=O)ccc1F 32022,C(=O)(C1=CC2C=CC1C2)N(CCCCCNC(=O)CCC1CCCOC1)C 32023,N1(C(CC)=O)CC2(CC(NC(c3ccc(-c4ccccc4)c(F)c3)=O)C2)C1 32024,C12(C(=O)NCc3ccc(C)cc3C)C3CCC(CC13)C2(F)F 32025,c1(C(c2nnnn2CC(F)F)NCc2c(CC)noc2C)ccc2ncsc2c1 32026,c1(SCC)ccc(NC(=O)NCC2(OCC)CCOC2)o1 32027,C1(C)(CC)C=C(C(=O)N2CC3CC3(C(N3CCN(C4CC4)CC3)=O)C2)C1 32028,C1(CCC(C)C)C(=O)N1.C(C(=O)N(C)CCN(C)C)SCC 32029,C1(CC)CC(C(=O)NC2CC=C(C)CC2)CCN1C(=O)C(F)C(C)(C)O 32030,CCCCC(CCC)C(=O)NC1CC1C1CCCCC1C(=O)OC(C)(C)C 32031,c1(C(=O)OC)ncc[nH]c1=NC1CCCN(C(=O)C=CC2CCCO2)C1.C=O 32032,C1(NC(=O)Cn2cc(CO)nn2)COC2(C1)CN(C(c1c(F)cccc1Cl)=O)C2 32033,C(=O)(C(CNC(=O)CC1CSC1)CC(C)C)NC(C#C)(C)C1CCC1 32034,CC1(CNC(=O)CCN2CCCC2)CCN(C(C2NC(=O)OC2C)=O)C1 32035,N1(C(c2nc(OC)c(C)s2)C(=O)NC2CC2)CCCC2CCC(C)CC12 32036,C(C(CC(F)(F)F)NC(c1cnc(O)o1)=O)NC(CCC1CCC(=O)NC1)=O 32037,N1(C(CN(C(c2ccoc2C2CC2)=O)CC)=O)CCCC(CN(C)C)C1 32038,c1(CC)c(C(=O)NCC2(F)CC(NC(c3cc(N)ccc3C)=O)C2)cccc1C 32039,N1(C(C)C(=O)NC2CCCC2NC(=O)CC2(N(C)C)CCC2)CCCCC1=O 32040,c1(C(N2CC(C)(NC(c3c(SCC)nccc3)=O)C2)=O)cc(O)ccc1C 32041,N1(C(C2=NOC(C)C2)=O)CC(NC(=O)CCCCNC(N)=O)C(C2CC2)C1 32042,c1(C(=O)NC2CCC(CCNC(C=C(COC)C)=O)C2)cc(F)ncc1OC 32043,c1(C(=O)NC2(C(C)C#N)CC2)cnc(CNC(C2CCCOCC2)=O)nc1 32044,c1(C(N2CCCC(CNC(C(CCC)C)=O)C2)=O)ccc(Br)cc1C(C)=O 32045,CC1(C)OCCOC1C(=O)NCCC1CCN(C(=O)COC2CCCC2)CC1 32046,CCC(C)(C)CCCC(=O)NCC1(C(N2CCC(CC)CC2)=O)CC12CCC2 32047,CCS(=O)(=O)CC(=O)NCC1CCN(C(c2cc(F)nc(F)c2)=O)C1 32048,C(CN=c1[nH]cc(C)s1)c1c(SCCC)cccc1.N1(CC)CCC(O)CC1 32049,CN1CCC(C2(C(=O)NC3(C)CCCN(C(c4ccc(Cl)s4)=O)C3)CC2)C1 32050,C1(NC(c2c(CC)c(C)sc2)=O)CCCN(C(=O)CC(C)n2ccnc2)C1C 32051,C#Cc1cccc(C(N2CCSCC2C(=O)N(C)C(C)C2CC2)=O)c1 32052,C(=O)(C1=C(C)NC2=NCCCC2=C1)NCC1N(C(COCCCCC)=O)CC1 32053,CCC(CNC(=O)C=Cc1cnccn1)(CC)C(=O)NCCC1CCCC(C)C1 32054,N1(C(C2CN(C(C3N(C)C(=O)CC3)=O)CC(F)C2)=O)CCN2CCOCC2C1 32055,c1(CC(=O)N(C2CN(C(c3nonc3N)=O)CC2F)C)cncnc1O 32056,C(=O)(CC(O)C(C)CC)NC(CC=C)C(=O)NC(C1CC1C(=O)OC)C 32057,c1(CC)ccc(C(=O)NC2CN(C(=O)C(C)CN(C)C)CC2CC)cn1 32058,c1(N2CCC(C)(CCO)C2)ccc(S(=O)(=O)NC(CO)C2CC2)cc1Br 32059,C1(NC(=O)C(c2cccs2)NC(C23CC2CNC3=O)=O)C2CCCCCC12 32060,c1(C(=O)NC(CNC(C(C)=CC)=O)(C)C2CC2)cc(C)c(-c2ccc(Cl)cc2)s1 32061,C1(CC#C)(C(=O)N(C(=O)CCC=C=C)CCCCC)CCCCO1 32062,n1(CCS(C)(=O)=O)ccc(=NC(=O)C2CCCC(F)C2)[nH]1 32063,c1(C(=O)N)[nH]ccc1-c1cccs1.N1(C(CC(C)CN(C(=O)CSS)C)=O)CCCCC1 32064,c1(C(C(=O)NCCCCNC(C(SC)SC)=O)F)ccccc1 32065,CC(=O)CCCC(C)C(=O)N1CC(C)CC1C(=O)NCC(C)OC(F)F 32066,C(=O)(C(C(C)C)n1cncn1)N(CC(CNC(C(CC)n1cncn1)=O)(C)C)C 32067,C(=O)(C(O)CC(C)(C)C)NC(CCCNC(c1c(C)n(CC(F)F)nc1)=O)C 32068,c1(C(=O)NC(c2ccc(Cl)cc2)C)ccc(F)c(-c2cc(F)nc(F)c2)n1 32069,C1(C(N2C(CCNC(c3ccn(COC)n3)=O)CCC2)=O)CCCCC(F)(F)C1 32070,N1(C(c2cc(CCC)[nH]n2)=O)CCC(C)C(NC(c2ncc(N(C)C)cn2)=O)C1 32071,C1(NC(CCSCCN(C(CSCC=C)=O)C)=O)CCCC(O)C1 32072,C1(C(=O)NC2CCN(c3ccc([N+](=O)[O-])cc3)C2)CCCC2(C1)CC2(F)F 32073,CC(C(=O)NCCN1CCCOCC1C)C(C)(C)c1ccccc1 32074,C(C(C)(C)CNC(C1(Cl)CC1(F)F)=O)N(C(=O)CCCc1cccs1)C 32075,c1(C(=O)NC2C3(CC(NC(C(C=C=C)C)=O)C3)C2)ccc(C(C)=O)nc1C 32076,c1(C(=O)NCC(CCCC)NC(=O)CC(CC)SC)ccc(C(F)(F)F)c(F)c1 32077,C(C)(CCCNC(=O)C(F)(F)c1nccs1)NC(C(C)NC(C)=O)=O 32078,C12(C(=O)NC(CCCCC)C)CCC(CN(C(c3n[nH]c(C)c3O)=O)C1)C2 32079,Cc1c(C=CC(=O)N(C)CC2CCCN2C(C2CCOCC2)=O)cnn1C 32080,Nc1ccc(-c2cn(CCCNC(c3cnc(C4CC4)o3)=O)nn2)nc1 32081,C1(CNC(c2coc(O)n2)=O)CC(O)CN1C(=O)Cc1ccsn1 32082,C(=O)(CCC(=O)NCC1CCOC1C(=O)NCC1(O)CCC(C)C1)NC 32083,CCC(CC)(CC)C(=O)NC1CC2CC1N(C(C1CC1c1ccccc1Cl)=O)C2 32084,c1(OCCC)c(Cl)cc(NC(c2cnc(OC)c(F)c2)=O)cc1Cl 32085,Cc1c(OC(F)(F)F)cccc1C(=O)NC1CCN(c2ccnc(O)c2)CC1 32086,CC(C)S(=O)(=O)CC(=O)NCC1(CNC(C2CCCO2)=O)CCC1 32087,c1(C(=O)NCCCC(C)NC(=O)C(C)C#N)cncc(C(=O)OC(C)(C)C)c1 32088,C1(CNC(CCCC=C)=O)CC2CCC1N(C(=O)Cc1cc(C)cs1)C2 32089,C1(CNC(C2CCC(C)(C)C2)=O)(CO)CCN(C(=O)CC2SC(=N)NC2=O)CC1 32090,C1(SCC(=O)NCCN(CC(C)O)C(c2ccsc2C(F)F)=O)CCOC1=O 32091,c1(CN2CCC(NC(c3cc(Cl)ccc3Cl)=O)C(O)C2)cncc2ccccc12 32092,C1(NC(C(CC(C)C)N(C)C)=O)COC2(C1)CN(C(=O)Cc1ccncc1Cl)C2 32093,CC1(C)CC(C(=O)NCC(O)CF)N(C(=O)C=Cc2ccco2)C1 32094,C1(CCNC(=O)Cn2cccc2)CCCN(C(c2sc(Cl)cc2Cl)=O)C1 32095,c1(C(N2CC(CC(C#C)C)C2)=O)cc(F)c(C)cc1Cl 32096,N(C1CCc2ccccc21)C(=O)Nc1nccc(C=NO)n1 32097,C1(C(C)C)CCC(C(=O)NCCC(C)NC(=O)CCC(C)N(C)C)CC1 32098,C(=O)(C(F)(F)C(C)O)NC(CNC(c1c(C(=O)OC)nn(C)n1)=O)C(C)(C)C 32099,Cc1cn2cc(NC3(CO)CCN(C(=O)C(=O)NS(=O)(=O)C4CC4)C3)ccc2n1 32100,c1(C(=O)NC23C(CN(C(C(C=C)(C)CC)=O)C2)C3)ccc([N+](=O)[O-])c(N)n1 32101,N1(C(c2ccc(C)cc2)=O)CCCN(C(=O)C(C)c2cc[nH]n2)C(CO)C1 32102,C1(CC)CN(C(c2sccc2C)=O)CCN1C(C1CCC12CCC2)=O 32103,C1(C(N2CC(=C)C2)=O)CC(=O)CN1C(=O)CCc1cccn1C 32104,C1(NC(CC(CCC)(C)C)=O)CC(C2CCN(C(=O)C(C)c3ccco3)CC2)C1 32105,C1(N(C(CN(C)CC)=O)C)CCC2CN(C(c3ocnc3C)=O)CC12 32106,C(CC(=O)NCC(CO)NC(=O)CC1CC(OC)C1)OCC#C 32107,c1(C(=O)NCC2N(C(CC(C=C)C)=O)CCC2)csc2c(O)ccnc12 32108,c1(N2CCC(NC(c3cc(I)ccc3Br)=O)C2)ncnc2ncc(Br)cc12 32109,c1(C(=O)NCC(C)CNC(=O)CCn2cnccc2=O)ccc(N)c(Cl)c1O 32110,CCC(C)CCCC(=O)N1CC(NC(C2CN3CCC2CC3)=O)C(C)C1 32111,Cc1c(C2CC2)nc2ccc(Br)cc2c1C(=O)N(C)C.C12CN(CCO1)C(=O)C2 32112,c1(SCC)ccc([N+](=O)[O-])cc1C(=O)NC1CN(C(=O)C#CC2(C)CC2)CC1C 32113,CC1(C)c2[nH]nc(NC(c3ccc(F)c(Cl)c3)=O)c2CN1C(c1nc[nH]n1)=O 32114,C1(c2ccccc2)(CC(=O)NCC2CN(C(=O)Nc3ccccn3)C2)CCCO1 32115,c1(C(=O)NCC(CC)NC(c2cnccn2)=O)nonc1N 32116,Cc1nc2c([nH]1)CC(C(=O)N(C)CCNC(c1ccc(C(C)C)o1)=O)CC2 32117,Cc1ncc(C(N2CCCCC2CCC(=O)NC(C)CS(C)(=O)=O)=O)c(=N)[nH]1 32118,Cc1ncc(NC(=O)CC2C3CN(C(=O)C(N4CCOC4=O)C)CC23)cc1Br 32119,Cc1cc(N2CCC(NC(C3CCCC3(C)C)=O)C(F)C2)nc(S(C)(=O)=O)n1 32120,c1(C(=O)NC2CC(CNC(C(C)(O)C3CCC3)=O)C2)cc(Cl)nc(Cl)c1 32121,C=C(C)CC(C(=O)NCC1CC(C)(C)CN1C(=O)Cc1cnn(C)n1)NC(C)=O 32122,c1(C(=O)NCC2CCCN(C(C(C)(C)CC#N)=O)C2)cc(F)cc2nc[nH]c12 32123,C(=O)(C1CCCn2cnnc21)N(CCCNC(=O)CC1CCCS1(=O)=O)C 32124,Cc1nc(C(N2CCC(C(=O)N(C)C)C2C)=O)c(C)s1.C1(C2CC2)C(=O)N1 32125,C#CCC(CC(=O)N1CC(NC(=O)CCOCC)C(C(F)F)C1)c1ccccc1 32126,C1(NC(C)=O)CCCC(NC(c2cc(-c3ccccc3)[nH]n2)=O)CC1 32127,N1(C(C(C=C)O)=O)CC(C(N2C(C(=O)OC)CC2C)=O)CC(C)C1 32128,Cc1coc(C(=O)NC(C)(C)C(C)NC(c2cc(C(N)=O)no2)=O)c1C 32129,C1(C(=O)NC2CN(C(c3cccc(Cl)c3Cl)=O)C2)CCC2CC2CC1 32130,C1(C(N(CCCC(=O)NC(CCOC)COC)C)=O)CC=NC=CN1CC 32131,CCCCCCCCCCC(=O)NC(C)CN(C(=O)C(c1ccc(Cl)cc1)O)C 32132,c1(C(N2CCC3CCC(C2)N3C(=O)CSC(F)F)=O)cc2cccc(F)c2o1 32133,c1(C(N2CC(N(C(C=CC(C)C)=O)C)C(F)C2)=O)cc2nccn2c(O)n1 32134,C1(CNC(CCC(C)C)=O)CC2CCC(C1)N2C(=O)C(C)SCc1cccnc1 32135,c1(OC(C(=O)NC2(C=C)CC2)C)ccccc1Br 32136,c1(C(N2C(C#C)CCC2)C(=O)NC2CC(F)(F)C2)cccc2[nH]ncc12 32137,c1(C(N2CC(COC)N(C(c3n[nH]c(C)c3F)=O)CC2)=O)cnn2ccn(C)c12 32138,CC1(CNC(=O)CC2(CNC(C3OC4CCC3C4)=O)CC2)CCCCO1 32139,CCCCC(CNC(C1CC(OC)(OC)C1)=O)NC(=O)CC1CCC(=O)N1C 32140,C1(CNC(=O)CCC2CCC(=O)N2)CN(C(=O)C2CC2)CCC12CCC2 32141,c1(-c2c(C)nc(CC)s2)cncc2sc(C(=O)Nc3cc(C)c(F)cc3Br)cc12 32142,c1(CC(=O)NC(C2CN(C(C(C)c3cc[nH]n3)=O)C2)C)cccc2cn[nH]c12 32143,CC1(C)C(C(=O)NCC(P(C)(C)=O)c2ccccc2)(CN)C1(C)C 32144,C(=O)(C(F)(F)CC(C)C)NC(CNC(c1c(C)nc(CO)s1)=O)CO 32145,C1(CNC(CC(C)C2CCCO2)=O)CCN(C(=O)C(C)(C)n2ccnn2)CC1 32146,c1(C(N2CC(SC)C(NC(=O)CCSC(F)(F)F)C2)=O)ncnc2c1ccn2C 32147,c1(-c2cc(C)cc(OCC)c2F)cccc2[nH]nc(C(=O)NC(C)(C)CO)c12 32148,Cn1ccc(S(=O)(=O)NCc2cnc(OCC3CCCN3)cn2)n1 32149,C#CCCCC(C)C(=O)N(C1CC(C#N)C1)CC(=O)NCC1CCC(=O)NC1 32150,N1(C(C2CN(C)C2)=O)CCC2C(CCN2C(=O)CCc2ccc(F)cc2Cl)C1 32151,C1(C(N(C)Cc2cnc(C)s2)=O)CCN(C(c2cnc(C(C)C)nc2)=O)CC1O 32152,N1(C(C(c2n(C)cnc2)O)=O)CCN(C(c2cocn2)=O)C(CO)C1 32153,c1(OC)cc(C)cc(C(=O)NCC2CC(O)CN2C(=O)CC(=O)N(C)C)c1C 32154,c1(C(=O)NCC2CC(F)(CNC(C(CC#C)C)=O)C2)cc(C)c(C)nc1C 32155,c1(C(=O)NC2C(NC(CC)=O)CCC2)sc(O)nc1C 32156,c1(OC)nccc(C(=O)NC2(CO)CN(C(=O)C(CCSC)NC(=O)C3CC3)C2)n1 32157,C1(CNC(C2CCN(CC)CC2)=O)CC2(C1)CN(C(=O)C=CC(=O)NC1CC1)C2 32158,Cc1c(CN(C)C(=O)NCCC2COCCO2)cccc1F 32159,N1(C(=O)NC(Cc2ccoc2)CC2CCOCC2)CCC2(CC1)CSC2 32160,N1(C(CC(C)SC)=O)CCC2(CC1)CN(C(=O)CC1COCCO1)C2 32161,c1(CNC(C2(CCC)CC2)=O)nc(CNC(=O)CNC(=O)CN(C)C)cc(O)n1 32162,C1(NC(CNC(C(CC)CC)=O)=O)CC2CC(NC(C3CNC(=O)C3)=O)CC2C1 32163,C1(CC=C)(NC(=O)CSCc2nccn2C)CCN(C(C23CC(F)C2C3)=O)CC1 32164,Cc1nc(NCC(n2cc(C3CC3)nn2)C)cc(N2CCOC(C3CCC3)C2)n1 32165,C(=O)(C1=C(C(=O)N2CC(N(C(=O)Cc3ccon3)C)C2)CCC1)OC 32166,N1(C(C2N(C)CC(O)C2)=O)CCOCCC1C(=O)N(CCCN=[N+]=[N-])C 32167,c1(C(=O)OCc2cc(CC(=O)OC)no2)sc(C)c(Br)c1C 32168,c1(OC)cnc(NC(C2CC23CN(Cc2cc(C)[nH]c2C)C3)=O)c(F)c1 32169,N1(C(C2C(=C)CC2)=O)CCN(C(=O)CC2CC3CCC(C2)C3)CC12CCC2 32170,C(=O)(C1=NOC2COCC12)N(C(C)CNC(C1C2(CC2)C12CC2)=O)C 32171,C(N=c1cc(C)nc(C(=O)NC)[nH]1)C1CCC(NC(CNS(NC)(=O)=O)=O)C1 32172,N1(C(C2C(=C)C2)=O)CCC(O)C(NC(=O)Cc2csc(-c3ncccn3)n2)C1 32173,CC(CC(N)=O)C(=O)NCC(C)(C)CC(=O)NC1CC2C=CC1C2 32174,Cc1cc(F)sc1C(=O)NC1(c2ccccc2)CCN(C(c2nonc2N)=O)C1 32175,N1(C(C2(NC(c3c(F)cncc3F)=O)C(C)CCC2)=O)Cc2cccnc2C1 32176,Cc1ccc(N(CCCNC(=O)C2=CC3CCCC23)C(C)C)c([N+](=O)[O-])c1 32177,CN1CCC(CC(=O)NCC2COCC2NC(c2ccc(C(F)F)nc2)=O)C1=O 32178,C(c1ccc(C(N)=O)o1)=CC(=O)NCC(CC)N(CC(CCC)C)C 32179,c1(CC(N2CC(O)(CN(C)C(c3cccc(F)c3O)=O)C2)=O)cc(Cl)ccc1Cl 32180,CC1CN(c2nnnn2C)CCC1CNC(=O)Cc1ccnc(F)c1 32181,c1(C(=O)NC(C2CCN(C(C3C(CC)C3)=O)C2)C)ccc(Cl)nc1 32182,C1(C(=O)NCC2C(C)(C)C(NC(c3ccc(Cl)o3)=O)C2)CCc2[nH]nc(O)c2C1 32183,C1(CNC(C(C)OCCCC)=O)CCCCN(C(=O)CC2(CSC)CC2)C1 32184,N1(C(C2N(C)CCOC2)=O)CC2(CCN(C(C3C4CCN3CC4)=O)CC2)C1 32185,CCC(C(=O)N(C1CC1)Cc1cc(OC)cc(OC)c1)C(C)(F)F 32186,C1(C(=O)NC(C)CCNC(C2CN(C(=O)OC(C)(C)C)C2)=O)CC2C(C1)C2(C)C 32187,C1(NC(CN(CCOC)C)=O)CN(C(=O)C(c2ccc(Cl)cc2)C)CC12CC2 32188,N1(C(=O)Cc2cn[nH]c2)CCCC(C2CN(C(C3COCCC3(F)F)=O)C2)C1 32189,C(CC(C)C)(C(=O)N1CC(N2CC(NC(=O)CC3(CSC)CC3)CC2=O)C1)OC 32190,c1(C(N2C(C)CC(NC(C3CCCC3(C)C)=O)CC2)=O)cncc(N=[N+]=[N-])c1 32191,N1(C(CN(C)S(N)(=O)=O)=O)C2CCC1CN(C(c1ccc(N)cc1)=O)CC2 32192,C(=O)(N=c1[nH]nc(C(C)(C)C)s1)NCC1CCCN(C(C)C)C1=O 32193,C1(CNC(CCN(C)CC)=O)CCCCN1C(c1onc(C)c1C)=O 32194,c1(C(=O)NC2C(NC(CC3OCC(C)(C)OC3)=O)C2)ccc(Cl)c(Cl)c1O 32195,c1(C(N2CCCC(N(C(c3cnco3)=O)CC)C2)=O)cnn2cccc(Cl)c12 32196,c1(C(=O)NCC2(NC(COC(CC)C)=O)CCCCC2)cn2cnnc2cn1 32197,n1(CC)cc(Cl)c(C(=O)NC2(CF)CCN(C(=O)CSc3cnn(C)c3)C2)n1 32198,C#CC1CC1C(N(C1CC(NC(C2CC(OC3CC3)C2)=O)C1)C)=O 32199,N1(C(c2c(C)nsc2N)=O)CC2(CC(C(=O)NCC3(F)CC3)CO2)C1 32200,c1(C(N(C2CCCN(C(C(C)(C)OCC)=O)C2)C)=O)nc(O)nc(O)c1F 32201,CC(C)(C)CC(F)C(=O)N1CC(CNC(=O)CSCC(F)F)C(F)(F)C1 32202,CC1(C(N2CC(C3CCCO3)C2)=O)CN(C(C2CCC(=O)C2)=O)C1 32203,Cc1oc(C(=O)NC(C)CN(C)C(C2CC2(C)C)=O)cc1S(=O)(=O)N(C)C 32204,N1(C(c2cc(C(=O)OC)co2)C(=O)NCCC)CCC2CC12C(=O)OC 32205,c1(CC(=O)NC2CC(NC(c3ccnnc3O)=O)C2)cc(F)cc(F)c1Br 32206,N1(C(CC(C=C)C)=O)C(C)CC2CN(C(=O)C(C3(O)CCCC3)F)CC12 32207,C1C(F)(F)CCC(=O)N2CCC(CC2)c2cn1nn2.C(CO)(CC(C)(C)C)OC 32208,Cc1c(S(N)(=O)=O)cnc(NC(c2ccc(Br)cc2)C(F)(F)F)c1Br 32209,c1(C(N2CC3C(NC(c4ncn(C)c4)=O)(C3)C2)=O)c(F)cc(F)cc1Cl 32210,c1(C(=O)NCC(C)CNC(=O)C(C)N(C)C2CC2)cccc2cncn12 32211,C1(C(=O)NC(C#C)C2CCC2)C2CC3C(C2NC(=O)CCCCSC)C13 32212,c1(CC(C(=O)OC)Nn2cc(C3CC(F)(F)C3)nn2)ccc(OC(F)(F)F)cc1 32213,c1(CN2CC(NC(c3c(C)ccc(Br)c3)=O)C(C#N)C2)ccc2nc[nH]c2c1 32214,C(C(=O)N(C)Cc1cnccc1C)(C(C)(C)C)NC(C(C)=C(CC)C)=O 32215,N1(C(COc2cccc(OC)c2)=O)CC2CC(NC(=O)C(C#N)C(C)C)C(C2)C1 32216,c1(C(=O)NCCN(C(c2cc[nH]c2)=O)CC)nccc2ccn(C)c12 32217,C1(NC(C=C(C)C)=O)CN(C(c2snnc2C(C)C)=O)CC1C 32218,C1(CC)CN(C(C2CN3CCC2C3)=O)CC1C(=O)NC1CN(c2ncco2)C1 32219,N1(C(C(CCCC)O)=O)CCN(C(=O)CCOCC(C)(C)C)C2(CCC2)C1 32220,C1(C)(C(=O)NCC(=C2CN(C(CCCOC(C)C)=O)C2)F)CCCS1(=O)=O 32221,C1(CC(N2C(CNC(C3(C)CCCO3)=O)CCC2)=O)COCCN1CC(F)(F)F 32222,c1(C(N2C(C(N(C(=O)Cc3cnccc3C)CC)CC)CCC2)=O)cnc(C)nc1 32223,CC1CC2CCCC2N1C(c1sccc1CNC(=O)C(N1CCOCC1)C)=O 32224,N1(Cc2cc(C)[nH]c2C)CC2(CCN2C(c2c[nH]c(C(C)(C)C)c2)=O)C1 32225,C1(C(=O)NCC2(C(N)=O)CN(C(C(C)C#N)=O)C2)CC2(CC(=O)N2)C1 32226,O=C1COc2c(C(=O)NC(CNC(C3C(F)(F)C34CC4)=O)C3CC3)cccc2N1 32227,C1(CCNC(=O)CCCN2CCCC2)CC(F)(F)CN1C(=O)Cn1cnnc1 32228,c1(C(=O)NC2(C)CC(NC(C3(CC(F)F)CCC3)=O)C2)ccncc1O 32229,C(c1cnc2ccccc2n1)=CC(N1CCC(NC(C2C(C)C2)=O)C12CC2)=O 32230,S(=O)(=O)(c1ccc(NC2CCOC(C(C)C)C2)cc1Br)NCC(C)(C)OC(C)C 32231,c1(C(=O)NCC(C)(CC(C)C)NC(C(CC(=C)C)C)=O)cn2cc(C)ccc2n1 32232,C1(CCC(=O)NCC(C)(C2CC2)OC)CCCCN1C(c1cccnn1)=O 32233,c1(C(=O)Nc2n[nH]cc2C(F)F)ccc(-c2ccccc2)c(F)c1 32234,C1(CNC(CC=C(C)C)=O)CC2(CCN(C(c3cn(C(C)C)cc3C)=O)C2)CO1 32235,CCC(C(C)(C)O)NC(c1cnn(CCNC(C2CCC(CC)C2)=O)c1)=O 32236,C(=O)(CCCCC(N)=O)NC(C(=O)NC1CCCN(C)C1)CO 32237,C(N=c1[nH]c(=NCCNC(C2CCCCC2)=O)[nH]c2ncn(C)c12)c1n(C)ccc1 32238,C#Cc1ccnc(C(N2CCN(C(=O)C(CC)CC=C)C(CC(F)F)C2)=O)c1 32239,C1(F)(CNC(C(CCCC)C)=O)CCCN(C(=O)Cc2ccc3ocnc3c2)CC1 32240,CC1(C)CC(CNC(=O)C(F)=C2CCC2)N(C(=O)CC2CC3CC3C2)C1 32241,C(=O)(CCC(C)S(C)(=O)=O)NC(CNC(c1c(C)nn(C2CC2)c1Cl)=O)C1CC1 32242,CCC(C)C(C(=O)N1CCOCC1)OC.N12CC(c3nn[nH]n3)(C1)C2=O 32243,c1(C(=O)NCC2CN(C(CC(CC)C3CC3)=O)CC2O)cccc2scnc12 32244,CC(c1ccccc1Cl)=CC(=O)NC1CC(CNC(c2cc(C)nc(C)n2)=O)C1 32245,Cc1ccc(O)c(C(=O)NCCCNC(c2ccn(C)n2)=O)n1 32246,c1(C(=O)Nc2c(C)[nH]nc2Cl)cc2n(n1)CCCN(Cc1cc(F)ccc1I)C2 32247,N1(C(C=CC=CCC)=O)CC(F)(F)CC1CNC(=O)CCCc1ccc(Br)cc1 32248,c1(C(C(=O)NC(=O)Nc2cn(CC)nc2)N2CCC2C2CCC2)nn(CC)cc1Cl 32249,N1(C(c2ccc(CCC)[nH]2)=O)CC(NC(c2cccc(N)c2)=O)CC1(C)COC 32250,C1(C(=O)OC)C2CC1N(C(=O)C=C1CCN(C(=O)C=CC3CCCC3)C1)C2 32251,c1(N2CCN(C)C(C)(C)C2)nc(N2CCOCC(C)(C)C2)nc2c1SCC2 32252,N1(CC)CC(C(=O)NC(C)CNC(C2(Oc3ccccc3)CC2)=O)NC1=O 32253,C(CCCCCC(=O)NC1CC(CC(=O)OC)C1)n1cc(-c2c(C)ncs2)nn1 32254,N1(C(COC)=O)CCCC2(NC(c3ncc(C(F)(F)F)s3)=O)CC2C1 32255,C(CC(=O)NOCCC(C)O)(C(F)(F)F)NC(C1(COCC)CC1)=O 32256,c1(C(N2CCC(C)(NC(c3nc(C)oc3)=O)CC2)=O)cnc(O)c2cncn12 32257,C(CC(C(=O)NC1(CC)CCC1)NC(=O)Cc1ccc(C)s1)=CC 32258,c1(C(N2C3CC(CC(NC(C(C=C=C)C)=O)C3)C2)=O)ccc2ccncc2n1 32259,C(CNC(c1cc(OC)cs1)=O)(CCC)NC(C(C)=C(CC)C)=O 32260,C12(C(N(CCN(C)C(C3(n4ccnn4)CC3)=O)C)=O)CC(C1)C(C)(C)O2 32261,C1(F)(C(N(C(CNC(c2n(CCC)ccc2)=O)C2CC2)C)=O)CCCCC1 32262,N1(CCNC(C2CN(C(c3c(CC)cno3)=O)CC(C)C2)=O)CC2(CCOCC2)C1 32263,O=C1CN(C(c2ccnc(N3CCCCC3)n2)C2CCOC2)C(=O)N1.N1CCCC1 32264,N1(C(CNC(CCC)=O)=O)CCC(C2CCCN(C(c3coc(Cl)c3)=O)C2)C1 32265,Cc1cnc(N(C23CC(N)(C2)C3)C(C23CCC(CC2)CC3)=O)nc1C 32266,C(=O)(CCCCCF)NCC1CCCC(NC(CN2C(C)CCC2)=O)C1 32267,C1(CCO)CCCN1NC(=O)C=Cc1cocn1 32268,N1(C(c2cc(CCC)[nH]n2)=O)CCCC(N2CCN(C(C3CCOC3)=O)CC2)C1 32269,Cc1ccnc(C(C)(C)C(=O)NC(C)CN(C(=O)C(F)OC(F)(F)F)C)c1 32270,N1(C(c2c(C)c(F)ccc2)=O)CCCC2CN(C(=O)C3=CCCS3)CCCC12 32271,C#CCC(CC(=O)N(C)CC1(C)CCCO1)NC(C12CCCC1OCC2)=O 32272,c1(OCC(=O)N(CCC)CCN(C(=O)C(C)=C(C)C)CC)cccc(O)c1 32273,N1(C(C(OCC)OCC)=O)CCC(C(=O)NC2CCC2C(F)(F)F)C(O)C1 32274,C(=O)(CCC(C)(C)N1CCOCC1)N1CCCC(CNC(CC(CC)OC)=O)C1 32275,C1(CC)CCCN1N(C)C.N1(CCNC=O)CCCC1=O 32276,c1(C(N2C(C)CC(NC(=O)CCOCC3CCC3)C2)=O)cc(F)cc2nc[nH]c12 32277,CN1CCCC1C=CC(=O)NCC1(O)CCN(C(c2cscn2)=O)C1 32278,c1(C(N(c2cccc3c[nH]nc23)C2(C#N)CCC2C(=O)O)=O)ccc2c(c1)CCC2 32279,C1(C(N(C2CN(C)C2)C)=O)CC12CCN(C(c1cscc1Cl)=O)CC2 32280,C(=O)(CCCCCC#N)NCC1C(NC(c2ccc(OC)nc2OC)=O)CC1 32281,N1(C(C(Cn2ccnn2)NC(CCCOC)=O)=O)CC2C(C1)C2(C)C 32282,c1(C(=O)NC2C(CNC(COCCC=C)=O)CCC2)cc(C)nc2ccnn12 32283,N1(C(Cc2c(C)ccs2)=O)CC(C2CN(C(c3cc4ncccc4s3)=O)C2)C1 32284,C12(C(=O)NCC=CCCOC)CC1CN(C(=O)C(C)=NOCC#N)C2 32285,c1(C(N2CCCC(N(C(=O)C(F)C(F)(F)F)CC)CC2)=O)cc(C)nc(Cl)c1N 32286,C1(C(=O)NCC(CC=C)NC(C2CC2c2cn(C)nc2C)=O)CCCCN1N=O 32287,C1(C)(C(N(C2CC(C#N)C2)CC(=O)NCCC2(C)N=N2)=O)CCOC1 32288,C(C(O)C(=O)NC1CCC1CNC(=O)C(=O)NCCCC)=CC 32289,Clc1ccc(CCCCN(c2ccccc2)c2ccccn2)cc1Cl 32290,C(CC(=O)NOCC1CCC1)C1CC(NC(CC2C(C)C2)=O)C1 32291,C1(O)(CN(C(c2cnc(OCC)s2)=O)C)CCN(C(=O)C2=CCSC2)C1 32292,N1(C(N(C2CCCC2NC2CCCCC2)CCOC)=O)CCCCCC1 32293,CCCCC(C)C(=O)N1CCCCC1C1(NC(=O)CCNC(C2CCC2)=O)CC1 32294,N1(C(C(C)(C)OC)=O)CC2(C(=O)NCC(CC3CC3)CO)CC1CO2 32295,c1(SC)nc(N2CCC(NC(=O)CCc3cncn3C)C(F)C2)cc(C(F)F)n1 32296,C(=O)(C1=COCCC1)NC1CCN(C(c2c(C)nsc2)=O)C1 32297,N1(C(CN(C)C(C2CCN(c3ccncc3)CC2)=O)=O)CC(N(C)C)C(O)C1 32298,C1(NC(CN(C(C(C)OCCCC)=O)C)=O)CCC(C(C)O)CC1 32299,Cc1cnc(C)c(C(=O)NCC2CCCN2C(=O)CCCNS(C)(=O)=O)c1 32300,c1(-c2nc(-c3scc(C)n3)nn2CC(C)(C)CO)cc(Cl)ncc1Cl 32301,C1(CNC(CC(CCC)CC)=O)CCCC2(CN(C(c3ccnnc3)=O)C2)O1 32302,c1(OC)ccoc1CNC1CC(C(N2CCCC2C(F)(F)F)=O)C1 32303,Cc1c(C(N2CC(NC(=O)C(C)(C)C)CCC2C)=O)cc(Br)cc1N 32304,S(=O)(=O)(C1COC(C)(C)C1)NC(CNC(NOCCCOC(C)(C)C)=O)=O 32305,CCN=C(NCc1cccc(OC(F)F)c1)NCC1CCC(C)C1 32306,C12(NC(c3ccc(=O)oc3)=O)CCC1CN(C(=O)CC1C=CCC1)C2 32307,O=C(N=c1cc(C2CCOC2)[nH][nH]1)C1CN(S(=O)(=O)CCC(F)(F)F)CCC1O 32308,N1(C(C(=O)NCC)=O)CC(CNC(C2CCC(N(C)C)CC2)=O)C(O)C1 32309,C12(NC(C(CC=C)CC=C)=O)CCCCC1N(C(c1cccc(F)c1F)=O)CC2 32310,Cc1cc(C(=O)NC(C(C(=O)NCC2CN3CCC2C3)C)C)sc1C 32311,c1(C(N(CCCCNC(=O)COC2CCOC2)C)=O)c(Cl)ccc(O)c1N 32312,c1(CSC(C(=O)NCC(C)(C)NC(C2C(OCC)CC2)=O)C)ccccc1Cl 32313,N1(C(c2ccc(C(N)=O)nc2)=O)CCN(C(=O)C2=CCSC2)C2CCCCC12 32314,N1(C(C2N(C(c3c(C)oc(CO)c3)=O)CC(=O)NC2)=O)CCOC2(CCC2)C1 32315,C#Cc1ccc(C(=O)NC(C)C(C(C)C)NC(=O)CN(C)CCC)c(F)c1Cl 32316,C1(CNC(C2(COC)CCC2)=O)CCC(C)(C)CN1C(c1ccc(C)nc1)=O 32317,C(C1=NOC2CC12)NC(=O)NCC(=O)Nc1ccc(C(CC)=O)cc1 32318,C(=O)(C1Cc2ccccc21)N1C(CN(C)C(c2csc3nnsc23)=O)CCCC1 32319,Nc1[nH]c(=O)c(Cl)nc1C(=O)NCC1CCN1C(c1ocnc1C1CC1)=O 32320,Cc1nc(C(=O)NC2(CNC(C3(CN(C)C)CC3)=O)CCCC2)c2n1CCCC2 32321,N1(C(C(C2CN(C(C3CC=C(C)CC3)=O)C2)O)=O)CCC(C)(O)C(O)C1 32322,N#Cc1cnccc1COC(c1ccc(-c2ccc(Cl)cc2)nc1O)=O 32323,CC(CF)CC(=O)NCc1cn(C2COCC2NC(C2CC(C(C)C)C2)=O)nn1 32324,n1(CC)ccnc1C(=O)NCCC1CN(C(=O)CC2(c3ccccc3)CC2)C1 32325,C(CC(C)C)(C(=O)OC)Sc1ccccc1CC(=O)OC.C12CN(CC1C#N)C2 32326,N1(C(=O)Nc2cccc(-c3nccc(C)n3)c2)Cc2c(F)cccc2C(C)(C)C1 32327,C12(NC(c3cc(O)cc(Cl)c3)=O)CCCC1CN(C(=O)CC1CCCC1(F)F)C2 32328,CC1CCCCN1CC(N1CCN(C(=O)Nc2nccn2C)CC1)C 32329,C=CCC(CC)C(=O)NC1CN(C(C2C3CCC2(c2ccco2)C3)=O)CCC1C 32330,Cc1cc(C(N2CCC(C)(CNC(C3CC4CC3CC4O)=O)CC2)=O)ccc1O 32331,C12(C(=O)NC(C(C(C)C)NC(c3cnc(S)nc3)=O)C)CC3CC1C2C3O 32332,c1(SCC(=O)NC2CCN(CCC)C2)nc(C)cc(C)n1.C1(N)CC1C1CCC1 32333,c1(C(C(=O)NC(C(C)C)CNC(c2nnsc2C(F)F)=O)C)cc(F)cc(F)c1 32334,N1(C(CCc2c(C)cccn2)=O)CCCN(C(=O)C2=CCOCC2)CCC1 32335,c1(C(=O)NCC#CCNC(=O)COCC2CCC2)cn2ccnc2cn1 32336,N1(C(C(C)OC)=O)CCCC(N(C)C(c2ccc(-n3cncn3)cc2)=O)C1 32337,c1(C(=O)NC2(C)CCN(C(CSCCN(C)C)=O)C2)ccc2c(c1)CNC2=O 32338,c1(C(=O)NCC(CNC(C(C2CCCOC2)OC)=O)O)c(F)ccc(F)c1F 32339,c1(C(=O)NC2CCC(CNC(c3c(C)cc[nH]3)=O)C2)cc(F)cc2nccnc12 32340,c1(OC(C)C)ccccc1-c1nc(Cc2cn[nH]c2)n(Cc2ccccc2Cl)n1 32341,C1(C)(CC)CCN(C(C2CCC(NC(=O)C(O)CCN(C)C)CC2)=O)C1 32342,C1(NC(c2ccc3occc3c2)=O)CCCC12CCN(C(c1cncs1)=O)CC2 32343,c1(C(=O)NCC(CNC(C2(COC)CCOCC2)=O)C)nc(C)ccc1OC 32344,C1(NC(CC2CC(C)C2)=O)C2CC3C1C3C2C(=O)NC1Cc2ccccc2C1 32345,C(=O)(C(Cc1ccc(O)cc1)C(F)(F)F)NC1C(CNC(CCC=C)=O)CC1 32346,C(=O)(C1=CCCOC1)NCCC1CC(NC(C2CC(N3CCCC3)C2)=O)C1 32347,Cc1cc(C(=O)Nc2cccc(CNC(c3scnc3C3CC3)=O)c2)cnc1O 32348,CC1C(C(=O)NC2CCN(C(=O)C=Cc3cnc[nH]3)C2)OC2CCCCC12 32349,CC(=O)CCCC(=O)NCC12CC1CN(C(c1ccc(C)n1C)=O)C2 32350,C1(C(N2C(CNC(=O)C(=O)NCCC(C)C)C(O)C(O)C2)=O)CCCC(F)(F)CC1 32351,CCC(F)(F)C(C)(C)C(=O)N1CCC(C(C)NC(C2(C#N)CC3CC3C2)=O)C1 32352,c1(C(N2C3CCC(NC(c4cnc(Cl)s4)=O)C(C3)C2)=O)cnc(O)c([N+](=O)[O-])c1 32353,C(=O)(CCNC(c1cnsc1)=O)NC1C(C)C1 32354,c1(C(=O)NC2CCN(C(c3c[nH]cc3Br)=O)C2)ccc2c(c1)CCC2(F)F 32355,CC(C)CC(C)(CNC(=O)CCOC1CN(C(=O)CCc2ccoc2)C1)N(C)C 32356,Cc1cc(NC(=O)CC2CCN(C(c3cc(Cl)ccc3O)=O)C2)nc(Cl)c1 32357,N1(C(C(C)C)=O)CC(NC(c2ccc3ncoc3c2)=O)C(S(C)(=O)=O)C1 32358,c1(OC)ccc(C2(CNC(=O)C(C)OC3CC=CCC3)CC2)cc1OC(F)F 32359,c1(C(N(C2CN(C(C3(OC)CS(=O)(=O)C3)=O)C2)C)=O)cc2c(C)c(F)ccc2[nH]1 32360,Cc1cn2ccc(C(=O)NCCCN(C(=O)CCNC(N)=O)C(C)C)cc2n1 32361,N1(C(C2CCN(C(C)=O)CC2)=O)CCC2(CCN(C(c3nc(C)sc3C)=O)C2)C1 32362,N1(C(CCCOC)=O)CC(NC(=O)CN(C)S(N)(=O)=O)CCC1C 32363,c1(OC)cc(NC(c2cc(-c3ccnc(F)c3OC)cs2)=O)c(C)cn1 32364,N1(C(C2C(C)(Br)C2)NCc2nnc(CC3CC3)s2)C(=O)c2ccccc2C1=O 32365,c1(OC)cc(NS(=O)(=O)CC(C)C)nc(Nc2ccc(C(F)(F)F)nc2)n1 32366,N1(C(c2c(CC)non2)=O)C2CCCC1CC(NC(c1cnnc(O)c1)=O)C2 32367,C1(COC)CN(C(=O)CCc2cnc(O)[nH]2)CCN1C(=O)CS(C)(=O)=O 32368,C(=O)(CN=c1[nH]c(C)cs1)NCC1N(C(c2nc(COCC)sc2)=O)CC(F)C1 32369,c1(C(N2CC(O)(CCNC(C3(F)CC3)=O)C2)=O)cc(F)ccc1Br 32370,C1(CNC(CCC(=O)NC)=O)C(C)CCCN1C(=O)CCC(C)CN(C)C 32371,N1(C(c2c(C)cc(CNC(C3CC34CCCC4)=O)o2)=O)CCCC2C(=O)NCC12 32372,N1(C(C(C)OCCC(C)C)=O)CCCN(C(=O)C=Cc2cnc[nH]2)CCC1 32373,C1(C(N2CCC(O)(C(C)CNC(=O)CC3CC=CC3)C2)=O)(COC)CC=CCC1 32374,C1(NC(CC2C(OC)COCC2)=O)CCCC2CN(C(=O)CCCC(F)F)CC12 32375,C1(NC(CC(C)C(F)F)=O)COC2(C1)CN(C(C1CC=CC1)=O)C2 32376,N1(C(CC2(OC)CC2)=O)CC(NC(=O)CCc2ccc(OC)nc2)C(C)(C)C1 32377,c1(CC)nc(Cl)nc(N2CCC(NC(C3CCC(NC(C)=O)CC3)=O)CC2)c1Cl 32378,N1(C(Cc2ccn(C(C)C)n2)=O)CCC(C)C1CNC(=O)CC(C)C1CC1 32379,c1(COC)c[nH]ccc1=NC1CC(NC(=O)C=C2CCCCCC2(F)F)C1 32380,CC(C)CC(C)(CNC(=O)C=Cc1ccn(C)c1)NC(c1cn2ccnc2s1)=O 32381,n1(CC)nc(C)c(C(=O)OC)c1C.n1(CCCC)nnnc1C(CC(C)SC)N 32382,O=S(=O)(c1ccc(F)c(Br)c1F)Nc1cccc(-c2ccccc2)c1 32383,C#CCC(CO)NC(C1(CCNC(=O)CCOCC2CC2)CCC1)=O 32384,C1(C(=O)NC2CCN(CC(C)C)CC2)CC2(C1)CN(C(C1CC(C)(F)C1)=O)C2 32385,C(CC(O)C(=O)NCC1(F)CC(NC(=O)C(C)Cc2cccc(F)c2)C1)SC 32386,C1(NC(c2ccc(C(C)C)cc2O)=O)CN(C(=O)CCS(C)=O)C2(CCC2)C1 32387,c1(OC)cc(C(N2CCC2(C)C(=O)NCC2CNC(=O)CO2)=O)cc(Cl)c1 32388,c1(C(N2CCC(C3N(C(C(CCCC)F)=O)CC3)C2)=O)cc(F)c(O)c(F)c1 32389,C12(CNC(C(CC=C)NC(C)=O)=O)CCC(CC1)N2C(=O)C(F)(F)COC 32390,c1(C(=O)NCC(CC)NC(c2c(NC)cccc2F)=O)cc(C)ccc1Br 32391,c1(NC)cccc(CCC(=O)N2CCC2CNC(=O)CC2(CSC)CC2)c1 32392,CC(C)C(C)C(=O)NCC(C1CC1)NC(c1ccc(OC(F)(F)F)cn1)=O 32393,N1(CC(=O)NCCCN(C(C2C(C)COCC2)=O)C)CCCc2sccc2C1=O 32394,c12cccc(c1F)C2.C1(CC(=O)N(C)C)CCCN(CC2CC2)C1 32395,CC1=C(C)CC(C(N2CCC(C(=O)NC3CNC(=O)C34CC4)C2C(C)C)=O)CC1 32396,c1(NC(C(CC)C)C)ccc(S(=O)(=O)N2CCC(C)(C)CC2)c(Cl)c1 32397,c1(C(=O)NC(C(=O)NC2(CSC)CC2)C)c[nH]c(=N)c(C)c1 32398,CCC(C)(C)C(O)C(=O)N1CC(C2(NC(=O)C(C)COC(C)(C)C)CC2)C1 32399,CCC(CC(=O)NCc1ccc(CCNC(=O)CN2CSCCSC2)cc1)OC 32400,C1(CCCC)CCN(C(C2CC(CC=CCNC(=O)Cn3cccc3)C2)=O)C1 32401,C(=O)(C(C)(C)CCC)N(CC=C)C(C)=O.C1(=O)CN1.C1CCNC(=O)CSCC(=O)N1 32402,N1(C(c2cccc(C)n2)=O)CCC2CCN(C(c3cc(Cl)ccc3Cl)=O)CC2C1 32403,c1(C(=O)NCC(C2CCC2)NC(C(C=C)O)=O)cccc2c1CCC2 32404,Cc1cc(S(N)(=O)=O)cc(C(=O)N(C(C)CNC(=O)CCCCC#N)C)c1C 32405,N1(C(c2c(NC)cccc2)=O)Cc2ccc(C(=O)NCC(C)(C)F)cc2C1 32406,Cc1ccc(-c2cc(C(N3CCCC(N(C(=O)C4=CCCS4)CC)C3)=O)n[nH]2)cc1 32407,C(=O)(N=c1[nH]sc2c(Br)cccc12)NC(C(C)C1CC1)OC 32408,CCC(F)(F)CC(=O)N1CCCC1Cn1cc(N2CCCC(CCO)CC2)nn1 32409,c1(CNC(C2(NC(C3CC(C#N)C3)=O)CCOC2)=O)ccc(N2CCCC2)cc1 32410,c1(C(N2CCC(CC(=O)Nc3onc(C)c3Br)C2)=O)cc(F)ccc1[N+](=O)[O-] 32411,CCN=c1ccc(C(=O)NC2CC2NC(c2ccc(C(F)(F)F)s2)=O)c[nH]1 32412,N1(C(CC2(NC(c3cccc4cncn34)=O)CCC2)=O)CCCC(F)(F)CC1 32413,C(C(CC(F)(F)F)NC(C1CCC(=O)N1C)=O)NC(CCSCC(C)C)=O 32414,C1(CNC(C=CC(C)C)=O)CC2(CC(NC(=O)C(C)(C)C3CCCC3)C2)C1 32415,C(=O)(C(C)S(N)(=O)=O)NC1CCN(c2ccc(CC(=O)OC)cc2)CC1 32416,C=CCC(CC(F)F)C(=O)N1CCN(C(=O)CCC(CC)CC)C(CC(F)F)C1 32417,N1(C(C2C(C)(C)CC2)=O)CCC2(CCN(C(c3cnc(C(N)=O)cn3)=O)CC2)C1 32418,c1(C(=O)NCC(CNC(c2csnn2)=O)CO)ccc(-n2cncn2)cn1 32419,N1(C(c2ncn(C)n2)C(=O)NC2CCOC2)CCC(CCC2(O)CC2)CC1 32420,N1(C(C2C(C)C2)=O)CCC(CC(C)(C)NC(=O)Cc2nccn2C)CC1 32421,CC1CN(C(=O)COCCF)CC1NC(=O)C(C)Cc1cccc(N(C)C)c1 32422,c1(C(=O)NC2CC(N(C(C(C3CC3)OCC)=O)C)C2)cc(C(=O)OC)[nH]n1 32423,c1(C(=O)NCC(CC)NC(C2CCN(C)C2)=O)nncc2ccccc12 32424,Cc1ccc(O)c(C(=O)NC(c2cnn(C)c2)C(N2CCC3CC23)=O)c1 32425,c1(OC)ncnc(C(=O)NCCCOCCNC(C2CCNC2=O)=O)c1F 32426,Cc1ccc2ncc(C(N3CCC(C)C3CNC(=O)C(C)(C)CC(F)F)=O)n2c1 32427,C1(NC(c2c(C)nn(C)c2F)=O)COC2(CCN(C(=O)CS(=O)(=O)N(C)C)C2)C1 32428,CCCC(CCNC(C1CCC1CNC(C1(OC)CCOC1)=O)=O)CCC 32429,CCCC(CCC)CC(=O)NC(c1cn(C)nn1)C(N1CCC(O)CC1)=O 32430,C(CCCCCC(=O)NCCc1nncs1)NC(c1cn(CC)nc1)=O 32431,c1(N2CCC=C(C(=O)NCc3cc(C)c(O)c(C)c3)C2)ccnc(S(C)(=O)=O)n1 32432,C1(CCC)(NC(c2csc(C)c2)=O)CCCN(C(c2cccc(=O)n2C)=O)C1 32433,c1(C(=O)NC2CCC(NC(C(CC)(C)OC)=O)C2)cc(OCC2CC2)ncc1Cl 32434,N1(C(Cc2c(C)nc[nH]2)=O)CC(NC(=O)C2=CCOCC2)CC12CCOCC2 32435,n1(CC)nc(C(C)C)cc1C(N1CC2CC1C2NC(=O)CSC1CCOC1=O)=O 32436,c1(C(=O)NC2C(CNC(C(C)c3ccsc3)=O)C2)ccc(Cl)c(F)c1O 32437,C1(C)(N)CN2CCC1CC2.C12CCCC1C(=O)N(C)CC(=O)NC2.CO 32438,Cc1cnccc1C(C)C(=O)NCCN1CCC(NC(=O)C(N)=O)CC1 32439,c1(CC(=O)NC(C(C)NC(C2(CC)CC2)=O)C)cccc(C(=O)OC)c1 32440,n1(CC)cnc2c(NCC3CN(C(C4CCOC(C)C4)=O)C3)nc(Cl)nc12 32441,c1(C(N)=O)csc2c1CCN(Cc1cc(C(F)(F)F)ccc1Cl)C2 32442,C1(C(=O)NCC(CC)NC(=O)CSCC(C)C)CCOC1C(C)C 32443,C1(O)(C(N2C(Cn3cc(C(CC)(O)CC)nn3)C=CC2)=O)CCCC(C)CC1 32444,C(=O)(C(C)(C)C(=O)NC1CN(C(=O)CC(=O)OCCC(C)C)CC1C)NC 32445,c1(C(N(CCCC)CC)=O)nn(C)c2c1CCC2.c12coc(n1)N(CC)C2=O 32446,Cc1c(C(=O)NC2CCCC(NC(c3occc3F)=O)C2)ccn1C(C)C 32447,Cc1cccc2c1CC(C(=O)NCC(C)CNC(=O)C(O)C1CCC1)N2 32448,c1(CNC(c2cc(C(=O)OC)n(C)c2)=O)ccc([N+](=O)[O-])cn1 32449,c1(NC(=O)NCCC#CCC)cnc2ncccc2c1 32450,c1(C(=O)NC2CCC(NC(C34CSC(C3)C4)=O)C2)cc(O)nc2ccccc12 32451,c1(C(=O)NC2CN(C(CC3(c4ccccc4)C(C)(C)C3)=O)C2)ccc(O)c(Cl)n1 32452,N1(C(CCCC)=O)CC2CC1CN(C(=O)C(C(C)C)NS(=O)(=O)c1cnn(C)c1)C2 32453,C1(CNC(=O)Cc2cc(Br)cs2)CN(C(=O)CC2CCC2)CCO1 32454,N1(C(C2CC(=C)C2)=O)CC(CNC(=O)C=Cc2cc(Cl)cc(Cl)c2)OC(C)(C)C1 32455,C1(NC(CCCC#C)=O)CC12CCC(NC(=O)C=Cc1ccsc1)CC2 32456,CC1(C)OCCC1NC(=O)CCC1CC(NC(=O)CCC2CCCCC2)C1 32457,N1(C(C(=O)N(C)C)=O)CCCC(CC(=O)NCc2cccc(CO)n2)C1 32458,C(=O)(CCC(=O)N(C(CNC(c1sc(N(C)C)nc1Cl)=O)C1CC1)C)NC 32459,C1(CNC(C2CCCC(C(N)=O)C2)=O)(NC(c2cc(F)n[nH]2)=O)CCCCCC1 32460,C1(NC(C#CC(C)C)=O)CCCC2CN(C(c3coc(C(C)(C)C)n3)=O)CC12 32461,C1(C(N2CC(C)(CNC(=O)Cc3csnn3)OCC2)=O)OCC2CCCC1C2 32462,CC1CC(NS(=O)(=O)c2cccnc2NCC2(CO)CCC2)c2nccn21 32463,N1(C(C2(CC#C)CCCCO2)=O)CCCCCC(NC(c2ccoc2Cl)=O)C1 32464,C(CC(C)N=c1nc(C#N)[nH]cc1C)NC(CCCCC(=O)NC)=O 32465,c1(C(=O)NCC23CC2CN(C(=O)CCC2CCCCC2)C3)ccn2ccsc12 32466,N1(C(Cc2ccc(C(C)=O)cc2)=O)CCC(NC(c2cnn(C)n2)=O)C(F)C1 32467,N1(C(C(CC)C)=O)CCN(C(=O)CCCCCF)C(CC(=O)NC)C1 32468,Cc1cnc(NC(c2csc3ccccc23)(C)C)c(S(=O)(=O)NCCCCO)c1 32469,N1(Cc2ccc(S(N)(=O)=O)s2)CCC2(COC(=O)N2)C1 32470,c1(Cc2cnc(NC(c3cc(C)nn3C)=O)s2)ccccc1[N+](=O)[O-] 32471,C1(NC(=O)C(O)C2CC2)CCN(C(c2cnn(-c3ccccc3)n2)=O)C1 32472,C1(CCC(=O)N(CC(CC)NC(N2C(C(=O)CCC)CSC2)=O)C)CCC(=O)N1 32473,CC(C)=C=CC(=O)NCCC1(C(=O)NC(C)CC(C)(C)C)CC1 32474,C(c1ccnc2ccccc12)=CC(=O)NC1CCCC1NC(C1CC2CC2C1)=O 32475,S(=O)(=O)(c1cncc(Br)c1)NC1CN(C(C(c2ccccn2)C)=O)CC1F 32476,C(CCCCCN(C(=O)CC1CC=CCC1)C)NC(C1(COC)CC(=O)C1)=O 32477,c1(C(COC(C(C)NS(CC)(=O)=O)=O)=O)ccc(C)cc1C 32478,c1(CCC(=O)N(C)CCOCCN(C(=O)CCC2CCOC2)C)cccnc1 32479,CC1CCC(C(=O)N(C(c2ccccc2)C(=O)NCCNC(=O)C(C)(C)C)C)S1 32480,c1(OC)ccc(S(=O)(=O)N2CC3CCN(Cc4ccc(C)c(F)c4)CC3C2)cn1 32481,C1(C2N(C(C(C)(C)NC(COCC)=O)=O)CCC2)CCCN(C(=O)COC(C)=O)C1 32482,N1(C(c2c(CC)nns2)=O)CCC(C)(C)C1C(=O)NCCc1ccc(C)cc1 32483,c1(C(=O)NCCCNC(C(C)OCCC=C)=O)ccc(F)c2[nH]ccc12 32484,c1(C(=O)NCC2(O)CN(C(c3ncnc(C)c3C)=O)C2)cc(F)cc(Cl)c1N 32485,CC1CN(C(=O)CCCN2C(=O)CNC2=O)CC(C)N(C(=O)C2=NNC(=O)C2)C1 32486,C1(CNC(C(CCC2CCCC2)N(C2CC(F)(F)C2)C)=O)CCCN(C)C1=O 32487,c1(OC)ccc(CCN(C(=O)C(N2CCN(CC(C)(C)C)CC2)=O)C)cc1OC 32488,Cc1ccc(CC(=O)NCCC2CN(C(=O)C=Cc3cccs3)CCO2)cc1 32489,N1(C(c2c(C#C)c[nH]n2)=O)CC(F)(F)CC1(C)CNC(c1c[nH]cc1C1CC1)=O 32490,C=C=CC(C)C(=O)N(CC(=O)N(C)CC1COC(=O)N1)C1CC1 32491,Nc1cc(C(=O)N(CCCNC(c2nc(C3CC3)cs2)=O)C2CC2)cc(F)c1 32492,c1(OC)cc(C(=O)NCC2CN(C(C3CCC=CCC3)=O)C2)cc(C2CC2)c1 32493,Cc1c(OCC(=O)NC23CC(CNC(c4ccc(C5CC5)o4)=O)(C2)C3)cccc1Cl 32494,c1(CC)nn[nH]c1C(=O)N(CCCNC(c1ccc(CN(C)C)s1)=O)CCO 32495,N1(C(C)=O)CCc2cc(NC(=O)C(N3CCC4CCC4C3)=O)ccc21 32496,c1(C(=O)NCC2CCCN(C(C(C)(C)CCl)=O)C2)ccc([N+](=O)[O-])cc1O 32497,C1(Cn2c(C(c3nccs3)NCc3cnc(CO)[nH]3)nnn2)CCCCCC1 32498,C12(CNC(c3n(CC)ncc3)=O)CC(CO1)N(C(=O)C(C)OCC(C)C)C2 32499,C1(C)(CNC(c2c(OC)nsc2OC)=O)CN(C(=O)CCC(C)C)C(C)(C)C1 32500,C(CN=c1cc[nH]c(=NCC(C)OC2CCS(=O)(=O)C2)[nH]1)OC 32501,C(=O)(C(=O)C(C)(C)CC)N(CCC(=O)NCC(C)N=[N+]=[N-])CC=C 32502,Cc1cc(C(N2CC(F)CC2C(=O)NCC2CC(=C3CC3)C2)=O)nc(O)n1 32503,C(=O)(C(C(C)(C)C)N(C)C)N1C(C2(NC(CCOCC)=O)CC2)CCC1 32504,C1(C2CCCO2)(C(=O)OCCS(=O)(=O)N(C)C)CCCO1 32505,N1(C(C(CCCC)NC(=O)Cc2cn(C)nc2C)=O)CC2(CCOCC2)C1 32506,C1(C(N)=O)CC(F)(F)CN1C(C(=O)NCc1cccs1)C1CC12CC2 32507,C(=O)(CC1=NNC(=O)C1)NC(C)(C)CCCNC(C1(n2nccn2)CC1)=O 32508,C1(C2(C)CC2)(C(=O)NC(C2C(C(N(CC#C)CC#C)=O)C2)C)CC1 32509,c1(N(C)Cc2c(C)cccc2F)cccc(S(=O)(=O)N2CCC(C(C)O)C2)n1 32510,CCC(CC(=O)NC1CCC1NC(c1ccc(C(C)C)o1)=O)C(F)F 32511,C1(CC(=O)N(C)CCNC(c2c[nH]nc2Br)=O)CCCNC(=O)C1 32512,c1(C(N2C3CC(CN(C(C(CC=CC)C)=O)C3)C2)=O)cnn2c1OCC1(CC1)C2 32513,N1(C(C2C(c3ccn(C)n3)C2)=O)CCOCC1CC(=O)NS(=O)(=O)CC1CCC1 32514,C1(CC)C(=O)NCCN1C(C1CCC(NC(C2CCCN2C)=O)CC1)=O 32515,c1(OC)ccc(C(C)C(=O)NCC(c2ccccc2OC)N)cc1OC 32516,N1(C(C(c2cc(C)c(F)cc2)=O)=O)CC2CN(C(=O)C(O)O)CC2C1 32517,Cc1ccc2c(c1)C(C(=O)NC1CCC(NC(=O)COCC3CCCC3)C1)C2 32518,c1(OC)ccc2cc(C(N3CC(N(C)C)C(SC)C3)=O)ncc2c1 32519,C1(CNC(C(C)CNC(=O)Cc2ccc[nH]2)=O)CC12CCOCC2 32520,c1(C(C(=O)NC(C2CC(C)(C)C2)C(=O)OC)F)c(F)cccc1F 32521,c1(C(=O)NCC2(CN(C(C(CC=C)CC)=O)C)CC2)ccc(Cl)c(OC)c1F 32522,CCC(C(=O)NCCCOCCCNC(=O)C(C)C1CCCC1)C(C)C 32523,Cc1ccc(C(=O)N(CCCCCC(=O)NC(c2csc(C)n2)C)C)c(O)n1 32524,N1(c2cc(C(C)C)nc(Cl)n2)CCCC(C2CC2NC(C2(C)CC2(F)Cl)=O)C1 32525,c1(N(C2CC3(CNC3)C2)C(=O)OC(C)(C)C)cc(Br)cc2ccccc12 32526,c1(C(=O)NCCC2(NC(CN3CC(C)(OC)C3)=O)CC2)ccc(F)c2c1CCC2 32527,CC1(C(N2CCCC(NC(=O)CSC3CC3)CC2)=O)CCCS1(=O)=O 32528,C1(C(=O)NCC(C)(C)NC(c2ccc(CC(C)C)s2)=O)Cc2cccnc2C1 32529,Cc1cc(C(=O)NCC2CCN(C(=O)CCOC3COC3)C23CC3)nc(C)c1 32530,C1(NC(c2c(CC)nc[nH]2)=O)CC2CCC1(N=c1[nH]nc(-c3cnccn3)o1)C2 32531,C1(NC(C2(C)CCNC2=O)=O)CCCN(C(C2CC(F)(F)CS2)=O)CC1 32532,c1(NC(Cn2cc(NC(COCC(=O)OC)=O)nn2)=O)cccc(Br)c1[N+](=O)[O-] 32533,N1(C(C2N(C(CC(CC)SC)=O)CCC=C2)=O)CCC(C)=C(F)C1 32534,C1(CNC(CS(CC)=O)=O)CC(C)(C)CN1C(c1ccc(SC(F)F)cc1)=O 32535,Cn1ncc2nc(Cl)nc(NC3CCCC34CN(C(=O)C3=CCSC3)C4)c12 32536,C1(C(=O)NC(C(=O)OC)C)CC12CC(NC(=O)Cc1cn[nH]c1)C2 32537,C1(C)(C(N2CCC(C(C(=O)NCc3c(C)nn[nH]3)C)C2)=O)CCN(C)C1 32538,c1(N2CCN(C(C(=O)N(CC#C)CC=C)C)CC2)ncnc2sc(C)nc12 32539,c1(C(C(=O)NC(C(C)C)CNC(=O)CC2CC3CC3C2)(C)C)ccccc1F 32540,c1(C(=O)NC(c2c(C)cccc2)CF)cccc2c1CNC(=O)N2 32541,C(=O)(CC(Cl)Cl)NC1(C(=O)NCC(=O)NCC#C)CSC1 32542,O=S(=O)(C=Cc1cccc(Cl)c1)Nc1cc(OC(F)F)ccc1OC 32543,c1(C(=O)NC2(CNC(C(CC#C)O)=O)CCCCC2)ccc(F)c(O)c1F 32544,CC(C)(C)CC(F)C(=O)N1CCC(CCNC(c2ccnn2C2CC2)=O)CC1 32545,c1(OC)ncc(C(=O)NC2CC2NC(C2CCC(C(N)=O)N2C)=O)cc1Cl 32546,N1(C(C2C(=C)C2C(=O)OC)=O)C(C(=O)NCCOCCC)CCC12CC2 32547,Cc1nc2ccc(C(N3CC(NC(C4CCC(=O)O4)=O)C3)=O)cc2n1C 32548,c1(N2C(c3c(C)noc3C)CCC2)nc2cc(Cl)ccc2s1.c1nnnn1C 32549,n1(CCC)ccc(C(N2CC(NC(=O)CCC3CC3(F)F)C2)=O)n1 32550,N1(C(c2sc3cc(C)sc3c2)=O)CCC(C2CCN(C(=O)CC#N)CC2)C1 32551,C1(O)(CNC(C2(C(C)C)CC2)=O)CCCN(C(c2ccc(O)cc2Cl)=O)CC1 32552,C1(CNC(=O)C(C2CCCCC2)=O)CNCCC1c1cccc(F)c1 32553,N1(Cc2c(OCC=C)cccc2)CC2CN(C(C3CC4CCC3O4)=O)CC12 32554,C1(CNC(C(C)SCCCC)=O)C2CN(C(=O)C(C)Sc3ccc(F)cc3)CC12 32555,n1(CC)cc(CNC2CCN(c3cc(O)ccn3)C2)c2cccnc12 32556,CCC(F)(F)CC(=O)N1CCC(C(C)(O)CNC(C23CC(C(C)C)(C2)C3)=O)CC1 32557,N1(C(C2C(C)(C(F)F)C2)=O)CCN(C(=O)CCC2CC2)CC12CC2 32558,c1(-c2onc(CC)n2)cccc(CNC(=O)CC2(NC(C)=O)CCCC2)c1 32559,N#Cc1cccc(CCOC(=O)C(C2CCCCC2)=O)c1 32560,Cc1cnn(C)c1C(N1CCC(C(C)(C)NC(=O)CCn2cccnc2=O)C1)=O 32561,Cc1ncnc(C)c1C(=O)NCCC1CN(C(c2cnc(C(C)(C)C)nc2)=O)C1 32562,C=C(Cl)CCC(=O)N1CC(CCNC(C2CC3CCC2C3)=O)(OC)C1 32563,C1(C)(C(=O)NCC2N(C(CCC(C)C#N)=O)CC2)CCCCNC1=O 32564,c1(CC)ccc(C(=O)OC)cc1CC.N12CC(CC(CO)C1)C2=O.C12CC1NC2 32565,c1(C(N2CCN(C(c3cn4c(n3)CCC4)=O)C3CC23)=O)ccc(F)c(Br)c1 32566,C(=O)(C1=CC(C)(C)C1)NC(c1c(OC)cccc1)CNC(C1(SC)CC1)=O 32567,C1(CNC(C=CCCC(C)C)=O)CCN(C(=O)C2=CCOCC2)CC1C 32568,c1(C(N2CCC(C(CNC(C(C)C)=O)(C)C)CC2)=O)ncnc2ccsc12 32569,C=CC(CC)CC(=O)N1CCN(C(=O)CN2CCCCC(=O)C2=O)C(CCO)C1 32570,c1(CC)nn(C)c(CC)c1C(=O)NCC=C1CCN(C(=O)C(C)S(C)(=O)=O)CC1 32571,c1(C(N2C(C(C(N3CCCC(CF)C3)=O)(C)C)CCC2)=O)ccc[n+]([O-])c1 32572,N1(C(c2c(OC)cnnc2)=O)CCN(C(=O)C(C)Cc2ccco2)C(C)C1C 32573,C1(C2=CCCCCC2)(C(N(CCCNC(c2c(C)onc2CO)=O)C)=O)CC1 32574,C1(N(C(CCN(C(=O)CC=CC(C)(C)C)C(C)C)=O)C)CCCC(O)C1 32575,c1(C(=O)NC(C2CCCN(C(c3cscn3)=O)C2)C)cc(C#N)c(O)nc1N 32576,N1(C(C2N(C(C)=O)CCC2)=O)CCC12CN(C(=O)CCCn1ccnn1)C2 32577,N1(CC(=O)NC2CCCC23CN(C(=O)Cc2ccsn2)C3)CCn2ccnc2C1 32578,N1(C(C(C(=O)OCC)OC)=O)CCC(O)(CCOC)CC1.C12CCN(CC1)C2=O 32579,c1(CC(=O)N(CC(=O)NC(C)Cc2ncn(C)n2)CC#C)cccc(C)n1 32580,Cc1c[nH]c(C(=O)NCCOCCC(=O)NCC(C)CCCO)c1C 32581,c1(OC)cc(O)ccc1NC(c1cnc(C2CC2)nc1C)=O 32582,c1(CC(N2CC(N(C(C(C=C)O)=O)C)C(C)(C)C2)=O)cnc2ccccc2c1 32583,C1(C(=O)NC2C=CCN(C(=O)C(c3ccccc3)F)C2)CC2CC(O)C(C1)C2 32584,C=CCCCCCCC(=O)NCC1CC(F)CN1C(=O)CC1CC(F)C1 32585,N1(C(C(CC)(C)COC)=O)CC2C1CCCN2C(c1cc2ccsc2n1C)=O 32586,Brc1ccc2c(c1)CC2NCc1cc(-c2ccccc2)ccn1 32587,C1(C(=O)NC(C)CCCNC(c2cc[nH]c2)=O)CC(S(C)(=O)=O)C1 32588,C12(CC(=O)NCC3(COC)CCCC3)CCC1CN(C(=O)C1=CCCCC1)C2 32589,c1(OC)ccc(C(O)C(N2CCC(F)(NC(=O)CCN3CCOCC3)C2)=O)cc1 32590,c1(C(=O)NC(CC)CN(C(=O)Cc2ccoc2C)C)occ(C)c1C(=O)OC 32591,C(=O)(CC(C)N(C(=O)C(c1ccncc1)C)C)N(CCC(C)C)CC(C)C 32592,N1(C(CC2CCN(C)CC2)=O)CC2(NC(C3COC(=O)N3C)=O)CCCC2(F)C1 32593,c1(OC)cc(OC)c(C(N2CC(NC(=O)C(C)CF)C(O)C2)=O)c(N)c1 32594,Cc1cc(Br)c2ncnc(N3CCCC(c4ccno4)C3)c2c1 32595,Cn1cc(Cl)cc1C(C1CC1)N.C1(CN2CC(c3nnnn3C)C2)CC(C)(C)CO1 32596,c1(C(=O)OCC)cc(CNCCc2cccc(SC)c2)c(C)s1 32597,N1(C(c2ccc(CSC)o2)=O)CC2CCC(C1)N2C(=O)CCC1CCCO1 32598,n1(CC)nc(C(N2CCC(C(C)NC(C3CCCC3C(C)C)=O)C2)=O)c(C)n1 32599,C1(CC(=O)NCC(CC2CC2)CO)CC=CCC1.C12CN(C1)C(=O)CO2 32600,CC1CC(NC(c2ccc(Br)c(O)n2)=O)CN(C(C2CCC(=O)C2)=O)C1 32601,N1(C(C(C=C)(C)C)=O)CCC(NC(c2ccc(OC)cc2OC)=O)C(C(C)C)C1 32602,C(=O)(C(F)(F)CCn1ccnn1)NC(CC(C)NC(=O)CC1CC(O)C1(C)C)C 32603,C1(NC(C(C)=C2CCCC2)=O)CCN(C(=O)C=Cc2ccncc2)C1C 32604,C1(CNC(c2c(C)cnnc2)=O)CN(C(=O)CC(C)c2ccco2)CC1(C)C 32605,Cc1cccc(-c2cc(C(=O)N(C(C)CN(C)C(C3CC3C(F)F)=O)C)on2)c1 32606,C12(C(=O)NCCc3nn[nH]n3)CC(CN(C(C3CC4(CCC4)CO3)=O)C1)C2 32607,n1(CC)nc(C)c(C(N2CC(NC(C3(O)CCSC3)=O)C(CC3CC3)C2)=O)c1Cl 32608,C1(N2CCOCC2)(C(N(CCN(CC)CC)CC)=O)CCCC1 32609,C(C)(CO)(C(=O)N(CCC(O)CO)C1CC1)NC(C(c1ccnn1C)C)=O 32610,C1(CNC(C(c2cccc(F)c2)C)=O)CC2CCC1N2C(=O)C=Cc1ccoc1 32611,c1(CCC(N2CC(C)(NC(C3C4CC4C4CC34)=O)C2)=O)cnc2ncccn12 32612,N1(C(c2c(CC)onc2)=O)CCN(C(=O)CS(=O)(=O)N(C)C)CC(CO)C1 32613,Cc1ncnc(O)c1CC(N1CCC1CNC(C1(O)CC(F)(F)C1)=O)=O 32614,C1(C(=O)NC(C)CCNC(C2(C#N)CC2)=O)OCC2COCCC12 32615,C(CCC(N)=O)(C(=O)N1CC(C)(c2cn(CC3CCCOC3)nn2)C1)N(C)C 32616,Cc1c(C(N2CC(O)(CCNC(C3CCN(C(C)=O)C3)=O)C2)=O)c(Cl)nn1C 32617,N1(C(CCC(NN(C)C)=O)=O)CCC2(C=C(C(=O)N3CC(F)(C#N)C3)C2)C1 32618,C1(CNC(C(C)OCC(C)C)=O)CC(C(=O)NCC2CCCC2N(C)C)CO1 32619,n1(C(C)C)ccc(CC(N2CC(NC(c3ccsc3Br)=O)C2)=O)n1 32620,Cn1cc(CCC(=O)NCC2CCCN2C(c2ncsc2C(F)(F)F)=O)nn1 32621,CCC(C)N(OC)C(=O)CC1CC(NC(C2CCC(=O)N(C)C2)=O)C1 32622,CC(C)C(CCCC(=O)O)NC(=O)CC1COCC1(C)C 32623,N1(C(Cc2cc(OC)ncc2)=O)CC(C2CC2(F)F)C1 32624,c1(C(=O)NCC(=O)NCC(O)CC2CCCO2)cncc([N+](=O)[O-])c1 32625,c1(C(N(CCNC(c2c(CC)onc2)=O)CC)=O)cc2cccn2cn1 32626,N1(C(C(CC)NC(C)=O)=O)CC(CNC(c2cncc(C(C)(F)F)c2)=O)C(C)C1 32627,c1(CC(=O)NCC2CN(C(c3c(Cl)ccc(N)c3)=O)C2)noc2ccc(F)cc12 32628,C(CC(C)C)(C(=O)NCC1CCCC1NC(c1ccncc1OC(C)C)=O)OC 32629,C(=O)(CCC(C(C)C)NC(c1cc(C(C)C)[nH]n1)=O)NC(C(=O)NCC(C)C)C 32630,C(=O)(C#CC1CCCOC1)NC1CC2CN(C(c3n(CCC)ccc3)=O)CC21 32631,c1(-c2ccc(C)o2)nnc(NSc2nc3ccccc3nc2Cl)c2ccccc12 32632,c1(C(=O)NC2C(C(=O)O)CN(C(CNS(C)(=O)=O)=O)C2)cc(C(F)F)ccc1F 32633,C(C(C(=O)NCc1cnn(CCF)c1)C(C)C)NC(c1ncc(C)nc1)=O 32634,c1(C(=O)NCc2c(CC)cns2)cc(-c2cccnc2)ncn1 32635,C1(C(=O)NCC(CC)NC(C2CC(=O)N(C)C2)=O)CC(C)(C)C1C(F)(F)F 32636,N1(CC2C(C#C)CCCC2)CCOC2(CCCN(C(=O)C(F)C(F)(F)F)C2)C1 32637,CC(O)C(C)(C)C(=O)N1CCC(=CCNC(=O)Cc2c(F)cccc2F)CC1 32638,C1(CS(Oc2cnncc2C(N2CC3C(C(N)=O)C3C2)=O)(=O)=O)CC2(CCC2=O)C1 32639,N1(C(CCCOC(C)(C)C)=O)CC(C2CN(C(=O)CN3CCCCCC3=O)C2)C1 32640,N12CC3(CC(C3)C1=O)C2.c1(N(C)C)cnc(C(C)(C)F)nc1 32641,N1(C(C(C(C)C)NC=O)=O)CC2(CC(NC(=O)CSc3cnn(C)c3)C2)C1 32642,c1(C(=O)NCC(CNC(C(C)CN2CCCCC2)=O)CO)cccc(N)c1F 32643,N1(C(CC(C)OC)=O)CCN(C(=O)CC2CC2)CC1c1cc(F)ccc1F 32644,C=CCC(C(=O)NC(CN(C)C)CCO)NC(c1ccon1)=O 32645,c1(C(=O)OC)c(NC(C2CCCN(Cc3nccn3C)CC2)=O)sc(C)c1C 32646,CC(C)CC(C)CC(=O)N1CC(C)N(C(=O)CC2CC(C)(C)CO2)CC1C 32647,Cc1ncc(Cl)c(C(N2CCC(O)(CNC(C3CC4COCC4C3)=O)C2)=O)n1 32648,Cc1cc(C(=O)NC23CC2CN(C(C2(C)CCOC2)=O)C3)c2n[nH]cc2c1 32649,c1(C(N2CCC(C)(NC(c3cc(C(C)C)on3)=O)C2)=O)cc2n(n1)CCCC2O 32650,c1(C(=O)NCC2CCN(Cc3c[nH]c4cccnc34)C2)ccc2c[nH]nc2c1 32651,c1(CC2(NC(CONC(CN(C)C)=O)=O)CC2(C)C)cccc2[nH]ccc12 32652,c1(C(=O)NCC2(C)C(C)CN(C(=O)C(F)F)C2)ncccc1S(C)(=O)=O 32653,CC1CCC(C)(C)N1C(C1CCN(c2ccncn2)CC1)=O 32654,c1(C(CNC(c2c(CC)c[nH]n2)=O)NC(=O)CCC(C)C)ccc(N(C)C)cc1 32655,CC1CCN(C(C2CC(O)(C#N)C2)=O)C(C)C1NC(C1CN(C(N)=O)C1)=O 32656,c1(C(=O)NCC23CN(C(CC(=O)OCC)=O)C(CC2)C3)nc2cc(F)ccc2s1 32657,C1(C(C(C)NC(=O)N(C)Cc2ccco2)(C)C)Cc2ccccc2O1 32658,CC(C)(O)C(F)C(=O)NCC1CN(C(C2CC(=O)N2)=O)C1 32659,c1(C(N2CCN(c3nc(C)cc(SC)n3)CC2C)=O)ccnc2c1OCO2 32660,c1(CC)ccccc1-c1cn(CC2CCCC2NC(c2cnn(C)c2)=O)nn1 32661,c1(C(=O)NC(CNC(c2ccc(C)nn2)=O)C2CCC2)c(C)nn(C(C)C)c1C 32662,c1(C(N2CCC(N(C(=O)C(N)=O)CC)C2)=O)cc(C)c(C)c(S(N)(=O)=O)c1 32663,CC1CCC(NC(c2cccnc2O)=O)CN1C(=O)CC1(NC(C)=O)CC1 32664,CC(CN=c1[nH]c(=NCC2CC23CCC(F)(F)CC3)[nH]c2c1CCCC2)C1CC1 32665,C1(OC)CCC(CC(N2CC3CC3(NC(=O)CC3CC(C)C3)C2)=O)CC1 32666,C1(CNC(N2CCCC(CCOC)CC2)=O)CCC2(CCC2)CN1C 32667,C1(Cc2cn(C(C(=O)NCC=C=C)C)nn2)CCC(CC)CC1 32668,N1(C(c2nc(C(C)OC)sc2)=O)CCCC1(C)CNC(c1ccnn1C)=O 32669,CC1(C)CC(C(N2CCN(C(c3coc(C#N)c3)=O)C(CO)C2)=O)C(C)(C)O1 32670,C12CCCC(C1)NC2=O.C1(SC)CN(C(=O)C(C)S)C1 32671,C1(C2CN(C(CCOCCOC)=O)C2)CCN(C(c2cccnn2)=O)CC1 32672,c1(C(=O)NC2CCCC(NC(c3c(N)c(F)ccc3)=O)C2)cccc2sccc12 32673,c1(C(N(CCN(C(C2(O)CC3CCC2C3)=O)CC)CC)=O)ccc2cn(C)nc2c1 32674,CCCCC(O)CC(=O)NC(C(N1CCCC(C)C1)=O)C1CC1 32675,N1(C(C2CCC(=O)N2)=O)CCCN(C(C23CCC2C3)=O)CC1 32676,C1(NC(CC(COC)C)=O)CC2CC1CN(C(=O)Cc1c(C)noc1C)C2 32677,C(c1ccc(C(F)F)o1)=CC(=O)NCC(CCNC(Cc1cn(C)nc1)=O)O 32678,N1(C(c2nc(CNC(CC(CCC)C)=O)oc2C)=O)CCc2ncsc2C1 32679,C#CCCCC(=O)N1CCCC(NCCC(=O)C(c2ccccc2)OCC)C1 32680,N1(C(C2N(C(C(C)NC(N)=O)=O)CC3CC32)=O)CCCC(CO)CC1 32681,CC(CCCc1ccccc1)C(=O)N1CCC(N(C(=O)C2=C(Cl)CC2)C)CC1 32682,c1(OC)cc(C(N2C3CCC2C(NC(=O)C=Cc2cc[nH]n2)C3)=O)c(Cl)cc1Cl 32683,Cc1ccc(F)cc1C(N1CCOCC1CCNC(C1(F)CCCN(C)C1)=O)=O 32684,C(=O)(C1=NOC(NC(=O)CC(C)n2ccnc2)C1)NCCCNC(COC)=O 32685,Cc1cc(CC(=O)NC2COCC2NC(=O)CC(C)F)ccc1CO 32686,C1(C2=CCOCC2)(CNC(C(C(F)(F)F)c2cccnc2)=O)CC1 32687,C(=O)(C(CCC1CCC1)NC(c1cnnn1C(C)C)=O)NCc1ncc(C)[nH]1 32688,c1(C(=O)N(C2(O)CNC2)C(C2CC2)C2CC2)c[nH]nc1-c1ccccc1 32689,Cc1cc(-c2nn[nH]n2)c(C)cc1C(=O)NCc1ccon1 32690,c1(CC)nc(C)c(C(=O)NC2CCCC(NC(=O)CCC#N)C2)c(C)n1 32691,C1(CNC(=O)NC(C#CC)(C)C2CCC2)(CNC(=O)OC(C)(C)C)CCC(=O)N1 32692,c1(CC)nc(C)c(CC(=O)N(C(C)CNC(C2CS(=O)(=O)CCO2)=O)C)c(C)n1 32693,c1(OC)ccc(CC(=O)NCCC2CCCC2(C)C)c(O)c1 32694,N1(C(C2N(CCCC)CCCC2)=O)CC(NC(c2cc(C)[nH]c2C)=O)C(C)(C)C1 32695,C(=O)(C1=CCCN(C(=O)CC=C(Cl)Cl)C1)N1CC(C)(OC)C1 32696,C1(C)(C(N(C(N(CC(C)O)C(C)C)=O)C(C)C)=O)CCN(S(C)(=O)=O)CC1 32697,c1(C(=O)NC(CC)CNC(=O)C=CS(C)=O)cnc2cnc(Cl)cc2c1 32698,N1(C(c2c(C)coc2)=O)CCC2(CCN(C(=O)CC3COCCOC3)C2)C1 32699,c1(C(=O)NCCC(C)N(c2nccnc2F)C)cncc2nc[nH]c12 32700,C=C(Cl)C(C)(C)C(=O)NCC(C1CCCN(C(c2ncncc2F)=O)C1)(C)O 32701,C(CC(O)CO)N(C(=O)CC1(NC(C2(C)CCCO2)=O)CCC1)C 32702,c1(CC)conc1CC(=O)NCC(C)NC(c1sncc1C)=O 32703,C1(NC(c2cc(F)c(Cl)cc2F)=O)CCCCCN(C(c2cc(CO)[nH]n2)=O)C1 32704,C=CCC(CC(F)F)C(=O)NCC(C)(C)CN(C)C(c1cc(SC)ccc1C)=O 32705,c1(C(N2C(CNC(C3CC(OC)C3)=O)CN(C)CC2)=O)cc(F)c(C#N)c(F)c1 32706,CC1CN(C(=O)CCCF)CCC1CNC(c1cc(Cl)ccc1Cl)=O 32707,c1(CC(=O)N(CCCNC(C2CC(CN3CCCC3)C2)=O)CCO)cnc[nH]1 32708,C(CCCCCC(=O)N(C)CC1CCCC1O)NC(c1n(CC)nc(C)c1)=O 32709,c1(C(=O)NC(C2CCCN(C(=O)CCNC(=O)CO)C2)C)ncnc(O)c1F 32710,CC(CO)(C1CCC1)NC(=O)NC1CCC1OC(C)(C)C 32711,C1(CCNC(C=COCC)=O)CCN(C(c2cn(C)c(=O)cn2)=O)C(C)C1 32712,N1(C(c2nc(CC)sc2N)=O)CC(CNC(=O)CCN2CCCCC2)C2(CC2)C1 32713,C(c1ccc2[nH]ccc2c1)=CC(=O)NC(C)CCNC(c1csnn1)=O 32714,C1(CCC(=O)N(CC(C)N(C(CCCC)=O)C)C)CCCC(O)C1 32715,N1(C(=O)C2=CCCSC2)CCN(C(=O)Cn2ncnn2)C2CCCCC2C1 32716,C=C(Br)CCC(=O)N1CCN(C2CC2NC(c2snnc2C)=O)CC1 32717,c1(C(=O)NC(CCNC(C(CCC)NC(C)=O)=O)C)cc(Cl)cc(C(F)(F)F)n1 32718,N1(C(CCC)=O)CC2CCC(C1)C(NC(=O)C1=CC(C)(C)C1)C2 32719,C1(N(CCNS(CC)(=O)=O)C(c2ccn(C)n2)=O)CC2CCC(C1)N2 32720,C1(NC(C2(OC)CCCCC2)=O)CCN(C(c2cc(Cl)c[nH]2)=O)CC1C 32721,n1(CC)ccnc1C=CC(=O)NCCC1CN(C(C2CC(CC(=O)OC)C2)=O)C1 32722,S(=O)(=O)(c1cc(C)c(-c2ccccc2C#N)cc1C)NCCC(CC)OC 32723,CC1=C(CNC(=O)CC2C=CC(NC(=O)C(c3ccccc3)O)C2)COCC1 32724,c1(C(N2CC3C(NC(C=CCOC)=O)CC(C3)C2)=O)ccc2cc(Cl)ccc2n1 32725,c1(C(=O)NC2CCCC(N(C(=O)C3=CCCOC3)C)C2)cccc2nccn12 32726,Cc1nnc(CCC(=O)NC2CC(CNC(=O)C(c3ccc(Cl)cc3)=O)C2)n1C 32727,C(=O)(CCC(C)(C)NC(c1cccc(F)c1N)=O)N(CC(C)(O)C1CC1)C 32728,N1(C(c2cn(CCC)nc2C)=O)CCC(C)(NC(c2n[nH]c(C)c2C)=O)CC1 32729,C(CCO)(C(C)(C)O)NC(c1cc(CNC(C2(CSC)CC2)=O)on1)=O 32730,CCC(O)C(F)(F)C(=O)N1CC(F)(CNC(=O)C(C)(C(=O)OC(C)(C)C)OC)C1 32731,c1(NC(=O)NC(C)CCCCN)ncc2c(n1)CCC(C(F)(F)F)C2 32732,N1(C(CC(CC)C2CC2)=O)CCC2C(NC(c3c(C)nn(CC)c3Cl)=O)CC12 32733,Cc1cc(Cl)ccc1C(N1CC(CNC(c2cnc3n2CCC3)=O)C2(CC2)C1)=O 32734,c1(C(=O)NCC23N(C(C(C)=C4CCC4)=O)CC(C2)C3)ccc(C)cc1N=[N+]=[N-] 32735,c1(C(=O)NCCCNC(c2c(C)ccc(OC)n2)=O)nccc2c1NCCC2 32736,c1(CNC(C2CC=CC(n3cc(C4(O)CC4)nn3)C2)=O)ncc([N+](=O)[O-])cn1 32737,CC(C)(C)CC(=O)NC(C12CCC(CC1)C2)CNC(C1(Cl)CC1)=O.C1C(=O)N1 32738,c1(N(c2c(OC)c(F)ccc2)C(C2CC3CCCCN3C2)=O)ccnc2ccnn12 32739,c1(COC)nc(NC(C)C(OC)OC)cc(N2CCC(CCCO)CC2)n1 32740,N1(CC(N2CC3C(C(N(CCN(C)CCO)C)=O)(C3)C2)=O)C(=O)CCCC1=O 32741,c1(CCC(=O)N(CC(C)NC(=O)CCC(F)F)C)ccccc1NC(N)=O 32742,C1(C(N2CCC(O)(CN(C(c3c(C)cc(CC)o3)=O)C)C2)=O)CCCCCN1C 32743,CC1OCCCC1C(=O)N(C)CCN1CCN(C(=O)CC2OCCO2)CC1 32744,Cc1cc(=NC2CN(CC3CC3)C2)[nH]c(N2CCc3n[nH]cc3C2)n1 32745,CCC(CC)CC(=O)NC(C(=O)NC1CCOCC1O)C1CC1 32746,C(C(C)C)(C(O)C(=O)NCC=CC(=O)NCC1CCC(C)(C)O1)OC 32747,C1(C(N(CC(O)COC)CC)=O)CCC(C)(C)N(C(=O)CN2CC(=O)NC2=O)C1 32748,N1(C(c2c(CC)noc2)=O)CCC2(CCCCN(C(C3CCOC(C)C3)=O)C2)C1 32749,Cc1cc(N)cnc1C(=O)NCC(C)NC(c1cnsc1C)=O 32750,CC1CC(NC(c2cnc(-c3cccnc3)s2)=O)CN(C(C2CC(F)(F)C2)=O)C1 32751,C(C)(C)(CCC(=O)NCCCCOC(C)C)NC(C(COCC)C)=O 32752,C1(CNC(C(C)OCC=C)=O)CCN(C(C2CC2c2cccc(Cl)c2)=O)CC1 32753,C1(NC(c2cnn(C(C)(C)C)n2)=O)CCC(C)(CNC(=O)C=Cc2ncc[nH]2)C1 32754,C12(NC(CCc3n(C)ccn3)=O)CCCCC1CN(C(=O)CCNC(=O)CO)C2 32755,N1(C(C(CC=C)C)=O)CCC2CN(C(c3ccccn3)=O)C(C)C12 32756,C(CCC(C(=O)N1CCC1C(N)=O)NC(=O)CN1CCCC1=O)OC 32757,C1(C(N2CC(N(C)C(c3cnn(C)c3)=O)C(C)(C)C2)=O)(OC)CCCCCCC1 32758,C1(C(=O)NC(C(C)C)CNC(=O)CC2CCN(C)C2=O)CC(=O)OC1(C)C 32759,C1(CN=C(NC(C)C)NC2CCN(CC(F)(F)F)C2)CSc2ccccc2O1 32760,CC1(C)OCC2CC12C(N1CCC(C)(CNC(c2ncc[nH]2)=O)C1)=O 32761,n1(SCCOCCCC)cc(C(C)(C)O)nn1 32762,N1(C(c2c(C#C)cnn2C)=O)CCC2(CCC2)C(NC(c2ccccc2F)=O)C1 32763,C1(C(=O)O)C(CN(C)C(C23CCC(CC2)C3(C)C)=O)C2CCC1(C)C2(C)C 32764,CCCC(CNC(=O)CCC1CCCCC1)NC(c1sncc1C)=O 32765,C1(NC(c2ccc(C)cc2C)=O)CN(C(=O)Cc2csc(C)n2)C2(CCCC2)C1 32766,C1(NC(C2CC(=C)C2)=O)CC2CCC1C(NC(c1ccoc1C(C)C)=O)C2 32767,c1(C(=O)NCC(c2cccs2)N(C)C)ccc2c(c1)CCCN2 32768,c1(C(=O)NCCCN(C(=O)CN2CCOCC2)CCO)ccc(O)cn1 32769,CCCC(C(C)CC)(c1nnnn1-c1ccc(F)cc1)NCc1ncsn1 32770,C1(C)(C(N2CCC(NC(C(c3ccnn3C)C)=O)C2)=O)CCCS1(=O)=O 32771,c1(CC)oc(C)cc1C(=O)N(C(C)CC(=O)NCCC(F)F)C 32772,c1(NC(C2C(OC)CN(S(=O)(=O)C(C)C)CC2)=O)cc2nc(F)ccc2o1 32773,Cc1sc(=O)n(CC(N2CCC(NC(C3CC3(C)C)=O)C2(C)C)=O)c1C 32774,N1(C(=O)C#CC2CC2)CCC2CCN(C(c3cn(-c4ccccc4)cn3)=O)C2C1 32775,c1(C(=O)NCC(CNC(C(C)OC2CCOC2)=O)O)cccc(CO)c1 32776,C(=O)(C1CCCc2nnn(C)c21)N1CCCN(C(C(C2CCC2)OCC)=O)CC1 32777,N1(C(=O)NC(C(=O)OCC)C)CC2(CNCCCCl)CCCCC2(C#N)C1 32778,CC1(C)CCOC1C(=O)NC1CCCN(C(=O)CNC(=O)N(C)C)C1 32779,c1(C(=O)NC(C)CNC(=O)CCCc2cncs2)cc2c(O)ncnc2cn1 32780,Cc1cc(NC(C2C=CC(NC(C3CC3F)=O)C2)=O)cc(-c2nn[nH]n2)c1 32781,C(=O)(C1Cc2ccc(C)cc21)N1CCN(C(CNC(CCC)=O)=O)CC(O)C1 32782,N1(C(c2c(C)nc(C(F)(F)F)o2)=O)CC2(CCN(C(=O)C3=CSCS3)CC2)C1 32783,N1(C(c2c(CC)onc2)=O)C2CCC1CC(CNC(c1cnn(C)c1OC)=O)C2 32784,C(=O)(C(C(C)(C)C)OC)NCCC(=O)NC1(c2c(OC)cccc2)CCOCC1 32785,C(=O)(C(F)CC(C)C)NCCN(C(=O)CCC1CCCN(C)C1)CCC 32786,C=CC(CC)CC(=O)N1CCC(C)C(NC(=O)C=Cc2cnc(OC)cn2)C1 32787,C1(NC(CCn2ccc(C)n2)=O)C2CC3CN(C(C4OCCCO4)=O)C1C3C2 32788,C1(C(N2CCC(CN(C(=O)C3=CCCCCC3)C)C2)=O)CC12CCC(=O)CC2 32789,C1(NC(C2CC(=C3CC3)C2)=O)CC(C(=O)NCC2(CO)CCCC2)C12CCC2 32790,C(=O)(CC(O)CCSC)NC1CN(C(c2c(-c3cn(CC)nc3)n[nH]c2)=O)C1 32791,C12(NC(c3nc(C(C)C)oc3)=O)CCCN(C(=O)C3=CCC3)CC1C2 32792,c1(CNC(C2ON=C(C)C2)=O)cccc(CNC(c2cnc(C3CC3)[nH]2)=O)c1 32793,c1(C(=O)NCC(CC=C)NC(c2ccccc2CO)=O)c(C(C)C)cccc1F 32794,c1(CS(C)=O)cccc(C(=O)NC2CC(NC(=O)C=CC(F)F)CC2O)c1 32795,CC1(NC(c2csc(-c3ccsc3)n2)=O)CN(C(C2CCC2)=O)C1 32796,N1(C(Cc2nc(C)sc2)=O)CCC(N(CCCCCc2ccncc2)C)CC1 32797,c1(C(N2CCC(N(C(=O)CC3COCCO3)C)C2)=O)cc([N+](=O)[O-])cs1 32798,c1(OCC(=O)N(C2CCN(C(C(C)=CC3CC3)=O)C2)CCO)c(C)cccc1Cl 32799,C1(C)(C(=O)NCCCN(C(C2CCc3ncnn3C2)=O)CC)CC(C2CC2)=NO1 32800,N1(C(C(C)(C)OCC)=O)CCN(C(c2c[nH]cc2CC)=O)CC(O)C1 32801,O=S(=O)(c1cccnc1NCC1CC2(C1)OCCO2)N1CCCC1CF 32802,c1(C(N2CC(C)N(C(c3ccc(N(C)C)nc3)=O)CC2)=O)ccn2ccnc2n1 32803,Cc1onc(-c2cccc(Cl)c2)c1C(=O)NC1CC(C)(NC(c2coc(Cl)n2)=O)C1 32804,c1(NC(C2N(C(c3ccn(C)c3)=O)CC=C2)=O)cnc2[nH]cnc2c1 32805,c1(CNC(=O)NC(c2cccs2)Cc2cn(C)nn2)cc(Cl)ccn1 32806,c1(-c2cn(CC3N(C(CC(CC)C(F)F)=O)CC3)nn2)ccc2nccnc2c1 32807,C(=O)(CCS(=O)(=O)c1ccc(OC)cc1)N(CCNC(C(CCCC)(C)F)=O)C 32808,c1(C(=O)NC(C(C)NC(c2cccc3ccsc23)=O)C)ccc2c(c1)CCOC2 32809,c1(C(N(C(CC(=O)N)C)C)=O)cc(F)c(O)c(Cl)c1.Cc1cc(CC=O)on1 32810,N1(C(Cc2cc(C)no2)=O)CCCC(C2CC2NC(c2cc(C(N)=O)cs2)=O)C1 32811,c1(C(=O)NC2CCC(NC(C3CC34CCCCC4)=O)C2)cccc2c1CCC2 32812,N1(C(CC23C(C)(C)C(CC2)CC3)=O)CCCC(C2(NC(=O)C(O)C3CC3)CC2)C1 32813,c1(CNC2(c3n(CCOC)nnn3)CCN(C3CC3)C2)n[nH]c2c1CCCC2 32814,c1(C(N(CCCCN(C(C(COC)OC)=O)C)C)=O)ccc2c(c1)C(C)C(C)O2 32815,C1(C(N2C(C(=O)NCc3cccnc3O)CCC2C2CC2)=O)CC2(C1)CC(O)C2 32816,C1(C(N2CCC(N(C(=O)CN3CSCC3=O)C)CC2)=O)C(C2CC2)C1(F)F 32817,c1(-c2n(CC)c(N3CC(C)(C)OCC3C3CC3)nn2)ccc2c(c1)ncn2C 32818,CCC(C(=O)OC)NC(c1csc(CNC(c2cccn2C2CC2)=O)c1)=O 32819,CC(C)C(C)C(CNC(C1CCSCC1)=O)NC(c1cc(=O)n(C)o1)=O 32820,N1(C(CC(C)(C)OC)=O)C(CC(=O)NCC2CCC3(CC3)C2)C2CCCC12 32821,C(=O)(C1=CC2(CCOC2)C1)NCC1(NC(c2c(C)ncnc2)=O)CCCCCC1 32822,Fc1ccc(Cl)c2[nH]cc(CNc3ncc(Cn4cc(Br)cn4)s3)c12 32823,N1(c2c(C)c(NCc3c[nH]ccc3=N)ncn2)CCOc2cc(Cl)ccc2C1 32824,c1(C(=O)NCCC(C)N(C)C(c2cnsc2)=O)cccc(N)c1 32825,C1(C(N2CC(O)(CCNC(c3scc(C)c3Cl)=O)C2)=O)CCn2nnnc2C1 32826,C1(NC(C2CC(=C)C2)=O)C2CC1N(C(C1CCN(CC(F)F)CC1)=O)C2 32827,CC(=O)C(C)(C)CC(=O)NC(C1CN(C(C2CS(=O)(=O)C2)=O)C1)C 32828,C1(CNC(c2n(CCOC)ncc2)=O)CC2CC2N1C(C1CCCOCC1)=O 32829,C1(CC=C)(NC(=O)CC(C)CF)CCN(C(=O)C=Cc2ccccc2)CC1 32830,c1(SCCC(=O)N2CCCC2CC2=CCSC2)nnnn1C1CCCCC1 32831,C1(NC(c2c(C)sc(Br)n2)=O)CC2CC(C1)N(C(=O)C=C1CCCC1)C2 32832,C1(C(=O)NC(C(=O)NC(CC=C)C2CC2)(C)C)CC2(C1)CC(O)C2 32833,C(=O)(C(C(C)C1CCOC1)N1CCC2CC2C1)NCCC(=O)NCCOC 32834,C(C(=O)CC(C)CC(C)C)O.c1(CCC)ccccc1 32835,N1(C(c2csc(Br)n2)C(=O)NCC2CC2)CC2CC1CN2Cc1cccs1 32836,c1(CC(C)C(=O)N2CCC(C(C)(C)NC(C3CCOC3)=O)C2)ccc(Cl)cc1Cl 32837,CC1(NC(C2(C)CCN(C(=O)OC(C)(C)C)C2)=O)CCCC1(F)F 32838,C#CCC(CC(=O)NCCOC1(C)CCC1)NC(C1CC12CCCC2)=O 32839,CC(F)(F)C(F)C(=O)NCc1ccc(C(=O)NOCCCCCC2CC2)s1 32840,Cc1ccc(CNC(C23CC(SC(C)(C)C)(C2)C3)=O)c(N2CCC(O)C2)c1 32841,C1(C(=O)OC)C2CC(CN(C(=O)C(=O)NC(C3(CSC)CCOCC3)=O)C2)C1N 32842,C1(CNC(C=CC(=O)OCC)=O)CC(C(=O)N2CCC(CO)(OC)C2)=NO1 32843,C=CCC(CNC(C1CC1C#N)=O)C(=O)N(CCOCC)CC 32844,CCCCC(C)CCC(=O)NCCC(C)NC(c1cc(C)nc2ccnn12)=O 32845,C1(CN(C)C(C23CCC(C2)C3)=O)CN(C(C2CC(F)(CF)C2)=O)CCO1 32846,C(=O)(C(C)CCCc1ccccc1)NC1CN(C(CCC(=O)OCC)=O)C(C)C1 32847,c1(CC)ccc(C2CCN(C(C(=O)NCCCSC)c3cn[nH]c3)C2)cc1 32848,N1(C(c2ccc(N)cc2O)=O)CCC2(CCC2)C(CNC(=O)Cc2cscn2)C1 32849,N1(C(c2n(CC)nnc2)=O)CCN(C(=O)CCc2ccc(Cl)s2)CC1C 32850,c1(C(N2CCCC(c3onc(C)n3)C2)C(=O)NC(C)C)sc(C#N)cc1C 32851,C1(C)(COC)CC(NC(c2c(C)cccc2F)=O)CN1C(c1ccoc1Cl)=O 32852,N1(C(CC(CNC(c2ccc(CC)cn2)=O)C2CCC2)=O)C(C)CCC1(C)C 32853,C1(OC)CC2(C1)CN(C(c1csc(CNC(C3(CF)CC3)=O)c1)=O)C2 32854,c1(C(=O)NC(CCNC(c2ccn(CC)n2)=O)C)ccc(C2CNC(=O)C2)cc1 32855,CCC(C)C(C(=O)N1CCC(O)CC1C(N1CC(CC)(CO)C1)=O)OC 32856,C(CC1=CCN(C(c2cc(N)nc(Br)c2)=O)CC1)NC(C1C(=C)C1)=O 32857,C(CC(O)CC(=O)N1CC2C(NC(=O)C=CC3CCCC3)C2C1)SC 32858,N1(C(=O)CCc2ccccc2)CCCC(C2CCCN(C(C3CC(O)CN3)=O)C2)C1 32859,N1(C(COCC)=O)CCCC(C)(CNC(=O)C2=CCCC2C)C1 32860,C=C(C)CCC(=O)N(CCCNC(C1CCN1CC)=O)Cc1cccnc1 32861,c1(CNC(NC2C(OCC)CCCC2)=NCC2CC2)ncc(Br)cc1Br 32862,c1(C2(C(COC(=O)CC3CCCOC3)=O)CC2)ccc(Cl)c(F)c1 32863,C1(C(N2CC(N(C)CC)C2)=O)CC1C1CN(C(C2CCSCC2)=O)C1 32864,CC1=CN2C(C(=O)NCCCCN(C)C(C3CC4CC4C3)=O)(C=C1)CC2 32865,N1(C(CN(C)CC)=O)CC2CC(NC(c3coc4c3CCCC4)=O)CC1C2 32866,Cc1ccc(-c2nc(CC(=O)NC3CC(C)(NC(=O)C(C)C(C)C)C3)cs2)cc1 32867,c1(C(N2CCC(NC(CCS(=O)(=O)NC)=O)C(F)C2)=O)cnc2c(c1)CCCO2 32868,C1(NC(c2coc(C(F)F)c2)=O)CCN(C(c2nocc2C(=O)NC)C)CC1C 32869,c1(CCC)ccc(C(=O)NCC(C)N(C(=O)CSCCC#N)C)cc1.N1(C)CCCC1 32870,C(=O)(C(O)C(F)(F)F)NCC1CC(C)N1C(=O)CC(C)(C)C 32871,CCC(Cc1ccccc1)C(=O)N1CC(C)(NC(=O)CCC(=O)NC)C1 32872,N1(C(C2(CS(C)(=O)=O)CCC2)=O)CCCC2CC(NC(c3cc4sccc4s3)=O)C12 32873,Cc1nc(O)ccc1C(N1CCC(C)C1C(=O)Nc1cnn(CCF)c1)=O 32874,C1(NC(C=CCC)=O)CCN(C(c2c(OC)noc2C)=O)CC12CCC2 32875,c1(OC)ccc(C(N2CCCC2C(C)(C)NC(=O)CC2CN(C)CC2O)=O)nn1 32876,CCCC(F)C(=O)NCCOCCCN(C)C(C1CCC1C#N)=O 32877,C(C(=O)NCC1CCN(C(C2CCOCC2(C)C)=O)C1)(c1ccccc1)=C(C)C 32878,CC(C)CC(CC(C)C)C(=O)NCCC(C)N(C(=O)CCc1ncc(F)cn1)C 32879,CN1CC(CC(=O)NCc2nncs2)CCC1C(F)(F)F 32880,c1(SC(=O)CN2C3CC(c4c(COC)ncs4)CC2CC3)nc2ccc(C)cc2[nH]1 32881,C1(CNC(C(C)(C)SC)=O)CN(C)CCN1C(c1cc(Cl)sc1Cl)=O 32882,Fc1coc2c(CNc3ccc4nc(C(F)F)oc4c3)ncnc12 32883,CC(F)(F)C(C)(C)CC(=O)N1CC(NC(C2CCS(=O)(=O)C2)=O)CC12CCC2 32884,C(=O)(C1Cc2ccccc21)NCC(CCCC)NC(=O)C(F)OC(F)(F)F 32885,c1(C(N(CCC(=O)NCCN(C)C)CCC)=O)cn(C2CC2)nc1C 32886,N1(C(c2nccc(N)c2)=O)CC2(CCC(CNC(=O)Cc3cnns3)O2)C1 32887,C1(C(=O)NCC2(NC(c3cnc(-c4ccco4)s3)=O)CC2)CCC2(CC2)C1 32888,C1(O)(CN(C(C2CCN(C)C2)=O)C)CCN(C(=O)CCc2cnn[nH]2)CC1 32889,c1(NC(c2ccn(CC(F)F)n2)c2nnnn2CCC2CC2)cccc2[nH]ccc12 32890,C1(C)(COC)CC(NC(C2CN(C)C2)=O)CN1C(=O)CCc1nncs1 32891,CCCC(CCC)CC(=O)N(C(C)C(=O)NCCCCCO)C1CC1 32892,c1(C(=O)NC2(CNC(C3C(CC)C3)=O)CC2)cncc(Cl)c1C 32893,N1(C(c2c(CC)noc2)=O)CC2CC(C)N(C(c3cn(C)nc3Br)=O)C2C1 32894,c1(OC)cc(F)cc(C=CC(N2CCC2CNC(c2c[nH]cc2C(C)C)=O)=O)c1 32895,c1(C(N2CC3(CC(NC(C4(F)CCOC4)=O)C3)C2)=O)ccc2nc(O)oc2c1 32896,C#Cc1cc(F)c(C(N2CCN(C)C(CC)C2)=O)c(F)c1 32897,N12CC3CCCC3(C1)C(=O)Nc1c(cc[nH]1)C2=O.c1(SCC)ccnc(F)c1 32898,C1(OCC)CC2(CCN(C(=O)CC=CC(C)(C)C)C2)C1.C12C(C1(C)C)NC2=O 32899,c1(NC2(C)CC(NC(C(C)Sc3ccccn3)=O)C2)ccnc2ncnn12 32900,CC(C)(CC1CC1)C(=O)NCC1CCN1C(c1c[nH]cc1Br)=O 32901,C1(C)(CNC(c2c(C(C)C)c[nH]n2)=O)CCCN1C(=O)COC(F)F 32902,C(=O)(N=c1ccn(C(C)(C)C)[nH]1)C1CC(N(C(=O)C(C)(C)C2CCC2)C)C1 32903,C(=O)(CCCCN=[N+]=[N-])N1CC(C(C(N2CCC(OCC)CC2)=O)O)C1 32904,Cc1cc(CC(=O)N(CCCNC(C2(C)CCOC2C)=O)C(C)C)cc(C)c1 32905,N1(C(c2ccc(CC)cc2O)=O)CCC2(CC(NC(=O)C(C)OCOC)C2)C1 32906,Cn1nncc1CC(=O)NN(CC(=O)NCCOCC(F)(F)F)CCO 32907,c1(C(N2CCC(CNC(C3C(OCC)C3)=O)C2)=O)ccc(-c2ccc(Cl)s2)cn1 32908,C1(NC(c2ccsn2)=O)C2CC3C1C3C2C(N1CC(n2cccn2)C1)=O 32909,N1(CC(=O)OC(C(=O)Nc2c(C)nc[nH]2)C)CCN(c2ccc(F)cc2)CC1 32910,C(=O)(C(O)C(F)(F)F)N1CC(N2C(CN(C)C)COCC2)C2C(C1)C(=O)C2 32911,c1(C(=O)NCCOCCCNC(CC2C(C)C2)=O)ccc(N(C)C)nn1 32912,c1(NC(C)Cn2cccn2)ccnc(N(C)CC2CC2(F)F)n1 32913,C1(N(C(CC2(CC)CCC2)=O)C)CC2CCC(C1)N2C(c1occ2c1CCC2)=O 32914,C=CCCCCCCCCCNC(=O)N(CCC(F)(F)F)CC 32915,N1(CC2CCCN(c3nc(C)cc(=NCC)[nH]3)C2)CCc2c(C)cccc2C1C 32916,N12CCC(C1)CC2=O.c1(CC2(CNC(C(C)=O)=O)COC2)ccccc1 32917,c1(CC(CC2(N(CCN3CCCC3)CC)CC2)=O)cn(CC(=O)C(C)C)nn1.OC 32918,c1(C2(NC(C(C)CN3CCCC3)=O)CC2)cccc(O)n1 32919,S(=O)(=O)(c1ccc(Br)cc1)NCC(=O)NCCNC(c1cccc(CO)c1)=O 32920,N1(C(c2c(CSCC)cccc2)=O)CC(C2CN(C(=O)CCCCC(N)=O)C2)C1 32921,N1(C(c2nnn(C(C)(C)C)n2)=O)CCCC(n2cc(-c3ccnc(Br)c3)nn2)C1 32922,N1(C(Cc2nc(C(C)OC)sc2)=O)CC(NC(=O)C(C)C)C(C2CC2)C1 32923,c1(CC(=O)NC(CC)CN(C(=O)C(C2CC2)SC)C)cc(F)ccc1C 32924,N1(C(CC(C=C)(C)C)=O)CCC2(CCCCC2NC(C2CCC(C)(CC)O2)=O)C1 32925,N1(C(c2ccn(C(C)C)n2)=O)CCOC(C(C)NC(c2cncn2C)=O)C1 32926,C(C(C(C)(C)C)NC(=O)Cc1csc(C(F)(F)F)n1)NCC1(C)CCCO1 32927,CCC(C)(C)CCNC(=O)C=CC(C)(C)NC(=O)C(C)C(F)F 32928,c1(COC)ccc(CNC(=NCC2CCCCCC2)NC2CCS(=O)(=O)C2)cc1 32929,Cc1c(CCNC(CC(C)C)c2nnnn2C2CCCCC2)cccc1Br 32930,N1(C(C23CN(C(c4cc(C)c(C)s4)=O)C(C2)CO3)=O)CCCC(C2(C)CC2)C1 32931,C(CCF)(C(=O)NCCC1CCCCO1)NC(c1cc(C)[nH]c1)=O 32932,C(=O)(C1=C2CCCN=C2NN1)NC(CCCOC)c1cccnc1 32933,C1(COC(C(CCC)NC(=O)OC(C)(C)C)=O)CCCS(=O)(=O)C1 32934,C1(COC)CN(C(c2cc(C#N)oc2C)=O)CCN1C(=O)C1=C(Cl)CCC1 32935,C1(OC)CCn2cc(C(=O)N(C)CCN(C(=O)CC3OCCC3C)C)nc2C1 32936,C(c1cncnc1O)=CC(N1CCC(C(C)NC(=O)CC(F)(F)F)C1)=O 32937,N1(C(Cc2cc(C)[nH]n2)=O)CCOCC(C)(CNC(C2CCC2C(C)(C)C)=O)C1 32938,N1(C(C(c2n(C)cnc2)O)=O)CCOC(C2CN(C(=O)CC3CC=CCC3)C2)C1 32939,C1(CC)CCC(C(N2CC(N(C)C(c3ccc(-c4ccccn4)s3)=O)C2)=O)C1 32940,N1(C(CCc2cn(C(C)(C)C)nn2)=O)CC2CCC1C(O)C2.N12CC(C)(C)C1C2 32941,c1(C(N(CCCCNC(C(CCC)O)=O)C)=O)cc(F)cc2c1NCCC2 32942,C1(C(N2C(CCNC(C(COC)(C)C)=O)CCC2)=O)CCCC1P(C)(C)=O 32943,c1(C(=O)NCCN(CCOC)C(c2nnn(C)c2C)=O)cc2ncn(C)c2cn1 32944,c1(C(N(C)CC2(NC(=O)CCCN3CCCCC3)CC2)=O)ccc2nonc2c1 32945,Cc1cc(C(=O)NCCC2(NC(=O)CCC(=O)N(C)C(C)C)CCCC2)c(C)cn1 32946,Cc1nn(CCC#N)c(C)c1C(=O)N(CCc1cn(CCCS(N)(=O)=O)nn1)C 32947,CC(C(C)(C)C)=CC(=O)NCCN(C(=O)CCCCCCC)CC1CC1 32948,c1(C(=O)NC(C(C)NC(c2cccc(OC)c2O)=O)C)cc2nc(F)ccc2o1 32949,S(=O)(=O)(c1cccc(=NCC2C(F)(F)C23CCC3)[nH]1)NC(CCCCC)(C)C 32950,[N-]=[N+]=NC1CCC(C(=O)NC2CCN(C(c3cc(-c4cccs4)on3)=O)CC2)C1 32951,C(c1cnc2ccccc2n1)=CC(=O)NC1C2CN(C(C(C)(C)CO)=O)C1CC2 32952,c1(C(=O)NCCC2(OC)CN(C(C(CCC)C)=O)C2)cc(Cl)c(Cl)cc1OC 32953,Cc1cc(C(=O)NC2CN(C(=O)CNC=O)CC2(C)C)c2nc(C)n(C)c2n1 32954,C1(C(C)C)(Nc2ccccc2NC(N2CC(CCC)SCC2)=O)CCC(O)CC1 32955,S(=O)(=O)(c1ccc(Br)cc1NC(c1ccccc1)CF)N(C)CC1CN(C)C1 32956,C(c1cccc(F)c1)=CCC(=O)NC1COCCC1NC(c1cccnc1)=O 32957,c1(N(CC(c2ccccc2)CO)C)ncnc(NCc2nnc(C)s2)c1C 32958,Cc1cc(=NC2CCS(=O)(=O)C2)[nH]c(=NCCCC(=O)N2CCCCC2)[nH]1 32959,N1(C(CC2CCC(NC(C3(OCC)CCOC3)=O)CC2)=O)CCC(O)C(C)C1 32960,C1(C(=O)NC(CN2CCCC2)CO)(CO)CCN(C(C2CC=CCC2)=O)C1 32961,c1(C(N2CC(C=C)C(NC(c3[nH]nnc3C)=O)C2)=O)nn(C)c2c1C(O)CCC2 32962,N1(C(C2(C)COC2)=O)CCCC2CN(C(=O)C(C#N)C3CC3)CC12 32963,N1(C(C2C(C)CC(=O)N2)=O)CCC2(C1)CN(C(=O)CC1CCCC(F)(F)C1)C2 32964,c1(CNC(=NC)N(C)Cc2conc2CC)cccc2c1OCCO2 32965,c1(CC)ccc(NC(=O)C(CC2CCCC2)NC(C2CCC(COC)O2)=O)cc1 32966,CC(CC(C)(C)C)C(=O)NCCNC(=O)CC1CCC(C)(C)CO1 32967,C1(C(N2CC(N(C(CCC#C)=O)C)C3(C2)CC3)=O)CC2CCC1CC2(F)F 32968,n1(CCCC)ncc(C(=O)NCC2(Nc3nnc(C(C)(C)C)s3)CC2)c1C 32969,N1(C(CN(C)CO)=O)CCC(C2CCCCN2C(=O)COCC2CCCO2)CC1 32970,C(=O)(C(C)(O)C(F)(F)F)NC(c1n(C)ncc1)C(N1CCC(N(C)C)C(F)C1)=O 32971,C(=O)(C(C)CC(F)(F)F)NCC1CN(C(CN(CCC#C)C)=O)CC1(F)F 32972,N1(C(C2N(C)CCC2)=O)CCC(C2CCC2)(NC(=O)C=CC2CC2)CC1 32973,CCC(CC)CCCC(=O)N(C(CNC(C1CC(=O)N(OC)C1)=O)CC)C 32974,N1(C(C(CC(C)C)O)=O)CCc2nc(O)cc(C(=O)NCCc3nccs3)c2C1 32975,C(=O)(CCCS(N)(=O)=O)NCC1CC(NC(C=Cc2ncc(C)[nH]2)=O)CC1O 32976,N1(C(Cc2c(OC)ccnc2)=O)CCOCC(NC(C2CCCC(OC)C2)=O)C1 32977,c1(C(=O)NCCC(C)NC(c2c(OC)cncc2)=O)cc(Br)c(C)nc1O 32978,C(=O)(C(CC(C)(C)C)c1ccccc1)N1CC(CC(=O)OC)CC1(C)C 32979,c1(C(N2CC(C)C(NC(C3CN4CCN3C(C)C4)=O)C2)=O)cc(F)c(F)cc1F 32980,Cc1nc2sccn2c1C(N1CCC(C)(CNC(C2CC3CC3C2)=O)C1)=O 32981,C1(CNC(CC(C)(C)C)=O)CN(C(=O)CSc2ccccn2)CCCO1 32982,c1(C(=O)NCC(C2CC2)NC(CC2(C#N)CCC2)=O)ccc2nc(O)[nH]c2n1 32983,C1(NC(=O)C2=CCCC2)C2CC3C1C3C2C(=O)NCc1cccc(F)c1O 32984,C(=O)(C(C(C)C)n1cc(Br)cn1)NCCNC(C1C(OCC)C1)=O 32985,CC(=NOCC#N)C(=O)N1CCN(CC(=O)NCc2cc(C)ncn2)CC1 32986,N1(C(CCC)=O)CC(OC)CC1(C)CNC(c1ccc(C)nc1O)=O 32987,C1(C(N(CCF)CC)=O)CCC(NC(=O)C=C(C)C)CC1 32988,C1(O)(CCNC(CC(=O)NCC=C)=O)CCN(C(=O)C(C)=CCO)CC1 32989,C12(CCCOC1)CO2.c1(CC)nnc(Cn2nnnc2C2(N)CCCC2)o1.CC 32990,C(C(C)(O)CC(=O)N1CC2(CC2)CC1CC(=O)N(CC(C)CO)C)OC 32991,N1(C(COCc2c(C)ncs2)=O)CCC(C)C(NC(C2CC(C)(C)C2)=O)C1C 32992,c1(C(N2CC(CNC(C3CN(S(N)(=O)=O)C3)=O)C2)=O)cnc2c(c1)CCCO2 32993,c1(C(=O)NCC2(OC)CN(C(C(CSC)O)=O)C2)cc(C)c2nc(C)nn2c1 32994,C#CC1(C)CCCN(C(=O)C(C)N(CCC)C(c2cnn(C(F)F)c2)=O)C1 32995,N1(C(C2CC(OC)C2)=O)CC(NC(c2cc(C)cc(O)n2)=O)C2(CCC2)C1 32996,c1(OC)cc(CC(=O)NC23CC2CN(C(c2nccnc2Br)=O)C3)ccn1 32997,C1(CC(=O)N(CC(C)O)CCNC(C=C(CCC)C)=O)CCCC(F)(F)C1 32998,C1(NC(C(Cc2c(C)n[nH]c2C)C)=O)CCCCN(C(c2coc(O)n2)=O)C1 32999,C1(COC)(NC(c2cnn(C)c2F)=O)CCN(C(=O)CC2CCCO2)CC1 33000,N1(Cc2n(C)ccn2)CC2CCC(C1)N2C(c1ncccc1F)=O 33001,CC(C)CCC(C(=O)NC1CCN(CCF)C1)NC(=O)C=Cc1nccs1 33002,Cc1cc(Cl)c(CN2CC(CC(N3CCC(=O)CC3)=O)C2)c(Cl)c1 33003,CCCC(C)CN(C(=O)C(C)N(C(=O)CC(C)n1cccc1)C1CC1)C 33004,C1(C(=O)NCCCN(C)C(C23CCCC2C3)=O)CCc2ncccc2C1 33005,c1(C(N2CCCCC2C)C(=O)NC(C(=O)OC)C)cc2c(Br)cccc2o1 33006,c1(C(N2CC(CNC(C=CC(C)C)=O)C3C2C3)=O)cccc2c1CCC2=O 33007,C1(CNC(C(C)OC)=O)COCCN1C(c1cc(-c2ccco2)no1)=O 33008,C1(CNC(=O)Cn2cncn2)CN(C(C2CC3CC(=O)C2O3)=O)CC1(F)F 33009,c1(C(N(CCNC(=O)C(C)OCC(F)(F)F)CC)=O)cn2nc(C)cc2[nH]c1=O 33010,c1(CC)cc(C(N2CCCCC2CNC(=O)CC2CCC(C3CC3)O2)=O)sc1C 33011,Cc1cc(C(N2CCC3(CC3C(=O)NCCCC3CCCCC3)C2)=O)nc(C)n1 33012,CN1N=C(C(=O)NC(C(N2CCCC(NC(N)=O)C2)=O)c2ccoc2)CCC1=O 33013,C(=O)(CCC(F)(F)F)NC1C(NC(c2c(-c3cn(C)nc3)nccc2)=O)C1 33014,N1(C(c2c(CC)con2)=O)CCCN(C(c2cc(C(F)F)c(Cl)cn2)=O)CC1C 33015,N1(C(=O)Cn2ccc(C(F)F)n2)CC2CN(C(C3CC3(F)F)=O)CC2C1 33016,Cn1cnc2c1CCCC2C(=O)NC1CCN(C(=O)CN2CSCC2=O)CC1F 33017,C1(NC(=O)NCC(N2CCCC2=O)C)CN(C)NC1=O 33018,c1(C(=O)NCC(CO)NC(CS(C)(=O)=O)=O)cccc(S(=O)(=O)C(F)F)c1 33019,C1(CCNC(c2cc(C)nnc2)=O)CN(C(C2C(C)(C)OC2(C)C)=O)CC(C)O1 33020,C(CC(C(C)C)NC(=O)CCc1ccc(Cl)nc1)N(C(c1c(CC)ccs1)=O)C 33021,c1(C(=O)NCC2CCN(C(C#CC(=O)N(C)C)=O)CC2)cc(Br)ccc1OCF 33022,N1(C(C(=O)NCc2ccc(OC(F)F)c(OCF)c2)=O)CC2CC1CN2CC(F)F 33023,C(=O)(C(C(C)C)SC)N(C1CCN(C(=O)C(c2ccccc2)SC)CC1)CC#C 33024,c1(C(=O)NCC2C(NC(C(C)OCC=C)=O)CC2)c[nH]c2ccc(C#N)cc12 33025,N1(C(C)C(=O)NCCCN(C(=O)C=Cc2ccco2)C2CC2)C(=O)CCC1=O 33026,c1(C(N2CCC(NC(C3N(N=O)CCC3)=O)C2)=O)cc(C2CC2)cc(F)c1 33027,Nc1cc(Cl)ccc1C(N1CC2(C1)CN(C(c1coc(C(N)=O)c1)=O)C2)=O 33028,CCCCC(O)C(=O)NCCCC(CCC)NC(c1cc(CCC)n(C)n1)=O 33029,c1(CCC)occ(C)c1C(=O)NC1CC1C(=O)N(C)CC1CCCS1 33030,c1(CCNC(c2nc(CC3CC3)cs2)=O)cccc(I)c1 33031,C1(OC)CN(C(c2ncncc2F)=O)CC1NC(c1ccc(N(C)C)nn1)=O 33032,Nc1c(F)ccc(F)c1C(N1CCCOC(CNC(C2CC2C2CCC2)=O)C1)=O 33033,c1(CC2(CNC(C3CN(C(Cc4nnc(C)o4)=O)C3)=O)CC2)ccc(F)cc1 33034,Cc1nc(N(C(C)CCNC(C2(C3CCCO3)CC2)=O)C)[nH]c(=N)n1 33035,C1(NC(C)=O)CCC(C(=O)NCCN2CCCC2=O)OC1 33036,Cn1nc(-c2cn(CC3CC4(CC4)CO3)nn2)cc1N 33037,c1(N2CCC3(CC(NC(C(CC)C)=O)C3)C2)ncnc2ccc(S(C)(=O)=O)cc12 33038,CC1(CNC(c2cc(C(F)F)no2)=O)CCN(C(C23CC(O)C2C3)=O)CC1 33039,c1(C(N(CCC(C)NC(c2ccoc2C2CC2)=O)C)=O)csc(C(N)=O)n1 33040,c1(-c2nc(C(C)SCC)nn2CC)cnn2c1CC(C)CC2 33041,c1(CC(N2C(CNC(c3cn(CC)nn3)=O)C(C)CC2)=O)c(O)nc(=N)[nH]c1C 33042,c1(C(=O)NC2(CC#C)CC2)ccc(CNC(=O)CC(Cl)Cl)nc1 33043,C1(CC)CN(C(C(=O)NCc2cccc(Br)c2)C2CC2Cl)CCN1C 33044,C1(CNC(C=CSC)=O)CN(C)CCN1C(=O)Cc1ncccc1C 33045,C(c1cccc(F)c1)=C(C(=O)NC1C=CCN(C(c2c(CC)onc2C)=O)C1)F 33046,Cc1cccc(C(O)C(N2CCOC(CN(C(=O)Cc3nnc(C)s3)C)C2)=O)c1 33047,N1(C(c2cc(OC)nc(C)c2)=O)CCC(N=c2nn[nH]n2C)C(C)C1 33048,C1(CNC(C(C)OC(C)=O)=O)CCC(C(=O)N(C2CC3CC3C2)C)CC1 33049,C1(C(=O)NCCC2OCCN(C(CC3C(OC)CC3)=O)C2)CCCCC12CCC2 33050,C(CC(O)CC(=O)NCCN(C(=O)C(C(C)(C)C)C1CCC1)C(C)C)SC 33051,c1(CCC)cc(C(=O)N(C)Cc2ccc(Oc3ccccc3Cl)cc2)cc(O)n1 33052,c1(C(=O)NC)ccc(CNC(c2csc(NC(=O)OC(C)(C)C)c2)=O)nc1 33053,CCCCC(C(=O)N1CCCOC(CNC(=O)CCc2scnc2C)C1)N(C)C 33054,Cc1ccc(C(N2CCC(N(C(=O)C(C)c3cncs3)C)C2)=O)cc1 33055,c1(C(=O)NCC2N(C(c3cccc(N)c3C(F)F)=O)CC2)cc2cccnc2[nH]1 33056,c1(N2CCC(CC)(CC)C2)nc(=NCC(C)(C)N2CCCC2)[nH]c2ncn(C)c12 33057,C1(Cn2cc(C(C(C)(C)C)O)nn2)CCCN(C(=O)C(c2cscn2)N(C)C)C1 33058,c1(OC)cccc2c1OCCC2NS(=O)(=O)c1cccc(F)c1C(=O)O 33059,c1(OC)ncccc1S(=O)(=O)N1CCN(C(=O)Cc2cccnc2Cl)CC1CO 33060,N(C(=NC(C)C)N1CCCCC(S(C)(=O)=O)C1)C(C#C)C(C)(C)OC 33061,N1(C(c2c(OC)cc(C)cn2)=O)CC(NC(=O)C2=CCCC2C)C(N=[N+]=[N-])C1 33062,Brc1c(-c2noc(CSc3cccc4nccn34)n2)cc(Br)c2nsnc12 33063,C(=O)(C#CC1CCCOC1)NCC1C2CN(C(c3cc(C(C)=O)c(O)cc3)=O)CC21 33064,c1(C(N(C)CC2CCN(C(=O)Cc3cncc(F)c3)C2)=O)cnc(N)c(N)c1 33065,Cc1ccc(C(=O)N(C)CC2CCCN2C(=O)CC2CC(CF)C2)cc1N 33066,c1(-n2cc(C3OCCN(C(=O)NCC4(O)CCOC4)C3)nn2)ccc2c(c1)CC2 33067,C#CCCC(C(=O)NC1(CC)CC(C)(C)C1)NC(C1CC2C=CC1O2)=O 33068,N1(C(=O)OC(C)(C)C)Cc2ccc(CNC(c3ccc4nn[nH]c4n3)=O)cc2C1 33069,c1(C(=O)NCC2N(C(c3c(C)con3)=O)CC(O)C2)ccc2nc[nH]c2n1 33070,N1(C(C2C(CC)C2)=O)CCCN(C(C2CCC(Oc3ccncc3)C2)=O)CCC1 33071,N1(C(CCC=C)=O)CCOC(CC(=O)N(C2CC2(C)C)C)C1 33072,C(CCP(C)(C)=O)NC(C1(N(C(=O)CCC2CCC(=O)C2)C)CC1)=O 33073,N1(C(c2n(CC)cnn2)=O)CC2CCCC2(NC(=O)CCc2n[nH]c(=N)s2)C1 33074,C1(CCCCNC(C(C)NC(CC)=O)=O)CCN(C(=O)Cc2ncoc2C)CC1 33075,C1(NC(C(C)NS(CC)(=O)=O)=O)CN(C(C2CCS2(=O)=O)=O)CCC1C(F)(F)F 33076,C(CC(C(=O)NC1CCN(C(C)=O)C1)NC(C1CCCSC1C)=O)=CC 33077,CC1(NC(=O)CC2CCCOC2)CN(C(=O)CC2(O)CC2)C1 33078,C1(F)(CNC(c2c(C)nco2)=O)CCCN(C(c2ccnn2C2CCC2)=O)C1 33079,CCC(C)C(CO)NC(=O)C(CC1CCOCC1)NC(c1cc(C#N)cs1)=O 33080,CCC(C)CCCCC(=O)NOCC(=O)NC(C)C(=O)NC 33081,C(=O)(C(C)(C)CO)NC(C)C(C)NC(=O)CCOc1cccc(Br)c1 33082,C(=O)(CCCCc1cnc[nH]1)NC1CC(NC(CCNC(C)=O)=O)C1 33083,C1(NC(CC(CC)C)=O)(CC)CCN(C(=O)CC23CCC(CC2)CC3)CC1 33084,Cc1cc(CNc2ccccc2CN2CCC(n3cc(I)cn3)CC2)ccn1 33085,C1(C(=O)Nc2c(OCCC)cccc2)CCN(C(c2ccccc2Cl)C)CC1O 33086,CC1CC(NC(c2ccns2)=O)CN1C(c1cc(Cn2cccn2)on1)=O 33087,c1(C(N2CC3C(NC(C(CC)OCC)=O)(C3)C2)=O)cc(C(C)C)nc(O)c1 33088,N1(C(Cn2c(C)ccn2)=O)CCOC2(C1)CN(C(C1CC(=O)N(O)C1)=O)C2 33089,n1(CC)c(C)cc(C(=O)NC2(CO)CCN(C(C3CC(C(F)(F)F)C3)=O)C2)c1C 33090,N1(C(c2n(C(C)C)ncc2)=O)CCOC2(C1)CN(C(=O)C(C)CS(C)=O)C2 33091,CCC(C(=O)OC)C(=O)NCC(CC)NC(=O)CC1(c2ccon2)CCC1 33092,c1(CO)ccncc1.C12CCN(C1)C(=O)C1(CC1)OC(C)C(=O)N2CCC 33093,N1(C(C2(CC)CCOC2)=O)CCCC(C)(CNC(c2csc(CC(C)C)n2)=O)C1 33094,c1(OC)ccc(CCC(=O)NC2CN(C(=O)CN(C)CCO)C3CC23)c(OC)c1 33095,C(=O)(CC1OCCc2ccccc21)N1C(C(=O)NCc2c(F)cccc2Cl)CC1 33096,C1(OC)CC2CCC(C1)N2C(=O)C1=CCN(C(=O)CC2CCCCN2C)C1 33097,c1(C(N(C2CCCN(C(C3CNC(=O)C3)=O)C2)C)=O)cc(Br)cc2nc[nH]c12 33098,N1(C(COCCCOC)=O)CC2(C1)SCCC2NC(=O)C(O)P(C)(C)=O 33099,O=C(C1=CC2(CCOC2)C1)N1CCCCC(CNc2cnc(F)cn2)C1 33100,c1(C(N(C)CC2(CNC(=O)C(C)(C)Br)CC2)=O)cn(C)nc1-c1ccco1 33101,c1(NC(C2CN(C(C3CCCCS3)=O)CC2CO)=O)nccnc1-n1ccnc1 33102,CCC(C#N)(CC)C(=O)N1CC(NC(=O)Cn2nc(C)ccc2=O)C(C)C1 33103,c1(C(=O)NCCC(=C)CNC(C23CCCCC2C3)=O)cc(C)cc(C)c1C 33104,N1(C(C(CC)N(C)C)=O)CC(NC(=O)CCc2cccnc2F)C(C)(C)C1 33105,C1(NC(C2C(CNC(C3(C#N)CC3)=O)CCC2)=O)CC2C(O)C(O)CC12 33106,c1(NCC(C2CCN(C(CC3CCC(C)C3)=O)CC2)(C)C)nccc(C#N)n1 33107,C(C)(CCC(=O)NC(c1nnc(O)n1C)C)NC(CCOCCC)=O 33108,c1(C(=O)NCC(CN(C(C(CC(C)C)C)=O)C)O)cc(Br)cc(F)c1F 33109,N1(C(CCSC)=O)CCCC2(CCN(C(c3c(N)cc(Cl)cc3Cl)=O)C2)C1 33110,CN1N=CC(CC(N2CCOCC2CCNC(=O)CCC(N)=O)=O)C1=O 33111,c1(C(=O)NCCCN(C)C(c2cc(Cl)sc2Cl)=O)csc(S(N)(=O)=O)c1 33112,Cc1c(C(N2CCCC2Cn2cc(CC3(O)CCSC3)nn2)=O)sc2nccn12 33113,C1(C(N(CC(C(C)C)OC)C)=O)CC2(CC2)CN1C(c1cc(C)ccc1F)=O 33114,c1(C(N2C3CC(CNC(C(CCC)(C)C)=O)C2CC3)=O)cc2n(n1)C(C)CCC2 33115,c1(CC(=O)NCCNC(CCOc2ccc(C)cc2)=O)ccc(F)c(F)c1 33116,C(CC(=O)NC(Cn1cncn1)CC)(C(F)F)NC(C1(OCC)CCC1)=O 33117,C(CC(=O)NC(C1CN(C(c2nc[nH]c2C(F)(F)F)=O)C1)C)(C(F)(F)F)OC 33118,N1(C(C2C3CCC(F)C23)=O)CC2CCCC2(C(N2CCCCC2CO)=O)C1 33119,c1(C(=O)OC)nc(CCNC(=O)CC(c2ccc(F)cc2)C)n(C)n1 33120,N1(C(CC(C=C)(C)C)=O)CC(NC(c2cnn(C(C)C)c2)=O)C(N=[N+]=[N-])C1 33121,C1(C)(CNC(CC2C=CC(NC(CC(C)SC)=O)C2)=O)CC(C)=NO1 33122,N1(C(C(C)OCC)=O)CCCC12CCCN(C(C1(C)CCCCCC1)=O)C2 33123,C1(C(=O)NCC2(CNC(=O)C(C)Cn3ccc(C)n3)CC2(F)F)(OC)CCSC1 33124,Cn1cc(CNC(C2CCCCC2NC(C2CCCCC2)=O)=O)ccc1=O 33125,C(=O)(CC(C(F)(F)F)N(C)C)NC1(C(=O)NC(C(CC)C)CO)CCOCC1 33126,c1(NC(C=CCN(C(=O)CC2CCOC(C3CC3)C2)C)=O)c(Cl)cccc1Cl 33127,CCCC(C(=O)NC(C)CC)NC(=O)CC1CC2CC2C1 33128,C1(NC(=O)CCc2cnccn2)CC2CN(C(c3cscc3Cl)=O)CC2C1 33129,n1(CCC)ccc(S(=O)(=O)NNC(=O)C2CC2c2ccc3c(c2)OCO3)n1 33130,c1(C(=O)OC)c(C=CC(=O)N(C2C3CCC2CNC3)C(=O)C(=O)CCl)cnn1C 33131,C1(C(N2CCC(CC)C2)=O)N(C(c2snnc2C)=O)CCC1(C)C 33132,c1(CCNC(c2c(-c3c(OC)csc3)ncs2)=O)ccc(Br)cc1F 33133,c1(C(=O)NCCC2CN(C(CC(C)C)=O)CC(C)O2)coc2c1NC(=O)CCC2 33134,c1(OC)cc(C#N)ccc1CN1CC2CC(C1)N2C(c1ccc2c(c1)OCO2)=O 33135,C1(C(=O)NC2CC(CCNC(c3cn(C)c(=O)cn3)=O)C2)CCCC1S(C)(=O)=O 33136,CC1CCC(N(C)C(c2cc(C(F)(F)F)co2)=O)C1 33137,C(CS(=O)(=O)CC(=O)NC1CN(C(=O)CCc2ccncn2)CC1(C)C)OC 33138,C1(NC(=O)CCc2ccco2)CC2CC1CN(C(c1noc3c1CCCC3)=O)C2 33139,C(=O)(C1c2c[nH]nc2CN1C(=O)C(CO)N(C(=O)C1CC1)CC)N(C(CC(C)C)CO)C 33140,C(CCN(C)C(c1cc(F)cc(Cl)c1)=O)(C(C)(C)C)NC(C1C(C)OCCO1)=O 33141,C1(N(C(c2c(C)nco2)=O)C)CCCC(NC(=O)C(c2cc(Br)co2)=O)C1 33142,N1(C(c2c(CC)nn[nH]2)=O)CCC2(CC1)CN(C(c1nn[nH]c1Cl)=O)CC2CO 33143,N1(CC)CCN(C(C(=O)NCCOC)C2COC2)CC1(C)C 33144,C12(NC(C(CC3CCCC3)NC(C3C(C#N)C3)=O)=O)CCCCC1OCC2 33145,N1(C(Cc2c(C)con2)=O)CCC(NC(C2CCS(=O)(=O)CC2)=O)C12CCC2 33146,CCCC(C(=O)NOC)NC(C1CC(O)CN1C(=O)OC)=O 33147,C1(NC(c2cc(C(N3CCC(F)(F)C3)=O)on2)=O)CC2(CO)COC1C2 33148,c1(NC(CNC(=O)C(N2CCCC(C(O)C(F)(F)F)C2)=O)=O)cccc(O)c1 33149,Cc1nc(N2C(C)CC(CNC(c3ccoc3Br)=O)C2)c2c(C)c(C)sc2n1 33150,C1(C)(C(N(CC#C)CC=C)=O)CC(O)CN1C(c1cnnn1CC)=O 33151,C1(CN2CCC(Cn3ncc(CO)c3)CC2)COC2(CCC2)CO1 33152,C1(C2(O)CN(C(c3oc(SC)cc3C)=O)C2)(CNC(C(C=C=C)C)=O)CC1 33153,c1(OC)cc(CNC2CC2C(N2CC(OC)CC2CO)=O)c(Cl)cn1 33154,N1(C(Cc2ccc(NC(C)=O)s2)=O)CC(C)CN(C(=O)COCC(F)F)CC1C 33155,c1(OCC)cc(CNC2CCC(C)(C(C)C)C2)ncn1 33156,c1(C(N2CCN(C(=O)C=CBr)C(C3CCC3)C2)=O)cccc2nonc12 33157,C1(CNC(CSCC)=O)N(C(c2cc(C(C)(C)C)on2)=O)CCCC1(C)C 33158,C1(NC(=O)NCC=CCCC)CC(=O)N(c2ccc(OC)cc2)C1 33159,N1(C(C(CC)NC(C)=O)=O)CCCN(C(c2ncccc2C(=O)OC)=O)CC1C 33160,C1(OCc2cn(C3(NC(CCC(=O)OCC)=O)CC3)nn2)CC(C)(C)OC1=O 33161,C1(C(=O)NCC(CNC(CNC(=O)OCC)=O)F)CCCN1S(C)(=O)=O 33162,C1(C(=O)NC2CCC(OCC)CC2)C2CCC(C2)C1NC(=O)C1=CCCC1C 33163,N1(C(C=COCC)=O)CCC(NC(c2cc(Br)c(C(F)F)s2)=O)CC1C 33164,c1(C(=O)NCC2CCN(C(c3c(C)nc(C)o3)=O)C2)c(C)cc(F)cc1Br 33165,N1(CC(=O)NCc2ccsc2)CCC(C2CNC2)CC1 33166,N1(C(c2cc3c(s2)CCC3)=O)CC2CC(C1)N(C(=O)C=Cc1cccs1)C2 33167,C1(C(=O)NCC(CCC)(C)O)CCC2(CC2)N1C(=O)CC1(O)CCCCC1 33168,Cc1ccc(NC(C2CN(C(C3CCCCN3C)=O)CC(F)(F)C2)=O)c(C#N)c1 33169,Cc1cc(CNC(C2(CCNC(=O)COCCCF)CC2)=O)c(C)s1 33170,C1(NC(CCC=CC)=O)CC(O)CN(C(c2cnn(C3CCCCC3)c2)=O)C1 33171,C(=O)(C(O)C(C)(C)C)N1CC(C(C(=O)NC2CC(C(=O)NCC)C2)OC)C1 33172,C1(C(=O)Nc2ccc(C(CC(=O)OC)N)cc2)C2C=CC(C2)C1CO 33173,Cc1ccc(C(C)C(=O)NCC2CN(C(=O)C=Cc3cn(C)nn3)CCO2)cc1 33174,n1(CC)cc(C(=O)NCc2c[nH]nc2C2CCN(C(=O)COC)C2)cn1 33175,Cc1cnc(C(=O)NC(Cc2cnn(C)c2O)C(=O)N(C(C)C(C)(C)C)C)cn1 33176,C1(CNC(c2nc(COC)sc2)=O)(CO)CCCN(C(C23CCC2C3)=O)C1 33177,Cn1ccnc1S(=O)(=O)Nc1nc(CC(N2CCCCC2)=O)cs1 33178,c1(C(N2CCCC(C)(NC(C(C)n3ccnc3)=O)C2)=O)ccc2sncc2c1 33179,N1(C(CS(C)(=O)=O)=O)CCC2CCC12CNC(=O)CCOc1ccc(F)c(Cl)c1 33180,CCC(F)(F)CC(=O)NCCn1cc(C(=O)NCC2CC(=O)NC(C)C2)nn1 33181,N1(C(C2N(C(=O)CN3CCC(C)C3)CCC(C)C2)=O)CCCC(C2(C)CC2)C1 33182,N1(C(CCNC(=O)NC)=O)C2CCC1CC(CNC(=O)CC1(C)CC1)C2 33183,C1(C(=O)NC(C)Cc2cccnc2)CC(NC(C2CCCN2C(C)C)=O)C(O)C1 33184,Cn1cnc2cc(CC(=O)NCC3CC(NC(C4CCCC4)=O)C(O)C3)ccc12 33185,C(C(=O)N(CC(C)(C)CNC(c1nocc1C1CC1)=O)C)(C(C)C)SCC 33186,C1(NC(C(C)NC(COC)=O)=O)(CNC(C2CN(C)CCO2)=O)CCCCCC1 33187,CN1N=C(C(=O)NC2CCCCC2CC(=O)NCCC2(C)CC2)CCC1=O 33188,C1(C(N2C(CNC(c3c(C(=O)OCC)[nH]cc3C)=O)CC2)=O)CCCC(C)(C)O1 33189,C1(C)(NC(N2CC(c3nc(-c4nc(CC)sc4)on3)OCC2)=O)CC2(CCC2)C1 33190,c1(C(=O)NCC(CC=C)NC(=O)C(C)(C)C(=C)Cl)cc2c(C)cc(Cl)cc2[nH]1 33191,C1(CC(=O)NC(C2CCN(c3ncccn3)CC2)C)CN2CCN1CC2 33192,N(C1CCc2c1ccc(F)c2F)C(CCSc1ccc(C)cc1O)=O 33193,N1(C(c2c(C)ccnn2)=O)CC(F)(F)CC1CCNC(=O)CN1CSCC1=O 33194,n1(CC)cnnc1C(=O)NCCOC1CN(C(=O)CCC2CCC(C)O2)C1 33195,c1(NC2(CNC(C3C(C)(COC)C3)=O)CCCC2)nc(C)nc(O)c1C 33196,c1(C(=O)NC(CNC(c2cc(C)ncc2)=O)(C)C)cc(N2CCCC2)nc(Cl)c1 33197,CCS(=O)(=O)CC(=O)N1CC(CNC(c2cc(F)n(C)n2)=O)CC1C 33198,N1(C(C=C(CCN(C)C)Cl)=O)CCOC2(C1)CN(C(C1CCCN1N=O)=O)C2 33199,c1(C(N2CC(=C(CNC(C3C(=C)C3)=O)F)C2)=O)n[nH]c(C(C)(C)C)n1 33200,C1(CNC(C2CC(F)CN2Cc2c(CC)n[nH]c2)=O)CN2CCN1CC2 33201,N1(C(C(c2cccs2)SC)=O)Cc2ccnc(Cl)c2C1 33202,C(=O)(C1CSc2ccccc21)n1c2ccc(c(F)c2)c1=O.C(CF)OC 33203,Cc1ccc2[nH]cc(CC(N3CC(NC(C4(C(N)=O)CC4)=O)CC(O)C3)=O)c2c1 33204,c12ccc(cn1)C(c1nnnn1C)N2.C1(COC)CCCC1Oc1ccccc1 33205,C1(C(=O)NCC2(C(N)=O)CN(C(c3ccc(F)c(Cl)c3)=O)C2)CC2C(C1)C2(C)C 33206,C1(SC(C(=O)N)C2CCCC2)(CCNC(=O)Cn2cc(CO)nn2)CCCCC1.CO 33207,C1(NC(CCC=C=C)=O)CCCN(C(c2cscc2C#N)=O)C1C 33208,c1(CC)cnc(O)c(C(N2CC(O)(CNC(c3n[nH]cc3C(F)(F)F)=O)C2)=O)c1 33209,N1(C(C(C)OCCOC)=O)CCC2CC12C(=O)NCC(C1CC1)SC 33210,CC(C)CC(CNC(c1cocc1C(N)=O)=O)C(=O)NC(C)CC1CCC1 33211,c1(NC(C)C)cccc(C(=O)NC2CN(C(=O)C(C)=C3CCC3)CC2C)c1 33212,CCCC(CCCNC(=O)CC1CCCCCO1)NC(=O)CNC(=O)C(C)(C)C 33213,N1(C(c2scc(CNC(c3c(C)ocn3)=O)c2)=O)C2CCC1COC2 33214,c1(OC)cc(C(N2C3CCC2CC(NC(=O)CN(C)C)C3)=O)c(C)c(Br)c1 33215,c1(C(N(C2CC(NC(C3CCC(C)CC3)=O)C2)C)=O)cccc2nncn12 33216,C1(F)(CNC(c2n(CCC)ccc2)=O)CCN(C(=O)COCC2CCC2)C1 33217,N1(C(C2C3(CN(C(c4c(C)nn(C)c4C)=O)C3)C2)=O)C2CCC1CN(C)C2 33218,c1(CC(=O)OCC)cccc(Br)c1NC(=O)C(=O)Nc1ccn(C2CCCC2)n1 33219,CC1(C)Cn2[nH]c(=NC(=O)c3c[nH]nc3-c3ccc(F)c(Cl)c3)cc2CO1 33220,CN1CCC(NC(=O)CCC2CCC(NC(=O)CSC3CC3)C2)C(C)(C)C1 33221,c1(C(N2CCC(O)(C(=O)OC)C2)C(=O)NCCC)cc(Br)c(Br)o1 33222,C(=O)(CC(C)(C)C)NC(C)C(N1CCC(C(=O)Nc2cc(Cl)c[nH]2)CC1)=O 33223,N1(CC)CCOCC1C(=O)N(CC(O)CN(C(=O)CCN1CCNC(=O)C1)C)C 33224,C(CCN=C(NCC(C)C1CCC1)NCC(N1CC(C)OC(C)C1)(C)C)OC 33225,c1(CC)cccc(Br)c1C(N1CCOCC1C(N1CCCC1CC(=O)NC)=O)=O 33226,c1(C(N2CCCC(N(C(CCC(CC)C)=O)CCF)C2)=O)cccc2nsnc12 33227,C(CCC(=O)N(C)CCOCCCN(C(=O)C(C)CSc1ccccc1)C)=CC 33228,C1(C(N2CCC(N(C(c3cn(C)nc3O)=O)CC)C2)=O)CCc2nnc(O)n2C1 33229,c1(C(N(CCCN(C)C(C2CCC(CCO)CC2)=O)C)=O)cc2sccc2[nH]1 33230,N1(C(C2(CCC)CC(=O)C2)=O)CCC2(CC1)CC2C(=O)NC1CC2(CCC2)C1 33231,C1(C(=O)NCC2N(CC)CCC2)CN(C(C2CCC3(CCC3)C2)=O)CCN1C 33232,N1(C(c2c(C)cn(C)c2)=O)CC(C)CN(C(=O)Cn2cnnc2)CC1C 33233,C(=O)(C(C)(O)CC)NCCCN(C(CCCSC)=O)C1CCCC1 33234,C1(NC(C2C(CCC)C2)=O)CN(C(c2ccc(-n3cnnn3)cc2)=O)C(C)(C)C1 33235,C(CCS(C)=O)(C(=O)N1CC2C(NC(c3ccc(O)cn3)=O)C2C1)N(C)C 33236,c1(CC)onc(C(=O)NCC2(C)CCN(C(c3ncc[nH]c3=O)=O)C2)c1C 33237,C1(CNc2n(CC3C(NC(Cc4cc(CC)sc4)=O)CC3O)nnn2)C2CCC(C2)C1C 33238,C(=O)(C1CCCc2ccnn21)N1C(C)CC(NC(C2(OC)CCS(=O)(=O)C2)=O)C1 33239,Cc1nc(NC(C2CC2NCc2cc(F)ccc2O)=O)c(Br)nc1Br 33240,c1(C(=O)NC2CCC(CCNC(CC(C=C)C)=O)C2)c(C)nc2sccn12 33241,c1(C(=O)NC2C(C)CN2C(=O)C=Cc2ccco2)ccnc(OCCO)c1 33242,C(CC1=CCOCC1)NC1(c2nnnn2CC2CCOC2)CC(CC(C)C)C1 33243,N1(C(CSCC=C)=O)CCC(NC(c2cc(C3CC3)[nH]c2C)=O)CC1C 33244,C1(CNC(CCc2cnc(C)s2)=O)CN(C)CCN1C(=O)CCc1cnc[nH]1 33245,N1(C(C(CC=C)(C)O)=O)CC=C(C(=O)NC(c2nc[nH]n2)C2CC2)CC1 33246,CC(=Cn1ccnn1)C(=O)NCC12CCC(CN(C(c3cccnc3O)=O)C1)C2 33247,N1(C(c2cc(C)sn2)=O)CC2(CCN(C(=O)CCC3CCCC(O)C3)CC2)C1 33248,c1(OC)cncnc1-c1ccc(-c2nccn2CC2CCCCC2NC(C)=O)s1 33249,C1(C(=O)NC2N(CC)CCC2)CCN(CC(=O)N(C)C2CC2)CC1 33250,c1(C(N2CC=CC(NC(c3ncc(C)cc3C)=O)C2)=O)cc2c(O)cccc2[nH]1 33251,c1(-c2nc(-c3cc(C(c4ccco4)=O)on3)on2)cc2c(nn1)CCCC2 33252,C(=O)(C(C)N(CC(F)(F)F)C)NCCN(C(C1C(CCC)C1)=O)CC1CC1 33253,CCN=c1[nH]c(C(N2CCN(C)C(CNC(=O)C(C)OCCOC)C2)=O)cs1 33254,c1(CNC2CC3N(CCOC)C(CC3)C2)c[nH]c2ncc(Br)cc12 33255,N1(C(=O)OCC2N(CC)CCCC2)C(CO)CCC12CC2 33256,C1(CNC(C2COC(=O)C2)=O)CC(F)CN1C(=O)C(F)F 33257,CC1(C(=O)NC2CC3(C2)CC3NC(=O)CCc2cnccn2)CC2CCC1O2 33258,CCC(CC(F)(F)F)C(=O)NC(CCN(C(=O)CC(C)(C)O)C)C(C)C 33259,N1(c2n(CC=C)c(C(O)CCOC)nn2)CCC(C)CC(C)C1 33260,C1(NC(c2c(C)coc2C)=O)CN(C(c2ccnc(O)c2)=O)CCC12CCC2 33261,Cc1cc(C(N2CCN(C(=O)Nc3ccccc3)CC2)=O)nc(-c2cccs2)n1 33262,Cc1nc2sn(CC(C3CCS(=O)(=O)CC3)(C)C)c(=O)c2c(C)c1C.C(C(C)C#N)N 33263,C1(C(N2CC(NC(C3(O)CC(F)(F)C3)=O)C(O)C2)=O)CCOCC12CCC2 33264,N1(C(c2nc(CCC)sc2)=O)CC2ON=C(CNC(c3nc(C)oc3C)=O)C2C1 33265,CC(C)CC(CN(C)C)NC(C1(F)CCN(C(=O)CCCC2CC2C)C1)=O 33266,CCCC(C)(O)CC(=O)N1C2CCC1C(CNC(=O)CC1(C(F)(F)F)CC1)C2 33267,N1(C(=O)CCc2nccs2)CCCCC1C(N1CCOC2CC12)=O 33268,c1(CC(=O)NC(C(C)NC(c2cc(C)c(C)nn2)=O)C)ccc2ncsc2c1 33269,c1(C(C(=O)NCCCC2N(C(COCC#C)=O)CCC2)O)cccc(C)c1 33270,N1(CC(N2CCC(NC(=O)Cc3nc[nH]n3)(CO)C2)=O)CCS(=O)(=O)CC1 33271,N1(C(CC(=O)NC2CC2)=O)CCC(C(=O)NCc2cccc(F)c2)C12CCC2 33272,N1(C(C(CC)OC)=O)CCCCC2(CCN(C(=O)OC(C)(C)C)C2)C1 33273,c1(NC(=O)CC2CCCN(Cc3ccccc3OCCO)C2)ccc(F)c(Br)c1 33274,c1(C(CC)(C)NC(=O)NC2(Cn3cnnc3)CC2)ccc(F)cc1 33275,Cc1cc(CN2CC(F)(F)CC2C(=O)Nc2nc(Cl)nc(Cl)n2)cnc1Cl 33276,C=CC(CCC)CC(=O)NC12CCC(NC(=O)C(O)CC(F)(F)F)(CC1)C2 33277,N1(Cc2n(CC)ncc2)CCC2CN(C(c3ccc(F)c(C)c3F)=O)CCC12 33278,N1(C(CSC)C(=O)OC)CC(CCO)OCC12CC2 33279,C(C)(C)(CCC(=O)N1CCOC(CC(N)=O)C1)NC(C(CC)C)=O 33280,CCCCCC(O)CC(=O)NCCN(C(=O)Cc1ccccc1S(C)(=O)=O)C 33281,C1(OC)CC(CC(=O)NCC2CN(C(=O)CC=C(Cl)Cl)CCO2)C1(C)C 33282,N1(C(c2scc(C)c2)=O)CCC2(CC1)OCCC2NC(=O)C(F)C1CCC1 33283,C(=O)(CC1C(=O)Nc2ccc(Cl)cc21)OCC(=O)Nc1ncc(C)s1 33284,S(=O)(=O)(c1cc(F)cc(Br)c1)N(C(=O)C(C)Oc1ccc(F)cc1)C(C)C 33285,N1(C(C(CSC)O)=O)CCC=CC1C(=O)N(CC1CC1)CC1CC1 33286,c1(N2CCCC3(NC(c4nccnc4Cl)=O)C(C2)C3)ncc2cccnc2n1 33287,C(C)(C)(CCCNC(=O)CC1CC2C=CC1C2)NC(C1CN(C)C1)=O 33288,c1(C(N2CC(NC(=O)C=C(C)C)CC(OC)C2)=O)nn(C)c2c1CC(F)(F)CC2 33289,c1(C(=O)NC2CC(n3cc(C4(C)CC4)nn3)C2)cncnc1C1CC1 33290,c1(C(=O)NCCC2CC(NC(c3n[nH]cc3Br)=O)C2)ccc2scnc2c1 33291,C1(C#N)(OC)CC(C(=O)NC(CNC(c2c(Cl)n[nH]c2C2CC2)=O)C(C)C)C1 33292,N1(C(CCCCCCC)=O)CCc2ccccc2C1CCNC(=O)CN(C)C 33293,N1(C(CCCCCN(C)C)=O)CC(NC(C2OCCCO2)=O)CC12CCCCC2 33294,C1(C2CC2)(CNC(CC2(OC)CCCCC2)=O)CCN(C(=O)C2=C(C)OCC2)C1 33295,C=CC1CN(C(=O)C(OC)SC)CC1NC(=O)C(F)C(C)C 33296,c1(NC(N(CC(O)CO)CC)=O)cccnc1Sc1cnc(C)nc1 33297,CCC(O)C(C)C(=O)NC1CCC(CNC(c2c(C)noc2C)=O)C1 33298,N1(C(C2CC(C#N)C2)=O)CCCC(NC(=O)C=CCF)C1 33299,C(=O)(CS(=O)(=O)C1CC1)NC(C(C)C)CCN(C(=O)Cc1ccn(C(F)F)n1)C 33300,Cc1cc(NC(C2COC(C)(C)CO2)=O)ccc1NC(=O)CN(C)S(N)(=O)=O 33301,CCC(C)(C(=O)N1CC(NC(=O)Cc2ncc(F)cc2F)C(O)C1)C(N)=O 33302,CN1CC(C(=O)NCC(C)(C)NC(=O)C=CC(F)F)CCC1=O 33303,N1(C(c2ccc(Br)o2)=O)CCC2(CCN(Cc3cccnc3Cl)C2)C1 33304,c1(CCNC(c2n(CC)nnn2)C2(CC)CCCC2)nc2ncc(Br)cn2n1 33305,C1(NC(C=CCCC)=O)CCCC2CN(C(=O)CCc3cnn[nH]3)CC12 33306,C1(CNC(C2N(CC)CC2)=O)CCC2(CCC2)CN1C(=O)C(Cl)=CCl 33307,c1(CCC)nnsc1C(N1CC(CCNC(c2cnn(CC(C)C)c2)=O)C1)=O 33308,c1(SCC(NOCCCC(=O)OC)=O)cccc(C#N)c1 33309,C1(CNC(c2cscn2)=O)CCN(C(c2cc(O)ncc2F)=O)CCC1(F)F 33310,c1(NC(CC2(C)CC2(Cl)Cl)=O)ccnc(-n2cc(-c3ncoc3C3CC3)nn2)c1 33311,Cc1cc(Cl)nc(Cl)c1NC(C1CC(C)CCN1C(=O)COC1CCCC1)=O 33312,C(=O)(CCCCCN(C)C(C1CC12CCCCC2)=O)NCC1CN(CC)C(=O)O1 33313,Cc1ccc(C(=O)NCC2(C(C)NC(C3CNC(=O)O3)=O)CC2)c(O)n1 33314,c1(C(=O)NCCCC(C)NC(=O)C2CC2)cccc(OCc2ccccc2F)c1 33315,CCCC(C#N)NC(C12CC(n3cc(C4CCC4)nn3)C1C2)=O 33316,C1(C(N(CCCNC(c2ccnn2C(C)C)=O)CC)=O)CCCC(CF)C1 33317,C(c1ccoc1)=CC(N1CCC(NC(=O)C(Cl)(Cl)Cl)C1)=O 33318,C1(OCC)CC(CO)(OCCOC(C2CCC(c3ccccc3)CC2)=O)C1(C)C 33319,N1(C(Cc2cc(C)ns2)=O)CCCN(C(=O)CCC(CF)CF)C(C)C1 33320,c1(N2CC(C)C(CO)CC2)nccc(=NCCc2cccc(N)c2)[nH]1 33321,N1(C(CN(CCCCCC)C)=O)CC(NC(=O)C=CC(C)(C)C)C2(CCC2)C1 33322,c1(SC)nccc(C(=O)NCC(C2CC2)N(C)C(c2coc(C(C)C)n2)=O)n1 33323,c1(C(=O)NCCC2N(C(CCCC)=O)CC(OC)C2)cnc2sccc2c1 33324,C(C(CC(F)(F)F)NC(c1cccc(O)c1Cl)=O)NC(CCN(CC)CC)=O 33325,N1(NC(CCC2CCN(C(c3c(C)con3)=O)C2)=O)CC(=O)NCC1C(N)=O 33326,C#CCCC(O)C(=O)N(C(C)CNC(=O)C(C1CCCC1)NC(C)=O)C 33327,C1(C(=O)NC2(CF)CN(C(c3cc(C)no3)=O)C2)CCCC2(CCC2)O1 33328,N1(C(c2nc(CC)oc2)=O)CC2CC3CC2C1C3NC(c1ccn(CCF)n1)=O 33329,C1(CNC(c2cnn[nH]2)=O)CN(C(C2C3(CC3)C23CC3)=O)CC12CC2 33330,CC1CC(C(=O)N2CC(NC(=O)C#CC3CCC3)CC2CO)=NO1 33331,CC1CN(C(=O)C(c2ccc(Cl)cc2)O)CC1NC(=O)C(C)C1CCOC1 33332,C1(C(N(C)C)=O)C=CCN1C(=O)CCCN(C(=O)CC1CCCN1C)C 33333,c1(O)ccccc1C(C)CC.C12CC(CCS1)NC(=O)NCNC2=O.C(C)(C)(C)O 33334,c1(CCCCC)ccc(C(=O)NCC(CCOC)NC(=O)C(C)=C(C)C)o1 33335,C1(NC(c2c(CC)noc2C)=O)CC2CC(NC(=O)C(C3CCOCC3)F)C2C1 33336,Cc1cccc(C(=O)NCC2CC(C(=O)N3CC(C)(C#N)C3)=NO2)c1C 33337,Cc1ccc(CNC(C2C(O)CCN2C(C2CCC(C)(C)OC2)=O)=O)c(O)n1 33338,N1(C(C(C#N)C2CC2)=O)CCOC2(C1)CN(C(c1c(F)cccc1F)=O)C2 33339,C#CCCCCCC(=O)NC(C)(CNC(=O)CSc1cccc(F)c1)C(C)C 33340,c1(OC)cc(F)c(C(N2CC(C)(NC(=O)CC3(N(C)C)CCC3)C2)=O)c(F)c1F 33341,C(=O)(CC(C(F)F)NC(c1conc1C)=O)N1CC(F)(CC)C1 33342,N1(C(c2cncc(OC)n2)=O)CC(C(=O)NCC(O)C(C)(C)C)CC(C)C1 33343,N1(C(CCc2ncc(C)[nH]2)=O)CC(NC(=O)C=CC=CCO)C(C)C1 33344,N1(C(c2cc(C)[nH]c2C)=O)C2CCC1CN(C(c1cccc(C3CC3)n1)=O)C2 33345,CC1=C(C)CC(C(=O)NC2CCCC2CC(=O)NOCC(N)=O)CC1 33346,N1(C(C(C2CCOC2)NC(c2nc(CCC)oc2)=O)=O)CCC12CCCC2 33347,c1(C(=O)NC2CC(NC(c3coc(Br)n3)=O)C2)ccc(-n2ccnc2)cc1 33348,c1(COCC)nc(C(=O)N(C(CNC(c2ccc(Cl)o2)=O)C2CC2)C)cs1 33349,c1(CCNCC(C)CS(C)=O)c[nH]c2cccc(Br)c12 33350,Cc1ncnc(C(N2CCC(NC(C3CC(F)(CO)C3)=O)CC2C)=O)c1C 33351,C(C(O)CC(=O)O)ONC(c1cc(-c2ccc(F)cn2)on1)=O 33352,C1(C(=O)NCCn2c(C)cnn2)CCC(C)(C)N(C(=O)COCCCN(C)C)C1 33353,C1(O)(C(C)NC(CC=C(C)C)=O)CCN(C(=O)CCC(=O)c2ccc[nH]2)C1 33354,c1(C(N2C3C(NC(c4c(Cl)ccc(SC)c4)=O)C(C3)C2)=O)c(N)ccc(F)c1C 33355,C1(C(=O)NC(C)CNC(c2nc(C(C)(F)F)cs2)=O)CCC2C(C1)C2(F)F 33356,C12(NC(CNC(C)=O)=O)CN(C(C3(Br)CC3)=O)CC1CS(=O)(=O)C2 33357,C1(NC(c2c(OC)noc2C)=O)CC2CC1CN(C(c1ccccn1)=O)C2 33358,C1(NC(Cn2c(C)nnn2)=O)CC2CC(C1)N(C(=O)C(C)OC1CCCCC1)C2 33359,C(=O)(C1=CCOCC1)NCCCNC(=O)CC1CC(C(F)F)C1.C1(N)CC(=C2CCC2)C1 33360,C1(CN(C(C2CC(N(C)C)C2)=O)CC)CCCN(C(c2cscc2C)=O)C1 33361,C1(CC(=O)NCC2(CNC(c3ncc(C)cn3)=O)CCCC2)(OC)CCOCC1 33362,C(=O)(CCCC(C)NC(=O)CC(C(C)C)OC)NCC(C)OCC=C 33363,Cc1ccc(C=CC(N2CC(C3(NC(c4ccc(F)s4)=O)CC3)C2)=O)cn1 33364,N1(C(c2cnn(C)c2)C)CCC2(CC1)CC(CNS(=O)(=O)c1ccncc1)C2 33365,Cc1cn2cc(C(=O)NC(CNC(=O)CC3CC=CCN3C)CO)cc(F)c2n1 33366,c1(C(=O)NCCC2(NC(c3ccc(O)cc3)=O)CCCC2)cnc2ccnn2c1 33367,C(=O)(CC(O)CC(C)C)N1C2C(NC(c3ccc(OC)c(C4CC4)c3)=O)C(C2)C1 33368,C1(C(=O)NC(Cn2cc(COC)nn2)C)(NC(=O)CC(C)COC)CCCOC1 33369,C1(CC=C)(NC(C2CC(N(C)C)C2)=O)CN(C(c2cc(C3CC3)on2)=O)C1 33370,C1(C(c2nnnn2C)NCc2ccc(OCC(F)(F)F)nc2)(CC)CCCCO1 33371,Cc1cc(C(=O)NC2CC(CCC(=O)NCC(F)(F)CO)C2)n(C)n1 33372,C1(C(=O)NC(CNC(c2cccc(SCC)c2)=O)CO)NC(=O)OC1(C)C 33373,CCC(C)C(C(=O)NC(CCO)CC(C)C)NC(=O)Cc1c(C)cnn1C 33374,N1(C(C(CC)NC(N)=O)=O)CCN(C(=O)CC2(C#N)CC2)C(C2CCCCC2)C1 33375,C(N=c1cc(C(C)(C)C)nc[nH]1)C1CN(C(c2cc(C)oc2)=O)CC1(C)C 33376,c1(C(C)C)ncc(C(c2nnnn2CC(F)F)NCC2CCCCC2)[nH]1 33377,N1(C(CCCOCC=C)=O)CCCC(O)(CNC(C23CC2COC3(C)C)=O)C1 33378,c1(C(=O)NCCCN(C(=O)CCCl)CC)cc(Br)c(OC)s1 33379,N1(C(CC(C)F)=O)CCC(NC(=O)COc2cccc(F)n2)C(CO)C1 33380,c1(C(N2CC(Cn3cc(CC=C)nn3)OCC2)=O)nccc2cc(Br)ccc12 33381,CC1=C(C(=O)NC(C)CC2CCN(C(C3(C)CCCO3)=O)CC2)C(C)(C)CCC1 33382,c1(CC(c2ccccn2)NC(C(NS(N)(=O)=O)C2CC2)=O)ccc(Cl)cc1 33383,C(=O)(CC(C)C(F)F)NC(C)C(CO)NC(c1cnc(C(C)(C)C)s1)=O 33384,Cc1ccc2c(C(=O)NCC(C)CNC(=O)C(C(C)C)C3CCC3)n[nH]c2c1 33385,c1(CN(CCOCCN(C(Cc2cc(C)no2)=O)C)C)ccc(I)c(O)c1 33386,C(CC(C(=O)NC1(C(=O)NC2CCCC2(C)C)CC1(C)C)OC)OC 33387,C(C1CCCc2cccnc21)c1n(-c2c(OC)cccc2)nc(-c2cc[nH]n2)n1 33388,c1(N(C(C(n2c(C)nnn2)c2ccccc2)=O)C)cc(F)cc(Cl)c1 33389,N1(C(CCCCCNC(C(CC)COC)=O)=O)CCn2ccnc2C1 33390,n1(CC(=O)NCC2COCC2NC(=O)CCCC(F)F)cc([N+](=O)[O-])ccc1=O 33391,C1(C(=O)NC(C)CC(C)NC(c2sccc2F)=O)(Cc2cnn[nH]2)CCOCC1 33392,C12(C(=O)Nc3c(CCC)cccc3)CC(CO)(CN1C(=O)CSc1nc[nH]n1)C2 33393,c1(C(N2C3CN(C(C=C(C)C4CC4)=O)C(C3)C2)=O)cc2scc(C)c2[nH]1 33394,C1(CC=C)(NC(=O)C(CC)OC)CCCN(C(c2ccc(C(C)=O)[nH]2)=O)C1 33395,CC(C)C#CC(=O)NC12CC1CN(C(c1ncncc1Br)=O)C2 33396,c1(C(=O)NC(C)CN(C(=O)Cn2cnnn2)C)ccccc1-c1ncc[nH]1 33397,N1(C(C(C)=C(CC)C)=O)CCCC2C1CCN2C(=O)C(C(C)(C)C)NC(N)=O 33398,N#Cc1cnc(CN2CC2)cc1N1CCC(O)(C(N)=O)CC1 33399,C#CCCCC(C)C(=O)NC1CCCCN(C(c2ccc3nccn3c2)=O)C1 33400,C1(C)(C(=O)NCC2(O)CN(C(c3c(OC)ccc(F)c3)=O)C2)CCC(C)=C(C)C1 33401,CCC(CNC(=O)C(C)=O)NC(=O)COCC1CCOC1 33402,c1(NCC23CCC(NC(=O)OC(C)(C)C)(CC2)CC3)cc(CO)ccc1[N+](=O)[O-] 33403,c1(C(CNC(C2(NC(c3cc(Cl)no3)=O)CCCC2)=O)O)cccnc1 33404,c1(C(N(CC(=O)NCC2C(OC)CC2)CC2CC2)=O)ccnn1C(F)F 33405,c1(OC)cc(F)c(C(=O)NC2COCC2NC(=O)C(c2ccnn2C)O)c(F)c1 33406,N1(C(c2cccn(C)c2=O)=O)CC2CN(C(c3cnns3)=O)CC(F)(F)C2C1 33407,CC1CCCCN1CC(=O)N(C(=O)COc1ccc(C(N)=O)cc1)C1CC1 33408,c1(C(C)C)nn(C)c(NC(=O)CC2CCCC(NC(c3cccnc3)=O)C2)c1Cl 33409,c1(OC)cc(Cl)c(Cl)cc1C(=O)NCCC(C)NC(C1C=CCC1)=O 33410,C1(NC(COC(CC)(C)C)=O)CCC2(CC2)N1C(=O)CN(C(=O)COC)C 33411,C1(C)(N(C)C)CCN(C(C2CC(=O)CN2C(C2CN(C(N)=O)C2)=O)=O)C1 33412,C1(C(N2C(CNC(=O)C#CC(C)C)CC(OC)C2)=O)Cc2ccc(C)cc2S1 33413,c1(C(=O)NC2C(NC(c3[nH]n(C)c(=O)n3)=O)C2)c[nH]c2c(Cl)cccc12 33414,C=C(Cl)C(C)(C)C(=O)NCC(O)CCNC(C1CC1CCC)=O 33415,C1(CC)CCC(C(=O)N(C(C)CCNC(=O)C=CC2(C)COC2)C)O1 33416,c1(C(C)C)c[nH]cc1C(=O)NCC(C)(C)NC(c1ccncc1)=O 33417,CC1SCCCC1(c1nnnn1CCOC)NCC1CCN(C2CC2)C1.C1(CC)CC1 33418,C(=O)(C(C)(C)OC)NC1CC(C(C)NC(C(C2CC2)OCC)=O)C1 33419,CC1=NS(=O)(=O)NC=C1C(=O)N1CC(CCNC(C2CCCC3CCCN23)=O)C1 33420,c1(C(N2C(C(=O)NCC3(O)CC(C)(C)C3)CSCC2)=O)cc([N+](=O)[O-])c[nH]1 33421,C12(C(=O)NCC(CCNC(C=C(CCC)CCC)=O)O)CC1CCC2(F)F 33422,Nc1nc(C(=O)NCC2(O)CN(C(C3CCC4CCC34)=O)C2)cnc1Br 33423,C1(NC(c2cc(F)c(F)c(F)c2)=O)CC1C1CCCN(C(c2coc(O)n2)=O)C1 33424,C1(NC(=O)CCc2cc(F)ccc2Br)CN(C(C2(F)CC2)=O)CC(F)(F)C1 33425,N1(C(C(C(C)C)C#N)=O)CCN(C(=O)CNC(=O)C(F)(F)F)CC(O)C1 33426,CC1CN(C(=O)CCc2cocn2)CCC1NC(=O)C(c1cnn(C)c1)C 33427,c1(CC(N2CC(CC(=O)Nc3cc(Cl)ncc3Cl)C2)=O)ccc2c(c1)CCO2 33428,c1(C(N2CC(N(C)C(c3cc(F)cnc3O)=O)C(F)C2)=O)c(F)ccc(F)c1F 33429,c1(C(=O)NCC(CC)NC(=O)C=CC2C(C)C2(Cl)Cl)n[nH]c2c1CCCC2 33430,c1(CC)nnc(C)cc1C(=O)NCC1CN(C(c2cnc3n2CCC3)=O)CCO1 33431,C(=O)(C1COc2ccc(Cl)cc21)NC1C(CNC(c2c(CC)occ2)=O)CCC1 33432,N1(C(C2CCC(CNC(C3CC4CCC3O4)=O)CC2)=O)CCC(O)C(F)C1 33433,C1(C(=O)NCCC2CCCN2C)(NC(C(C=C)O)=O)CCCCC1 33434,N1(C(c2c(OC)cccc2F)=O)CCc2ccccc2C(NC(=O)C(C)(F)F)C1 33435,c1(C(=O)NC(c2ccc(Cl)cc2)CNC(C(C)O)=O)cnc(O)cc1C(F)(F)F 33436,C(=O)(C1c2c[nH]nc2CN1C(=O)CC1CCOC1=O)NCc1c(C)cc(C)nc1 33437,C1(CC(=O)N(CCCNC(c2c(C)cncc2)=O)C)CC2CCC1CC2 33438,c1(N(C)Cc2c(C)ccc(Cl)c2)nc2c(c(=NCCC3CC3)[nH]1)SCC2 33439,CCC(C)C(COC)N=c1[nH]c(=N)[nH]c(=NCCC(C)(C)N(C)C)[nH]1 33440,N1(C(Cc2ccn(C)n2)=O)CCCC(C)(C)C1CNC(=O)Cc1ccsn1 33441,CC(C)(C)CCC(=O)NCCCC1CCCCN1C(C1CCC2(CCC2)C1)=O 33442,c1(C(=O)OCc2cnc(OC)c(F)c2)c(Cl)cccc1[N+](=O)[O-] 33443,Cn1ccnc1C(=O)NC1(C2CCCN2C(=O)CCSCc2nccn2C)CC1 33444,C1(CNC(CCc2ncc(C)[nH]2)=O)CC(NC(c2sc(C)cc2Cl)=O)C1(C)C 33445,n1(C(C(=O)N(CCC(=O)NCC2(C#C)CC2)C)C)ccc(C)n1 33446,C1(CC(=O)NCCCC(=O)OC)CCCCN1C(=O)C(C1CCCCC1)=O 33447,C1(NC(C(C(C)C)SCC)=O)CC2(CCN(C(C3CCCN3N=O)=O)C2)C1 33448,Cc1nc(C(=O)NC2CC(NC(=O)CC3CCC(=O)NC3=O)C2)c(C)n1C 33449,C1(NC(CONC(C(C)N(C(C)=O)C)=O)=O)C2CCCC1COC2 33450,C(=O)(C(O)CC(C)(C)C)N(CCCNC(c1c(OC)c(Cl)c(Cl)s1)=O)CCO 33451,C1(CC)C(NC(=O)C(c2cn(C)nc2C)C)CCN1C(=O)C=CC1CCC1 33452,Cc1nn(CC(=O)NC2CC2NC(C2(C)CC(C)(C)C2)=O)c(C)c1Cl 33453,c1(C(=O)NCC2N(C(c3ccn(C)n3)=O)CC=C2)cc2cc(Cl)cnc2[nH]1 33454,c1(CC(=O)NCC(C)(O)CNC(=O)CCc2cnc[nH]2)c(F)cccc1F 33455,C1(C(N2CC3C(NC(C4CC5COCC5C4)=O)(C3)C2)=O)CC2(C1)CC(F)(F)C2 33456,c1(C2C(C(=O)NCC#CCNC(C3C(Br)(C(=O)OCC)C3)=O)C2)cccnc1 33457,C1(NC(CCC2(C)CN(C(C3CC(=O)C3(C)C)=O)C2)=O)CCCC2(C1)N=N2 33458,N1(CCc2cn(CC)nc2)CC(=O)N(Cc2c[nH]nc2C2CCC2)C1=O 33459,C(=O)(CCCC(=O)NCCC1(NC(=O)C(C)NC(=O)CO)CCCC1)NCC 33460,C1(NC(CCSCC)=O)CC(NC(c2ccc(OC)cc2C(F)F)=O)C12CCC2 33461,c1(CCC)nc(C(=O)N(CCCCN(C)C(C2(C)CCC2)=O)C)cs1 33462,c1(C(=O)NCCCN(C(=O)Cc2nc[nH]n2)CC)cc2ncccc2s1 33463,c1(OC)cccc(NC(C2COCC2NC(=O)CCc2cccn2C)=O)c1 33464,C1(CC(=O)N(C2CC(C#N)C2)CC(=O)NCC(C#C)OC)CCOC1(C)C 33465,c12ccc(cc1)C(=O)NCCc1cc(no1)C(C)ONCC(=O)N(C)C2.C(C)(C)OC 33466,C1(CC)C(C(=O)NCCN2CCNC(=O)C2)CCN1C(=O)C(F)C1CCCC1 33467,C(=O)(CCCN=[N+]=[N-])N1C2(C(=O)NC3CN(CCC)C3)CC2CC1 33468,C1(C(N2C3(CN(C(C4CCOCC4)=O)C3)CC2)=O)CC2CC(O)C(C1)C2 33469,C(CCCCCN(C(=O)COCC(F)F)C)NC(C(CC)NC(C)=O)=O 33470,CCCCC(CC)C(=O)N1CCC(=CCNC(C2CC3CC3C2)=O)CC1 33471,N1(C(CC(CC#C)NC(C2CCCCC2(C)C)=O)=O)CC(=O)NC2(CC2)C1 33472,N1(C(CCc2cccc(C)c2)=O)CCN(C(=O)CCc2ccncc2)C2CCC12 33473,c1(C(=O)NC2CN(C(C(CO)NC(C(C)C)=O)=O)C2)ccc2c(c1)CCN2C 33474,C1(O)(CC(=O)NCCSC)CCN(Cc2ccc(F)c(OC)c2)CC1 33475,C(=O)(CC(C)(C(F)F)N(C)C)NC(CN(C(c1ccc(C)cn1)=O)C)C 33476,Cc1cc(CC(N2CCCC2CNC(c2ccn(C)n2)=O)=O)ccc1Cl 33477,C1(C(=O)NC(C)(C)CNC(=O)C=CC2(C)COC2)CS(=O)(=O)CCO1 33478,c1(CC)cc(C)c(C(=O)NC2COC(C3CCNCC3)C2)o1 33479,CC1(N(C(=O)Cc2ccco2)CC2CC2)CCN(C(c2ccc(NC)cc2)=O)C1 33480,c1(SC(C(=O)NC(CNC(c2cc(CCC)on2)=O)C)C)ccc(F)cc1 33481,C1(C(=O)NC2CN(C(=O)Cn3cccn3)CC2O)SC2C=CC1CC2 33482,C(=O)(CC(C)(C(F)F)N(C)C)NC1C(O)CCN(C(CC=CC=C)=O)C1 33483,N1(C(C2N(C(C(C)n3cncn3)=O)CSC2)=O)CCCC1(C)CC1CCC1 33484,N1(C2CCN(C(CC=C)=O)C2)CCN(C(C2CC23CCOC3)=O)CC1=O 33485,C12(C(=O)Nc3cccc(C)c3)CCCN(c3ncc(F)cn3)CC1C2 33486,C1(CC#C)CN(C(=O)COC2CN(C(=O)CSC(C)C)C2)CCO1 33487,c1(N(CCN(C)CC)C)noc(-c2cnn(-c3cnccn3)n2)n1 33488,C(C(CC(F)(F)F)NC(=O)C1=NOC(C)C1)NC(C(NOC)=O)=O 33489,c1(CNC(c2nc(CC)oc2C)=O)ccc2c(c1)CN(C(=O)C(=O)N1CCCC1)C2 33490,N1(C(C(C2CCC2)OC)=O)CCC(N(C(=O)C=CC2CCCCC2)CCO)CC1 33491,c1(C(CNC(CC=CC)=O)NC(=O)Cn2nnc(=N)[nH]2)cccc(C(F)(F)F)c1 33492,N1(C(C2N(CC)CCOC2)=O)CCCCC(N(C(=O)Cc2ccccc2C)C)C1 33493,c1(N(C)Cc2ccno2)nc(N2CC3C(C2)C3(F)F)nc2c1CCC2 33494,c1(CC)cncc(C(=O)N(C)CCOCC2(C(=O)CN)CCCO2)n1.C1CC1 33495,C1(C(=O)NC(c2cnn(C)c2)CO)(OC)CCN(C(C2CC(O)CN2C)=O)C1 33496,C(=O)(C#CC1CCCO1)N(CCNC(c1c(CC)cccc1)=O)C(C)C 33497,N1(C(C(=O)NC2C(C(C)C)CCCC2)=O)CCOC2(CCS(=O)(=O)C2)C1 33498,Cc1cc(O)nnc1C(=O)NCC1(C)CCN(C(=O)CC2CCC(C)C2)CC1 33499,C1CC(OC)C(=O)N1.c1(CC)cc(C(=O)NCC(C)(C)OCCO)n(C)n1 33500,C1(NC(c2[nH]c(=NC)sc2)=O)CN(C(c2ccnnc2S)=O)C2(CCCCC2)C1 33501,C1(CNC(=O)C(c2ccc(Br)cc2)F)CC1C1CCNCC1 33502,C(CCS(=O)(=O)c1ccc(Cl)cc1)N1CC2C(C(=O)OCC)(CCC2)C1 33503,N1(C(CCCCN(C)C)=O)CCC2(CCCN2C(=O)Cc2cccs2)CC1 33504,N1(c2nc(C)c(Br)cn2)CC(NC(c2ncc(Cl)s2)=O)CC(C)(C)C1 33505,N1(C(c2c(OC)oc(C)n2)=O)CCC12CN(C(=O)CC1CC3CCC1O3)C2 33506,C(=O)(CCC(=O)C(C)(C)C)N1C(C(=O)NC2CC(N(C)C)C2)CC(F)(F)C1 33507,Cc1ccc(C)c(OCC(N2CC(O)(CNC(c3csc([N+](=O)[O-])c3)=O)C2)=O)c1 33508,C1(CNC(Cn2cc(C(C)O)nn2)=O)CN(C(=O)CCOC(F)F)CC1C 33509,Cc1ncc(C(F)(F)F)cc1C(=O)NC1CC(NC(=O)C=Cc2ccc[nH]2)C1 33510,c1(CNC(C2(NC(c3c(CC)ocn3)=O)CCC2)=O)oc(C)nc1C 33511,c1(C(=O)NCC2(NC(c3c(CC)nns3)=O)CCCC2)cc(C2CC2)nn1C 33512,c1(C(c2n(CC=C)nnn2)NC(C)(C)C(=O)NC)cc(C(=O)OC)cc(CC)c1 33513,CCC(C(=O)NC(CCSC)C(=O)NCC1(C#N)CCCCC1)C(F)(F)F 33514,N1(C(CC2(C)CC2)=O)CCN(C2CCN(C(=O)C=CC3CCC3)CC2)CC1 33515,Cc1nc(C(=O)NC2CC(CCC(=O)NC3(CN(C)C)CC3)C2)c(C)o1 33516,C1(CNC(=O)C=CCn2cncn2)CCC(CNC(=O)Cn2cnnc2)CC1 33517,Cc1nn(C2CCOCC2)cc1C(=O)NCC1(NC(=O)C=CS(C)=O)CCCC1 33518,CCCCCC(=O)NC12COC(CNC(C3CC3[N+](=O)[O-])=O)(C1)C2 33519,N1(C(C2(C)CCN(C)C2)=O)CCN(C(c2cc(Cl)c[nH]2)=O)CC(CO)C1 33520,c1(C(=O)NC(CO)C2CNC2)cc(S(=O)(=O)C(F)(F)F)ccc1F 33521,C(=O)(C(C)C(F)(F)F)NCCC1N(C(CCOc2cccc(C)c2)=O)CCSC1 33522,C1(NC(c2cc3cnccc3[nH]2)=O)CCCC12CN(C(c1ccnc(Cl)c1)=O)C2 33523,c1(C(=O)NC2(C)CCCN(C(c3cc(C)on3)=O)C2)cc2cnccc2o1 33524,c1(OC)c(C(=O)OC(C)C(C)n2ccnc2)oc2ccccc12 33525,C(CCCOC)(C(=O)N1CC(C(C)C)C1)NC(c1nn(CC)c(O)c1)=O 33526,c1(CN(C)CC2CCN(C(=O)Cn3nnnc3C(C)(C)C)C2)cc2cnccc2o1 33527,N(C(=NCCCCl)NCc1nc(-c2ccccc2Cl)n[nH]1)CCC1CC(=O)NC1 33528,C1(N(CC(=O)N(CC(C)C)CC)C)CCOC1 33529,N1(C(C(N2CCC(C)C2)=O)=O)CCC(O)(N(C(=O)C(c2ccccc2)F)C)CC1 33530,C1(CC(=O)NC2(c3cccc(Br)c3)CC(=O)C2)(C(=O)OC)CCCNC1=O 33531,c1(C(C)(C)OC)nc(=NC2CC(NC(=O)Cn3cc(C)cn3)C2)s[nH]1 33532,Cc1c(Cl)cc(C(=O)OCCCC(=O)OC(C)(C)C)cc1Br 33533,CCC(C(=O)N1CC(NC(c2csc(C)c2OC)=O)C1)C(C)C 33534,C1(CC)CN(C(=O)CC(C)C(C)C)CCN1C(C1CC(F)C1)=O 33535,C1(NC(CSc2ccc(OC)cc2)=O)CN(C(=O)Cc2csc(S)n2)C(C)(C)C1 33536,CCC(C(=O)N1CC(CN(C)C(c2cccc(NC(=O)C3CC3)c2)=O)C1)C(C)O 33537,C#CC1(NC(=O)CCCCN(C)C(c2coc(C(N)=O)c2)=O)CCCCC1 33538,C1(NC(c2ccccc2-c2nc[nH]n2)=O)CN(C(C2CC2(F)F)=O)CC1C(F)F 33539,C(=O)(C1=C(Cl)CCCC1)N1C(CNC(C2(COC)CCCO2)=O)CC(F)C1 33540,C1(NC(c2nc(C(C)NC(CC(C)C)=O)oc2)=O)CCN2CCC1C2 33541,C(CC(O)CCc1ccccc1)NC(c1n(CCOC)nnn1)c1cccnc1 33542,CCC(C)C(C(=O)NCC1COCCN1C)N(C(=O)CCC(C)OC)C 33543,N1(C(c2ccc(C(C)C)o2)=O)CC2CC(NC(=O)C(F)(F)C(C)O)C1C2 33544,C1(CNC(C(CCOC)C)=O)CCC2(CN(C(C3CCOC(C)C3)=O)C2)O1 33545,C(=O)(CCc1ccc[nH]1)NCCN(C(=O)CCOC1CCCC1)C 33546,CN=c1cc(C(=O)NC2CCC(CCNC(=O)Cn3nnc(=O)[nH]3)C2)cc[nH]1 33547,c1(N(C)C)ccc(C(=O)NC2CN(C(C3(C)CCC(=O)C3)=O)CC2F)cc1 33548,N1(C2CN(C(c3cnc(C)s3)=O)C2)CCN(C(c2cc(C(F)F)on2)=O)CC1=O 33549,C1(CNC(Cc2n(C)ccn2)=O)CN(C(C2(O)CCCCC2)=O)CCO1 33550,Cc1cc(C(N2C(CNc3ccc(C(N)=O)c(C)c3)CCC2)=O)cc(=O)o1 33551,CC(C)(CS(N)(=O)=O)C(=O)N1CCN(C(c2ccn(C3CC3)n2)=O)CC2(CC2)C1 33552,C(C(CC(C)C)C(=O)NCC1CN(C)CCN1C(c1ccc(=N)[nH]n1)=O)OC 33553,C=CC(C(=O)N(C1CCN(C(c2cnccn2)=O)C1)CC)NC(=O)OC(C)(C)C 33554,C(N=c1nnc(C)c(C)[nH]1)C1CN(C(c2ccc(C)c(F)c2)=O)CC1C 33555,N1(CC(COc2ccc(C)cc2)O)CCc2[nH]c3ccc(F)cc3c2C1 33556,N1(C(c2cc(C(N)=O)sc2)=O)CCN(C(=O)C(F)(F)C2(O)CCC2)CC1C1CC1 33557,c1(NCCC(=O)NC)nc(=NCC(C(C)C)N(C)C)[nH]c2c(C)nn(C)c12 33558,c1(CC(C(=O)NC(C)CN(C(=O)C=CC(F)(F)F)C)C)cccc(Br)c1 33559,C(CC(C)C(=O)N(C1CCN(C(C2(n3cc(Cl)cn3)CC2)=O)C1)CCO)=CC 33560,C1(C(=O)NCC(C)NC(c2cc(Cl)ncc2N)=O)CCc2cc(F)ccc2O1 33561,CC1CC(NC(=O)Cc2ccc(F)cc2)CN1C(=O)CC1CCS(=O)(=O)C1 33562,CCCC(CCCNC(c1cc(Br)nn1C)=O)NCc1ccccc1 33563,Cc1cccc(C)c1NC(=O)C(c1cc(Br)ncc1F)N1CCC(C(F)F)CC1 33564,C(=O)(CC(CC)CCC)NCC1CCCN(C(C(C#C)(C)C)=O)C1 33565,CC(C)CCC(F)C(=O)NC1CC1CNC(c1cc(C(N)=O)n(C)n1)=O 33566,c1(COCCC(=O)N(C2CCCN(C(CSC)=O)C2)C)nc2ccccc2s1 33567,Nc1nc(C(N2CC(NC(c3cnns3)=O)CC(O)C2)=O)cnc1Br 33568,C(=O)(C(C)(F)CCCC)NCCCCC(C)NC(C(C=C)(C)CC)=O 33569,c1(N2C(C)CC2CO)nc2ccsc2c(=NCc2ncc3c(n2)CCC3)[nH]1 33570,c1(C(N2CC3(CC3C(N3CC4C(CO)C4C3)=O)C2)=O)cccc(Cl)c1Cl 33571,c1(C(N(CC(CC)NC(C2(CF)CCC2)=O)C)=O)c(C)nc2sc(C)nn12 33572,C1(CNC(c2cc(COC)no2)=O)CCCCN(C(=O)C(c2cncn2C)O)C1 33573,CCCC(CC)C(=O)N1CC2C(CC(=O)NC3CCN(C(C)=O)CC3)C2C1 33574,N1(C(c2nc(CCC)sc2)=O)CC(CNC(=O)C=CC2CC2)C2CC12 33575,Cc1cccc(-c2cccnc2NCC(N2CCN(C)CC2)=O)c1C 33576,N1(C(CC(C)OC)=O)CCN(C2CCCN(C(C3CCCC(O)C3)=O)C2)CC1 33577,CC1(C)CC(C(N2CCC2C2CCCC2)=O)CCN1C(=O)Cc1cn[nH]c1 33578,C1(NC(C(C)CC(C)(C)C)=O)C2CC3CN(C(c4cc(F)ccc4F)=O)C1C3C2 33579,CC1CCN(C(=O)C(c2cnn(C)c2)NC(=O)C(F)F)CCS1 33580,c1(NC(C2C(C)CCCC2)=O)cnc2ccc(F)cc2c1 33581,CC1CCN(C(c2cc(O)nn2C)=O)C1CNC(c1ccc(C2(C)CC2)cc1)=O 33582,c1(C(C)(CO)N(C(=O)NCC2CCN(C)C2)Cc2ccco2)cccc(C(F)(F)F)c1 33583,c1(N2CCC(CCOC)C2)ncnc(NC(COC)CC(C)C)c1C 33584,C1(CNC(C(CCCOC)C)=O)CC2COCC2N1C(C1(C)CCCO1)=O 33585,c1(C(N2CCCC(C(CNC(CCCOC)=O)(C)O)C2)=O)cnc(C)c(N)c1 33586,c1(OC)cnc(C(=O)NC(C)C(N2CCC(N(C)C)(CO)C2)=O)cn1 33587,C1(C(=O)NC2COCCN(C(CN3CCC(C)(C)C3)=O)C2)CCCC2(CCC2)O1 33588,Cc1cc(F)cc(C)c1C(=O)NC1CCN(C(c2ccc(Cl)nc2N)=O)C1 33589,c1(SC2C(OC)CS(=O)(=O)C2)nc2ccc(Br)nc2[nH]1 33590,N1(C(c2cn(C)nc2)=O)CC=CC(NC(C2CCCC2(C)C)=O)C1 33591,Cc1cc(C(=O)NC(CNC(=O)CC2CC2c2ccccc2)C2CC2)on1 33592,c1(C(N(CC(CO)(CO)NC(CC2CCC(C)O2)=O)C)=O)n[nH]c2c1CCCC2 33593,C1(CNCC23C(CN(C(=O)Cc4cnc[nH]4)C2)C3)COc2ccccc2O1 33594,C#Cc1ccc(C(=O)NC2(COC)CCN(C(=O)C(C(C)C)NS(C)(=O)=O)C2)nc1 33595,C=CCCCC(=O)NCC(CC=C)NC(=O)C(=C1CCCCC1)F 33596,c1(C(N2CCC(C)(NC(=O)Cc3cccc(O)c3)C2)=O)oc2ccccc2c1Cl 33597,N1(C(c2nc(CC)oc2C)=O)CCC2CN(C(c3cn(C)nc3OC)=O)CC12 33598,C=C(C)CCC(=O)NCC(CO)NC(=O)CC(C)C 33599,C(=O)(C(C(C)O)NC(=O)Cc1cn[nH]c1)NCC1(C(C)C)CCCC1 33600,C(=O)(C1=CCCCO1)N1CCN(C2CCCN(C(CSC)=O)C2)CC1 33601,c1(C(=O)NC2C(C)N(C(=O)Cn3ncnn3)CC2)cc2c([nH]1)CCOC2 33602,CC(C)(CCC(=O)N(C1CCC1)C1CC1)NC(=O)CC1CC=CC1 33603,CCCCC(CCCC)C(=O)NC1(CNC(=O)C(O)CC(C)C)CCCC1 33604,Cc1nncc(C(N2CC=C(CNC(C3CCO3)=O)CC2)=O)c1C 33605,C(C)(CNC(C1CCNC1=O)=O)(CO)NC(CCC)=O 33606,C1(OC)CCCCCC1Nc1ccc(-c2ccc(C)nc2O)cn1 33607,c1(C(N2CCC(NC(C3N(CC)CCC3)=O)C2)=O)nc2ccc(C)cn2c1N 33608,C(CC(F)(F)CC(=O)NCCn1cc(Cl)c(C(F)(F)F)n1)NC(=O)OC(C)(C)C 33609,c1(-c2cc(C(=O)NC(c3c(OC)cccc3)CO)on2)ccc(C)c(C)c1 33610,C=CC(CC)CC(=O)N1CC(NC(C2CCCN(C)C2)=O)C1 33611,c12ccc(cc1)N(C)C(=O)C(=O)NC(C1CC1)C2.Cc1nnc(CCC2CC2)o1 33612,CC1(C(=O)NC2CC(CNC(=O)CCn3ccnc3)C2)CC(C#N)C1 33613,c1(OC)ccc(NCc2cc(C)c(-c3ccc(CO)cc3)s2)cc1C 33614,C1(N(C)C)(C(=O)NCC(O)CCNC(=O)CCC2CCC2)CCOCC1 33615,C1(C(N2CCC(C)(CN(C)C)C2)=O)CCCN(C(=O)Cn2ccnn2)CC1 33616,c1(C(=O)NC2(c3cn(C(C)C)nn3)CCOC2)cc(NC(C)C)ccn1 33617,C1(C2CCCC2)(NC(C2C(C)CCN2C(=O)C(C)c2cc[nH]n2)=O)CC1 33618,C(C(=O)NCc1cccs1)(C(C(C)C)OC)N1CCCC(C(=O)OC)C1 33619,C(=O)(C1=NOC2(C1)CN(C(C)=O)C2)NCC=C(C)C1CCN1C(=O)OC(C)(C)C 33620,c1(NC(c2ccoc2)C)ccc(S(=O)(=O)NC2CC3CCC(C2)S3)cc1F 33621,c1(C(N(CCCN(C(C(CSC)O)=O)C)C)=O)ccc2c(c1)CC(=O)NC2 33622,CN1CCN(C2CCN(C(=O)C(=O)Nc3nsnc3N3CCC3)C2)CC1.C(=O)O 33623,C1(NC(C2N(C)CCOC2)=O)CN(C(c2cccc(Cl)c2)=O)C2(CCC2)C1 33624,C1(CNC(C(C)Sc2nncn2C)=O)CCCC(NC(=O)CCn2cccn2)C1 33625,N1(CC)CC(C(N2CC3CC2C3NC(=O)CSc2n[nH]c(C)n2)=O)CCC1=O 33626,N1(CC)CCCCC1C(=O)N(C1CCN(C(=O)CCSc2ccccc2C)C1)C 33627,c1(C(=O)NCCC23C(CN(C(CCOCC)=O)C2)CC3)sc2ccccc2c1C 33628,c1(C(=O)NCC(C)CNC(=O)CCn2cc(Cl)cn2)ccc([N+](=O)[O-])c(O)c1 33629,c1(NCC2CN(C(CC3C(C)=NOC3=O)=O)C2)nc(C)c(C#N)cc1Cl 33630,c1(C(=O)NC(C)CNC(=O)COCCOc2cn[nH]c2)ccc2c(c1)CC(C)O2 33631,N1(CC)CC(C(=O)NC(C)CC2CN(C(C3CCCN3CC(C)C)=O)C2)CC1=O 33632,c1(CC(N2C(C)CC(CNC(c3cnc(O)s3)=O)CC2)=O)c[nH]c2cccnc12 33633,N1(C(c2nc(C)n(C)c2)=O)CCCC(NC(c2[nH]ncc2C#N)=O)CC1 33634,CCCC(CC)C(=O)NCc1cccc(C(=O)NCC2CCN(CC)CC2)n1 33635,N1(C(CC(C(C)C)C)=O)CCCC2(CCN(C(=O)Cn3cnc([N+](=O)[O-])n3)C2)C1 33636,N1(C(C(C)(C(C)C)OC)=O)CC(C2CCN(C(C3CC34CCCC4)=O)CC2)C1 33637,c1(Cn2cc(CS(CCC)(=O)=O)nn2)cc(C)ccc1S(N)(=O)=O 33638,CC(C)(C)C1=NOC(C)(C(=O)NC2CN(C(=O)CCCCC#N)CC3(CC3)C2)C1 33639,CC1CN(C(=O)CC#N)CC1CNC(=O)C(c1ccccc1F)(C)C 33640,CNS(=O)(=O)NCC(=O)NCC1(C(N)=O)CN(C(=O)CC2CC(C(F)F)C2)C1 33641,c1(NC(COC)=O)ccnc(C(N2CC(NC(C34CC(F)(C3)C4)=O)CC2C)=O)c1 33642,C1(CCC(=O)NC(CN(C(C(C)=C(CC)C)=O)C)CC)CCC(=O)NC1 33643,C1(C(=O)NCC2(COC)CN(C(C(C=C)C)=O)C2)CCC2(CCC2)C1 33644,C(=O)(C(O)CC(C)(C)C)N1CCC(N(C)C(c2cc(-n3cnnc3)ccn2)=O)C1 33645,N1(C(C2(CNC(c3cc(C)sn3)=O)CCC2)=O)CC(C)(C)OC(C)(C)C1 33646,Cc1cnc2c(C(=O)NCC(CO)NC(C3CC34CCCCC4)=O)cnn2c1 33647,C(CC(O)C(=O)N1CCN(C(=O)CCNC(c2ncccc2C)=O)CC1)SC 33648,c1(C(N2CC(O)(C(C)NC(C3CCCCC3)=O)C2)=O)ccc(N)o1 33649,CC1Cc2cccc(C(=O)N(C(CNc3ncc4ccnc-4[nH]3)C3CC3)C)c2O1 33650,c1(C(N2CCC(C(C)NC(CCc3scc(C)n3)=O)C2)=O)cncc2nc[nH]c12 33651,c1(NC)ccc(C(=O)NCc2cncc(C(=O)NC3(C)CC(O)C3)c2)cc1 33652,c1(CNC(N(C(C(=O)OCC)C)C)=O)ncncc1C 33653,C1(C(=O)NCC2CCCC2CF)(NC(=O)COC2CCCC2)CC(F)(F)C1 33654,S(=O)(=O)(c1cnn2ccc(NCC3CCCCC3O)nc12)NC(c1ccco1)C 33655,C(c1cccc(F)c1)=CC(=O)NCCCCCNC(Cc1cn(C)nn1)=O 33656,c1(C2C(NC(=O)NC(CCOC)CC(F)(F)F)C2)cc(C)ccc1C 33657,c1(C(=O)NC(CN(C(COCCCOC)=O)C)(C)C)cnc2ccccn2c1=O 33658,C1(O)(C(C)NC(=O)CC(C)c2ccco2)CCN(C(C2CC(=O)N2)=O)C1 33659,CCCC(CCCNC(=O)CC1COCC1(C)C)NC(c1cnc[nH]1)=O 33660,C1(NC(C(CC)CC)=O)CCC(C)N(C(=O)C(c2cccc(Br)c2)C)C1 33661,c1(OC)c(C(N2CCC2CNC(c2cc(C)c(C)cn2)=O)=O)cc(Cl)cc1Cl 33662,Cc1cccc(Br)c1C(C(=O)NC1CC1c1ccco1)NC(c1nn(C)cc1C)=O 33663,c1(C(=O)OC)ccc2c(c1)C1(CC1)CN2C(c1cnc2sccn2c1=O)=O 33664,Cc1cccc2c1OCCN(C(=O)C(C)(N)CC(C)C)C2 33665,CCCS(=O)(=O)C(C)C(=O)NCC1CC2(C1)CN(C(C1CC1(C)C)=O)C2 33666,C1(C(N2CCC(N(C(COCCC#C)=O)CCO)CC2)=O)CC2(C1)CC1(CC1)C2 33667,c1(C(=O)NC(CNC(c2cncc(CC)c2)=O)CO)cc(C(C)C)ccc1N 33668,c1(C(N2CCC(C(F)(F)F)C2)C(=O)NCCCC2CC2)ncc(Cl)s1 33669,N1(C(C2CCCC(OC)C2)=O)CCC(F)(CNC(C2CCC=CCC2)=O)CC1 33670,CC(CC(F)(F)F)C(=O)NCCNC(C1CCCN(C(=O)C#CC2CCC2)C1)=O 33671,C=CC1(C(=O)NCC(C2CC2)SC)CCN(C(C2CC(=C3CC3)C2)=O)C1 33672,C1(NC(COCC#C)=O)CCCCCC1NC(c1ccc(N)c(SCCC)c1)=O 33673,C1(COC)(CNC(=O)COC(C)C)CCN(C(=O)CNc2ccncc2)CC1 33674,c1(C(=O)NC(c2cccnc2)C(=O)NCC2(N(C)C)CC2)cnc(C2CC2)o1 33675,Cc1ncc(C(=O)NCC(C)(C)NC(=O)C(Cc2ccsc2)NC=O)[nH]1 33676,c1(NC)ccc(C(F)(F)F)cc1C(=O)NC1CN(C(C2COC(=O)N2)=O)C1 33677,C(=O)(N=c1cc2ccccn2[nH]1)C1(C)C=CCN1C(c1ccccn1)=O 33678,c1(NC(C)C)ccc(C(=O)N(C2CCN(C(c3coc(Br)n3)=O)CC2)C)cn1 33679,c1(C(=O)NCCC(C)N(C(=O)CCC#N)C)cnoc1C1CCOCC1 33680,N1(C(CSC(C)(C)C)=O)CCN(C(=O)C(F)C(C)(C)O)CC1c1cn[nH]c1 33681,Cc1cc(C(=O)NCC(C)(CO)NC(=O)CCc2cc(Cl)no2)ccc1Cl 33682,C1(CCNC(=O)CCCN(C)C)(OC)CN(C(=O)CCc2nc(C)no2)C1 33683,c1(C(N(C)CC2(O)CCN(C(CC3(C=C)CC3)=O)C2)=O)c(OC)ncnc1C 33684,c1(C(c2ccoc2)O)nn2c(c1CNCC(O)COc1ccc(Cl)cc1)CCC2 33685,c1(C(=O)NCCN(C)C(C2(C(F)F)CCOCC2)=O)c(F)cncc1Cl 33686,CN1C(=O)CCC(c2nc(C3(c4ccccc4F)CC3)no2)C1c1ccccc1F 33687,N1(C(CSCCCC)=O)CCC(C)(CCNC(C2CC(C)C2)=O)C1 33688,Cc1nn(C)c(C)c1C(N1CC2CC(C1)C2NC(=O)C(C)N1CCC1)=O 33689,C1(CCNC(c2cc(C)on2)=O)CCN(C(C2CCCN2C=O)=O)CC1(F)F 33690,C1(C(C)=O)C(C(=O)NC2CC2NC(c2cc(C)co2)=O)C1(C)C 33691,N1(C(c2cnc(CC)o2)=O)CC(C(N2CCCC(C)(F)C2)=O)C2(CC2)C1 33692,Cc1ccnc(C)c1CNC(=O)C(C1CCOC1)NC(c1nccs1)=O 33693,C1(CC)CN(C(C2(NC(=O)CC(C)CN(C)C)CCOCC2)=O)CC(=O)N1 33694,c1(SCC)cccnc1C(N1CCOC(CN(C)C(C2CCC(=O)O2)=O)C1)=O 33695,S(=O)(=O)(c1cccnc1N1CCC(OC2CCCOC2c2cn(C)cn2)C1)NC 33696,CCCCC(F)C(=O)N(C1CC(NC(c2c[nH]c(=N)nc2CC)=O)C1)C 33697,CCC(C)(C)C(=O)C(=O)N1CC(F)(C(=O)NC2(C(C)O)CC2)C1 33698,c1(C(=O)NC2C(CNC(c3c(CC)c[nH]c3)=O)CCCC2)cn(C)c(=O)cn1 33699,c1(C(N(C(CNC(C2CCC(=O)O2)=O)C2CC2)C)=O)cc2ccccn2n1 33700,C1(C)(C(=O)NCC(CCOC)NC(=O)C=CC2CCC2)CC(=O)N(C)C1 33701,c1(CCC)cccc(NC(c2sc(C)cc2C)=O)c1.C12COC(C1)CNC2=O 33702,C(=O)(C(CCN(C)C)NC(C1COCC(C)O1)=O)NC(C#C)C(C)C 33703,C1(OC)CCCC(CNC(=O)C=CCN(C(=O)Cn2cncn2)C)C1 33704,C1(C2CCCC2)(C(=O)NC2C3(CCN(C(c4cc(Cl)nnc4O)=O)C3)C2)CCC1 33705,C(=O)(C(O)C(F)(F)F)N1CC(O)(CNC(c2ccc(CC)s2)=O)C1 33706,CC1COCCCN1C(C1CN(C(C2CCCC2)=O)C(C)(C)C1)=O 33707,Nc1cnc(Cl)c(C(N2CCOCC(NC(c3ccc(F)s3)=O)C2)=O)c1 33708,c1(C(CNC(c2ncn(CC)c2)=O)NC(=O)CC(C)SC)cccc(OC)c1 33709,c1(CNC(C2CCN(C(C3CCCN3C=O)=O)CC2)C)cc(O)c(O)c(O)c1 33710,c1(C(N(C2CCC(NC(C3CCC(F)C3)=O)CC2)C)=O)cc2cnn(C)c2s1 33711,C1(CCC(=O)N(CC(F)F)C2CC2)(NC(C=CC(C)C)=O)CCC1 33712,C1(CN2CCC(C(=O)NCCC3(O)CCCOC3)(CC)C2)CCC(C)(C)CC1 33713,c1(CC(=O)NCC(CC)(C)NC(=O)CCC2CC(F)(F)C2)ccc(Cl)c(C)c1 33714,N1(C(CCC(=C)C)=O)CCN(C(=O)C(C)CCC)C(c2cn[nH]c2)C1 33715,c1(C(N2CC(CC)C(c3cnn(C)c3)C2)=O)cnc(CC(=O)O)[nH]c1=N 33716,c1(C(=O)NCCC2CN(C(=O)C=CCO)C2)cccc2cncn12 33717,C#Cc1cc(C(=O)NCCNC(C2CC[Si](C)(C)CC2)=O)cc(F)c1 33718,N(C(=NCC(C(C)C)OC1CCCC1)NC(C)C1CC1)Cc1cccc(C)n1 33719,C1(c2nn(C(CC)CC)c(-c3nc(C)c(C)s3)n2)CCC(F)(F)CC1 33720,c1(OC)sc(C(=O)NCC(C)NC(=O)CNC(=O)CNC(C)=O)nc1C 33721,c1(Nc2ccc(OC)cc2CC#N)nc(C)nc2scc(SC)c12 33722,C1(NC(CSC(C)C)=O)COCCC1NC(c1cccnc1-n1nccn1)=O 33723,c1(C(=O)NCCNC(C2C(NC(=O)OC(C)(C)C)CC2)=O)ccc(Cl)o1 33724,C=C1CCN(C(=O)C(COC)OC)C(C(=O)NCc2ccc(C)c(C)n2)C1 33725,Cc1ccc(C(=O)NC2(CNC(c3cc(C(=O)O)sc3C)=O)CC2)c(O)n1 33726,c1(CC)cccc(CC)c1C(N1CC(NC(=O)C(C)C2CC2)CC(CC)C1)=O 33727,c1(C(N2CCC(OCCC(N)=O)CC2)C(=O)NCC(C)C)cnc(Br)n1C 33728,N1(C(c2c(CCNC(C3CNC(=O)C3)=O)n[nH]c2)=O)CC2(CNC(=O)OC2)C1 33729,c1(CC(=O)NCC(Cn2cc(CCO)nn2)OC)cc(Cl)cc2c1OCC2 33730,CC1(C)OCCOC1C(=O)NCC1(O)CN(C(C2(F)CC=CC2)=O)C1 33731,N1(C(c2ccc(C)[nH]2)=O)CCN(C)C(CNC(=O)C(c2cccnc2)O)C1 33732,N1(C(C(c2ccncc2)C)=O)CC(CNC(=O)CC(C)(C)C)CCC1C 33733,C1(CNC(C(C(C)C)C)=O)CN(C(c2cnc(Cl)c(N)c2)=O)C2COCC2O1 33734,C1(C)(OC)CCCN(C(=O)C(C)(CNC(c2ncoc2C)=O)CC)C1 33735,CN1CCOCC1C(=O)N(C)Cc1ccc(CNC(=O)CN(C)C2CC2)cc1 33736,CCC(CC(C)C)C(=O)NCCN(c1ncc([N+](=O)[O-])cn1)CCOC 33737,N1(C(C(C(CC)C)OC)=O)CC2CCC(C1)N2C(=O)C(N1CCN(C)CC1)(C)C 33738,c1(C(N2CC(Cn3cc(CCNC(C)=O)nn3)C2)=O)cc(F)cnc1O 33739,c1(C(=O)NC(CC)CNC(=O)CN2CCCC2C)ccc2cnoc2c1 33740,C1(CC(C)(F)CN(C(=O)C2=COCC2)CCO)CCC(C2CCC2)CC1 33741,C1(CC(=O)NCC(CNC(=O)CCc2nccs2)F)CCCCC12CC2 33742,N1(C(C(CC)c2ccccc2)=O)CC(CNC(=O)CC(C)(F)F)C2(CC2)C1 33743,c1(CNC(C2C(CNC(C(CN(C)C)N(C)C)=O)C2(C)C)=O)cccc(O)c1 33744,c1(SC)cc(C)c(C(N2CCC(CF)(NC(c3cnsc3)=O)C2)=O)s1 33745,c1(CNC(C2(CC(C)C)CC2)=O)ccc(CN(C)C(C2C(F)(F)C23CC3)=O)cc1 33746,c1(C(=O)NC23CC(CN=c4c(C)cnc[nH]4)(C2)OC3C)cc(C#N)c(N)cc1O 33747,CC1CCN(C(C2CCCC2)=O)C1C(=O)NCCC1CCC(C)(C)O1 33748,N1(C(c2ccc(C)cc2)C)CCC(NC(=O)C(C)NC(c2cccs2)=O)C(C)C1 33749,C1(COC)(CNC(=O)Cc2c[nH]nc2O)CCCN1C(C1CNC(=O)N1)=O 33750,c1(C(N2C(CCN(C(=O)Cn3nccn3)C)CCCC2)=O)c[nH]c2nccc-2c1 33751,c1(OC)ccc(O)c(CNCCCc2ncn(C)n2)c1 33752,Cc1c(C(=O)NCC2CCN(C(c3cnc(Cl)[nH]3)=O)C(C)C2)nc2sccn12 33753,C(CCC(C)N(C(=O)C(N1CCOC1=O)C)CC)NC(C(C)n1ncc(C)c1)=O 33754,Cc1nnc2n1C(C(=O)N1CC(Cc3cn(CC4CCOC4)nn3)C1)CC2 33755,N#Cc1cnn(CC(=O)OCC(=O)Nc2ccc(Cl)cc2)c1 33756,FCCN=C(NCc1cn(CC(F)(F)F)cn1)N1CCCC2(CCCNC2=O)C1 33757,C1(CNC(C2N(C)C(=O)NC2)=O)C(O)C(O)CN1C(c1ccc(F)cc1)=O 33758,c1(CC(N2CC3(CCN3C(c3ccc[nH]3)=O)C2)=O)cc(Cl)cc(Cl)c1 33759,O=C(C1=CCCC1)N1CCCC1CCCNC(C12CC(CN1C1CC1)C2)=O 33760,C1(C(N2CCC(NC(C3CC=CC3)=O)(CO)C2)=O)CN2CCN1CC2 33761,C=CCCC(CC(C)C)C(=O)NC(C)CN(C(=O)COc1cccc(C)c1C)C 33762,N1(C(c2ncc(OCC)nc2)=O)CCCC(N(C)C(c2csc(C)c2N)=O)CC1 33763,Cc1cccc(CC(N2C(CNC(=O)C3=NOC(C)C3)CCC23CCC3)=O)c1F 33764,c1(CN2CCC(N(C(C=CC(C)C)=O)C)CC2)ccc([N+](=O)[O-])cc1O 33765,C(CCCC(=O)NC1(C)CCN(C(=O)C2=COCC2)C1)OCC 33766,c1(C(N(CC(C)NC(CC(=C)Br)=O)C)=O)ncccc1S(=O)(=O)CC 33767,N1(C(C2(CCN(C)C)CC2)=O)CCC2(CC1)CC2NC(=O)C(c1cccnc1)O 33768,c1(NCC2C(C)(C)CN(C(=O)CCc3cccs3)C2)nc2c(F)cc(Cl)cc2s1 33769,N1(C(c2c(CC)con2)=O)CCC(NC(=O)CCCN(C)C)C1c1ccccc1 33770,Cc1ccc(C#N)cc1NC(=O)C(C)N(C(=O)CSc1nc[nH]n1)C1CC1 33771,C(CC(C)C(=O)NCC1CC1NC(c1ccnnc1C)=O)=CCC 33772,Cc1cc(Cl)c(Cl)cc1C(=O)NCCC1CCCCN1C(C1CC12CCCC2)=O 33773,N1(C(c2cc(CC(C)C)[nH]n2)=O)CCCOC(CNC(=O)C=CC(N)=O)C1 33774,c1(NC)cc(Cl)ccc1C(=O)NCC1(CO)CCN(C(=O)CNC(C)=O)C1 33775,C1(CC)CNC(=O)CN1C(C1CCC(NC(=O)COC2CC(=O)NC2=O)CC1)=O 33776,C(CC(CC)C(=O)N1C(CC(=O)NCc2cn(C)nc2OC)C2CCCC12)=CC 33777,C1(CC(N2CCCC(O)(CNC(COCCC)=O)C2)=O)CC2CCC(C1)N2C 33778,N1(C(C2(OC)CC2)=O)CC2(CCN(C(=O)Cc3nnc(C)o3)C2)C1 33779,C12(CNC(c3cncc(C(N)=O)c3)=O)CCCC1N(C(=O)C=CC1CC1)CCC2 33780,c1(OC)ccc(C(C)C(N2CC3CC3(CNC(=O)C(C)C3(O)CCC3)C2)=O)cc1 33781,O=C(C1=NOC2(CCN(C(c3c(F)ccc(F)c3F)=O)C2)C1)NCC1CCOC1 33782,C#CC1CCCCN1C(C1OCCC1NC(=O)CN(CC(C)(C)C)C)=O 33783,CCC(CC(=O)N1CCCC(CC)C1C(=O)NCc1c(C)noc1C)C(F)F 33784,C1(C(N(CC(CC)(C)OC)C)=O)(C(C)C)CCN(C(c2coc(C3CC3)n2)=O)C1 33785,C1(CC(N2CCC(NC(COCCN(C)C)=O)(CO)C2)=O)CC2CCC1CC2 33786,c1(C(N2CC(NC(CS(C)(=O)=O)=O)C(F)(F)C2)=O)ccc2nc(Br)sc2c1 33787,S(=O)(=O)(c1cc(C(N2CCN(C(=O)CSC(F)F)C(C3CC3)C2)=O)co1)N(C)C 33788,N1(C(C(C)SC(C)C)=O)CC2CC2(C(=O)NC2CC3CCC2O3)C1 33789,C1(NC(c2c(C)cc(F)cc2)=O)CC2CC(NC(=O)C(C)(C)C3CCC3)CC2C1 33790,c12[nH]c3ccccc3c1CC1(CC)COCC(CCCNC2=O)CNC1=O 33791,N1(C(CCCOCC)C(=O)NC(CC(C)C)C(=O)OC)CCC(S(N)(=O)=O)C1 33792,c1(OC)cc([N+](=O)[O-])cc(CN2CCC(NC(=O)CC(C)(C)O)C(F)C2)c1O 33793,C1(C)(N(C(=O)CO)C)CC(NC(=O)CC2(NC(=O)C(c3cccnc3)O)CC2)C1 33794,CCC(O)(CC)CCN=C(NCc1ccc(C(N)=O)o1)NC(C)CCC1CC1 33795,N1(C(C2(CC=C)CCCC2)=O)CCOCC(NC(=O)CSC2CCOC2=O)C1 33796,c1(C(=O)NCC2(O)CN(C(C3(C(=O)NC)CC3)=O)C2)cc(Cl)c(OC)cc1Cl 33797,C1(NC(c2nc(C(C)NC(C3C(C=C)OCC3)=O)oc2)=O)CCC2(CCC2)CC1 33798,c1(C(N(C(C)CNC(c2sccc2CN(C)C)=O)C)=O)ncc(Cl)nc1Cl 33799,Cc1c(I)c(NC(N2CCCC(OC(F)F)C2)=O)nn1C 33800,O=C(CCCS(=O)(=O)NCCC1(O)CCCOC1)Nc1ccccc1 33801,Cc1cc(C(=O)N(CCCNC(=O)CC(=O)NC2CC2)CC2CC2)ccc1O 33802,C(C)(C(CO)NC(c1ncoc1C(C)C)=O)NC(C(c1ccccc1)OC)=O 33803,c1(OC)cc(C(=O)NCC(C)NC(=O)C2CCSc3ccccc32)ccc1C#N 33804,c1(OCCCNC(C(=O)NCCCOC)C)c(C)ccc(C)c1C 33805,c1(C(N2CCN(C(C(CC)C)=O)C3C2CC3)=O)cnc2c(c1)CCC(=O)N2 33806,CC1CCN(C(=O)C=C(Cl)Cl)C1CNC(c1ccc(Sc2nc[nH]n2)o1)=O 33807,N1(C(c2onc(C)n2)=O)CC2CCCC1C2CNC(=O)C(C)(C)C(N)=O 33808,CC1CCC(c2cn(CCC3CCSC3)nn2)CC1 33809,c1(C(N(CC)CC2CCOC2)=O)n[nH]cc1CNC(=O)C(C)=C(C)C 33810,C(=O)(C(F)CC(C)(C)NC(=O)CCC1CCOCC1)N(C)Cc1nccs1 33811,Cc1ccc(C=CC(=O)NC(C)CCCc2cccnc2)cn1 33812,Cc1c(N)ccc(C(=O)NCCN(C(c2csc(Cl)n2)=O)CC2CC2)c1C 33813,N1(CC(N2CCCC(C(=O)OC)C2)=O)CC2CC1CN2C(c1ccnnc1C)=O 33814,N1(C(C(CCC)CC)=O)CC2(CNC(=O)C(F)OC(F)(F)F)CC1CCO2 33815,CC1CC(C(N2CCC(NC(c3coc(Cl)n3)=O)C(C)C2)=O)CC(=O)N1 33816,c1(NC(=O)Cn2cc(-c3ccc(OC(F)F)nc3)nn2)cncc(OC(F)F)c1 33817,C(c1ccc(OC)cn1)=CC(N1CCC(N(C(=O)CC2(C)CC2(Cl)Cl)CC)C1)=O 33818,CCCC(C(=O)N(CC(C)NC(C1(n2ccnc2)CCCC1)=O)C)C(C)C 33819,CCCC(C(=O)N(C)CCN(C(C1(OC)CCSC1)=O)C(C)C)C(C)C 33820,C1(NC(=O)CC2CSC2)CC(O)CN(C(c2cnn(-c3nccs3)c2)=O)C1 33821,C1(NC(C(CC)N(C(C(CCC)=CCC)=O)C)=O)CCCOC1(C)C 33822,N=c1nc(N2CCC(C3CC3)C2)[nH]c(=NCc2ccc3c(c2)CCCC3)[nH]1 33823,Cc1cc(C)c(C(=O)NC2CCN(C(c3cc(C(C)C)[nH]n3)=O)C2)c(=O)o1 33824,Cc1n[nH]c(C)c1C(C)C(=O)NCC1(CO)CCN(C(C2(C)CSC2)=O)C1 33825,C(CC(C)C)(C(=O)NC1CC(NC(c2c(C)cccc2C)=O)C1)NC(C)=O 33826,C1(NC(c2sc(CC)c(C)c2)=O)CC2CCC1N2C(=O)CSCC1CCCCO1 33827,C1(NC(Cn2ncc(C)c2)=O)CC2CCC1C(NC(=O)CC1CC=CCC1)C2 33828,C1(CC(=O)N(CCC(=O)NCC2CSCCO2)CC)CC2CCC1O2 33829,CCC(F)(F)CC(=O)N1CC2(CNC(c3nnn(C(C)(C)C)n3)=O)CCC1C2 33830,CCC(CC(=O)N1CCC1COC)NC(=O)CCc1ccccc1O 33831,c1(CC)ncc(Cl)c(C(=O)NC2(CN3CCN(C(=O)CC(C)O)CC3)CC2)n1 33832,C1(O)(C(C)NC(Cc2c(C)con2)=O)CCN(C(c2cnc(N(C)C)o2)=O)C1 33833,CC1(C)OC2CC(C(=O)NCC3CC3NC(=O)CC3(N(C)C)COC3)CC2O1 33834,C1(C(N(CCN(C)C)Cc2c(F)cccc2Cl)=O)C2(CCC2)C12CCC2 33835,c1(CNC(C2C(=C)C2)=O)cc2n(n1)CCN(C(=O)Cc1ccc(C3CC3)cc1)C2 33836,N1(C(c2c(C)ncn2C)C(=O)NCCSC)CC2CCCCC2C1C 33837,O=C1CCOC(C(=O)NCC(CC2CCCC2)C(=O)NCCCCn2ccnc2)C1 33838,c1(CC)nc(C)ncc1C(=O)NCC1(F)CCN(C(=O)CCC2CCCO2)CC1 33839,N1(C(C2CC(C)OC2)=O)C(C)CC2CN(C(C3CC(N(C)C)C3)=O)CC12 33840,N1(C(CC2CCN(C)C(=O)C2)=O)CC2CCC1CN2C(CC(C)(C)C#N)=O 33841,C1(NC(C23C(C)(C)C(CC2)CC3)=O)CCCC2CN(C(c3cc(Br)co3)=O)CC12 33842,C1(CC)CN(CC(c2ccc(CN)cc2OC)=O)C(C)CO1.c1(OC)ccccc1C 33843,Cc1nccc(C(=O)NC2(C(=O)NC3CNC(=O)OC3)CCC2)n1 33844,N12C(CCC13CC3)C(=O)N(CCCC(=O)OC)CC2=O.C(COC)OC 33845,C(=O)(CCCC(=O)N1CCOCC(CNC(=O)C(C)CC(F)F)C1)OCC 33846,C1(O)(C(N2CC(O)(CCNC(C3(C)CCC(C)C3)=O)C2)=O)CCCC(C)(C)C1 33847,CC(C)C(C)C(CNC(c1cnc[nH]1)=O)NC(C1CSC1)=O 33848,CC1OC(C)(C)OC1(C)CNC(N1CCN(c2cc(C3(C)CC3)no2)CC1)=O 33849,C(CC(N)=O)(C(=O)NCC1CCC2(CC1)CC2)NC(c1cccc(C)n1)=O 33850,Cc1cc(Cl)ccc1CC(N1CCC(NC(=O)CCNC(=O)C2CC2)C(F)C1)=O 33851,C#CCC(C)(C(=O)NC1CN(C)CC12CC2)NC(=O)CSCC(F)F 33852,c1(C(N(CCCNC(COCC)=O)C2CC2)=O)cnc2sc(C)c(C)n2c1=O 33853,c1(C(C(=O)OC)(F)F)ccc(NC(=O)Cc2ccccc2)cc1 33854,N1(C(C2=NOC(C)C2)=O)CCC2(CC1)CN(C(c1cn(C)cc1C(F)(F)F)=O)C2 33855,c1(N(CCOCC=C)C)[nH]c(=NC(C)c2ncccc2OC)nc2sccc12 33856,N1(C(=O)CCCn2cccc2)CCOC(Cc2cn[nH]c2)C1.c12ocnc1C2 33857,c1(OCC)ccc(C(=O)NCC2(CNC(C3(C)CC3(C)C)=O)CCCC2)cn1 33858,c1(C(=O)NC(CC=C)CNC(C2CC3(CCC3O)C2)=O)ccc(F)c(C)c1O 33859,CC(C)CC(C)CC(=O)NC(CNC(=O)Cn1cc(CN(C)C)nn1)CC(C)C 33860,c1(C(N2CCCC(CNC(C3(OC)CCC3)=O)C2)=O)cc(=N)[nH]c(Cl)n1 33861,C=CCC(CC(=O)NCCC1CC(OC)C1)NC(=O)C(N1CCNC1=O)C 33862,C(=O)(C#CC1CC1)N(C1COC(C(=O)NCCc2ccco2)C1)C 33863,N1(C(C=CC=CC)=O)Cc2ccccc2C(NC(C2CCc3nccn3C2)=O)C1 33864,N1(C(c2cc(C)c(C)o2)=O)CCN(C)CC1CNC(c1nocc1C1CC1)=O 33865,Cc1nc(C(N2CCCC2CCc2cn(C3C4CC5C(C4)C35)nn2)=O)sc1C 33866,C1(C(=O)NCc2sccc2Cl)CC(F)(F)CN1C(c1ccccc1O)=O 33867,Cc1c(NCc2cscc2Cl)ncnc1N1C2C=CCC1CC2 33868,C1(N(C(CC=C)=O)CCC)CCN(C(=O)C(C)C=C)C1 33869,N#CCCCC(=O)NC1C=CCC(C(N2CCN(c3ncccn3)CC2)=O)C1 33870,C1(NC)CCC(NC(=O)CCN(CCO)C(=O)OC(C)(C)C)CC1 33871,C1(NC(C(C)N(C)C)=O)CC2(C1)CC(NC(c1cncc(-c3cnn(C)c3)c1)=O)C2 33872,CCC(CC(=O)N(C)CCNC(c1nccc(C)c1N)=O)C(F)F 33873,C(=O)(N=S(C)(=O)C1CC(O)C1)C1(N(CCC(=O)OC)CC)CCOC1 33874,C1(C(C)C)COCCN1C(c1cc(-n2cccn2)ccn1)=O.C12CC1CNC2=O 33875,N1(C(=O)C=Cc2cnc[nH]2)CC2(CCC2)CC1C(=O)N(CCC)CC1CCCO1 33876,C1(OC)CC(CNC(=O)C(F)C(C)C)N(C(C2CC(F)C(=O)N2)=O)C1 33877,C1(NC(=O)CNC(C2CCCC2)=O)CCCCN(C(c2ncsc2Br)=O)C1 33878,CC(C)C(C)(C)C(=O)N1CC2CC2(CNC(c2cccc(N(C)C)c2)=O)C1 33879,Cc1cc(C(=O)N(C2CCN(C(c3ccc(F)cn3)=O)CC2)CCO)cc(F)c1C 33880,c1(OC)cccc2c1CC(C(N1CC(C)N(C(=O)CCCF)CC1C)=O)CO2 33881,C#CCC(O)C(=O)N(C1CCN(C(C2(COC)CCCO2)=O)CC1)C 33882,C1(C(=O)NC(C(=O)OC)C(C)C)CC2CN(C(=O)Cc3cccnc3C)CC2C1 33883,CC(CC(=O)NCCN(C)C(c1cnc2sccc2c1)=O)P(C)(C)=O 33884,N1(C(CC)=O)CCC(C2CCN(C(c3cc(F)c(Br)c(F)c3)=O)C2)CC1 33885,C(=O)(C(C)S(N)(=O)=O)N1CCC(NC(c2ccc(C)cc2)=O)C1C 33886,c1(-c2c(SC)ncnc2)ccccc1S(=O)(=O)C(=O)OC.C1(C(F)(F)CO)(N)CNC1 33887,C(C(C)CC(=O)N1CC2C(CNC(c3ccncc3SC(C)C)=O)C2C1)OC 33888,C1(CS(=O)(=O)NCC2CC(N3CCC3)C2)CC2C(C1)C2(F)F 33889,C(=O)(C1CCc2scnc21)N1CC(CN(C)C(c2ccn(C)c2)=O)C2(C1)CC2 33890,N1(C(C2CCC(CC)O2)=O)CCc2nc(CNC(c3ccc(F)cn3)=O)sc2C1 33891,C1(NC(c2n(C)ncc2)=O)CC2CC1CN2C(c1ccncc1F)=O 33892,c1(C(=O)NCC2C(NC(c3c(N)cccc3F)=O)C2)ccc(F)cc1[N+](=O)[O-] 33893,c1(N2CCC(NC(C)=O)CC2)cc(C)c(S(=O)(=O)NCC2CCCC(C)C2)cn1 33894,N1(C(COCC=C)=O)CC(NC(C2CCCCC(=O)N2)=O)CC12CCOCC2 33895,N1(C(C2SCCS2)=O)CCC2(CCCN(C(c3cc(C4CCOC4)[nH]n3)=O)C2)C1 33896,C1(N(C)C(C2CC(=O)N(C3CC3)C2)=O)CCN(C(C2C3COCC23)=O)CC1 33897,C1(O)(CNC(C2C(C)CC2)=O)CCCN(C(c2ccc(F)c(CO)c2)=O)C1 33898,c1(C(N2CC(O)(C3CCCN3C(C3(C4CCCO4)CC3)=O)C2)=O)ccnc(Cl)c1 33899,C(=O)(C(C)(C)O)O.C(C(C)(C)CC1CCOCC1)OCCOCCOC 33900,c1(NCCC2(c3ccc(-c4cn(CCCC)nc4)cc3)CC2)c(C)cccc1F 33901,CC(C)CC(CC(=O)NC12CC3CCC(C1C2)N3C(C1(F)CCC1)=O)CC(N)=O 33902,C1(NC(C=Cc2cc(OC)ns2)=O)CC2CCC(C1)N2C(=O)Cc1c[nH]nc1C 33903,c1(C(N2CCC(C(=O)NC(COC=C)C)(C(C)C)C2)=O)cn2c(n1)CCC2 33904,CC(C)CCC(C)N=c1[nH]c(=NC2COC3(CCC3)C2CO)[nH]c2ncn(C)c12 33905,CP(C)(=O)C(O)C(=O)NC1CCCC1NC(c1ccc(F)c(NS(C)(=O)=O)c1)=O 33906,N1(C(=O)OC(C)(C)C)CCC2(C1)CN(C(c1cnoc1-c1ccco1)=O)CCO2 33907,C1(NC(C(C)Sc2nnnn2C2CCCC2)=O)CCC(NC(C2(C)CC2C)=O)CC1 33908,c1(-c2nn(-c3cnc(C)s3)c(Cc3nccn3C)n2)ccc(C)cc1C 33909,C12(CC(=O)NC(C3CCN(C(CCOCCOCC)=O)C3)C)CCC(CC1)OC2 33910,c1(CC(C)C)ccc2cc(C(=O)NC3CCNCC3)[nH]c2c1 33911,c1(C(=O)NC2CCCCN(C(C3C(OC)CCCC3)=O)C2)cc2c([nH]1)CCOC2 33912,N1(CC(=O)N(C(c2csc(C)c2N)=O)C2CC2)C(=O)NC2(CCCCC2C)C1=O 33913,c1(C(=O)NC2CCN(C(c3c(OC)ccs3)=O)C2)ccc(C2CC2)c(OC)c1 33914,N1(C(=O)C(F)C2CCOC2)CC2(CCN(C(C3(CC4CC4)CCCO3)=O)CC2)C1 33915,C1(NC(CN(C)S(N)(=O)=O)=O)CN(CC(c2ccccc2)c2ccncc2)CC1O 33916,C1(C(=O)NC2C(C)(C)CCC2)CC1C1CN(C(=O)COc2ccccc2)C1 33917,C(C(=O)NC1CC2(C1)CC2C(=O)NCC1(C#N)CC1)(C(C)C)NC(C)=O 33918,CC1CCC=C1C(=O)N1CCN(CCCNC(C2CC2Br)=O)CC1 33919,c1(CC(N2C3(CN(C(c4ccnc(CO)c4)=O)C3)CC2)=O)cccc([N+](=O)[O-])c1 33920,Cc1csc(C(=O)NC2CN(C(=O)CCc3ccc[nH]3)CC2F)c1Cl 33921,c1(C(CC)=O)cc(=NC2CCCC(NC(C3(C)CCCCCC3)=O)C2)[nH]c(Cl)n1 33922,N1(C(C=COCC)=O)CCN2C(=O)C(NC(=O)CC3CSC3)CC2C1 33923,CC(C)(C)C(C)(O)C(=O)N1CCCN(C(c2coc(C(C)(C)C)n2)=O)C(CO)C1 33924,c1(C2(C)CC2)ccnc(NC2CCCCC2NC(=O)C2=CC(C(F)(F)F)C2)n1 33925,C1(C(N(CC)Cc2ccc(O)cc2)=O)CCCN(C(c2cnoc2C)=O)CC1 33926,c1(C(=O)Nc2cnn(CC)c2C(=O)O)cc([N+](=O)[O-])ccc1Cl 33927,C1(NC(c2c(C)n(C)nc2)=O)C(C)CN(C(=O)CC(C2CC2)C2CC2)CC1C 33928,C1(CNC(c2c(C)cc(O)nc2)=O)CN(C(=O)CC(C)C2CC2)CCC1(F)F 33929,CC1(C)CN2CCC1NC2=O.c1(COC(=O)OC)ccccc1.C(N)C(F)(F)F 33930,C1(CNC(c2c(C)snn2)=O)CC(NC(=O)Cc2sccc2Cl)C1(C)C 33931,c1(OC)cc(NC(C2CNCCN2Cc2cnc(N(C)C)nc2)=O)c(Br)cc1Br 33932,C(c1cccc(F)c1F)=CC(=O)NC1CCCC(CNC(C(C)O)=O)C1 33933,CCC(C(C)C)C(C(=O)NCCC)N1CCC(c2ccc(N)cc2)CC1 33934,C1(NC(=O)NCC(C)N(C(=O)C(C)=C(C)C)CC)CC(=O)N(c2nccs2)C1 33935,C1(C(=O)NCCCC(C)(C)NC(c2cncc(C3CC3)c2)=O)CN2CCC1CC2 33936,Cc1ccc2c(C(=O)NCCCN(C(C3SCCCS3)=O)C3CC3)c[nH]c2c1 33937,N1(C(CNC(C)=O)=O)CCN(CCN(C)C(C2CC2Cl)=O)CC1 33938,C12CC(C1(c1cccnc1)NC(=O)CC)O2.C1(COCCCN)CCOC1 33939,N1(C(Cc2cccc(C)c2)=O)CCN(C(=O)Cc2ccccc2F)CC(CO)C1 33940,C1(N(C(C2CC(OCC)C2)=O)CC)CCN(C(=O)Cc2ccc(C)nc2)CC1F 33941,N1(C(C=Cc2cn(C)nc2)=O)Cc2ccccc2C1CNC(c1cnnn1C)=O 33942,c1(SC)nc(N2CC3CC2CN3C(=O)C=Cc2ccccc2)c(Br)c(C)n1 33943,c1(OC)cccc(-n2cc(CNC(=O)CN3CC(C)(C)C3)nn2)c1C 33944,c1(C(N2CCN(C(c3cccnn3)=O)C(C3CC3)C2)=O)ccc(Br)c(F)c1 33945,c1(C(N2C(CNC(C=CCC)=O)CC(F)C2)=O)cc2cc(Cl)cnc2o1 33946,C1(C(=O)NC(COC)C)CC(O)CN1C(=O)CN1CCOCC1 33947,n1(CCOC)nc(COc2ccccc2C)nc1-c1ccnc(OC)c1 33948,N1(C(CN(CCC)C)=O)CC2CCCC2(C(=O)NC2(CC3CC3)CCC2)C1 33949,C1(C(=O)NCC2CC(NC(c3c(COC)cc[nH]3)=O)C2)CCS(=O)(=O)C1(C)C 33950,N1(C(CCSC)=O)CCC2C(NC(=O)C(c3ccnn3C)C)CC12 33951,C1(SCCNC(c2cnco2)C)CCS(=O)(=O)C1 33952,N1(C(CC(C)C(F)F)=O)CC2(CCN(C(=O)C=Cc3ccn(C)c3)C2)C1 33953,C1(CCOC)(NC(c2ccon2)=O)CCN(C(C2CCOC2C)=O)C1 33954,C#CCCC(C)(c1nn[nH]n1)N(C1CCCC1)CCCN(C)C 33955,N1(C(CN(C)Cc2ccccc2)=O)CCCCC1CCNC(c1cnccn1)=O 33956,C1(C(=O)OC)COC2(CCC2)CN1CCC(C)F 33957,N1(C(c2ccc(Cl)cc2Cl)=O)CC2CCCC(N=c3cnc(F)c[nH]3)C2C1 33958,N1(C(c2ncc(F)cc2F)=O)CC2CCN(C(C3CC4CCC3O4)=O)C2C1 33959,C12(CNC(c3ccc(Cl)cn3)=O)CC1CN(C(c1cccc(=O)o1)=O)C2 33960,N1(C(C2(SCC)CC2)=O)CC(NC(c2cnc(CC3CC3)s2)=O)C2(CC2)C1 33961,N1(C(C2=NOC(C)C2)=O)CC2(CCCC2)CN1C(=O)C#CC1CCC1 33962,c1(C(=O)NC2CC(NC(CCCC)=O)C23CCC3)cc2cnc(Cl)cc2s1 33963,c1(N2CCC(NC(c3cccc(C(C)C)c3)C)C2)ccc(S(=O)(=O)N(C)C)cn1 33964,c1(C(C)C)nc(=NCCCCC(C)NC(c2ccc(C(F)F)c(F)c2)=O)s[nH]1 33965,c1(C(=O)NC2CCC(CNC(c3cc(C)oc3)=O)C2)ccc([N+](=O)[O-])n1C 33966,C12(NC(C(C)OCC=C)=O)CCCC1(F)CN(C(c1[nH]nc([N+](=O)[O-])c1Cl)=O)C2 33967,N1(C(c2c(CC)nn(C)c2)=O)CCC(C)C(NC(=O)CSCCN(C)C)C1C 33968,c1(NC(CC2CCN(C(CC=CCC)=O)C2)=O)cccc(C2CC2)c1F 33969,C1(NC(CSCC(=O)NC2C(O)CC2O)=O)CC2CCC(C1)C2=O 33970,CC1CN(C(=O)CCCSC(C)(C)C)CCCN1C(=O)C(C)CC1CCC1 33971,C1(N(C)C)(C(=O)NCC(CNC(=O)C(F)=C2CCCC2)CO)CCCOC1 33972,C#CC1(NC(C2C=CC(NC(=O)CCCOCC)C2)=O)CCCCC1 33973,N1(C(C2(C)CCCCNC2=O)=O)CCOC2(CCN(C(=O)C=CCF)C2)C1 33974,C=CC(C)(O)CC(=O)N(CC(C)O)CCNC(=O)Cc1sc(C)cc1C 33975,c1(OCCC)ccc(Cl)cc1CC(N1CC2C(NC(=O)C3=C(Cl)CC3)C2C1)=O 33976,c1(Oc2ccc(CCO)c(Cl)c2)ccnc2cc(F)cnc12 33977,c1(OC)ccc(CNC(C(C)(C)OC)c2nnnn2CC(F)F)cc1C#N 33978,O=C1CCCC(NC(=O)CC2COCCN2Cc2ccc(Cl)o2)C(=O)N1 33979,C1(C(=O)NC2CC(CNC(C3(F)CC4(CCC4)C3)=O)C2)CC2(C1)CC(F)(F)C2 33980,c12ccc(cc1)s2.C1(CNC(CSC)=O)CC(C)N(C(=O)CN2CCCCC2)C1 33981,C1(CC(N2CC(N(C(c3ncc(C)cn3)=O)C3CC3)C2)=O)Cc2ccc(Br)cc2C1 33982,C(=O)(C(C(=O)Nc1cccc(CNC(=O)C(COC)OC)c1)C(C)C)OCC 33983,N1(C(=O)C=CC2CC2)CCCC1CC(=O)NCC(C(=O)N(C)C)N1CCC1 33984,C#Cc1ccc(CCC(=O)NC2CCN(C(c3cnn(C)c3)=O)C23CC3)cc1 33985,c1(C(=O)NCCNC(C(F)OC)=O)c(Cl)c([N+](=O)[O-])nn1C 33986,N1(C(C2CC23CCOC3)C(=O)NC(C)C)CCc2ccc(F)c(F)c2C1 33987,C1(C2CCN(C(c3cc(C)n(CC(F)(F)F)n3)=O)C2)(NC(CCNC(C)=O)=O)CC1 33988,C1(NC(c2c(CC=C)cccc2)=O)CCCN(Cc2cn(C)nn2)C1C 33989,CCC1=NOC(C(=O)NC2CC2NC(c2cn(CCO)nn2)=O)C1 33990,C1(NC(c2ncn(CC)n2)=O)CN(C(c2sccc2CC#N)=O)CC1C 33991,CC(C)(CC(=O)NC1CN(C(=O)CS(=O)C(F)(F)F)CC1n1ccnn1)C(F)F 33992,CCCCC(C(=O)NC1CC2CC1CC2CO)NC(=O)C(C#N)CC 33993,c1(OC)ncnc(Cl)c1NC(=O)CC1(Nc2ccc(C)cc2Cl)CCC1 33994,C1(CNC(CCC(=C)C)=O)CN(C(C2CC(OC3CC3)C2)=O)CCC12CCC2 33995,C1(CNC(c2cnc(CCC)s2)=O)CC2CCC(C1)N2C(=O)CC1CCCOC1 33996,Cc1ccc(Cl)c(C(=O)NC23CC2CN(C(=O)C(C)(C)CN2CCOCC2)C3)c1 33997,CC1(C)OCCC1(O)C(=O)NC1CCC(CC(=O)NC2CC23CCC3)CC1 33998,c1(C(N(C)CC2(CNC(c3c(C)csc3)=O)CC2)=O)nc(C)n(C)n1 33999,N1(C(c2nc(C)oc2C)=O)CCCC2(C1)C(NC(=O)CCNC(N)=O)CCN2C 34000,c1(CNC(C(=O)OCC)CCF)ccc(OC)c(N)c1F 34001,CC1(NC(C23CC(CN2C(c2cc(N)cc(F)c2)=O)C3)=O)CN2CCC1CC2 34002,c1(CN(C(=O)C(CCc2ccccc2)C(=O)O)CC)cc(Cl)cc(Cl)c1 34003,C1(NC(C(C)OCCN(C)C)=O)CCSC12CN(C(=O)CCC1CCCO1)C2 34004,N1(C(CC2CC(OC)C2)=O)CC(C(N)=O)(CNC(c2cc(C(N)=O)c[nH]2)=O)C1 34005,c1(CNC(c2c(C)n(C)cn2)=O)ccc2c(c1)CN(C(=O)C(F)C(C)C)C2 34006,Cc1c(CC(N2CCCC2C2(C(=O)NCC3CCOCC3)CC2)=O)cnn1C 34007,c1(OC)cnnc(C(=O)NCC(O)CC(=O)NCC(C)SC)c1 34008,C1(NC(C2(CCO)CC2)=O)CCCN(C(C2(C(F)(F)F)CCOCC2)=O)CC1F 34009,N1(C(CC=C)=O)CCCC2(C1)CN(C(C1OCCOC1(C)C)=O)CCO2 34010,C(N=c1ccc(-c2ccccc2)c[nH]1)c1c(C)cc(Cl)cc1.N(C)C 34011,C1(NC(CN(C(=O)CN(CC(C)(C)C)C)C(C)C)=O)CCOC(C(C)C)C1 34012,c1(NCC(=O)NC2(CNC(CCOCCN(C)C)=O)CC2)nn(C)cc1Br 34013,Cc1nsc(C(=O)NC(C2CCCN(C(=O)C(C)(C)C3CCC3)C2)C)c1N 34014,CCC(C)CCC(=O)NCc1ccc(C(N2CC(OCCF)C2)=O)cn1 34015,CCC(CC(=O)Nc1cnn(CC2CC2)c1)NC(=O)CC1(C)CC1 34016,C1(CN(C(C(C)OCC)=O)C)CCCN(C(c2ccc(SC3CC3)cc2)=O)C1 34017,N1(C(C(C)NS(CC)(=O)=O)=O)CC(NCC2CCC2)CC(C)C1 34018,C1(C(=O)NC(CN(C)C(=O)OC(C)(C)C)(C)C)CC(C2CC2)=NO1 34019,C=CC(C)(CC)NC(c1c[nH]nc1C(C)(C)OC)=O 34020,N1(C(c2cnn(C)c2)C(=O)NC(C(=O)OC)CC(C)C)CCCC(C2CCC2)C1 34021,N1(C(=O)OC(C)(C)C)CC2CCC(Nc3cc(F)ccc3CC(N)=O)C2C1 34022,C1(NC(C(=O)N(C)C)=O)CCC2CCN(C(c3ccccc3SCCO)=O)C1C2 34023,c1(OCC)cncc(C(=O)NC(C2CN(C(=O)Cc3cc(Cl)cs3)C2)C)c1 34024,C1(C)(CNC(C2(CCC=C)CC2)=O)CCN(C(c2ncoc2C)=O)CC1 34025,C(=O)(CS(=O)(=O)C(C)C)NC1CCC(CNC(C(C2CCOC2)OC)=O)C1 34026,c1(N2CC3(CN(C(c4c(OC)nccc4)=O)C3)C2)ncnc2scc(C)c12 34027,C1(CCNC(C(c2ccc(C3CC3)cc2)C)=O)CCC=CCC1 34028,Nc1nc(C(=O)NC23CC(C2)N(C(=O)CCOCC(F)F)C3)ccc1[N+](=O)[O-] 34029,N1(CCC(=O)Nc2ccc(Cl)cc2)CCC2COCCC12 34030,CCC(C)(C)C(C)OC(C1CCCN1C(=O)OC(C)(C)C)=O 34031,C#CC1(NC(C2CC(NC(c3csc(F)c3)=O)C23CCC3)=O)CCCCC1 34032,N12C3CCC1CC(C3)NC2=O.c1(CC)ccc(Br)cc1C(=O)NCc1nccs1 34033,C1(O)(Cc2ccc(Cl)cc2)CCN(c2nocn2)C1.c1(CC(=O)N(C)C)ccsc1Br 34034,C1(C#N)(C(=O)NC(C)C(C)NC(c2cccnc2C(F)(F)F)=O)CC1(C)C 34035,Cc1csc(Cl)c1C(=O)NCCCN1CCN(C(=O)CSc2ccncc2)CC1 34036,c1(CNC2C(CNc3cc(C)c(I)c(C)c3)CCC2)ccc2c(c1F)OCCO2 34037,Cc1c(C(=O)NCCC(C)(C)NC(C2CC2(C)C(F)F)=O)cnc2ncnn12 34038,n1(CC(=O)NCC(CNC(CC(CC)OC)=O)C)cccc([N+](=O)[O-])c1=O 34039,c1(C(N(C(C)C)C)C)nc(C(O)CC)nn1-c1ccc(Br)cc1 34040,O=C(C=CCC(F)(F)F)NCc1cncc(Br)c1Cl 34041,C1(CC(=O)N(C(COC)C)C)CCN(C(=O)CC=C(Cl)Cl)C1(C)C 34042,C(=O)(C1=CCCCCC1)NC(CCCC=C)C(=O)NC(CCC)C(=O)N(C)C 34043,c1(Cc2n(-c3cnc(C)s3)nc(COC3CCCN3C)n2)ccc2ccccc2n1 34044,N1(C(CC(OCC)OC)=O)CCC2CCCC12CNC(C1CCC(OCC)C1)=O 34045,C(=O)(C(C)(CNC(c1nn(C)cc1Cl)=O)CC)NCCOCC 34046,N1(C(CN2CC(C)C2)=O)CCC2C(C1)CN2C(=O)C(N1C(=O)CCC1=O)C 34047,c1(C(N2C(C)CN(C(C3CC(=C4CCC4)C3)=O)CC2)=O)cc2occc2n1C 34048,CC1C(NC(C2CCCCS2(=O)=O)=O)CCCN1C(C1CCCC1)=O 34049,C1(CC)CCC(C(=O)N(C)CC2CCCN2C(c2cnsc2)=O)CC1 34050,c1(C(=O)NCC2CCCN2C(C2CC(CCO)C2)=O)cc2c(F)c(Cl)ccc2[nH]1 34051,c1(C(=O)NC(COC)CNC(c2cnn(CCO)c2)=O)cnc(Cl)n1C 34052,C(=O)(C1=CCCCC1C)N1CCCC(NC(COCC(C)C)=O)CC1 34053,N1(C(C2CCN(c3n(C)ccn3)C2)=O)CC2(CCN(C(C3CC3(C)C)=O)CC2)C1 34054,C(=O)(CCCS(=O)(=O)NC(=O)Nc1nc(C)no1)OC 34055,C1(C(=O)NC(CCC)C)CCC2(CC1)CN(C(=O)C(C)OC)C2 34056,C1(C2(NC(c3cc(C(=O)OC)[nH]c3)=O)CC2)CCCCN1C(c1n[nH]c(C)n1)=O 34057,C1(F)(C(=O)NC)CCN(C(=O)C(=O)Nc2ccc(OCC3CCCO3)cc2)C1 34058,N1(C(C2(CC=C)CN(C(=O)CN3CC4CC4C3)C2)=O)CCc2oc(C)nc2C1 34059,c1(C(=O)NCC(C)NC(=O)C(c2ccccc2F)C)cccc(N)c1Br 34060,C1(NC(N2CCCC(n3ccc(C)n3)C2)=O)CCC(F)(F)C(C)(C)O1 34061,c1(C(=O)NCC(CCOC)NC(C2CC3CC3C2)=O)oc(COC)nc1C 34062,CC1CCCCN1CCNC(=O)C(CC1CC1)NC(c1ccc(CC#N)cc1)=O 34063,C(=O)(C(CC(C)C)NC)N1C(C(N2CCCC(CCC=C)C2)=O)(C(C)C)CCC1 34064,N1(C(Cc2ccn(CC)n2)=O)CCCCCC1CNC(=O)C(C)(CC)CO 34065,C(=O)(C1OCCc2ccccc21)N(CCCOCC(F)(F)F)C(C)C 34066,N1(C(C(Cc2ccoc2)NC(CNC(=O)NC)=O)=O)CC(CO)C1(C)C 34067,c1(C(C(=O)NCC#CCNC(C2(C)CCNC2=O)=O)N(C)C)c(F)cccc1F 34068,N1(C(C=COCC)=O)CC(NC(c2cc3n(n2)CCC3)=O)C(C)(C)C1 34069,c1(C(N2C(CCNC(C(C)OCC(C)C)=O)CCC2)=O)noc2ccc(Cl)cc12 34070,N1(C(C2N(C)CCN(C(C(c3ccn(C)c3)C)=O)C2)=O)CCCC(C)(C)CC1 34071,C1(CC(C)(C)C#N)C(=O)N1.N1(CCS(C)=O)CCC(CC#N)CC1 34072,c1(C(=O)NC(CNC(CC(C)n2ccnc2)=O)C2CC2)ccc(P(C)(C)=O)cc1 34073,c1(-c2ccc(C(F)F)o2)nc(C2CCC2)nn1CCCO 34074,C1(CNC(c2c(C)cccc2C(C)C)=O)CCN(C(C2CC2CF)=O)C12CCC2 34075,c1(OCC2C(NC(c3cc(-c4ccccc4)[nH]n3)=O)CCC2)ccc(Cl)cc1Br 34076,C1(C(N2CCCC(Cn3cc(CC(C)O)nn3)C2)=O)CCc2nc(O)[nH]c2C1 34077,c1(N(CCCC)C)ccc(C(F)(F)F)cc1S(=O)(=O)N1CCCC2CC2C1 34078,CC(C)C(C)C(C)CC(=O)NC(C1CCN(C(=O)Cn2cnc(=N)[nH]2)CC1)(C)C 34079,CCCC(O)C(=O)NC1(C)CC1.C12CCN(CC1)C2=O.C(C)(C)(C)O 34080,N1(C(C(CSC)O)=O)CC(C(N2CCCN(C)CC2C)=O)C2(CCC2)C1 34081,C1(NC(C(COCC)(C)C)=O)COC2CN(C(=O)C(F)C(C)(F)F)CC12 34082,C(=O)(C1CC(=O)c2ccccc21)N1C(C)(CNC(C(C)NC(N)=O)=O)CCC1 34083,Cc1cc(C(=O)NC2CN(C(C3(C)CCCCCC3)=O)CC2(C)C)nc(C)c1 34084,C=CC(C)(CC)C(=O)N(CCCNC(=O)CNC(=O)COc1ccc(F)cc1)C 34085,Cc1cncc(C(=O)NC2CCCC2NC(=O)CCF)c1Cl 34086,c1(C(=O)NCC(C)(CO)NC(=O)C(F)CC2CCCCC2)cc(Cl)ccc1O 34087,C1(C(=O)NCC(n2ccnn2)C)CN(C(=O)CN2CSCC2=O)CC(C)(C)C1 34088,Cc1oc(Cl)nc1C(=O)NC1(CCCC(=O)NC2CC(C(F)F)C2)CCC1 34089,CC1CC(NC(=O)C(C)(F)C(C)(C)F)CN(C(=O)CCS(C)(=O)=O)C1 34090,N1(C(=O)Cc2c[nH]nc2O)CCC2CCN(C(c3ccc(Cl)cc3O)=O)CC2C1 34091,N1(C(c2c(C)noc2)=O)CC(NC(C2CCC(N(C)C)CC2)=O)C2CC12 34092,C1(NC(C2CCC3CC23)=O)CN(C(c2cnc(Br)s2)=O)CC12CC2 34093,C1(NC(=O)COC2CCOC2)CC(F)CN(C(c2c[nH]nc2C(F)(F)F)=O)C1 34094,N1(C(N2CCN(C)CC2C(C)(C)C)=O)CCOC2(CCCN(C(=O)C3CC3)C2)C1 34095,C(=O)(CCC(=O)NCC1(CNC(C2CC2C(F)(F)F)=O)CC1)c1cn(CC)nc1 34096,CC(C)CC(C)(O)C(=O)NCC1CC1NC(C1(CCc2ccccc2)CC1)=O 34097,C1(=O)C(F)CC2CN1C2.c1(COCC(=O)NCC2CN(C)C2)ccccc1 34098,c1(C2(C(=O)NCCOCCN(C)C(=O)C3CC3)CC2)ccc(F)c(Cl)c1 34099,CC1=CC(O)CN(C(=O)NC(c2nc(C(=O)OC)sc2)C)C1.C1CC1 34100,C1(C(=O)OC)CC(F)(F)CN1N(CC(F)(F)F)CC.c1nccs1 34101,c1(C(N2CC3N(C(CN(C)C)=O)C(C3)C2)=O)cc2ccc(Cl)cn2c1 34102,c1(CC)ncc(C(=O)NC(CO)C(C)NC(c2ccncc2C)=O)c(O)n1 34103,Cc1cc(C(=O)NC2CCCC23CN(C(=O)C(F)C(F)(F)F)C3)cc(N)c1Cl 34104,C1(C(=O)NC(C)CN=[N+]=[N-])CC(N=[N+]=[N-])CN1C(C1CCNC1=O)=O 34105,C(=O)(C(F)C(C)(C)O)NC1C(CNC(C2(CC#C)CC=CCC2)=O)CC1 34106,c1(C(=O)OC)cc(C2CCCN(C(=O)C=CC(C)C)C2)cnc1OC(C)(C)C 34107,C1(C(C)C)CCC(C(=O)N(CCNC(=O)C(C)N2CCC2)CCN(C)C)CC1 34108,c1(CC)noc(C(=O)NC2CCN(C(C3CC(OC)C3)=O)CC2)c1C 34109,c1(C(N2CC(C)C(CNC(c3cnc(O)c(F)c3)=O)C2)=O)cnc2c(c1)NCC2 34110,c1(C(N(CC(CC)NC(c2cccc(OC)c2)=O)C)=O)cn(C2CC2)nc1C 34111,CCC(O)C(C)(C)C(=O)N1CCN(C(=O)C(C)(Cl)Cl)CC(O)C1 34112,c1(C(=O)NC2C(C(=O)NC(CC=C)C(=O)OCC)CC2)cc(C)nc(O)n1 34113,c1(COC(c2cccc(COCc3ccccc3)c2)=O)cc(CCO)cc(Br)c1 34114,Cc1ccsc1C(N1CCCC1CCNC(=O)C(C)SC(F)(F)F)=O 34115,C1(CNC(c2c(OC)nsc2OCc2ccccc2)=O)CC2(CC(=O)CCO2)C1 34116,N1(C(CCCCC=C)=O)CCCCC12CN(C(c1cn(CCC3CC3)nn1)=O)C2 34117,O=C(C1Cc2ccccc21)N1CCC(N2CCN(C(C3(CO)COC3)=O)CC2)C1 34118,N#CC1(C(=O)NC2CC(NC(C34CCOCC3C4)=O)C2)CCSCC1 34119,N1(C(CCCOC(C)C)=O)CCC(NC(=O)CC2CCCN(C)C2)CC1C 34120,N1(C(CN(CCC)C(C2CC=CCO2)=O)=O)CC(O)CC1CC(C)C 34121,c1(C(N2CCC(NC(C)=O)CC2)C(=O)NCCCCCC)nn(COC)nc1Br 34122,Cc1cc(Br)cc(C(=O)NC2(CCO)CN(C(C3CC(C)CO3)=O)C2)c1C 34123,N1(C(C2(CNC(=O)CC(C)(C)O)CC(=C)C2)=O)CCCCC(C)C1 34124,C1(C)(C(N2CC(CNC(c3c(C)occ3)=O)C2)=O)OC(C)(C)OC1C 34125,C(=O)(C1CSc2ccccc21)NCCC1(C)CCN(C(C2CC(O)C2)=O)C1 34126,C1(CNC(CCCC#CC)=O)CC12CCN(C(C1CC3CCC(C1)N3C)=O)CC2 34127,C1(C(N2CC(F)(CNC(C3N(CC)CCC3)=O)C2)=O)CCc2cn(C)nc2C1 34128,N1(C(CC(COC)(C)O)=O)CCCC2(NC(=O)C=CS(C)(=O)=O)CCCC12 34129,N1(C(c2cnc(C3CC3)s2)=O)CCN(C(c2cnn3c2OCC3)=O)C(CCO)C1 34130,c1(SC)ncc(C(=O)NC2CC3CN(C(c4ocnc4C4CC4)=O)CC23)c(O)n1 34131,CC1(C)CCCC(C(N2CC3(CC(CC(=O)Nc4cnccc4CO)C3)C2)=O)C1 34132,C(C(=O)NCC1CC(NC(=O)Cc2ccc(OC)cc2)CCO1)(C(C)C)OCC 34133,c1(C(=O)NC(C(=O)NC(CC=C)CO)C2(O)CCC2)n[nH]c(C)c1Cl 34134,C1(NC(CC=CC)=O)(CF)CCN(C(c2cn(CCCC)nc2C)=O)C1 34135,C(C1=NCC(C)(C)O1)NC(C1CN(c2c(OC)cccc2)C(=O)C1)=O 34136,C1(CCNC(C(C)(C)OC)=O)CN(C(=O)C(C)NC(c2ccoc2)=O)CC1C 34137,N1(C(C2C(C)OCCO2)=O)CCCC(C)(NC(=O)C(=O)N2CCCC2)C1 34138,CC1CC(NC(=O)CC(C)(C)F)CN(C(c2cncnc2)=O)C1 34139,c1(C(N(CCNC(C2(C)C(C)CCC2)=O)CC2CC2)=O)cnn2c1CCC2 34140,c1(C(N2C(CNS(C)(=O)=O)CC3CC32)=O)cccc(C2CCCOC2)c1 34141,N1(C(CC=C=C)=O)CC2CC1C2NC(=O)Cc1ccccc1 34142,N1(C(c2n(CCOC)ncc2)=O)CCCC1(C)C(C)(C)CNC(=O)C(O)C1CCC1 34143,c1(C(N(CCCOCCNC(C2CCC(F)C2)=O)C)=O)nnn(C)c1N 34144,C1(C(F)(F)F)(OC)CCCN(C(C(=O)NC(C)C)c2nccs2)C1 34145,c1(C(=O)OC)ncccc1-c1cn(CC2CCC(NC(C3CC(F)C3)=O)C2)nn1 34146,C1(NCc2c(C)nsc2)C2CN(C(N(C)C(C3(C(=O)C4CC4)CC3)=O)=O)CC12 34147,CCC(CCOC)C(=O)NC1(CCC(=O)NC2COC(C(F)F)C2)CCC1 34148,C(=O)(C(C)(C)CC(F)(F)F)N(CCNC(C(CCC)N(C)C)=O)CCC 34149,N1(C(C(c2cccc(Cl)c2)C)=O)CCN(C(c2ccc(Cl)cc2N)=O)CC1C 34150,c1(C(=O)NCC2N(C(C(c3ccccc3)OC)=O)CC(O)C2)cnc(C)cc1Cl 34151,C1(COC)COCCN1CCc1cc(-c2ccccc2)no1 34152,c1(C(=O)NCC2(O)CCN(C(C3C(c4cc(C)on4)C3)=O)C2)cccc(=S)n1O 34153,c1(C(N(C2CN(C(c3ccc(C)nc3C3CC3)=O)C2)C)=O)cc(F)c(F)cc1C 34154,c1(C(=O)NC(C2(O)CN(C(C(CC)N(C)C)=O)C2)C)cc2nccnc2cc1C 34155,C=Cc1cncc(C(=O)NC(C2CCOC2)CNC(c2c(C)cncc2F)=O)c1 34156,N1(C(C(C2CCN(C(c3cnn(C4CC4)c3)C)C2)F)=O)CCC2(COC(C)C2)C1 34157,c1(C(N(C2CCN(C(=O)CC3CC3)CC2)CCCC)=O)ccc(Cl)cc1.c1cccs1 34158,c1(N2CCCC(c3c(C)cccc3)C2)nc(NCC23CC(CO2)C3)c2ccsc2n1 34159,c1(OC)c(F)ccc(F)c1C(=O)NCC1CCC2(CCC2)C1NC(=O)C(N)=O 34160,C1(C(=O)NCC2(C)CC(F)(F)CNC2)CCc2n[nH]cc2C1 34161,c1(C(=O)NC2CC(NC(C=C(C)C(C)C)=O)C23CCC3)coc2ccccc12 34162,C(=O)(C(F)(CNC(C1(C#N)CCCOC1)=O)C(C)C)NC(C(=O)N(CC)CC)C 34163,N1(C(c2c(C)onc2Cl)=O)CC(NC(c2cccc3nc[nH]c23)=O)C2(CCC2)C1 34164,C(C(CC(C)C)C(=O)N1CC(NC(C2(c3cccs3)CC2)=O)C(C)C1)OC 34165,N1(c2nc(Cl)nc(C)c2F)CCC2(CC1)OCCC2NC(=O)Cn1nnnc1C 34166,c1(CN2CC(N(C(c3ncsc3C(F)(F)F)=O)C3CC3)C(F)C2)ccc2nc[nH]c2c1 34167,C1(CNC(C(C)c2cncs2)=O)CCCC1NC(=O)C(C)(C)O 34168,N1(C(=O)NC2CCOC(c3ccccc3)C2)CCN2CCOCC2C1 34169,c1(CCC2CC2)c[nH]nc1CCOCC#C.C1C(=O)N1CC1(CCC)CC1 34170,CC(C)CCC(C)NC(=O)CCC(=O)NC(=O)OC(C)(C)C 34171,Cc1cc(C(N2CCCC(N(C(=O)C(C)CC3CC3)C)C2)=O)ncc1Cl 34172,CC1OC(=O)NC1C(=O)NC1CCCC(NC(c2cc(Br)sn2)=O)C1 34173,c1(SC)cc(NC2CCN(C(=O)C(C(C)C)C3CCC3)CC2C)nc(SC)n1 34174,N1(C(C2CCC(=C)CC2)=O)CCC2CCN(C(c3cc4sc(Cl)cc4[nH]3)=O)CC12 34175,Cc1noc(C)c1C(C)C(=O)N(C)CCOCCO.C(CC(=O)O)NC 34176,c1(C(=O)Nc2ccsc2C(=O)Nc2nn[nH]c2C(F)(F)F)cnncc1Cl 34177,N1(C(C2N(C(CC3C(C)CCC3)=O)CCCC2(C)C)=O)CC23CCC2(COC3)C1 34178,c1(C(N(C(C)CNC(=O)C(c2cncnc2)C)C)=O)cnc2cnn(C)c2c1 34179,CC(N=c1cc[nH]cc1S(=O)(=O)N1CCCC(CN2CCC2)C1)c1ccc(Br)o1 34180,Cc1ccc2nc(SCCCNC(C3COCCN(CCN=[N+]=[N-])C3)=O)cn2c1 34181,C(=O)(CC(CNC(=O)CC1CSC1)C1CCC1)NC1(CN(C)C)CC1 34182,C1(NC(c2n(CC=C)nnn2)(C2CCCOC2)C)CCC2(CC1)CSC2 34183,N1(C(Cc2c(C)noc2)=O)CCC2C1CCCN2C(C1CCCCO1)=O 34184,C(CC(O)C(=O)NCCCC1CN(C(c2cn(CC(F)F)cn2)=O)CCO1)SC 34185,c1(C(C(=O)NCCC(=O)OCC)N(c2ccccc2)C)nc(Cl)sc1Cl 34186,C=CC(CC)C(=O)NCC1(C(=O)NCC2CC2Cl)CCC1 34187,C(CC(C(=O)NCc1cn(C2CC2)cn1)NC(=O)CC1CNC(=O)O1)SC 34188,S(=O)(=O)(c1ccc2cccc(Cl)c2c1)NCC(C(=O)OCC)C1CCOCC1 34189,c1(SC(F)F)cccc(-c2cncc(CNCc3ncccc3Br)c2)c1 34190,c1(OCCN(C(C=NOC)=O)C)cccc(C#N)c1.C1CN(C)CC1 34191,N1(C(C(C)O)=O)CCC(C2CC(NC(=O)CCc3ccn(C)n3)C2)CC1 34192,N1(C(c2c(C)nc(C)o2)=O)CC2CCN(C(=O)CC3CCC(C)CO3)CC12 34193,c1(C(=O)NCCN(C(c2c(C)ccc(C)c2)=O)C)nc2ccccc2cc1C1CC1 34194,C(=O)(C(C)(C)S(C)(=O)=O)NC(C)CNC(=O)CCOc1ccccc1C(N)=O 34195,C(=O)(C1=CCCC1(C)C)N1CCN(C(Cn2cc(C(C)=O)nn2)=O)CC1CO 34196,C1(NC(C2(CC)CCOC2)=O)CCCCCC1NC(=O)C(F)(F)c1csc(C)c1 34197,c1(CC(C(=O)N2CC(CC(F)F)C2)NC(C2(C#N)C(C)C2)=O)ccccc1Br 34198,N1(C(COCCC#C)=O)CCC(F)(F)C(CNC(c2sccc2CN(C)C)=O)C1 34199,C(N=c1ccn(C2CC2)[nH]1)(c1cc(C)ccc1C)c1n(CCOCC)nnn1 34200,C(=O)(C(C#N)C(C)C)N1CCCC(NC(Cc2c(C)cnn2C)=O)C1 34201,C1(C(C)C)CN(C(C2(C(F)F)CCCC2)=O)CCN1C(c1csc(C2CC2)n1)=O 34202,c1(C(N(CC(CC)NC(C(CC=C)NC(C)=O)=O)CC)=O)cc(F)ccc1C 34203,N1(C(CCN(CCC)C)=O)CC=C(C(C)(C)C(=O)NC2CC(C3CC3)C2)C1 34204,C=CCC(CN1C(=O)C1C)NC(=O)CC1(N(C(C)=O)CCNC(C)=O)CCC1.SC 34205,C1(OC)(CNC(c2cnoc2C)=O)CCN(C(=O)C2=COCCC2)CC1 34206,N1(C(c2c(SCC)cncc2)=O)C2CCC1C(CNC(=O)Cn1ccnc1C)C2 34207,N1(C(C2(NC(=O)C(C3CCCCC3)O)CC(O)C2)=O)CCC12CCSCC2 34208,c1(CC(=O)N(CC(C)C)CCN(c2ccccc2)C)ccccc1-c1nn[nH]n1 34209,C1(C(=O)NCc2nnc(C)s2)CN(C)CCN1C(=O)CC(C)C1CCCC1 34210,C=CC1CN(C(=O)COCC(F)F)CC1NC(=O)CCc1ncc(F)cn1 34211,c1(C(=O)NC2CCN(C(C3(P(C)(C)=O)CC3)=O)C2)n[nH]c2ccc([N+](=O)[O-])cc12 34212,N1(C(CC2(NC(C=CC(C)C)=O)CCCCC2)=O)CC2(C)CC1CCO2 34213,N1(CC2(c3ccc(OC)cc3)CC2n2cc(CN)nn2)CCC2(CC1)CN(C)C2 34214,NS(=O)(=O)c1ccc(C2(C(=O)NC3CCC3NC(C3(CO)CC3)=O)CCC2)cc1 34215,C1(C(=O)NCCSCC=C)CC2(CC2)CN1C(=O)NC(=O)C(Cl)(Cl)Cl 34216,Cc1nscc1C(=O)N(C)CCNC(=O)CC1CCC(C)O1 34217,C1(C(=O)NCCC(C)N(C)C(c2cn(C)nn2)=O)CCC(C)(C)C1 34218,C1(NC(Cn2nc(C)n(C)c2=O)=O)CC12CCN(C(C1OCCC1C)=O)CC2 34219,N1(C(c2cc(C)c(Br)cn2)=O)CCN(C(C2(CO)CC2)=O)CC(C)(F)C1 34220,Cc1cc(NC(=O)NC2(c3ccccc3)CCOC2)cnc1C 34221,CCC(C(=O)NCC1(C)CCCN1C(=O)C1=NOC(C(C)(C)C)C1)C(C)C 34222,c1(CCC(=O)NC(C2CCN(C(c3c(C)nn(C)c3)=O)C2)C)c(Cl)cccc1Cl 34223,CCCN=C(NCC1CCN(C(=O)NC)C1)NCCc1ccc(NC(C)=O)cc1 34224,C1(C(N(C)CC2C3CN(C(=O)Cc4ccccc4)CC23)=O)C2CCC3C(C2)CC13 34225,C1(NC(c2c(C)nccn2)=O)CN(C(c2cnc(S)nc2)=O)CC12CCC2 34226,C(=O)(C1=C(C)OCCS1(=O)=O)NC1CN(C(C(CC)CC(F)F)=O)CC1C 34227,c1(C(=O)NC2CN(C(C(C)N(C)C)=O)CC2C)cc(F)c2nc(O)ccc2c1 34228,C1(CCC)CCC(C(N2CCCC(CNC(c3cnc(C(C)O)s3)=O)C2)=O)CC1 34229,C1(NC(c2c(C(C)C)scn2)=O)CN(C(c2c[nH]ccc2=O)=O)CC2(CCC2)C1 34230,C(C(C)C(=O)NC(C(=O)NCCCC1CC1C)C1CC1(C)C)OC 34231,C12CC13CCN(CC3)C2=O.C1(CN(c2ccccc2)C(C)=O)CCCC(=O)C1 34232,Cc1cc(Br)ccc1CC(=O)NC1CCC1NC(C1CCCCN1C)=O 34233,c1(-c2cn(C3(NC(C(CC)C4CC4)=O)CCOCC3)nn2)ncc(Br)cc1CO 34234,C1(C(=O)NCCCCC2CN(C(c3c(C)cc(C)[nH]3)=O)C2)CC12CCCOC2 34235,c1(OC)cc(C(=O)NC2CN(C(c3coc(C)n3)=O)C2)c(N)c(Br)c1 34236,C=CCC(C(=O)N1CC(C(=O)N(C(C)CN(C)C(C)=O)C)CC(C)C1)C(C)C 34237,C1(C(CC)=O)CCCC1OC(=O)C1CC1 34238,Cc1nc2ccnn2c(C)c1C(=O)NC1CC(C)(NC(=O)CCn2cnnn2)C1 34239,C1(N(C(C(=O)NCCOC)=O)C)CCCN(C(C2(OC(C)C)CC2)=O)CC1 34240,N1(C(CCC(=O)OCC)=O)CCC2(CCCN2C(=O)Cn2cc(C)cn2)C1 34241,CCCC(C(=O)NCCCOCCNC(C1CCc2nnnn2C1)=O)S(N)(=O)=O 34242,N1(C(c2n(CC#C)cnn2)=O)CCCC(C(=O)NC2CC(CC(C)(C)C)C2)C1 34243,N1(C(c2nc(Cl)cs2)=O)CC(C2(N=c3[nH]nc(C4CC4)o3)CC2)C1 34244,C1(C(=O)NCC(C)CN(C)C(c2ncsc2C2CC2)=O)COC2(CCC2)C1 34245,C(=O)(C(CNC(C1CC=CC(O)C1)=O)CC(C)C)N1CCC(NCC)CC1 34246,N1(C(c2c(C)nns2)C(=O)NC(C)(C)C)CCCC(F)(CO)C1 34247,N1(C(c2ncc[nH]c2=O)=O)CC2OCCN(C(C3CC3c3cccnc3)=O)C2C1 34248,C1(C(F)(F)F)(C(=O)NC(CCNC(Cc2c(C)scc2)=O)C)CC2CCC1C2 34249,CC(C1OCCc2sccc21)N(CC(=O)N(C)CC1CCC1)C 34250,N1(C(CC2(C)N(C(c3cnc(CC)o3)=O)CC2)=O)CC(=O)NC(C)C1 34251,c1(NCC2(CNC(c3cc(F)cc(F)c3F)=O)CCC2)ccncc1[N+](=O)[O-] 34252,N1(C(C(C(C)(C)C)OC)=O)CCCC(C2CN(C(=O)C(=O)NCC3CC3)C2)C1 34253,N1(C(c2c(CC)nn(C)c2)=O)CC2CC1CN(C(c1nocc1Cl)=O)C2 34254,Nc1cc(Cl)nc(Cl)c1C(N1C2CCC1C(NC(=O)CC1CC1)C2)=O 34255,C(CC(C)C(=O)NC(C1CN(C(=O)CCc2conc2C)C1)C)=CC 34256,CC1CN(C(C2CCCN2C=O)=O)CC1NC(C1(N(C)C)CCC1)=O 34257,CC1OCCC1(C)C(N1CCC(C(=O)NCC(C2CC(C)(C)C2)O)CC1)=O 34258,C1(C(=O)OCC)CCN(C2CC2)C1=O.c12nnc(o1)s2 34259,C1(CN(C)C(C2(S(N)(=O)=O)CC2)=O)CC(F)CN1C(=O)CSc1nc[nH]n1 34260,c1(SCC)ccccc1CC(=O)N(C)CC1(C)CCCC1NC(=O)C(C)OC 34261,c1(C(N(CC(C)NC(C(CNC(C)=O)(C)C)=O)C)=O)cc2sccc2cn1 34262,c1(NCC2CC(C)OC(C)C2)[nH]c(=NCC2(n3ccnn3)CC2)nc2sccc12 34263,c1(C(=O)NCC(c2ccccc2)NC(c2onc(C)n2)=O)ccc(O)nn1 34264,c1(C(N(CC(CC)NC(C(CC)CC2CCCC2)=O)C)=O)ncc2ccccn12 34265,C(N=c1ccnc(CN2CCN(Cc3cn(C)nc3OC)CC2)[nH]1)C1CC(=C)C1 34266,c1(CN(C(C2CCCN(C(c3coc(C)n3)=O)C2)=O)CC)ccc(O)cc1 34267,N1(C(C#C)C)CCCN(C(=O)Nc2ccc(SC)c(SC)c2)CC1 34268,c1(OC)cc(NC(c2ccnn2C)(c2nnnn2C2CCCC2)C)sn1 34269,N1(C(CC(C)(C)O)=O)CC2(CC(C(=O)Nc3ccc(F)c(F)c3)CO2)C1 34270,c1(C(N2CC(O)(CNC(C34CC(F)(C3)C4)=O)C2)=O)cccc(F)c1O 34271,C(=O)(CC(C)CC(F)(F)F)NC(C)CCNC(c1cc2cc(Cl)ccn2n1)=O 34272,C1(CNC(C(CC)C)=O)CCCCN1C(c1cccc(-c2ccoc2)c1)=O 34273,N1(C(c2c(C)cccn2)=O)CC(C)CN(C(c2ccc(F)c(N)c2F)=O)C(C)C1 34274,N12CCCC(C)(C1)C2=O.c1(C(CNC)O)ccccc1.C1(CC)(CN)CC1 34275,c1(C(C)C(=O)NC2CCC(NC(C3(F)CC3C)=O)CC2)ccc(S(N)(=O)=O)cc1 34276,c1(C(=O)NC(CNC(CC(C)CC(C)(C)C)=O)CO)ccc2c(c1)C(=O)CCO2 34277,C1(NC(COCCC)=O)CN(C(=O)CCc2scnc2C)CCC1F 34278,C1(NC(CCC=C)=O)CN(C(=O)COc2ccon2)CCC1C 34279,C(C(CC(=O)NCC1(CCCO)CC1)NC(=O)C(C)(C)CSC)OC 34280,C(=O)(CCCCN(C(=O)C=Cc1nccs1)C)NC(CC)(C)CO 34281,N1(C(C(CSC)OC)=O)CCCC(C)(C(=O)NC(C)(C)C(O)CO)C1 34282,c1(CC(=O)N(C2CCCN(C(c3cccnc3)=O)CC2)CC)c(F)cncc1Cl 34283,C1(C(=O)NCCCCNC(CN(CC(=O)NC(C)C)C)=O)CCc2nc(C)cn2C1 34284,C(=O)(C(C(CC)CC)OC)NC(CC)CN(C)C(c1cnn(CCC#N)c1C)=O 34285,c1(C(=O)NC2C(NC(C=CCOC)=O)C2)cccc2oc(C)cc12 34286,c1(C(=O)NCC2CCC(NC(c3c(C)ocn3)=O)C2)cnc2c(c1)CCOC2 34287,C1(NC(CC(C(F)F)NC(c2c(C)ccnc2C)=O)=O)CC(C2CCCC2)C1 34288,C1(c2nnnn2C2CCCCC2)(Nc2c(OC)nc(C)cc2)COC2(CCC2)C1 34289,C12(CC=C)CCN(C1)C(=O)C(C)O2.C(=O)(CCC=C(C)C)NCc1ccccc1 34290,c1(C(=O)NC(C(C)(C)OC)C)ccc(CNC(=O)Cn2cc(C#N)cn2)nc1 34291,c1(CN(C(n2c(NCC(=O)OC)ccn2)=O)OCC)cnc(CC)[nH]1 34292,N1(C(C(C2SC(=N)NC2=O)C)=O)CC2OCCN(C(C3CN(C)CCO3)=O)C2C1 34293,C(c1cccc(C)c1)=CC(=O)N(C)CC1N(c2c(C(=O)OC)nccn2)CCC1 34294,N1(C(c2cc(COC)no2)=O)CCN(C(C2CCC(=O)O2)=O)CC2(CC2)C1 34295,C1(NC(c2cc(CC)ncc2)=O)CCN(C(=O)Cc2cncnc2)CC(C)(C)C1 34296,N1(C(CCCCOCCC=C)=O)CC(NC(=O)CSc2cn[nH]c2)CC(C)C1 34297,c1(CN(C)C)nn(C)cc1NC(=O)Nc1ccccc1C(C)(F)F 34298,N1(C(c2nc(COC)oc2)=O)CCC(CC)C1CNC(=O)C=CSC 34299,N1(C(C)=O)CCCOC(CNC(=O)CCOC2CCC2)C1.C12(CC(O)C1)C(=O)N2 34300,N1(C(C(C=C)c2ccccc2)=O)CCN(C(c2cnc(CC)s2)=O)CC1CC1CC1 34301,n1(CC(=O)NCC2(CNC(C3(C)C(C)OCC3)=O)CCC2)nc2c(n1)CCCC2 34302,c1(OC(C)C(=O)NC(C)(C)CO)cccc(C(F)(F)F)c1 34303,CCCCC(C)(F)C(=O)NCC(C)N(C(=O)CN1CCOCC1)C 34304,N1(C(C2(C)COC2)=O)CCC2C(NC(=O)CCSCC(N)=O)C2CC1 34305,N1(C(C(CC)N(CC)CC)=O)CC2CCC(NC(=O)C=CSC(C)(C)C)CC2C1 34306,C1(NC(c2ccc(SC(C)C)cc2)=O)CC2CC1CN2C(=O)CN(C)CCO 34307,c1(CNC(C(CSC)O)=O)ccc(CNC(=O)C(C2CC2)SC)c(F)c1 34308,N1(C(c2c(CC)n[nH]c2)=O)CC2CN(C(c3sccc3COC)=O)CC(C1)O2 34309,c1(C(N(CC(CC)NC(=O)CCNS(C)(=O)=O)CC)=O)cc(SCC)cc(F)c1 34310,C(=O)(C1CCCn2c(C)nnc21)NC(CC)CNC(c1ncncc1F)=O 34311,c1(CC(=O)NCC(CC)NC(=O)COc2ccsn2)csc(C(C)(C)C)n1 34312,CCCCC(CC)(c1nnnn1CC1CCOCC1)NCc1n[nH]c(C)n1 34313,c1(N2CCCC(C)(NC(c3cc(SC)oc3)=O)C2)ccn2ccnc2n1 34314,c1(C(=O)NC2(CCOC)CCN(C(c3cnn(C)c3)=O)C2)cc(C)cnc1C 34315,c1(C(N2C(CC)C(NC(c3cnn(C(C)(C)C)c3)=O)CC2)=O)ccc(=N)[nH]c1Cl 34316,N1(C(=O)C(c2ccccc2)O)CCN(Cc2cnc(C3CC3)nc2)C2CC12 34317,C1(CNC(CC2CC(SC)C2)=O)CCCCC1NC(c1nnccc1C)=O 34318,N1(C(C2(CC=C)CCCCC2)=O)CC2CC(CNC(C3C=CCCC3)=O)C2C1 34319,c1(C(=O)NCCC(=C)CNC(c2ncccc2C)=O)nn(C)nc1Br 34320,C1(CNC(c2n(C(CC)C)nc(C)c2)=O)CCCCN(C(C23CC(C)(C2)C3)=O)C1 34321,c1(CCNC(C2C(NC(C(c3ccccc3)OC)=O)COC2)=O)ccncc1C 34322,C1(Nc2cccc(NC(C(=O)NC3CCC(C#C)C3)=O)c2)CCCCN1N=O 34323,CC(C)CCCCCCC(=O)N1CCC2C(NC(=O)CS(=O)(=O)N(C)C)C2C1 34324,c1(N2CC(C(=O)NC)OCC2)ccc(S(=O)(=O)NCc2csc(Br)n2)c(Cl)c1 34325,C=CC(F)(F)C(=O)N1CC(OC2CCN(C(=O)C(C)N(C)C)CC2)C1 34326,Cc1cc(Cl)cc(C)c1OCC(=O)NC(C)CCCNC(=O)C(C#N)C1CC1 34327,CCC(C)CCC(=O)N(CCCCCNC(C12CCCC1C2(F)F)=O)C 34328,C(=O)(NNC(=O)C(O)c1ccccc1)c1c(C)nc[nH]1 34329,C(=O)(C(CCSCC(C)C)NC(c1cccs1)=O)N1CC(=CCC)C1 34330,CCCCC(C)(c1nnnn1C1COC1)NCc1ccc(OC(F)F)nc1 34331,c1(C(=O)NCC2(C(=O)NOC(c3ncccn3)C)CC(=C)C2)ccncc1OC 34332,N1(C(CSC)=O)CCN(CC2CCCN(C(=O)C(C)CF)C2)CC1 34333,CCC(CNC(=O)C(=O)Nc1cc(Cl)ccc1C(F)(F)F)CC(F)F 34334,C1(C(=O)NCC(C=C)(C)C)CN(C(=O)CCc2ccnn2C)CC1F 34335,N1(C(Cc2c(C)cccc2C)=O)CC(C)(C)CCC1CNC(=O)C(O)C(C)C 34336,c1(CN(C)C(=O)Nc2cc(-c3ccccc3)[nH]n2)noc(C2CCC2)n1 34337,CN1CCOCC(NC(=O)CCOCCNC(=O)CC2CCCN(C)C2)C1 34338,c1(CC)c(C(=O)NC2CCC(NC(c3cc(O)nc(OC)n3)=O)C2)cccc1C 34339,C1(C(N(CCCNC(C=C(C)c2cnn(C)c2)=O)C)=O)CCc2nncn2C1 34340,C1(C)(NC(C=CCOCCOC)=O)CCN(C(=O)CCc2cc(Cl)no2)C1 34341,C1(OC)C2CCN(C(c3cncc(C)n3)=O)C2C1(C)C 34342,C1(NC(C)=O)CCN(C(C2CC(NC(c3ccns3)=O)C2)=O)C1 34343,C1(NC(c2cc(C)c(Br)o2)=O)(CO)CCCN(C(c2nonc2N)=O)C1 34344,c1(CNC(Cn2cc(C(C)OC)nn2)=O)cccc(C#N)c1 34345,C12(C(=O)OC(C)C(=O)n3cccn3)CCN(C1)S(=O)(=O)C2 34346,c1(OC)cc(C)c(C(N2CCC(C)(CNC(C3CCC(=O)N3)=O)C2)=O)c(C)c1 34347,C1(F)(C(N(CCNC(C2(N(C)C)CCCOC2)=O)C2CC2)=O)CC2(CCC2)C1 34348,Cc1ccc(CNc2cc(C(=O)O)c(C)[nH]2)c(N(C)C)c1 34349,N1(C(C2C(CCOC)C2)=O)CCC(C)(C)C1CC(N1CC(S(C)=O)C1)=O 34350,c1(C(N(CCCNC(=O)C=C(C)C)CC)=O)cc(F)c(F)c(O)c1F 34351,c1(C(=O)NC(C(=O)N(CC#C)CC)C2CCCO2)c[nH]c(=NC)s1 34352,c1(C(=O)NCC2(CC(=O)NCC(CCC)C)CC2)c(C)n[nH]c1C 34353,Cc1c(Cl)ccc(C(N2CC(OCCNC(c3sccc3F)=O)C2)=O)c1O 34354,S(=O)(=O)(CC(=O)N1CC(NC(C2CCCN2C(=O)C(C)C)=O)C(C)C1)N(CC)CC 34355,N1(C(C(C(C)C)C)=O)CCC(CNC(=O)C(C)(C)CN2CCN(C)CC2)C(C)C1 34356,c1(SC)c(C(=O)N(C)CC2(O)CN(C(C3C4CC4C4CC34)=O)C2)cnn1C 34357,C(=O)(C(C)(CC)OC)NC1C(C(N(CCC)CCN(C)C)=O)C1(C)C 34358,C(=O)(C(O)CN(C)C)NCCN(C(C)C)C(c1csc(-c2ccccc2)n1)=O 34359,C1(CC(=O)NC(C(C)(C)OC)C)N(C(=O)Cc2cccnc2F)CCC1(C)C 34360,N1(C(CC2(C(=C)F)CCC2)=O)CCC(C2CN(C(C3(C4CCCO4)CC3)=O)C2)CC1 34361,c1(C(=O)NC(C2CCN(C(CNS(NC)(=O)=O)=O)C2)C)cnc(O)c(C)c1 34362,N1(c2snc(-c3c(C)cccc3)n2)CCCN(C2CCN(C(=O)C(C)(C)F)C2)CC1 34363,N1(C(c2cc(OC)n(C)n2)=O)CCN(C(C2CCNC2=O)=O)C(C2CCC2)C1 34364,Cc1ccc(CN2CCC3C2CCCN3S(=O)(=O)c2ccccn2)c([N+](=O)[O-])c1 34365,c1(C(=O)NCC(CO)NC(c2n(CC)ncc2)=O)c(F)cc(C)cc1F 34366,CC(C)CC(F)(F)C(=O)N1CC2CC1CN2C(=O)Cc1c[nH]c2cnccc12 34367,Cc1cnn(C)c1C(=O)N(C)CC1(CNC(C2COCC(C)O2)=O)CC1 34368,c1(C(N(C2CCN(C(c3cc(C)ns3)=O)C2)CCO)=O)nc(=O)n(C)[nH]1 34369,N1(Cc2ncc(-c3cccc(OC)c3)o2)CCC(c2nn[nH]n2)C1(C)C 34370,c1(C(N(CC(=O)NC(C)C(O)C(C)C)CC)=O)ncnc(O)c1F 34371,Cc1ccc(O)c(C(=O)NC(C)(C)CN(C)C(C2CC2(C)C(C)C)=O)n1 34372,C1(NC(c2nccc(SC)n2)=O)CN(C(=O)CC2COCCO2)CCC1C 34373,C1(C)(CNC(C(C=C)OC)=O)CCCN1C(c1cc(C(F)(F)F)nn1CC)=O 34374,CC(C)CCCCCC(=O)NC(C1CCN(C(C2CC(C)N(C)C2)=O)C1)(C)C 34375,c1(C(=O)NCCC(C)N(C(CC2(CC)CCOCC2)=O)C)ccc2cnoc2c1 34376,CC(CN(C)C)CCC(=O)N1CCCC(C(=O)NCC2CC3OC2C2CC32)CC1 34377,C(N=c1nc(C2CCOCC2)[nH]s1)C1CCN(C(C(CCSC)O)=O)C1 34378,c1(C(N(CCN(C(c2cc(C)nnc2O)=O)C)C)=O)c(Cl)ccc2c[nH]nc12 34379,c1(C(C)C)cc(C(=O)NCC(O)CNC(=O)C(F)=C2CCCC2)ccc1Br 34380,C1(CCNC(=O)CCCF)COCCN1C(c1ccc(C(O)C(F)(F)F)cc1)=O 34381,c1(C(=O)NC(C2CN(C(c3ccc(C)cn3)=O)C2)C)n[nH]c2ccc(Br)cc12 34382,c1(C(=O)NCC(CNC(CCC(c2ccc(C)cc2)=O)=O)C)cc(C)cnc1F 34383,C12(C(=O)NCC(CC)NC(C3CCSCC3)=O)CC1COC2(C)C 34384,C12(CNC(c3cc(N(C)C)ncc3)=O)CCC1CN(C(C1CNC(=O)C1)=O)C2 34385,c1(C(=O)NC(CNC(Cc2c(C)nc[nH]2)=O)C)cc([N+](=O)[O-])c[nH]1 34386,CC1(C)CC(C(=O)NC2CCCC(O)C2O)CCN1C(=O)C1=CCSC1 34387,N1(C(C(CC=C)NC(C)=O)=O)CC2CC(C(=O)N(CC(C)O)CCOC)(C2)C1 34388,CCC(CC(=O)NC12CC1CN(C(c1cocc1C)=O)C2)c1ccccc1 34389,c1(NCCC(C)NC(C2CCOC3(CCC3)C2)=O)cc(=O)n2ccccc2n1 34390,N1(C(c2c(OCCOC)nccc2)=O)CC(CNC(=O)C(C)COC)C2(CC2)C1 34391,Cc1cccc2nc(C(=O)NC(C3CN(C(=O)C=Cc4nccs4)C3)C)cn12 34392,N1(C(c2cnc(COC)s2)=O)CCCC(CNC(=O)COCCCF)CC1 34393,C1(C2CCN(C)CC2)(C(=O)NC(C(C)NC(C=Cc2cccc(C)c2)=O)C)CC1 34394,C#CCCCCC(=O)NCCC1CCN(C(=O)CCCCCN(C)C)C1 34395,Cc1cc(CNC(C(N2CC(C(F)(F)F)C(C)C2)=O)=O)ccc1F 34396,c1(NC(CN(C2CC(C#N)C2)C(c2[nH]cc(C)c2)=O)=O)cc(C)ccc1CO 34397,Cc1oc(C(F)(F)F)nc1C(=O)OC(C)Cc1ccc(F)cc1 34398,C1(CNC(c2c(CNC(c3ccc(C)[nH]3)=O)noc2)=O)CCC2(CC2)C1 34399,N1(C(CCC#C)=O)CC(CNC(=O)CCC2CCC2)CCC1C 34400,C(=O)(CS(=O)(=O)CC(C)C)N1C(CC)C(NC(C23CC2COC3(C)C)=O)CC1 34401,c1(C(C(=O)NC(C)(C)C)N(CC(CC)(C)OC)C)c(Br)ccc(C)c1F 34402,C(C(C)(C(C)C)NC(c1ccc(CC)nc1)=O)NC(CC1(CC=C)CCCC1)=O 34403,CC1CC(C)(C)CCC1NCCCN(C=O)CC1CCC(F)(F)CC1 34404,O=CN1CCOCC1C(=O)NCC(CO)NC(=O)Cn1ncccc1=O 34405,c1(OC)cc([N+](=O)[O-])ccc1CCN=C(NCC1CC1C)NCC(C)OC 34406,c1(Cc2onc(C)n2)ccc(Oc2ccc(CNC(C(C)C)=O)cc2)cc1.C(C)(C)O 34407,C12(C(=O)NCc3cn(C4CN(C(CSCC=C)=O)C4)nn3)CCCCC1C2 34408,c1(C(=O)NC2(C)CCN(C(=O)C(O)C3CCCC3)C2)csc2c(O)ccnc12 34409,N1(C(C(CC)C)=O)CC2CC(O)C1C2NC(c1cc(C2CCOCC2)[nH]n1)=O 34410,c1(C(C)C(=O)NCC2(C(C)NC(C3CC(C)(C)C3)=O)CC2)ccc(F)cc1F 34411,N1(C(c2n(CC#C)cnn2)=O)CCC(C#C)(C(=O)NC2CCN3CCC2C3)CC1 34412,C1(NC(Cc2cc(C)on2)=O)COCCN(C(=O)C(C2CC(F)(F)C2)O)C1 34413,N1(C(c2cn(CCC)nc2C)=O)CCC(F)(CNC(=O)Cc2nnc(C)s2)CC1 34414,N1(Cc2cnc(C)n2C)CCC2(CC1)CC2C(=O)NC(CC(=O)O)C(=O)O 34415,C1(F)(CNC(CC2CC(C)C2)=O)CC(NC(=O)CSC(F)F)C1 34416,Cn1nc(C(F)(F)F)c(CN2CCC(F)(C(=O)NCCCO)CC2)c1Cl 34417,CC(CC1CCCCC1)C(=O)NCC(c1ccccc1)C1CCC1 34418,C#CCC(C)(C)C(=O)N1CCN(C)C(CNC(=O)CCC2CCOCC2)C1 34419,c1(OCC(=O)NCCN(C(=O)CC2CCC(=O)O2)C2CC2)ccc(Br)cn1 34420,c1(N2CCCC(C(C)NC(=O)C=CBr)C2)cc(Cl)nc(-c2ccccn2)n1 34421,N1(C(CCC(CC)C)=O)CCCN(C(c2cnccn2)=O)CC1C(C)C 34422,c1(C(=O)NC(C2CN(C(=O)C3=COCC3)CCO2)C)cc(Cl)cc(Br)c1 34423,c1(Nc2nnc(C(=O)OCC)s2)ncnc2c(C)csc12 34424,Cn1cc(C(=O)NCC(C)(C)CC2CN(C(C3CC3c3cccs3)=O)C2)nn1 34425,c1(N2CCN(C(=O)OC(C)(C)C)CC2=O)ccc(F)cc1C1CC1 34426,C1(CC(=O)NC2CN(C(c3c(C)cc[nH]3)=O)C(C)(C)C2)CC2(CCCC2)CO1 34427,C1(F)(C(N2CC(CN(C)C)C2)=O)CN(C(=O)COc2ccn(C)n2)C1 34428,N1(C(CN(C(C(C)C2(O)CCC2)=O)C)=O)CCN(C(C2COCC2(C)C)=O)CC1 34429,c1(CNC(C2(OC)CNC2)C)ncc(C(F)(F)F)[nH]1 34430,c1(C(C)NC(=O)C(=O)NC(CNC(=O)OC(C)(C)C)C(C)C)ncccc1C 34431,c1(C(=O)NC(CNC(CC(CC)SC)=O)C)ccc2c(c1)CCN2C(C)=O 34432,N1(C(CCOCC#C)=O)CCC(CNC(=O)CN(C)C2CC2)C12CC2 34433,C1(N(C)CC2CCCC2)CC2CC1CN2C(c1ccn(C)n1)=O 34434,CCCC(C(=O)N1CCC(NC(=O)CNC(=O)C(C)(C)C)C12CCC2)C(C)C 34435,C1(CCNC(C2(Cl)C(C)(C)C2)=O)CC(F)(F)CN1C(=O)COc1ccc(Cl)cn1 34436,C(=O)(C1=CCC(NC(=O)Cc2ccns2)C1)NC(C)CC(F)(F)F 34437,CC1CN(C(=O)CSCCC(F)(F)F)CC1NC(c1nc(Cl)cs1)=O 34438,N1(C(C(C)n2cccc2)=O)CCC2(CCC(NC(=O)C(F)(F)CC3CC3)C2)CC1 34439,C1(NC(c2cncc(C(N)=O)c2)=O)CCCN1NC(=O)C(C)c1ccsc1 34440,CC1C(NC(C2(C)CCC(=O)NC2)=O)CCCN1c1ccnc(C#N)n1 34441,C(=O)(C(C(C)(C)C)NC(CN(CC(=O)NCC=C)CC)=O)C1C(CC)CCCC1 34442,C(=O)(CCCCC(C)C)N1CC2C(CN3CC(c4ccc(C)nc4)OCC3)C2C1 34443,c1(C(N2CC3C(NC(=O)CC(C4CC4)C4CC4)(CC3)C2)=O)cn2c(n1)CCCC2 34444,C1(NC(CC(=C=C)C)=O)CCC2CCN(C(c3ccc(F)c(C)c3Cl)=O)C1C2 34445,c1(CN2CCCC(NC(c3scc(C)c3)=O)C2)cc(Br)ccc1F 34446,c1(NC(c2cc(-c3cccc(C(C)=O)c3)[nH]n2)=O)ccc(Cl)c(CO)n1 34447,C(CNC(C1(C(N)=O)CCC1)=O)(CCNC(=O)CC1CCCC1C)OC 34448,CC(O)C(F)(F)C(=O)NC1COCCC1NC(c1cc([N+](=O)[O-])n[nH]1)=O 34449,N(C(=NCC1=CCCCC1)NCC1(C#N)CCC1)CC1N(CC)CCC1 34450,C(=O)(C(C)(C)C(C)O)NCCCN(C(COCc1c(C)ncs1)=O)C 34451,N1(C(C(C)OCCC=C)=O)CC(NC(c2nocc2C(C)(C)C)=O)CC1(C)C 34452,N1(C(C(C)C2CC2)=O)CCN(C(=O)CN(C(c2ccco2)=O)C2CC2)CC1 34453,N1(C(CN(C(c2c(CCC)n[nH]c2)=O)C)=O)CC(N(C)C)C(C)C1 34454,Cc1ncc(C(=O)NC(C)(C)C(=O)NCCC2CCCCO2)cc1C#N 34455,C1(CC(=O)NCCCNC(C2C(c3cn(C)nc3)OCC2)=O)NC(=O)NC1=O 34456,c1(C(=O)NCC2(CNC(c3ccc(NC)c(F)c3)=O)CC2)nn(C)cc1[N+](=O)[O-] 34457,C1(CN(C)C(C2CC(C#N)C2)=O)CCCN(C(=O)C(O)CF)C1 34458,N1(C(C2CC(C)(C)N2)=O)CCC(S(=O)(=O)C(F)F)C1 34459,C(=O)(CCC(C)OC(=O)CCc1c(N)cnn1C)OC(C)C 34460,c1(C(=O)OC(C)(C)C)ccc(NNC(=O)NCCCS(C)(=O)=O)c(F)c1 34461,C1(CC)CN(C(=O)COCCF)CCN1C(=O)CC(C(F)F)c1ccccc1F 34462,n1(C(C)C)cncc1C(=O)N(CCCNC(=O)CC1CCCO1)C 34463,N1(CCC2(OC)CN(C(=O)C3=C(Cl)CCOC3)C2)CC(C)OC(C)(C)C1C 34464,C1(O)(CC(N2CC(N(C(C3(C(=O)OC)CC34CC4)=O)CC3CC3)C2)=O)CCCCC1 34465,c1(CNC2CC(OC)C2OC)cnc2ncccn12 34466,N1(C(C(C)(C)C)=O)CCCC(C(=O)NC2CCN(C(=O)Cc3ccoc3)C2)C1 34467,[N-]=[N+]=NC1CCC2(C(=O)NC(CO)CCCCNC(c3cncc(F)c3)=O)CC12 34468,N1(C(c2cc(C(C)C)n(C)n2)=O)CCCC(C2CC2NC(C2CC=CCO2)=O)C1 34469,C1(CNC(C(CC)OC)=O)CN(C(=O)C(CC(C)C)OC(N)=O)CCCO1 34470,c1(C(N2C(CCNC(c3coc(SC)c3)=O)CC(OC)C2)=O)nnc(O)cc1O 34471,C1(C)(CN(C(C(C2CCCC2)OC(=O)CCS(C)=O)=O)C)CCCC1NCC 34472,c1(OCC(=O)NCCC2CCC(NC(=O)C3=CCC3)C2)cccnc1 34473,C=CC(C)(CCOC)C(=O)NCCN(C(=O)C1=COCCO1)CCC 34474,c1(C(=O)NC(C)C(CO)NC(C2CC3CCC(C2)O3)=O)cccc2c1ncn2C 34475,C(C(O)CC(=O)NCC1CC12CC2)NC(=O)CCc1ncccn1 34476,C1(N(C(CC(C)CF)=O)C)CCC2(CC1)CCN(C(c1ccc(F)cc1O)=O)C2 34477,c1(NC(C=CC(C)NC(c2c(C)noc2)=O)=O)ccccc1C(C)C 34478,C1(NC(C2C(C(=O)OC)C2)=O)CCN(C(=O)CC2COCCOC2)C12CCC2 34479,CC1(C)NC(=O)CC1C(N1CCCC(NC(=O)Cc2ccc(F)c(F)c2)CC1)=O 34480,CC(C)CC(CNC(=O)CCCC#N)C(=O)NCCCC1CC1C 34481,CC(C)CC(C(=O)NC(C)CNC(=O)CN1CCN(S(C)(=O)=O)CC1)C(N)=O 34482,C1(N(C(COCC=C)=O)C)CC2CCC(C1)N2C(C1(CC)CCOCC1)=O 34483,N1(CC(=O)NCC(C)N(C)C(c2cc(C(C)(C)C)n[nH]2)=O)CC(=O)N(C)C1=O 34484,c1(OC)ccc(N)c(C(N2CC(C(C)NC(C3C4CCC(F)(F)C34)=O)C2)=O)c1 34485,C1(CNC(C(C2CC2)OC)=O)CN(C(=O)CCN2CCNC(=O)C2)CC(C)(C)O1 34486,c1(C(=O)NCC2C(C)CN(C(C3CCCCO3)=O)C2)cc(Br)c(F)cc1N 34487,CCCN=C(NCc1ccc(F)cc1Cl)NC1CN(C2CC2)CC1C 34488,C1(CCC#C)CCCN1C(=O)C(C1CCN(C(C2CC(=O)C2)=O)C1)C 34489,N1(C(C2CCC(C(C)(C)C)CC2)=O)CCCCCC1CNC(C1CCCSC1)=O 34490,c1(CN(C(C2CCC2NC(C2CCCSC2)=O)=O)CC)ccccn1 34491,CC1(CCO)CCN1C(=O)C(c1ccco1)NC(C1CC(CF)C1)=O 34492,Cn1ncc2ccc(CN3CCCC(C(=O)Nc4cc(C#N)c(Br)cn4)C3)cc12 34493,c1(CC)cc(N)ccc1C(=O)NCCC1CCN(C(C2(C)CCCC2C)=O)CC1 34494,C1(NC(c2coc(C3CCC3)n2)=O)COC2(C1)CN(C(c1cc[nH]n1)=O)C2 34495,C1(C(=O)NCC2CCCN(C(c3cncc(Cl)c3)=O)C2)CC1C1CCCC1 34496,N1(C(=O)CC2(C3CC3)CC2)CCCC(C2CCN(C(C3(F)CCCC3)=O)CC2)C1 34497,C(=O)(C#CC1(C)COC1)NCC1CN(C(Cn2ccc(C)cc2=O)=O)CC1O 34498,N1(C(C2C(OCC)C2)=O)CCC(NC(=O)CCn2cccnc2=O)C(CO)CC1 34499,C1(NC(C(C2(O)CN(C(C(F)=C(C)C)=O)C2)F)=O)C(O)C2CCOC12 34500,c1(OC)cc(OC)cc(CNC(C2CC3CCC2CC3)=O)c1 34501,C12(CNC(c3cc(CC)n(C)n3)=O)CC(CO1)N(C(=O)C(C)CO)C2 34502,C(=O)(CCCC(C)CC)NC1(C(N2CCCCC(CCC)C2)=O)CCOCC1 34503,c1(C(N2CCC(O)(C(C)NC(=O)CC3CC(F)C3)C2)=O)n[nH]c2c1CCC2 34504,c1(C(N(C)CCN(C)C(C2CCCS(=O)(=O)C2)=O)=O)cncc2n[nH]cc12 34505,C=Cn1nccc1C(=O)NC1CC(OCC(=O)NCCCc2cnc[nH]2)C1 34506,C1(C#CC(=O)NCC(C(C)(C)C)NC(c2conc2C)=O)(CC)CC1 34507,C1(C2CC2)(NC(CCNC(c2nn(C)c(O)c2)=O)=O)CCOC1 34508,c1(OC)cc(NC2CC(CNC(=O)C(C)CCOC)C2)ccc1[N+](=O)[O-] 34509,CCC(CC(=O)NC1(CCC(=O)NCc2cn(C)cn2)CCCC1)C(C)C 34510,N1(C(C(C)O)=O)CCC(n2cc(C(=O)N(CCC(F)(F)F)CC(N)=O)nn2)CC1 34511,C1(OCc2cn(C(C)C)nn2)CCCN(C(=O)CC2CCCC(O)C2)C1 34512,C=CC1CN(C(c2ncsc2C)=O)CC1NC(=O)C(C)(C)C1CC1 34513,C1(NC(C(c2c(C)ccnc2)(C)C)=O)CC2(C1)CC(CNC(C1CC1(F)Cl)=O)C2 34514,CC1(C2CC2C(N2CCC(C(=O)Nc3ccc(O)c(F)c3)C(O)C2)=O)COC1 34515,n1(C2(N3CC(CN=[N+]=[N-])C3)CC2)cc(C2CC2)nn1 34516,C(=O)(CC(CC)CCCC)NC(CC#C)CC(=O)NCC1(C)CC(C)=NO1 34517,CCC(CC(=O)NCC1(C(N)=O)CN(C(=O)C(C)n2ccnc2)C1)c1cn[nH]c1 34518,Cc1nn2cc(C(N3CCC(N(C(=O)C(c4ccccc4F)C)C)C3)=O)nc2s1 34519,N1(CC(N2CCC(NC(=O)CC3CCSCC3)C2)=O)C(=O)CNC1=O 34520,N1(C(c2c(SC)nccn2)=O)CCC2(CCC(NC(c3nccn3C)=O)CC2)C1 34521,CC1C(NC(=O)C(CCN(C)C)NC(c2ncccc2N)=O)CCCN1C 34522,n1(CCC)cc(CN2CCC2(C)C(=O)NC(C2CCCC2)C)cn1 34523,C1(CC)CCC(C(N2CCC2CC(=O)NCC(C)O)=O)CC1 34524,C(=O)(C1=Cc2ccccc2C1C)NC(C)CCCNC(=O)C1=C(Cl)CC1 34525,Cc1ccc(C(N2CC=CC(NC(=O)C(c3ccccc3)O)C2)=O)cc1F 34526,Cc1ccc(Cl)cc1NC(=O)C(N1CCOC(CCC(=O)OC(C)(C)C)C1)=O 34527,N1(C(c2cc(C)ncn2)=O)CCC(CO)C(NC(c2ccc(C(N)=O)cn2)=O)C1 34528,C(=O)(C1=CS(=O)(=O)CCC1)N1CCC(C(C)NC(=O)C(C)CF)CC1 34529,c1(C(=O)OC)cc(Cl)c(NC(=O)CSc2c(F)cc(F)cc2F)c(Cl)c1 34530,c1(CC(N2CCCC(CNC(CCc3ncc(C)[nH]3)=O)C2)=O)ccc(F)cc1F 34531,N1(CCC)CCSC(C(=O)N(CC)CC2CCCCC2)C1 34532,C1(C(N2CC(C(C(N3CCC3(C)C(C)C)=O)OC)C2)=O)CCC(F)C1 34533,N1(C(c2cc(C3CC3)no2)C(=O)NCC(C)C)CCN(C)c2ccccc21 34534,c1(NC(CC=CCNC(C2C(C)(C(F)F)C2)=O)=O)cnc2ccccc2c1 34535,C1(C(=O)NCCCOCCN(C)C(C2CC23CCC3)=O)CCCN(S(N)(=O)=O)C1 34536,N1(C(Cc2cn(CC)nc2)=O)CCCC(C)C1CNC(=O)Cc1c(C)cnn1C 34537,c1(C(=O)NC2(CNC(=O)CCF)CCC2)cc(Cl)c2c(c1)OCCCO2 34538,N#Cc1ccnc(NC2CC(CC(=O)NCc3ccccc3F)C2)n1 34539,c1(-n2cc(-c3ccc(N)cn3)nn2)cccc2c1C(=O)NC2=O.Cc1oncc1N 34540,C=CCC(CNC(C1CCC(=O)N1)=O)C(=O)N1C2CCC1CC2 34541,c1(CC(N2CC(NC(C=CS(C)=O)=O)CC2(C)C)=O)ccc(Br)cc1C#N 34542,CCCCC(C(=O)NCCCCCNC(c1ccnc2ccsc12)=O)C(C)C 34543,N(C(=NCCC1OCCO1)NCC(F)F)C(c1ccccc1)C 34544,C(=O)(CC(O)CCCCC)N1CCC(=C)CC1C(N1CC(CC(=O)OCC)C1)=O 34545,C(C)(CS(C)(=O)=O)(C(=O)NC(c1c(C)nn(C)c1N)=O)OC 34546,Cc1cc2ccc(C(=O)NC3(C4CCN(C(=O)CNS(C)(=O)=O)C4)CC3)cn2c1 34547,C1(NC(Cc2c(C)ccs2)=O)CCCN(C(c2ccccc2C(C)(F)F)=O)C1C 34548,C1(NC(C2N(CC)CC2)=O)CCSC12CN(C(C1CCN(CC3CC3)CC1)=O)C2 34549,c1(CC(=O)NC2CC(NC(C(C3CC3)SC)=O)C(O)C2)ccc(O)c(C)c1 34550,N1(C(c2c(C)ccs2)=O)CCC2CN(C(=O)CN(C3CCCC3)C)CCC12 34551,Cc1cc(NC(C2CN(C(=O)C(c3cncnc3)C)CC2(F)F)=O)c(C)cc1O 34552,C1(NC(=O)C=CCN2CCOCC2)CC2(C1)CN(C(C1CCC3(CCC3)C1)=O)C2 34553,N1(C(c2sc(NC)nc2C)=O)CCc2c(ccc(NC(=O)C=O)c2F)C1.CCO 34554,c1(C(=O)NCCCC(C)NC(C2CN3CCC2CC3)=O)nn(C)c2c1CCCC2 34555,c1(-c2nc(-c3cc(CC)oc3C)on2)cn2cc(Cl)ccc2n1 34556,C(=O)(CC(F)(F)CC)NC(CCC)CNC(C1(C(=O)OCC)CCC1)=O 34557,Cc1cnc(N)c(C(N2CCCC2CN(C)C(C2CCC3(CCC3)O2)=O)=O)c1 34558,Cc1nn2cc(C(=O)NC3(CCNC(=O)Cc4csc(S)n4)CCCC3)nc2s1 34559,C#Cc1cccc(C(N2CCN(C(c3cc(C)nnc3O)=O)C(CC)C2)=O)c1Cl 34560,N1(C(C(CC)(C)C)=O)CC2CCCC(C1)N2C(=O)Cc1cccc2c1CCC2 34561,c1(N2CCC(CNC(C(CC)(C)CC)=O)C2)nc(C)nc(C)c1C 34562,N1(C(C(CC)n2cncn2)=O)CC2CCC1CN2C(c1cccnc1)C 34563,c1(C(=O)NCC2C(CNC(c3nc(CCCC)sc3)=O)C2)cc(COC)ncn1 34564,c1(OC)ccccc1C(=O)NCC(C(C)C)NC(c1cnn(C(F)(F)F)c1)=O 34565,N1(C(=O)OC(C)(C)C)CC2CCCN(CCc3cccc(F)c3Cl)C2C1 34566,c1(COCCC(=O)N(C2CCN(C(C3CSC3)=O)CC2)CCC)ccc(F)cc1 34567,C(=O)(C(C)(C)CCC#N)NCC1(F)CC(NC(c2c(C)nco2)=O)C1 34568,CCC(O)C(F)(F)C(=O)OCC1CC1C(F)F 34569,Cc1ocnc1CC(=O)N(CCCCCNC(=O)CC(C)n1cccc1)C 34570,C(CCCC(C)NC(=O)CCCc1ccsc1)NC(C1C(C(C)=O)COC1)=O 34571,c1(CC(=O)NC2CCCC(CN=c3[nH]nc(O)s3)C2)cccc(Cl)c1Cl 34572,c1(CCNC(C(C)Oc2ccc(Br)cn2)=O)cccc(S(N)(=O)=O)c1 34573,C1(NC(C)=O)CCCCC12CCN(C(c1cc3c(Cl)cc(F)cc3[nH]1)=O)C2 34574,c1(NC(=O)NC)ccc(C(=O)NCCC2CCC(NC(=O)CCSC)C2)cc1 34575,c1(SCC)cc(C)ccc1NC(=O)C(=O)NC1(C(C)OC)CC1 34576,n1(CCC(=O)NC2CC(C)(NC(C(CCC)NC(C)=O)=O)C2)cnc(C)cc1=O 34577,N1(C(c2ncn(CC)n2)=O)CCC2CC12C(=O)NCCCc1c[nH]nc1C 34578,C1(C(=O)NCCOC2CN(C(CC3(C=C)CC3)=O)C2)CCS(=O)(=O)C(C)C1 34579,N1(C(C23CC(OC)C2C3)=O)CC(NC(c2cc(C(C)C)on2)=O)C(O)C1 34580,CC(=O)CCN=C(NCCCCCN(C)C)N1CCC(C2CC2)C1 34581,N1(Cc2c(-c3c(OCCC)cccn3)cn(C)n2)C2CCCC1CC(N(C)C)C2 34582,c1(OC)cc(C)c(C)cc1C(=O)NCC1CC(NCc2ccc(SC)o2)C1 34583,CC(C)(CCNC(C1CCC1F)=O)NC(=O)COC1CCCC1 34584,Cc1cc(NC(c2nnnn2C)(C2CC=CCC2)C)cc(C2CC2)c1.c1(C)ccco1 34585,C1(C2CCN(C=O)CC2)(NC(c2coc(Cl)n2)=O)CC1.c1(C2CCC2)cn[nH]n1 34586,C1(CCOCCC(=O)NC(C)CN(C)C)CCCNC1 34587,N1(C(CCOCCOC)=O)CC(O)CC1C(=O)NC1CCC(NC(C)=O)CC1 34588,c1(C(N2C(C)CC2C(=O)NC2CCCCC2)=O)ccn2cncc2c1 34589,c1(C(=O)NCC2CCN(C(C(Br)=C(C)C)=O)CC2C)ccc2nc(O)oc2c1 34590,N1(C(C(=O)NCCCC(=O)OCC)C2(CCC(O)CO)CC2)CCOC(CC)C1 34591,C1(CC(=O)NCC2C(NC(C3CN(S(CC)(=O)=O)C3)=O)C2)CCC(F)(F)CC1 34592,CC(C)CC(F)C(=O)N(CCCCCNC(c1nn(C)cc1Br)=O)C 34593,Cn1cnc(C(N2CCCCC2CNC(C2CCCC2(F)F)=O)=O)cc1=O 34594,C12(NC(c3ccc(O)nc3)=O)CCCC1N(C(c1ccc3nccn3c1)=O)CC2 34595,N1(C(CCCC)=O)CCOCCC1C(N1CCC(OC2CC2)C1)=O 34596,CC1CN(C(C2CCOC(C)(C)C2)=O)CCN1C(=O)CC1CCCOCC1 34597,c1(NC(C2(OC)CCN(C(c3cocc3C)=O)C2)=O)ccc(O)c(Cl)c1 34598,C(=O)(C(CCC1OCCO1)C(=O)NC1CC2CCC1O2)OC(C)(C)C 34599,c1(CNC(Cn2cc(CN(CC=C)CC=C)nn2)=O)ccc2[nH]ncc2c1 34600,C1(NC(CC2CC(=C)C2)=O)CC2CCC1(NC(=O)CN1CC3CC3C1)C2 34601,Cn1ncc(=NC(=O)C2CC23CCN(Cc2ccc(C(=O)O)s2)C3)[nH]1 34602,c1(C(N(C2CCCC(NC(C3CC(F)C3)=O)C2)C)=O)c(F)c(F)c(F)c(F)c1F 34603,N1(C(C(c2ccccc2)N(C)C)=O)CCC2(CCCC2NC(C23CC2C3)=O)CC1 34604,Cc1cnc2cc(C(N3CCCC3C(C)NC(=O)CC(F)(F)F)=O)nn2c1 34605,N1(C(C2(COC)CCCC2)=O)CCC(C2CC2)(NC(=O)C(O)C2CCCC2)C1 34606,C1(C2(O)CCOC2)(C(N(C)CC2CCN(C(c3ccc(C4CC4)o3)=O)C2)=O)CC1 34607,C1(NC(C2C(CNC(c3cc(C)n(C)n3)=O)C2)=O)CC(C2CCC2)C1 34608,C1(NC(COC(C)C)=O)CC2CN(C(C3CC(Cl)(Cl)C3)=O)CC2C1 34609,C1(NC(c2c(C)noc2)=O)CC2CCC1N2C(=O)C=CC1CCC1 34610,C=CCC(CC(C)C)C(=O)NCc1ccc(C(=O)NC(C)C(C)n2cccn2)o1 34611,N1(C(C(C(C)C)CN(C)C)=O)CCN(C(=O)CCCC(N)=O)C2(CCC2)C1 34612,CC(CC(=O)N1CCC(C(=O)NCC(C)(C)N2CCCC2)O1)N(C)C 34613,C1(NC(CCN(C(C)=O)C)=O)CCN(C(=O)CC2CC3(COC3)C2)C1C 34614,C1(NC(c2c(CC)cno2)=O)CCCCC1NC(=O)C(c1ccnn1C)OC 34615,c1(CC)oc2ccccc2c1C(N1CC(CNC(=O)C(C)CSC)C(F)(F)C1)=O 34616,CC(COC(=N)O)N=c1[nH]c(=NC(C)c2cc[nH]n2)[nH]c2ncn(C)c12 34617,Cc1nc(CC(=O)N(C)CC2(O)CN(C(C3(NC(N)=O)CC3)=O)C2)co1 34618,C(=O)(CCCCBr)NCC(C)NC(c1c(C)nn[nH]1)=O 34619,c1(OCCC(C)NC(=O)Nc2nn(C)cc2-c2cn[nH]c2)cccc(F)c1 34620,CCCC(C)CC(=O)NCC1(O)CCCN(C(=O)CCc2nc(CCC)no2)C1 34621,c1(NC(=O)Cc2ncc(-c3ccc(Br)cc3)[nH]2)ccc(F)c([N+](=O)[O-])c1 34622,c1(C(N(C)CCNC(C2CS(=O)(=O)CC(=O)N2)=O)=O)cccc2cnnc(O)c12 34623,Cc1sc(Cl)nc1C(=O)NCCCCCCNC(C1(C)COCCO1)=O 34624,c1(C(=O)N(c2nc(SC)nc(C)c2)C2CC2)cc(=O)n(CCO)c(O)n1 34625,C1(CC(=O)N(CCCN(C(=O)CC=C(C)C)CCC)C2CC2)CCC(C)C1 34626,c1(C(=O)NCCCCCN(C(=O)CC2CC2(C)C)C)cnn2c(Cl)cccc12 34627,Cc1cc(C(N2CC(NC(C3CCOCC34CCC4)=O)C(C)C2)=O)cc(C)c1Cl 34628,CC1CN(C(=O)CSS(C)(=O)=O)CC1NC(=O)CCCc1ccsc1 34629,n1(CC)cc(Cl)c(C(=O)NC2CCC2NC(c2cnc[nH]2)=O)n1 34630,N1(C(C2C(C)C2)=O)CCCC(C)(CNC(C2CC(=O)N(c3ccccc3)C2)=O)C1 34631,N1(C(c2cc(CCC)[nH]n2)=O)CCN(C(C2CCC(=O)N2)=O)CC1C(C)(C)C 34632,S(=O)(=O)(c1c[nH]c2nc(Cl)ccc12)NCC1CCC(CC)C1 34633,C1(CNC(CCNC(=O)OCC)=O)CC2(CCC2)CN1C(C1CC1(Cl)Cl)=O 34634,C1(CCC(=O)NC(C(C)C)=O)CC(C(=O)OC(C)(C)C)CO1 34635,O=S(=O)(c1ccncc1)N(C1C2CCC1CNC2)C1CCCCC1(F)F 34636,CC(CS(C)(=O)=O)C(=O)N1CC2CC(NC(c3ccc(N(C)C)nc3)=O)C(C2)C1 34637,C1(CNC(c2ccc(C(C)(C)C)[nH]2)=O)CN(C(C2CCC3CC23)=O)CCC1(F)F 34638,CC(CCC(C)(C)C)N=c1[nH]c(=N)[nH]c(=NCCc2cn(C)nn2)[nH]1 34639,Cc1c(C(=O)NCC(O)CNC(=O)CC2CC3(CC3)C2)sc2nccn12 34640,c1(CC(=O)NC(CC)(C)CNC(=O)Cc2cccs2)ccc2scc(C)c2c1 34641,c1(CCC)nnc(S)n1CC(=O)NC1CCCC(CNC(=O)C(O)CCSC)C1 34642,CC(C)CC(C)(CNC(C1(OC2CCOCC2)CC1)=O)NC(=O)CC1(C#N)CC1 34643,C=CCC(C)(C)CNC(=NCc1ccnn1C)NCc1ccsc1Br 34644,OC1COCCN(c2nnc(C3CCCCO3)n2CC2CCCC2)C1 34645,c1(CCC(=O)NCCOCCCN(C(=O)C(=O)C(C)(C)C)C)cc(Cl)cc(Cl)c1 34646,CC1CC2(CCN(C(c3cc(CNC(=O)C(=O)NC4CC4)cs3)=O)C2)CO1 34647,N#Cc1ccc(CC(=O)NCC2CCN(C(=O)CCN3CCCC3)C2)cc1 34648,C(c1ccc(F)cc1)=CC(=O)NCC1CC(F)(CNC(C2(F)CC2(Cl)Cl)=O)C1 34649,c1(C(CCC(N2CCC(N3CCOCC3)C2)=O)O)ccc(Br)cc1.c12cn(nn1)C2 34650,N1(CCOCC)CCN(C2CCN(C(=O)CC(N)C3CCCC3)C2)CC1 34651,C1(CN(C(C(n2ccc(C(F)(F)F)n2)C)=O)C)CC(F)CN1C(c1ccco1)=O 34652,CCC(CC)(CN=c1c(C)c[nH]cc1[N+](=O)[O-])NC(C1CC(=O)N1)=O 34653,N1(C(C2C(C(C)C)C2)=O)CCC2(CCC(CNC(=O)Cn3ncnn3)O2)CC1 34654,CN(C)N=Nc1ccccc1NC(c1csc(-c2ccc([N+](=O)[O-])cc2)n1)=O 34655,C1(N(C)C)CCCN(C(=O)C(C)(N)C(F)F)CC1 34656,N1(CCc2ccc(OC)c(Cn3cccn3)c2)CCOCC12CCC2 34657,C1(C(=O)NC(C2CCN(C(Cc3ncc(C)o3)=O)CC2)C)CCCC(C)(C)C1 34658,C(=O)(C1=CC2CCCCC12)N(CC(CN(C(Cc1c(OC)cccc1)=O)C)O)C 34659,c1(C(=O)NCC2(NC(c3ccc(O)nc3)=O)CCC2)cccc2c1OCO2 34660,Cc1c[nH]c(C(=O)NCC(C)(C2CC2)NC(c2cnc(C(N)=O)s2)=O)c1 34661,Clc1ccc(CNc2cnn(C3CCC3)n2)c(I)c1 34662,N1(C(C2CCC(COC)C2)=O)CCN(C(c2cnc(C)s2)=O)CC(O)C1 34663,C(C(C(=O)N(CCO)C(C)C)n1cc(CCCC(N)=O)nn1)OCC.OC 34664,CC1CCN(C(=O)Cc2nc(=N)[nH][nH]2)C1CNC(c1cscc1C1CC1)=O 34665,C12(C(N3C(C)CC(NC(=O)CC4(CO)CC4)CC3)=O)CCCCC1CCCC2 34666,C#CC1CC2CCC1N(C(C1CC(O)CN1C(=O)CC(F)(F)C(F)F)=O)C2 34667,c1(C(C(C)(C)C)N(C(=O)NCCC2(OC)CCC2)CC2CC2)cccc(C)c1 34668,c1(C(N2CCC(F)(CNC(c3ncn(CC)n3)=O)CC2)=O)cc[nH]c2nccc1-2 34669,c1(C(N2CCC(O)(c3onc(C)n3)C2)=O)nc(C(F)(F)F)ccc1Br 34670,n1(CC(=O)NCC2(O)CCCN(C)C2)cnc2ccc(F)cc2c1=O 34671,c1(N2C(NC(c3nn(C)cc3Br)c3n(CC=C)nnn3)CCC2)nnc(C)n1C 34672,C(CCOCCO)(C(=O)N(C(C(N)=O)C1CC1)C)NC(C=CCC)=O 34673,C1(CCN(C)C)(C(C2CCCC2)C)CCCC1.C(C(C)(C)CO)N 34674,CCC(CC)(CNC(=O)C(=O)NC1CC(C)N(C(C)=O)C1)OC(=O)OC(C)(C)C 34675,Cn1c(Br)cnc1NC(N1CCN(c2ccc(Cl)nn2)CC1)=O 34676,c1(OC)ccc2c(c1)CCC2(C)CNc1nc(OC)ccc1Cl 34677,C(=O)(C#CC1CCCCC1)N1CC2C(NC(=O)COc3ccc(Cl)c(F)c3)(C2)C1 34678,c1(OCC)ccccc1C(=O)NC(C)CCCNC(c1cscc1CC)=O 34679,Cn1cc(C(N2CCC(O)(CNC(C3CCC(=O)N3)=O)C2)=O)c2cc(F)ccc12 34680,Cc1cc(C(=O)NC2CC23CC(NC(=O)CSc2cccs2)C3)c(C)n1C 34681,C#CC1CCC(NC(c2csc(CNC(c3ccc(CO)cc3)=O)c2)=O)C1 34682,N1(C(C(N2C(CC)CCC2)=O)=O)CCOCC1CN(C(=O)Cc1ccsc1)C 34683,C(=O)(CCC(=O)NN(C)C)NC1C(CO)CCN(C(COCCCC)=O)C1 34684,c1(C(=O)NCC23CC2CN(C(C2CC=CC2)=O)C3)cccc2cccn12 34685,c1(C(=O)NCC(C(C)C)NC(C2(F)CC2C)=O)ccc(SC(F)(F)F)nc1 34686,N1(C(C2COC(C)(C)O2)=O)CC(NC(C2(F)CCOCC2)=O)CC2(CC2)C1 34687,C1(NC(CC(=C)C)=O)C(C)CN(C(=O)CN2CCCCCC2)CC1C 34688,c1(CC(C)NC(=O)C(N)=O)ccccc1CNC(=O)CC1(O)CCOC1 34689,N1(C(C(C)(C)OC)=O)CCCC2C1CCN2Cc1cc(Br)ccc1Br 34690,c1(CC(=O)NCC2C(NC(C(CC)O)=O)CC2)c(C)nn(CC(C)C)c1C 34691,CC(C)C(CC(=O)N(C1CC(CO)C1)C)NC(C1CC2CC(=O)C1O2)=O 34692,C(CCC(C)C(=O)NCC1(C(=O)NOCCCO)CCOC1)OC 34693,c1(C(N2C(CNC(C3CC34CCCC4)=O)CC(O)C2)=O)cnn2c1CCC2 34694,CC1(C(=O)NC2CN(C(c3ccc(SC(F)(F)F)s3)=O)CC2O)CC=CCC1 34695,C1(CC2(NC(c3c(C)nns3)=O)CC2)CNCCOC1 34696,C1(NC(CCCC=C)=O)CN(C(=O)CCCCC(C)(C)C)C2(CCCOC2)C1 34697,c1(CC)nc(C(N2CC(NC(C3CC(F)(CO)C3)=O)C2)=O)c(C)o1 34698,C(C)(C(=O)NC1(C)CCC(C2OCCO2)CC1)(C(C)C)OC 34699,c1(C(=O)NC2CC(CNC(CCSCCCC)=O)C2(C)C)cc(Cl)ncc1F 34700,N1(C(c2c(NC(CCOCCOCC)=O)c[nH]n2)=O)CCOC(C)(COC)C1 34701,c1(C(N(C2CCN(C(C3CC34CC4)=O)CC2)CC#CC)=O)ncncc1Cl 34702,c1(C(N2CCC(NC(=O)CCC3CC3)C23CC3)=O)ccc2cnnc(O)c2c1 34703,C(CC(C(=O)NCc1cncs1)NC(=O)C=CC(F)F)=CC 34704,c1(C(N2CC(NC(c3c(C)nn[nH]3)=O)C3C2C3)=O)cnc(N)c(N)c1 34705,Cc1ccc(CNC2CC3(C2)CC(C(=O)NCc2ccc(C#N)cc2)C3)c(O)c1 34706,N1(C(CC(C)SC)=O)C2COCC1CC(NC(=O)C(C)=NOCC#N)C2 34707,c1(CSCC(=O)NC(C(C)NC(C(C)CN(C)C)=O)CO)nnc(S)n1C 34708,C1(CCC)CN(C(C2CC2(C)C(F)F)=O)CC1C(=O)NC1CCC(O)CC1 34709,c1(OC)ccc(CC(=O)NCCC2CCCN2C(C2CC2(F)F)=O)cc1 34710,C(=O)(C(O)C(C)(C)CC)N1CC(NC(CCC=CC)=O)C2(C1)CC2 34711,C1(C(N2CCN(C)C(CNC(c3cccc(Cl)c3)=O)C2)=O)CCc2n[nH]cc2C1 34712,C1(C(C)NC(c2cc(Cl)c[nH]2)=O)CCCCN1C(=O)CCCc1ccccc1 34713,N1(C(C(c2nc(C)sc2)=O)=O)CCOC(C)(CNC(=O)CCCc2cnn[nH]2)C1 34714,c1(C(=O)NC(c2c(C(=O)NC3(C(=O)NC)CCC3)con2)C)cc(O)nc(C)n1 34715,CN=S(C)(=O)c1cccc(CNC2CCN(C(=O)OC(C)(C)C)CCC2CO)c1 34716,C#Cc1ccc(C(=O)NC2CC(CNC(c3cn(CCCC)nc3C)=O)C2)cn1 34717,c1(C(N2CCC3CN(C(=O)CCc4cc[nH]n4)CC32)=O)ccc2nc(S)oc2c1 34718,CC1(C)OCCOC1CC(=O)NCCOCCCNC(=O)CC1OCCCO1 34719,C12(NC(C(=C)F)=O)CCC(NC(=O)Nc3nnc(-c4ccc(Cl)cc4)s3)(CC1)C2 34720,N1(CCc2c(C=C)cccc2)C(=O)CN(CC2CCC3CC23)C1=O 34721,C1(CCNC(C2C(C)C2)=O)CCCN(C(c2cocn2)=O)C1 34722,C1(c2n(C)nc(Br)n2)C2CCC(C2)CN1Cc1cn(C2CCOC2)nn1 34723,Cn1cnc(CNc2cccc(OCC3CCCCC3)c2)cc1=O 34724,c1(CNC2(C(c3ccccc3Cl)O)CCCC2)c(Cl)ccc(Br)c1F 34725,c1(NCC2(F)CC(NC(CCc3onc(C)n3)=O)C2)cc(=O)n(C(C)C)c(O)n1 34726,C1(CC(=O)NCC(C)(C2CCC2)NC(c2cc[n+]([O-])cc2)=O)CCC(=O)CC1 34727,C1(C2CCN(C(=O)C(F)=CC3CC3)C2)(NC(c2n[nH]c(C)c2Br)=O)CC1 34728,c1(C(=O)NCC2(OC)CN(C(C3(CC)CCCCO3)=O)C2)ccc(C)cc1Cl 34729,c1(CN(CCC(=O)OCC)C(=O)NCCCCCC)ccc(C)cc1OC 34730,C(=O)(C(CCC(C)C)N(C)CC)N1CCC(NCc2ccc(CC)cc2)C1 34731,N(C(=NCCC(=O)N(C)C)N1CCCC(CC(N)=O)C1)CC(C)C(F)F 34732,C#CCCC(=O)N(CCC(C)(C)NC(C1CC(N(C)C)C1)=O)CCO 34733,c1(OC)ccc(S(=O)(=O)NCC2(F)CCCN(C(=O)C(C(C)C)OC)C2)cn1 34734,C(CC(C(=O)NC(c1nc(C)no1)CO)NC(=O)CCCc1ncco1)OC 34735,c1(CC(=O)NCC(C)NC(CC(c2cccc(OC)c2)C)=O)ccc(F)c(C)c1 34736,CC(C(=O)NCc1ccc(CNC(=O)C=CCN2CCCC2)cc1F)S(N)(=O)=O 34737,C12(C(NOC(c3ccc([N+](=O)[O-])cc3)C)=O)CCOC1CS(=O)(=O)C2.N1(C(C)C)CCNCC1 34738,N1(C(C(CC#C)(C)C)=O)CC2CCC1C(CNC(C1(c3ccn(C)n3)CC1)=O)C2 34739,N1(C(CCCNC(C2CC3(CC3)CO2)=O)=O)CCCC(F)(CO)C1 34740,c1(C(=O)NC(CC(C)NC(c2c(C#C)c[nH]n2)=O)C)noc2c1CCCC2 34741,Cc1nc(O)nc(O)c1CC(N1CCCC(CNC(C2(C(N)=O)CCC2)=O)C1)=O 34742,c1(C(C)=O)ncc(C(N2CCCC2CNC(=O)CC23CCCC2C3)=O)s1 34743,NC1CC2(CCC2)Oc2ccccc21.N=c1[nH]nc(-c2nn[nH]n2)[nH]1 34744,C1(C(N2CC(C(C)O)C2)=O)CN(C(=O)CCc2cncs2)CC2(CCC2)C1 34745,c1(C(=O)NCCCNC(C(c2ccc(F)cc2)C)=O)nccc(C#N)c1F 34746,c1(CC(=O)N(C2CCCCC2NC(C2CC(F)C2)=O)C)c[nH]c2cc(Cl)ccc12 34747,c1(OC)ccccc1OC(C1CCCN(CC2(C)CC2)C1)=O 34748,CCCCCCCCC(F)C(=O)OCC.C(=O)(C1CCCc2nncn21)N 34749,c1(CNc2cccc(NC(CCCCCC#N)=O)c2)ccc2c(O)nncc2c1 34750,C=CC(C)CC(=O)NCCOCCOCCNC(C1CCCCO1)=O 34751,N1(C(CCC(C)OC)=O)CCCC(F)(C(=O)NC2CC(C)C2)C1 34752,C1(CC#C)CCCCN1C(C1CCN1C(=O)CC1CCOC1)=O 34753,N1(C(C(CC)(C)F)=O)CCC2(CC1)CN(C(C1CC(=C3CCC3)C1)=O)C2 34754,O=C(C#Cc1ccccc1)NCC1(C(=O)NCc2cccc3c2OCO3)CC1 34755,C(c1ccccc1)=C(C(=O)NCC1C(NC(CCC=C)=O)CCC1)CC 34756,n1(CC)cccc1CCNC(c1nnnn1C1CCOC1)c1cnoc1 34757,c1(C(=O)NC2CC(NC(C(C(C)O)(C)C)=O)C2)nnc2n1CCCCC2 34758,Cc1coc(C(C)(C)C)c1C(N1CC(N(C(=O)C(F)C2CCOC2)C)C1)=O 34759,c1(C(N(C(C)CNC(=O)Cc2ccc(Cl)nc2)C)=O)cc(Cl)c(F)c(Cl)c1 34760,N1(C(C2(C)N(C(c3c(CC)noc3)=O)CCC2)=O)CCc2ncncc2C1 34761,C1(C(N(CC(C)NC(=O)CCc2cnc[nH]2)C)=O)CC2(C1)C(F)(F)C21CC1 34762,C(CO)(CC(F)(F)F)NC(C(c1n(C)ncc1)NC(C1OCCC1(C)C)=O)=O 34763,C(=O)(CC1=CCN(C(C23CCC(OC)C2C3)=O)CC1)NCC(C#C)OC 34764,C1(C(C)NC(C2CCCCN2S(C)(=O)=O)=O)CCCN(C(c2coc(Cl)c2)=O)C1 34765,N(C1CCOc2ccc(Cl)cc21)Cc1ccc(F)cc1Nc1ncc(C)cn1 34766,N1(C(c2c(C(C)C)sc(Cl)n2)=O)Cc2nccn2CC(NC(=O)CC(C)O)C1 34767,C#Cc1ccc(CNC(c2coc(CNC(=O)Cc3ccsn3)c2)=O)cc1 34768,N1(C(c2c(C)scc2)=O)CCN(C(=O)CSc2ccccc2)CC1CC1CC1 34769,CC(C)S(=O)(=O)CCCN1CCC(NC(C2CN3CCN2C(C)C3)=O)C(O)C1 34770,CC(C)(Cc1cccc(Cl)c1)C(=O)N1CCN(Cc2nc[nH]c2C(F)(F)F)CC1 34771,c1(COC)cc(C(N2CCC2CNC(c2ccccn2)=O)=O)on1 34772,c1(SC(C(=O)NCC(CNC(C2(CC(C)C)CCC2)=O)(C)C)C)ccc(Cl)cc1 34773,S(=O)(=O)(c1ccncc1)NC1CCN(C(C2CCC(OC)CC2)=O)CC1F 34774,CC1c2c[nH]nc2CCC1C(N1CCC(CNC(=O)CC2=CCCC2)C1(C)C)=O 34775,N1(C(C(CCC)NC(N)=O)=O)CCN(CC(=O)NCC2CC2)CC1C 34776,c1(C(=O)NC(C)C(=O)NC(c2nc[nH]n2)CO)cc[nH]c2nccc1-2 34777,c1(C(=O)NC2C(NC(c3cc(C)nc(C)n3)=O)CCCC2)ccc([N+](=O)[O-])n1C 34778,C1(C(N2CCN(C(CSCC#C)=O)C(CF)C2)=O)OCC2COCCC12 34779,c1(C(=O)NCC(CC)NC(c2snnc2C)=O)cccc2cnsc12 34780,C1(CNC(c2ncc(NC)nc2)=O)CCN(C(C2CC(=O)C23CCC3)=O)CC1C 34781,Cc1ccc(C(=O)NCC2CCN(C(C34CCC3C4)=O)C2)cc1 34782,c1(C(=O)NC(CC)CN(C)C(c2cc(C)nnc2O)=O)nccn2cc(C)nc12 34783,N1(C(c2n(CC)ccn2)=O)CCC(C(C)C(N2CCCC(CO)C2)=O)CC1 34784,C1(C(N2CCN(CCN(C(=O)CC3CCC3)C)CC2)=O)CCCC12OCCO2 34785,C1(CC(C)NC(C(=O)N(CCC(=O)NCC2CC2)CC)=O)CCCCC1 34786,N1(C(CNC(CC)=O)=O)CC(NC(=O)Cc2ccccc2C)CCC1C 34787,N1(CCC(C(C)C)(C)C)CCCC2CCN(C(=O)OC(C)(C)C)CC12 34788,C1(CC(=O)NCCCN(C(=O)CCN2CCCC2=O)C)C=CCCC1 34789,C(C(F)(C(=O)N1CC(C)(OC)C1)C(C)C)NC(c1ccc(=NC)[nH]c1)=O 34790,C(=O)(C(CCN(C)C)NC(c1ccc(O)nc1)=O)N1CC(O)(CC)C1 34791,c1(C(C(=O)NS(=O)(=O)C2(c3ccon3)CC2)n2cccn2)ccc(O)cc1 34792,C1(C(N2CC(C)C(NC(C3(C(C)(F)F)CC3)=O)C2)=O)CC1C1CCOCC1 34793,CCC(COC)C(=O)NC1CC(C(=O)NCC(=O)NC2CCC2)C1 34794,c1(CC)nc(C)c(C(=O)NC2CCC(N(C)C(c3cocc3C)=O)C2)o1 34795,N1(C(NOCC(=O)N(C)Cc2cnn(CC(F)(F)F)c2)=O)CCCCC1=O 34796,C(=O)(C(C)CC(=C)C)NC1(CC#C)CCCCC1.c12cc(no1)C(=O)NC2 34797,N1(C(CSC)=O)CCN(C(C2CCCN(C(=O)CC3(C)CC3(Cl)Cl)C2)=O)CC1 34798,Cc1nc(O)nc(C)c1C(=O)NC1COCCN(C(=O)CCC(=O)OC(C)(C)C)C1 34799,c1(CC)nc(C(C)C)ccc1C(=O)NCCCNC(c1ccn(C2CCC2)n1)=O 34800,c1(C(=O)Nc2ccc(O)cc2Br)ccc2ncc(-c3ccc(F)nc3F)n2c1 34801,c1(COCC(=O)NCC(C2CC2)NC(C(C)NC(CC)(C)C)=O)ncc[nH]c1=O 34802,N1(C(c2c(OC)nccc2)=O)CCCC(N(c2cnc(C#N)cn2)C)CC1 34803,c1(C(N(C2CCN(C(C3CC3(F)F)=O)C2)CC)=O)c2c(nn1C)CCC2 34804,c1(C(N2C3CN(C(=O)Cc4cn[nH]c4)C(C3)C2)=O)nc2cnccc2s1 34805,C(CC(C)(C)CC(=O)N1CSCC1C(=O)NCC(C)(C)OCCO)OC 34806,Cc1cncc(C(N)C(=O)NC(C)CC2CCNCC2)c1 34807,C1(C(N2CCC(NC(CC(C=C)CC)=O)C(C)C2)=O)CCC2(CC1)CNC(=O)C2 34808,CC1(C(=O)NC2CC2NC(=O)C(c2ccc(F)cc2)(F)F)CCC(O)CC1 34809,N1(C(COCC)=O)CCN(C(C2CCCCN2C(=O)CC)=O)CC1CCOC 34810,c1(C(N2CC(C=C)C(NC(=O)COc3cn[nH]c3)C2)=O)csc2ccc(F)cc12 34811,C(CCCCC(=O)NC1CCC(C(N)=O)CC1)N(C(=O)C(=O)C1CCCC1)C 34812,Cn1ccc2sc(C(N3CCCCCC(NC(c4csnn4)=O)C3)=O)cc12 34813,C1(OC)CC(NC(=O)C(=O)NCCCC(=O)Nc2ccc(C(F)(F)F)cn2)C1(C)C 34814,c1(OCN=c2n(-c3cccc(C)c3)[nH]nn2)cccc2c1nc(O)n2C 34815,c1(C(N2CC(NC(C3(OC)CCOC3)=O)C(O)C2)=O)c(N)sc(C)c1C 34816,CC1=N[Si](C)(C)CCC1NC1CC(C)(c2ccccc2)C1 34817,c1(CC)c(C(C)NC(c2nn(C)cc2C)=O)oc2ccccc12 34818,C1(NCc2scc(CN(C)C)n2)CCC2(CCCNC2)C1 34819,c1(C(N2CC(C(C)NC(c3cnc(CC)s3)=O)OCC2)=O)cc(O)ccc1N 34820,CC1CN(C(C2CC2c2ccc(Br)cc2)=O)CCN1S(=O)(=O)c1cccs1 34821,C=CCN=C(NCCN(S(C)(=O)=O)C1CC1)N1CC(C(C)C)c2ccccc21 34822,Cc1cccc2nc(C(=O)NC(C)(C)C(C)NC(C3CNC(=O)N3)=O)cn12 34823,c1(C(=O)NC(C(C(C)C)NC(CSCCOC)=O)C)cnc2ncnn2c1O 34824,c1(C(=O)NCC2(O)CN(C(Cc3cc(C)no3)=O)C2)cc(C)c(O)c(N)c1 34825,CCC(CC)C(C)C(=O)N1CCC(C(=O)NC(c2ccnc(C)n2)C)(CF)C1 34826,c1(C(N2CCC(C(C)NC(c3cnsc3)=O)C2)=O)cc(OC(F)F)n(C)n1 34827,C1(C(=O)NCc2c(C)ccs2)C2CC3C(C2NC(=O)C(C)C(F)F)C13 34828,c1(C(=O)NC(C)CCNC(c2cccc(CO)n2)=O)nsc2c(Cl)cccc12 34829,N1(C(c2cnc(C(C)(C)Cl)s2)C(=O)NCCOC)CCCCC1C 34830,Cc1ccc(C(CNC(c2occc2C)=O)NC(c2scc(C)c2C)=O)cc1 34831,O=C1CCCC(C(=O)NCC(CC(=O)N2CCC(CF)CC2)C2CCC2)CC1 34832,C1(NC(Cn2ncc(C#C)c2)=O)CN(C(=O)C(C)CC(C)C)C(C)(C)C1 34833,c1(CC)cnc(C)nc1N1CCC(CNC(=O)CN(C)CCOC)C1 34834,C1(CN(C)C(c2cc(Cl)cn2C)=O)CN(C(c2cc(CO)[nH]n2)=O)CCO1 34835,CC1CCC(C)(C(=O)NCC(=C2CN(C(C3CC4CCC3C4)=O)C2)F)CC1 34836,Cc1c(C)c(C)c(C(=O)NCC2CCCC2NC(=O)CCOC2CC2)c(C)c1C 34837,c1(C(=O)NCC2N(C(CCCC#C)=O)CC2)ccc(NC)c(C(F)(F)F)c1 34838,c1(C(=O)NC(C(=O)NCc2ncc(C)[nH]2)C2CC2)cncc(C#N)c1 34839,Cc1ccc(CC(CO)NC(c2cnc[nH]2)=O)nc1 34840,c1(C(N2CC(C(C)(C)C)N(C(=O)CC3C=CCCC3)CC2)=O)nccn2ccnc12 34841,C1(CC(C)NC(=O)C#CC2CC2)CCN(C(=O)CC23COCC(C2)C3)CC1 34842,C1(NC(C(C)n2ccnc2)=O)CCN(C(c2ccn(O)c(=O)c2)=O)C1(C)C 34843,c1(C(N2CC(C)C(NC(c3csc(O)n3)=O)CC2)=O)cncc2c(O)nccc12 34844,C(CCC(C(=O)NCCc1cccc(C)n1)N(C)C)NC(C1C(=C)C1)=O 34845,n1(CC(=O)N(C2CCN(C(=O)CCCc3nncn3C)C2)CC)cnnc1O 34846,Cc1cc(C(=O)NC2CCC(C)N(C(C3SC4C=CC3CC4)=O)C2)ccc1O 34847,C1(CC)CN(C(c2cc(F)ccc2F)=O)CCN1C(c1cc2[nH]ccc2s1)=O 34848,C1(C(=O)NC(C(C)NC(c2ccnnc2)=O)C2CC2)CC(C)(c2ccccc2)C1 34849,C1(CCC)CCCCC1NC(c1csc(CNC(C2(CO)CCCCC2)=O)c1)=O 34850,CC1(C(N2CCCN(C(=O)CCC3CCCCO3)CC2)=O)COCC1(F)F 34851,c1(N2C(C)(CNC(=O)Cn3cc(CO)nn3)CCC2)ccc2c(n1)CCCC2=O 34852,c1(C(N(CCN(C(=O)C(c2cncn2C)N(C)C)C)C)=O)cnc(C2CCC2)[nH]1 34853,C(=O)(C1=C(Cl)CCCC1)NCC1(COC)CCCN1C(C1CC12CCC2)=O 34854,c1(C(N2CCC(COC)(NC(C3(CF)CC3)=O)C2)=O)cc(Cl)cc(C(F)(F)F)n1 34855,N1(C(C#CC(C)C)=O)CCC(C)(NC(=O)CCc2nnc(O)nc2O)CC1 34856,c1(OC)c(Cl)ccnc1NC(C1CN(Cc2ccc(F)c(F)c2)CCS1)=O 34857,N1(C(C2(C)CC2(Cl)Cl)=O)CCC(O)(Cn2ccnn2)CC1 34858,C(CC(C)(C)Cc1cn(C2CCCN(CCOC)C2)nn1)OC 34859,N1(C(=O)NC(C)C(=O)NC2CCC2)CCN(C2CCC2)C(C)C1 34860,C1(NC(c2ccc(OC)c(O)c2)=O)C2CC(O)C1N(C(c1cscc1F)=O)C2 34861,C1(NCC2C(OCC)CCCC2)CC(C2CCOC2)C1 34862,N1(C(C2(C)CNC(=O)C2)=O)CCCN(CCNC(c2c[nH]nc2C(F)F)=O)CC1 34863,CN1CCC(CC(N2CCCC(CCNC(C3CC3OC(C)(C)C)=O)C2)=O)CC1 34864,C(C(N=[N+]=[N-])C(=O)N1CCC(C)(NC(=O)CC2CCCCC2O)C1)OCC 34865,N1(C(CCC2CC(OC)C2)=O)CC2CC(Nc3ncnc(Cl)c3F)CC1C2 34866,Cc1cc(F)ccc1CC(=O)NC(CNC(=O)CC1CCCC(=O)N1)CC(C)C 34867,C(C(O)C(=O)NOCCN(C)C)NC(c1c(CC)[nH]cc1)=O 34868,c1(C(=O)NC2(C(=O)NC(CC(=O)OCC)C)CCC2)c[n+]([O-])c(C)cn1 34869,C1(C)(CC(=O)NCC=CCNC(C2(c3cccs3)C(C)C2)=O)CCCO1 34870,c1(NC(Cn2c(C)cnc2)=O)cccc(CNC(c2cncc(N)n2)=O)c1 34871,N1(C(c2c(N)cc(Cl)nc2Cl)=O)Cc2nccn2CC(NC(C2(F)CC2)=O)C1 34872,Cc1cc(C(=O)NC2(CC(N3CCC(NC(N)=O)C3)=O)CCCCC2)cc(C)c1N 34873,N1(C(c2nccc(C)c2N)=O)CCOC2CN(C(=O)CC3C=CCCC3)CC12 34874,c1(C(N2C(C)CC(CNC(C(C)=C3CC3)=O)C2)=O)coc(S(C)(=O)=O)c1 34875,CCCCCC(C)CC(=O)NC1CCCC1NC(C1CC2(C1)OCCO2)=O 34876,C(CNC(C1CCC1)=O)(C(C)C(C)C)NC(Cc1c(C)cccc1)=O 34877,C=CC1(C(=O)NCC(C)(C)CNC(c2ccn(C3CC3)c2C)=O)CCCCC1 34878,C1(NC(c2ccc(C3CC3)cn2)=O)C2CCC1N(C(=O)C(C1CCCCC1)O)C2 34879,CC(C(C)(C)CN(C)C)NC(c1cn(CCNC(c2ccn(C3CC3)n2)=O)nn1)=O 34880,CC(C(=O)N1CCN(C(=O)CN(C)CCO)C(c2ccncc2)C1)C(C)(C)C 34881,Cc1cccc(C(N2CCCC2C(N2CCOC(C3(C)CC3)C2)=O)=O)n1 34882,c1(C(=O)NCCCCC(CO)NC(C(C)SCC)=O)ncc2ccccn12 34883,N1(C(C(C(=O)OC)(C)C)=O)CCC2(CC1)OCCC2NC(=O)C=CC1CCCO1 34884,C(=O)(C(C)(C)C(F)F)NC1CNCC(COc2ccc(NC(=O)OCC)cc2)C1 34885,C1(C(C)NC(C2CNC(=O)C2)=O)CN(C(=O)CN2CCCCC2)CCO1 34886,c1(C(N2C(CNC(C3C(C)C3)=O)C=CC2)=O)cn(C)nc1C(C)(F)F 34887,CC(CC(=O)NCC(O)CNC(C1(F)CCCC1)=O)NC(=O)NC1CCCC1 34888,c1(C(=O)NCC(CNC(c2ccc(C(C)C)nc2)=O)(C)O)cc(CO)ccc1Cl 34889,N1(C(CCCOCCC)=O)CCC(NC(c2ccc(OC)cc2C)=O)CC1C 34890,c1(CC)ccc(C(=O)NCC(C)N(C(=O)C(c2ccccc2C)C)C)c(C)n1 34891,N1(C(c2c(CC)occ2C)=O)CC(C(N2CC(CC3CC3)C2CC)=O)CCC1(C)C 34892,C(CNC(C1CC(=O)NC1(C)C)=O)(C(=O)N=c1cc(C)n(CCO)[nH]1)OC 34893,C(=O)(C1=C(C)OCCC1)N1CCC(C(=O)NC(CCC)CC)C1CC 34894,c1(C(=O)NCCNC(c2onc(C)c2C)=O)cccc(C2CC2)c1Cl 34895,C1(C(=O)NC(C2CCN(C)C2)C)(CO)CN(C(C2CCN(S(C)(=O)=O)C2)=O)C1 34896,c1(N(C(=O)CCCCBr)C2CCNCC2F)ncnc2n[nH]c(Br)c12 34897,Cc1cc(C(=O)NCCC2CCCN(C(=O)CC3(C)CCCO3)C2)cc(F)c1C 34898,C#Cc1ccc(C(N2CCCC2CNC(=O)CC(N2CCCCC2=O)C)=O)o1 34899,N1(C(C(C)C(C)(F)F)=O)CC2(CCCC2CNC(=O)C(C2CCOCC2)O)C1 34900,C1(C(=O)NC(C2CN(C(=O)C#CC3CCC3)C2)C)CC2(CCC2=O)C1 34901,CCC(CC(=O)N(C)CCOCCC(N1CC=CC1C(=O)NC)=O)SC 34902,Cc1ccccc1CCC(=O)NC1(CNC(=O)C(C)C#N)CCCC1 34903,CC(C)S(=O)(=O)C(C)C(=O)NCCN(C(=O)CCCCN1CCCC1)C 34904,c1(C(=O)NCCCCNC(=O)C(c2ccccc2)F)cn(C2COC2)nn1 34905,c1(OC)cc(Cl)ncc1C(=O)NC1CCCC1C(=O)Nc1cc(O)ncn1 34906,CC1CC2CN(C(c3cccnc3O)=O)CC2N1C(=O)CCCC1CCCC1 34907,C1(CC(=O)NC(CNC(C(Cc2ccccc2)OC)=O)C)CCC(=O)N1C 34908,N1(C(Cc2cc(C)on2)=O)CCC(C)(CNC(=O)C(C2CCOCC2)C)C1 34909,c1(C(N(C)CC2CCCCN2C(=O)C=CC2CCCC2)=O)ccc2ccnn2c1 34910,CCC(F)(F)CC(=O)NCC1CC1NC(=O)C(c1ccnn1C)O 34911,c1(C(=O)NC2CCCCCC2C(=O)NC2CC(CF)C2)cccn2nccc12 34912,C1(C2CC2)(C(=O)NCC(C)CNC(=O)C(=C2CCCCC2)F)CC=CC1 34913,C(=O)(C(C)(C)C(F)(F)F)N(C(C(=O)Nc1c(Cl)ccc(OC)n1)C)C 34914,c1(C(=O)NCCOC2CN(C(C3CC34CCCOC4)=O)C2)cn2cccnc2n1 34915,CCC(C)(CNC(c1cc(C)c(F)cn1)=O)C(=O)NOCC(O)C(C)C 34916,c1(C(N(C2CN(C(=O)CC3CC3(C)C)C2)C)=O)ccc(OC2CCCC2)c(Cl)c1 34917,C1(CC)(CC)CC(C(=O)NCCCOCCC(=O)NCC2CCCOC2)C1 34918,CCC(C)CCC(=O)N1CCC(NC(=O)C=Cc2cn(C)cn2)C1 34919,N1(C(c2c(CC)ccs2)=O)CC(CNC(c2cnnc(O)c2)=O)CC1(C)C 34920,C1(NC(c2ccc(F)c(Cl)c2)c2n(C(C)C)nnn2)CCCCC1S(C)(=O)=O 34921,c1(COC)ccc(C(=O)N(C(C)CNC(C2(CC#N)COC2)=O)C)o1 34922,N1(C(C2CC(C)(CC)C2)=O)CCC2CN(C(c3[nH]c(O)nc3C)=O)C2C1 34923,Cc1nn(C)c(C)c1CC(=O)NC1CN(C(C2CC2F)=O)CC1C 34924,Cc1nc(=NC(=O)CCNC(c2nnn3c2C(=O)NCC3)=O)o[nH]1 34925,N1(C(CN(CCC)C)=O)CCC1CC(=O)NCCOc1cnsc1 34926,N1(C(Cn2ccc(C)n2)=O)CCC12CN(C(c1nc(O)sc1C)=O)C2 34927,C(C(C)(C)CCC=C)N(C(CCC=CCC)(C)c1nnnn1C1CCOC1)C1CC1 34928,C1(C(N2CCC(O)CC2)=O)CC2(CCN(CCCc3cnc4ccccn34)CC2)C1 34929,N1(C(C(c2ccccc2)OC)=O)CC(NC(=O)C(CC)N2CCCC2=O)C(C)C1 34930,C1(NC(C(COC)O)=O)Cc2ccccc2C1NC(=O)Cc1cc(C)ns1 34931,O=C1CCN(Cc2ccc(N3CCOCC3)nc2)c2cc(Br)ccc2N1 34932,C1(C2CCN(C(=O)CC(C)C(C)(C)C)C2)(NC(CC(C)C)=O)CC1 34933,C=CC(C)(CC)C(=O)NCCC(F)(F)Cn1cc(C2CC23CC3)nn1 34934,c1(C(=O)NCCNC(CCC=CC(C)C)=O)cc(S(N)(=O)=O)c(F)c(F)c1F 34935,c1(C(=O)NC(CCNC(CC2CCC(C#N)C2)=O)(C)C)cc(F)cc([N+](=O)[O-])c1 34936,C1(C2CCN(C(=O)CNC3CC3)CC2)(NC(c2c(C)ccc(F)c2O)=O)CCC1 34937,Cc1nc(Cl)[nH]c(=NCC2CCN(C(c3cnc4ncccn34)=O)C2)c1[N+](=O)[O-] 34938,c1(C(=O)NCC(CC)NC(c2ccc([N+](=O)[O-])s2)=O)cnc2c(c1)c(C)nn2C 34939,C1(C(N2CC3C(NC(=O)Cc4ccsc4Br)(C3)C2)=O)CCCC1C1CC1 34940,Cc1[nH]c(C(=O)Nc2cccc(NC(N)=O)c2)c(C)c1NC(=O)C(C)NC=O 34941,C(=O)(CC(C)(C)OC)N(CCCNC(c1csc(-c2cn[nH]c2)n1)=O)CC 34942,C(=O)(C(O)(c1ccccc1)SC)NCC(CC)NC(=O)C(C)(C)c1ccccc1 34943,Cc1cc(=O)n(CCC(=O)N(C2CCC(NC(=O)CC(C)(C)C)C2)CCO)cn1 34944,CCCC(C(=O)OC)C(=O)N1CC2C(CNC(c3nc(O)nc(O)c3F)=O)C2C1 34945,c1(CC(=O)NCC2C=CC(NC(=O)NC3(c4cccs4)CC3)C2)ccccc1 34946,C1(CNC(C(C#C)(C)C)=O)CN(C(=O)CCn2ccnc2)CC(C)(C)O1 34947,CCCC(C)CCCC(=O)N1CC=C(CNC(=O)C(CC)OC)CC1 34948,C1(C(=O)NCC2CCC(C(=O)N(C)Cc3c[nH]nc3C)CC2)(OC)CCCOC1 34949,N1(C(=O)CC2CCC(F)(F)C2)CCC2CN(C(c3ccc(Cl)cc3Cl)=O)CC2C1 34950,c1(-c2cccc(OC)n2)ccc2oc(C(=O)NCC3(C(F)(F)F)CC3)cc2c1 34951,c1(CC)noc(CC)c1CC(N1CC(NC(=O)CC2CCCCO2)C(O)C1)=O 34952,C1(NC(C=CSC)=O)CCC2CC1CN2C(=O)CC1CCOC(C)(C)C1 34953,Cc1nc(C(C)C)nc(N2CCCC2CNC(c2cn(CCO)nn2)=O)c1Br 34954,C1(NC(C(C2CC2)SC)=O)CCCC1NC(=O)Cn1ccc(Br)n1 34955,CC(C)CC(F)(F)C(=O)N1C2CCC1CC(CNC(C1CC(C)CO1)=O)C2 34956,C#CCC(C)(C(=O)NCC1CC1Cl)NC(c1cc(C#N)cs1)=O 34957,C1(C(N2C(CNC(CNC3CCCC3)=O)CC2)=O)CCc2ncnc(C)c2C1.CO 34958,CCCCCCC(=O)N1CC(NC(c2oncc2C)=O)C(C(F)F)C1 34959,C(C1=CCN(C(C2CC(C)CN(C(=O)Cc3cncs3)C2)=O)CC1)OC 34960,CC1=C(C(=O)N2CC3CCC3(CNC(C3CC3c3cncs3)=O)C2)CCCO1 34961,CC1C(NC(=O)CCC2CCC(C)O2)CCCN1C(c1cn(C)c(=O)n1C)=O 34962,C(=O)(CC1c2ccccc2C(=O)N1C)NCCCCNC(CC1CC(SC)C1)=O 34963,Cc1ccc(C(C)CC(=O)NC2CC(C)N(C(=O)C(C3CCOCC3)C)C2)cc1 34964,S(=O)(=O)(c1ccc(=NCCS(=O)(=O)N2CCCC2)[nH]c1)N1C(CCC)C=CC1 34965,c1(C(N(C(CNC(C(CC)=CCCC)=O)C2CC2)C)=O)cc(Cl)cc(F)c1F 34966,Cc1cc(C(N2CC(C)CCC2CNC(c2cn(C(C)C)nn2)=O)=O)c(C)nc1C 34967,C(C)(C(O)C(=O)OCc1nnc(-c2ccc(C(F)(F)F)cc2)o1)OC 34968,C(=O)(C1=CC(C)CC1)NC(C)CCNC(c1ccn(C2CCC2)n1)=O 34969,C12(C(=O)NC3CCC(C(=O)OC)C3)COC(C1)C(NC(C1CNC(=O)N1)=O)C2 34970,CC1CCN(C(C2(CF)CC2)=O)CC1N(CC(C)C)C.C1(C=O)CCN(C2CC2)CC1 34971,CC1CN(C(c2cnc(Br)s2)=O)CC1NC(C12CC(C#N)(C1)C2)=O 34972,C12(COC)CC(NC(=O)CSS(C)(=O)=O)(CN1C(=O)CCc1cccnc1F)C2 34973,C12(C(=O)NC(COCC(C)C)C(=O)O)CC3CC(C1)CC(O)(C3)C2 34974,CCCC(C(=O)N(CCC(=O)OC)OC)NC(=O)C(CO)C(C)(C)C 34975,c1(C(N2CCC(N(C)C(C3CCCCCCC3)=O)CC2)=O)c2c(nn1C)CCSC2 34976,c1(C(N(c2ncc(CCC)cn2)C2CC(N)C2)=O)cc(C(F)(F)F)ccc1F 34977,c1(CNC(C(C2CN(C(C(C)OCC)=O)C2)OC)=O)cnc(CC(C)C)[nH]1 34978,C1(OC)C=CCN(C(C2(CNC(c3cocc3C(N)=O)=O)CC=CC2)=O)C1 34979,Cc1cnc[nH]c1=NCCCC(C)NC(c1cnn(CCN(C)C)c1)=O 34980,c1(NC2C(C)CCN(C(c3c[nH]c(C(N)=O)c3)=O)C2)ncnc2sccc12 34981,C1(C(=O)NC(CCCCC)C)CN(C(C2(O)CCOCC2)=O)CC12CC2 34982,c1(C2(C(=O)Nc3cccc(CCC)n3)CC2)ccc(F)cc1Br 34983,N1(C(C(C(C)C)SC)=O)CC2(C1)C(NC(=O)Cc1csnn1)CCS2(=O)=O 34984,C=CCC(C)(C)CC(=O)NC1CCCC1NC(=O)C=C(C)C1CC1 34985,CCC(CC(=O)NC(CCOCC)C(=O)N1CCC=C(Br)C1)C1CC1 34986,c1(OC)cc(Cl)cc(N)c1C(=O)NC(c1sc(C(C)(C)SC)nc1C)C 34987,C1(C(N(C)Cc2ccns2)=O)CCC(C2CC2)N1C(c1ccc(C#N)s1)=O 34988,c1(C(N2CCC(C#N)CC2)C(=O)NCc2ccccc2)ccc2ccccc2n1 34989,CCCCCC(O)C(=O)NCc1cc(-c2ccc(C#N)cc2)nn1C 34990,C1(CN(C(=O)Cc2sccc2C)CC)CCCCN1C(=O)CN1CCC(F)(F)C1 34991,c1(C(N2CCC(CCNC(C(C)CC(F)F)=O)C2)=O)cccc2c1CC(=O)N2C 34992,C1(N(C(CC(=O)NCC#C)=O)C)CCN(C(=O)C(C)CSC)CC1 34993,N1(C(C2(CC)CCC2)=O)CC2CC2(CNC(=O)C(C)Sc2ccc(OC)cc2)C1 34994,c1(C(C)C)ccc(C(=O)Nc2cccc(NC(=O)CCC3CNC(=O)N3)c2)cn1 34995,Cc1oc(-c2ccccc2F)nc1C(=O)NCC(O)CN(C)C(c1cncs1)=O 34996,C(=O)(NNC(=O)C1CC1(F)F)N(C1CCCC1c1ccc(Cl)cc1)C 34997,Cc1c(C(=O)NC2CN(C(=O)CC(C)NC(N)=O)CC2F)cnc2ncnn12 34998,N(C1CCCc2c1cnn2C(C)(C)C)Cc1cc(C)cc([N+](=O)[O-])c1 34999,C(=O)(C1CCc2ccc(Br)cc21)NCC(Cn1cc(-c2c(C)ncs2)nn1)(C)C 35000,c1(C(N2C(C(N3CCC(C(C)(C)O)CC3)=O)CC2)=O)cc([N+](=O)[O-])n[nH]1 35001,C1(NC(C2CCC(NC(CCC3C(C)C3)=O)C2)=O)CC2CC1CC21CC1 35002,C(CC(C)C(=O)NCC(O)CNC(c1ccnc(NC(=O)NC2CC2)c1)=O)=CC 35003,C(=O)(CC(C(F)(F)F)N(C)C)N1CCC(F)(C(=O)NC(c2nnc(O)o2)C)C1 35004,O(NC(=O)C(C1CC=CCC1)NC(C1C2CCC(F)C12)=O)CC(C)(C)O 35005,c1(NC(C2C(C(=O)Nc3c(C#N)ccs3)C2)=O)cccnc1[N+](=O)[O-] 35006,N1(C(c2c(C)noc2N)=O)CC2(CCC2NC(=O)Cc2cc(Cl)cc(Cl)c2)C1 35007,c1(N(C2CC(N)C2)C(c2c(F)ccc(Cl)c2Cl)=O)ncnc2cc(Br)sc12 35008,CCCC(C)CCCC(=O)NCC1CN(C(=O)Cc2cc(Cl)n(C)n2)CC1(C)C 35009,CC1CN(C(c2ccncc2F)=O)CC(C)CN1C(C1CC12CCSCC2)=O 35010,Cc1cc(C=CC(N2CC(NC(C3CC3(Cl)Cl)=O)C(C)(C)C2)=O)c[nH]c1=N 35011,C(CN=C(NCC1CC12CC(OC)C2)NC1CCN(C2CC2)CC1)OCC 35012,c1(OC)ccc2ccccc2c1NC(C1CNCCN1Cc1cncs1)=O 35013,C(=O)(CCC(C)(C)[N+](=O)[O-])N1CCC(CNC(C2(CC)CC2(F)F)=O)C12CC2 35014,N1(C(C(COC)OC)=O)CCN(C2CCCN(C(=O)C=C(C)C(C)C)C2)C(=O)C1 35015,C12(C(=O)NCC3CCN(C(c4cccnc4S)=O)C3)CCC(O1)c1ccccc12 35016,C1(NC(CN2CC(CC)C2)=O)CN(C(=O)C(C)Cn2cccn2)CCC1C(F)(F)F 35017,N1(C(CCC(=C)C)=O)CCC(Cn2cc(CC3(O)CCSC3)nn2)C(F)(F)C1 35018,c1(CC)cc(C(=O)NC2CC2CNC(c2cncc(N)n2)=O)cc(O)n1 35019,CCC(C)C(=O)C(=O)NC1COCCC1C(=O)N(CCC(N)=O)CC 35020,N1(C(CNC(C2C(C)C2)=O)=O)CCC(C(=O)N(C2CSC2)C)(CF)C1 35021,c1(C(=O)NCC2C(N(C)C)CN(C(CC3C(CC)C3)=O)C2)c(Cl)ccnc1C 35022,S(=O)(=O)(c1c[nH]c(=NCCC2CC2(Cl)Cl)cc1C)N1CCC(OC(=O)NC)CC1 35023,C12(C(=O)NC3C(OC)CN(C(C(CC=C)C)=O)C3)CC3(F)CC(F)(C1)CC(F)(C2)C3 35024,Cc1cc(C(N2CC(C(=O)NCCN3CCCCC3)C2)=O)cc(C(F)(F)F)c1 35025,c1(C(=O)NC2CCCC(NC)C2)c(F)cc(Cl)cc1Cl 35026,C1(O)(CN(C)C(C2(CF)CC(F)(F)C2)=O)CCCN(C(=O)COCCCF)C1 35027,c1(OC)ccc(F)cc1CC(N1CC(N(C)C(C2CCCC(C)CC2)=O)C1)=O 35028,c1(Cn2cc(CCCCNC(C(C)CCN(C)C)=O)nn2)csc2ccccc12 35029,c1(C(=O)NCCC2N(C(C3CC(C#C)(O)C3)=O)CCSC2)cncc2c1CCC2 35030,N(C1CCOc2ccc(O)cc21)C(c1c(C)cco1)C 35031,Cc1ccc2c(c1)C(=O)N(CC(=O)NCC1COCCN1C(=O)C=CCO)C2=O 35032,N1(C(C2CC(C)OCC2)=O)CC=C(C(=O)Nc2cccc(C#N)c2)C1 35033,c1(C(=O)OC)cccc(C(N2CCCC(CO)(NC(C3(Br)CC3)=O)C2)=O)c1O 35034,N1(C(C(CO)N(C)C)=O)CC(NC(=O)C=Cc2ccccc2)CC1(C)C 35035,N1(C(c2ccc(C(C)C)cc2)=O)CCCC(C)(NC(C2CCC3CC2CO3)=O)C1 35036,CCCCC(O)CC(=O)N1CCC(C)C1C(=O)NOCC(C)(C)O 35037,C1(NC(CC2CC(C)(C)OC2=O)=O)CN(C(c2ccnc(O)c2)=O)C2(CCC2)C1 35038,Cc1noc(CN(C)C(=O)NCc2ccn(CC(F)(F)F)n2)n1 35039,C(CN=c1[nH]c(=NCC(=O)NC(C)C)c2ncccc2[nH]1)C1CC(C)OC(C)C1 35040,C(CCCC(=O)N1CC(O)CC1C)NC(c1c(CCC)[nH]cc1)=O 35041,C1(C(N2C3CC(NC(C(CCC)C)=O)(C3)C2)=O)CC(C(C)C)=NO1 35042,C1(C(N(CC(C)(C)NC(COCCCC(C)C)=O)C)=O)CCCCC1(F)F 35043,N1(C(=O)NC2CN(C(=O)OC)C2)CCC(C(C)(C)C)(Cn2cc(C)cn2)C1 35044,N1(C(c2c(C)cc[nH]2)=O)CCC(CCN(C)C(c2nocc2Br)=O)CC1 35045,c1(OCC)nccc(C(N2CCC2CNC(c2nc(C)ncc2Cl)=O)=O)c1F 35046,CC1(C)OC2(CN=c3ccnc[nH]3)CC1(C(=O)NC1(CO)CCS(=O)(=O)C1)C2 35047,N1(Cc2n(CCC)nnn2)CCC(NC(c2nsnc2O)=O)C(O)C1 35048,C(=O)(CC(C)C(=O)OC)Nc1cc(CC)ncc1.C12(CCCO1)C(=O)NC2 35049,c1(NC(c2c(C(C)C)nns2)=O)ccccc1I 35050,c1(NCCc2ccc(OC)cc2)cc(Cl)nnc1OCc1ccc(C(C)(F)F)cc1 35051,C1(C(=O)NC(CC)CN(C)C(c2ccc(C)cn2)=O)CC(O)CN1C(=O)NC 35052,C1(C)(C(=O)OCC)CCCN1C(=O)CCn1cc(C(=O)OC(C)(C)C)cn1 35053,c1(C(=O)NCC2C3CN(C(C4C(OCC)C4)=O)CC32)c(F)cc(F)cc1Cl 35054,N1(C(C(CSC)(C)C)=O)CCC(CNC(C2CCCC(CF)C2)=O)C(O)C1 35055,c1(C(N(CC(CNC(C(C)SCCCC)=O)C)C)=O)ccc(-n2ccnn2)cc1 35056,c1(C(N2C(CC(=O)NCC(C)C3CC3)C3CCCC32)=O)cc2ccccc2o1 35057,CC1CCC=C1C(=O)N1CCC(C)(C)C1CC(=O)NOCCCF 35058,c1(CC)cccc(NC(=O)NCC2CCCN2C(c2ccsc2SC)=O)c1O 35059,O=C(O)CCC(F)(F)C(=O)N1CC2CC1CN2Cc1ccc(F)cc1 35060,c1(SCC(C)(C)C2CCCO2)cc(Cl)cc(Cl)c1.C1(=O)C(C(=O)N(C)C)N1C 35061,N1(C(CCOCCC)=O)CCCC2CN(C(c3cncc(NCC)c3)=O)CCC12 35062,C=CCC(C)C(=O)NCC1CCCN1C(=O)Cn1ncccc1=O 35063,c1(OC)cc(C(=O)NC(C)CC(C)NC(c2cnn(CCO)c2)=O)ccc1Cl 35064,C1(C(N2CCC(O)(CC)C2)=O)COCCN(C(=O)COCC(=O)NC)C1 35065,C1(C(=O)NC2(C)CCN(C(C(CSC)O)=O)CC2)Cc2ccccc2S1 35066,C1(CN(C(C(C2CCCC2)NC(C(C)=C(C)C)=O)=O)C)C(C)(C)C1(C)C 35067,CC(C(=O)N1CCC(O)(CN(C(=O)C(C)(C)C)C)C1)C(F)F 35068,C(=O)(C(F)(F)C(C)O)NCC(c1cc(F)cc(Cl)c1)NC(Cc1c(C)ncs1)=O 35069,c1(NC(CC2C(C)CCC2)=O)ccc(N2CCC(F)(F)C2)cn1 35070,C=C=C(C)CC(=O)NC1(c2ccccc2)CCN(C(=O)CSCCC)C1 35071,C(CC(C)(C)C(=O)NCC(C)CN1CCOCC1)NC(C=CCC)=O 35072,c1(NC(C2C3CN(C(CCCC(C)C)=O)CC32)=O)cc(Cl)c(Cl)cc1C#N 35073,N1(C(c2nc(CC)oc2)=O)CCC2(NC(=O)CCCc3cc(C)no3)CC2C1 35074,c1(OC)ccc(CNC(=O)Nc2ccnn2-c2c(F)cccc2F)c(O)c1 35075,C1(C(=O)NCCCC2CCCN2C(=O)CN2CCSCC2)CCCCCC1(F)F 35076,N1(C(C2CC(C)SCC2)=O)CCN(C(=O)Cn2cccc2)CC1CO 35077,c1(NCc2csc3ccc(OC)cc32)[nH]c(=NCC2(OC)CC2)nc2ncn(C)c12 35078,c1(OCCCC)c(C(=O)N(CC(C)C)Cc2cnc(C)nc2C)cccc1Br 35079,C(C)(CC(=O)NC1(CCC(=O)NCC(O)CCC2CC2)CCCC1)=C(C)C 35080,Cn1cncc1C1CC1NC(=O)CC1(C)CCN1C(=O)CSCC(F)F 35081,C1(NC(C=C(C)C(C)C)=O)CCN(C(=O)C(C)SC(F)(F)F)C1C1CC1 35082,N1(C(CCN(C(C)=O)C)=O)CCC(CN(C(=O)C(F)(F)c2cnccn2)C)CC1 35083,CN1N=CC(CC(=O)N(CC(CO)(CO)NC(=O)CC2CCCC2)C)C1=O 35084,CCC(CC)CCCC(=O)N1CCC2CN(C(c3nnn4ccccc34)=O)C2C1 35085,N12CCC(C)(CC1)C2=O.c1(CNC(C(C)C(F)F)=O)cc(C(F)(F)F)cc(F)c1 35086,Cc1ccc(CCCC(=O)NC2CCCC2CNC(=O)Cc2csnn2)s1 35087,C12(C)CCC(C1)N(C(=O)C(C)C)C2.C1(N2CC(C(=O)OC)C2)CCCCC1 35088,N1(C(Cc2c(C)nc[nH]2)=O)CCN(C(=O)CCC2OCCO2)CC1c1cn[nH]c1 35089,C(=O)(C1=CS(=O)(=O)CCC1)NC1CN(C(C(C2CC2)OCC)=O)CC1(C)C 35090,CCC(C)CC(C)C(=O)NC(c1cccnc1)C(=O)NCCN1CCNC1=O 35091,c1(CC(=O)Oc2cc(C3CCC3)ccc2Br)noc2ccc(Cl)cc12 35092,N1(C(CCC(N)=O)=O)CCCC1C1CCCN1C(=O)Cc1nnc(O)s1 35093,C1(CNC(C(N2CC(C)C2)C)=O)(CNC(C2(C)CCSCC2)=O)CC12CCC2 35094,c1(C(=O)NCC2(OC)CN(C(c3cc(C)ncc3C)=O)C2)ccn(O)c(=O)c1 35095,C1(C)(C(=O)NC2CCC(NC(c3ccc(CC)[nH]3)=O)C2)CCC(C)(C)CC1 35096,C(=O)(C(CO)C(C)(C)C)NCc1c(C(=O)NCC(C(=O)NC)(C)C)occ1 35097,C1(NC(c2c(CC)n[nH]c2)=O)CCCN(C(=O)C(C2CCC(=O)N2)C)CC1 35098,c1(C(C(=O)OC(C)(C)C)N(C)C)ccc(Br)cc1.c12cn(nn1)CC(=O)N2 35099,O=C(CCCNC(c1cccnc1)=O)NCC1CN(C(c2cc(Cl)c[nH]2)=O)C1 35100,c1(CN(C)C)c[nH]c(C(=O)NC2CC2NC(=O)COCC2CCCO2)c1 35101,N1(C(C2(COCC)CC2)=O)CC(C2CCCCN(C(=O)CC3COCCO3)C2)C1 35102,c1(C(=O)NCCC2CC(NC(c3cn(CCC)nc3C)=O)C2)nnc(O)cc1O 35103,N1(Cc2c(C)n(C)nc2)CC2(CN(C(c3ccc(Br)cc3CO)=O)CCO2)C1 35104,C(=O)(CCCCC(=O)NC1CN(C(=O)CSc2nnnn2C)CC(C)(C)C1)NC 35105,N1(C(CC(C)F)=O)CCC2(CC(NC(c3ccc(CCN(C)C)cc3)=O)CO2)C1 35106,N1(C(Cn2c(C)ccn2)=O)CCC(O)(CN(C)C(C2(C)CCCC2C)=O)CC1 35107,CC(C)CCCNC(=O)CCc1cccs1.C1C(C)CC(=O)N1C 35108,N1(C(C(C)(C)NC(=O)NCC)=O)CC(NC(c2nnccc2C)=O)C(C)(C)C1 35109,C12(C(=O)NCCN(C(C3(CC#C)CCOC3)=O)C(C)C)CC(CO)(C1)OC2C 35110,O=C(CCCC(F)(F)F)NC1CC(O)CN(C(=O)COC2CCOC2)C1 35111,c1(NC(C2CC3(C2)CC3F)=O)oc2ccccc2c1C(=O)NC(COCC)CC 35112,c1(OC)ccc2cccnc2c1CN(C=O)C(c1cccs1)C1CC1.c1ccncc1 35113,c1(C(C(=O)NCCC#N)N(CC)CC2CCCO2)nc2c(s1)CC(C)CC2 35114,CCCCCCC(C)C(=O)NC(C(=O)NC1CC(F)(F)C1(C)C)C(C)C 35115,C12(C(N(CCC(=O)NC(CC=C)C3CC3)C)=O)COCC1C2 35116,N1(C(c2noc(CNc3ccnc(SC)c3)n2)=O)CCCCC1Cc1ccccc1 35117,C1(CNC(C2CC(OC)C2)=O)COCC1NC(=O)CCOc1cccnc1 35118,CN=c1ccc(C(=O)NCC2CCN(C(=O)C(C)(C)c3csc(C)c3)CC2)c[nH]1 35119,c1(OC)cc(CC(N2CCCC(C)(NC(=O)CCCC3CC3)C2)=O)ccc1C 35120,c1(C(N2CC(CC=C)(NC(c3ncc[nH]3)=O)C2)=O)cnn(C(C)C)c1C 35121,N1(C(c2cccc(Cl)c2)=O)CC(C2CCCN(C(C3CCCCS3)=O)C2)C1 35122,c1(C(=O)NC(Cn2c(CC)ncc2)C)ccc(Br)cc1N=[N+]=[N-] 35123,c1(CN(C(C2C(C)C2)=O)C)ccc(CO)cc1 35124,C1(F)(C(=O)OC)CN(C(=O)CONC(c2cccnc2)=O)C1 35125,N1(C(C(CC)OCC)=O)CC(N=c2nc(C(C)(C)C)[nH]s2)CC(C)(C)C1 35126,N1(C(Cc2c(C)nsc2)=O)CCCC2(NC(=O)COCCCC(C)C)CCCC12 35127,N1(C(C2N(C(C)=O)CC(O)C2)=O)CC(NC(=O)Cc2[nH]cnc2C)CC(C)C1 35128,N1(C(COCC=C)=O)CC2CCC(C1CO)N2C(c1ccc2c(n1)CCCC2)=O 35129,c1(C(N2CCC(NC(C(C)OCCCC)=O)C2)=O)ncccc1C(F)F 35130,C1(CNC(C(C(=C)Cl)(C)C)=O)C(C2CC2)CCN1C(c1ccc(Cl)cc1)=O 35131,C12(NC(=O)COC3CC(F)(F)C3)CCN(C(c3cccc(O)c3Cl)=O)CC1C2 35132,C#CCCC(C(=O)NCC(C)C#N)NC(=O)CCCCCN(C)C 35133,n1(CC)cnc2[nH]c(=NCCCN=c3cc[nH]cc3)[nH]c(=NC(C)c3ccco3)c12 35134,C1(NC(CC(C(C)C)C)=O)CCCC12CCN(C(=O)C(C)CS(C)(=O)=O)CC2 35135,c1(C(=O)OCC2CC2)ccc(Br)c(CC(N2CC(=O)NCC2C(F)F)=O)c1 35136,O=S(=O)(c1cccc(F)c1F)N1CC2CN(Cc3cccnc3Cl)CC2C1 35137,c1(C(=O)ON2CC(C(C(=O)NC3C(C)CCC3)O)C2)c[nH]nc1[N+](=O)[O-] 35138,N1(C(c2cnc(COC)s2)=O)CCN(C(=O)CC2CN(C)C2)C(C)CC1C 35139,N1(C(C=C(CC)CC)=O)CC2(CC2)CC1CNC(=O)C(C)SC(C)C 35140,C(=O)(C(C)(C)CCOC)NC1CCCC(NC(C2(COC)CC(=C)C2)=O)C1 35141,Cn1ccc(C(N2CC(C(=O)NCCCCCCF)CC2(C)C)=O)cc1=O 35142,C1(CC(N2CC(NC(c3c(C)nn(C)c3)=O)C(C(F)F)C2)=O)CCOCC1(C)C 35143,CC1(C)CC(O)(C(=O)NCCCNC(C2CC2C2CCCO2)=O)C1 35144,C1(C(=O)NCc2cc(C(=O)N(C)CC3CCN(C)C3)n[nH]2)(OC)CCC(C)C1 35145,Cc1cc(F)c(C(N2CC3CN(C(=O)C(n4ccnc4C)C)CC23)=O)c(F)c1 35146,Cn1nc(C(=O)NC2CCCC2NC(C2CCC3CC23)=O)c2c1CCC(C)(C)C2 35147,N1(C(C(CC)C)=O)CC2CCC(C(=O)NCCc3ncn(C)n3)(C2)C1 35148,Cc1nccc(C(=O)NCC2(NC(=O)CNC(C3CCCCC3)=O)CCOC2)c1N 35149,N1(C(Cc2ccc(C)o2)=O)C2CCC1CC(CC(C)NC(=O)C(C)CCO)C2 35150,c1(CC(=O)NC2CN(C(CC(c3c(C)n[nH]c3C)C)=O)C2)c(F)cccc1Cl 35151,S(C1CCc2c(F)cccc21)C(c1cccc(NC(N)=O)c1)=O 35152,C1(C(N2CCC3CN(C(C4CC4OC)=O)CC3C2)=O)CC2(CCC(CO)CC2)C1 35153,C(CC(C(=O)N1CCC(NC(=O)OCC)C1)NC(=O)Cc1cn[nH]c1)=CC 35154,CCCCCC(C)CC(=O)NC(CNC(=O)CN1C(=O)C(C)C(C)C1=O)C(C)C 35155,CCC(C)C(O)C(C)C(=O)NC(C)CCC(=O)NCCc1ccccn1 35156,CCC(C)(C)C(C)CC(=O)NC1(CNC(=O)C=Cc2cc(Cl)ccc2Cl)CCC1 35157,C1(CNC(C2CCC(CC)O2)=O)CC(NC(c2cnc[nH]2)=O)CC1O 35158,N1(C(=O)CN2CCCC2)CC2CN(C(c3cccc4cc[nH]c34)=O)CC2C1 35159,N1(C(CC(COC)C)=O)CCCCC(CNC(=O)C=C2CCC(C)(C)CC2)C1 35160,N1(C(c2c(C)cccc2F)=O)CC(NC(=O)Cc2ccon2)CC2(CC2)C1 35161,CCCCCCC(F)C(=O)N(CCCNC(=O)C(C(C)C)Oc1ccccn1)C 35162,c1(C(=O)NCC2N(C)CCN(C(=O)C=C3CC3)C2)cnn2ccn(C)c12 35163,C=CCCCCC(=O)N1CC(CC(F)C(=O)NCc2ccc(C)o2)C1 35164,C=CCC(CC)C(=O)N(C)CCOCCN(C)C(c1cnc(N(C)C)o1)=O 35165,c1(C(C)C)cc(C(F)(F)F)ccc1Nc1n[nH]c(-c2ccccc2)n1 35166,Cn1nccc1C(=O)NCCC(O)CNC(c1c[nH]c(Br)c1)=O 35167,CC1CCN(CCC(=O)NCCCCCCNC(c2ccnc(OCF)c2)=O)CC1 35168,CCC(CCCC(=O)N1CCCCC1CCO)NC(=O)C(C)(C)SC 35169,Cc1nn(C)c(C)c1Cn1cc(CCNc2nccc(OC(C)C)c2F)nn1 35170,N(C(=S)N1CC(C(c2ccccc2)=O)CC(C)C1)CCc1ccc(C)c(C)c1 35171,CC(C)CC(CNC(=O)C1=CCCCO1)C(=O)NC(C1(O)CCCC1)(C)C 35172,S(=O)(=O)(c1cc(C(=O)NCCNC2(C(C)C)CC2)ccc1Cl)NC(C)C 35173,c1(CC(N2CC(CCNC(COCCOCC#C)=O)C2)=O)nc(C)c(C)s1 35174,C1(C(N(CCNC(=O)C(C)(CC)C(F)F)CC)=O)CCc2ncnc(C)c2C1 35175,C1(C(=O)NCCCOCCC(=O)N(CCC#C)CCOC)C(C)(C)C1(F)F 35176,C(C1=NOC2COCC12)SCC(C(=O)N1CCCC1)NC(=O)CCCC1CC1 35177,CC1CCC(CNC(=O)Cc2cc[nH]c2)N(C(=O)CN2CCC(CO)CC2)C1 35178,c1(OCCC(=O)NCCN(C)C(C2CC3(C2)CC3F)=O)cccc(F)c1 35179,c1(C(=O)OCC)cc(C(=O)NCC2CC2CNC(=O)Cc2ccco2)n(C)n1 35180,C12(C(=O)NC3C=CCN(C(COC4(C)CCCC4)=O)C3)CCCN(CC1)C2 35181,c1(C(N2CC3(CCN3C(C3(F)CCCCC3)=O)C2)=O)ccc(Cl)c(F)c1F 35182,c1(OCCCN(C(=O)C(=O)NCCC(F)(F)F)CC)ccc(Br)cc1 35183,C1(CC(N2CC(C3CC3)C2CO)=O)CN(C(=O)Cc2cc[nH]c2)CC12CC2 35184,N1(C(c2cc(C)ncc2)=O)CC2CN(C(=O)CCc3ccc(Cl)cc3F)C2C1 35185,N1(C(C(CO)N(C)C)=O)CCC2(C1)CN(C(=O)CS(=O)(=O)C(C)(C)C)CCO2 35186,N1(C(C(CC)(C)OC)=O)CC2=C(C1)CN(C(c1cnc(C(C)(C)C)[nH]1)=O)C2 35187,c1(C(=O)NC(c2ncc[nH]2)CC)cc(CNC(=O)Cc2csnc2C)[nH]n1 35188,N1(Cc2c(OC)cco2)CCCC(NC(c2cnc(Cl)cc2I)=O)CC1 35189,C(=O)(C(C)(C)CC(F)F)NCc1c(C(=O)NCC(C#C)OC)con1 35190,c1(C2(C(=O)NC(C3CCN(Cc4ccccn4)C3)C)CC2)ccccn1 35191,C(=O)(C(O)C(F)(F)F)N1CCC(CC2N(C(C=C(C)C)=O)CCC2)CC1 35192,c1(NC2CCN(C(C=C(C)Cl)=O)CC23CCC3)ncnc2cccc(C)c12 35193,c1(C(N2C(CNC(CSCC)=O)CC(C)CC2)=O)n[nH]c2cc(C)ccc12 35194,N1(C(C2(COC)CCC2)=O)CC2CCC1C2NC(=O)CCc1ccc(Cl)cc1 35195,C1(CNC(C(c2ccc(F)cc2)OC)=O)CN(C(c2ccc[nH]2)=O)C(C)(C)C1 35196,CC1CN(C(=O)CC23CCC(CC2)C3)C(C)CN1C(C1(N2CCOCC2)CC1)=O 35197,C(C1OCc2ccccc21)N(C)C.n12nnnc1C(=O)NC1CC2C1 35198,C1(NC(CCCCOC)=O)CC2(C1)CN(C(=O)CC1C(C(=O)OC)C1(C)C)C2 35199,c1(OC)ccc(C)nc1C(=O)NC1CC1CNC(c1ccc(C(C)C)cc1C)=O 35200,C1(NC(C2C(C)CCS2)=O)CCC(NC(=O)C(C)(C)c2ccc(Cl)s2)CC1 35201,c1(NC(C2(C)CCN2C(c2c(O)cccc2O)=O)=O)cccc2sccc12 35202,N1(C(c2c(CC)[nH]cc2)=O)CCCC(NC(c2csc(S(N)(=O)=O)c2)=O)C(F)C1 35203,N1(C(C(C(CC)C)O)=O)CCCC2(C1)CN(C(c1nc(O)c(C)s1)=O)CCO2 35204,c1(COC)cc[nH]c1C(=O)NC1(CNC(=O)C(C)NC(C2CCC2)=O)CCCC1 35205,C(c1cccc(F)c1)=C1CCN(Cc2c(CSC)cccn2)CC1 35206,c1(C2C(C(N3CCCC3Cc3cn(Cc4cscn4)nn3)=O)C2)sccc1Cl 35207,N1(C(C(c2ccc(Cl)s2)C)=O)CCC(NC(=O)Cc2ccc(O)c(Cl)c2)CC1C 35208,Cc1cc(C)n(CC(=O)NCCC2COCCN2C(=O)C(C2CCCCC2)O)n1 35209,c1(CCN=C(NC2CC(SC)C2)NCCc2cccs2)ccc(S(N)(=O)=O)cc1 35210,c1(C(N2CC3(CN(C(c4ccc(C)s4)=O)C3)C2)=O)cc(N)cc(C)c1F 35211,c1(-c2onc(CCCOc3ccc(Br)cc3)n2)cccc2ncsc12 35212,CCC(C(=O)NCC1CC(C)CN(C(=O)C(n2nccc2C)C)C1)C(F)(F)F 35213,CN1CCN(C(C2CC(O)CN2C(=O)C(F)C(C)(F)F)=O)CC12CCC2 35214,N1(c2c(C(=O)OCC)cnc(SC)n2)CCC2(CC(NC(=O)COC)C2)C1 35215,C1(C(N(C(CO)C2CC2)C)=O)CC12CCN(C(=O)CCC1(C)N=N1)C2 35216,c1(C(C)(C)C)nnc(N(C(=O)NC(C2CN(C3CCOCC3)C2)=O)CC2CC2)s1 35217,C1(=O)C(CC(N)=O)N1.Cc1nonc1CC(=O)NC(C)(C)COC1CCCCC1 35218,c1(OCC)ccc(C(c2cccs2)NC(CCO)CC(C)C)cc1OCC 35219,C(N=c1cc(C(C)(F)F)nc[nH]1)C1(CNCC=C(C)C(C)(C)C)CC1 35220,C(=O)(CCCCN(C)C)NCC1C(NC(COC(C)=O)=O)CCC1 35221,CCCC(C(O)C(=O)NCC1CCC=CO1)NC(c1n[nH]c2c1CCC2)=O 35222,N1(C(c2nc(CC)[nH]n2)=O)CC(NC(C2(C(F)(F)F)CC2)=O)CC1C 35223,N1(C(C(CC)C#N)=O)CC(O)(C2CCN(C(=O)Cc3cn4ccsc4n3)CC2)C1 35224,CC(C)S(=O)(=O)CC(=O)NC1CC(N(C)C(c2cnoc2C2CC2)=O)C1 35225,N1(C(CN2CCC(=O)CC2)=O)CCOCC(NC(c2ccn(CCF)n2)=O)C1 35226,c1(C(N2CC3C(N(C(C(C)NC(N)=O)=O)C)C3C2)=O)cc2cc(F)ccc2o1 35227,C(C)(C)(CCCC(=O)NC(C(C)C)C1CC1)NC(c1ccc(OC)cc1)=O 35228,c1(NC(C2C3CN(C(C4CCC(C)CO4)=O)CC32)=O)nc2cc(F)ccc2s1 35229,C1(CC)CCCCCCN1C(C1CCOCCN1C(c1cc(CO)ccn1)=O)=O 35230,N1(Cc2cncc(OC)c2)CC2CC(C1)N(C(=O)CC1CC=CCC1)C2 35231,C1(C(=O)NCc2nocc2C(=O)NCc2cccc(F)c2)CCCCC1O 35232,C12(CNC(C3(C)COCCO3)=O)CCC1CN(C(c1cc3occc3[nH]1)=O)C2 35233,C12(NC(C3CNC(=O)N3)=O)CCC(C1)N(C(=O)CCCCNC(N)=O)C2 35234,c1(C(CNC(=O)CCn2cccn2)NC(C(C)NC(=O)NC)=O)ccccn1 35235,C(CC(=O)NCCC1CN(C(c2nc(Br)c[nH]2)=O)C1)(C(F)(F)F)OC 35236,Cc1cc(C(=O)NCCN(C(=O)C(c2ccc(Cl)cc2)C)C)c(C)[nH]1 35237,C1(C(=O)NCC2(C(C)C)CC2)C2CC3C(C2NC(C2(C(N)=O)CC2)=O)C13 35238,N1(CC(=O)NC(C)CN(C(=O)CCc2cscc2Br)C)CCCCCC1 35239,N1(C(c2c(C)nc(CC)o2)=O)CCC(NC(=O)C(C)NC(=O)NC)C(CO)CC1 35240,c1(CC(=O)NC(C(C)C)CCN(C)C(C2CC(C)(C)C2)=O)ccccc1[N+](=O)[O-] 35241,Cc1cc(Br)ccc1CC(=O)NCC1CC2CC2N1C(=O)CNC(=O)CC#N 35242,c1(N(C)C)ccc(C(N2CCC2CNC(c2cnc(Cl)cc2N)=O)=O)c(F)c1 35243,c1(NC(C2CC(F)CN2C(=O)Cc2c(F)cccc2F)=O)cccc2c1OCO2 35244,c1(C(=O)NC(CC(C)NC(C2CC(CC)C2)=O)C)ccnc(C(F)F)c1 35245,c1(OC)cc(C(=O)NC(CNC(=O)CN2CC(C)C2)C2CC2)[nH]n1 35246,c1(N(C2C(C)SCC2)C2CCCC2)ccc(S(=O)(=O)N2CCCCC2)c(Br)c1 35247,C12(C(=O)NC3(C(=O)NC)CCC3)CC(C)(CN1NC(c1nc(C)oc1C)=O)C2 35248,C1(C(N(CCCOCCNC(COCC#C)=O)C)=O)COc2cc(O)ccc2C1 35249,CC1CNc2c(C(=O)NCCN(C)C(C3CCC(N=[N+]=[N-])CC3)=O)cnn2C1 35250,C1(N(C2CCOC2C)C(c2cccc(OCC)c2)=O)CCNCC12CC2 35251,C(C1CN(C(=O)CCN(c2ccncc2)C)CC1C(=O)NCC)=CC 35252,c1(C(C(=O)NC(CC)(C)CNC(=O)Cn2cc(C3CC3)nn2)C)ccccc1F 35253,N1(c2c(C(C)=O)cccn2)CCC(NC(=O)C(C)n2cnnn2)C(O)C1 35254,Cn1nc(C(N2CCOC(CC(=O)NCCOCC3CCCC3)C2)=O)cc1Cl 35255,c1(C(C)(C)C)cc(C(=O)OCCNCCOCC(O)CO)cs1 35256,C1(C(=O)NC(C2CCOCC2)C#C)(CC)CCN(C(=O)CCc2conc2C)C1 35257,N1(C(CCOC)=O)CC2CCOC2(CNC(c2cc(OC)cc(C(C)C)c2)=O)C1 35258,N1(C(c2c(CC)ncs2)=O)C(CNC(c2cc(C(C)C)no2)=O)CC2CC12 35259,C(=O)(C1CCCc2cn(C(C)C)nc21)NCC(CNC(c1c(C)nns1)=O)F 35260,c1(OC)ccc(C(C)=CC(=O)NC2CC2CNC(c2csc(C#N)c2)=O)cc1 35261,CC(C)C(C(=O)NC1CN(C(C)C)CC1C)C(C)NC(=O)C=Cc1ccccc1 35262,c1(-c2n(C(CCCC)C(=O)NC)nc(CC3CCC3)n2)csc2cccc(F)c12 35263,C1(NC(CCC(=O)NC)=O)(CNC(c2cccnc2F)=O)CCCCC1C 35264,N1(C(C2CC2C2CCC2)=O)CCCCC2(CCN(C(C3(C(F)F)CCC3)=O)C2)C1 35265,c1(C(=O)NC2C(CNC(=O)Cn3cnnc3O)C2)cc2ccc(Cl)c(F)c2[nH]1 35266,c1(C(=O)NC2CCCN(C(c3noc(CC)c3C)=O)C2)ccc(Cl)cc1OC 35267,Cc1ccc(S(=O)(=O)NC(Cn2ccnn2)C(=O)N2CCCC2)cc1C 35268,C1(CNC(c2cnn(C)n2)=O)C(C2CC2)CCN1c1ncnc(Cl)c1F 35269,CC1(C)C(CC(=O)NCCC2COCCO2)CCN1C(C1CCCCCC1)=O 35270,C(C(C(=O)NCC1CC(F)(C(=O)OC)C1)N(C)C)OC.C12(CC1(F)F)C(=O)NC2 35271,N1(C(c2ccn(CCC)n2)=O)CC2CC2C1CNC(c1ccnnc1C)=O 35272,c1(C(=O)OC)ccc(C(=O)NCCNC(=O)C(C)NC(C2CCCC2)=O)cc1 35273,c1(C(=O)NCC2(O)CN(C(C3(C(C)C)CNC(=O)C3)=O)C2)nn(C)c(Cl)c1Cl 35274,c1(NCC2CN(C(C3CN(C)C3)=O)CC23CCC3)ncnc2c1nnn2C 35275,CON(C(=O)CCCC(C)NC(=O)C(n1ccc(C)n1)C)C1CCOCC1 35276,N1(CC)CCOC(C(=O)NCCn2cc(C(=O)N(C)CC3(O)CN(C)C3)nn2)C1 35277,c1(C(N(CC(CC)NC(C2(c3cccs3)CC2)=O)C)=O)cnc(O)n(C)c1=O 35278,O=C(C1=CCCN(C(c2cc(F)c(Cl)c(Br)c2)=O)C1)NC1COCC1F 35279,C12(C(=O)NCCNC(=O)CC3CCOC3=O)CC3CC(C1)CC(F)(C3)C2 35280,Cc1c(C(=O)N(C)CCC2CCCCN2C(=O)C#CC2CC2)cccc1CO 35281,c1(C(=O)NC(CCCC)CNC(c2ccco2)=O)cccc(OC)c1OC 35282,C(CC(=O)NC(C1CCCC1)CN(C)C)N(C)C(=O)OC(C)(C)C 35283,c1(C(=O)NCCC(=C)CNC(c2cc(Br)c(C)o2)=O)cccc(CC)n1 35284,c1(OC)cncc(C(=O)NCC(CNC(=O)CC2C=CCCC2)CO)n1 35285,C12(C(=O)NC(C)Cc3cnoc3)CC(n3cc(CCCN(C)C)nn3)C1C2 35286,C(=O)(C1CCCc2cccnc21)N1CCC(N(C(=O)CC(C)C)CC#C)CC1 35287,Cc1ccc(NNC(=O)CN(C)C(C2CCC(=O)N2)=O)cn1 35288,N1(C(c2ccc(NC(C)=O)nc2)=O)C2CCC1CN(C(=O)COC1(C)CCC1)C2 35289,c1(C(N2C(CN(C(=O)COCC3CC3)C)CCC2)=O)ccc(F)c2ccncc12 35290,C=CC(C)(O)CC(=O)NC1C2CC(NC(c3nc(CC)c[nH]3)=O)CC12 35291,C1(CCOC)CCCCN1C(=O)C(N1CCC(Cn2cnnc2)CC1)=O 35292,c1(C(=O)NC(CNC(C2(C)CCC(C)C2)=O)C)cnn2ccccc12 35293,C1(C(N(CC(CCC)C)C)=O)CC12CCN(C(c1n[nH]c(=N)[nH]1)=O)C2 35294,c1(C(N2CCC(CC(F)F)CC2)C(=O)NCCSC)cc2ncccc2o1 35295,N1(C(C(=O)NCc2ccc(-c3c(C)nc(CC)s3)cc2)=O)CCCSCC1C 35296,CC1(F)CCC(C(=O)NC2CCCC2NC(c2ccc([N+](=O)[O-])o2)=O)CC1 35297,CC1(C)CCC(NC(c2ccn3ncccc23)=O)C(CNC(=O)C(N)=O)C1 35298,c1(C(N2CC(c3ccccc3C)OCC2C)C(=O)NCCOC)cccc(F)c1C 35299,CC(C)(C)C(O)C(=O)N(CCNC(C1C(c2ccccc2)C1(C)C)=O)C1CC1 35300,Cn1nc(C(=O)NC2CCC(NC(c3coc(CC4CC4)n3)=O)C2)cc1C#N 35301,N1(C(CCSCC(=O)OC)=O)Cc2ccc(C(=O)NCc3cnccn3)cc2C1 35302,c1(OC)ccc(S(=O)(=O)N2CC3CC2CN3C(c2ccc(Br)c(F)c2)=O)cn1 35303,N#Cc1ccc(C=CC(N2CCC(NC(c3cn4c(n3)CCC4)=O)CC2)=O)cc1 35304,CC(CCCNC(C1(C)CC1)=O)NC(c1nc(I)cs1)=O 35305,Cc1nc2cc(C(=O)NCC(C)NC(c3ccc(Cl)nn3)=O)ccc2o1 35306,CSC1=C(C(=O)NCC(C2CC2)N(C(=O)C(CO)c2ccccc2)C)CCCC1 35307,C1(C(=O)N(C)CCOCCN(C)C(c2c[nH]cc2C2CC2)=O)(CC)CC1(F)F 35308,C1(NC(=O)NCCC(C(F)(F)F)OC)CCN(C)C2(CC2)C1 35309,C1(NC(C(CC)NC(C)=O)=O)CCN(C(=O)CSCCC(C)C)C1C 35310,c1(C(=O)OCC)c(OC)cc(NC(C2C3CN(c4ncc(F)cn4)CC23)=O)cc1I 35311,c1(N(CCC)CCNC=O)cc(N(C(c2csc(C)n2)=O)C2CC2)n[nH]1.CC 35312,C12C3CCC(C3)N1C(=O)N2.c1(C(=O)C(=O)NC(C)(C)C)ncc(CO)s1.CC 35313,c1(CCC)onc(C)c1C(=O)NC(C1CN(CCOCC(F)(F)F)C1)C 35314,C12(CNC(C(C)(C)CNC(=O)CC3CC4CC4C3)=O)CC=CC(C1)OC2 35315,C=Cn1nccc1C(N1CCSCC1C(=O)NC(CC=C)C1CC1)=O 35316,c1(C2C(C(N3C(C(=O)NCCC(=O)O)CC3)=O)C2)ccccc1OC(F)(F)F 35317,Cc1ncncc1C(=O)NCCn1cc(CNC(C2CC2C(C)(C)C)=O)nn1 35318,N1(CCNC(c2c(C)occ2)=O)CCC(NC(c2c[nH]c(=S)cn2)=O)CC1 35319,C1(NC(C(C)C2(O)CCC2)=O)CCCCCC1NC(c1cc(F)cc(Cl)c1)=O 35320,CC1CC(C(=O)N(CCCCCNC(=O)C2=CC(C)(CO)C2)C)=NO1 35321,C(CCC1CC1)(C(=O)NC1CC1)NC(C1(COC)CCCO1)=O.C1CCNC1=O 35322,C12C3CC(O)C1N(C3)C(=O)CN2.c1(C=CC(=O)NC2(C(C)C)CC2)cscn1 35323,CC1(CNC(=O)C=Cc2ccco2)CN(C(=O)CCN2CCC(F)C2)CCO1 35324,C(=O)(C#CC(C)(C)CNC(C1(C)CC1(F)F)=O)NC1C(C)COC1 35325,CCCN=c1[nH]c2c(c(=NC(C)c3cnccn3)[nH]1)CSC2 35326,c1(C(=O)NC2C(C)CN(C(C3CCCC(C(C)(C)C)C3)=O)C2)ccc([N+](=O)[O-])o1 35327,N1(C(c2nc(C)oc2C)=O)CCN(C(c2cc(=O)c(O)c[nH]2)=O)CC(O)C1 35328,N1(C(C=CC)=O)CCC2(CC1)CC(NC(=O)C(C)Sc1nnnn1C1CC1)CO2 35329,CCC(C)(CC)NC(C1CCC(CNC(=O)Cc2cnnn2C)O1)=O 35330,C(=O)(C(C(C(C)C)OC)N1CCC(N(C)C)C1)NC1(CO)CCOC1.CCCO 35331,C(C(C)(CNc1cnc(N(C)C)n1C)C(=O)OC)SC 35332,c1(C(C(N2C(C(N)=O)CC2)=O)NC(c2ccco2)=O)ccc(Cl)cc1Cl 35333,C1(C(N2CCC(CNC(CCS(C)=O)=O)C23CC3)=O)COc2cc(F)ccc2C1 35334,N1(C(c2cc(OCC)cc(F)c2)=O)CC2(CC(NC(=O)CCC3(C)CC3)CO2)C1 35335,c1(C(N2CCCC(NS(CC(=O)OCC)(=O)=O)C2)=O)ccc2nccn2c1 35336,C1(N(C)C)CC(CO)CN(C(c2ccc(Br)o2)C(=O)NCc2ccccc2)C1 35337,c1(N2CCC(NC(=O)OCC)CC2)nc(N(CCCF)C)nc2c1cnn2C 35338,c1(NC2CC(C3C(=O)NC(=O)N3)C2)ncnc2c1CCC2 35339,CC1C2C(CCN2C(=O)C=CCN2CCCC2)CN1C(=O)CCOC1CCOC1 35340,c1(C(N2CC(C=C)(CC(=O)NCCOC3CCOC3)C2)=O)ccc([N+](=O)[O-])[nH]1 35341,C1(C(=O)NCC2CCN(C(C(C)Cc3cccc(F)c3)=O)C2)CCCC(=O)N1C 35342,C(=O)(C1=CC2CCCCC12)N1CC(CNC(=O)CC2(O)CCC2)C(C(F)(F)F)C1 35343,c1(NC(C2N(C(CC3CN(C)C3)=O)CCC2O)=O)ccc(C(=O)N(C)C)c(F)c1 35344,N1(C(c2cc(C)ncc2C)=O)CC2CCCC(C1)N2C(c1cccc(N)c1O)=O 35345,C1(CNC(C2CCCN(C(CC3(C(=O)OC)CC3)=O)C2)=O)CCC12CCOCC2 35346,C(=O)(C(F)CCC(C)C)NCC(CC(=O)N1C(C#C)CC1)C 35347,C(=O)(C1CCCc2sc(=N)[nH]c21)N(CC(CNC(C(CCC)C)=O)(C)C)C 35348,N1(C(C2N(C(C)C)CCC2)=O)CC(O)CC1CNC(=O)CC(=O)NCC1CC1 35349,N1(C(Cc2ccc(C#N)cc2)=O)CC(NC(=O)C=CC(N)=O)C2(CCOCC2)C1 35350,C1(C(N(C(CNC(c2cc(C(F)(F)F)no2)=O)C2CC2)C)=O)CCCSS1 35351,C1(C(=O)NCc2ccc(C3CCC3)cc2)CCCN(C(C2(C3CC3)CC2)=O)CC1 35352,c1(C(=O)NC2C(OC)CN(C(=O)CCC3CCCC3)C2)n[nH]c2cccnc12 35353,N1(C(C2(CCOC)CCC2)=O)CC(CCNC(c2cnc(CC)[nH]2)=O)OC(C)C1 35354,C(C(C(F)(F)F)N1CCN(C(=O)CC2C=CCC2)CC1)NC(COCC)=O 35355,c1(C(N2CC(N(C(=O)CC3CC(C(F)F)C3)C)C2)=O)coc(Cl)c1 35356,C1(CC(N2CCC(CN(C(=O)CN3CCCCC3)C)CC2)=O)CCCCC12CC2 35357,c1(C(=O)NCCC(C)NC(c2ccc(Cl)o2)=O)oc2ccccc2c1CO 35358,c1(CNC(c2ccc(Cl)c(F)c2)(C)C)cccc(F)c1C#N 35359,C1(C(=O)NCC(C(C)C)NC(c2cn3c(n2)SCC3)=O)CCC(S(C)(=O)=O)CC1 35360,C(=O)(C(F)CCC(C)(C)C)N(CCNC(CN(C1CC1)CC)=O)CC1CC1 35361,c1(CCC)ccc(C(=O)NC2COCCC2NC(C2CC(F)C2)=O)cc1[N+](=O)[O-] 35362,C(=O)(CC(O)C(C)(C)C)NC1CCC(NC(C2ON=C(C)C2)=O)CC1 35363,CCCCC(C(=O)NCC=C(C)C)NC(=O)CCC(N)=O 35364,c1(N(C(c2ccn(C)c2)C(=O)N(CC)C2CC2)C)nnc(C2CC2)n1C 35365,c1(C(N2CCCC(CC(=O)Nc3nccc(C)c3)C2)=O)cc(Br)cnc1O 35366,c1(CC(=O)NC2CN(C(=O)CC3(O)CCOC3)CC2O)cc(F)cc(Cl)c1 35367,N1(C(C(C)(C)SC)=O)CCN(C(CNC(=O)CC2CN(C)C2)C(F)F)CC1 35368,c1(C(N2CC=CC(NC(C(F)=C(C)C)=O)C2)=O)cccc2ncnc(O)c12 35369,C(=O)(C1=C(Cl)CCC(C)C1)N(CCOC)CCNC(c1cc(C)c(N)cn1)=O 35370,c1(C(=O)NC(C)Cn2cc(C3CCN(C)C3)nn2)ccc2c(c1)COCO2 35371,CCCC(C)(O)CC(=O)N1C2CCC(C2)C1C(=O)NC(c1ccccc1)CF 35372,N1(C(CCC(C)C)=O)CCOCC2(COCCN2C(=O)C2=CC3CCCC23)C1 35373,c1(CC)ccc(C(=O)NC2CCC(NC(C3(F)CCC3)=O)C2)[nH]1 35374,C(C(CC(C)(C)C(=O)OC)NCc1cn(-c2cc(C)cc(C)c2)nn1)OC 35375,C12(CNC(C(C(C)C)C)=O)CCC(CN(C(=O)CCCc3nccs3)C1)C2 35376,Cc1[nH]c(C(=O)NCCCO)c(C)c1C(=O)Nc1cnc(Cl)cn1 35377,C(=O)(N1CCCc2nncn21)C1C(C)CN(C(=O)CC2(n3cccn3)CC2)C1 35378,C1(S(N)(=O)=O)(C(=O)NCC(C)NC(c2ccccc2OCC(N)=O)=O)CCCC1 35379,c1(OC)cnc(F)cc1C(=O)NCC(C)(CO)NC(=O)C=Cc1ccc(O)cc1 35380,Cc1cccc(C(=O)NCCC2CN(C(=O)COC3(C)CCCC3)C2)c1Cl 35381,C(=O)(C1=NOC2(CCN(C(C3CCSCC3)=O)C2)C1)Nc1cc(C(=O)OC)no1 35382,N1(C(C(C)n2cnnn2)=O)CCN(C(=O)C#CC2CC2)C(CC(F)F)C1 35383,c1(C(=O)NC(CC)CNC(=O)CCc2ccc(F)nc2)cncc2cccnc12 35384,C1(C(=O)NCC2(NC(=O)Cc3cccs3)CCC2)CC12CCSCC2 35385,C(=O)(C(O)C(C)OC)N(C1CCN(C(C2(CF)CCC2)=O)CC1)CCC 35386,c1(CC(N2CC(C(C)(C)O)(CNC(CSC)=O)C2)=O)ccc(S(=O)(=O)NC)cc1 35387,C#CC1(C)CCCN(CC(=O)CCOC)C1 35388,C1(CC)C(C(=O)NCC2(CC(=O)OC)CC2)CCN1C(c1cnsn1)=O 35389,c1(C(C)=O)ccc(C(N2CCC(C3CCCN3C(c3csc(CF)n3)=O)C2)=O)o1 35390,c1(CC)nn[nH]c1C(=O)NCC1(NC(=O)C(COC)OC)CC1 35391,c1(C(=O)NCC(CC)NC(=O)CCC(C)OC)ccc(N)c(CC(C)C)c1 35392,C(=O)(CCCCN(C)C(c1ccc(CO)o1)=O)NCc1nnc(C)o1 35393,C(=O)(C1=NNC(=O)C1)NCC(CC(=O)N(C(CC(CC)C)C)C)O 35394,c1(CNC(C(C(C)O)NC(=O)CC(C)(C)O)=O)ccc(C#N)cc1 35395,c1(C(N2CCC(NC(c3ccccn3)=O)CC2C2CC2)=O)cncc2sccc12 35396,c1(CCC(=O)NC2CC(NC(CCS(C)=O)=O)C2)nnc(S)nc1O 35397,CC1(C)CC2(CC2C(=O)NCC2(NC(c3ccc(F)c(CC#N)c3)=O)CC2)C1 35398,C(=O)(CCC(C)(C)F)N1CCCC(NC(C2C(C(=O)OCC)CC2)=O)C1 35399,C1(CNC(=O)CSc2ccsc2[N+](=O)[O-])CCN(C(C2CC2F)=O)C12CCC2 35400,c1(CC(=O)NC(C2CCCN(C(=O)CC3CC3)C2)C)ccc(F)c(F)c1 35401,C1(C(N2CCC(NC(C(CC)=CC)=O)C(C)C2)=O)CCCC2CCCN12 35402,CC1(C)CCCC(C(=O)NC2CCCC23CN(C(c2snc(Cl)c2Cl)=O)C3)CC1 35403,CC(C)(CCC(=O)NCc1nc(=O)o[nH]1)NC(=O)C(c1ccccc1)F 35404,c1(CC(C(=O)NC2(CCNC(CC3CC(OC)C3)=O)CC2)C)ccc(F)cc1 35405,N1(C(=O)OC(C)(C)C)CCC(C2CCN(C(=O)C(C)(Cl)CCl)CC2)C1 35406,N1(CC)C(=O)CCC1CCNC(=O)NCCOCCN1C(=O)CNC1=O 35407,C1(C)(CCC(=O)NCCCN(C(C)C)C(C2CC(F)C2)=O)CCC(=O)N1 35408,n1(CC(=O)NC2C(NC(c3ccc(CSC)o3)=O)C2)cc(Br)c(C)n1 35409,O=C(CS(=O)(=O)CC1CCCO1)NC12CC(NC(=O)C(c3ccccc3)F)(C1)C2 35410,C12(C(=O)NCC(=O)NC(CNC(c3c(OC)cccc3)=O)C)CC(C)(CCO1)C2 35411,Cn1cc(CN(CCC(=O)O)CCn2cc(-c3cnn(C)c3)nn2)nn1 35412,c1(C(=O)NC2CC(O)(CNC(=O)CC3CCCS3(=O)=O)C2)cc2c(s1)CCC2 35413,CC(C)S(=O)(=O)CCCN1CC=CC(NC(c2coc(Cn3cccn3)c2)=O)C1 35414,c1(OC)cccc2c(Oc3cccc4c(Br)cccc34)ccnc12 35415,C=CC1CN(C(=O)Cn2cc(C3CC3)nn2)CC1NC(c1cc(C)c(C)[nH]1)=O 35416,N1(C(COCC(C)C)=O)CCC2C1CCCN2C(=O)Cc1ccc2c(c1)CCC2 35417,C=C(Cl)CC(C(=O)NOCCOCCOC)N(C(=O)C(C)NC(C)=O)C 35418,C1(CC=C)(C(=O)NCCC(O)C2CCCC2)CCN(C(=O)C=Cc2cocn2)C1 35419,Cc1ccc2n[nH]cc2c1C(N1CC(C)(NC(c2cnc(O)c(Br)c2)=O)C1)=O 35420,N1(C(C2CC(NC(C3N(C)CC(C)(C)C3)=O)C2(C)C)=O)CC2CCC(C1)C(=O)N2 35421,C1(NC(c2cc[nH]c2)=O)CCN(C(c2cc(=O)n3ccsc3n2)=O)CC12CCC2 35422,C(=O)(C1CCCc2c[nH]nc21)N1CC2C(NC(CN3C(=O)CC(C)(C)O3)=O)C2C1 35423,c1(CC(=O)NC(C)CCNC(=O)C(C)C2CCCO2)ccc2nonc2c1 35424,C1(CNC(CP(C)(C)=O)=O)CC2CC(C1)CN(C(=O)COCC(F)(F)F)C2 35425,C1(C(=O)NC(C)CCOC)(CC)CCCN(C(c2cc(CO)nn2C)=O)C1 35426,c1(C(=O)NC2C(NC(c3c(C)nc(COC)s3)=O)C2)cc([N+](=O)[O-])c(C)cc1Cl 35427,c1(C(=O)OC)ccc(C(=O)NC2CCC(NC(=O)CS(N)(=O)=O)CC2)nc1 35428,c1(CCC(=O)NC(CC)CNC(C2CCC(F)(F)CO2)=O)nc2ccccc2o1 35429,C(C1(C)COC1)=CC(=O)NCCN(C(C1C(C)(C(=O)OCC)C1)=O)CC 35430,N1(C(C2CCCN(CC)C2)=O)C2CCC(C2)C1CNC(c1ccc(O)nc1)=O 35431,N1(C(C2C(C)(COC)C2)=O)CC2(COC(CNC(=O)Cn3nc(C)nc3C)C2)C1 35432,N1(C(C(C)(C)c2ccccc2)=O)CCCC(NC(=O)Cc2ccccc2)C1 35433,CCC(CC(C)C)C(=O)NCCC1(O)CN(C(=O)Cc2ccn(CC)n2)C1 35434,O=C1CCc2cccc(NC(=O)NC3CC(CO)C34CCC4)c21 35435,C1(C)(NC(CCCCCN(C)C(c2cccn(C)c2=O)=O)=O)CCC(=O)NC1=O 35436,C1(N(C)C(C2(C(C)(C)C)CCC2)=O)CCN(C(=O)COc2ccsn2)C1 35437,c1(C(=O)NCC2C(C(=O)NC(c3c(C)nccn3)C)CCO2)ccn(C)c(=O)c1 35438,C1(C(=O)NC(C(=O)NC)(C)C)CC2CC1CC2NC(=O)C(CO)N(C)C 35439,N1(C(C(CC2CC2)NC(C2(CN(C)C)CC2)=O)=O)CCC(O)CC1 35440,C=C1CCN(C(c2ccn(C)c2)=O)C(C(=O)NC2(CO)CCCCC2)C1 35441,C1(CC)CN(C(=O)C=Cc2cccnc2)CCN1C(=O)COCC(=O)NC 35442,N1(C(c2c(C)cc[nH]2)=O)CCCC2C1CCCN2C(C1CCC(N(C)C)CC1)=O 35443,c1(C(=O)NCC2(O)CN(C(C(CSC)O)=O)C2)cncc(N2CCCC2)n1 35444,N1(C(C2CCN(C(c3n(CC)ccn3)=O)C23CC3)=O)CCC(O)CC(C)C1 35445,N1(C(C(C)=CC2CC2)=O)CCCC(C)C1CNC(=O)CCC1CC1(C)C 35446,CC1CS(=O)CCN1C(=O)C(C1CCN(C(=O)C=C2CCCCC2)C1)F 35447,C12(NC(=O)C3CC3)CC(C(c3cccc(F)c3)c3ccco3)(C1)OC2C(F)(F)F 35448,C(COC(C)C)(C(=O)O)NC(N(C(CC)=O)C)=O 35449,c1(C(=O)NCCCC(C)NC(CCNC(COC)=O)=O)ccc(C)nn1 35450,Cc1ncc(C#N)cc1NC(c1conc1CNC(C1(C)CCC(C)C1)=O)=O 35451,N1(C(CCC(=C)Cl)=O)CCC2CN(C(C3(C)CCCNC3=O)=O)CC2CC1 35452,C1(CCOC)CN(C(=O)CC2CS(=O)(=O)C2)CCN1C(c1cnc(S)[nH]1)=O 35453,c1(OC)cc(S(=O)(=O)Nc2nc(Nc3cc(C)ccc3C)cs2)c(F)cn1 35454,C(CC(C)C(=O)N1CCN(CCN(C(=O)Cc2n[nH]c(=NC)s2)C)CC1)=CC 35455,CC(C)CCC(F)C(=O)NC1(CCC(=O)N2CCC2CC2CCCC2)CCCC1 35456,c1(OC)ncnc(C(=O)NC2(C)CN(C(C3CCOC(=O)CC3)=O)C2)c1F 35457,N1(C(C(c2cn(C)nc2)O)=O)CCCC2(C1)CN(C(c1cnc3sccn13)=O)C2 35458,CCC(Cc1ccccc1)C(=O)NCC1(F)CN(C(=O)C(c2cnccn2)C)C1 35459,CCCC(CC)C(=O)NCC(O)CCNC(c1cc(=O)c(Br)c[nH]1)=O 35460,N1(C(Cn2ncc(C)c2)=O)CC=CC(C(=O)NC2CC(CO)C3CC23)C1 35461,CC(CC(F)F)C(=O)N1CCC(CNC(c2cccc(CO)n2)=O)C1 35462,CC1(C(=O)NCC2CC(NC(C3CC(=O)N(O)C3)=O)C2)CS(=O)(=O)C1 35463,C1(C(C)NC(C2(CC)CCCC2)=O)CCN(C(C2CC2(Cl)Cl)=O)CC1 35464,C(CC(C)(C)OC)(c1n(CCC)nnn1)NCc1cnn(C2CC2)c1C 35465,CCCC(C)(CCCN(C(=O)Cc1nc2c(s1)COCC2)C)C1OCCO1 35466,N1(C(Cn2c(C)c(Cl)cn2)=O)CCCCC(C(=O)NCc2ccnc(C#N)c2)C1 35467,c1(C(=O)NC2CC(C)(NC(CC(=C)Br)=O)C2)c(O)nnc2c1CCC2 35468,C(C)(CCCNC(=O)C=CCOC1CCOCC1)NC(CSCCCC)=O 35469,C(=O)(NNc1cccc2ccsc12)C1N(C(=O)OC(C)(C)C)C2C(O1)CCC2 35470,N1(Cc2nc(-c3ccc(C)cc3)on2)CC2CCCCN2c2ccccc21 35471,c1(C(=O)NCCCCCCNC(CN2C(C)CCC2C)=O)cc2occc2n1C 35472,c1(C(=O)NC2CC(F)(CNC(CCOC)=O)C2)c(F)ccc(F)c1N 35473,N#CC1(C(N2CCN(C(C3(S(N)(=O)=O)CCC3)=O)CC2)=O)CC2CC2C1 35474,N1(C(C2CCC(C(N)=O)CC2)=O)CCN(C(=O)C2=COCCC2)CC1C(F)F 35475,Cc1cc2[nH]c(COCCOCC=O)cc2o1.C1(NC(ON)=O)CCC1 35476,CC(=O)CC(C)(C)C(=O)N1CCC(C)C(CNC(C2CN(C)CC(C)O2)=O)C1 35477,C1(C(N2CCC(C(C)OC)CC2)=O)CC2CCC1N2C(c1csc(C)c1)=O 35478,CN=c1[nH]c(=NCCCc2nc(C)cs2)[nH]c(=NC2CCOC(C(C)C)C2)[nH]1 35479,c1(C(N(CCCCN(C(CCn2c(C)ncc2)=O)C)C)=O)ccc(F)c(Cl)c1F 35480,c1(CNC2CCC(C(N(c3c(Cl)cccc3I)C)=O)CC2)cc2ccccc2s1 35481,N1(C(C(c2c(C)ccnc2)(C)C)=O)CCCC(C)C1CNC(c1nccn1C)=O 35482,c1(C(N2CCN(C(c3ccc(C(C)=O)nn3)=O)C3C2C3)=O)c[nH]c2ccccc12 35483,N1(C(C2CC(NC(=O)CCC3CC3(F)F)C(O)C2)=O)CC2(CCC2)C12CCC2 35484,C1(CNC(CC2C(C)CCO2)=O)CCC2CN(C(c3cnc(Cl)[nH]3)=O)CCC2C1 35485,N1(C(CC)=O)CCC(C)(CNC(=O)C(C(C)C)NC(C)=O)C1 35486,C(=O)(C(C(C)(C)C)N(C)C)NCC1(CNC(C(C)n2cnnn2)=O)CC12CCC2 35487,c1(OC)ccc(CC(=O)NCCC(O)CNC(C2CNC(=O)N2)=O)cc1O 35488,C=CCC(CNC(C1(C)CC(=C)C1)=O)NC(c1cc(C2CC(F)(F)C2)[nH]n1)=O 35489,C=C(Cl)CC(C(=O)NC(c1nccn1C)C)NC(=O)Cc1ccn(CC)n1 35490,C1(NC(C(F)=C(C)C)=O)C2CC3CN(C(c4cc(O)c5ccoc5c4)=O)C1C3C2 35491,Cc1ccc(C(=O)NCC(C)(CO)NC(=O)CC2CCC2(C)C)c(O)n1 35492,c1(OC)c(C(N2CCCCC(Cn3cc(C4CCC4)nn3)C2)=O)ccc(Cl)c1Cl 35493,c1(OCC)cc(C(N2CCC(=CCNC(=O)CCC3CC3)CC2)=O)cc(F)c1 35494,Cc1ccc(Cl)c(C(=O)NCC2CC2NC(=O)Cc2ccco2)c1N 35495,N1(C(C(CSC)OC)=O)CCC(NC(=O)Cc2nc3ccccc3s2)C(C)(C)C1 35496,C1(NC(C(C)NC(=O)CC2CNC(=O)O2)=O)(CO)CC2CCCC12 35497,CCCCCCCCCC(=O)NCC1CC2(CC2)CN1C(=O)C(O)C(F)F 35498,N1(CCNC(c2nc(C(C)(C)C)oc2)=O)CCCN(C(C2CC2(F)Cl)=O)CC1 35499,CC1CC(C(F)(F)F)n2nc(C(=O)NCC3CC4(CC4)CO3)cc2N1 35500,n1(CC=C)nnnc1C(c1cc(C(F)(F)F)cs1)NCC(C)OC 35501,Cc1nc([N+](=O)[O-])cn1CC(=O)NCCC(C(C)C)NC(C1CCOC(=O)N1)=O 35502,C1(CN=C(NC(CC)CO)NCC(F)F)COC2(CCC2)CO1 35503,c1(C(=O)NC2C(NC(C(C)(C)OC(C)C)=O)C2)ccc(Cl)c(F)c1O 35504,O(C1CCCc2c(F)cc(F)cc21)C=O.C12(CCCCC1)C(=O)N2C.CC=CC 35505,C(=O)(C(C#N)C(C)C)N1C(SCCCn2cc(-c3n[nH]c(C)c3C)nn2)CC(O)C1 35506,N1(C(Cc2nc(COC)sc2)=O)CC2C(NC(=O)C(C)n3ccnc3)C2C1 35507,c1(C(N2C(C(=O)OC)CCOCC2)C(=O)OC)ccc(C)c(F)c1F 35508,C1(NC(C2N(C(c3c(C)noc3)=O)CCSC2)=O)(CO)CC2CCCC12 35509,c1(C(=O)NCC(C)CNC(C23CC(C)(C2)C3)=O)cc2c(o1)CCCNC2=O 35510,C1(CNC(c2c[nH]c(=N)o2)=O)CCC2(CCC2)C1NC(=O)CCCc1cccs1 35511,N1(Cc2n(CC)cnc2)CC(CC(=O)NC(=O)NC)c2ccccc21 35512,Cc1nc(Cl)nc(N2CC3CC(NC(C4CC5CCCC45)=O)CC3C2)c1C#N 35513,C1(C(=O)NCC2C3CN(C(=O)C(C)OC)CC23)(CC)CCCCC1 35514,n1(CC#C)cccc1C(=O)NCCCNC(=O)C(C)OCc1ccccc1 35515,C1(C(N(C2CCN(C(C(CCN(C)C)(C)O)=O)C2)CCO)=O)CC2CCCC(C1)C2 35516,N1(C(C(CC=C)NC(C)=O)=O)CCC(C)N(C(=O)CSCCCN(C)C)CC1 35517,CN1CCN(C(=O)CCc2cc(F)ccc2Br)C(CNC(=O)C(N)=O)C1 35518,c1(OC)ccc([N+](=O)[O-])cc1-n1cc(CN(C(=O)C(C2CCC2)OC)C)nn1 35519,c1(C(N(C)CCC2CCCCN2C(=O)CCC(N)=O)=O)ccccc1P(C)(C)=O 35520,N1(C(c2c(OC)ccnc2)=O)CCCC(NC(=O)CC(C)(C)C#N)C1C 35521,N(C(=NCCCSC1CC2CCC2C1)NCC(C)(C)C)CCC(=O)N(C)C 35522,CCCCCCCCOCC(=O)NC(C)CNC(C1CCC(NC(N)=O)CC1)=O 35523,n1(CC)ncc(Cl)c1C(N1CCCCC1CCN(C(=O)C(C)CC1CC1)C)=O 35524,Cc1ccc(Cl)cc1CNC(=O)CCN(C(=O)CN1CCC(C)C(C)C1)C 35525,CC1CN(C(C2CC(O)(CNC(C3(C)CCC3)=O)C2)=O)CC(C)(C)C1 35526,CC1(NC(C23CC(CN2C(C2(CCN=[N+]=[N-])CC2)=O)C3)=O)CCOC1=O 35527,C1(CNC(Cc2ccc(C)o2)=O)CN(C(C2CC2C)=O)C(C)(C)C1 35528,C1(NC(=O)Cc2ccc(Br)s2)CN(C(=O)CCC2CC2)CC1O 35529,c1(C(C(N2CCC(CC(=O)NCCC(=O)N(C)C)C2)=O)=O)ncc(F)cc1F 35530,C1N=C2N=C(C=C(C)N2)C(=O)NC2CCCC12.N1(C(C)=O)CCC(C)(CO)C1 35531,N1(C(c2scc(OC)c2OC)=O)CCN(C(C2OCCO2)=O)CC2(CC2)C1 35532,c1(C(=O)NC2(CCC)CCN(C(CC=C)=O)CC2)cc2c(cnn2C)nc1C 35533,C1(CC)CN(C(=O)C(=O)NC23CC(C(F)F)(C2)C3)CCN1C(C)=O 35534,N1(C(C=CC2COC(C)(C)O2)=O)CC(NC(=O)C=CC2CCCO2)CC(C)(C)C1 35535,C=C(Cl)CC(C(=O)NCC1C(CO)C1(F)F)NC(=O)C(CSC)OC 35536,N1(C(c2c(CC)noc2)=O)CC(CNC(c2cccc(C)c2)=O)CCC1C 35537,c1(C(N(C(CC(=O)OCC)c2ccccc2)CCC)=O)ccc(COC)o1 35538,c1(C(=O)NCc2occ(C(=O)NCC(C(CC)C)C)c2)ccnc(C)c1N 35539,c1(C(N2C(CCNC(CCCCCC=C)=O)CCC2)=O)cc(N)c(F)c(F)c1Cl 35540,c1(CC(=O)N(CCNC(=O)CCOCC(F)F)CC)cncc(Br)c1 35541,C(c1cn(CCCNC(C2CCN(c3ccc(Cl)cn3)CC2)=O)nn1)=CC 35542,C1(NC(=O)Cn2cc(CO)nn2)CCC(F)CC1.C12CCC(C1)C(=O)N2C 35543,C12(C(N3CCC(NC(c4cc(C)cc(O)c4)=O)C3)=O)CCC(C)(CC1)OC2 35544,N1(C(C23N(C(C(CC)COC)=O)CC(C)(C2)C3)=O)CCC2CC1C(=O)O2 35545,C1(NC(CC(C)F)=O)CC(F)CN(C(c2cncc(N3CCCC3)n2)=O)C1 35546,Cc1ccc2sc(C(=O)NCC3(O)CCN(C(=O)CCCCC(N)=O)C3)cc2c1 35547,N1(C(CNC(=O)CC2CC(CF)C2)=O)CC2CCCC(C1)N2C(c1cc[nH]c1)=O 35548,c1(C(=O)NCCC(=O)NCCC2CCN(C(C3CCC3)=O)C2)cnccc1Cl 35549,C(=O)(CCC(=O)NCC1CN(C(c2csc(CO)n2)=O)C1)Nc1nnc(CC)s1 35550,C12(C(N(CCN(C(C3CC3(C)C(C)C)=O)CC)CC)=O)CC(C)(C1)OC2(C)C 35551,CC1(C)CC(C(=O)NC2CCC([N+](=O)[O-])CC2)CN(C(C2(C)CCSCC2)=O)C1 35552,C1(NC(=O)CC2=CCCC2)CCCC2CN(C(=O)Cc3ccc(O)c(F)c3)CC12 35553,C1(C(=O)NC2(c3ccc(F)cn3)CC2)CC2c3ccccc3C1c1ccccc12 35554,Cn1nnc(C(N2CC(=C(F)CNC(c3cc(F)c[nH]3)=O)C2)=O)n1 35555,N1(C(c2c(C)occ2)=O)CCC2CC(CNC(C3CCC(C)CC3)=O)CCC2C1 35556,CC(C)CC(C(=O)N(C(C)CC(N)=O)C)ONC(=O)C1(C(N)=O)CC1 35557,C1(CC(C)C)(C(N(CC(C)NC(CCC=CC)=O)C)=O)CCNC1=O.C(C)(=O)O 35558,C1(CC)CN(C(=O)OC(C)(C)C)CCC1CNCc1coc(C)n1 35559,c1(C(CC)O)nc(C2CCC(=O)N2C)n(-c2nc(C)nn2C)n1 35560,N1(C(CCCCOCC)=O)CCN(C(c2ccnnc2NC(C)C)=O)C(C)C1C 35561,C1(F)(C(=O)OCC)CN(C(=O)C(C2CC2)SC)CC1CN 35562,N1(C(c2onc(CC)n2)=O)CC2(CCN(C(=O)Cc3cccs3)CC2)C1 35563,c1(C(=O)NC2C(CNC(C(C)NC(c3ccoc3)=O)=O)CC2)cc(Cl)c(Cl)n1C 35564,c1(OC)ccc(F)cc1C(=O)C(=O)NC1CCN(C(c2ccc(C)o2)=O)C12CC2 35565,N1(C(c2ccc(C)c(I)c2)=O)CCOCC(F)(CNC(=O)Cc2ccn(C)n2)C1 35566,C1(C(=O)NCC(CC=C)NC(c2cc(CCC)oc2C)=O)CC2C=CC1C2 35567,CC(C(=O)NC(C(=O)NCC1(CO)CCC1)c1cccs1)OC1CCCC1 35568,C(=O)(CCCC(C)(C)C)N1CCC(CN(C(=O)Cc2cn3ccsc3n2)C)C1 35569,Cc1cc(O)nnc1C(=O)NCC1CC(NC(=O)C(C)(C)c2nncn2C)C1 35570,c1(CC)c(NC2CCN(C(C3(F)CCOC3)=O)CC2C)nc(C)nc1Cl 35571,N1(C(c2nnn(CC)c2C)=O)CCC(C2(NC(c3[nH]ccc3C)=O)CC2)CC1 35572,[N-]=[N+]=NCCCC(=O)NCC1(O)CC(CNC(=O)CCc2csc(=N)[nH]2)C1 35573,c1(C(=O)NCCC(=O)NCCNC(c2cc(C)c(C)[nH]2)=O)cc2ccccc2o1 35574,C1(CN(C(=O)C(C)(O)C2CCC2)C)CCCN1C(=O)COCc1cccnc1 35575,N1(C(C(CC)OCC)=O)CCC2(CCCN2C(=O)C(c2ccccc2)SC)CC1 35576,n1(CC)nc(C)cc1C(=O)NCC1CC1NC(=O)C(C)(C)n1ccc(C2CC2)n1 35577,C1(CC)CCN(C(c2ccc(SC)s2)=O)C1C(=O)Nc1cnn(C)c1SC 35578,N1(C(C(C2CCOC2)NC(c2c(CC)ncnc2)=O)=O)CCC(CO)C(O)C1 35579,N1(C(Cn2c(C)nc(C)n2)=O)CC2(COC(CNC(=O)CN3CCSCC3)C2)C1 35580,N1(C(c2cnn(C(C)C)n2)=O)CCC2CN(C(c3cnccn3)=O)CCC2C1 35581,C(=O)(CCS(=O)(=O)C(F)(F)F)NCCCC(C)NC(C(CC)(C)OC)=O 35582,C=CCC(C)C(=O)NCC1(C(=O)NCCSC2CC2)CC=CC1 35583,CC(C)(C(=O)NCC(O)CNC(C1(n2ccnn2)CC1)=O)C(F)(F)F 35584,Cc1c(F)ccc(C(=O)NC2CCC(NC(C3CCCCC3C)=O)CC2)c1C 35585,C1(NC(C(C)OCCCCCC)=O)C=CCN(C(=O)CC2(C3CC3)CC2)C1 35586,Cc1cc(C)c(C=CC(=O)NC2(CO)CCN(C(=O)C3=CCCS3)CC2)cc1C 35587,C(=O)(C1=CCC2CCC1N2C(=O)CC1CCCNC1=O)N1CCC(C)(O)CC1 35588,C1(CCNC(CCc2cc(OC)no2)=O)COCCN1C(c1coc(SC)c1)=O 35589,N1(C(c2nscc2Br)C(=O)NC(C2CC(N(CC)CC)C2)=O)CC2CCC2(C)C1 35590,c1(C(=O)NC2CN(C(C(CCCC)N(C)C)=O)CC2C)c(Cl)ccc2ccoc12 35591,c1(NC)ccc(S(=O)(=O)N(CCN(C(c2cc(CC)on2)=O)C)CC)cc1 35592,CCC(CC)CCCC(=O)N1CC2CCC1C(CNC(=O)CC1COCCO1)C2 35593,N1(C(c2scc(CNC(C(C=CC)O)=O)c2)=O)CCc2c(cnn2C)C1 35594,CC(=O)CCN=C(NCC1COC(=O)O1)NCC1CCCCS1 35595,C12(CNC(C3CCN(C(C4CC45CCCC5)=O)CC3)=O)CCC(CC1)O2 35596,C(N=c1nc(C(=O)OC)c(Cl)c[nH]1)C1CCCC(NC(C(CCC)(C)CC)=O)C1 35597,c1(OC)cc(C(=O)NC(CNC(C2CCCC23CC3)=O)C2CC2)c(F)cc1N 35598,C(=O)(C(C)C(O)CC)NCC(CC=C)NC(c1cncc(SC)c1)=O 35599,C1(CNC(C=Cc2n(C)cnc2)=O)CCN(C(=O)C=CC(=O)NC2CC2)C12CC2 35600,c1(C(=O)NC2CN(C(C(CC)OC3CCCCC3)=O)CC2F)cc2sccc2[nH]1 35601,c1(C(N(CCNC(C2N(C(C)=O)CCOC2)=O)C)=O)c([N+](=O)[O-])cnn1CCO 35602,C1(CNC(c2c(CC)noc2)=O)CN(C(C2CC3CC3C2)=O)CCC1C 35603,Cc1cc(C(N2CCOC(C(C)NC(C3CCCCO3)=O)C2)=O)cc(C)c1F 35604,C1(NC(C(CC#C)C)=O)CS(=O)(=O)C2CN(C(=O)CNC(=O)OCC)CC12 35605,C1(C(=O)NC2CC(NC(C3CC4(CC4)C3)=O)C2)CCC12CCCO2 35606,c1(C(=O)NCC(CNC(c2cncc(OC)n2)=O)C)cc(C)c(Cl)cn1 35607,S(=O)(=O)(c1ccnc(CN)c1)NS(C)(=O)=O.c12ccc(cc1)c(=O)[nH]2 35608,C12CCC(C1)n1cc(nn1)C1(CCCC1)C(=O)N2C.C1(CCCO)(CSC)CC1 35609,N1(C(C(C)C#N)=O)CCC2(CC1)CN(C(c1ccc3nn[nH]c3n1)=O)CCO2 35610,c1(C(=O)NC2C(NC(C3CCC(=O)NC3)=O)C2)ccc2c(c1)C(=O)CCO2 35611,C1(c2nnnn2C(C)C)(Cc2cn(CC)nc2)CC(C)(C)C1.C1(=O)NCCN1 35612,CC1CC(CNC(=NCCN2CCCC2(C)C)NCc2ccccc2)CC(C)O1 35613,N#Cc1cc(NC(C2CC2C(=O)NCCc2ccc(Br)s2)=O)c(F)cc1F 35614,C1(C2CCOCC2)(C(=O)NC2CCC3CCNC23)CC1 35615,C(C(C(=O)NCCN(C(=O)C(C)(C)n1ccnn1)C)C(C)(C)C)OCC=C 35616,C(CC(C(=O)Nc1ccc(C2CC2)nc1)OC)NC(COCCCCC)=O 35617,Cc1c(C(F)(F)F)n[nH]c1C(=O)NC(C)CN(C(=O)C(n1cc(Cl)cn1)C)C 35618,C(=O)(CCCCCC#N)NCC1(C(=O)NCC2(C)CCN(C)C2)CC1 35619,c1(C(=O)NCCCC(C)NC(c2ccncc2Cl)=O)cccn(C)c1=O 35620,c1(C(N2CC(NC(C3(COC)CC3)=O)C(C3CC3)C2)=O)oc2ccccc2c1Cl 35621,c1(CNCC2N(CC(C)C)CCC2)n[nH]c2cc(F)ccc12 35622,c1(N(C)Cc2ccn(C)n2)nc2c(c(=NCc3nc4ccccc4s3)[nH]1)COC2 35623,CCC(CCC(=O)N(CC(C)(C)CSC)C)NC(=O)CC(CC)SC 35624,C1(CC(C)NC(C=C(COC)C)=O)CCN(C(=O)C(N2CCCCCC2)C)CC1 35625,c1(NC(C2CN(C(Cc3nc(C)on3)=O)CC(F)C2)=O)ccc(C#N)cc1Br 35626,C1(CNC(C(C)(CO)OC)=O)CN(C(=O)CCc2nnc(O)nc2O)CC1(C)C 35627,c1(C(=O)OC)[nH]c(C)c(C(=O)N(C2CCC(NC(C3CC(C)C3)=O)CC2)C)c1C 35628,c1(C(=O)NCCCC(C)NC(c2cc(CC3CC3)on2)=O)cc[nH]c(=N)c1 35629,N1(C(C(CN=[N+]=[N-])NC(=O)CCCn2ccnn2)=O)CC2CCC(O)C2C1 35630,n1(Cc2cc(OC)ncc2CSCC(=O)OC(C)(C)C)cnc2ccccc12 35631,c1(CC)ncc(C(=O)OCCSc2cccnc2)c(C)n1 35632,c1(OC)nccc(C(=O)NCc2occc2C(=O)NC(c2ccncc2)C)n1 35633,C1(F)(CNC(CN(C2CC2)CC)=O)CCCN(C(=O)CS(C)(=O)=O)CC1 35634,c1(C(=O)NCC(=C)CCNC(c2cncc(N(C)C)c2)=O)cccc2ccnn12 35635,c1(CN2CCN(Cc3cc(OC)ncn3)CC2)ccc(C(F)(F)F)c(F)c1.C1CCN1 35636,C1(COC)(CNC(C2CC(N(C)C)C2)=O)CN(C(=O)C(n2ccc(C)n2)C)C1 35637,N1(C(c2cc(CC)ncc2)C(=O)NCC2CCOC2)CCCC(C)(C)CC1 35638,c1(CC(N2C(C)CC(NC(CC(CC)C3CC3)=O)C2)=O)ccc(O)c(C)c1 35639,C(=O)(CCCCCNC(=O)CCCOc1ccc(Br)cc1)N(C)C 35640,c1(C(=O)NCC2(F)CCC(NC(COCCC(C)C)=O)C2)cccc2occc12 35641,NC(=O)C1CN(C(C2CC3(C2)CC3(F)F)=O)c2ccccc21 35642,C(C)(CCC(=O)N1CCN(C2CCC(NC(C3(C)CCN(C)C3)=O)C2)CC1)OC 35643,c1(C(=O)OCC)cc(Br)c(Cl)nc1N.c12cc(ccc1C)C(=O)N2 35644,C1(C(N(C(C=C)C)C)=O)CCCCCC1NC(C1CC1(F)F)=O 35645,C(C)(C)(CC(=O)NC(C1CN(C(=O)CC2CCCS2(=O)=O)CCO1)C)SC 35646,c1(C(=O)NC2C(NC(CN(C)C(N)=O)=O)CCCC2)cc(N)ccc1Cl 35647,N1(C(CCS(C)=O)=O)CCC2C(C1)NC1(CC1)C(=O)N2.c1(NC(N)=O)ccccc1 35648,C1(C(N(CCNC(C2CC2CC2CC2)=O)C2CC2)=O)CCN(c2cnccn2)C1 35649,c1(C(=O)NC2CCCC2CC(=O)NOCCCC2CC2)cc[n+]([O-])cc1 35650,N1(CC(=O)NCC(C(C)C)NC(=O)CC2CCCCN2C)CCC(=O)NC1=O 35651,c1(C(N(CCCN(C(=O)C=CC2CCOC2)C)C)=O)cc(C(F)(F)F)cc(N)c1 35652,C(=O)(CC(C(C)C)NC(C1CN(CC)CCO1)=O)N(CC=C)C 35653,C1(C(=O)NC2C(NC(C=CC(=O)OCC)=O)CC2)CC(=O)N(c2cnn(C)c2)C1 35654,C1(C)(NC(C(C(C)O)NC(C2C(=C)C2)=O)=O)CC2(CCC2)C1 35655,C(=O)(CS(=O)(=O)CCC)N1CC(CCNC(CCC=CCC=C)=O)OC(C)C1 35656,C1(N(C(=O)CN2CCSCC2)C)CCCC(NC(=O)C=CC2CCCC2)C1 35657,N1(C(C2(C3CC3)CCC2)=O)CCCN(C(N)=O)CC1.Cc1ccc(CC(=O)OC)o1 35658,C12(COCC(=O)NC3CC(C(=O)NCCCC4CCOC4)C3)CCC1C2 35659,N(C(=NCCCF)NCC1(C)CCC(=O)N1C)C1CC(c2c(C)cccc2)C1 35660,Cc1nc(NC(C2CC(C)CN2Cc2cnn(C)c2C)=O)cc(Cl)n1 35661,C1(CNC(C(CC=C)(C)C)=O)CC2CCC(C1)N2C(=O)CC1CC(C)C1 35662,Cc1nnc(NC2CCCC(NC(=O)C(C)CC(N)=O)C2)c(C#N)c1C 35663,c1(CN(C)C)ccc(C(=O)NC2COCC2CNC(=O)CN2CCCC2=O)o1 35664,C1(CC(=O)N(CCN(C(=O)CCC2CCOC2)C)C)CC2(CC2)CO1.c1(C)cnc[nH]1 35665,CC1=CC(NC(=O)CCOCCCNC(=O)C=Cc2cn(C)nn2)CCC1 35666,CC1CC2CN(C(=O)CCCCNC(=O)CCNC(=O)CCC(CF)CF)CCN2C1 35667,N1(C(C2CCCN(C(C(C)CC3CC3)=O)C2)=O)CC2(COCC(=O)N2)C1 35668,N#Cc1ccc(C(=O)NC2CCCC2CNC(=O)Cc2cccc(F)c2)o1 35669,C(=O)(CCC1CCc2ccccc21)OCCCCCOC(C)C 35670,C1(NC(=O)C=CC2CCCC2)CCN(C(C2CCCS2)=O)CC1F 35671,c1(NCCCCN(C)C2CC2)[nH]c(=NCCn2ccnn2)nc2scnc12 35672,n1(CCNC(CSCCC#N)=O)cnc(C(=O)NCC(C2CC2)OC)c1 35673,N1(C(c2cc(CC(C)C)on2)=O)CCCN(C(=O)CN2CCN(C)CC2)C(C)C1 35674,C(=O)(CC1=CCOCC1)N1CCC(C(C)(C)NC(=O)Cc2cccc(C#N)c2)C1 35675,C(N=c1cc(NCCSc2cc(F)ccc2Br)nc[nH]1)C1S(=O)(=O)CC1 35676,Cc1ccc2cc(C(N3CCC4CCC(C3)N4C(=O)COCCF)=O)ccc2n1 35677,CCC(C)CCC(=O)NC1CC2(NC(c3cccc(N(C)C)c3)=O)COC1C2 35678,C1(N(c2n(C)nnn2)CCO)CCN(C(=O)NC2(CF)CC2)CC1.c1ccccc1 35679,c1(C(=O)NCC(CC)(C)NC(=O)Cn2cccc2)cccc(C2CC2)n1 35680,c1(CCC(N2CC(OCCNC(C(C)=C(C)C)=O)C2)=O)ccc2ncccc2c1 35681,N1(Cc2ccc(C(=O)OC)o2)CC2C3C=CC(O3)C2C1.c12ncc(cn1)C(=O)NC2 35682,c1(C(=O)OCCOC(C2CCOC2=O)=O)ccc(-c2nc(=O)o[nH]2)cc1 35683,C1(CCC)(C(=O)NCC(CCOC)NC(=O)CCCCSC)CCNC1=O 35684,N1(C(COCCCC)=O)CC2ON=C(CNC(c3cccc4c3OCO4)=O)C2C1 35685,CCCC(C)CC(=O)NCCC(C)NC(=O)CSc1cc(F)ccc1F 35686,c1(C(=O)NCC2N(C(CCCC(=C)C)=O)CCC2)ccc2cc[nH]c2n1 35687,c1(OC(F)F)ncc(CNCCCC2CCC2)cc1Cl 35688,c1(N(C)C)ncnc2cc(C(=O)Oc3c(Cl)cccc3Cl)ccc12 35689,n1(CC(=O)N(C(C)CNC(c2ccc(-c3ccccn3)o2)=O)CC)cnc(=N)[nH]1 35690,CN=c1[nH]c(=NCc2ccccc2OC)[nH]c(=NCCC2CC3CCC2O3)[nH]1 35691,N1(C(C)=O)CCC2(CCC2NC(c2ccc3ncccc3n2)=O)CC1 35692,C#CCCCCCC(=O)NC1(CCOC)CCN(C(=O)C(c2ccccc2)O)C1 35693,C1(COC)(NC(=O)C=CSCc2ccco2)CCN(C(=O)Cn2nc(C)nc2C)C1 35694,N#CC1(C(=O)NC2CN(C(c3ccn4nccc4c3)=O)CC2F)CC12CCCC2 35695,c1(C(=O)NCCC(C)NC(c2c(CC)nns2)=O)ccc(C#N)n1C 35696,N1(C(C(=O)NCCC)CC2CCC(F)(F)CC2)CCCC2CN(C)CCC12 35697,C1(NC(CC(C)F)=O)CC12CCC(NC(=O)CCc1cn[nH]c1)CC2 35698,C(C(C(=O)N(C)CC1CCCCN1C(C1CCOC(=O)CC1)=O)C(F)(F)F)OC 35699,Cc1ccc(C=CC(=O)NCCCNC(c2c(-c3cccs3)noc2C)=O)cn1 35700,c1(OC)ncc(C(=O)NCC(CC(C)C)NC(c2cc(C)co2)=O)c(C)n1 35701,C(=O)(C(C)(C)CN(C(=O)Cc1ccsn1)C)NCCS(CC)=O 35702,N1(C(C2N(C(C)C)CCC2)=O)Cc2ccccc2C(NC(c2ns[nH]c2=O)=O)C1 35703,CC1(C(N2CCC(O)(CCNC(C3CCC4(CC4)C3)=O)C2)=O)COC(=O)N1 35704,c1(C(N2CCC(=C(C)CNC(=O)CC3CCCS3(=O)=O)C2)=O)ccc(N)c(Cl)c1 35705,c1(C(N(C(CNc2ncc(C#N)cc2Br)C2CC2)C)=O)cnc2c(c1)ncn2C 35706,c1(NC(=O)NC(CC2CCCC2)CO)cccc2nc(O)nc(O)c12 35707,CC(C)CC(CNC(=O)CC1CCCCOC1)C(=O)NCC1(C)COCCO1 35708,N1(C(c2nn(SCC)c(O)c2)=O)CCOCC(NC(=O)CN(S(=O)(=O)CC)C)C1 35709,N1(C(C2(C)CCC2)=O)CC2COCCC2(NC(=O)CC2CCNC2=O)C1 35710,C1(C(N2C(COC)CCCC2)=O)CCN(C(=O)CNC(N)=O)O1 35711,C1(NC(C2C(OCC)C2)=O)CN(c2nnc(C(N)=O)s2)CC2(CC2)C1 35712,c1(C(=O)NCC2C(NC(=O)C=CC3CCC3)CC2)cnc2[nH]ncc2c1 35713,Cc1c(C(=O)NC(CO)C(=O)NCC2CSCCO2)ncn1C 35714,CC(C)C(O)C(=O)NC(c1ccc(C(F)(F)F)cc1)C(N1CCOC(CN)C1)=O 35715,N1(C(C(CCC)O)=O)CCC2(CC1)CC2C(=O)NC(c1ccc(Cl)cc1)C(=O)OC 35716,CN1CCC(C)(C(=O)NCC2CCN(C(=O)Cc3cn[nH]c3)CC2O)CC1 35717,c1(C(N(CCN(C(C2CC(=C3CCC3)C2)=O)CC)CC)=O)c(C)n[nH]c1C 35718,C(C(C(=O)NCC1(C2(O)CCC2)CC1)C(C)(C)C)NC(C(COC)OC)=O 35719,c1(C(=O)NC(C)C#N)ccc2c(-c3cscc3C#N)nn(C)c2c1 35720,N1(C(C23CSCC2C3)=O)CC=CC(NC(C2(n3cnnn3)CC2)=O)C1 35721,C1(NC(c2ccn(C(C)C)n2)=O)CC2CC1N(C(c1ccc(O)nc1Cl)=O)C2 35722,Cn1cc(C(=O)NC2CCC(NC(C3(C)CCCCO3)=O)CC2)c(C(F)F)n1 35723,C#CC1CN(C(C2(F)CCCN(C(=O)C3=NNC(=O)C3)C2)=O)CCO1 35724,C1(C(=O)NC2(CC(=O)NC(C#C)CC3CC3)CC2)Cc2ccccc2C1 35725,C(=O)(C(C)(C)F)N(C1CCC(NC(=O)COc2ccsc2)C1)C 35726,N1(CC#C)CCC(OC(=O)NCCNc2ccccc2)C1 35727,c1(CC(=O)N(C2CC2CF)C)ccc(NS(C)(=O)=O)cc1.C12CCN(C1)C2=O 35728,C12(C(=O)NC(C(C)F)C)CC(CCO1)N(C(C1CN(C)C(=O)N1)=O)C2 35729,CCC(C)(C)C(=O)N(C)CC1C2CN(C(=O)CNC(c3cccs3)=O)CC12 35730,c1(C(N2CC(N(C(C3(CC)CC3(F)F)=O)C)C2)=O)ccccc1S(C)(=O)=O 35731,CCCC(C)(C)C(=O)NC(c1ccccc1)CNC(=O)CCCc1ccncc1 35732,c1(C(=O)NCC2CN(C(C3CCC(=O)NC3)=O)CC2O)[nH]cc2c1CCC2 35733,N1(C(Cn2nnc(C)n2)=O)CC=C(C(=O)N2CCC(OC3CC3)CC2)CC1 35734,C(=O)(CCCCC(F)(F)F)NC1C(C=C)CN(C(=O)Cn2cnnc2)C1 35735,C(CC(C(C)(C)C)NC(c1cc(-c2c[nH]c(=N)c(C)c2)no1)=O)OC 35736,CCCCCCC(c1nnnn1CCOC)Sc1c(C)nn(CC(F)(F)F)c1Cl 35737,Cc1cnc(F)c(C(N2CCC(NC(c3cc(C(N)=O)ccn3)=O)C2C)=O)c1 35738,Cc1nnsc1C(=O)N(C1CCN(C(=O)C(C)Cc2ccccc2)C1)C 35739,CN1C(=O)OC2CN(C(=O)C(c3cn(C)nn3)NC(=O)C=CC(F)F)CC12 35740,c1(C(=O)NCCCN(C(C(C(=O)OC)OC)=O)C2CC2)cc2n(n1)CC(F)C2 35741,C12(C(=O)OC)CC1CN(C(=O)CC(O)CNC(c1cc(C3CC3)[nH]n1)=O)C2 35742,c1(C(N2C(C(=O)O)CCC(C)C2)=O)coc2c1CN(C(=O)CC1CCC1)C2 35743,C1(C(N2C(CN(C(C(N3CCCC(O)C3)C)=O)C)CCC2)=O)CCC(F)(F)CC1 35744,N1(C(CSCc2ccc(C)cc2)=O)CCC(C2CCCN(C(=O)C(C)O)C2)C1 35745,c1(C(=O)NCC(CC)NC(c2cnsc2C)=O)n[nH]c(C)n1 35746,C(=O)(C1=CCCCCC1)N(CC(CNC(c1c(C(=O)OC)c(C)[nH]n1)=O)O)C 35747,n1(CCCC)nccc1C(=O)NC1(C2CCCN2C(=O)C(C)N(C)C(C)=O)CC1 35748,CC1=C(C(=O)C(=O)CCCCCC#N)COCC1.C1(CN)(C)CC1(F)F 35749,CCCC(C)CC(=O)NCC(O)CNC(=O)COc1ccc(CC#N)cc1 35750,N1(C(C=CC(=O)OC)=O)CC2CC(C(=O)NCCc3cnco3)CC2C1 35751,C1(NC(=O)CC2CC(C(F)F)C2)CN(C(=O)Cc2cncs2)CC1C1CC1 35752,N1(C(=O)NCCCC)C(C)CN(c2ncnc(C)c2F)CC1C 35753,Cc1ccc(C=CC(=O)NC2CC2NC(c2cnc(C(C)(C)C)s2)=O)cc1C 35754,c1(C(=O)NCC(C)CNC(=O)CCNC(C2CC(CCO)C2)=O)ccccc1 35755,c1(OCC)ccc(NC(c2occc2COC)=O)cn1.C12CC(C1)NC(=O)C2 35756,N1(C(C(CC)(C)COC)=O)CC(NC(c2cnn3ccccc23)=O)C2(CCC2)C1 35757,C1(C(=O)NCC(C2CCCC2)CNC(=O)CCCCC2CC2)CCC(CO)CC1 35758,CC(C)CCC(=O)N1CC(NC(=O)CCC(C)O)CC1C 35759,CC#CCC(C(=O)NC(C1CN(C(C2(O)CC2)=O)C1)C)NC(=O)OC(C)(C)C 35760,Cc1cc(F)cc(Br)c1C(=O)NC1CC2CCC(C1)N2C(C1CC1C#N)=O 35761,c1(C(=O)NC(CC(F)F)C(=O)NCC(O)CCO)ccnc2cc[nH]c12 35762,c12cccc(c1)S(=O)(=O)NC2=O.Cc1cccc(NCCCS(N)(=O)=O)c1C 35763,c1(-c2c(NC(C3(c4ccc(C)c(Cl)c4)CC3)=O)cccc2)c(C)c(C)n(C)c1C 35764,C#CC1(NCC)CCN(C(C)(C)C)CC1.C12CN(C)C(C)(C1)C(=O)O2 35765,c1(SCC(=O)N(CCN(C(C)C)C(c2cc(Cl)c[nH]2)=O)C)ccc([N+](=O)[O-])cc1 35766,C1(S(C)(=O)=O)(C(=O)NC(C2CCOC2)CNC(CC=CC=C)=O)CC1 35767,c1(C(=O)OCC)nnc(NC(C2CCN2C(=O)C(C)(C)n2cccn2)=O)s1 35768,c1(C(N(C2CC(NC(C3CCCO3)=O)C2)C)=O)c[nH]cc(F)c1=O 35769,N1(C(CCC#C)=O)CCC2CCC(NC(=O)C(F)CC3CCCC3)C12 35770,CC1(C)CCC(C(N2CC3CC3(CNC(c3ccc(Cl)o3)=O)C2)=O)O1 35771,N1(C(c2scc(C(C)=O)c2)=O)CC(O)CC1CNC(=O)CCOC1CCOCC1 35772,c1(C(N(C)CC2(O)CN(C(CC=CC=C)=O)C2)=O)cc(S(N)(=O)=O)cs1 35773,CCC1=NOC(C(=O)NCCC(O)CNC(=O)C(F)(F)CO)C1 35774,CC1(F)CN(C(c2c(Cl)ccnc2F)=O)CCN(C(c2c(F)ccnc2Cl)=O)C1 35775,c1(CC)ccc(C(N2CC(C(C)NC(=O)C=Cc3cncn3C)C2)=O)cc1CC 35776,N1(C(CSC)=O)CC2CC(C(=O)NCCC(O)CO)C(C2)C1 35777,C1(NC(c2cnc(NC(C)=O)o2)=O)CCCCN(C(C2(C)CCCNC2=O)=O)C1 35778,CCCCCCCCCC(=O)NC1CN(C(c2cc(C(N)=O)c[nH]2)=O)CC1(C)C 35779,C(=O)(CC(C)(C)CNC(C1C(C)(C)C1(F)F)=O)NCc1nc(CC)sc1 35780,C12(C(=O)NCC(CN(C)C(C3CC4CC4C3)=O)O)CC(C)(C1)OC21CCC1 35781,C(=O)(C(CO)C(F)(F)F)NC(CCC=C)C(=O)NC1CCOC1C 35782,C(=O)(C(F)C(F)(F)F)N(C)CCNC(C1CCC(Oc2ccncc2)C1)=O 35783,C1(C(N(CCCF)C)=O)CCCCN(C(C2(N(C)C)CC2)=O)C1 35784,CC1CC(=O)NC(C(N2CC(NC(c3cn(CCC(C)(C)C)nn3)=O)C2)=O)C1 35785,c1(-c2c(CN(CC(O)CO)CC)nccc2)ccn(C(C)C)c(=O)c1 35786,c1(C(N2C(CC)CN(C)CC2)=O)ccc(S(=O)(=O)NC(C)C)cc1 35787,c1(CN=C(NC(C#C)C(C)(C)OC)NC2CCC2)ccc(C#N)cc1Cl 35788,CCC(C)C(C(=O)NCC(C)(C)CNC(=O)CN(c1ccccc1)C)OC 35789,Cc1cc(C)c(C(=O)NC2CC23CC(NC(C2CCC(C)(C)O2)=O)C3)[nH]1 35790,C(C(=O)NCCC#N)(C(C1CCC1)NCc1cc(C)on1)N(CC(C)C)C 35791,CCCCCC(CC)C(=O)NC(CNC(c1nocc1C)=O)CO 35792,c1(C(=O)NCC(CN(C(C(CC)n2nccc2C)=O)C)O)cc2cccnn2n1 35793,c1(C(=O)NC2C(NC(C(C)O)=O)COC2)cnc(C(c2ccco2)C)nc1O 35794,CCCC(C(=O)NC)NC(=O)C=CC(C)NC(C1CC(C)(C(=O)OC)C1)=O 35795,N1(C(CCNC(=O)C=CCl)=O)C(CNC(=O)Cc2ccon2)CC2CCCC12 35796,c1(CN(CCC(=O)NCC(O)CCC(F)(F)F)CC)nccc(C)n1 35797,C1(CN(C(=O)CC(F)(F)F)CC)CCCCN1C(C1CCC1n1cccn1)=O 35798,N1(C(C=CS(C)=O)=O)CC(NC(=O)Cc2cccc3c2CCC3)C(C2CC2)C1 35799,C(C(C)C(C)C(=O)NCC1(C(=O)NC2CCC(=O)N(C)C2)CC1)OC 35800,C1(CN(CC(C)(C)Cn2cc(-c3c[nH]c(C(=O)O)c3)nn2)C(C)(C)C)C(F)(F)C12CC2 35801,CCC(Cc1ccccc1C)C(=O)N1CC(NC(c2csc(CO)n2)=O)C(C)C1 35802,C1(CNC(CC2CC(C)C2)=O)CCN(C(=O)C(c2nccn2C)=O)CC1 35803,c1(C(N2CCC(NC(C3CCCOCC3)=O)CC2)=O)cc(F)c(O)c(F)c1 35804,C1(CC=C)(NC(C2CCC(=O)N2C)=O)CCN(C(c2ocnc2C2CC2)=O)C1 35805,C1(C=O)(COC)CN(C(c2ccc(CO)o2)=O)C1.N(CC)CC1CC1 35806,N1(C(C2(C)N(C(Cc3c(C)ocn3)=O)CC=C2)=O)CCC(N=[N+]=[N-])C1 35807,N1(C(C(C)N=[N+]=[N-])=O)CC2CCCC2(CNC(c2cnnc(O)c2)=O)C1 35808,C(=O)(C(C)(C)CCCO)N(C1CCCO1)CC1CCN(C(C(C(C)(C)C)O)=O)CC1 35809,Cc1nocc1NC(=O)CNC(=O)CNC(c1ccc(F)s1)=O 35810,N1(C(CC2CC(=C)C2)=O)CCCC(O)(CN(C(=O)CCCn2cccn2)C)C1 35811,C1(C(=O)NC(C)CNC(C2CC(=O)N(c3nccs3)C2)=O)C2C3CCC(C3)C12 35812,N1(C(C(CC)(CNC(C2CCOC(=O)CC2)=O)CC)=O)CC2(COCC(=O)N2)C1 35813,N1(C(=O)NCC2CCCNC2)CC2CCCC(N)C2C1 35814,c1(C(=O)NCC(C)(C)Nc2nc(COC)nc(Cl)c2)ccc2c(c1)nc(O)n2C 35815,c1(OC)cc(C(=O)NCC23CC2CN(C(c2n[nH]cc2C)=O)C3)nc(Br)c1 35816,C1(C)(CNC(CN(C)C(N)=O)=O)CN(C(=O)CC2CCCC23CC3)CCO1 35817,C1(CNC(CCC(C)OC)=O)CN(C(c2nnn(C(C)C)c2C)=O)CC(C)(C)C1 35818,N1(C(C2OCC(C)(C)C2)=O)CC2CCN(C(c3nccc(Cl)c3O)=O)C(C2)C1 35819,c1(C(=O)NCC2(C(N)=O)CN(C(C3C4CCCOC34)=O)C2)ccc(Cl)c(F)c1F 35820,c1(OC)cccc(CC(=O)NC2CCCC(NC(c3cocn3)=O)C2)c1F 35821,N1(C(Cc2c(C)n(C)cn2)=O)CC(NC(C2(Cl)CC2(F)F)=O)CC(C)C1 35822,C1(C(=O)NC(C2(O)CCN(C(=O)CC3CC3)C2)C)C2CCC1(c1ccccn1)C2 35823,c1(CC)ccc(C(=O)NCC(CO)NC(c2ccc(C)cc2C)=O)cc1C#N 35824,n1(CC)cncc1COC(=O)CCc1cc(C)on1 35825,c1(C(=O)OCC2(OC)CCSCC2)c(Cc2ccccc2)oc2ccccc12 35826,c1(C(N2CC3CN(C(c4c(C)noc4C)=O)CC32)=O)c(F)cc(F)cc1Br 35827,CC1(C)CCC(C(N2CCOCC2c2cn(Cc3cccc(Cl)n3)nn2)=O)O1 35828,CC(C)(CC1CCOC1)C(=O)NCC(=O)NCC1CCN1CC1CCOCC1 35829,N1(C(CCC(C)SC)=O)CCC(NC(C2(C(F)(F)F)CC(F)(F)C2)=O)CC1C 35830,C1(NC(C2(OCC)CCSCC2)=O)COCCN(C(c2csnc2Cl)=O)C1 35831,N1(C(=O)CCc2cc[nH]n2)CCC2(CCCN2C(c2ccccc2Cl)=O)C1 35832,O=C(CC1CCNc2ccccc21)NCCN1CCN(C(C23CC(C2)C3)=O)CC1 35833,N(C1=NC2CCCCC2S1)c1cc(N2CC3(CC(COC)OC3)C2)nc(C)n1 35834,C(C(C)(C)CNC(=O)C(CC1CC1)NC(=O)CCOC(C)=O)OC.C(C(C)(C)C)O 35835,c1(C(=O)NC2CC(NC(C3(CCO)CC3)=O)C23CCC3)nnn2c1CSCC2 35836,C(=O)(C1=CCS(=O)(=O)C1)N(C)CC1CCCN1C(=O)CC1CCCC(=O)N1 35837,C#CCC(CC(=O)NC(c1cccc(C)c1)C)NC(c1ccc(O)nc1)=O 35838,c1(C(N2C(C3CCN(C(Cc4n(C)ncc4Cl)=O)C3)CCC2)=O)coc2c1COC2 35839,Cc1nn(CC(N2CC3CC3(CNC(=O)C(C)(C)C3CCCCO3)C2)=O)c(=O)o1 35840,C1(C(=O)NCC2(OCC)CCC2)CC2C=CC1N(C(=O)C1=CCCCC1C)C2 35841,N1(C(C2CCC(C)O2)=O)CC(CNC(c2cc3ccccc3o2)=O)OC(C)(C)C1 35842,C1(N(C(CN(c2ccccc2)CC)=O)C)C2CN(C(=O)C(F)=C(C)C)CC12 35843,N1(C(C=CC)=O)CCC2(NC(c3cccc(Br)c3C)=O)CCCCC12 35844,c1(C(N2CCCC(C(=O)Nc3cnc(Cl)nc3)C2)=O)cnc2ccccn12 35845,N(C1CCc2cc(CNC(c3cn(C)nc3C)=O)ccc21)C(C(CCC#C)O)=O 35846,c1(C(=O)OC)ccc(C(=O)NC2CC3C=CC2C3)c(C(C)C)c1 35847,CC1(NC(c2nsnc2O)=O)CCN(C(C2CC3CC2C3)=O)C1 35848,C1(c2ccc(OC)cc2)CSCCCN1Cc1sncc1Br 35849,C1(C(=O)NC2COCC2NC(c2cnc(O)s2)=O)(OC)CCOCC1 35850,Cc1nc(Cl)ncc1NC(=O)CC1C2CCC(C2)N1C(=O)COC1CCOC1 35851,C(CC)(CC(=O)N(C1CCOC1C)C1CC1)N(C(CC=CCC)=O)C 35852,S(=O)(=O)(c1cccc(CNC(c2oc(C)nc2CN)=O)c1)N(CC)CC 35853,Cc1cc(F)ccc1C(=O)N(C1CCCN(C(=O)CCc2scnc2C)C1)C 35854,Cc1cc(C(=O)N(CCCCNC(c2ccc(CO)nc2)=O)C)c(Cl)cc1F 35855,N1(C(C2(C)C=CCN2C(C2CN(C)CCN2C)=O)=O)CC2(CO)CC2(CO)C1 35856,C(CC(=O)N(CC(C)CNC(c1csnc1C1CC1)=O)C)(C(C)C)OCC 35857,CC(=O)n1ccc(CNC2CC(C(=O)NCc3ccc(Cl)cc3)C2)c1 35858,c1(OC)nccc(C(=O)NCC2CN(C(C3(n4cncn4)CC3)=O)C2)c1F 35859,c1(NC(C2C(NC(c3c(C(C)C)cccc3)=O)CCC2)=O)cccc2c1OCO2 35860,C(c1cnn(C)c1)=CC(=O)NCC(COC)NC(c1csnn1)=O 35861,c1(C(=O)NC(C)C(CO)NC(c2cnc3ccccn23)=O)cccc2nn[nH]c12 35862,c12cc(Br)ccc1NCC2.n1(CCSC)nnnc1C(c1sccc1Br)OC 35863,CCCCN=C(NCC1(O)CCC1)NCC1CCCCN1S(C)(=O)=O 35864,CC1CN(C(=O)CNC(c2cc(CSC)cn2C)=O)CCCN1C(C1CCC1)=O 35865,C(=O)(CC(C)CN(CC)CC)N(CCNC1(C(N)=O)CC1)CC 35866,C1(NC(c2cc(CC)sn2)=O)C=CCN(C(c2nonc2N)=O)C1 35867,c1(C(=O)NC(CC)CNC(C2CC3CC2C3)=O)cc(C(C)C)cc(C(C)C)c1O 35868,c1(OC)ccc(F)c(-c2ccnc(NC(C3CC(C)(C)C3)=O)c2)c1 35869,CCC(C)CC(C(=O)NC1CN(C(C23CCC(C2)C3)=O)C1)NC(=O)OC(C)(C)C 35870,CCC(C)(C)OCC(=O)NCC(C)CN(C)C(C1(C(C)(C)O)CC1)=O 35871,N1(C(c2c(C)nccn2)=O)CCN(C(=O)CC2(O)CCOC2)C(CC2CC2)C1 35872,C1(NC(CCCC(N)=O)=O)CC2CC1CN(C(C1(c3cnccc3Cl)CC1)=O)C2 35873,N1(C(C2(CC)CCCC2O)=O)CC2CCC1CN2C(=O)Nc1c(C)cccc1C 35874,C1(NC(c2cc(SC)c(C)o2)=O)(CNC(c2nccn2C)=O)CCCCC1C 35875,C1(C2CCN(C(=O)CCOCC(F)F)CC2)(NC(CC2C(C)CCC2)=O)CC1 35876,CC1(CNC(C2CC(C(F)(F)F)C2)=O)CCN(C(C2CC(F)(F)C2)=O)C1.C(F)F 35877,Cc1ncc2n1CCC(C(=O)NC1(CF)CCN(C(c3ccncc3Cl)=O)C1)C2 35878,C#CCCCCCC(=O)N1CCC2CN(C(=O)C(F)(F)C(O)CC)CC12 35879,CCCCC(C)CCC(=O)N(CC(=O)NCCOCC1CCOCC1)CC 35880,c1(C(N2C3C(NC(C4CC(OCC)C4)=O)CC(C3)C2)=O)sc2ccccc2c1Cl 35881,c1(OC)cccc(C(N2CCC(O)C(F)C2)C(=O)NCCC#N)c1Br 35882,c1(NC(C2(CC)CCOC2)=O)ccc(NC(=O)C(n2cc(C)cn2)C)cc1C 35883,C12(CNC(CC(C)SC)=O)COCCN1CCN(C(C1CN3CCN1CC3)=O)C2 35884,CSC1=C(C(=O)NCCC2(CNC(=O)C(n3ccnc3C)C)CC2)CCCC1 35885,N1(C(c2n(CC)ncc2)=O)CC(NC(c2cncc(Cl)c2)=O)C(O)C1 35886,N1(C(Cc2cn(C)nc2)=O)CC(NC(C2CC3CCC3C2)=O)C2(CC2)C1 35887,C1(C(=O)NCC23CN(C(CCN(C)CCO)=O)C(C2)CO3)CNc2ccnn2C1 35888,C1(CC)CCN(C(C2C3CN(C)CC23)=O)C1CNC(c1ccsc1OC)=O 35889,C1(N(C(C=Cc2ccc(SC)s2)=O)C)CN(C(C2(CCF)CCC2)=O)CC12CC2 35890,c1(C(C(=O)O)C2(C3CN(C(CC(F)(F)F)=O)C3)CC2)ncccn1 35891,C1(CNC(C2(CC(=O)OC)CC2)=O)C2CCCC1N(C(c1[nH]cnc1C)=O)C2 35892,c1(OC)ncnc(C(C)C)c1-c1nc(C2CCC(F)(F)CC2)nn1C 35893,CCCCCCCCC(=O)N1CCC(C(C)NC(=O)CC2(O)CCOC2)CC1 35894,N1(C(C2(CC=C)CC2)=O)CCC2(CC1)CC2(CO)CNC(=O)COC 35895,Cc1nc(NC2(CNC(C3CN4CCN3C(C)C4)=O)CC2)c2cc[nH]c2n1 35896,Cc1c(C(=O)NC2CC23CC(NC(C2CCC4CC24)=O)C3)oc2ccc(F)cc12 35897,c1(C(=O)NC2C(O)CCN(C(C(C)CC(C)(C)C)=O)C2)ccc2c(c1)OCCN2 35898,C1(OC)CC(CNC(=O)C(=O)Nc2cccc(F)c2)N(C(c2ccc[n+]([O-])c2)=O)C1 35899,c1(CC)cc(C(=O)NC2CCCC2CC(=O)NCCCC(C)(F)F)ncn1 35900,c1(C(=O)NC2C(NC(c3cc(C)nc(C)c3)=O)COC2)cc2nccn2c(O)n1 35901,C1(C(=O)NC2CCN(C(Cn3c(C)nnn3)=O)C2)CCc2nc[nH]c2C1 35902,N1(C(CC2COCC(C)O2)=O)CCCCC2(C1)CN(C(=O)CCn1cccc1)C2 35903,C1(NC(=O)CC2CC2C(F)(F)F)CCCCN(C(=O)C=Cc2ccccc2)C1 35904,CCCC(C(=O)NCC1(C)CCCN1C(=O)C(F)C(C)C)OCC 35905,C(CC)(CCC)(c1nnnn1CCCSCC)NC1(C)CC(=C)C1 35906,S(=O)(=O)(c1ccc(NCCCC(C)(C)C)c(F)c1)N1C(C(C)C)CC(O)C1 35907,CCCC(C)(O)CC(=O)N1CC(CC(C)NC(c2cc(C3CC3)ccc2Cl)=O)C1 35908,N1(C(C(C)=C2CC2)=O)C2CCC1C(C(=O)NC(c1ccns1)C)C2 35909,c1(C(N2CCC(C(C)O)C2)=O)cc2ncc(-c3ccn(C)c3)cc2[nH]1 35910,N1(C(C2(C)COC2)=O)CCN(C(=O)Nc2cc(Cl)cc(Cl)c2)C2CC12 35911,N1(C(c2nc3nc(C)cc(C)n3n2)C(=O)NCC=C)CCC(C2CC(F)(F)C2)C1 35912,c1(C(=O)NCC(C)N(C)C(c2ccncn2)=O)coc2ccc(O)cc12 35913,CC(CCc1ccccc1)CC(=O)NC(C)(C)CCNC(c1ncccc1Cl)=O 35914,Cc1[nH]nc(CNC(=O)C(c2cccs2)NC(=O)C=Cc2cncs2)c1C 35915,c1(OC)cc(C(N2CCC(CC(=O)OCC(C)C#N)C2)=O)on1 35916,N1(C(C=NOC)=O)CC2CC(NC(C3(C4CCCO4)CC3)=O)C2C1 35917,C1(COC)CN(C(c2cc(Br)c(C)cn2)=O)CCN1C(c1cnc(O)[nH]1)=O 35918,c1(C(=O)NCCC2N(C(CSc3onc(C)n3)=O)CCC2)c(C)cccc1C 35919,Cc1c(C(=O)NCC(O)CCNC(=O)C(C)C(C)C)cnn1CCN(C)CCO 35920,Cc1ccc(C(N2CCCC(C)(NC(=O)Cc3cscc3F)C2)=O)c(Cl)c1 35921,C1(C(=O)NC2(C(C3CCC3)=O)CC2)(CNC(=O)Cc2cc[nH]n2)CC(F)(F)C1 35922,N1(C(=O)NCc2ccc(C(=O)OC)o2)CCOC(C2CC(F)(F)C2)C1 35923,C(=O)(C1CCCn2cncc21)NC1CCN(C(C(=O)NCCC(N)=O)=O)CC1 35924,n1(CC(=O)N(CC(C)OC)CC)ccc2ncc(Br)cc12 35925,N1(C(CCC2C(C)(C)C2)=O)CCOC2(CCC(Nc3ncc(Br)cn3)CC2)C1 35926,N1(C(C)C)CCCC1CC(=O)N(C)CC1CCN(C(c2ccsn2)=O)C1 35927,C1(CCNC(CC(C)O)=O)COCCN1C(c1cncc(CO)c1)=O 35928,c1(C(N(CCNC(CCC#C)=O)C)=O)c(Br)ccc(OC)c1C 35929,[N-]=[N+]=NC1CN(C(C2CC2F)=O)CC1NC(c1c[nH]nc1-c1cnn2c1OCC2)=O 35930,Cc1[nH]c(C)c(C(=O)NCC2CN(C(c3cn(C(F)F)cn3)=O)CC2C)c1C 35931,c1(CC)onc(C)c1C(=O)NC1CCCN(C(=O)COCCCCC)C1 35932,Cc1ncc(Cl)cc1C(N1CC(CC(C)NC(c2cncc(F)c2Cl)=O)C1)=O 35933,N1(C(C(C(CC)C)O)=O)CC(NC(C2OCC2(C)C)=O)CC(C)(C)C1 35934,c1(SCc2cn(CC(C(=O)NC(C(C=C=C)C)=O)O)nn2)ccc2sccc2c1 35935,c1(C(=O)NCC2N(C(C3CC(C)(C)O3)=O)CCN(C)C2)ncnc2c1ccn2C 35936,C1(CCC)(CO)CCN(C(=O)C(CNC(=O)C(F)(F)COC)CC2CC2)C1 35937,c12cc3c([nH]cnc-3n1)N1CCC(=CCNC(=O)COC2=O)CC1.C(C)(=O)OC 35938,c1(C(=O)NC(CNC(c2ccc(C)nc2O)=O)(C)CO)nccc2ccccc12 35939,C1(C(N2CCCC(=C)C2)=O)CC1C1CN(C(=O)CC2C(=O)NN=C2C)C1 35940,Cc1cc(F)ccc1CNC(C1CC2(CC2)CN1C(=O)C(Cl)Cl)=O 35941,O=C1NC(=O)C2C3CCC(CC3Nc3cccc(F)c3[N+](=O)[O-])C12 35942,CC(C)=C=CC(=O)NCc1ccc(C(C)NC(=O)CCN2CCOCC2=O)cc1 35943,C(C(C(=O)N1CCOCC1CO)C(C)C)NC(c1cn(CC)nc1C)=O 35944,C1(CNC(=O)Cn2cnnc2)(NC(c2cc(Br)no2)=O)CCCC1 35945,C1(SC)CN(C(=O)CCN2CCCS2(=O)=O)CC1NC(=O)C#CC1CC1 35946,C1(C(=O)OC)CN(C(=O)CCCn2cc(CC3(O)CC(C(=O)O)C3)nn2)CC1F 35947,C12CCCCN(C1)C2.C(=O)(C(O)Cc1cn(CCC2(F)CC2)nn1)OC 35948,CC(CC(=O)NC1C=CC(CNC(=O)CCc2cnn(C)c2)C1)c1cnn(C)c1 35949,c1(OC)cc(C#N)ccc1C(=O)NC1CS(=O)(=O)CC1NC(c1ccncc1)=O 35950,C#CCCCCCC(=O)NCCCN1CCN(C(=O)CC2CSCCO2)CC1 35951,Cc1nc(C(C)NC(C2CCN(C(c3c[nH]nc3C)=O)C2)=O)n[nH]1 35952,c1(C(=O)NCCCCNC(C2CCCN(C(C)=O)C2)=O)cc(F)c(F)c(F)c1 35953,C1(C(=O)NC(CCC)Cc2ccccc2)CC2CC(=O)C1O2 35954,C1(CN(C(C2CC(F)C2)=O)CC)CCCN(C(=O)C2=CCSC2)C1 35955,C(=O)(CCCCC(C)(C)C)N1CCC(NC(COCc2ncc(C)o2)=O)C1(C)C 35956,Cc1nc(C2CCCCC2)nc(O)c1C(=O)NCC(C)C1CC1 35957,c1(C(N2CCC(NC(c3c(C=C)cnn3C)=O)C2)=O)c(Cl)ccc(F)c1F 35958,N1(C(c2n(CC#C)cnn2)=O)CCC(C)C1NC(C1CCOC1=O)=O 35959,C1(O)(C(=O)NC2CCN(C(C3CC(C(=O)OC)C3)=O)C(C)C2)CCC(C)(C)CC1 35960,N12CCC(F)(CC1)NCC(F)C2=O.c1(C(C(=O)N(CC)CC)C)cncnc1 35961,C1(N(C(C(=O)N(C)C)=O)C)CCCN(C(c2coc3c2COC3)=O)CC1 35962,n1(CC(=O)NC2C(NC(=O)CCc3ccon3)C2)ccccc1=O 35963,N1(C(C2CC(CCC)C2)=O)C2CCC(C(=O)N(C3COCC3(C)C)C)C1CC2 35964,N1(C(CCCOC(C)=O)=O)CC(F)(F)CC1CCNC(=O)COC1CC1(F)F 35965,Cn1nc(CC(N2CCCC2CCNC(=O)CC23COCC(C2)C3)=O)cc1Cl 35966,C1(C#N)(C(N2C(C)CN(C(CCC(C)OCC)=O)C(C)C2)=O)CC2CCC1CC2 35967,c1(OC)cc(C(=O)NCCN(C(=O)CCCc2cccc(Cl)c2)CC)cc(Cl)n1 35968,C1(C(=O)NCC2(OC)CC2)CCCCC1NC(=O)C(C)(C)C1CC1 35969,C1(C(=O)NC2C(NC(c3c(OC)ccs3)=O)CCCC2)CC2(CCCO2)C1 35970,Cc1cccc2c1CC(C(N1CCC(N(C)C(C3(C#N)CC(C)C3)=O)CC1)=O)O2 35971,Cc1c(C(=O)NC2CCC(NC(=O)CC(O)C(C)C)CC2)cccc1F 35972,c1(C(N(CC(C)NC(CC2ON=C(C)C2)=O)C)=O)cn(C)c(C)cc1=O 35973,N1(Cc2c(C)ccs2)CCCC(C(=O)NCC2=CCCCC2)C1 35974,c1(SC)ccc(C(=O)NC(C2CCCC2)CNC(C2C3CCCC23)=O)cc1 35975,N1(C(C=C)=O)CCCC1CC(=O)NC(c1ccccc1)Cc1cccnc1 35976,CN1CCC(C)(NC(=O)NCC(O)Cn2cccn2)C1=O 35977,C1(CNC(c2c(SC)cccn2)=O)CN(c2cnc(F)cn2)CC2(CCC2)O1 35978,C(=O)(CCCC(F)(F)F)NC(CCNC(C1(OC)CCSC1)=O)C 35979,c1(CC)cc(C(=O)NCC2CCCN(C(=O)CC3CC(F)C3)C2)cc(O)n1 35980,N1(C(C2(COC)CCCO2)=O)CCCN(C(c2cnn(C3CCC3)c2C)=O)CC1 35981,C1(CNC(=O)Cc2ccc(Cl)s2)CN(C(C2CC3(CCCO3)C2)=O)CC12CCC2 35982,N1(C(CCC=CC)=O)CCOC(C)C1C(=O)NCCC(C)C(C)C 35983,[N-]=[N+]=NC1COCC1NC(=O)Cn1cc(CN2CC3CC3C2)nn1 35984,C1(C(=O)NCC(CC=C)NC(=O)COC2CCCC2)CC2(COC(=O)N2)C1 35985,n1(CC)cc([N+](=O)[O-])c(C(=O)NCC(C)(C)OCCNC(=O)CSSC)n1 35986,N1(C(c2cc(OC)c(C#N)cc2)=O)CCC2CCC(C1)N2C(C1CC1CF)=O 35987,C1(C(=O)NC(CCC)C(=O)N2CCOC3CC23)CCCCC1(C)C 35988,CC(CC(C)NC(C1(n2ccnn2)CC1)=O)NC(=O)Cc1cc(C(F)F)no1 35989,N1(CC(=O)NC2CC(CNC(c3ccc(CC4CC4)cc3)=O)C2)CCCCC1=O 35990,C1(NC(C2CC(=C)C2)=O)(COC)CCCN(C(c2ccc(F)c(Cl)c2)=O)C1 35991,c1(CC)cc(C(N2CCC(CCNC(c3cn(C(F)F)cn3)=O)CC2)=O)nn1C 35992,C(=O)(C(C)CCC(C)(C)C)SC1CC(C(=O)OC)C1.c1(C2CN2)ncc(F)cn1 35993,CC(C(=O)N1CC2CC2(CNC(c2cccc(F)n2)=O)C1)S(=O)c1ccccc1 35994,c1(N(C)Cc2cccc(NC3CC(O)C3)c2)nccc(N2CCOCC2)n1 35995,N1(C(c2n(CC#C)ccc2)=O)CC(NC(c2cc(CC)cc(F)c2)=O)C2CC2C1 35996,c1(C(=O)NC(C2(CNC(=O)Cn3cnnc3)CC2)C)ccc(CN(C)C)o1 35997,N1(C(c2ccc(C(C)=O)cc2)=O)CCC(CO)C(NC(c2cc(C)[nH]n2)=O)C1 35998,S(=O)(=O)(c1cc(C(=O)N(C)CC2(OCC)CCC2)ccc1C(F)(F)F)NC 35999,Cc1ccc(C)c(C(=O)NC(C2CCCN2C(=O)Cc2cc(F)ccc2Cl)C)c1 36000,N1(C(C2C(c3n(C)cnc3)C2)=O)CC(C)(C)OCC1CNC(=O)CP(C)(C)=O 36001,C(=O)(C(F)C(C)(C)O)NC(CC(=O)NCCN1C(C)COCC1)(C)C 36002,N1(C(Cn2ncc(C)c2)=O)CC2CC1CN2c1cc(-n2ccnc2)ncn1 36003,c1(C(=O)NC(C(=O)NCc2onc(C)n2)(C)CO)c[nH]c(C)cc1=O 36004,N1(C(CC(C)P(C)(C)=O)=O)CCCOC2CCCC12 36005,Cc1nn(C)c(C(=O)NC(C2CN(C(=O)OC(C)(C)C)C2)C)c1C1OCCO1 36006,C(=O)(C(CCCC(=O)SC)OC)N(CCN(C)C(=O)OC(C)(C)C)CC 36007,C(=O)(CC(C(F)F)NC(=O)Cc1ncn(C)c1C)N1C(COCC#C)CCC1 36008,c1(CNC(C2CCN(Cc3cnc(N(C)C)o3)C2)=O)ccc(F)c2ccccc12 36009,C(=O)(C(O)C(C)(C)C)NCC1(O)CN(C(C2(CC=C)CCC2)=O)C1 36010,Cc1cc(C2(F)CCN(C(=O)NCc3ccnn3C3CC3)C2)cc(C)c1 36011,C=CCC(C)(C)CC(=O)NCC1CCCC(NC(c2cncc(C)c2)=O)C1 36012,N1(C(C2C(CC)C2)=O)CC2(CC(NC(=O)C=CCOC(C)(C)C)CO2)C1 36013,n1(CC(N2C(CNC(=O)CCc3cnccn3)CCC2)=O)c(C2CC2)nnc1S 36014,C(c1c(Cl)nc2sccn12)=CC(N1CC(NC(C2CC3C=CC2O3)=O)C(O)C1)=O 36015,c1(CNC(=O)NCC2C(C)CCN2C(=O)CC(C)(C)C)cccn2cnnc12 36016,Cc1nc(O)nc(C)c1C(N1CC2(CCN(C(=O)CC3CCSCC3)C2)C1)=O 36017,Cc1ccc(F)cc1C(N1CCC(CCC(=O)NCC2C(C)C2C)C1)=O 36018,CCCN=C(NCC1(C2CC2)CC1)NC1CCN(CC)C(C)C1 36019,CC1CCN(C(=O)CCn2cccc2)CC1NC(c1ccnc(OC(F)F)c1)=O 36020,Cc1cc(C(=O)NCC2(O)CCCN(C(=O)C=C(Cl)Cl)C2)c(C)n1C1CC1 36021,c1(-n2c(C(C)SC)nc(COC(F)F)n2)cccc2nc[nH]c12 36022,C12(NC(CCCC#C)=O)CCN(C(c3cc(C(F)(F)F)ncn3)=O)CC1C2 36023,c1(C(N2CC(NC(C3CN(C)C(=O)C3)=O)C(O)CC2)=O)nccn2nccc12 36024,c1(C(=O)NCC2CCCN(C(C3CC(C)C3)=O)CC2)cn(C)c(=O)nc1O 36025,C(CCCCC(=O)N1CCOCC(CNC(C2CC23CC3)=O)C1)OCC 36026,C1(C(N2CCC(CC(C)C(=O)O)CC2)=O)CCCC(F)(F)CC1 36027,C1(C(N(CCC(=O)OCC)CC(C)C)=O)CC2(CC2)CN1C 36028,C1(N(C(C)(C)C)C)CCCN(CCNC(=O)C(F)Cc2ccccc2)CC1 36029,C1(NC(C2CC2C2CCCN(C(C3CC34CC4)=O)C2)=O)CCCCC12OCCO2 36030,C1(NC(C2C(C)=CCS2)=O)CN(C(c2csc(C)n2)=O)CC1(C)C 36031,C12(CCNC(=O)COCc3ccccn3)CCC(C1)N(C(C1CC=CCO1)=O)C2 36032,N1(C(C(C)c2cccs2)=O)CCC2(CCN(C(c3cnn(C)n3)=O)CC2)C1 36033,c1(SCC#N)cccc(C(=O)NCC(O)CNC(=O)CCN2CCCC2)c1 36034,Cc1cc(C(N2CCC2C(=O)Nc2cnc(Br)c(C)c2)=O)ccc1O 36035,CCCCC(F)C(=O)N1CCC(C(=O)NCCSCC(=O)OC)C12CC2 36036,c1(C(=O)NC2CCCN(Cc3ccc[nH]3)CC2)cn2c(Cl)cccc2n1 36037,c1(OC)cnc(C(=O)NCCC2(C)CCN(C(=O)CC3(C)CCCO3)C2)nc1 36038,C1(NC(CCOC)=O)CC2CCC(C1)N2C(c1cnc(O)c2ccsc12)=O 36039,N1(C(C2=CCCC2(C)C)=O)CCC2CCN(C(c3ccc(CO)nc3)=O)CC12 36040,CC1C(C(N2CCSCC2)=O)CCN1Cc1cn(C)nc1C(F)F 36041,C=CC(C)(CC)C(=O)NCC1CC1CNC(c1nc(N(C)C)nc(=N)[nH]1)=O 36042,C(=O)(CCCc1cccnc1)NC(CN(C(c1cnccn1)=O)CC)C 36043,N1(CC(=O)NC23CC(CNC(Cc4c(C)n[nH]c4)=O)(C2)C3)C(=O)C(C)C(C)C1=O 36044,c1(C(=O)NC(C2CCN(c3cc(Cl)ncn3)C2)C)nc2cnccc2s1 36045,c1(CC)nn(C)cc1C(=O)NC1CCN(C(=O)Cc2cnc[nH]2)C1C(C)C 36046,C12(NC(c3c(C)ccs3)=O)CCCN(C(C3(CS(C)(=O)=O)COC3)=O)CC1C2 36047,C1(CC(=O)Nc2nc[nH]n2)OCCCC1(C)C.C1C(O)CCCC(C)=CC(=O)N1 36048,CCCCC(O)C(=O)NCC1(C)CCN(C(=O)CCCC(O)c2ccccc2)C1 36049,N1(C(CCOCCNC(Cc2c(C)scc2)=O)=O)CCOC2CCCC12 36050,C(=O)(CN=c1cc[nH]cc1)N1CCC(C(=O)Nc2c(OCC)cccn2)C1(C)C 36051,C1(C(=O)NCC(C(=O)NC)C)CC(C)(C)CN1C(=O)CC1CCCOC1 36052,N1(C(c2n(C)ncn2)=O)C2CCC1C(CNC(C1CCOC(C)(C)C1)=O)C2 36053,C(CCCCNCCc1cc(C(=O)OC)no1)SC 36054,c1(C(=O)NC(CCNC(c2c(CC)nn[nH]2)=O)C)cc(Cl)ccc1OC 36055,c1(C(N(C)CC2CCCC(NC(c3coc(O)n3)=O)C2)=O)nnc(O)cc1O 36056,N1(C(CCCc2ccc(OC)cc2)=O)CC2CC(C1)N(C(=O)CN(C)C1CC1)C2 36057,Cc1snnc1C(=O)NCCOC1CCN(C(c2cnn(-c3nccs3)c2)=O)C1 36058,C1(NC(CN(C)CC)=O)(CC)CN(C(=O)CC(C)c2ccccc2)C1 36059,CCC(C)(COC)C(=O)NC1CN(C(c2cccc(F)c2C)=O)CC1F 36060,CC1Oc2ccc(C(N3CCN(C(C4(C)CCCCCC4)=O)CC3)=O)cc2NC1=O 36061,N1(C(CC2C(C)(C)OCC2)=O)CCC2CN(C(c3ccnc4ccnn34)=O)CC12 36062,c1(C(=O)NCc2ncoc2CCNC(C2(CCF)CCC2)=O)ccnc(S)c1 36063,c1(OC)ccc(Cl)c(C(=O)NC(C)CCNC(C2CC(C3CCC3)C2)=O)c1 36064,c1(C(=O)NC2(CO)CCN(C(C34CC(C)C3C4)=O)C2)cc2ccc(Cl)cc2o1 36065,c1(C(C(=O)NCC2N(C(c3cnoc3)=O)CCC2)F)ccc(F)cc1 36066,c1(N2CCC(CCC)C2)ccc(S(=O)(=O)N2CCCN(C)CC2CC)cc1Cl 36067,N1(C(CSCC)=O)CCC(NC(c2ccc3c(c2)CCO3)=O)C(F)(F)CC1 36068,n1(CC)ncc(C(=O)NCC(C)NC(c2c[nH]c(=N)s2)=O)n1.n12cc(nn1)C2 36069,CCC(C)CC(C(=O)NC(CO)C(N)=O)NC(=O)CCc1nncs1 36070,c1(C(N2CC(C)N(C(c3csc(Cl)n3)=O)CC2)=O)cc2ccsc2c(=O)[nH]1 36071,c1(C(=O)NCC(C(C)C(C)C)NC(C#CC(C)C)=O)nn(C)cc1[N+](=O)[O-] 36072,N1(C(=O)Cn2ncnn2)CCCC1C1(C(=O)NCCn2cncn2)CC1 36073,c1(C(C(=O)OCC(N2CCN(CC)C(=O)C2)=O)N(C)C)ccc2n[nH]cc2c1 36074,C1(NC(C(CC)NC(C)=O)=O)CN(C(=O)C(C)(C)OC)CC2CC12 36075,c1(C(=O)NCCN(C(=O)C(C)C(C)O)C(C)C)cc[nH]c2nccc1-2 36076,C(=O)(CC(C)C(F)F)NCCC(CC)(C)NC(c1cccc(CO)n1)=O 36077,CC1C2CCC(C2)C1C(N1CC2(C)CC1(C(=O)N(C)C1CC1)C2)=O 36078,Cc1ccc(F)c(C(N2CCC(NC(c3ncsc3S(N)(=O)=O)=O)CC2)=O)c1F 36079,C1(CN=C(NCC(=O)NC(C)C)NCC(Cl)C(F)(F)F)CC(O)C12CCC2 36080,CC(CC(=O)NC1CCN(CC(=O)NC(=O)Nc2cccs2)C1)C1CCCC1 36081,C=C(Cl)CCC(=O)N1CCC(C(C)(O)CNC(c2ccn(CCOC)n2)=O)CC1 36082,C(=O)(C(CC)CC(F)(F)F)N1C(CCCNC(C(C#C)(C)C)=O)CCC1 36083,O(C1CCCc2ccccc21)CC(=O)N(CCCNC(C1(O)CC1)=O)C 36084,Fc1cc(Nc2nccc(NCCCNC3CCCC3)n2)cc(C(F)(F)F)c1 36085,c1(C(=O)NCC(C(C)C)=O)ccc(F)cc1I 36086,C1(C(=O)NC2(CC=C)CC=CC2)CN(C(c2c(O)cccc2F)=O)CC(C)O1 36087,N1(C(C2CCC(CCC)CC2)=O)CCCC2CN(C(=O)Cc3ccsn3)CCC12 36088,c1(C(Cc2cn(C3CCN(C(=O)CCOc4cccs4)C3)nn2)O)ccccc1 36089,C1(NC(c2cc(OC)ncc2)=O)CC2CN(C(C3CCOC3)=O)CC2C1 36090,C1(C)(NC(COC2(C)CCC2)=O)CCCN(C(C2COC3(CO)CC2C3)=O)C1 36091,c1(C(=O)NCC2(CO)CC(CNC(C3CN(C(C)=O)C3)=O)C2)cc(C(=O)O)n[nH]1 36092,CC(C)=C=CC(=O)NCC1(NC(=O)C(c2ccccc2)F)CCOCC1 36093,C12(C(=O)NCC3C(NC(c4n(CCCC)ncc4)=O)C3)CCC(OCC)(CC1)C2 36094,N1(C(C(COCC)C)=O)CC2CCC1C(CNC(c1cncc(NC)c1)=O)C2 36095,N1(CC(=O)NC(c2ccc(-c3ccc(Cl)cc3Cl)nc2)C)CCc2[nH]nc(O)c2C1 36096,c1(C(=O)NC(CN(C(c2ccn(C3CCC3)n2)=O)CC)C)nc(C)sc1C 36097,C1(CC(=O)NC(CC)CN(C)C(c2cnc(C3CC3)o2)=O)C=NN(C)C1=O 36098,c1(C(=O)NCCN(C(C(CCC)O)=O)C(C)C)cccc(S(=O)(=O)CC)c1 36099,C12(NC(c3n(C)cnc3S(N)(=O)=O)=O)CN(C(C3CCC3)=O)CC1CS(=O)(=O)C2 36100,Cc1cc(C)c(C(=O)NCC2(O)CC(NC(=O)Cn3ccnc3)C2)o1 36101,C1(CNC(CCCOCC=C)=O)CN(C(c2cn(CC=C)nn2)=O)C(C)(C)C1 36102,c1(C(N(CCCN(C(=O)CSC2CCCC2)C)C)=O)cc(F)cc(Cl)c1 36103,CCC(C(=O)NCC1CCCC1C(=O)NC1CCOCC1O)C(F)(F)F 36104,C1(CN(C(c2nc(OCC)oc2)=O)C)CN(C(c2csc(O)n2)=O)CCO1 36105,N1(CCNC(CCCOC)=O)CCN(C(=O)CCCn2ccnn2)CC1 36106,C(C1CCN(C(=O)CCCN=[N+]=[N-])CC1)=CC(=O)NCc1nc(C(C)C)on1 36107,N1(C(c2c(C)nco2)=O)CCCC(C)(C(=O)Nc2cn(C)nc2C(F)(F)F)C1 36108,C1(C(=O)NCC(C)(C)OCCNC(C2CC2Cl)=O)Cc2ccccc2C1 36109,C1(C(N2CCC3(C(NC(c4ccoc4Cl)=O)C3)C2)=O)COC2COCC2O1 36110,Cn1ncc2c1CN(C(c1ccc(Cn3cc(CC(N)=O)nn3)o1)=O)C2C(=O)O 36111,c1(C(=O)NC2C(NC(C(C(C)C)N(CC)CC)=O)CC2)c(F)cccc1Cl 36112,n1(CCC(=O)N(CCCN(C)C(C2CSC2)=O)C)sc2ccccc2c1=O 36113,CN1CC2(CCN(C(C3(C)CC4(CC4)C3)=O)C2)CC1=O 36114,N12CCC3(CC(C3)C(=O)NC3(CC3)C1=O)C2.C1(CCCO)(COC(C)C)CC1 36115,C1(CNC(C(=O)NCC)=O)C2CCC(C2)N1C(=O)C(C)(C)C1CCCCC1 36116,C1(NC(c2cnn(C3CC3)c2)=O)CC2CN(C(=O)C3=COCCO3)CC2C1 36117,N1(C(c2c(N)cn(C)n2)=O)CC(NC(c2cc(Cl)n(C)n2)=O)CC2(CC2)C1 36118,N1(Cc2ncc(C)s2)CCC(C(C)NC(c2ccncn2)=O)CC1 36119,C1(C(=O)NCCCCCNC(c2cc([N+](=O)[O-])c[nH]2)=O)C2CS(=O)(=O)CC12 36120,N1(C(C2C(C)CC2)=O)CC2CCC(C1)N2C(=O)C(c1cccc(Br)n1)(F)F 36121,c1(C(=O)NC(CC(C)NC(=O)C(C)NC(c2ccco2)=O)C)cc(C#N)cs1 36122,c1(SC)ccc([N+](=O)[O-])c(C(=O)NC2CC(CCNC(=O)CC(C)C(C)C)C2)c1 36123,C(=O)(CCC(=O)N1CCCCC1C(C)NC(C1CN(CC(C)C)C1)=O)NCCC 36124,C1(C(=O)NCCC)CCN(Cc2cccc(I)c2)CC1F 36125,C1(CC)CCCCN1Cc1nn[nH]n1.c12ccn(n1)CCN2 36126,C1(NC(CSC(C)C)=O)CC2(CCN(C(c3csc(C4CC4)c3)=O)CC2)C1 36127,CN1C2CCC1CC(C(N1CC(N(C(=O)Cc3ccsc3Cl)C)C3(CC3)C1)=O)C2 36128,Cc1cc(CC(=O)NCC2C=CC(NC(c3nccn3C)=O)C2)n(C)n1 36129,C1(C(=O)NCc2ccc(C)c(C)c2)N(C(=O)CC=C(Cl)Cl)CC12CCCC2 36130,Cn1nc(CO)c2c1CN(C(c1ncc(I)cn1)=O)CC2 36131,C1(NC(C2CCCO2)=O)CN(C(=O)CCCCC(F)F)C2(CCC2)C1 36132,c1(C(CC)C)ccc(C(=O)NC2CC(F)(CNC(C3(C)CCC(=O)N3)=O)C2)cc1 36133,c1(OC)cc(CC(N2CCC(C)(NC(c3cc(C(C)C)on3)=O)C2)=O)cc(Cl)c1 36134,N1(C(CCCCOC)=O)CC2(CCCCN2C(C2(C)CC3CCC2O3)=O)C1 36135,N(C1CCCn2cnnc21)C(=O)Nc1ccc(C2CCC2)nc1 36136,Cc1ccc(CC(=O)NCCC2CC(NC(=O)Cn3cnnc3)C2)cc1Cl 36137,Cc1ccc(S(=O)(=O)N2CC(C)NC(C)C2)cc1NC(=O)C(N)C1(C(C)C)CC1 36138,c1(CC(=O)NC(C2CN(C(C3CC4(C3)CC4F)=O)C2)C)nn(C)c2ccccc12 36139,C1(C(N(C)Cc2ccon2)=O)CCN(C(=O)CCc2csnn2)C1 36140,C(=O)(CC(=O)N(CCC(=O)NC1(C)CC1C)OC)OC 36141,C(=O)(CC(c1ccccc1)C1CC1)NCCCCNC(C(=O)NCC(F)(F)F)=O 36142,c1(CC(=O)NC2CCN(C(=O)Cc3cc[nH]n3)C23CC3)ccc([N+](=O)[O-])cc1 36143,C(=O)(CCS(=O)(=O)c1ccccc1)NC(CC)CN(C(=O)C(C)CC1CC1)CC 36144,CCCC(CC)CC(=O)NC1CN(C(=O)CNc2cccc(C#N)c2)CC1O 36145,C1(F)(CNC(=O)NC(C2(CCc3ccon3)CC2)C)CC1C 36146,C(=O)(CCCN(C)N=O)NCCC1CC(OC)CN1C(=O)C(C)NC(C)=O 36147,C(=O)(CCCCN=[N+]=[N-])NCC(CN(C(C1(C2(C)CC2)CC1)=O)CC)(C)C 36148,N1(C(CN(C)C(C2(C)CCCS2)=O)=O)CCN(C(c2nccn2C)=O)CC1 36149,N1(C(CC2N(C(C=C(CCC)C)=O)CCOC2)=O)CC(C2CC2)(COC)C1 36150,N1(C(c2ccc(C)c(F)c2)=O)CCCCCC(NC(C2(C)CC2(F)F)=O)C1 36151,C#CCCC(C(=O)NC1CC12CCC2)NC(c1cc(C)no1)=O 36152,N1(C(CC2CCC(NC(c3occ(C)c3)=O)C2)=O)Cc2cccc(C)c2C1 36153,Nc1ncc(C(=O)NC2CC(NC(c3ccccn3)=O)C2)cc1-c1ccccc1 36154,c1(C(N2C(CN(C)C(c3scc(Cl)c3Cl)=O)CCC2)=O)cccc(=O)n1C 36155,CCCC(C(=O)NC1(CO)CCOCC1)c1ccc(Cl)cc1.C12CCC1NC2=O 36156,N1(C(CCC(=O)NC)=O)CCN(C(c2coc(C(C)=O)c2)=O)C(C)C1 36157,C1(C(N2CC(C3(NC(C(C)SC)=O)CC3)C2)=O)CCc2n[nH]cc2C1 36158,Cc1cc(C(N2CC(C)(NC(=O)CC3CCCOCC3)C2)=O)cc(N)c1 36159,C(=O)(C1CCCn2c(C)cnc21)NCCC1CCCN(C(CCC#CC)=O)CC1 36160,N1(C(C)C)CC(NC(=O)CCCN(C(=O)CC2CSCCO2)C)C(C)C1 36161,c1(N(CCOC)C)cccc(CN2CCCC2C2CCCC2=O)c1 36162,C1(CC(=O)NCC(N2CCCCC2)=O)CCN(C(C2CC(F)C(=O)N2)=O)CC1 36163,CC1CC=C(C(=O)N2CCCC(CCC(=O)NC3(C)CCCCC3)C2)CC1 36164,c1(NC(C)=O)ccc(C(N2CC(CNC(c3c[nH]cc3C)=O)C2)=O)c(C)c1 36165,N1(C(C2CC(=O)C2)=O)CC2(CCCC2)C1C(N1Cc2ccncc2C1)=O 36166,C1(C(C(=O)N(C(C#C)C2CCC2)C)C)CCN(C(c2cc(COC)sn2)=O)C1 36167,C=CCC(F)(F)CN(C(=O)C(C1CCN(C(=O)C(C)C2CC2)CC1)C)C 36168,c1(C(=O)NCCOCCN(C(C2(CC#C)CC2)=O)C)cc2c(cc1Cl)CCCC2 36169,c1(C(=O)NC2CCC(CCNC(c3c(OC)csc3)=O)C2)cn(C)c(=O)cc1C 36170,Cc1ccc2c(c1)CCC2C(=O)NCC1CCCC1NC(=O)CCC1(C)CC1 36171,C1(CN(C(c2ccc(OC)s2)=O)C)CN(C(c2nccnc2Cl)=O)CCO1 36172,N1(CC)CC(C)OC2(CCN(Cc3c(C)nc(-c4ccccc4)n3C)CC2)C1 36173,c1(CC)nc(C)c(C(=O)N(C)CCOCCN(C)C(c2nc(C3CC3)cs2)=O)s1 36174,C12(CNC(=O)CC3CC(F)C3)CCC(NC(C3CC4CCC4C3)=O)(CC1)CO2 36175,c1(C(=O)Nc2cccc(Br)c2)cnc2n1CCN(C(=O)Nc1occc1Br)C2 36176,C1(CNC(c2ccnc(CO)c2)=O)CC2CC2N1C(=O)COCC1CCOCC1 36177,C1(NC(C=Cc2cc(OC)ns2)=O)CCCN(C(c2cccc(F)c2F)=O)C1C 36178,c1(C(C)NC(C2CN(C)C2)=O)ccc(CNC(c2ccc(C#N)[nH]2)=O)cc1 36179,N1(C(c2cc(OC)cc(Cl)c2)=O)CCC2(CCCN(CCn3cccn3)C2)C1 36180,N1(C(c2cccc(C#C)c2)=O)CC(C2CN(C(=O)C(C)(C)CCCO)C2)C1 36181,c1(C(=O)NCC2CCCCC2NC(C2CCCCS2)=O)cnn2c1C(=O)NCC2 36182,C1(C(N2CCC(NC(c3ccc(C(=O)OC)s3)=O)C2)=O)CC(C)(C)CN1C 36183,C(=O)(CCCCC#N)N(CCC(C)NC(=O)CC1CCC(F)(F)C1)C 36184,C1(CNC(C(C#C)(C)C)=O)CCCC2(CCN(C(c3nc(C)oc3C)=O)CC2)O1 36185,c1(CN(C(C(=O)OCC)C)C(C2CCCCC2)=O)cc(F)ccc1O 36186,N1(C(C(C)OCC#C)=O)CC(NC(=O)CCn2cc(C)cn2)C(C)C1 36187,n1(CC#C)cccc1C(=O)NC(C)CNC(c1cc(C2CCC2)no1)=O 36188,c1(CC(=O)NCCC(C)NC(CC(CC)OC)=O)cccc(F)c1F 36189,c1(OC)ccc(F)c(C(=O)NCC2CC3(CC3)CN2C(=O)CC2CNC(=O)C2)c1 36190,C1(NC(C(CC)CC(C)C)=O)CCCC12CCN(C(=O)CC1CC(F)(F)C1)CC2 36191,N1(C(c2c(C)[nH]cc2)=O)CCC(CO)C(NC(=O)Cc2cn(C)cn2)C1 36192,C1(=O)C(O)CCN1.n1(CC(=O)N(C2CCN(C(C)=O)C2)CCC)nnc(=O)[nH]1 36193,C=CC1CN(C(=O)CC(C)F)CC1NC(c1cc(COC)cs1)=O 36194,C1(NC(C(c2ccc(O)cc2)C)=O)CN(C(=O)C(C)(C)OC(C)C)CC(C)(C)C1 36195,C=C(Cl)C(C)(C)C(=O)NCC(CC)NC(c1cccc(N2CCC2=O)c1)=O 36196,N1(C(c2c(CC)c[nH]n2)=O)CC2CCN(C(=O)CC3OCCCC3(C)C)CC12 36197,N1(C(C(C)(C2CC2)OC)=O)CCN(C(C23CC2COC3(C)C)=O)CC(O)C1 36198,N1(C(C(c2ccccc2)C)=O)CC(NC(c2c[nH]c(=O)cn2)=O)C(C)C1 36199,N1(C(C2(CC)CCCC2O)=O)CCC12CN(C(=O)CCCc1ccccc1)C2 36200,CCCCCC(C)(C)C(=O)NCCC(C)NC(=O)C(n1cc([N+](=O)[O-])cn1)(C)C 36201,C(CCCCCCCO)=CC1C(C)(C)N(C(=O)CCCCCC#N)CC1.c1(N)nn[nH]n1 36202,C#CCC(CC(=O)NC1CC2(NCc3cn(C)nn3)COC1C2)c1ccccc1 36203,C(=O)(CC(C)C(C)C)NC1(CCN(C)C(C2(OC)CCCC2)=O)CCC1 36204,c1(C(N2CC=CC(NC(C=CCN(C)CC)=O)C2)=O)cc[nH]c2nccc1-2 36205,C(c1cccc(C)c1)=[SH]CC(=O)C(C)=O.c1(N)ccccc1Cl.C12CN(CC1F)C2=O 36206,C1(C(=O)NC2CCCC(NC(c3c(OCC)nccc3)=O)C2)CC2(C1)CC2(F)F 36207,C1(C(=O)NC2(COC)CC2)CC12CC(NC(=O)CCC1CCOC1)C2 36208,c1(OCC)ccccc1OCCCN1CC2C(C(=O)NCCCO)C2C1 36209,C1(C(=O)NC)C(C2CC2)CCN1C(=O)C(=Cc1c[nH]cn1)F.C1(OCC=O)CCCC1 36210,C(CC(CC)C(=O)NC(c1cnn(C)c1)C(=O)NC(COCC)C(C)C)=CC 36211,Cc1ccc(C(CNC(C2(n3ccnn3)CC2)=O)NC(=O)CSC(F)F)cc1 36212,O(NC(=O)C(O)CNC(=O)C(O)C(F)(F)F)C(C=C)C 36213,n12nnc(n1)C2.c1(CNC(=O)NC2(c3cccs3)CC2)cnnn1-c1ccccc1 36214,c1(C(=O)NC2CC3(CC(NC(C4C(C(=O)OC)C4)=O)C3)C2)ccnc2[nH]cnc12 36215,N1(C(C2(C(=O)OC)C(=C)CC2)=O)CCCCC(NC(c2nn(C)cc2Cl)=O)C1 36216,C(=O)(C1CCCc2ncc(C)n21)N1CCC(NC(CCc2nnc(CC)o2)=O)C1 36217,c1(OC)ccc(C(=O)C(=O)NC2CCC(NC(=O)C=C(C)C)C2)cc1OC 36218,CC1CC(F)(F)CN1C(=O)C=CC(C)(C)NC(=O)C=CC1CCC1 36219,CCCC(C(=O)OC)C(=O)N1CCC(C)(C(=O)NC(c2cncnc2)C)C1 36220,C=CC1(C(=O)NCC2(C)CCCCC2)CCN(C(=O)C=C2CCC2)C1 36221,c1(C(=O)NCC2(F)CC(NC(CC(CN(C)C)O)=O)C2)ncnc2sccc12 36222,C=C=CC(C)C(=O)NC1(C)CC(NC(=O)CCc2nc(-c3ccoc3)no2)C1 36223,C(=O)(C(C)(C)CC#N)NC1C(NC(c2c(SC)cn(C)n2)=O)COCC1 36224,N1(C(C(C)NC=O)=O)CCCC(CN(C)Cc2nn(C)cc2Cl)C1 36225,c1(C(=O)NCC2C(CNC(CNS(CC)(=O)=O)=O)C2)cc2oc(C)c(C)c2[nH]1 36226,c1(OCC)ccccc1C(=O)NC(c1cnc[nH]1)C 36227,C1(C(=O)NCC2OCCN(C(C3N(C(C)=O)CCC3)=O)C2)CCCC(=O)N1C 36228,c1(CNC(CCOCCNC(C2(C(=O)OC)CC2)=O)=O)nnc(CO)s1 36229,C1(C(=O)NC2CCC(NC(c3ccccc3F)=O)CC2)(COC)CCOCC1 36230,C=CC(CCC)CC(=O)NCC1CC(F)CN1C(c1cc(F)c(N)c(F)c1)=O 36231,N1(C(C2CCN(C)C2=O)=O)CC2CN(C(c3cnc4ccsc4c3)=O)CC2(C)C1 36232,C1(CC(N2CC(C(C(=O)NCCNC(=O)NC)C)C2)=O)CCCCC1O 36233,N1(C(CC(C)NC(=O)C=C(Cl)Cl)=O)CCCCC1C1(NC(=O)CC(C)(C)C)CC1 36234,C1(C(=O)NCC2(NC(c3ccc(C)o3)=O)CC(OC)C2)CC12CCCCC2 36235,c1(-n2ncc(CS(=O)(=O)NCCC(=O)OC(C)(C)C)c2)ccc(Br)cc1 36236,CCC(CNC(C1(NC(=O)CCn2cncn2)CC1C)=O)CCO 36237,Cc1ccc(C(=O)NCC2(F)CCN(C(=O)CCCC3CC3C)CC2)c(O)n1 36238,N1(C(C(C)OC)=O)CC(NC(C2CCC(C(F)(F)F)O2)=O)C(C(F)F)C1 36239,C(=O)(C(COC)CC(C)C)NC1(CC=C)CN(C(=O)C(C)=CC(C)(C)C)C1 36240,C12(C(=O)NCC3(C)OCCN(C(Cc4nnc(C)o4)=O)C3)CCCCC1C2(F)F 36241,Cc1ncnc(C(=O)N(C(CC(C)C)C(=O)NCC(c2ccnn2C)O)C)c1C 36242,C1(CNC(C(c2ccccc2Cl)OC)=O)CCCN(c2nc(CCOC)ns2)C1 36243,c1(CNc2c(C(=O)Nc3c(C)cnc(O)c3)cc(Cl)nc2)c(Br)ccc(Cl)c1F 36244,C(=O)(C1CCCc2sccc21)NC1(C)CCN(C(C2CCC(OC)CC2)=O)CC1 36245,c1(C(N2CC(CNC(c3[nH]nnc3C3CC3)=O)C2)=O)cc2c(F)cc(F)cc2[nH]1 36246,c1(C(=O)NC2CC(CNC(C(CC)n3cncn3)=O)C2)cc(C)nc(O)n1 36247,C1(CC(=O)NCC(C2CCN(C(=O)C=Cc3cc[nH]n3)CC2)C)CCCCN1C 36248,C(=O)(C1COc2ccccc21)NCCN(C(CSCCC)=O)CCOC 36249,CC1CCC(CC(=O)NC2CCC(NC(c3cnn(CCC(F)(F)F)c3)=O)C2)O1 36250,c1(C(N(CC(C)NC(=O)C(C(=O)OC)OC)CC)=O)cc2nc(=O)ccn2[nH]1 36251,N1(C(c2sc(C)cc2C)C(=O)NCC)CCN(C)c2ccc(C)cc21 36252,CC1(C(=O)NCCCCCNC(c2cc(CC3CCC3)c[nH]2)=O)CCC(=O)NC1 36253,C1(C(N2CC(NC(C(C)(C)C3CC3)=O)C(O)C2)=O)CCn2ccnc2C1 36254,c1(CC(N2CC(C)C(CNC(=O)CCC(=O)NN(C)C)C2)=O)ccc(C#N)cc1 36255,c1(C(=O)Nc2c(C(=O)OC)scc2)ccccc1N1CCNC1=O 36256,C=C=CC(C)C(=O)NC(CNC(c1cc(C)n(CC(F)(F)F)n1)=O)CC=C 36257,n1(CC(=O)NC2CCCCN(C(=O)CC3(O)CCOC3)C2)ccc(O)nc1=O 36258,C1(NC(c2cncc(OC)n2)=O)CN(C(c2cc(C)c(C)o2)=O)C(C)(C)C1 36259,C(=O)(C#CC(C)(C)C)NC(C(C)C)CNC(=O)CN1CCNC(=O)C1 36260,CC1(CNC(=O)CC2CCSCC2)CCCN(C(C2CC3(C2)CC32CC2)=O)C1 36261,c1(N2CC(C)CN(C)CC2)ccc(S(=O)(=O)NCc2ccc(=N)[nH]c2)cn1 36262,N1(C(CCOCC#C)=O)CC2OC(C1)C2.C(=O)(C(C)OC)NCC1CC1 36263,Cc1cc2cc(F)ccc2n1Cc1ncc(F)cc1C 36264,CC(C)CC(O)CC(=O)N1CC(C)C(C)(CNC(C2(C(C)C)CC2)=O)C1 36265,Cc1ccc(C(=O)NC2CCC(C)N(C(c3ccnc(F)c3F)=O)C2)cc1N 36266,c1(C(N(CCn2cc(-c3ccc(C)s3)nn2)C)=O)ccc(-c2cccs2)cn1 36267,C1(C(C(C)C)NC2(CCOC(C)C)CC2)(CO)CCCCC1 36268,N12CC3C(C3C1)CC2=O.c1(C(c2ccncc2)CNC(C)=O)ccc(Cl)cc1 36269,c1(CN(C2CC(=C)C2)C)c(C)nn(C2CCCCO2)c1C 36270,CC1CCCN(C(=O)CC(C)(C)C)C1CNC(=O)C=Cc1ccn(C)c1 36271,C1(CNC(N(OC)Cc2ccccc2)=O)CCC2(CC1)NC(=O)OC2 36272,Cc1cc(C(=O)NCC(CO)NC(=O)CCc2cccs2)n(C)n1 36273,c1(OC)cc(CC(N2CCC(NC(C3CCCOCC3)=O)C2(C)C)=O)ccc1C 36274,C1(CNC(CCC(=C)Cl)=O)CN(C(c2c(N)cc(Cl)cc2F)=O)CC2(CCC2)O1 36275,CCC1=C(C(=O)NCCN(C2CCCC2)C(C2CCCC(F)C2)=O)SCCO1 36276,Cc1cc(O)ncc1NC(C1CCC(C2CC2)N1C(c1nnn(C)c1N)=O)=O 36277,CC(C)C(N=[N+]=[N-])C(=O)N1CCC(C)C1C(=O)NCCOC1CC1(F)F 36278,C1(NC(CSc2cccc(OC)c2)=O)CC(F)(F)C12CCC2 36279,N1(c2nccc(=NCc3c(C)occ3)[nH]2)CCN(C)CC2(C)CCCC12 36280,C1(CCN(C(C(C2CC2)OC)=O)C)CCCC2CC12.c1c(=O)n1 36281,N1(C(C2CCCC2)C)CC2CCC1C2CC(=O)NNC(=S)N 36282,Cc1cc(C(N2CC(NC(c3cc(C4CCCC4)[nH]n3)=O)C3CC23)=O)c(C)cn1 36283,c1(NCCCOc2c(C)cccc2)cc2[nH]nnc2cc1F 36284,C(=O)(C(CNC(c1oncc1CC)=O)CC(C)C)NC1(CC#C)CCC1 36285,C1(CCCNC(C2CCC3CC23)=O)CCN(C(=O)Cc2ccccc2F)CC1 36286,CC1CN(C(c2cc(C(C)(C)C)on2)=O)CC(C)C1NC(c1n[nH]c(C2CC2)n1)=O 36287,N1(C(C2CCOC2)=O)CCCC(Cn2cc(C3CC=CCC3)nn2)C1 36288,C=CCC(CC)C(=O)N1CC2CCC2(CNC(=O)CNC(=O)CC(C)(C)C)C1 36289,C1(NC(CCCC=C)=O)CC2CC1N(C(=O)CCc1ccsc1Cl)C2 36290,N1(C(C(C(C)(C)C)n2cc(CC3CCCNC3)nn2)=O)C2CCC1CC(F)C2 36291,c1(NC2C(C)(C)OCC2)c(-c2ccc(Cl)cc2)nc2ncccn12 36292,c1(-n2c(CC(F)(F)C(F)(F)F)nc(CCN(C)C)n2)ccnc2ccccc12 36293,c1(C(N2CCN(C(c3c(C)n(C)nc3)=O)C(C)CC2)=O)cccn2c(O)nnc12 36294,CCC(C)(C)C(C)CC(=O)NC1CCC1CNC(=O)Cn1cnc(C#N)n1 36295,CCC(CCC(=O)N1CCC(C(C)(F)F)CC1)OC 36296,C(C(O)CC(=O)NCCCCCF)NC(CCC1C(C)(C)C1)=O 36297,C1(C(NOCC(=O)OCC)=O)CC(NC(=O)CC2CCCN2C)C1(C)C 36298,C1(OCCO)COC(C)(C)CN1c1nc(C)cc(NCc2c(OC)cccc2)n1 36299,C(=O)(C(F)CC(C)(C)NC(=O)CCCCCF)N1CCCC(C(C)C)CC1 36300,c1(C(=O)NCC2N(C(C3C(C)=C3)=O)CCC2C)cnc(F)cc1C 36301,C1(NC(COCC2N(C)CCC2)=O)COCCN(C(=O)CO)C1 36302,c1(OC)ccc2[nH]cc(C(=O)NC(C)CC(C)NC(=O)CSC3CC3)c2c1 36303,N1(C(C(C)OCC(C)C)=O)CCC2(CCC2)C(NC(=O)CSC2CC2)C1 36304,C#CC1CN(C(=O)Cc2ccc(Cl)s2)CCN1C(c1cc(C(C)(C)C)[nH]c1C)=O 36305,C#CC1(C(=O)NCC2(CCNC(c3ccc(F)o3)=O)CC2)CCCC1 36306,C(CCCC(C)(C)C)c1nnc(CC(C)(C)NC=O)o1 36307,c1(CNC(CC2N(C(CC(C)c3ccco3)=O)CC2)=O)ccc(O)cc1 36308,C1(NC(CCOC)=O)CC=C(C(=O)NCC2CC3C=CC2O3)C1 36309,N1(C(Cn2c(C)nc(C)n2)=O)CCC2(CC1)CCN(C(C1(CC3CC3)CC1)=O)CC2 36310,N1(C(C(=O)NCC=C)C(C2CC2)OCC)CCC2(CC1)NC(=O)NC2=O 36311,c1(C(=O)NC(CCNC(c2c(CC)ncnc2)=O)C)ccc(C(C)(F)F)nc1C 36312,CN1CCN(C(c2cc(CNC(=O)CCc3ccsc3)[nH]n2)=O)CC1CO 36313,Cc1nc(N)c2c(C)c(C(=O)NCc3ccc(CC4CC4)cc3)sc2n1 36314,N1(C(COCCCC)=O)CCc2sc(CNC(c3nc(C)c(C)s3)=O)nc2C1 36315,c1(CC)ncc(C(=O)NC2COCC2NC(=O)CCC2CC2(F)F)c(C)n1 36316,C12C(C3CC3)CCN1C2=O.c1(CNC(C2CN(C(N)=O)C2)=O)csc(C(C)=O)c1 36317,C(C)(C)(C(=O)NCC(C1CC1)NC(=O)C(c1nc(C)cs1)C)SC 36318,C(C(=O)Nn1cccn1)N(C(C)CC(N)=O)CC 36319,N1(Cc2cc(C)c(Br)cc2C)CCC(N=c2[nH]cnc3cnn(C)c23)C1 36320,c1(C(=O)NC2CCN(C(C3CCNC(=O)C3)=O)CC2)ccnc2ncccc12 36321,C1(CC)CN(C(=O)C(C2CCC2)NC(c2ccnnc2C)=O)CCO1 36322,N1(C(Cc2cc(C)no2)=O)CCC2CCN(C(C3CC3C(C)(C)C)=O)C2C1 36323,c1(NC2(CNC(C3CC(CC)OCC3)=O)CCC2)ncc(S(C)(=O)=O)cc1Cl 36324,C#CCN(OC)C(=O)CC1CC(NC(=O)CSc2ccncc2Cl)C1 36325,CCC(O)C(C)(C)C(=O)NCC1CCN(C(=O)CSCCC(C)C)C1 36326,Cc1c(C(=O)NC2CCC2CNC(C2COC(=O)N2)=O)[nH]c2c(C)cccc12 36327,C1(C(=O)OCc2c(OC)nn(C)c2)CN(C(C2CC3CCC3C2)=O)C(C)(C)C1 36328,CC1(C)C(NC(C2COC(=O)C2)=O)CCN1C(=O)COC1CCCC1 36329,c1(CNC(C(CCC)CC)=O)ccc2c(c1)CN(C(C1CCN1S(C)(=O)=O)=O)C2 36330,C#Cc1ccc(NC(c2cnn3c2CCCC3)c2nnnn2CC=C)c(C)c1 36331,C1(C(N2CC(C(CN(C)C(C34CC(CO)(C3)C4)=O)(C)C)C2)=O)CCCC(F)C1 36332,N1(C(C(=O)N(C)C)=O)CC2CCCCC2(CNC(C2(C)CC(C)(C)C2)=O)C1 36333,c1(NC(C(CC)(C)OC)c2nnnn2CCCF)ccc(C)c(S(C)(=O)=O)c1 36334,O=C1CCC(C(=O)NC2CC(C3CCN(CCN4CCCCCC4)C3)CC2O)=NN1 36335,C(=O)(C(C)(C)CCCSC)NC1CN(C(c2cccc(OC)c2F)=O)CC(C)C1 36336,C#Cc1ccc(C(N2CC(C)CC2C(=O)Nc2cnn(C)c2)=O)cc1C 36337,Cc1nc[nH]c2nc(NCC3(NC(c4cnc5n4CCC5)=O)CCCC3)cc1-2 36338,C(C)(N=c1[nH]c(=NCC(CO)C2CCCC2)c2c(ncn2C)[nH]1)c1ncc(C)s1 36339,C1(C(=O)NC(CN(CCC(C)C)C2CC2)=O)CCN(S(=O)(=O)N(C)C)C1 36340,C(=O)(C1=CC2C=CC1C2)NC1CCN(C(C(C)OC(C)(C)C)=O)C1C1CC1 36341,C1(CNC(c2c(OC)n(C)nc2)=O)C(C2CC2)CCN1C(c1nnn(C)n1)=O 36342,C1(C(N2CCC(CN(C(=O)COCC3CC3)C)C2)=O)CCc2n[nH]cc2C1 36343,n1(CC)ccnc1C=CCNC(C1CC(CNC(C2CCSC2)=O)C1)=O 36344,C(CCCCNC(c1ccn(C2CCOCC2)n1)=O)N(C(C)C)C(c1cnns1)=O 36345,Cn1cc(C(=O)NC2CCCN(C(=O)CCC3CC3(Cl)Cl)C2)c(O)n1 36346,NS(=O)(=O)c1ccc(C(N2CCC(CNC(c3nsnc3O)=O)C2)=O)cc1F 36347,N1(C(C(CC)C)=O)CC(CNC(c2sccc2C)=O)OC(C)(C)C1 36348,Cc1cc(N2CCCC(C)(NC(=O)CCC(F)(F)F)C2)ccc1[N+](=O)[O-] 36349,C(=O)(C(O)CCC(C)C)N1CC(C)(NC(C2CCCC(OC)C2)=O)C1 36350,N1(C(C(C)N(C)CC)=O)CCOC(C(N2CCCC(C)(C)C2)=O)CC1 36351,c1(NC(C)=O)cnc(C)c(C(N2CCCC2CNC(C2OCC2(C)C)=O)=O)c1 36352,C(N=c1[nH]c(=NC2CCCN(C)C2)c2cc(Cl)ccc2[nH]1)C1CC(=C)C1 36353,c1(C(=O)OC)cc(F)c(C(N2CCS(=O)CC2c2cnn(C)c2)=O)cc1F 36354,Cc1sccc1C(=O)NC(C1CCCN1C(=O)CSS(C)(=O)=O)C 36355,CC1CN(C(c2ccc3sccc3c2)=O)CC(C)CN1C(c1cscn1)=O 36356,N1(C(C(C)OCC)=O)CC(NC(=O)CCc2cnc(O)[nH]2)C2(CCOCC2)C1 36357,c1(OCC(=O)NC2CC(C)(NC(C(C(C)C)SCC)=O)C2)cc(C)ccc1F 36358,CCC(C)C(C)CCNC(=O)C(c1cccc(C(F)(F)F)c1)NCC(=O)N(C)C 36359,c1(CN(C2CCS(=O)(=O)C2)CC)cc(NC(C)C)ccc1OC 36360,c1(SC)nc(N2CCCCC2CCNC(=O)CN2C(=O)CNC2=O)cc(Cl)n1 36361,CCC(C)CC(C)C(=O)N(CC(=O)NC1C2CCN(CC2)C1C)C1CCC1 36362,c1(CC(N2CC(C3CC3C(=O)O)C2)=O)c[nH]c2ccccc12 36363,C1(O)(CNC(C(C)n2cccn2)=O)CCCN(C(C23CCCN2CCC3)=O)CC1 36364,c1(C(c2n(CC(=C)C)nnn2)NCCc2cccc(F)c2)cc(F)c(F)cc1F 36365,S(=O)(=O)(C1CCN(CC#Cc2cn(C)cn2)CC1)NC 36366,c1(OCC)ccc(CN2CC3CC3(C(=O)Nc3ccc(Cl)nc3)C2)c(C)c1 36367,C1(C(C)NC(c2cc(C(C)=O)[nH]n2)=O)CCCN(C(c2nnc(C3CC3)s2)=O)C1 36368,N1(C(C(CC=C)(C)C)=O)CCCN(C(=O)C(C2CCC2)OC)C(CO)C1 36369,c1(CCCC)cc(C(N(C(CO)CCC)CCN(C)C)=O)c(C)o1 36370,Cc1cc(C)c(C(=O)Nc2cccc(NC(C3CC3Cl)=O)c2)c(N)c1 36371,C1(O)(CCNC(c2nsnc2O)=O)CCCN(C(C2CC3CCC2C3)=O)C1 36372,N1(C(C(CC)OCC)=O)CCC(O)(C(C)CNC(=O)CCc2nccs2)C1 36373,c1(CN2CCN(C(CC)C(=O)OC)CC2)cc2ccc(C(C)=O)cc2n(C)c1=O 36374,C1(N(C(=O)CCNC(c2cccs2)=O)C)CCC(N=c2nc(C3CC3)[nH]s2)CC1 36375,C1(C(N(C2CN(C(c3cc([N+](=O)[O-])cn3C)=O)C2)C)=O)CCCCC(C)(C)C1 36376,c1(NC(c2cc(-c3c(OCOC)cc(F)cc3)[nH]n2)=O)c(C)cc(C#N)cc1Cl 36377,c1(OC)ccc(Cl)c(OC)c1C(=O)NCC1(C)CN(C(c2cc(C)nn2C)=O)C1 36378,N1(C(CN(C(c2n[nH]c(O)n2)=O)CC)=O)CCCC1C 36379,c1(C(=O)NC(CN(CCC)CC)C)occc1CNC(c1cocn1)=O 36380,Cc1cncc(C(N2CCOC(CN(C)C(c3cc(Br)oc3C)=O)C2)=O)n1 36381,C1(CNC(=O)C(N2CC3CCCC(C2)C3(F)F)=O)CCCC12NC(=O)NC2=O 36382,N1(C(c2cc[n+]([O-])cc2)=O)CCCN(C(=O)CN2CSCCSC2)C(CO)C1 36383,C1(CNC(CCN(C)CC)=O)(NC(=O)CCCCC2CC2)CCCCC1 36384,c1(C(N2C(CNC(C(CCC)(C)CC)=O)COCC2)=O)cc(C)cc2c1CCC2 36385,C1(NC(c2cnc(C(C)C)nc2)=O)CC2CCC1(NC(=O)CCC1CCCC1)C2 36386,c1(C(N2CC(C)(CNC(C(C(=O)NC)(C)C)=O)OCC2)=O)csc2ccccc12 36387,c1(C(=O)NC2CC(F)CN(C(=O)C(Cl)(Cl)Cl)C2)ccc2cccnc2c1 36388,c1(C(C)(C)N(C(C)C)C(c2cccc(F)c2)C2CC2)cc(F)c(Cl)cc1Cl 36389,C1(CCC)(CO)CCN(C(=O)CSCCNC(c2ccnc(OC)c2)=O)C1 36390,Cc1cc(C)c(C(N2CCOC(CCNC(=O)C(C)(F)F)C2)=O)c(O)n1 36391,C(CCC(C)CC(=O)N1CCCC(N(C)C(c2cncn(C)c2=O)=O)C1)=C(C)C 36392,CC1(C)CN(C(C2(c3ccno3)CC2)=O)CCN(C(C2(C)CCC(=O)NC2)=O)C1 36393,c1(CCC)cc(NC(=O)Cn2cc(C(=O)NC3CC(N(C)CC)C3)nn2)ncn1 36394,C#CCCCCC(=O)NCC1CCN(C(=O)CSC)C1 36395,N1(C(C=CSC)=O)CC2CCC(CNC(C3C4CCCCCCC34)=O)(C2)C1 36396,C1(OC)CC(NC(=O)C(C)Cn2ccnc2)CN(C(C2(n3nccn3)CC2)=O)C1 36397,c1(C(=O)NC2C(NC(C3(CCN(C)C)CC3)=O)CC2)cccnc1C(F)(F)F 36398,c1(NCC2C(C)CN(C(c3ccc(=O)n(C)n3)=O)CC2)c(F)cccc1[N+](=O)[O-] 36399,c1(CC)ccc(C(=O)NC(C2CC(F)(F)C2)CNC(C2CSCCS2)=O)o1 36400,N(C(=NCC1(CC2CCC2)CC1)N1CCC(C2CCC2)C1)C(C)C 36401,Cc1cccc(C2CC2)c1CN1CCCC(c2ccno2)C1.c1(=O)c(=O)[nH]1 36402,N1(C(CN(C(C(CC=C)CC)=O)C)=O)CC(C)CC(C)(C)C1 36403,Cc1nc(N2CCC(NC(=O)C(C)N3CCCC3)C(C)(C)C2)c(Cl)cc1C#N 36404,C12(NC(c3nocc3Cl)=O)CCCC1N(C(c1ccc(OC(F)F)cc1)=O)CC2 36405,C1(C(=O)NCCSC)CCN(C(c2coc(N3CCNCC3)n2)=O)CC1O 36406,C1(C(CNC(CC2CC(OC)C2)=O)(C)O)CCN(C(=O)CC2CCC(=O)N2)CC1 36407,c1(OC)cc(P(C)(C)=O)ccc1NC(=O)NC1CCN(c2ccc(F)cc2)C1 36408,Cc1cc(F)c(C(=O)N(CC(O)CN(C(=O)Cc2c[nH]ccc2=O)C)C)cc1F 36409,Cc1cccc(-c2csc(C(=O)NC(C)C(N)=O)c2)n1 36410,Cc1[nH]c(C)c(C(N2CCOC(CNC(=O)CC(C)C(F)F)C2)=O)c1C 36411,c1(C(N2CCC(NC(CC3(N(C)C)COC3)=O)CC2)=O)cc(S(N)(=O)=O)c(C)o1 36412,C1(CNC(c2c(C)cc(C)o2)=O)CCCN(C(=O)CN2CCC(C)C2)CC1 36413,C1(CC(C)C)CCCN(C(=O)CC2CCCN2C(c2cccc[n+]2[O-])=O)C1 36414,C1(CNC(c2ccc(OCCO)cc2)=O)CN(C(=O)COCCCF)CC12CC2 36415,C#CC1(O)CC(C(=O)NC2CCOC(c3ccnn3C)C2)C1 36416,N1(C(C(CSC)C)=O)CCN(C)CC1CNC(C1(C)CCC(=O)NC1)=O 36417,N1(C(COC)=O)CCC(CNC(=O)C(c2cncnc2)C)C(F)(F)C1 36418,c1(C(=O)NCC2CCC(NC(C3CC(OC)C3)=O)C2)cncc(SC)c1 36419,C(C(C(=O)N1CC(C(=O)NC2CC2)C1)N(C)C)NC(C1CC(SC)C1)=O 36420,C1(C(=O)NCc2cc(C)ncc2)COC2(C1)CN(C(C1CCC(=O)C1)=O)C2 36421,NC(=O)CCC(C(=O)O)NC(=O)CC(c1ccccc1)N1CCCC1=O 36422,c1(OCC(=O)NC(CC=C)CNC(C2CCCC2(F)F)=O)ccccc1C(F)F 36423,C1(C)(CC)C=C(C(=O)NC2CC(NC(C3C4CCC3CC4)=O)CC2O)C1 36424,C1(CN(C(C2CCN(CC)C2)=O)CCOC)CCN(C(C2CC(F)(F)C2)=O)CC1 36425,C(=O)(C(C)(C)c1cccs1)NC(C1CC(NC(=O)Cc2cnc[nH]2)C1)C 36426,C1(NC(CC(=O)N(C)C)=O)CN(C(=O)CCCc2ncc(Br)cn2)CC1O 36427,c1(C(=O)NC23C(CN(C(Cc4ccc(C)s4)=O)C2)C3)ccc2ncc(=O)[nH]c2c1 36428,CCCC(C(=O)N1CCC1C(=O)N(CC(C)(O)C1CC1)C)OC 36429,CC1CCN(CC(=O)NCC2CCC(N(C)C(C3(C4CCC4)CC3)=O)CC2)CC1 36430,C(=O)(C(C(C)C)SCC)NCCN(C(C1N(C(CCCC)=O)CSC1)=O)C 36431,CC1CN(C(=O)CCCN2CCCCC2)CC1NC(C1CCC(N(C)C)CC1)=O 36432,N1(C(C(C)c2ccsn2)=O)CCC2(CCC2)C(NC(=O)CCC2CC2)C1 36433,C1(O)(C(C(=O)NC2CC(NC(c3c(C)snn3)=O)C2)(F)F)CCOCC1 36434,N1(C(c2nc(CNC(C(CCC)NC(N)=O)=O)oc2)=O)CCC2(CCCN2C)C1 36435,c1(C(N2CC(OCCNC(CS(CC)=O)=O)C2)=O)cc(C(=O)OC)cc(O)c1 36436,c1(C(N2CCC(NC(C3CC=C(C)CC3)=O)C(O)C2)=O)cc(S(C)(=O)=O)c(C)o1 36437,C1(C)(CNC(NCC(CC)(C)C)=NCC2CCCCO2)CCCC1(F)F 36438,N1(CC(=O)NC2CCC(CNC(C3(N(C)C)CCC3)=O)C2)C(=O)CC(C)(C)C1=O 36439,C1(C(=O)NCC(C(=O)N2CC(OC(C)C)C2)O)CC2CCC2C1 36440,c1(C(N2CC(C)C(C(=O)NC3(C4CCCO4)CC3)C2)=O)cc2ncccc2[nH]1 36441,C(CC(O)C(F)(F)F)NC(C(CSC)(C)NC(c1cccc(F)c1)=O)=O 36442,Cc1nn2c(c1CNC(=O)Cc1ccsn1)CN(C(C1CCC(=O)C1)=O)CC2 36443,c1(C(=O)NCCC2(NC(c3c(C)coc3)=O)CCC2)nn(C)c2ccc(F)cc12 36444,C1(CN(C(c2ccc(COC)o2)=O)CC)CCN(C(C2C3CCCCC23)=O)CC1 36445,CC1CC(=O)NC(C(=O)NCc2ncoc2CCNC(C2CCCOC2)=O)C1 36446,c1(C(=O)NCc2c(C(N(C(CCC)C)C)=O)scc2)cc(OC)n(C)n1 36447,C1(CC)COCCN(C(c2cc(CNC(=O)C(C)SC(C)C)on2)=O)C1 36448,C1(C)(NC(CC2(COC)CC2)=O)CCN(C(c2ccc(C)c(N)c2)=O)CC1 36449,c1(C(=O)NCC(CC)(CC)NC(c2ccn(C)n2)=O)c(O)cc(F)cc1F 36450,C(=O)(C(O)Cc1ccccc1)NCCCN(C(=O)CC1CCCO1)C(C)C 36451,c1(-n2c(C(CC=C)CC)nc(-c3ccnn3C)n2)ccc(S(=O)(=O)CC)cc1 36452,C1(C(=O)NCCCC#C)CN(C(C23CCC(CC2O)C3)=O)CC(C)(C)C1 36453,C1(C(N(C)Cc2ccc(CC)o2)=O)CN(C(=O)C(C#N)(CC)CC)CC(C)(C)C1 36454,c1(NC(C2CC(F)(F)C2)C)[nH]c(=NC2CC2c2ccccc2)nc2scnc12 36455,Cc1ccc(=O)n(CC(=O)NCC(C)NC(=O)Cc2cc(Br)cs2)n1 36456,c1(C(C(C)NCc2cnn(C(F)F)c2)O)ccc(F)cc1F 36457,C=CC(CC)CC(=O)NCCC1CSCCN1C(c1n[nH]c(C2CC2)c1Cl)=O 36458,c1(OC)nc(C(=O)NCC(C)CNC(=O)CCC(=O)c2ccccc2)cc(O)n1 36459,N#Cc1c[nH]c(=NC(=O)C2CCC(C(=O)Nc3ncc(F)cc3Br)CC2)cc1F 36460,C(C(C)NC(=O)CCc1cc(C)n(C)n1)(C(C)C)NC(C1C(c2cc(C)no2)C1)=O 36461,C(=O)(C(CC(F)F)C1CCC1)NC1CC(CNC(=O)CCn2cncn2)CC1O 36462,C1(F)(C(=O)NCC(Cc2ccccc2)N(C)C(C2(CO)CC2)=O)CCOCC1 36463,c1(C(N(CCCCN(C(C(CSC)O)=O)C)C)=O)ccc2nnnn2c1 36464,N1(C(c2c(OC)cccc2)=O)CCC(C)C(CNC(=O)CCc2cccs2)C1 36465,CN1CCC(C(=O)N(C)CC2CCN(C(C3CCCC34CCC4)=O)CC2)S1(=O)=O 36466,Cc1cc(C)n(C(C)CNC(N2CCCC2CCCc2ccncc2)=O)n1 36467,c1(OC)cc(F)c(F)cc1NNC(=O)Nc1ccc(C(C)(C)C)nc1 36468,c1(C(=O)NC(C2N(C(C3CC(OC)C3)=O)CCC2)C)ncnc2c1CCC2 36469,CN1CCC(F)(C(N2CC3(CCC3NC(c3ccc(N(C)C)nn3)=O)C2)=O)CC1 36470,C1(NC(c2ccc(SC)cc2)=O)CCCC(NC(C2(c3cc[nH]n3)CC2)=O)CC1 36471,c1(CC(=O)NC2CN(C(C(P(C)(C)=O)O)=O)CC23CC3)cc(Cl)cc2c1OCC2 36472,C(=O)(C(O)C(C)(C)C)N1CCC(n2cc(CNC(C3CC(C)OCC3)=O)nn2)C1 36473,Cn1nnnc1SCCC(=O)NCC(C1CCCC1)NC(=O)Cn1cncn1 36474,c1(CC)c(C(N2CCCCC2CNC(=O)CCc2nncn2C)=O)ccn1C 36475,C1(C)(CC(=O)NC2CC(F)(C(C)(C)C)C2)CCS(=O)(=O)N1.C12CC1C(=O)NC2 36476,C(CCCCC(=O)N(CC(C)O)CCNC(C1CC(O)CN1C)=O)OCC 36477,C(=O)(C(C)(C)CCNC(=O)C(C)N1CC(C)C1)N1CC(C(CC)CC)C1 36478,C1(NC(C2(N(C)C)CC2)=O)CCN(C(=O)CCC2CC2)CC1F 36479,N(C1CCCc2ccoc21)C(C1N(C(=O)Cn2ncccc2=O)CCN(C)C1)=O 36480,C1(CNC(C2(CC)CC2)=O)CN(C(c2snnc2C2CC2)=O)CCC1(C)C 36481,C(C(C)C(=O)NCC(O)CNC(=O)CCOCc1ccccc1)NC(C)=O 36482,N1(C(C)C)CCCN(C(C2CCC(C(C)C)N2C(=O)C2=CCOCC2)=O)CC1 36483,CC1=CCSC1C(=O)NCc1ccsc1C(=O)NCCC(C)N(C)C 36484,C(=O)(CC1=NN(C)C(=O)C1)NCCN(C(C1(C(=O)OCC)CC=CCC1)=O)CC 36485,C1(O)(CN(C(CN2CC(C)C2)=O)C)CCCN(C(=O)CCS(C)=O)C1 36486,c1(N2C(CNC(c3cn(C(C)C)nn3)=O)CCCC2)ccc([N+](=O)[O-])cc1C#N 36487,c1(C(=O)NCC(C2CC2)NC(c2ccc(CC)c(N)c2)=O)cccc2scnc12 36488,c1(C(N2CCC3(CN(C(C(CC(C)C)OC)=O)C3)C2)=O)cc2nc(=O)ccn2[nH]1 36489,C1(C(=O)OC)CN(C)CCN1C(=O)CN(c1cccc(I)c1)C 36490,c1(C(N2CC(NC(C3C(=C)CC3)=O)C3(C2)CC3)=O)cc(Br)c(OC)cc1N 36491,c1(CC)cccc2[nH]c(C(N3CCC(CNC(=O)CSC)C34CCC4)=O)cc12 36492,CC1=CCC(C(N2CCCC2CCCNC(=O)CC(C)(C)C)=O)CC1 36493,c1(C(N2C3(C(N(C4CCCCC4)CC#C)=O)CC(C2)C3)=O)cc2ccccn2n1 36494,C1(NC(C(C2CCC2)OCC)=O)CC(OC)CN(C(c2cccc(SC)n2)=O)C1 36495,c1(C(CC)C)nccc(N2CC(C)(C)C2C2CCN(C(c3cncs3)=O)CC2)n1 36496,C1(C(=O)Nc2ccc(N(C)C)cc2)CCN(C(=O)NC2COC2)C12CCC2 36497,c1(C(=O)Nc2cccc(CNC(CCN(C)CCO)=O)c2)coc2ccccc12 36498,N1(C(C2CCC(CC)C2)=O)CCC(C=CC(=O)NC(CCO)C(F)F)CC1 36499,N1(C(C2CC(C#C)(O)C2)=O)CC(NC(c2cnn(CC(F)(F)F)c2)=O)CC1(C)C 36500,C(=O)(C(CC)CC=CC)N1CC(CN(C(CC2CC(=C)C2)=O)C)OCC1 36501,C1(NC(c2cccnc2C2CC2)=O)CN(C(=O)Cc2cccs2)CC1F 36502,C1(CNC(c2ccsc2)=O)CN(C(=O)CC2CCC3(CCC3)O2)C2(CCC2)C1 36503,C1(C(=O)NCC2(CNC(c3cnc(C)nc3)=O)CCCC2)CCC(C)(C)CC1 36504,C(=O)(CCCCCCCCC)N(CC(CNC(C1(CC#C)CCC1)=O)(C)C)C 36505,c1(C(N2CCC3(CCN(C(C45CC(F)(C4)C5)=O)C3)C2)=O)cnc2ncnn2c1O 36506,CCC(C)CC(C(=O)NC(C)C(C)SC)NC(c1cnc2n1CCC2)=O 36507,CCC(CC)C(C)C(=O)NC(C)(C(=O)NCC1=CCCCC1)C1CCC1 36508,C1(O)(CNC(C2(CC(C)C)COC2)=O)CN(C(=O)CCc2cnccn2)C1 36509,C1(CNC(c2c(C)scc2)=O)C(C2CC2)CCN1C(c1coc(C(C)C)n1)=O 36510,C1(NC(c2c(C#C)c[nH]n2)=O)CC2CC1CN(C(C1CCS(=O)(=O)CC1)=O)C2 36511,CC1CCC(NC(=O)C(C)(C)c2cncnc2)CN1C(=O)C=Cc1ncc[nH]1 36512,C1(CC#N)C(=O)C(=O)N1.c1(OCCCNC(COC(C)(C)C)=O)ccccc1 36513,C12CC3(CC3)CN1C(=O)C2.C1(COCCNC(C2CCC2)=O)CCCO1 36514,N1(C(=O)NCC(c2cnn(C)c2)OC)CCCC2(C1)OCc1ccccc12 36515,CCC(C)(C)CC(=O)NCC1CN(C)CCN1C(c1cc(Cl)ccc1OC)=O 36516,C1(O)(C(=O)NC2(CNC(=O)Cc3cc(C)ns3)CC(OC)C2)CC2CCC1C2 36517,C#CCC(CC#C)NC(=O)C(Cn1ccnn1)NC(=O)CC1CCNC1=O 36518,N1(C(C(Cc2cc[nH]n2)NC(c2cc(O)cc(=O)o2)=O)=O)CCC(F)(F)C(CO)C1 36519,C1(NC(COC(CC)C)=O)CC(C(F)C(=O)N(C2CC2(C)C)C)C1 36520,C1(CC)(NC(=O)C(c2ccc(F)c(Cl)c2)C)CCN(C(=O)C(C)S(N)(=O)=O)CC1 36521,CC(CC(F)F)C(=O)N(C1CCC(NC(=O)C(C)N2CCC2)CC1)C 36522,N1(C(c2c(C(C)(C)C)ccs2)=O)CC2CC1CN2C(c1n[nH]cc1Br)=O 36523,N1(C(C(C(C)C)n2cccc2)=O)CCN(C)CC1CNC(=O)CC1CC=CC1 36524,C1(NCc2c(CC)nsc2)CCc2nncn2C1 36525,c1(CNC(C(CC)CC)=O)nnc2n1CCN(C(C1(C(C)C)CCC1)=O)C2 36526,CC1(C)OC(=O)CC1C(=O)NC1CCCN(C(c2cnn(-c3nccs3)c2)=O)C1 36527,N1(C(C(CC2CN(C(C(CCN(C)C)O)=O)C2)F)=O)CC2(C1)CC(C)(F)C2 36528,N1(C(c2c(C)cco2)=O)CCC2(CC1)CN(C(C1CC(C)OC(C)C1)=O)CC2CO 36529,C1(NC(c2n(CCC)nnn2)(C)CCBr)CC(=O)N(c2ccc(Br)cc2)C1 36530,CCCC(C(=O)N1CC(CNC(c2cocn2)=O)(COC)C1)C(C)C 36531,C1(NC(=O)CC2CCCCC2)CC(F)CN(C(=O)C(F)F)C1 36532,C1(NC(c2c(C(C)C)nns2)=O)CCN(CCNC(C2CC2(Cl)Cl)=O)CC1 36533,N(C(=NCCC(=O)NC1CCCCC1C1CC1)NCc1ccccc1C#N)CC 36534,C(CCN=c1cc(C)nc(CC)[nH]1)N(CC)CC.c1ccc(C(F)(F)F)cn1 36535,C1(N(C)C(c2cc[nH]n2)=O)CC2CCC(C1)N2C(=O)Cc1csc(Br)c1 36536,N1(C(C(=O)NCC)=O)CCC2(CC1)COC(CNC(c1c(Cl)nn(C)c1C)=O)C2 36537,Cc1c(Cl)ccc(C(=O)NC2CN(C(c3cccc(=O)n3C)=O)CC2CO)c1O 36538,C1(NC(COC2C(CC)CCCC2)=O)CCN(C(c2cc(O)cs2)=O)C(C)C1 36539,Cc1nc(Cl)nc(N2CC3CCC2CN3C(c2ncc(F)cc2F)=O)c1[N+](=O)[O-] 36540,C(=O)(C(C)(C)C(C)(C)O)N1CCC(O)(CCNC(COCCSC)=O)C1 36541,Cc1nnccc1C(=O)NCc1cccnc1N1CCNC(=O)C1 36542,c1(COC)nnc(CNC(=O)NC(c2nnc(C)o2)C)s1 36543,n1(CC(=O)NCC2CN(C(c3ccccc3CO)=O)C2)nc(Cl)ccc1=O 36544,CC1CN(C(c2scnc2C(F)(F)F)=O)CCN1C(C1CC2(CCOC2)C1)=O 36545,c1(-c2occ(N(CCCCC(=O)O)C)n2)ccc(P(C)(C)=O)cc1 36546,c1(C(N2CCC(C)(c3cn[nH]c3)CC2)C(=O)NC(C)(C)C)cc(S(N)(=O)=O)cs1 36547,Cc1ccc2c(C(=O)NC3CCC(C)N(C(=O)CCOC4CC4)C3)ccnc2c1 36548,c1(Cn2c(NC(N(C(C#C)C3CCC3)C)=O)ccn2)ccc(Br)cc1F 36549,CC1CCC(NC(c2cc(N)ccc2F)=O)CN1C(=O)C=CC(=O)OC(C)(C)C 36550,C1(CN(C)C(C2(C(N)=O)CCC2)=O)CCN(C(c2c[nH]nc2C2CCOC2)=O)C1 36551,C1(C(N(C2CCN(C(c3conc3C3(C)COC3)=O)C2)C)=O)COC(=O)N1 36552,c1(C(N(CCN(C(=O)Cn2ccc(C)n2)CC)CC)=O)ccnc(F)c1OC 36553,c1(SC)cc(C(=O)NCC23CC2CN(C(c2ccnn2C2CC2)=O)C3)ccc1F 36554,N#Cc1c(C(=O)NC2CC(NC(c3n[nH]c4c3COCC4)=O)C2)cccc1F 36555,N1(CC(=C)C)CCCC(C)C1C(=O)C(C)N(C)C 36556,C1(C(C)NC(c2nc(CC)sc2)=O)CCN(C(c2cc(C3CCC3)[nH]n2)=O)CC1 36557,c1(NC(C2COCCN2Cc2cnc(Cl)c(F)c2)=O)cc2c[nH]nc2cc1F 36558,c1(CC(=O)NCC2(CNC(C3C(C#N)C3)=O)CC23CCC3)cccc2cnccc12 36559,Cc1cc(C(=O)NCc2cc[nH]c2C(=O)NCCc2cnn(C)c2)cc(C#N)c1 36560,N1(C(C=Cc2occ(C)n2)=O)CCCC(O)(CNC(=O)CC2CC3CC3C2)C1 36561,N1(C(c2c(CC)ocn2)=O)CCCC(C)C1CNC(=O)Cn1nc(C)n(C)c1=O 36562,C1(OC)CC2(C1)CN(C(=O)C(O)CCNC(=O)Cc1cncs1)C2 36563,C(CN=C(NCc1cc(O)cc(O)c1)NCc1cc(C)ccn1)N(CC)CC 36564,c1(CC(=O)NCC2(C(=O)NCC(C)Cn3cccn3)CCC2)cccn1C 36565,c1(C(=O)NCC2CN(C(CSCC#C)=O)CC2O)c(Cl)sc(C)c1C 36566,c1(NC2(CNC(CC(=O)OC)=O)COC2)cc(Br)c(F)cc1OC 36567,C1(OC)CC(NC(c2cc(C)ns2)=O)CN(C(C2CCC(=O)N2C2CC2)=O)C1 36568,C1(CC(=O)N(C2(C(N)=O)C(C)C2)C)CCCC1NC(=O)Cc1ccn(C)c1 36569,Cc1nncc(C(=O)N(C(C)CNC(=O)CCC2CCCCN2C)C)c1C 36570,C1(C(N(CCN(C(CC2C(OCC)COCC2)=O)C)C)=O)CC(=O)NC1(C)C 36571,N1(C(Cc2ncc(CC)[nH]2)=O)CC2(NC(=O)CCCn3cccc3)CC1C2 36572,c1(C(=O)NC(CC)CNC(=O)C(C)(CC)C(F)F)ccnc2ccc(Cl)cc12 36573,N1(C(C2CCCC(C)CC2)=O)CC2(CC(NC(c3ccnn3CCF)=O)CO2)C1 36574,C(CCC(N)=O)(C(=O)NCC1CCN1C(=O)C=CCN1CCCCC1)N(C)C 36575,C(C(C(=O)NCCNC(=O)CO)C(C)C)NC(CCC=C)=O 36576,C(=O)(CCC(=O)NN(C)C)NC1CC(C)CN(C(c2ccoc2Br)=O)C1 36577,c1(CC)nc(C)c(C(N2CC(C(=O)NC(C)(CO)C3CC3)(CC)C2)=O)o1 36578,C1(C(=O)CC2CC2C(=O)OC)CCCN(C(=O)C(=O)C(COC)=O)C1C 36579,N1(C(c2nccc(C)c2O)=O)CC2CCCC(NC(=O)CCSCC(N)=O)C2C1 36580,c1(C(N(C2COCC2CNC(=O)CCOC2CC2)C)=O)c(F)cccc1[N+](=O)[O-] 36581,N1(C(CC(C)(C)N(C(c2cc(CC)ncc2)=O)C)=O)CCN(C)C(C)C1C 36582,c1(C(N2C(CNC(c3[nH]cc(C(C)=O)c3)=O)CCC2)=O)cc(C)n(C)c(=O)c1 36583,C(=O)(C(C)(O)CC(C)C)NC(CC(=O)NCc1snc(CC)n1)C(C)C 36584,C(=O)(C#CC1CCOCC1)NC1CCC(CNC(C(c2ccccc2)C)=O)CC1 36585,C(CC(=O)NCC(c1cccnc1)O)(CC(C)C)NC(c1cccc(C)c1O)=O 36586,C1(C(=O)NC(C2CCCCC2)C#C)COCCN1C(c1ccnc(C)n1)=O 36587,CCCS(=O)(=O)c1ccccc1C(=O)NCCCCCNC(C1CC1F)=O 36588,Cc1nc(C(=O)NC2CC2CNC(=O)C=CC2CCCCCC2)c(C)n1C 36589,n1(CCC)nccc1C(=O)NC1CCC1CNC(C1CCC(C(=O)OC)C1)=O 36590,C1(C(c2n(CCSC)nnn2)NCCc2ccncc2)CC2CCC1CC2 36591,c1(OCC)ccc(C)cc1CN=C(NCC1(C#N)CCOCC1)NC1CC1C 36592,Cc1ccc(S(=O)(=O)NC2CCCC2C(N2CCC(O)C(C)C2)=O)c(F)c1 36593,N1(Cc2nnc(CC)s2)CC2(C)CN(C(=O)CCCCOC)CC2(C)C1 36594,c1(C(N2CCC(NC(c3cnc(=N)[nH]c3)=O)C2)=O)ccc2c(c1)CCCS2 36595,C1(N(C(CCN(C(CC(C)SC)=O)CCO)=O)C)CCOC(C)(C)C1 36596,C1(C#CC(=O)NC(CNC(=O)C=C(C)c2ccccc2C)C(C)C)(CC)COC1 36597,C12(CNC(C3OCCN(C)C3)=O)CCC(CNC(C3CC3[N+](=O)[O-])=O)(CC1)CO2 36598,c1(CNC(C(C)O)(C)C2CCOCC2)ccc(Br)cc1OOC(F)F 36599,N1(C(C)=O)CCC(CC(=O)O)C(NC(=O)Cc2cc(C)nn2C)C1 36600,C(=O)(NNc1cc2ccccc2cn1)c1c(-c2ccn(C)n2)ncs1 36601,Cn1ncc(C(=O)NC2CC3CC(C2)N(C(=O)C(C)(C)C)C3)c1S(N)(=O)=O 36602,CC(C)C(O)C(=O)N1CCSCC1CCN.c1(C(=O)NC2(C)CC2)ccncc1 36603,c1(CC)ccc(C)c(C(=O)NC(C)C(C)(C)NC(=O)CN2CCSCC2)c1 36604,CC1CCc2nc(C(=O)NCC3CCCC3NC(=O)CC(C)(C)O)ccc2C1 36605,C1(NC(c2nc(-c3c(C)cccc3)sc2)=O)(CNC(=O)C(N)=O)CC2CCC1C2 36606,Cc1ccc(F)cc1C(=O)N(C(C)CN(C)C(C1CC2(CCC2)CO1)=O)C 36607,n1(CCC)ncnc1CNC(=O)C(C)(C1CCC1)NC(=O)C(N1CCOC1=O)C 36608,c1(C(=O)NCCNC(c2ccc(S(C)(=O)=O)s2)=O)cccc2nc(Cl)cn12 36609,C(=O)(N=c1[nH]nc(C2CC2)s1)OC(C)(C)C.c12ccccc1CN2C 36610,C1(COC)(NC(=O)C=CC(F)(F)F)CCN(C(=O)Cn2cnc(=N)[nH]2)CC1 36611,Cc1nc(F)ccc1CNC(C1CCN(C(=O)C(CO)N(C)C)C1(C)C)=O 36612,CCC(N=c1ccnc(NC2CCN(CCC(C)(C)C)CC2)[nH]1)C(C)C 36613,C1(CC(=O)N(CCn2c(C)ncc2)C)COCCN1C(C1CCC(C)(C)C1)=O 36614,CC(C(=O)N1CCCC1CCNC(c1c[nH]cc1C(F)(F)F)=O)C(F)(F)C(F)F 36615,CCCCCC(F)C(=O)NCC1(O)CCN(C(=O)C(C)(C)c2cscn2)C1 36616,N1(C(C(C)NC(CC)=O)=O)CC(=O)NCC1C(=O)NCC1(O)CCN(C)C1 36617,N1(C(COC)=O)CCCC(C)(C)C1CNC(C1(Cc2ccc(F)cc2)CC1)=O 36618,c1(CC2(NC(COc3c(F)ccc(C)c3)=O)CCCC2)cn2ccccc2n1 36619,C1(CNC(CCCOCC)=O)CCCC(NC(=O)CCc2nnc(C(F)F)o2)C1 36620,c1(N2CC(CNC(c3cc(C)no3)=O)OCC2)ncnc2scc(C)c12 36621,c1(N2CCC(O)(C(C)NC(c3c(CC)nns3)=O)C2)ncc([N+](=O)[O-])cc1F 36622,C1(C(=O)NC(CCCNC(CCC(=O)NCC)=O)C)COCC(C)(C)O1 36623,N1(C(c2ccn(C)c2)=O)CCC(C(C)C(=O)NCc2ccncc2F)CC1 36624,CC(C)(C)CC(=O)NCC1CC(C(N2CCC(c3nc[nH]n3)C2)=O)CO1 36625,C1(C(=O)NCC(C)NC(c2cnn(C3CCCC3)c2)=O)OCC1(C)C 36626,C1(NC(c2ccc(OC)c(Br)n2)=O)CCc2ncc(Br)n2C1 36627,c1(C(=O)NC2(CC=C)CCN(C(=O)C(CC)SC)C2)cc2c(=O)[nH]ccn2c1 36628,n1(CC)cnc(C(=O)NC(CO)C(C)NC(=O)CCNC(C2CCOCC2)=O)c1 36629,C(=O)(C(F)CCC(C)(C)C)N(C1CCCN(C(C(CC)NC(C)=O)=O)C1)CCF 36630,Cc1cc(C(N2CCC(F)(CNC(C3CCCN3C3CC3)=O)C2)=O)nnc1C 36631,CN=c1[nH]cc(C(=O)N(C)CCN(C(=O)Cc2cnn(C(C)C)c2)C(C)C)s1 36632,C(c1ccc(F)c(Cl)c1)=CC(N1C(CNC(C2C(OC)CCC2)=O)CC(O)C1)=O 36633,C1(N(C(=O)C=CC(C)(C)C)CC)CCN(C(=O)C=Cc2csc(C)n2)CC1 36634,c1(OC2CN(CC(c3ccc(C(=O)O)cc3)O)C2)ccc(Cl)cc1[N+](=O)[O-] 36635,C1(CCNC(C(C)SC)=O)CCN(C(=O)CC2CC(C)(C)CC2)CC1 36636,N1(CCC)CC(NC(=O)C(C)(C)CNC(=O)CCC2CCCCC2)CC1=O 36637,C1(C2CCOCC2)(C(=O)NCC(C(C)(C)C)NC(C(C)CC(F)F)=O)CC1 36638,C1(CNC(C(CC=CC)NC(=O)CCOCC2CC2)=O)OC(=O)CC1(C)C 36639,Cc1cc(C)c(C(=O)NCCC(C)(C)NC(c2cc3c(ccn3C)[nH]2)=O)c(=O)o1 36640,C(=O)(C1=CC2(CN(C(=O)Cn3cnc(=N)[nH]3)C2)OC1)N(CCC#C)C 36641,C1(NC(C(CCC)=CCC)=O)CCCC(C(=O)NCCN2CCCOCC2)CC1 36642,C(C(F)(F)C(F)F)OCC1(OC)CCC1.C1(CON)CC1 36643,C1(CNC(C(CC)CO)=O)CCN(C(c2cnn(C3CCCC3)c2)=O)C1(C)C 36644,c1(C(N2C(CNC(C(C)SCCCC)=O)CC(C)(C)C2)=O)ccc2cnoc2c1 36645,c1(C(C)C)cccc(OCC(=O)NCCCCC(C)NC(=O)C=CCO)c1 36646,c1(C(N2CCCC(CC(N)C(F)(F)F)C2)=O)cc(Cl)ccc1I 36647,CCCC(C(=O)NCC1CCCCN(C(=O)CCN2CCOCC2)C1)S(N)(=O)=O 36648,Cc1noc(C(F)F)c1C(=O)NCc1cccc(CN(C(=O)C(C)(C)F)C)c1 36649,C1(NC(c2cc(C(C)=O)on2)=O)CCC(C)(CNC(c2cnccn2)=O)C1 36650,c1(CC(N2CC(O)(CNC(C3CC(CCC)C3)=O)C2)=O)sc(C)nc1C 36651,c1(OC)ccc(Cl)c(OC(F)F)c1C(N1CCC(C)CC1C)=O 36652,c1(C(N2CC(CNC(CC3(C=C)CC3)=O)C(C)(C)C2)=O)c(C)ccc(OC)c1N 36653,c1(N(C)CC2CCCCC2)nc2c(c(=NCC3CCC=CCCC3)[nH]1)COC2 36654,CCC(C)C(=O)NCC(=O)NCCN(C)C(C1CC(OC(=O)NCC)C1)=O 36655,N1(C(c2c(C)snc2)=O)C2CCC1C(CNC(=O)CCc1nc(=N)[nH][nH]1)C2 36656,CC1(NC(c2c[nH]nc2-c2ccncc2)=O)CCN(C(=O)CC=C(Cl)Cl)C1 36657,C1(C(=O)NCC23CC(NC(c4ccc(SC)s4)=O)(C2)C3)CC(C)(C)C1C(F)(F)F 36658,N1(C(CC(COC)C)=O)CCC2CCCC12C(N1CCCCC(N(C)C)C1)=O 36659,C=C(Br)CC(C)(C)C(=O)N1CC(CNC(=O)C(C)NS(C)(=O)=O)C(C)C1 36660,c1(N2CCC(C)OCC2)ccc(S(=O)(=O)NC2CCCC(CC(N)=O)C2)c(Br)c1 36661,C(CC1CC(=O)N1)OC(=O)CCn1ccnc1.c1(OC2(CF)CC2)ccccc1 36662,N1(CCNC(C(c2cscn2)N(C)C)=O)C(=O)NC(C)(c2ccc(Br)cc2)C1=O 36663,c1(-c2c(C(=O)NC(C)C(C)n3ccnc3)c[nH]n2)ccc2c(c1)CCCO2 36664,c1(C(N2C(CNC(c3c(C)nccc3)=O)CCCC2)=O)ccc(C(C)C)c(Cl)c1 36665,c1(C(CNC(=O)CCc2ccon2)NC(C2CCCS2)=O)ccc(Cl)cc1 36666,c1(C(N(CCNC(CNCC(=O)NC)=O)C)=O)ccc(N)c(OCCO)c1 36667,C1(C(=O)NC(CCN(C(=O)C=C2CCCCC2)C)(C)C)CC(C)(C)OC1(C)C 36668,C(=O)(C#CC1CCCCC1)N1CCCC(CCC(=O)NCC2(O)CCC(C)C2)C1 36669,C1(CC)CNC(=O)CN1C(=O)CC=CCNC(C1CC12CC2)=O 36670,C1(C(=O)NC2C(NC(C3(CC#C)CCCC3)=O)CCC2)CC2C=CC1C2 36671,c1(C(=O)NCCC2(NC(=O)C=Cc3ccncc3)CC2)cccn2cncc12 36672,Cc1ccc([N+](=O)[O-])cc1C(N1CCC2CN(C(C3(C#N)CC=CC3)=O)CC12)=O 36673,c1(N)nccc(C)c1O.C(=O)(CC(Cc1ccc(F)cc1)NC(=O)OC(C)(C)C)OC 36674,CCCCC(F)F.C1(=O)C(CCC2CC2)O1.C(C)(C)(C)OC=O 36675,C12(C(N3CCCN(C(=O)CNc4ncccn4)CC3)=O)CCCCC1C2(F)F 36676,C1(CC(N2CC3=C(CN(C(CC(C)SC)=O)C3)C2)=O)CCc2ccccc2C1=O 36677,C(c1ccc(C)cc1)=CC(=O)NCC1(C(=O)Nc2ccc(CC)cc2)CC1 36678,Cc1cc(F)cc(C(N2CC(N(C)C(C3CCOCC3)=O)C3(CC3)C2)=O)c1O 36679,C=CCC(Cc1ccccc1)C(=O)NCCCOc1c(F)cccc1F 36680,N1(C(C(C)SC)=O)CCC(CN(C(c2cnccn2)C2CCCC2)CC)C12CCC2 36681,N1(C(C=Cc2cc(C)no2)=O)CC2CCC(N(C(=O)C3=CCCSC3)C)C2C1 36682,c1(C(N2C(C)(C(=O)NC)CC(O)C2)=O)nccc2[nH]ccc12 36683,C(CNC(=O)Cc1ccccc1)(C(C)(C)C)NC(CCN(C)CCO)=O 36684,C1(C(=O)NCCCN2CC=CC2)CCC(O)CN1C(c1cc(C(F)F)[nH]n1)=O 36685,N(C(=NCc1ccccc1NC(C)=O)N1CCC(C)(F)C1)C(CC)C 36686,c1(N2C(CNC(c3c(C(C)C)con3)=O)C=CC2)ccnc(-c2ccccc2)n1 36687,C1(OC)(CNC(c2n[nH]c(C)c2O)=O)CCN(C(c2cn(CCO)nn2)=O)C1 36688,CC1CC2(CCN(C3CCN(C)C3=O)CC2)CN1C(C1CC1(Cl)Cl)=O 36689,c1(OS(NC(C)C)(=O)=O)cccnc1OC(N1CC(OCCO)C1)=O 36690,N1(C(c2c(C)ccc(C)c2Br)=O)CCC2(CC1)CC(NC(=O)CCC(C)C)CO2 36691,c1(C(=O)NCCCN(C(=O)C(CC)OCC)CCC)cc(C(N)=O)[nH]n1 36692,N1(C(CC2(OCC)CC2)=O)CCC(O)(C(C)NC(c2cnc(C3CCC3)o2)=O)C1 36693,C1(NC(c2ccnc(F)c2Cl)=O)CC2CC1CN2C(c1ccc[n+]([O-])c1)=O 36694,C#CCCCCCC(=O)NC1CC1CNC(=O)C1=C(C)OCC1 36695,N1(C(c2scc(C)c2C)=O)CC(CO)C2(C1)CN(C(C1CCN(C)C1=O)=O)C2 36696,C(=O)(C(C)(C)CCCF)N(CCC(=O)NCc1c(C)cc(O)cc1)CCCO 36697,N1(C(CCSCC)=O)CCCC(F)(C(=O)NC2C3CCCC23)C1 36698,C1(CNC(C2CC3(C2)CC3F)=O)COCCN1C(=O)Cn1cnnc1O 36699,CC1CN(CCCc2cc(Cl)no2)C12CCOCC2.c1(C(C)(C)O)cn(CC)nn1 36700,c1(OCCC(N2CCC(NC(c3c(C)nn(C)c3)=O)C2)=O)cc(Cl)cc(Cl)c1 36701,CC(=O)C(C)(C)CC(=O)N(C)CC1(c2ccccc2)CC1 36702,C(C)(CCC(=O)N1CCCCC1C1(NC(c2[nH]cnc2C)=O)CC1)SC 36703,N1(CC)CCC(NC(=O)C(F)CC2CN(C(C3(CO)CCCO3)=O)C2)C1 36704,C1(C(C)C)CCC(C(=O)NCC(c2cccnc2)O)N1C(c1cc(Cl)ccn1)=O 36705,C1(CNC(CC(C)SC)=O)CN(C(c2ccc(Cl)c(C)c2N)=O)CC12CCC2 36706,C(=O)(CCCCCNC(C)=O)NCC1CC(NC(COCCC)=O)C1 36707,C(=O)(C(C)C(C)(C)C)NCCCN(C(=O)C=Cc1cccc(CO)c1)CC 36708,c1(C(N)=O)ccncc1NC(=O)Nc1cc(CSC2CCCCO2)on1 36709,c1(CC)ccc(F)c(C(=O)NCC2CC(F)CN2C(c2nnc(S)n2C)=O)c1F 36710,C1(CNC(c2c(C)cncc2C)=O)COC(C)(C)CN1C(c1cc(Cl)cn1C)=O 36711,N1(C(C(N)=O)=O)CC2CC1CN(C(c1cc(C(N)=O)co1)=O)C2.N1(C=O)CCCC1 36712,C1(NC(C(=Cc2ccccn2)C)=O)C2CCC1N(C(c1cc(C(F)F)no1)=O)C2 36713,C1(C2CC2)(C(=O)NCC(c2ccccc2)CNC(C)=O)CC1 36714,CCCC(C)CC(=O)NCCCC(O)C(=O)NCc1cncc(C)c1 36715,C(CCCCCC(=O)N1CC2(CO)CC2(CO)C1)NC(c1c(NC)cccc1)=O 36716,c1(C(=O)NC2CC(CO)N(C(c3ncccc3F)=O)C2)ccc2c(c1)OCCO2 36717,Cc1c(NCCCN(c2ccccn2)C)nc[nH]c1=NCc1cc(Br)no1 36718,N1(C(C(C)OCC=C)=O)CCC(NC(=O)CC2(C)CCOCC2)C1C(C)(C)C 36719,c1(OC)ccc(C(C)C(N2CCCN(C(C3CC4(C3)CC4F)=O)CC2)=O)c(C)c1 36720,C1(C)(CC(=O)OC(C(C(C)C)n2cncn2)=O)CCCN(C(=O)OC(C)(C)C)C1 36721,c1(NCCCCCC(N)=O)[nH]c(=NCCCC2CCCCC2O)nc2scnc12 36722,c1(C(=O)NC(CCC)CNC(c2cncn2C)=O)c(OC)nsc1OC 36723,C#CCCCC(C)C(=O)N1CCOC(CC(=O)NC(c2n[nH]c(C)n2)C)C1 36724,C1(C(=O)Nc2cc(OC)c(O)cc2)CC12CCN(C(c1cc(O)n(C)n1)=O)CC2 36725,CCS(=O)(=O)CCN=c1[nH]c(N2CCCCC(C3CCOC3)C2)nc2c1COC2 36726,Cc1ccc(CC(N2CCC2CNC(=O)CN(S(C)(=O)=O)C)=O)c(Cl)c1 36727,C1(O)(N(C(=O)COC(C)(C)CC)CC#C)CCN(C(c2ccc(NC)cc2)=O)C1 36728,C(=O)(C=C1SCC(=O)N1C)NC1CCN(C(c2n(CCC)ccc2)=O)CC1O 36729,CC1CC(C(=O)NC2(CCNC(=O)Cc3ccc(Br)nc3)CCCC2)=NO1 36730,C(=O)(C1CCc2ccccc21)N1CCC(CNS(C(CC)C(C)C)(=O)=O)CC1 36731,c1(CC(=O)NCCC(C)NC(C2CC23CC3)=O)c[nH]c2ccc(Cl)cc12 36732,N1(C(=O)CC2CCCN(C(c3cnn(C(F)F)c3)=O)C2)CCC(CO)C(F)C1 36733,CC(CCCCNC(C1CCCCC1O)=O)NC(c1ccnc(C2CC2)c1)=O 36734,c1(CC(=O)NCC2C(NC(=O)Cc3sccc3Cl)CC2)ccccc1Cl 36735,c1(CNC(c2cc(C)ns2)=O)nc(C)c(C(=O)N(CC(=O)NC(C)(C)C)C)o1 36736,CC1=NOC(C)(C(=O)NC(CNC(=O)Cn2nc(C)cc2C(F)F)CO)C1 36737,C(C1=NOC2CN(C(=O)C=CS(F)(F)(F)(F)F)CC12)NC(=O)C1=C(Cl)CCC1 36738,C(CCC(=O)NNC(=O)NCc1ccc(N(C)C)cc1)c1cn(C)nc1 36739,C(c1c(C)noc1C)=CC(N1CCC(N(CCC)C(C2CCCN2C=O)=O)C1)=O 36740,N1(C(CC(CC)C2CCC2)=O)CCN(C(C2CCc3c[nH]nc3C2)=O)CC(O)C1 36741,N1(C(c2ccc(N)c(N)n2)=O)CCC(C2CCN(C(=O)CC3=CCCC3)C2)C1 36742,Cc1cc(OC(C)C(N2CCC(NC(=O)C(C)C#N)C2)=O)cc(C(F)(F)F)c1 36743,N1(C(C2(SC)CN(C(=O)C(C3CCOCC3)O)C2)=O)CC(C#N)(CCF)C1 36744,CC(CN=[N+]=[N-])NC(C1COCC1NC(=O)CC1(C)CCC1)=O 36745,C12(C(N(C)OCc3ccccc3)=O)CC(C)(CN1C(c1cnn[nH]1)=O)C2 36746,Cc1ccc(CN2CCCC2CNC(c2cc(F)cc(Cl)c2)=O)c(F)c1 36747,c1(OC)ccc(NC(C2CC3(CC3)CN2Cc2ccnc(F)c2)=O)c([N+](=O)[O-])c1 36748,C1(CNC(CCC#CC)=O)CN(C)CCN1C(C1CC1Cc1ccccc1)=O 36749,C1(CC)CN(C(c2cc[nH]n2)=O)CCC1NC(=O)Cc1ccccc1Cl 36750,CC(C)(CCCO)C(=O)NCCCCC(C)NC(c1c[nH]nc1[N+](=O)[O-])=O 36751,C(=O)(C(CNC(C1(C)CCSCC1)=O)CC=C)NCCOCCC=C 36752,Cc1nc(Cl)c(C)c(=NCC2CCCC2NC(c2cc(=O)cc[nH]2)=O)[nH]1 36753,c1(CN2CC(C)(C(=O)NC(c3ccc(Br)s3)C)C2)ccc(N2CCOCC2)cc1O 36754,N1(C(CN(CCC(F)(F)F)C)=O)CC(NC(C2CCSCC2)=O)CC12CCOC2 36755,C1(C(N2CC(O)(CCNC(=O)COCC(F)(F)F)C2)=O)CCC(C2CCC2)CC1 36756,N1(C(C(=O)OC)=O)CCC(C(F)CNC(=O)Cc2ccc(C(F)(F)F)cc2)CC1 36757,C(=O)(CC(C)c1ccco1)N(CCCN(C(=O)CC#N)C)C 36758,C=Cn1nccc1C(=O)NCC1CCC1NC(C1(C(N)=O)CC1)=O 36759,C1(N(C(C(c2ccccc2)C)=O)C)CCCCN(C(c2ccncc2F)=O)C1 36760,Nc1cc(=O)[nH]c2cc(C(N3CCC(CS(=O)(=O)F)CC3)=O)nn12 36761,C1(OC)CCC(CC(=O)NC2CCN(C(c3ccn(C)c3)=O)C2C(C)C)CC1 36762,c1(C(N2CCOC(C3CCCC3)(C3CC3)C2)=O)ccc(S(=O)(=O)C(F)F)cc1 36763,c1(C(N2CC(NC(c3nccc(OC)c3)=O)C(OC)C2)=O)cnc(N)c(Cl)c1 36764,N1(C(c2c(CCCC)ocn2)=O)CCN(C(=O)Cc2ccns2)CC1CO 36765,C(C(C)(C)C(=O)N1CCCC1CC1CN(C(N)=O)C1)NC(=O)OC(C)(C)C 36766,Cc1c(C(=O)NC(C2CCCN2C(=O)Cc2cn(C)nc2Cl)C)sc2nccn12 36767,c1(C(N2C(COC)CN(C(c3nc(Cl)sc3C)=O)CC2)=O)cc(C)cc(C)c1O 36768,O(C=CC(=O)N1CCCC1CN(C(=O)CC1CCC(=O)N1)C1CC1)CC 36769,c1(C(=O)NC(C2(O)CCCCC2)C(=O)NCC(CC)CCO)ccc(C#N)cc1C 36770,C(=O)(CC1CCC(C)(C)c2ccccc21)NCCCNC(C(COC)O)=O 36771,CN=c1[nH]ccc(C(N2CC3CCCCC3(CNC(=O)C3CC3)C2)=O)c1[N+](=O)[O-] 36772,c1(SC)ncc(C#N)c(N2CCCC(C(N3CCCC(CO)C3)=O)C2)n1 36773,c1(OC)ccc(C)c(C(C)NC2CCCCCN2C(=O)OC(C)(C)C)c1 36774,c1(CC)n[nH]cc1C(=O)NCC(N1CCC(C(=O)NCCOC)C1)=O 36775,C(CC(C)C)(C(=O)NC1CC(CCC(N)=O)C1)ONC(CSCC=C)=O 36776,C=CCC(C(=O)N(C(C)C(F)F)C)NC(C)=O.C1(=O)C(C)N1 36777,N1(C(=O)CC2C=CCC2)CC2(CCN2C(c2cc(-c3ccncc3)on2)=O)C1 36778,C1(CC(N2CC(CNC(Cc3cccc(SC)c3)=O)C2)=O)CCC2(CCC2)CO1 36779,CCCC(CCNC(=O)C(C)(C1CC1)N(C(=O)COCCF)C)C1CC1 36780,Cc1cc(O)ccc1C(=O)NCC1CCCN(C(=O)CC2CCCS2(=O)=O)CC1 36781,Cc1nn(C2CCOCC2)c(C)c1CNC(c1ccnc(Br)c1N)=O 36782,CC(CC(F)F)C(=O)NCC(O)C(=O)NC1CCCCCC1CO 36783,N1(C(C2CC(=O)NC(=O)N2)=O)CCC(CNC(=O)Cn2cc(Cl)cn2)C(F)(F)C1 36784,c1(CNC(C2C(CNC(=O)CC3CCCOC3)CCC2)=O)ccnc(O)c1 36785,Cc1nc(C2CCC2)sc1CC(=O)NC1(C)CCN(C(=O)C(C)NCCC(C)C)C1 36786,C1(C(=O)NC2C(NC(c3ccc(C(=O)OC)cn3)=O)C2)CCc2nc[nH]c2C1 36787,N1(C(CC2CC(=O)N2)=O)CC2(C1)CN(C(=O)COc1cc(Cl)ccn1)C2 36788,N1(C(c2nc(C(C)C)sc2)=O)CCN(C(=O)C(c2cnn(C)c2)C)C(CO)C1 36789,c1(-n2c(C(C(C(C)C)OC)NCCCCSC)nnn2)ccc(F)cc1 36790,CC1(CO)CC2(CCN2C(C2CNC(=O)CN2C(c2cc[nH]n2)=O)=O)C1 36791,C1(NC(c2nc(CC)oc2)=O)CC2CC1N(C(C1CCC(F)(F)CC1)=O)C2 36792,N1(C(C2(C)CC(=O)C2)=O)CCC(C)(C)C(CNC(c2c(F)cccc2F)=O)C1 36793,N1(C(C(CCNC(CC(CC)C2CCC2)=O)O)=O)CC2CCC(C1)O2 36794,N1(CCC)CCN(S(=O)(=O)N(C)C)CC1.c1(C2CNC(=O)N2)c(F)cccc1F 36795,N1(C(C2C(C(N(CC#C)C)=O)C2)=O)CC=C(CCNC(=O)CC2CCOC2)CC1 36796,c1(CC(=O)NC2CCCCCC2NC(=O)CC(F)(F)F)cccc2c1OCCC2 36797,C1(C(N(C)CC2CCN(C(=O)Cc3nccn3C)C2)=O)CCC(C)(C)CC1 36798,C1(CCC)CCN(C(=O)Cn2cc(CCN3CCCCC3)nn2)C1 36799,CC(C)CC(C)CC(=O)NC(C)CCN(C)C(c1nncn1C1CC1)=O 36800,N1(C(c2c(C)nc(CC)s2)=O)CC2(CCCCN(C(C3CN(C)C3)=O)C2)C1 36801,C1(C)(NC(c2c(C)n[nH]c2)=O)CCCN(C(=O)C(C)Oc2cccc(C#N)c2)C1 36802,c1(N(CC(C)(C)C(C)(F)F)C)ccc(S(=O)(=O)NCC2CCN(C)C2)cn1 36803,N1(c2nccc(C(=O)OC)n2)CCC2(NC(c3cn(C)nc3SC)=O)CCCC12 36804,c12cc(Cl)ccc1NC2(c1nnnn1C1CCOCC1)C.C1(C(C)C)CC1(Cl)Cl 36805,c1(-c2nc(C)c(C(=O)Nc3cc(F)c(Cl)cc3F)cc2)ccc2c(C)[nH]nc2c1 36806,c1(OC)cc(SC)ccc1CNC(Cc1sccc1Br)C(=O)O 36807,C1(N(C(C(C)NC(COC)=O)=O)C)CCC(NC(c2ccn(C)n2)=O)CC1 36808,C1(NCCCCN(C(Cn2cc(C(C)=O)nn2)=O)C2CC2)C=CCCCC1 36809,C1(NC(CSCC=C)=O)CC(OC)CN(C(=O)CCc2cc(C)nc(C)c2)C1 36810,c1(C(N2CCCC(F)(CNC(C3(Cl)C(C)(C)C3)=O)C2)=O)n[nH]c2cc(Cl)ccc12 36811,N1(C(CCCCCOC)=O)CC2CCCN(C(=O)CCC(C)(C)C)C(C2)C1 36812,C1(NC(c2cccc(C)n2)=O)CC2CC1N(C(=O)C(F)(F)CCn1ccnn1)C2 36813,C(=O)(C1=CCCSC1)NC1CCC(CNC(C2CCN(C(N(C)C)=O)CC2)=O)C1 36814,C1(C(=O)NCCC(=O)OC)CCC(C(C(=O)OC)N(C)C(c2csc(=N)[nH]2)=O)O1 36815,C(=O)(C1CCCc2ncccc21)N1C2CC(CN(C(C(CC)OC)=O)C2)C1 36816,c1(OCC)ncc(NC(=O)CC2CCCN(C(=O)C(C)C(C)C)C2)cn1 36817,CC(C)CC(F)(F)C(=O)NC1CN(C(c2c(Cl)nn(C)c2Cl)=O)CC2(CC2)C1 36818,C(=O)(CC(C)CC(=O)N(CCC(C)NC(c1ncc2ccccn12)=O)C)OC 36819,N1(C(C2CC(SC)C2)=O)CCCC(NC(c2ccn(C)c2C2CCC2)=O)C1C 36820,N1(C(c2cncs2)=O)CCCC(F)(C(N2CCCCC2CCCO)=O)C1 36821,c1(C(N2CCC(N(C(c3c[nH]nc3SC)=O)CC)C2)=O)cn2ccc(C)cc2n1 36822,C1(C(=O)NC2C(CNC(C3CC(OCC)C3)=O)C2)CC(O)(C(F)(F)F)C1 36823,C1(C(=O)NC(c2nccs2)C)CCCC12CCN(C(c1ccc[nH]1)=O)C2 36824,c1(C(=O)NC2(C)CCCN(C(=O)C3=CCSC3)C2)nc(Br)c2n1CCCC2 36825,N1(C(C)=O)CCN(C(C2COC(=O)N2C)=O)C(c2cccc(Cl)c2)C1 36826,Cc1ccc(C(=O)NC2CC(CNC(=O)C(O)CN(C)C)C2)c(C)c1Br 36827,c1(C(N2C(CNC(C=CC=CC)=O)CCC(C)C2)=O)ccc(OC)c(F)c1N 36828,C(=O)(C(F)CC1CN(C(C2CC2c2ccccc2)=O)C1)N(C(C)C)C1CC1 36829,C12(CNC(=O)COc3ccon3)COCCN1C(=O)CN(C(C1CCOC1)=O)C2 36830,c1(C(N2CC(O)(CN(C)C(c3cccn3C)=O)C2)=O)cccc(F)c1F 36831,CC1CN(C(=O)C(c2ccccc2)=O)CCC1NC(c1ccnc(C2CC2)n1)=O 36832,N1(C(C(C)C)=O)CCC=CC1C(=O)NOCC1CC1c1ccnn1C 36833,C1(NC(CCC#C)=O)CC2CC1CN(C(c1cc(C(F)F)no1)=O)C2 36834,c1(NC(C2(NC(CCOCC)=O)CCCC2C)=O)c(C)ccn(C)c1=O 36835,c1(C(=O)NC2CCCC(F)C2)cc2oc(Br)cc2s1 36836,CCC(C)CC(=O)N1CCC(O)(CNC(=O)CCN(C2CCCCC2)C)C1 36837,c1(CSC)cc(Br)ccc1CNC(C1CC(F)CN1C(=O)CCc1cnn(C)c1)=O 36838,c1(CCCC(=O)NCC(CC=C)NC(C2(COC(C)C)CC2)=O)ccc(O)cc1 36839,c1(C(N2CC(CC(C)NC(C3CC(=C)C3)=O)C2)=O)cc2sccc2s1 36840,N1(C(C(CC)N(C)CC)=O)CC2(CC(C(=O)NOC3CCCCC3)CO2)C1 36841,S(=O)(=O)(c1cnc(NCC2(Br)CC2)c(Cl)c1)N1CCCC(C(C)O)C1 36842,CC1(C)CN(C(C2CCN(C(C3CC(O)C3)=O)C2)=O)CC1O 36843,C(C(=O)NC(C)(CNC(=O)C=Cc1cn[nH]c1)CO)(C(C)(C)C)SC 36844,c1(C(=O)NC)ncc(NC(=O)C(C(C)C)NC(=O)CC(C)COC)cn1 36845,C12(C(=O)NCCC3N(C)CCC3)C(NC(C3CC4C=CC3C4)=O)C3CC1C2C3 36846,c1(CC(=O)NC2(C)N(Cc3nnc(C)o3)CC2)cccc(OC(F)(F)F)c1 36847,C1(CNC(Cc2cc(OC)ncc2)=O)CCN(C(C2CC=C(C)CC2)=O)C12CC2 36848,C12(CC)CCC(C(=O)NC3CCC(NC(C4(C)CC(F)C4)=O)C3)(CC1)CO2 36849,N(C(=NCC1CCC1)N1Cc2ccccc2C(F)(F)C1)Cc1c(OC)ccnc1 36850,N1(C(c2c(N)ncc(C)c2)=O)CC2CC3CC2C1C3NC(=O)CC1(CO)CC1 36851,c1(C(C(=O)NCCCC(C)NC(CCCCC)=O)(F)F)ccccc1C#N 36852,CC1CN(C(=O)C(C)(C)C2CCN(C(C3CC(F)CN3C)=O)C2)CC1O 36853,c1(NC(C2CCCN(C(C34CC(C)(CO3)C4)=O)C2)C)ncc(C#N)cc1F 36854,N1(C(CC2N(C(Cc3cn(CC)nc3)=O)CCC2)=O)CC2(CCC2)C1 36855,C(C(C)(C)C#CC(=O)NCC(O)CC(F)(F)F)NC(C(C1CCCCCC1)C)=O 36856,C1(C(N(C)CCOCCCO)=O)CCN(C(C2(N(C)C)CCCCC2)=O)CC1(C)C 36857,C1(NC(C(CNC(C2(CC#C)CCCO2)=O)C)=O)CCC(C#N)CC1 36858,Cc1c[nH]nc1C(=O)N(CCCNC(=O)C(Cc1ccccc1)N(C)C)C 36859,C1(OCC)CN(C(c2nccc(C)n2)=O)CC1CNC(c1ccc(CF)cc1)=O 36860,C(CCCC(=O)NCCC1(C)CCN(C(c2ccc(C(C)C)s2)=O)C1)(OC)OC 36861,N1(C(C(CC)SC)=O)CCSCC1CNC(=O)C(O)c1ccco1 36862,C(=O)(C1CCC(=O)c2ccccc21)N1CCCC(NC(CNC(CC)=O)=O)C1 36863,c1(CC(=O)NC2CN(C(C(C)C)=O)CC23CCC3)nn(C)c2ccccc12 36864,c1(C(=O)NCC2(C)OCCN(C(C3CN(C(C)=O)C3)=O)C2)cc2ncccc2[nH]1 36865,c1(SC)cc(C(=O)NCCCCCN(C(=O)C(C2CCCOC2)OC)C)co1 36866,c1(C(C(=O)NCCC(C)(C)NC(Cc2nnc(C)s2)=O)N(C)C)cccc(Cl)c1 36867,C1(OC)CC(NC(c2cc(C)nc(O)c2)=O)CN(C(=O)C(C)Cc2cnc[nH]2)C1 36868,C(=O)(CC(O)C(C)C)NC1C(NC(C(CC#C)C)=O)CCCC1 36869,N1(C(Cc2cn(CC)nn2)=O)CC(CCNC(=O)CCc2cncnc2)C(C)C1 36870,N1(C(C2(OC)CCSC2)=O)C2CCC(C2)C1CNC(c1cc(C)c(C)[nH]1)=O 36871,C(=O)(CC(F)(F)F)NCCC1(OC)CN(C(C2CCC(C)C2)=O)C1.C(C)(=O)O 36872,c1(C(c2n(CCCC)nnn2)Nc2cnccc2CO)ccc2nc(C)oc2c1 36873,Cc1c(N)cc(C(=O)NCC(C)NC(=O)C(c2cccc(Cl)c2)O)cc1[N+](=O)[O-] 36874,c1(C(=O)NC2(CO)CCCN(CC3(SC)CC3)C2)cc(C2CC2)nc2ccnn12 36875,C1(N(C)C)CN(C(C23CC2CCN3C(C2COC(=O)N2C)=O)=O)CC1(C)C 36876,N1(C(C(CNC(C2C=C(C)CS2)=O)OC)=O)CCOC(C)(C)C1C 36877,c1(CNC(CSCC)=O)ncoc1C1CN(C(C2CC2(F)Cl)=O)C1 36878,Cc1cc(O)ccc1CN1CCCC1CCC(=O)NCCC#N 36879,c1(C(=O)NC2C3(CC(NC(c4c(C)cc(Br)o4)=O)C3)C2)cc[nH]c2nccc1-2 36880,C(=O)(CCC(=O)NC(C1CCOC1)CNC(=O)Cc1csc(Br)n1)NC 36881,c1(CC(N2CCC(C(C)NC(=O)C(N)=O)C2)=O)cccc2ncccc12 36882,C(=O)(C(C)(C)CCCNC(=O)C(c1cnn(C)c1)C)N1C(CC)CCOCC1 36883,C(C(C)(Cn1cccn1)NC(C1(C(C)C)CC1C(=O)NCc1c[nH]nc1C)=O)OC 36884,c1(C(N2CCC(NC(C(CCSC)OC)=O)C(F)C2)=O)cc2oc(C)c(C)c2[nH]1 36885,c1(CNC(C(C)n2cnnn2)=O)cccc(C(=O)NCCC#CCO)c1 36886,CC1CCN(C(=O)C(C2(O)CCC2)NC(=O)COCCCN=[N+]=[N-])CC(C)O1 36887,CCCC(C)(C)C(=O)N1CC2C(CC(N3CC(=O)NCC3C)=O)C2C1 36888,N1(C(c2nncc(OC)c2)=O)CC(F)(F)CC1(C)CNC(c1ccc(Cl)cn1)=O 36889,CC1(C2CC2)NC(=O)N(CC(N2CC(NC(=O)Cn3nccn3)C3CC23)=O)C1=O 36890,c1(C(C(=O)NCCC2(C)CC2)N(C)Cc2cnc(CC)s2)ccc(C)cc1Cl 36891,C1(C)(CC)C=C(C(=O)N2CCOC(CC(=O)NCCOCC(C)(C)O)C2)C1 36892,C(=O)(C(CO)C(C)C)NCC(C(C)C)Nc1ncc(Br)cn1 36893,C(=O)(C1CCc2c[nH]nc21)N1CCCC(NC(=O)Cn2ncc(O)nc2=O)C1 36894,c1(C(=O)NC2CCCN(C(CC3(CSC)CC3)=O)C2)cc2cc(F)cc(F)c2[nH]1 36895,C1(=CC(=O)NC2(CC=C)CN(C(c3ccc(CO)o3)=O)C2)CCC(C)CC1.C(CSC)N 36896,C1(O)(CC#C)CC(C(=O)NC(C)C(=O)NCC(c2ccccc2)F)C1 36897,C1(O)(CN(C(C(C)CF)=O)C)CCN(C(C2CCCC2C(F)F)=O)CC1 36898,CC(=O)C(C)(C)CC(=O)N1CC=CC(C(=O)NCC=CCCOC)C1 36899,CCC(C)CCN=c1[nH]c(=NCC2(CO)CC3CCC2CC3)c2ncccc2[nH]1 36900,CC1(C(=O)NCC2CCCC(NC(=O)C(=O)NCC(F)(F)F)C2)CCC2CC2C1 36901,c1(CNC(c2c(C)cno2)=O)cccc2c1CCN(c1cc(O)nc(O)n1)C2 36902,c1(C(=O)NC2(C(=O)NCC3(COC)CCC3)CC2)ccc(OC)nc1OC 36903,C(=O)(C1=COCCC1)N(CCNC(CS(CC)=O)=O)CCc1ccccc1 36904,C1(C(=O)NCCC2C(C(=O)OC)C2)CN(C(C2COCCC2C)=O)CC1F 36905,Cc1cc(C2(C(=O)NC3CCCN(C(C4CC(C#N)C4)=O)C3)CCC2)cc(C)c1 36906,Cc1ccnc(NCCCCNC(=O)C(C)NC(c2ccoc2)=O)n1 36907,c1(NC(c2nc(NC(Cc3ccc(C)s3)=O)sc2)=O)cnc(N(C)C)nc1 36908,N1(C(C(C)(C)NCC)=O)CCCC(O)(CN(C(=O)C(C(C)C)NS(C)(=O)=O)C)C1 36909,N1(C(CCCCC(N)=O)=O)CC(NC(c2cccnc2)=O)CC12CCCOC2 36910,C(CN=C(NCc1cccc2c1OC(F)(F)O2)N1CC(O)C(C)(C)C1)SC 36911,c1(C(=O)NC(CNC(C2(OCC)CCC2)=O)C2CC2)scc(C)c1C 36912,CCCCC(O)C(=O)N1CCCCC1CN(C)C(C1(CC)CCCCCC1)=O 36913,Cn1cc(C(N2CCCCC2CNC(C2(Cl)CC=CC2)=O)=O)ccc1=O 36914,C(=O)(C#CC1(C)CCCO1)N(CCC(=O)NCC(CC)C(C)C)C(C)C 36915,c1(C(=O)NC2CC(C)(CNC(C3N(C)C(=O)CC3)=O)C2)cn(C)c(=O)nc1O 36916,c1(CN(CC(C)(C)C(=O)N(C2CCCCC2)C)C)cc(OC)c(OC)c(OC)c1 36917,C1(O)(C(C)C)CCN(C(=O)C=CC(C)NC(C2CCCC2O)=O)C1 36918,N1(C(c2ccn(CCCC)n2)=O)CCC2(NC(=O)C=CC3CC3)CCCCC12 36919,c1(C(=O)NC(C2CC(NC(=O)CC3CCOC3)C2)C)ccc(F)c(CO)c1 36920,C1(NC(=O)N(C)C)CCC2(C1)CN(C(=O)Nc1oc3ccc(C)cc3c1)C2 36921,c1(N(CC(C(=O)NC2CCC2)NC(=O)C(O)CN2CCCC2)C)ccc(Cl)cc1Cl 36922,C=CCC(CC=C)C(=O)N1CCC(C(=O)N(CCCCC)C)(CC)C1 36923,C1(NC(C(C)(C)OC)=O)CCC(C)C(C)C1 36924,c1(C(=O)NCC2(C(F)F)CCN(C(c3onc(C)n3)=O)C2)cnc2c[nH]nc2c1 36925,N1(C(CC2(CC=C)CCCC2)=O)CC(NC(=O)CCCF)CC(F)C1 36926,Cc1c(NC2(CCN(C)C)CC2)ncnc1N1CCC(Oc2ccc(F)cc2)CC1 36927,n1(CCC(=O)NCCCCCN(C(=O)CC2CC23CC3)C)ccc(O)nc1=O 36928,c1(C(=O)NCC2N(C(CC=CC=C)=O)CCC2)cncc(F)c1C 36929,c1(C(N(C2CCC(NC(=O)C=CCN(C)C)C2)C)=O)ccc(OC(F)F)nc1Cl 36930,CCCC(C)(CC)C(=O)NC1CC(CCNC(C23CCCC2C3(F)F)=O)C1 36931,C1(NC(c2c(OC)ccs2)=O)C(C)(C)C(NC(C2CCNC(=O)C2)=O)C1(C)C 36932,C1(NC(CCCCCC)=O)CC2CN(C(=O)C(=Cc3cccs3)C)CCN2C1=O 36933,CCC(CC)C(C)C(=O)NCC1CCN1C(=O)CCCOc1ccc(F)c(F)c1 36934,c1(-c2nc(C(C)Nc3cc(S(C)(=O)=O)co3)[nH]n2)ccc2ccccc2c1 36935,c1(CC(=O)NCCC2C(C)CCCC2)cc(Br)ccc1Cl 36936,Cc1cc(C(=O)NCCCCC(C)NC(=O)CCC2(C)CC2)cc(N)c1 36937,N1(C(CNS(C)(=O)=O)=O)CCC(C2N(C(=O)CO)CC2(C)C)CC1 36938,c1(CNC(C2CCN2C(=O)OC(C)(C)C)C)ncc(Cl)cc1Cl 36939,c1(OC)c(C(=O)NCCC(C)N(C)C(C2CC(SC)C2)=O)cc(Cl)cc1Cl 36940,N1(C(c2cnc(CC)[nH]2)=O)CCC2CCCN(C(c3cn(C)nc3CC)=O)C2C1 36941,C1(NC(C=NOC)=O)C2CCN(C(=O)C(C)Cc3cccnc3)CC12 36942,C1(C(=O)NCC2N(C(c3nc(C)sc3)=O)CCCC2)CC2CC1C1C2C1(F)F 36943,c1(NC(C(C2CCCCC2)NC(CC(=O)OC)=O)C)ncc([N+](=O)[O-])cc1C#N 36944,c1(C(C)C)cc(C(=O)NCC2CN(C(=O)CCSC(F)(F)F)C3CC23)ccc1F 36945,c1(C(N2C(CNC(c3c(CC)ncs3)=O)C=CC2)=O)cc2n(n1)CCC2 36946,c1(OC)ccc(Br)c(C(N2CCCC(O)(CNC(=O)C(C)SC)C2)=O)c1 36947,c1(C(=O)OC)ccc(C(=O)NCc2nnc(O)n2C2CC2)n1C 36948,C1(OCC)CC(NC(=NCCF)NCC(c2ccc(F)c(Cl)c2)(C)C)C12CCC2 36949,C1(CCC=C)(C(=O)NC(C)C(C2CC2)OC)CCCC1.C1(C)C(=O)N1 36950,c1(C(=O)NC(C2CCOC2)CC)ccc(Cn2cc(C(N3CCCC3)C)nn2)o1 36951,c1(C2C(n3c(-c4c(-c5n(CC)ccn5)n[nH]c4)ncc3)C2)ccccc1OC 36952,c1(CS(N2C(c3onc(-c4nccc(C)c4)n3)CCC2)(=O)=O)cc(Cl)ccc1Cl 36953,C1(NC(C(F)=C(C)C)=O)CCCC(NC(c2cc(Cl)n(C)n2)=O)C1 36954,c1(C(N2CC(C)N(c3nc4ccccc4o3)CC2)=O)cccn2ncnc12 36955,CC1CCC(O)(C(=O)NC2CCCN(C(=O)C(C)CN(C)C)C2C)CC1 36956,C1(C2CCN(C(=O)CCC3OCCO3)C2)(NC(c2c(CC)ccc(F)c2)=O)CC1 36957,c1(SCC)c(C)nn(C)c1N.C1(C)(N(C)C)CCN(C(C2CC(O)(C(=O)N)C2)=O)C1 36958,CC(C)C(CC(=O)N1CCC(O)CC1)NC(c1cocn1)=O 36959,CCC(CC(=O)NC(C(=O)NCC1(CC)CCCO1)C(C)OC)OC 36960,CC(C)C1=NOC(C(=O)NCC2CC3CCC2N3C(C23CC(C)(CCO2)C3)=O)C1 36961,CCC(C)C(O)C(=O)N1CCCN(C(c2[nH]c(-c3cccnc3)nc2C)=O)CC1 36962,c1(C(=O)NC2C(CNC(C(C)NC=O)=O)C2)ncc(F)cn1 36963,c1(N2CCCCC(CC)C2)cc(S(=O)(=O)N2CCCC(C(C)C)C2)ccc1C#N 36964,N1(C(CC2CC(C)OC2C)=O)CCCCC2(CCN(C(C3COC(=O)N3)=O)C2)C1 36965,CC1(C)CCCCCC1NCC1CCCNC1 36966,Cc1ccc(I)c(C(=O)NC2CN(C(=O)Cc3ccc(F)cc3F)CC23CC3)c1 36967,C1(NC(C2C(C(C)C)CN(C(=O)CC3CSCCO3)C2)=O)CCNC(=O)CC1 36968,CP(C)(=O)C(O)C(=O)NCCC1CN(C(=O)CCC2CC2(F)F)C1 36969,CC1CN(C(C2CC2C(C)(F)F)=O)CC1(C)C(N1CCC1c1ccccc1)=O 36970,C(C(C(=O)NOCc1ccc(F)cc1)C(C)(C)C)NC(C(CCC)C#N)=O 36971,N1(C(c2cc(OC)n[nH]2)=O)CC(CNC(=O)C(N2CCSCC2)C)C2(CC2)C1 36972,C1(C(=O)NCCCCN2CCOC2=O)Cc2ccc(Br)cc2N1 36973,c1(N2CC3CN(C(Cc4cc(C)cc(C)c4)=O)CC3C2)nc2ccc(Cl)cc2s1 36974,C=C(C)C(CC(=O)NCC1CCC1NC(=O)Cc1ccc(F)cc1F)OOCC 36975,C1(NC(c2n[nH]c(O)n2)=O)CCN(C(C2CCCC(F)(F)CC2)=O)CC12CCC2 36976,C1(C(=O)NCC=CCCC)(CF)CCN(C(=O)CCC=C(C)C)C1 36977,c1(C(N2CC(F)CC(NC(C3(C)N(C)CCC3)=O)C2)=O)cc2ccccn2n1 36978,CC(C)CC1CC1C(=O)NCCCOCCCNC(=O)CSC(F)F 36979,C1(CC(=O)NCCOC2CCN(C(C(C)(C)CC3CC3)=O)C2)CCCCC(=O)N1 36980,Cc1nn[nH]c1C(N1CCCC1CCNC(=O)CC1(CS(C)(=O)=O)CC1)=O 36981,c1(C(N2CC(CC)(NC(=O)Cc3c(C)cccc3Cl)C2)=O)cn2cnnc2cn1 36982,C12(NC(=O)NCC(COC(C)(C)C)O)CC3CC(C1)CC(CC(F)(F)F)(C3)C2 36983,c1(OC)c(C(=O)NCC2CCCN(C(=O)C(C)S(N)(=O)=O)C2)ccc(Cl)c1C 36984,N1(C(C2N(C(C(C)NC=O)=O)CC(F)C2)=O)CCOC(C)(C)C1 36985,c1(C(N2CC(CC(C)NC(c3ccncn3)=O)C2)=O)cc(N)cc(O)n1 36986,C1(NC(C(C)N(CC)CC)=O)CC2CC(C1)CN(C(c1ncccc1OC)=O)C2 36987,C(=O)(C(C)(C)CC(=O)OC)NCC1COCCN(C(c2c(CCC)[nH]cc2)=O)C1 36988,N1(C(CC(CC)CN(C)C)=O)CC2CCCC(C1)N2C(=O)C1=NOCC1 36989,N1(C(C=CC=CC)=O)C2CCC1(CNC(=O)CCCN1CCCC1)CC2 36990,c1(NC(=O)NC(C)(CCCC2CC(OCC)C2)Cn2cccn2)cnccc1C 36991,CC(C)CC(CNC(C1(C(F)(F)F)CC(F)(F)C1)=O)NC(c1ccccn1)=O 36992,C1(SC)CCCN(C(=O)CC2CC(NC(=O)C(C(C)O)NC(C)=O)C2)C1 36993,C1(NC(c2c(OC)cnc(Br)c2)=O)CC2(CCN(C(=O)Cc3ccno3)CC2)C1 36994,N1(C(CS(=O)(=O)N(C)C)=O)CC(NC(=O)Cc2ccc(O)cn2)CC12CCC2 36995,c1(C(N2CCC(Br)C2)=O)cnn2c1CN(Cc1ccc(F)cn1)CC2 36996,C1(C(N2CC(OCCNC(c3c(C(C)C)c[nH]c3)=O)C2)=O)CC(=O)NC(C)C1 36997,c1(CC(C)CN2CCCC2)cc(C(=O)O)cc(Cl)c1 36998,CC1CN(C(C2CN(C(C3(Cc4ccccc4)COC3)=O)C2)=O)CC1 36999,Cc1cc(F)ncc1NC(=O)NCC(C1CC1)N(C1CCOCC1)C 37000,N1(C(c2cc(COC)[nH]n2)=O)CC2CCC(C1)C2NC(c1cc(COC)cs1)=O 37001,c1(C(N2CCC(CSC)C2)=O)c(I)cnc(Cl)c1F 37002,c1(CC)cc(C(=O)NCC2(O)CC(CNC(C3(N4CCOCC4)CC3)=O)C2)on1 37003,c1(C(CC(=O)NC2CN(C(C3(C(=O)OCC)CC3)=O)CC2O)C)ccc(F)cc1F 37004,N1(C(c2c(CC)[nH]cc2)=O)CC2(C=C(C(=O)Nc3ccccc3)CO2)C1 37005,c1(-c2cc(C)ncc2)ccn2cc(C(N3CC(O)C(F)C3)=O)nc2c1 37006,N1(C(CN(C)C)=O)CC2CCCN(C(c3ccc4oc(O)nc4n3)=O)C2C1 37007,Cc1ccc(OCC(=O)NC2CCC23CN(C(=O)CCC(C)(C)C)C3)c(C)c1 37008,c1(C(=O)NCC(CNC(C(C)SCC)=O)F)cc(F)cc2nn[nH]c12 37009,Cc1cccc(C(=O)NCC(C)CN(C)C(C2CCC(C)(C)O2)=O)n1 37010,c1(C(CC)CC)cc(C(=O)NC2CC(CNC(=O)CN3CSCC3=O)C2)on1 37011,C=CC(CC)CC(=O)NCC(c1cccc(Cl)c1)N(C(=O)C(C)(C)CC)CC 37012,c1(CC)cc(C(=O)NCCC2CCC(NC(=O)Cn3cnnn3)C2)ccc1F 37013,c1(NC(CN2CCN(CC(=O)NC(CC)C)CC2)=O)c[nH]c2cc(F)c(F)cc12 37014,c1(C(=O)NC2CN(C(C3(C=C)CCCCC3)=O)CC(C)C2)cc2ncccc2o1 37015,C1(F)(c2cc(C)cc(C)c2)CCN(C(=NCC(C)C)NCC2=CCCC2)C1 37016,c1(C(=O)NC2CCC(NC(c3c(SCC)nccn3)=O)C2)cc(CC)ccc1O 37017,N1(C(C2CC23CC3)=O)CC2(C(=O)NCCSCCO)CCC1CC2 37018,c1(C(=O)OC)cccc(C(C(=O)OC)OCCC2NC(=O)NC2=O)c1 37019,c1(C(=O)NCC2COCC2NC(C2(C(F)F)CC2)=O)cn2cc[nH]c(=O)c2n1 37020,n1(CC(C2CCC(=O)N2)C)cc(CCN2CCOCC2)nn1 37021,C(=O)(C1=CCCOCC1)NC1CC(C)N(C(=O)CC(C)n2cccc2)CC1 37022,c1(C(=O)NCC(=O)NC2C(CNC(=O)CCn3cncn3)C2)ccc(Cl)cc1Cl 37023,c1(C(N2C(C(=O)NCCN(OC)C)CCC2C(C)C)=O)ncc(C)cc1F 37024,c1(NC(C2CC3CCCCC3N2C(c2ccoc2)=O)=O)ccc2nc(O)[nH]c2c1 37025,c1(C(N(CCC)CCNC(c2cnn(C)n2)=O)=O)ccccc1-n1cncn1 37026,N1(C(C2N(C(C)=O)CSC2)=O)CCCCCC(NC(c2csc3cncn23)=O)C1 37027,c1(C(=O)NC2CCN(C(C3CC(CC)(CC)C3)=O)C2)cc(C)c(Cl)cc1OC 37028,N1(C(C2CC(C(C)C)C2)=O)CCCC(C)C1CCNC(=O)CCC1CC(F)(F)C1 37029,C(=O)(CCCN=[N+]=[N-])NC1C(NC(c2nn(C(CC)C)c(C)c2)=O)COCC1 37030,N1(C(c2c(CC)non2)=O)CCC(CN(C(=O)CC2(COC)CC2)C)CC1 37031,c1(N2CCC3(CC(OC)C3)C2)nc(=NC(C)c2cc(C)oc2C)[nH]c2c1CCC2 37032,N1(C(C(CC)O)=O)CC2CCCC(CNC(c3cc(O)cc(=O)o3)=O)(C2)C1 37033,c1(C(C)=O)ccc(C)c(Cc2nc(C(F)(F)F)n3c2CC3)c1 37034,C1(NC(c2ccn(CC)n2)=O)CC2(C1)CC2NC(=O)CCc1ccc(C(F)F)o1 37035,c1(C(=O)NCCC2CC(NC(c3cn(CCO)nn3)=O)C2)cc(Cl)ccc1O 37036,C1(CC=C)(NC(C2CC3CC3C2)=O)CCCN(C(C2CC(=O)N(C3CC3)C2)=O)C1 37037,C1(C(NOCC=CC)=O)CCCN(C(=O)CCC2CC2)CC1 37038,c1(CC(C(=O)NC2CCC(NC(CCSCCC)=O)CC2)C)ccc(F)c(F)c1 37039,CCCCC(C)C(=O)N1CCN(C(=O)CCCOCC(C)C)CC1c1cn[nH]c1 37040,C1(C)(CCNC(c2n(CCCOC)nnn2)C(C)(C)OC(C)C)CCOCC1 37041,C(C(C)(C)CNC(c1nocc1Br)=O)N(C)C(C1C=CCCC1)=O 37042,C1(N(C(C(C2CC(C)(C)C2)OC)=O)C)C2CN(C(=O)CC(C)(F)F)CC12 37043,C(=O)(C1=CC2C=CC(C1)C2)NC(CC)CC(=O)NOC(CO)C(C)C 37044,c1(CCCNC(=O)NC(CCCCCC)C)ccccc1[N+](=O)[O-] 37045,c1(CNC(CC(C)n2cccn2)=O)ccccc1CNC(C1C(F)(F)C12CC2)=O 37046,C(=O)(C1=CS(=O)CCC1)N1C(CNC(C=Cc2c(C)ccs2)=O)CC(F)C1 37047,c1(OC)nccc(C)c1SCCCOC(=O)CC(O)C(=O)c1ccccc1 37048,c1(N(CC(=O)NCC(CCCC)NC(=O)CC(F)(F)F)C)ncnc2[nH]cnc12 37049,Cc1ccc2oc(C(=O)NC3CN(C(=O)CCNC(=O)CO)C4CC34)cc2n1 37050,C(=O)(C(=O)C(C)(C)C)NCc1c(NC(CC2(OC)CCOCC2)=O)cccc1 37051,CC(C)CC(C)(CNC(=O)CC1CCC2CC12)NC(c1cnc2n1CCC2)=O 37052,C1(CN(C(C(CC)C)=O)CCOC)CCCCN1C(=O)C=Cc1ncc[nH]1 37053,c1(NC(N)=O)cc(Br)cnc1N1CCCC(Cc2ccc(Cl)cc2)C1 37054,CCC(C)(C(=O)NC(CNC(=O)C=Cc1cccc(F)c1F)C(C)C)C(F)F 37055,C(=O)(C(CC)C(C)O)NCC(=C)CCNC(c1cnc(CC(C)C)s1)=O 37056,c1(C(N2CCOCC2C)C(=O)NC)ccc(Oc2ccc(C3CC3)cn2)cc1 37057,N12CCC3CC13C2=O.C12(Cc3nc(CN(C(=O)COCO)C)on3)CCC(CC1)C2 37058,N1(C(=O)OC(C)(C)C)C(C(=O)NCCc2ccc3nc[nH]c3c2)CC2CCCC12 37059,c1(C(=O)NCC(C2CCCN(C(=O)CCF)C2)(C)O)ccccc1F 37060,C1(NC(CCOCC)=O)CCC(CC(=O)NCCCC2CCCC2)C1 37061,C(=O)(C(O)P(C)(C)=O)N1CCC(CCNC(C(C)n2ccnc2)=O)C1 37062,C1(NC(C=CCCC)=O)CCS(=O)(=O)C12CN(C(C1CN(S(N)(=O)=O)C1)=O)C2 37063,c1(C(c2n(C(CC)(C)C)nnn2)NC2CC(=C3CC3)C2)nc(C)c(C)n1C 37064,c1(CCC(=O)NCC2C(C(=O)NC3C(CCOC)C3)CC2)nc(C(C)C)no1 37065,C1(c2nnnn2C2CC2)(NCCn2cc(C(F)(F)F)nn2)CN2CCCCC2C1 37066,CCC(C(=O)NC1CC1NC(=O)CCc1sccc1Br)c1ccccc1 37067,Cc1cnc(C(=O)N(C)CC2CCCN(C(C3CC3C)=O)C2)cc1C 37068,c1(OC)ccc([N+](=O)[O-])cc1C(N1CCC12CN(c1ncccn1)C2)=O 37069,c1(C(=O)NC2C(NC(C(CC)n3ccnc3)=O)C2)ccccc1C(C)=O 37070,N1(C(C(C)=C(C)C)=O)CC(C)OC2(CCN(c3ncc([N+](=O)[O-])cc3Br)C2)C1 37071,CCCCC(C(=O)NC1CCN(C(C2CCCCS2)=O)C1C(C)C)N(C)C 37072,N1(C(C(C)SC(F)(F)F)=O)CC(CO)C2(C1)CN(c1ncnc3c1cnn3C)C2 37073,C1(CNC(C2CN(CC)C(=O)C2)=O)C(C)CCCN1C(=O)Cc1cc(C)no1 37074,c1(O)ncc(F)c(NC2CC3CC(C2)N3C(=O)COCC(C)(C)C)n1.C(=O)(CC)OC 37075,C1(NC(C2(CC#C)CC=CCC2)=O)CN(C(c2ccco2)=O)CC1S(C)(=O)=O 37076,c1(SCC(N2CC(C(C)NC(=O)CCOC3CCCCC3)C2)=O)n[nH]c(O)n1 37077,Cn1nc(C(=O)O)c(C(=O)O)c1Cl.C12CC3CC(C3C1)NC2 37078,C(=O)(C1=NOC2(CCN(C(c3ccsc3Br)=O)C2)C1)N1CCN(C)C(=O)C1 37079,Cn1c(C(=O)NC2CC2CNC(c2c(F)cc(N)cc2F)=O)cc2c1CCOC2 37080,C(=O)(CCCC#CC)NC1CCN(C(C(C)OCC#C)=O)C1 37081,Cc1ccnc(C(=O)NCC2CCN(C(=O)C=C(Cl)Cl)C(C)C2)c1F 37082,c1(C(=O)NC(C2OCCN(C(c3nc(CC)sc3)=O)C2)C)ccc(OC)c(O)c1 37083,c1(C(=O)NC2CCCC(NC(C3CC(CC4CC4)C3)=O)C2)cccc2ccsc12 37084,CC(CC(=O)NCC1CCCN1C(c1ccc(CO)o1)=O)C(C)(C)C 37085,N1(C(CNC(C(CC)CC)=O)=O)CCCC(NC(c2ccc(F)c(Cl)c2)=O)CC1 37086,C1(C(=O)OC)CC(CC(N2CC(N3CCOCC3)C(CO)C2)=O)CN(C(C)(C)C)C1 37087,C1(CC=C)(NC(=O)CC(C)(C)C)CCCN(C(=O)CSc2ccc(C)c(C)c2)C1 37088,CN1CCCC(CN2C(=O)NC(Cc3ccc(F)cc3)C2=O)C1=O 37089,Cn1c(Cl)nc2cc(C(=O)NC3C=CC(C)(C)CC3)ccc12 37090,CCC(C)(C)CC(=O)N1CCCC(CCNC(C2CCC3(CCC3)C2)=O)CC1 37091,C(C1=NOC2CN(C(=O)C=Cc3cncs3)CC12)NC(=O)COCC1CCC1 37092,Cn1ncc2ccccc2c1=NCc1ccc2c(c1F)CCC2 37093,C#Cc1cn(C)nc1C(N1CCOC(CNC(=O)C(C)=CC2CC2)C1)=O 37094,c1(C(N2CC(C(C)NC(=O)CCc3cncs3)C(O)C2)=O)cc(F)cc(F)c1 37095,C(=O)(CCC(N)Cc1ccccc1)N(C(CCC)C)C 37096,C(=O)(CCC(=O)NCC1(O)CC(C(=O)NC(CC2CCCC2)CO)C1)NCC 37097,C1(NC(C2CCC3(CCC3)OC2)=O)CC2CCCC(C1)N2C(C1CSC1)=O 37098,C1(C(N2CC(C#N)(SC)C2)=O)(CC)CCCN1C(C1CCCOCC1)=O 37099,C(=O)(CC(CC)CC)NC(CCCC)CNC(c1ccnn1CC(F)F)=O 37100,c1(CC(=O)NCC(CO)NC(=O)CN2CC3CC3C2)cc(Cl)c2c(c1)OCCCO2 37101,N1(C(CCC(=O)NC)=O)CCC2CC2(C(N2CC(C)OCC2C)=O)CC1 37102,c1(C(C(=O)NC(=O)NC(C)C)NCCc2cn(CC)nc2)ccc(F)cc1 37103,c1(OC)c(Br)ccc(F)c1S(=O)(=O)N1CCC(O)(c2ccccc2Cl)CC1 37104,c1(CC)nc(C)cc(=NCC(C2CCCC2)NC(=O)C(C)CSC)[nH]1 37105,C12(C(N3C4(CN(C(c5cnc[nH]5)=O)C4)CC3)=O)CC3CC(CC(C3)C1)C2 37106,c1(C(N(C2CCN(Cc3cnc(Cl)cc3Cl)C2)C)=O)ccc(C#N)cc1 37107,C1(NC(c2ccnn2-c2ccncc2)=O)C=CCN(C(=O)C=Cc2ccc[nH]2)C1 37108,N1(C(c2cc(OC)ncn2)=O)CCC(CCNC(=O)COCC(C)C)CC1C 37109,c1(N2CCC(C(N(CC(C(=O)NCCSC)C)C)=O)C2=O)c(F)cccc1F 37110,C1(NC(CC2(C=C)CN(C(C3CC(=O)C34CCC4)=O)C2)=O)CC2C(C1)C2(F)F 37111,c1(C(CCCOC)C)nc(C2CCCN(C)C2)nn1-c1ccc(F)cc1 37112,n1(C(CC)C)ncc(C(=O)Nc2nccnc2SC)c1C 37113,C1(Cn2cc(C(CC)N(C)C)nn2)CC(SC)CN1C(=O)CSC1CCOC1=O 37114,C1(C(=O)NCCn2ccc(C(=O)NC3CCC(F)(F)C3)c2)C2CC3C(C2=O)C13 37115,CCC(O)C(=O)NC1CC(C(F)F)(NC(c2cnnn2C)=O)C1 37116,C12(C(N3CCN(C(CCCNC(=O)OCC)=O)C4C3C4)=O)CCC(C)(CC1)OC2 37117,C1(NC(C2N(C(C)C)CCC2)=O)C2CCC(C2)C1C(N1CCC(C)(F)CC1)=O 37118,c1(NC)ccccc1C(=O)NC1CC1NC(c1cnc(Br)s1)=O 37119,C#Cc1cncc(C(=O)NCC(C(C)(C)C)NC(=O)Cc2ccsc2Cl)c1 37120,N1(C(c2c(CC)nnc(C)c2)=O)CC2(COC(CNC(=O)C=NOC)C2)C1 37121,C(C)(CC(=O)NCCn1cc(CCN2CCOC2=O)nn1)(C(F)F)N(C)C 37122,N1(C(CC(=O)NC2(C)CN(C(c3ncc(CC)s3)=O)C2)C)C(=O)CCC1=O 37123,c1(CCC)nc(C)c(-c2nc(C(C)SC)nn2C2CCC(C)C2)o1 37124,C1(C(N(C2CC(SC)C2)C)=O)CCCCN(C(C2CCOC2(C)C)=O)C1 37125,C12CCN(C1)CC1CC(C1)C(=O)N2C(CC=CC=C)=O.C(=O)(CCC)NC 37126,Cc1sncc1C(=O)N(C(C(=O)N(C(C)C)Cc1ccccc1)C1CC1)C 37127,C1(NC(c2c(CCOC)n[nH]c2)=O)CCN(C(c2cscc2C#N)=O)CC1 37128,c1(CC(N2CC(C(=O)NCC3CC(=C)C3)(COC)C2)=O)ccc(C)c(F)c1 37129,c1(C(N(CCNC(=O)C(O)C2CC2)CC)=O)ccc(Br)c([N+](=O)[O-])c1 37130,C1(CC(N2CCCC(N(C)C(c3cc(Cl)no3)=O)C2)=O)OCCCC1(C)C 37131,Cc1cc(NC(=O)NC2CCN(C(N3CCOC3=O)C)C2)cc(C)c1Cl 37132,c1(C(=O)NC2CC(F)(CNC(C(CC)(C)C)=O)C2)cc(OC)c(OC)c(N)c1 37133,C1(C(=O)NCC2CCC(NC(c3n(CC)ccc3)=O)C2)CCc2nc(O)[nH]c2C1 37134,S(=O)(=O)(c1cc(Br)ccc1F)N1CC2C(C(N3CCCC4CCCCC34)=O)(C2)C1 37135,Cc1nnc(CCC(=O)N2CC2NC(c2csc(-c3ccc(F)cc3)n2)=O)n1C 37136,CC1c2cc(Br)ccc2CCN1CCSc1ccccc1F 37137,c1(CC(=O)NC2CC(F)(CNC(CCC(C)SC)=O)C2)ccc(C)c(F)c1F 37138,C(C)(C)(C(C)NC(=O)CC(C)c1cnn(C)c1)NC(C(C)C)=O 37139,C1(CNC(C(C2CN(C(C(C)C#N)=O)C2)O)=O)CCNC(=O)C1 37140,CN1C(=O)OCC1C(=O)NC1CN(C(c2cn(Cc3ccccc3)cn2)=O)C1 37141,C1(CNC(CCc2c(C)ncs2)=O)CN(C(c2cccnn2)=O)C2CCN1C2 37142,C1(C(=O)NCC(CC=C)NC(=O)CSc2ccccn2)CN(C)CCN1C(C)=O 37143,N1(C(c2ncccc2F)C(=O)NCCCSCC)CCC(C2(O)CC2)CC1 37144,CCC(O)C(=O)N1CCCC1C(=O)NC(C)Cc1cn[nH]c1 37145,CC1(C)CCC(O)(n2cc(C3COCCN3C(c3cccc(I)c3)=O)nn2)CC1 37146,c1(NC)nc(C)ccc1C(=O)NCC1CCCC(NC(=O)Cc2ccsc2)C1 37147,CCC(CN(C)C)CC(=O)NC1CN(C(c2cc(C)nc(O)n2)=O)CC12CC2 37148,C12(NC(c3c(COC)scc3)=O)CC1CN(C(=O)C(O)Cc1cnc[nH]1)C2 37149,CC1CN2CCN1C(C(=O)NC(C1CCN(C(=O)Cn3cccn3)C1)C)C2 37150,N1(C(c2cc(OC)cc(Br)c2)C(=O)NC2CC2)CCCC(C2(O)CCC2)C1 37151,Cc1ccnc(C(N2CCC(C(=O)NOCC3CCOC3)(C(C)C)CC2)=O)c1N 37152,CCC(C(=O)OC)C(=O)NC1CN(C(c2ccc(OC)cn2)=O)C1 37153,c1(C(=O)NCCN(C(=O)C(=O)NC2CC2)CC(C)O)ccc2c(O)nccc2n1 37154,Cc1ccc2ncc(C(=O)NCC3CC3NC(=O)Cc3cnnn3C)n2c1 37155,C(=O)(CN=c1cc[nH]cc1)NC(CC)CNC(=O)C1=C(C)OCC1 37156,N1(C(CCC2(C)CN(C(c3c(CC)nn[nH]3)=O)C2)=O)CCC2(CNC(=O)N2)C1 37157,N1(C(C(n2c(C)ncc2)C)=O)CCC(C(=O)NC2CC2(C)C)C1C 37158,C(=O)(C1=C(SC)CCCC1)NC(CC)C(=O)Nc1c(OC)cccc1C 37159,N1(C(c2c(CC)nco2)=O)CC(NC(c2ccc(N(C)C)cc2)=O)CC12CCC2 37160,CC1(C)C2CCC1(CC(=O)NC1(CF)CCN(C(=O)CCC3CCCO3)C1)CC2 37161,C#Cc1ccccc1CC(=O)N(C)CCNC(c1cc(C2CC2)on1)=O 37162,C1(NC(CCOCC)=O)CC2(CCN(C(c3cnn(CC)c3Cl)=O)C2)C1 37163,c1(NC(C)CN(C)C(C2CCCC(C)(C)CC2)=O)cccc(F)c1[N+](=O)[O-] 37164,c1(OC)nc2ccc(CNc3cc(NCC4CC4C(C)C)ncn3)cc2[nH]1 37165,N1(C(c2occ(C)c2C)=O)CCCC12CCN(C(=O)CC1CSC1)CC2 37166,C1(C(=O)NCCOCC(N)=O)(CC)CCN(C(=O)C(C)=C2CC2)C1 37167,c1(OC)cc(CC(=O)NC2(C)CN(C(C3CCC(CN(C)C)O3)=O)C2)ccn1 37168,N#Cc1ccc(C(=O)NCC(CC2CC2)C(=O)NCCc2cncs2)o1 37169,C12(C(N(C(CC)CC)CC)=O)CC(NC(=O)C(F)C3CCC3)(C1)C2 37170,N1(C2C(c3c(Br)ccc(C)c3)C2)CC2C(C1C(=O)NC1CC1)C2(C)C 37171,C1(C(N2C3C(NC(C(CCC)=CCC)=O)C(C3)C2)=O)CCC([N+](=O)[O-])CC1 37172,c1(C(=O)NC2C3CCN(C(c4c(CC)nc[nH]4)=O)C32)c(Br)ccc(OC)c1C 37173,c1(C(=O)NCCC2OCCN(C(CC=C)=O)C2)cc(OC)ccc1Br 37174,c1(N2CC(C)OCC2)nc(=NCCOc2ccncc2)[nH]c2c1SCC2 37175,C(c1ccc(C)cc1)=CCSC.C1(CC)C2CCN1C(=O)CNC2=O 37176,c1(SCCNC(NCC2CC=CCC2)=NCc2ccccc2)cc2occc2[nH]1 37177,c1(C(=O)NCC(C)(CC(C)C)NC(C(=O)NCCOC)=O)ccnc2[nH]ncc12 37178,c1(CC)cnccc1C(=O)NC(CNC(c1nccn1C)=O)C1CC1 37179,c1(C(C)C(=O)N(C2CCCC2)Cc2ccc(Cl)cc2)ccc2c(c1)OCO2 37180,C1(C(=O)NC(Cn2cc(C(CC)(C)O)nn2)C)CC(C(=O)OC(C)(C)C)=NO1 37181,C1(NC(C2CSC2)=O)CCC2CN(C(c3ccc(CO)cc3)=O)CC2C1 37182,Cc1ncc(CC(N2CCC(NC(=O)C(C)NC=O)C(C)C2)=O)c(O)n1 37183,c1(C(N2CCC(C)(CNC(C3CC(=O)N(O)C3)=O)C2)=O)cc2nc(=O)ccn2[nH]1 37184,N(C1CCCc2ccc(F)cc21)C(=O)NC(C)(CC1CCC1)C(=O)O 37185,Cn1cc(I)c(=NC(=O)C(N)n2cc(-c3ccc(F)nc3)nn2)[nH]1 37186,C1(C(=O)NC(CCC)CCO)CCCCN(C(=O)CC2CC(OC)C2)C1 37187,C(=O)(C(C)(O)CC(F)(F)F)N1CC(C)C(n2cc(-c3ccc(CO)nc3)nn2)C1 37188,C(C)(N=c1nc(N2CC3C(C(F)(F)F)C3C2)c2c([nH]1)CCC2)c1c(C)nc(C)[nH]1 37189,C(=O)(CCC(C)(C)C)NCC1OCCC(NC(CN2C(C)CCCC2)=O)C1 37190,c1(C(N2CC3C(CNC(Cc4c(C)noc4)=O)(C3)C2)=O)cnc2c(c1)CCCO2 37191,c1(N2CCCC(CC=C)(NC(=O)C=COCC)C2)nc2ncc(Cl)cc2o1 37192,CCC(CC(C)C)C(=O)NCC(O)CNC(c1ccc(Br)c(Cl)c1)=O 37193,c1(C(C(=O)OCC2C(OC)CCC2)(C)C)ccc(C(F)(F)F)cn1 37194,C12(C(=O)NCC(=O)N(C)CC)CC1CCN2C(=O)CC1CC2(CCC2)C1 37195,c1(C(=O)NCC2C(NC(CC3(C)CCCO3)=O)CC2)nccc(Cl)c1F 37196,N(C1CCCc2n[nH]cc21)C(C(C1CCOC1)NC(CCC(C)(F)F)=O)=O 37197,CCCCC(CCCC)C(=O)N1CC(NC(=O)C(C)(C)NC(=O)C(F)(F)F)C(C)C1 37198,C=CCN=c1nc(N2CCS(=O)(=O)NC2)c2ccc(OC)cc2[nH]1 37199,Cc1c(C(=O)N(CCCNC(=O)C=CC(=O)N(C)C)C)c(C(F)F)nn1C 37200,N1(C(c2cn(C(C)C)nn2)=O)CCC(C)(C)C1CC(=O)NC(C(O)CO)C1CC1 37201,C1(NC(C(=O)N(C2CC2)CC2ON=C(C)C2)=O)CCC(C)(C)C(C)C1 37202,c1(C(=O)NC2C(NC(c3c(CC)nc(C)o3)=O)COCC2)cc(C)nc(C)c1 37203,c1(C(N2CCC(F)(C(N3CCC(OC(F)F)C3)=O)C2)=O)ncccc1Br 37204,C#CC1CN(C(C2CC3(C2)CC(O)C3)=O)CCN1C(c1cc(C2CC2)on1)=O 37205,C1(NC(C2CC(CCO)C2)=O)CC1C1CCN(C(c2nnc(O)cc2O)=O)CC1 37206,C1(NC(C(CC=C)(C)N(C)C)=O)CCOC2(CCN(C(=O)COC(C)=O)CC2)C1 37207,CC1CN(C(C(=O)NCc2ccco2)C2CC2Cl)CC(c2ccsc2)O1 37208,CCC(N=c1nc(N2CC3CC2CN3C)c2[nH]ccc2[nH]1)c1ncc(C)[nH]1 37209,N#Cc1ccc(CN2CCC(O)(C(=O)Nc3cc(Cl)ccc3I)C2)cn1 37210,N1(C(C(C(=O)OC)(C)C)=O)CC2CCC1C1CN(C(=O)CNC(=O)C(C)C)CC21 37211,c1(NC(CCC2CCC(NC(c3[nH]c(=N)sc3)=O)CC2)=O)ccc2c(c1)OCC2 37212,N1(C(CC2C(C)(C)C2(C)C)=O)CC=C(CC(=O)NC2C=CCCC2CO)CC1 37213,c1(CC(=O)NCCN(C(C(COC)N(C)C)=O)CC(C)O)ncn2c1CCCC2 37214,Oc1ccc(Cl)c(F)c1-c1nc2ncccn2n1.CC 37215,C(=O)(C1=CCCCO1)N(C1CCCN(C(C(=CC2CCCC2)C)=O)C1)CC1CC1 37216,C1(C(=O)OC)CCC(C(CO)N(C(C)CNC(c2ccccc2OC)=O)C)CC1 37217,CC1(C)CC(O)(C(=O)NCC2CCCN(C(C3(c4ccccc4F)CC3)=O)C2)C1 37218,Cc1cccc([N+](=O)[O-])c1N1CCCC(C)(CNC(C2(CF)CCC2)=O)C1 37219,c1(C(=O)NCC(C(=O)OCc2onc(COC)n2)C)ccc(C)cc1 37220,C1(C(=O)NCC2N(C(C(CC(=O)OC)C)=O)CCCC2)CCC(C2CCC2)CC1 37221,CCC(C)C(CC(=O)N1CCC(N(C)C)C1(C)C)NC(c1cncc(OC)c1)=O 37222,N1(C(c2c(C(C)C)onc2)=O)CC2CCC2(CNC(C2CCS(=O)(=O)CC2)=O)C1 37223,N1(C(c2ccc(CC)s2)=O)CC=C(CCNC(C2CC2(F)Cl)=O)CC1 37224,CCCCCC(=O)N(CC)CC1(CNC(=O)CC2CC(OC)C2(C)C)CC1 37225,CC(CNC(=O)OC(C)(C)C(=O)O)C(C)(C)C 37226,C1(C(N2CCN(CC=C)CC2)=O)CNC(=O)CN1C(C1(CC2CC2)CCC1)=O 37227,C1(C(=O)NCCCN(CCC)C(c2cnn(C)c2Cl)=O)CC2C=CC1C2 37228,C1(C(=O)OC)(NC(CCCC(=C)C)c2nnnn2C)CCS(=O)(=O)CC1 37229,C1(CC(C)(C)C)CN(C(c2scnc2C(F)F)=O)CC1NC(=O)C=CCF 37230,N1(CC)CC(C(=O)NCCCNC(=O)CCc2ncc(C)[nH]2)c2ccccc21 37231,C(=O)(CC1=NN(C)C(=O)C1)N(C1CCCCC1)CCNC(C1C(C)SCCC1)=O 37232,C#Cc1ccc(Cl)c(C(N2CC(NC(=O)C(F)F)C(CC)C2)=O)c1 37233,N1(C(c2cc(CNC(CC(C)(C)OC)=O)no2)=O)CCCC2CC1C2(C)C 37234,CCCCCCN(CCNC(=O)CSCC)C(C1CC(F)(F)C1)=O 37235,O=C(C1=CCSC1)Nc1cnn(C2CCN(C(c3sccc3F)=O)CC2)c1 37236,Cn1nc2ccccc2c1C(N1CCCN(C(=O)Cc2ccns2)C(CO)C1)=O 37237,N1(C(C2C3CN(C)CC32)=O)CCC2CN(C(C3(C(F)(F)F)CC3C)=O)CC2CC1 37238,c1(C(c2nn(-c3cccc(OC)c3)c(Cn3cncn3)n2)C)ccc(F)cc1F 37239,C1(CNC(c2cc(CC)nn2C)=O)CC2(CCN(C(=O)C=CC3CC3)C2)CO1 37240,c1(CSCC)nc2ccccc2n1CC.C1(S)COCCC1C(=O)O 37241,C12CCC(C)(C)CN1C2=O.c1(C2(NC(CC(C)CF)=O)CC2)ccc(C#N)cc1 37242,CCCCC(C)C(=O)NCc1n[nH]cc1C(=O)Nc1conc1C 37243,c1(C(=O)OC)cc(C(=O)NC2CCCC2NC(=O)C(C(C)O)N(C)C)c(F)cn1 37244,N1(C(C(=O)NCC)=O)CCC2CN(C(c3ncnc(OC)c3F)=O)CCC2C1 37245,C12(CNC(C3N(C)CCC3)=O)CC(CO1)N(C(C1CCN(CCO)C(=O)C1)=O)C2 37246,Cc1nn(C)c2ncc(C(N3CCC4(NC(c5cnsn5)=O)CCCC34)=O)cc12 37247,N1(CC(N)=O)CCCC(N=c2[nH]c(=NCC3CCSC3)c3[nH]ccc3[nH]2)C1 37248,C(=O)(CC(C)CCC(=O)NCC(CC(C)C)NC(=O)C=Cc1cnc(C)s1)OC 37249,C(=O)(CCCC(C)(F)F)N(C(C)CNC(=O)CCc1ccco1)CC 37250,CC1(C)CC(NC(c2ccns2)=O)CN(C(=O)COCCO)C1 37251,C(c1cccc([N+](=O)[O-])c1)=CC(=O)NCCCN(C(=O)C(C)(C)C(F)(F)F)C 37252,Cc1nc(CO)ncc1C(=O)NC(CNC(=O)CC1CC(F)(F)C1)C(C)C 37253,C12(C(=O)NC(COC)C(=O)OC)CC(C)(CN1C(=O)C(F)C(F)(F)F)C2 37254,c1(C(N(CC(CC)NC(C2(O)CC(C)(C)C2)=O)C)=O)cc2cn[nH]c2cn1 37255,N1(C(CC(CC)C)C)CCCOC(CNC(c2ccccc2)=O)C1 37256,C1(C(=O)NC(CC(=O)NC(C)C)C)CN(C(=O)CCc2cn[nH]c2)CC12CC2 37257,c1(C(=O)NCC2C3N(C(C=C(COC)C)=O)C(CC3)C2)c[nH]c2nccc-2c1 37258,C1(C(=O)NC(CC)CN(C)C(c2sccc2C(F)F)=O)CCn2cnnc2C1 37259,CC(C)C(CO)C(=O)N1CCC(NC(=O)Cn2nnc(C3CC3)n2)C1C 37260,C(=O)(C(C)CC(C)C(C)=O)NCC1C(NC(c2c(OCC)cccc2)=O)C1 37261,C1(NC(=O)NCCSCCO)CCCC(C(C)=O)C1.C12CC1C2 37262,C(=O)(C(O)CC(F)(F)F)NCCCN(C(C1(C)CC(F)(F)C1)=O)CC 37263,c1(NCC2OCCN(C(c3c(C)coc3C3CC3)=O)C2)ccc(S(C)(=O)=O)cn1 37264,Cc1nc(CC(N2CCCC2Cc2cn(Cc3nccs3)nn2)=O)oc1C 37265,C1(NC(=O)C=CC2CCC2)CC2CCC1(NC(C1(F)CCCCC1)=O)C2 37266,c1(C(=O)NCCOCCN(C(C(=O)NCC)C)C)nccc(C)c1N 37267,C1(NC(C(C(C)C)C)=O)CC2(C1)CC(CNC(c1cc(C3CC3)nc(O)c1)=O)C2 37268,C1(CC(=O)NCC2(C)CC(NC(=O)CN3CC4CC4C3)C2)CCCCC1(F)F 37269,C1(CNC(C(CCSC)O)=O)CC2COCC2N1C(c1cnn(C(C)C)c1N)=O 37270,C1(C(N2C(C)(C(=O)OC)CC2)=O)CCN(C(C2C3CCCC23)=O)CC1(C)C 37271,C1(C)(C(=O)NC(C)Cc2ccco2)CCCCC1(C)C 37272,C(CC(O)C(=O)NCC1(F)CC(NC(c2ccc(C)nc2)=O)C1)SC 37273,C1(CC(=O)NCCN(C(c2cnsc2)=O)CC)CC(C)(C)CCO1 37274,c1(C(=O)NC2CC(NC(c3c(C)ncc(C)c3)=O)C2)ccc2ncnc(O)c2c1 37275,c1(C(=O)O)cc(C(N2CCC(c3cscn3)CC2)=O)nc2ccc(F)cc12 37276,C1(C(N2CC(CNC(CCC=C=C)=O)OCCC2)=O)CCOCC12CCCCC2 37277,C1(C)(C(N2CCOCC(NC(CCC=CC)=O)C2)=O)CC2CCC(C1)S2 37278,N1(C(c2ccc(Cl)c(Cl)c2)C(=O)NC(C)C)CC(C)OCC1(C)C 37279,c1(C(=O)NCCCNC(C2CCS(=O)(=O)N2)=O)cc(F)c(F)c(O)c1F 37280,C1(O)(C(C)NC(=O)Cc2ccn(C(F)F)n2)CCN(C(C2CNC(=O)N2C)=O)C1 37281,c1(C(N(CC(C)NC(c2ccnc(C(C)(F)F)c2)=O)C)=O)cncc(Cl)c1Cl 37282,c1(CC(CO)N(CC(=O)NCC2CCCCC2)C(C)C)ccc(C#N)cc1 37283,c1(C(C(=O)NC2CC(F)(CNC(c3cc(CF)on3)=O)C2)O)cc(F)cc(Cl)c1 37284,C1(NC(c2nc(C3CC3)n[nH]2)C)CCCOCC1 37285,N1(C(C(C(=O)OCC)F)=O)CCC(C)(CNC(c2ncn(C(C)(C)C)n2)=O)CC1 37286,N1(C(C=CC=CC)=O)CCCC(CO)(NC(=O)C(C)C2CCOC2)C1 37287,c1(C(C)OCC)nc(-c2oc(C(C)C)nc2C)n(-c2ccn(C)n2)n1 37288,CC1CN(Cc2cc(Cl)ccc2F)CCN1Cc1cccc(C(C)(C)C)n1 37289,C1(NC(c2c(C)n[nH]c2)=O)CCC2(CC1)CCN(C(=O)C(=O)C(C)(C)C)C2 37290,N1(C(c2cc3cscc3s2)=O)CCC(C2CCCN(c3ncncc3I)C2)CC1 37291,c1(C(=O)NC(C(=O)N2CCC(CC#C)C2)(C)CSC)cc(C)ncc1C 37292,N1(C(Cc2c(C)con2)=O)CCN(C(=O)Cc2ccccc2Br)C2CCC12 37293,C1(C(=O)NCC(C2CC2)OC)CCN(C(c2nc[nH]n2)=O)C1C 37294,Cc1ccc(F)c(C(N2CCC(F)CC2C(=O)NCC2CC(CN=[N+]=[N-])C2)=O)n1 37295,c1(C(=O)NC2CCCC2)occ2c1CCC2.Cc1cc(C(=O)N2CCC2)ccn1 37296,CC1CN(C(C2(C(C)(C)O)CC2)=O)CCC1C(=O)NCCC1CCC(C)(C)C1 37297,C1(CNC(C2CC(=C)C2)=O)CN(C(=O)CC2CCCN(C)C2)CCC12CCOC2 37298,C1(F)(C(=O)NC(C(=O)NC)C2CC2)CCCN(C(c2ccc(C3CC3)s2)=O)C1 37299,c1(C2CC(C(=O)NC(C3CN(C(C(C)OC)=O)C3)C)C2)ccccc1F 37300,C1(CNC(C(C)OCC(C)C)=O)C2CCCC1N(C(C1CCCS1)=O)C2 37301,C1(NC(C2(C)COC2)=O)CC(F)(F)CC1NC(c1ccc(CN2CCCC2)o1)=O 37302,Cc1ccccc1-n1ccc(C(=O)Nc2ccc(C(=O)N(C)C)nc2)n1 37303,CCCCCCC(C)(CC)NCc1ccc(-c2nn[nH]n2)cc1 37304,N1(C(C2C(C(=O)NCC#C)C2)=O)CCC(CC2CC2)CC1.c12cc(no1)NC2=O 37305,c1(CCC)cnnc(C(=O)NC2CN(C(c3cc[nH]c3)=O)CC2OC)c1 37306,c1(OC)cnncc1C(=O)NCC(O)CNC(C1(O)CCCCC1)=O 37307,C1(NC(=O)Cc2cscn2)CN(C(c2csc(O)n2)=O)C2(CCCCCC2)C1 37308,C1(C(C)C2CC2)C(=O)Nc2nc1ns2.C1(C(=O)OCC)(CC)CC1 37309,C1(CNC(C=Cc2n(CC)ncc2)=O)CCCC2(CN(C(=O)C(C)(C)SC)C2)O1 37310,Cc1nc(SCC(=O)NCCN(C(=O)COCC2(F)CC2)C)cs1 37311,[N-]=[N+]=NC1(C(N2CCC3CC2C(=O)O3)=O)CCN(C(c2cc[nH]n2)=O)C1 37312,c1(C(=O)NC2C(NC(C(C(C)C)F)=O)COC2)nc[n+]([O-])cc1Cl 37313,CCCCCC(=O)NCC(=O)NCC(C)CNC(c1ccccc1Cl)=O 37314,C1(C(=O)NC2(C)CC(C(=O)OC)C2)CC(F)(F)CN1C(=O)C(C)COC 37315,c1(SC)ccc(C(=O)NC2(CNC(=O)C#CC3CC3)CCCCC2)cc1 37316,CCCCCC(O)C(=O)N1CC2CC1(CNC(C1CC1CN(C)C)=O)C2 37317,c1(N(CCCNC(=O)OC)C)nc(N2Cc3ccc(C)cc3C2)nc2c1CCC2 37318,CCN=C(NCCc1ccsc1Br)NCC(c1ccoc1)O 37319,c1(C(=O)NCCN(C(=O)CC2(O)CCC2)CCOC)scc(C)c1C 37320,C(=O)(C1=CCCCO1)N1CCC(OCCNC(C2CC(Cl)(Cl)C2)=O)C1 37321,CC#CCCC(=O)N1CC(NC(=O)Cc2ccnn2C(C)C)C(n2ccnn2)C1 37322,c1(C(=O)NC2(CC=C)CCN(C(=O)C(CCO)NC)C2)oc2ccccc2c1C 37323,N1(C(CCCC#C)=O)C2CCCC1CC(CNC(c1ccccc1C)=O)C2 37324,c1(CCC(=O)NC2CN(C(c3cc(OC)ns3)=O)C(C)C2)c(C)nn(C)c1C 37325,C1(N(S(C)(=O)=O)C)CCN(S(C)(=O)=O)CC1.C12(N)COC(C1)C2 37326,c1(C(N2CCCN(C(C3(OC)CCSC3)=O)CC2)=O)cc2c(s1)C(C)(C)CCC2 37327,N1(C(C2=C(C)OCC2)=O)CC(NC(=O)C(C)CS(C)(=O)=O)C2(CCOCC2)C1 37328,C1(Cn2cc(C(CCC)=O)nn2)CC2CCCC2N1C(C1CC2CC1CC2=O)=O 37329,c1(OCC#CC(NOCCN(C)C)=O)ccc(F)c(Cl)c1.C(COC)N 37330,C1(C2CCCN(C(c3cc4ccc(F)cc4s3)=O)C2)(NC(CC2C(C)C2)=O)CC1 37331,O=C(C1=CC2(CCOC2)C1)N1CCC(F)C(NC(C2CC(O)(C(F)(F)F)C2)=O)C1 37332,N1(CC(=O)NC(CNC(CC(C)F)=O)(C)C2CC2)CCCNC1=O 37333,c1(CN(C)C(C2CCN2C(c2cc3sccc3s2)=O)=O)cccc(Cl)c1Cl 37334,N1(C(C(C)NC(=O)C(F)(F)F)=O)CCC2CN(C(c3ccccc3C#N)=O)CC12 37335,c1(C(=O)NC2C(C(C)(C)C)N(C(=O)CC3CC4(CCC4)C3)CC2)ccc([N+](=O)[O-])[nH]1 37336,C1(CNC(c2cc(CC)on2)=O)CC2(CC2)CN1C(=O)C(C)c1cncs1 37337,C(=O)(C(CCS(C)(=O)=O)OC)NC1C(NC(C(=CC2CCCC2)C)=O)CCCC1 37338,C1(C(N(CCC(=O)NC(COCC)CO)CCCO)=O)CCC(C2CC2)C1 37339,C1(C(=O)NC2(CC#C)CCC2)C=CCN1C(=O)Cc1csnn1 37340,c1(CC)cc(F)ccc1C(=O)NC1CC(NC(c2nc(C)ncc2Cl)=O)C1 37341,S(=O)(=O)(c1ccc(Cl)nc1)N1C(C(=O)NC(C)C2CC2)CC2CC21 37342,C1(C(=O)NS(CC#N)(=O)=O)(Nc2n[nH]c(C(F)(F)F)n2)CC2(CC2)C1 37343,C1(NC(CCn2ncc(C)c2)=O)CC2CC1N(C(=O)CCNC(=O)CO)C2 37344,Cc1cc(=O)oc(C)c1C(=O)NC(C)C(CO)NC(=O)C(C)CC(C)(C)C 37345,c1(-c2ccc(NC(C34CNCC3C4)=O)s2)cccc2ccccc12 37346,c1(C(C=O)N(C2(NC(=O)OC(C)(C)C)COC2)CC)cc2c(cc1Cl)NC(=O)C2 37347,c1(C(N(CCNC(CCC)=O)C(C)C)=O)nc2ccccc2cc1Br 37348,N1(C(C(CCCCC)O)=O)CCC2(CCC2)C(NC(=O)CN(C)C(N)=O)C1 37349,N1(C(C(CO)OC)=O)CCCC(CNC(c2cc(Cl)n[nH]2)=O)C1 37350,Cc1cc(F)c(O)c(OCC(C)Sc2ccccc2)c1F 37351,N1(C(CCCC)=O)CCN(C(C2(OC)CCCOC2)=O)CC(CO)C1 37352,C12(C(=O)NC3CC(C)(CNC(C=CC)=O)C3)CCCCC(=O)N1CCC2 37353,N1(C(Cc2nc(COC)sc2)=O)CCCN(C(=O)C(C2CCOCC2)O)CC1C 37354,S(=O)(=O)(c1cncc(Br)c1)NC1CN(C(C2(C)CCCC2)=O)CC1F 37355,c1(C(N2CCCC(NC(C(n3ccc(C)n3)C)=O)C2C)=O)ccc([N+](=O)[O-])n1C 37356,Cc1ccc(Br)c(C(N2CC(CNC(C3(F)CC3)=O)CC2C)=O)c1 37357,C1(C(=O)NC)(CNC)CCCN1C(=O)CC(=O)OC 37358,c1(OC(C)C)cnccc1Br.C12CC(OC(C)(C)C)C1NC(=O)N2 37359,c1(C(N(CCN(C(C)C)C(C2CC23CC3)=O)C)=O)cccc2cc[nH]c12 37360,Cn1c(C(F)(F)F)nnc1C1CCCN(C(=O)Nc2cnc(C(C)(C)C)nc2)C1 37361,C(=O)(C(CCSC)N(C)C)NC1(CC)CN(C(=O)CCNC(c2ccoc2)=O)C1 37362,N1(C(C2(C(N)=O)CC2)=O)CC(NC(=O)Cc2cncnc2O)C2(CCC2)C1 37363,N1(C(C(F)=CC)=O)CCCOC(CCNC(=O)CC2COC(C)(C)CO2)C1 37364,c1(C(=O)NCC(CO)NC(=O)CC2COCCO2)ccc(-c2nnc(S)o2)cc1 37365,C1(C(=O)NCCCC(C)NC(C(CNC(C)=O)(C)C)=O)CCC(C)=C(C)C1 37366,c1(C(N2C(CNC(C3C=C(C)CS3)=O)CC2)=O)cc(N)c(O)c(F)c1 37367,c1(OCC)ccc2ccccc2c1NCc1cc(C(=O)O)ccc1Br 37368,C(CCCC(=O)NC1CCC(NC(=O)CCSCC(=O)OC)CC1)OCC 37369,CC(C)CC(Cc1cn[nH]c1)N(C(=O)CC(F)F)C(=O)CC1CCCCCN1 37370,C(CCCCCC(=O)NOCC1CC1)NC(c1c(C)nccc1)=O 37371,O=C1CC(C(N2CCC(OCCF)C2)=O)N(C(=O)C(=C2CCCCC2)F)C1 37372,N1(C(C2(CC)CCCO2)=O)CC(NC(=O)Cc2cccs2)C(C)C1 37373,C(N=c1nc(C)c([N+](=O)[O-])c[nH]1)C1CCN(C(C(C(CC)O)C)=O)CC1C 37374,c1(C(=O)NCCCC(C)NC(=O)C(C)(C)C)cncc(C(=O)N(C)C)c1 37375,C1(NC(=NCc2nc(CO)sc2)NC2CCCC2)CCOC2(CCCC2)C1 37376,c1(C(N2C(C(=O)NCC3(C)N=C(C)SC3)CCC2)=O)cc(C#N)ccc1C 37377,c1(CC(N2C(C)C(NC(=O)C(CO)OCC(F)(F)F)CC2)=O)cc(F)cc(F)c1 37378,Cc1cc(F)cc(Br)c1C(=O)NCC1(c2ccccc2)CCN(C)C1 37379,C(=O)(C(CCOC)OC)NCC1(CN(C(CCOCC#C)=O)C)CC1 37380,N1(C(c2cccc(Cl)c2)=O)CC2(CCC(NCc3cnccc3Cl)C2)C1 37381,N1(C(C2N(C)CCCCC2)=O)CC2CN(C(c3cc4cc[nH]c4cn3)=O)CC2C1 37382,C1(CNC(=O)COC2CC2)C2CN(C(c3cc[nH]c3C3CCCC3)=O)CC12 37383,c1(OC)ccc(CNCC(O)CC2CCCC2)c(F)c1F 37384,C(=O)(C1=CCCC1(C)C)N1CCC(O)(CNC(CC2CCN(OC)CC2)=O)C1 37385,C1(C(=O)NCC(C)(C)NC(c2cc(OCC)n[nH]2)=O)C(O)C(=O)N(C)C1C 37386,C1(C)(C(=O)NC(C(C)NC(c2csnn2)=O)CO)Cc2ccccc2NC1=O 37387,c1(OC)ccc2c(c1)CC(C(N1CC3C(CNC(=O)CC(C)F)C3C1)=O)CO2 37388,c1(CC)ccc(F)c(C(=O)NCC2CCCC(NC(=O)CC3CCOCC3)C2)c1 37389,CC(C)CC(O)C(=O)NC(c1nc(C(=O)NOCCCC2CC2)co1)C 37390,N1(C(CCCCSC)=O)CCCC(C2CCN(C(=O)C3CC3)CC2)CCC1 37391,Cc1nc(C(N2CC(NC(c3ccnc(O)c3)=O)CC(F)C2)=O)c(C)n1C 37392,N1(C(C(n2cc(-c3c(Cl)ccc(C)c3)nn2)C)=O)CCC(C2CC2)C1CN(C)C 37393,C1(C(=O)NCC2CC(NC(CC3(CC(=O)OC)CC3)=O)C2)NC(=O)OC1(C)C 37394,N1(C(Cc2cc(C)on2)=O)CCC(NC(=O)CN(C2CCSC2)C)C(C)(C)C1 37395,C1(OCCOC)(CO)CCN(C(C2C3CN(c4ccnc(C)n4)CC23)=O)CC1 37396,C1(CC(=O)NC(C)C(=O)NC(c2ccc(Br)cc2)C)CCCCCC1 37397,C1(N(C)Cc2cncc(-c3ccc(Cl)cc3)c2)CCC(O)(c2cncn2C)CC1 37398,N(C1c2ccccc2CC1NC(=O)C(C)O)C(C=CS(CC)(=O)=O)=O 37399,CCCCCCCN=c1nc(N2CCC(c3nc(=N)[nH][nH]3)C2)c2ncccc2[nH]1 37400,C12(NC(=O)Nc3cc(C(N4CCOCC4)=O)cc(F)c3)CCC(O)(CC1)CC2 37401,N1(C(=O)OC(C)(C)C)CC=CC(C(=O)NCCCC2CC3CCC2C3)C1 37402,C(=O)(C#CC1(C)CCCO1)NCC1C2CN(C(C(C)CC3CC3)=O)C1C2 37403,N1(C(c2cc(C)cc(N)c2)=O)C2CCC1CC(CNC(c1cn(C)nc1Cl)=O)C2 37404,N(C(=NCCCCl)N1CCC2(CNC(=O)C2)C1)CC1C(C)(C)C1 37405,C(=O)(CC(C(F)(F)F)c1ccon1)NC1CC(CNC(=O)CCCC2CCCC2)C1 37406,C1(OC)CN(C(c2cn(C)nc2Cl)=O)CC1NC(c1ccccc1O)=O 37407,C1(N(C(C(c2cnn(C)c2)OC)=O)C)CCC2CN(C(=O)CCC(C)(C)C)CC12 37408,CC1CN(C(C2CCC(N(C)C)CC2)=O)CCN1Cc1cccc(C#N)n1 37409,Cc1ccc(CNC(=O)C(C)NC(C2COCC2(C)C)=O)cc1C 37410,N1(C(C(C2CCC(=O)N2)C)=O)CCC(NC(=O)CC2CCOCC2)C(C)(C)C1 37411,C1(n2cc(COC(C)C)nn2)CC2CCC1CN(C(C1CC1(C)C)=O)C2 37412,N1(C(C(N2CCSCC2)C)=O)CCCOC(CNC(=O)C=Cc2cccs2)C1 37413,Cc1sc(C(=O)NC2CCCC(NC(=O)CC(C)NC(N)=O)C2)cc1[N+](=O)[O-] 37414,c1(OC)c(C(=O)NC(C2CCCN2C(c2ncccc2O)=O)C)c(C)nn1C 37415,c1(C(=O)NC2CC(CCNC(c3c(OC)c(C)cs3)=O)C2)cn2ccnc2cn1 37416,Cc1cc(C(N2CC=C(CCNC(=O)CC(O)C3CC3)CC2)=O)c2n[nH]cc2c1 37417,C1(CCNC(CCC=C=C)=O)CCN(C(=O)CN2CCCS2(=O)=O)CC1(F)F 37418,C(N=c1cc(Cl)nc[nH]1)C1(O)CCCN(Cc2c(OC)nn(C)c2)C1 37419,CCCCC(O)C(=O)N1CCCC(NC(c2ccc(C(=O)OC)cn2)=O)CC1 37420,N1(C(C(c2ccc(C)o2)C)=O)CCC(C)N(C(=O)COc2cn[nH]c2)CC1 37421,C1(CCC(=O)NC(CN(C(C=CCN(CC)CC)=O)CC)C)CCOCC1 37422,C=CCC(CC)C(=O)NC1CCN(C(c2cnn(-c3ccccc3C)c2)=O)C1 37423,CCC(C)C=CC(=O)NCC(C)=CC(=O)NCCN(C)C(=O)C1CC1 37424,c1(NC(C)=O)c[nH]c(C)c1C(=O)NCC1CC(NC(c2nn[nH]c2Cl)=O)CCO1 37425,Cc1ccc2[nH]cc(CCC(=O)NCCOCCNC(=O)CC(O)C3CC3)c2c1 37426,c1(OCC)ccc2ccccc2c1NC(=O)C(=O)NC1CCc2nc(C)nn2C1 37427,CCCCC(C(=O)NCCCC(C)(C)C)NC(=O)C=CC(C)C 37428,N1(C(=O)OC(C)(C)C)CCCC1C(=O)NC1CCCC1NC(C1(C)CC=CC1)=O 37429,C1(NC(=O)C=CC=C(Cl)Cl)COCC1NC(c1n[nH]cc1Cl)=O 37430,CC(C)C1=NOC(C)(C(N2CCC(O)(CCNC(=O)Cc3cscn3)CC2)=O)C1 37431,N1(C(C2CC(=C)C2)=O)CC(OC)C(NC(C2CC(O)C2)=O)C1 37432,c1(CCC(N2CCC(CO)(NC(C3CC(O)C3)=O)CC2)=O)cccc([N+](=O)[O-])c1 37433,C(=O)(CC(F)(F)C(F)F)NCC(CN(C)C(C1(C)CCC12CCC2)=O)(C)C 37434,C1(NC(C2CCN(C)C2=O)=O)CC(F)CN(C(c2ccc(OCCF)cc2)=O)C1 37435,N1(C(CC2(CC(=O)OC)CC2)=O)CCCC(NC(=O)Cc2cccc(C)c2)CC1 37436,C(C(C(=O)NCCC1CC(=O)N(C)C1)C(C)(C)C)NC(c1cn(CC)nc1)=O 37437,CN1CCN(C(C2(F)CCCN(C(c3cc(N)cc(F)c3)=O)C2)=O)C(C2CC2)C1 37438,c1(-c2occ(C(=O)NC(C3CCOC3)CNC(CSCC)=O)n2)ccc(Cl)cc1 37439,C1(C(=O)NC(CC#CC)CO)CC(C)(C)CCN1C(=O)CCOC(C)=O 37440,C(=O)(CCCc1cncs1)NCC(CC)NC(=O)CSc1nc[nH]n1 37441,C1(C)(C(N2C(C(C)NC(=O)Cc3sccc3Br)CCC2)=O)COC(=O)C1 37442,c1(C(=O)NCC2N(C(C(COC)C)=O)CC(O)C2O)cn2c(n1)COCC2 37443,C1(CNC(N)=O)CC(C(F)(F)F)CN1C(=O)CCOC(c1ccccc1)=O 37444,c1(C(C(=O)NC(c2ccccc2)CNC(C(CC)F)=O)SC)c(F)cccc1F 37445,Cc1nccc(=NCC2CCC(NC(C3CCC(N=[N+]=[N-])CC3)=O)C2)[nH]1 37446,N1(C(CSC(C)(C)C)=O)CC(NC(c2ccc(F)cc2)=O)C(C(=O)O)C1 37447,c1(C(=O)NC(CCNC(c2c(C)c(CO)ccc2)=O)C)noc2ncccc12 37448,Cc1sc(C(F)(F)F)nc1C(=O)N(CC(C)(C)NC(=O)CC1C=NN(C)C1=O)C 37449,c1(C(=O)NC2(C(=O)NCc3ccnc(C)n3)CC2(C)C)cc(O)nc(C)n1 37450,c1(C(CC(=O)OC)NC(=O)NCc2sc(Cl)cc2Cl)ccccc1Br 37451,CC(C(=O)N1CCC(C2CCOC2)C1)S(=O)c1ccccc1.CC(C)(C)O 37452,C(C(C(C)(C)C)NC(=O)C(O)C1CCC1)NC(C=C(C)C(F)F)=O 37453,c1(C(C(=O)NCCC)N(C(C)C(F)(F)F)C2CC2)ccc(I)c(C)c1 37454,CCS(=O)(=O)CC(=O)NC(C)(CNC(=O)C(c1c(C)nn(C)c1C)C)C1CC1 37455,CC1(CC(N2CCOC(CNC(=O)CNC(N3CCCC3)=O)C2)=O)CCS(=O)(=O)N1 37456,O=C(C1CCc2nccn21)NCCC1CN(C(c2ncc3c(F)cccn23)=O)C1 37457,c1(OC)cc(N)c([N+](=O)[O-])cc1C(=O)OC(Cc1ccccn1)C(N)=O 37458,c1(COCC(=O)NCc2cccc(CNC(=O)C3=CCC3)c2)cc(F)cc(F)c1 37459,c1(N2CCC(CNC(C(c3cccnc3)C)=O)C2(C)C)ccc([N+](=O)[O-])cn1 37460,C(=O)(CCCCCS(N)(=O)=O)NC1CCCCN(C(c2c[nH]c(=N)s2)=O)C1 37461,c1(OC(C(CC)C)C)cc(C#N)ccc1OC(=O)OC(C)(C)C 37462,CCCC(C(=O)NCC1(O)CCCN(C(=O)C2=NOCC2)CC1)S(N)(=O)=O 37463,C(C(C)(C(=O)N(C1(C(N2CCSC(C)C2)=O)CC1)C)OC)OC 37464,c1(CCNC(c2n(C(C)C)nnn2)c2csc(-c3ccsc3)n2)ncccc1F 37465,c1(CC(=O)NCC2C(NC(C(C)OCCC=C)=O)CCC2)cn2ccccc2n1 37466,c1(CNC(CN(C)Cc2cccc(C#N)c2)=O)nc2c(O)nc(=O)n(C)c2[nH]1 37467,c1(C(N2CC(NC(c3coc(Cl)n3)=O)C(O)C2)=O)nc2ccccc2o1 37468,N1(C(C(CC)(C)F)=O)CCC2(CC1)CN(C(=O)C=Cc1ncc[nH]1)C2C(C)C 37469,N1(C(CC(C)NC(c2coc(SC(C)(C)C)n2)=O)=O)CCOCC(C(=O)OC)C1 37470,N1(C(CCC(C)=O)=O)CCC(O)C(C(=O)Nc2cc(C(F)(F)F)cc(F)c2)C1 37471,N1(C(CCC(C)OC)=O)C2CCC1CC(NC(=O)CC13CCC(CC1)OC3)C2 37472,c1(SC)nccc(=NC2CC23CC(NC(c2csc(NC(C)=O)n2)=O)C3)[nH]1 37473,Cc1c(F)ccc(N)c1C(=O)NCC12CC(NC(=O)C3=CCC3)(C1)C(C)O2 37474,C(C(CC1CC1)C(=O)NCC1CCN1C(C)(C)C)NC(c1c(C)ccs1)=O 37475,C(C(=O)N=S(C)(=O)c1cnn2c1CN(c1ncnc(O)c1Br)CC2)=C(C)C 37476,c1(C(=O)NC)cc(C)[nH]c(=NCC2CCC(NC(=O)C(C)(C)CC(F)F)C2)n1 37477,N1(C(C(CC=C)C)=O)CCOCC(F)(CNC(c2nc(OC)ccc2OC)=O)C1 37478,CN=S(C)(=O)c1ccc(C(=O)NCC2CCCCC2NC(c2cccs2)=O)cc1 37479,CC1CN(C(C2CSCN2C(C2(F)CCCCCC2)=O)=O)CC2(CCC2)O1 37480,Cc1cnc(F)cc1C(N1CC(NC(=O)C(O)CCn2cncn2)C(C)C1)=O 37481,N1(C(C2=C(C)CCC2)=O)CCC(C)(C)C(CNC(C2CC(C)(C)OC2(C)C)=O)C1 37482,C1(NC(=O)COCC(=O)NCC)CC2C(NC(COCCCCC)=O)C2C1 37483,CC1=NOC(C(=O)NC(c2cn(CC3CCN(C(=O)CNC4CC4)C3)nn2)=O)C1 37484,c1(OC)c(OC)cc(C(=O)NCCC2CC(NC(C3CCC(O)C3)=O)C2)cc1Cl 37485,C1(NC(CC(C)(C)N(C)C(C2C=CCC2)=O)=O)CCCC(O)CC1 37486,N1(C(CC)=O)CC2CCC1CN2C(c1[nH]c(CC)cc1-c1ccccc1)=O 37487,N(C1CCCn2ncnc21)C(CC1CC(NC(C(CCC(C)C)O)=O)C1)=O 37488,c1(CCC(=O)NC(C)(C)CNC(C2(N=[N+]=[N-])CC2)=O)cccc(F)c1 37489,C1(CNC(C(C)=C(C)C)=O)CCC(C)(C)CN1C(c1ccc(NC=O)cc1)=O 37490,C1(CNC(CCCC)=O)CCC2CN(C(C3CCCCC3OC)=O)CCC2C1 37491,c1(C(=O)NCC(C)CNC(C2(N(C)C)CCC2)=O)ccc(C(N)=O)cn1 37492,C1(C(N2CCC(CC(C)NC(=O)CC3CCCCO3)CC2)=O)OCC2CCCC12 37493,CCC(CCOC)C(=O)N(CCNC(=O)C(C)(C)n1cccn1)CCOC 37494,CC1(C)CCCC(N2CCCC(n3ccnc3-c3ccc(C#N)cn3)C2)C1 37495,CCC(CC1CCCCC1)C(=O)NCC1CCN(C(c2ccnnc2)=O)C1 37496,C1(NC(=O)C(C2CC2)C2CC2)CCC2CCN(C(=O)C(O)c3ccsc3)C1C2 37497,n1(CC)c(C2CCCN2CC(N2CCC(CCCc3nnc(C)s3)C2)=O)nnc1S 37498,N1(C(Cc2c(C)nc[nH]2)=O)CC(NC(=O)Cc2cc[nH]c2)CC12CCCCCC2 37499,CCC(C)(CN)C(=O)NC1CCN(C(C2CC2c2cc(F)ccc2F)=O)CC1 37500,C(=O)(C(CNC(c1cc(C#N)cs1)=O)C(C)C)N1C(C)(C(=O)OC)CC1 37501,C12(C(=O)NCC(CC)(CC)NC(c3cccc(OC)c3)=O)CCCC1C2(F)F 37502,CC1(C)CCCC(C(=O)NCCC2=CCN(C(c3ccc(C#N)[nH]3)=O)CC2)CC1 37503,c1(C(N(CCC(C)NC(C2CCCCN2C)=O)C)=O)cnc(O)c2ncccc12 37504,c1(C(=O)NCC(C)N(C(CC2CCC(C)O2)=O)C)ncccc1Cl 37505,CCCC(O)C(=O)N1CCCC1C1CCCN(C(=O)COCc2ncc(C)o2)C1 37506,C(CS(=O)(=O)c1cccs1)NC(=NCC=C)NCCCNC(=O)OC(C)(C)C 37507,c1(C(N2C3CC(NC(C(CCC)OC)=O)C3CC2)=O)cccc2c1nnn2C 37508,N1(CCC)CCC(C(=O)NCC2(CO)CCC2)C1 37509,C(C(C(=O)NC1CN(C(=O)CCC2CCC2)C1)OC(F)F)OC 37510,C=CCC(F)(F)C(=O)NC1CCCC(N(C)C(c2ncncc2N)=O)C1 37511,C(CC#CC(C)(C)C)NC(C(CNC(c1cc(CO)on1)=O)N(C)C)=O 37512,C1(C(=O)O)C(NCc2cn3c(n2)COCC3)C2(C)CCCCC12 37513,c1(C(=O)NC(C(C)N(CC)CC)=O)cc(CC2(c3cc[nH]n3)CC2)on1 37514,c1(NC(C2C(OC)CN(C(=O)C3=CCCCO3)C2)=O)c(C)cc(O)nc1C 37515,CC1(CONC(=O)C2(C3CCCO3)CCC2)CCCO1 37516,c1(C(=O)NC(CNC(C2CC(OC)C2)=O)C)ccccc1C1(C#N)CC1 37517,C=CC1CCN(C(C2CCN(C)C2=O)=O)C1.C1(C)(C)C(=O)N1 37518,N1(CC(=O)NC2CCC2NC(c2cscn2)=O)C(=O)c2ccccc2C1=O 37519,C1(NC(c2cncc(C(C)C)c2)=O)CN(C(=O)C(F)=CC2CC2)CC12CCC2 37520,C1(OC)CC(CNC(c2cc(C)[nH]n2)=O)N(C(C2(CF)CC2)=O)C1 37521,c1(OC)ccc(C(=O)NC2CC23CN(C(=O)OC(C)(C)C)C3)c(Cl)n1 37522,c1(C(=O)Nc2cccc(CNC(C(C)N(C)C)=O)c2)cc2c(cc1N)CCCC2 37523,c1(CC(=O)NC2(CC=C)CCN(C(=O)C(O)CF)C2)cn2cc(F)ccc2n1 37524,c1(CC(=O)NC2CC(C)(NC(C(C)NC(CC)(C)C)=O)C2)ccc(OC)cc1C 37525,C1(C(=O)NCC2OCCCN(C(C3CNC(=O)N3)=O)C2)Cc2cncn2C(=O)N1 37526,C#Cc1ccc(CC(N2CCC(C(N3CC4CCCC3C4)=O)C2CC)=O)cc1 37527,C(=O)(C(C)(CC)CC)N(CC(CNC(C(CCC)=CCC)=O)O)C 37528,C(=O)(C(F)C(F)(F)F)NCCCC(CO)NC(C=CCOCCOC)=O 37529,FC(F)C(c1ccoc1)NCCC(Cl)Cl 37530,CC1CN(C(c2cc(Br)ccn2)=O)CCN1C(=O)Cc1cc[nH]c1 37531,C12(F)CCC(C1)N2.c1(C(N(C)NC(C(C)OCC)=O)=O)ccc(C2(C)CC2)cc1 37532,c1(C(C(=O)NCC(C)N(C)C(C2(F)CCCCC2)=O)C)cncc(F)c1 37533,C(=O)(C1CCc2c[nH]nc21)N1C(C)CN(C(=O)CSc2cnn(C)c2)CCC1 37534,N1(C(C2(CCOC)CC2)=O)CCCC(C(C)NC(=O)CC(C)(C)OC)C1 37535,c1(OC)ccc(CC(C)(C)CNC(=O)C(c2ccc(Cl)cc2)CO)cc1OC 37536,CC(C)CC(CNC(c1csc(F)c1)=O)C(=O)NCCN1CCOC1 37537,N1(C(C(C)NC(=O)OC)=O)CC2(CCCN(C(=O)CC3COCCN3C)C2)C1 37538,C(=O)(CS(=O)(=O)C1CCCC1)N(CCN(C(C(C)C1=CCCC1)=O)C)C 37539,Cc1cc(S(N)(=O)=O)oc1C(=O)NCCN(C(c1c(C)n[nH]c1C)=O)C1CC1 37540,N1(C(c2n(C)ncc2C#N)=O)CCC2(CC1)CCN(C(C1CC1CF)=O)C2 37541,c1(C(=O)NC2CN(C(C(C(=O)OCC)CC)=O)C2)cc(=O)n(C)c2ccccc12 37542,c1(C(N2CCC(N(C(CCc3cc(OC)no3)=O)C)C2)=O)c(Cl)cncc1Cl.C(C)=O 37543,C1(C(=O)NCCC(C)NC(c2cnoc2C2CCOCC2)=O)CC(Cl)(Cl)C1 37544,Cc1cc(C(=O)N(CC(=O)NC(c2cnsc2)C)C)nc(C)c1 37545,C1(CNC(C2CN(C(=O)NC)C2)=O)CN(C(c2cc(O)ncc2F)=O)CC1(F)F 37546,C(=O)(C1=CC2C=CC1C2)NCC(CNC(=O)C(C)(C)C1(O)CCC1)OC 37547,Cc1cc(NC(=O)C(F)C(C)CN(C)C(=O)OC(C)(C)C)cc(C)c1Cl 37548,c1(C(N2CC(CC=C)(NC(=O)CC)C2)=O)nccc(C)c1F 37549,C1(C(N(C2CCN(C(c3nc(Cl)cs3)=O)C2)CCC)=O)CCC(C)(C)O1 37550,CCC(C(=O)N1CC(C(N)=O)(CNC(=O)CC2(O)CCOC2)C1)C(C)O 37551,C1(C(N2CC(CCO)(OC)C2)=O)CN(C(=O)CCC2CC2)CC1(F)F 37552,c1(C(C(=O)NCC(C)(C)NC(C(C)OCC(C)C)=O)C)ccc(Br)s1 37553,C1(CNC(C2N(CC)CCC2)=O)CN(C(C2CSC2)=O)CCC12CCC2 37554,c1(CC(=O)NCC(CC=C)NC(c2n[nH]cc2Cl)=O)cnc2ccccc2c1 37555,c1(N2CCC(O)(COC)C2)cc(C)c(F)cc1[N+](=O)[O-] 37556,c1(C(NC(NCC(=C)C)=NCCC2CC2(Cl)Cl)C)ccc(C#N)cc1F 37557,Cc1nc(=N)[nH]c(C)c1C(=O)NCCC(C)NC(C1OC(C)CC1C)=O 37558,C1(C(=O)NCc2cc(F)cc(C#N)c2)C2C(CN1Cc1c(C)ccnc1)C2(C)C 37559,CC1=C(C(=O)N2CCN(C)C(CNC(=O)COC3CCOC3)C2)S(=O)(=O)CCO1 37560,C(CN=c1[nH]c(=NC2CC3C(C2)C3(F)F)[nH]c2c1SCC2)OCCN(C)C 37561,N1(C(C2(C)CC(=C)C2)=O)CC2CCCC(C1)N2C(C1CC1C(=O)OC)=O 37562,c1(SC)cc(C)c(C(=O)N(C2CCN(C(=O)C(C)C(C)C)C2)C)o1 37563,C=CC1(C(=O)Nc2ccc(O)c(=O)cc2)CCN(C(c2cc(=N)[nH][nH]2)=O)C1 37564,c1(OCC)nccc(C(=O)NC2CCCCN(C(C3CC=C(C)CC3)=O)C2)c1F 37565,c1(CC)cc(OC)ccc1C(N1CCC(CNC(c2c[nH]c(=N)o2)=O)C(C)C1)=O 37566,C1(=O)CCCCCN1.C1(C(N2CC(CC)(OC)C2)=O)(COC)CCOC1 37567,c1(N(CC(C2CCC2)NC(=O)OC(C)(C)C)C(C2CC(F)C2)=O)ccc(Cl)cc1 37568,c1(C(=O)NCC2OCC(CNC(c3ccc(O)nc3)=O)C2)ccc2nn[nH]c2n1 37569,c1(CNCCN2CCN(C(c3cccc(C#C)c3)=O)CC2)ccc2ccoc2c1 37570,c1(OC)ccc(C(=O)NC2CCCC(NC(C3CCCCC3O)=O)C2)c(C)c1 37571,c1(CS(N2CCC(C(CC)C#N)CC2)(=O)=O)ccc(Br)c(OC(C)C)c1 37572,N1(C(C(C)C)=O)CC2CS(=O)(=O)CC2(NC(c2cc3cc[nH]c(=O)c3o2)=O)C1 37573,O=C(CCN=c1[nH]ccs1)NC1CCC(NC(c2cc(Cl)cc(Cl)c2)=O)CC1 37574,C(=O)(C1CCC(N)c2ccccc21)N1C(COC(C)(C)C)CCCC1 37575,C1(C(=O)NCC=CCNC(c2scc(C)c2C)=O)CCC2(CCC2)C1 37576,N1(C(CCOCCCOC)=O)CCN(C(=O)CSCCc2ccccc2)C2CC12 37577,N1(C(C(=O)Nc2ccc(C)cc2Br)C)CCC(C2CC(O)C2)CC1 37578,N1(C(CC=CC=C)=O)CCC2CC2(C(N2CC(OC(C)C)C2)=O)CC1 37579,C1(N(C(=O)C=CC2CC2)C)CN(C(C2CCN(CC(F)F)C2)=O)CC12CC2 37580,CC1(C)CCC=C(C(=O)NCC#CCNC(C2CC23CCOCC3)=O)C1 37581,c1(CNC(C2N(C(c3c(CC)n[nH]c3)=O)CC3CC32)=O)cccc(F)c1O 37582,N1(C(c2cncc(NC(CC)=O)c2)=O)CC2(CC(NC(=O)C(C)CCCOC)C2)C1 37583,c1(C(N2CCCC(C(C)NC(CC3(OC)CC3)=O)C2)=O)nccc(C)c1N 37584,C(=O)(CS(=O)(=O)C(C)C)NCC1(NC(c2cc(C)cc(O)c2)=O)CCOC1 37585,CCCCC(O)C(=O)N1CCNC(C(=O)Nc2nc(F)ccc2Br)C1 37586,N1(C(C2(CC)CCOCC2)=O)CC2(CCN(C(=O)Cc3cnnn3C)C2)C1 37587,c1(N2CC(C(C)C)OCC2)[nH]c(=NCC2CC2C2CCOCC2)nc2scnc12 37588,N1(C(c2ccc(OC)nc2)=O)CCC2(COC(CNC(=O)CC(C)C3CC3)C2)C1 37589,C1(C)(CC(=O)CC2CN(C3CCN(Cc4c(C)cnn4C)C3=O)C2)CCS(=O)(=O)N1 37590,N1(C(c2n(C=C)ncc2)=O)CCCC(NC(C2CC3CC3C2)=O)CC1 37591,C#CCCCCCCC(=O)N(CCCCCC(=O)Nc1cnccc1N(C)C)C 37592,c1(OCC)cc(CC(F)(F)F)[nH]c(=NCCc2ccc(OC)c(OC)c2)n1 37593,c1(CC)cccc(F)c1C(=O)NCC1CC(NC(=O)CC2(C)CCCC2)C1 37594,Cn1c(C(=O)Nc2csc(Br)c2)cc2c(=O)n3ccccc3nc12 37595,c1(NC(C(=O)NCC(CC(C)C)C)=O)ccccc1S(C)(=O)=O 37596,N1(C(c2ccc(SC)o2)=O)CCCC(C2CN(C(c3cc(O)cc(O)n3)=O)C2)C1 37597,c1(C(=O)Nc2c(C(=O)NCc3n(C)ccn3)n[nH]c2)ccc(I)c(O)c1 37598,C1(CNC(=O)C#CC2CC2)C2CCC1CN(C(c1nncs1)=O)C2 37599,C(CC(F)F)(C(=O)NOCCC(C)C)N(C(CC(CC)CC(C)C)=O)C 37600,c1(OCC=C)cccc(CN2CCCC(C(=O)Nc3cscn3)C2)c1 37601,N1(CC(=O)NOC2CCCCC2)CC(O)C(O)CC2(CCOCC2)C1 37602,c12cc(C(F)(F)F)ccc1S2.[N-]=[N+]=NCCCNC(=O)C(=O)NCCC(F)(F)F 37603,c1(CC(=O)NCC2CCCC2NC(C2CCOC2)=O)c[nH]c2ccccc12 37604,C1(C(=O)NCCC2CN(C(c3ccc(-c4nc(C)sc4)s3)=O)C2)C2CC2C2CC12 37605,c1(OCC=C)ccc(C(N2CCOC(CCNC(=O)C=CC)C2)=O)cc1OCC 37606,c1(C(=O)NC(CC(C)NC(c2n(C=C)ncc2)=O)C)cc(Cl)c(N)c(Cl)c1 37607,C(=O)(CCCN=[N+]=[N-])NCC(CC)(C)NC(c1ccncc1Nc1nccs1)=O 37608,Cc1cc(F)c(C(=O)NC2(C3CCCN3C(=O)C(O)C(C)(C)C)CC2)cc1F 37609,n1(C(C)C)cc(CN2CCCC2COCC2CC2)c(I)n1 37610,N1(C(c2ccc(C3C(C)C3)o2)C(=O)Nc2ccccc2)CCN(C2CC2)CC1 37611,O=C1OCc2cc(NC(C3CC34CCN(S(=O)(=O)C(F)(F)F)C4)=O)ccc21 37612,N1(C(c2c(N(C(C)C)C)cccc2)=O)CCN(C(=O)CCCCF)C2CC12 37613,n1(CC)c(C(=O)NC2CCCC2NC(=O)C(O)C2CCC2)nc2ccccc12 37614,c1(NC(C(C)C)=O)ccc(OCC(C)NC(=O)NCc2cnn(C)c2F)cc1 37615,N1(C(C(C(CC)C)O)=O)CCC2(CC1)CN(C(=O)CN(C1CC1)CC)CC2CO 37616,c1(C(N2CCC(NC(c3c(N)cn(C)n3)=O)CC2)=O)cccc2ccccc12 37617,CS(=O)(=O)c1cc(C(=O)N=c2nc[nH]n2C2CCCN(C(=O)OC(C)(C)C)C2)cs1 37618,C1(C(=O)OC)CCC(C(=O)NC(C)(C)C(C)NC(=O)CCCN(C)C(C)=O)CC1 37619,Cc1ccc(S(=O)(=O)N(CC(=O)NCC(O)CNC(=O)CC2CCOC2)C)cc1 37620,c1(CC)c(C(N2CCC(C)C2C(=O)NCc2cnn(C(C)C)c2)=O)ccn1C 37621,c1(N2CCC(F)(C(=O)Nc3cc(OC)cc(Br)c3)C2)ncc2ccccc2n1 37622,N(C1CCCn2ccnc21)C(C1(C)CCCN1C(=O)CC1(O)CCOCC1)=O 37623,c1(C(N2CCC(O)(CNC(C(CC)(C)CC)=O)C2)=O)noc(C)c1[N+](=O)[O-] 37624,C1(NC(CC2CC(OC)C2)=O)CCC(CNC(c2cc(N(C)C)on2)=O)C1.COC 37625,C(=O)(CCCC(=O)c1ccc(C)cc1)N(CC(CC)O)C1CC1 37626,CCC(O)CC(=O)N1CC(C(=O)NCc2coc(C)c2)C(C)C1 37627,O=C1NCC(Cc2ncc(Cl)cc2O)c2ccccc21 37628,C1(NC(C(CCC)NC(=O)C(O)CC2CCCC2)=O)CC2(C1)CC(C)(C)C2 37629,S(=O)(=O)(c1ccc(N2CCC(CCF)CC2)c(F)c1)N1CCSC(C)C1C 37630,C12(NC(C(C(C)NC(C3N(CC)CCC3)=O)C)=O)CCCN(CCC1)C2 37631,C1(C(=O)NCc2cc(C(=O)NC3CN(C(N)=O)C3)n(C)n2)(OC)CCC(C)C1 37632,c1(C(N2CC(C)C(CNC(=O)CC3CSC3)CC2)=O)c(Cl)ccc2ccoc12 37633,C(C(CC1CC1)C(=O)NCCC1COCC1O)NC(CSC)=O 37634,Nc1cc(F)cnc1C(=O)NCCC1CN(C(=O)CC2CCCNC2=O)C1 37635,C(CCF)(C(=O)N(C)CCO)NC(c1n(CC#C)cnn1)=O 37636,c1(C(N2C(CC)CN(Cc3cc(C4CC4)no3)CC2)=O)cc2c(C)snc2s1 37637,C1(C2CC2)(CNC(c2cc(C)nc(O)n2)=O)CCN(C(=O)C(C)OCC(C)C)C1 37638,CCC(C)(C)CCCC(=O)NC1CCC2CCN(C(=O)CCC(C)(C)F)C12 37639,c1(C(=O)NC2C(C)CCN(C(=O)CC3CCCS3(=O)=O)C2)ccc(N=[N+]=[N-])cc1 37640,C1(CC(=O)N(C2CCN(C(C3C(C)C3)=O)CC2)CCO)COC2(CCC2)CO1 37641,c1(C(N2CC(O)(CCNC(c3cncc(CO)c3)=O)C2)=O)cnn2ccncc12 37642,c1(C(=O)NCCC2CC(NC(C3C(CC)C3)=O)C2)cnc(S)n1-c1ccccc1 37643,c1(C(=O)NC2C(C(=O)NC(C(=O)NC)CC(C)C)C2)cc(Cl)cc(Cl)c1[N+](=O)[O-] 37644,C(C(C(C)C(C)C)NC(=O)C=Cc1cnn(C)c1)NC(CC1CC(CC)C1)=O 37645,c1(OC)cc(C)c(NC(=O)CC2C=CC(NC(=O)CCCC(C)C)C2)cn1 37646,c1(CC)nc(C(=O)NCC2CC2C(=O)NCCCN=[N+]=[N-])c(C)o1 37647,c1(C(C)C)ccc2cc(NC(=O)C(N3CCC(F)CC3)=O)ccc2c1 37648,CC(C)(O)C(=O)NNC(=O)c1cc(C(F)F)cc(F)c1 37649,c1(C2(C(=O)NCCOCCNC(c3cn(CC)nn3)=O)CCC2)ccc(O)cc1 37650,C(=O)(CCC(C)(C)N(C)C)N1C(C(C)NC(c2cnnc(CO)c2)=O)CCC1 37651,c1(CC(=O)NCC2N(C)CCN(C(C(C(C)C)SC)=O)C2)ccc2occc2c1 37652,N1(C(c2c(F)ncc(-c3cccc(C#N)c3)c2)=O)CCC2(CC1)CC(=O)NC2=O 37653,Cc1cscc1C(N1CCC(CCN(C)C)C1)=O.N12CC(C1)C2=O 37654,N1(C(c2c(C)onc2)=O)CCC2C(CCCN2C(=O)CN2CCC(C)(C)C2)C1 37655,c1(C(=O)NCCC(C)(C)NC(c2ccc(NC(C)=O)s2)=O)csc2nnsc12 37656,c1(OC)nc(N2CCC(NC(=O)CCCC(C)O)C2)nc2[nH]cnc12 37657,C1(NC(CC(C)OC)=O)COCCN(C(=O)CNc2ccc(O)cc2)C1 37658,C1(C(=O)NC(CCOC)CNC(=O)C(C)(C)OC(C)=O)CC2(CCCC2)C1 37659,c1(CCC(=O)OC)ccc(Br)cc1OC(F)(F)F.C12(C)CC(C1)NC2=O 37660,C1(NC(C=CCC)=O)CC12CCC(NC(c1ccc(C(F)F)o1)=O)CC2 37661,C1(NC(CN(CC)CC)=O)CCCC(NC(=O)C(C(C)CC)OC)CC1 37662,C(C(C)(F)CNC(c1ccc(C)s1)=O)NC(C(C1CC1)SC)=O 37663,C12CS(=O)(=O)CC1N2.c1(CSc2ccnc(C(=O)OCC)n2)cccc(Br)c1 37664,c1(C(N2CC(CN(C)C(c3ccnn3C3CC3)=O)C2)=O)conc1C1CCC1 37665,c1(C(=O)NCC(C2CC2)NC(C2CC(C)(F)C2)=O)cc(F)cc2cc[nH]c12 37666,O=C(CCC(=O)C1CC1)NC1CCOCC1C(=O)NC1C(O)CC1O 37667,N1(C(C(C(C)(C)C)O)=O)CCC2(CC1)CC(NC(=O)C(C)(O)C(F)(F)F)C2 37668,C(C(O)C(C)(C)C)C1(NC(CCC2(O)CC(NC(=O)OC(C)(C)C)C2)=O)CC1 37669,n1(CC(=O)CC2(CN(C(CSCC)=O)C)CC2)cc(C2CC2)nn1 37670,O=C(C1CSc2ccccc21)N1CCCCC(Nc2nc(Cl)nc3sccc23)C1 37671,C(C#Cc1cn(CC2CCC(F)(F)CO2)nn1)NC(c1c[nH]nc1C(F)F)=O 37672,N1(C(C(CC)Nc2ccco2)=O)CCN(C(=O)C(C)n2cccn2)CCC1C 37673,C(=O)(C(C)C(C)(C)C)NCCC1(OC)CN(C(c2n(CC)c(O)nc2)=O)C1 37674,N1(C(CC(C)(C)C)=O)CC2CCC1C1CN(C(c3c(N)ccc(F)c3F)=O)CC21 37675,C1(C)(NC(C(C(C)C)NC(c2sccc2C#N)=O)=O)CCC(=O)NC1=O 37676,C1(C(=O)NCC(C2CC2)SC)C2CC2CN1C(=O)Cc1cnccn1 37677,C1(Nc2c(C)c(Br)ccc2F)CCN(CCCOC(C)(C)C)CC12CCC2 37678,c1(C(N(CCCNC(c2cccc(OCC)c2)=O)C(C)C)=O)cc2[nH]ccc2s1 37679,C(C(=O)NCC1(C(=O)O)CNCCO1)(C(C(C)C)OC)OC 37680,C1(C(=O)NCC(C2CCCN2C(=O)CCn2cccn2)(C)C)COC2COCC12 37681,C(=O)(CC(C)CC(C)(C)C)NC(c1ccccc1)C(=O)NCCn1ncc(C)c1 37682,c1(OCC)cccc(OC)c1-c1nc(C(=O)N(C)C)c(C)s1 37683,Cc1cccc2c1OC(C(=O)OCc1c(C(F)(F)F)nc(=N)[nH]c1Cl)C2 37684,Cn1c(C(=O)NCC(CO)NC(C2CCC(C(N)=O)O2)=O)cccc1=O 37685,c1(C(N(C2CNCC(C)C2)c2ncncc2I)=O)cccc2nccn12 37686,C1(COC)CC2(CCN2C(=O)CCC2CCCCN(C(=O)CC3CC3(C)C)C2)C1 37687,C1(C(=O)NCC(CN(C(=O)C(C)CC(F)F)CC)(C)C)CCOC(=O)CC1 37688,N1(C(C(CCC)NC(C2CCOCC2NC)=O)=O)CCC(C)(CCO)CC1 37689,C1(C(N(CCCN(C(=O)C=C2CC2)C)C)=O)CCC(O)C1 37690,c1(C(=O)NCCCCCN(C(C(=Cc2ccco2)C)=O)C)nnc(S)n1C 37691,CC1(C)CC(C(=O)NC2CN(C(CCC3CCC(C=O)O3)=O)C2)=NO1.C(C)(C)C 37692,C1(COC)CC(CNC(=O)C(C2CCOCC2)O)N(C(=O)CCC2OCCO2)C1 37693,c1(N(C)CCO)cc(C(F)(F)F)ncn1.N12CC(C1)CC(=O)NCC1C(C1)C2=O 37694,CS(=O)(=O)c1ccc(F)c(C(=O)NCC2(NC(=O)CC3CC=CC3)CCOC2)c1 37695,CC(C)(CNC(C1C=CCN1C(C1CC(=C2CC2)C1)=O)=O)CN=[N+]=[N-] 37696,C1(S(N)(=O)=O)(C(=O)NC2C(CC)CN(C(c3[nH]c(O)nc3C)=O)CC2)CCCC1 37697,C=CCC(CC(C)C)C(=O)NCC1CCN(C(=O)C2Cc3ccccc32)C1(C)C 37698,c1(OC(C2C(C(=O)OCC)C2)=O)ccc(N2CCOCC2)cc1 37699,c1(C(N(CC(CNC(c2ccc(CC)cc2)=O)O)C)=O)c(Cl)cccc1[N+](=O)[O-] 37700,C(=O)(C1CSc2ccccc21)NC(CC)CNC(=O)CC(C)(C)C(F)(F)F 37701,C(C)(N=c1[nH]c(=N)[nH]c(=NCc2cc(C(F)(F)F)nn2C)[nH]1)c1nc(CC)sc1 37702,N1(C(C(=O)NCC=C)C)CCOCC(C(=O)NCCn2nc(C)cc2C)C1 37703,c1(C(=O)Nc2nscc2C(=O)NC2CC(=C)C2)ccc2nc(O)n(C)c2c1 37704,CN1CCN(C(C2(C(=O)O)CC2(F)F)=O)CC1c1cc(F)cc(F)c1 37705,C(=O)(C(O)CC[S+](C)C)NCCOC1CCN(C(C(C)(C)OCC)=O)C1 37706,CN=c1nc(C(N2CCCC(O)(CCNC(C3CCCO3)=O)C2)=O)cc(C)[nH]1 37707,C1(=O)C(N(CCN)C(C)C)C(C)O1.CCOC 37708,Cc1oc(C(N2CCOC(CCNC(C3CC3CF)=O)C2)=O)cc1Br 37709,C(C(CC(F)(F)F)NC(C1CCCN1N=O)=O)NC(=O)Cn1cncn1 37710,C1(NC(=O)CCC2CC2)C2CC3CN(C(=O)CCCc4ccccn4)C1C3C2 37711,CC1CC(NC(=O)C=Cc2ccc(C(F)F)o2)CN1C(c1ccc(C#N)o1)=O 37712,c1(CN(C(c2cscc2Br)C(=O)NCCCF)C)ccc(S(C)=O)cc1 37713,C(=O)(CCC(CF)CF)N1CC(C)(C(=O)NC2CC3CCC2O3)OCC1 37714,S(=O)(=O)(c1ccc(C)c(Cl)c1)NCC1N(C(c2ccc(C)cc2)=O)CCC1 37715,c1(C(=O)NC(c2cccc(C)c2)CNC(C(CC#C)C)=O)ccc2c(c1)CC2 37716,C1(CNC(C(C)NC(C)=O)=O)CCN(C(C2CC2C(N)=O)=O)CC1C 37717,C1(C(=O)Nc2ccc(CO)s2)CCCC12CCN(Cc1cc(Cl)c(F)cc1F)C2 37718,Cc1nc(Cl)[nH]c(=NC(C)CC(C)NC(c2ccc3cnsc3c2)=O)c1F 37719,N1(C(CC=C)=O)CC(NC(c2ccc([N+](=O)[O-])cc2)=O)C(C2CC2)C1 37720,C1(C(C)(C)NC(CC2CN(C(C)=O)C2)=O)CCN(C(c2ncsc2C2CC2)=O)C1 37721,N1(C(CC2ON=C(C)C2)=O)CCC(CF)(NC(c2cc(C3CC3)ccn2)=O)C1 37722,c1(C2C(C(=O)NCC3CC(NC(CCSC)=O)C3)CC2)ccc(F)cc1 37723,C1(O)(c2cn(C(C(N3CC4(C(OC)CCS4)C3)=O)C)nn2)CCC(F)(F)CC1 37724,c1(C(=O)NCC(C)NC(c2cccnn2)=O)c[nH]c2cc(Br)ccc12 37725,c1(OCC)nc(C(=O)NC2(C(=O)NC(CN(C)C)CCO)CC2(C)C)co1 37726,c1(C(=O)NCCCN(C(C)C)C(=O)C2CC2)cc2n(n1)CCN(C)C2 37727,c1(N2CCC(C#N)C2)nc(N2CCC(C3CCCCO3)CC2)c2c(n1)CCS2 37728,c1(C(C(=O)Nc2ccccc2)N(C(C)C)C)cccc(Cl)c1Br 37729,N1(C(c2ccc(=N)[nH]c2)=O)C2CCC1(CNC(C1CCN(C3CC3)CC1)=O)CC2 37730,c1(CN2CC(NC(C3(F)CCCC=C3F)=O)C2)ccc2cc[nH]c2c1 37731,CCCC(C)CCCC(=O)NCCCOCCCNC(c1cn(CCO)nn1)=O 37732,Cc1ccc(CC(N2CC(OCCNC(=O)C(C)CF)C2)=O)cc1Br 37733,c1(C(=O)NCC(CO)NC(CC2N(C)CCCC2)=O)cc2c(F)cccc2[nH]1 37734,N1(C(C(C)=C2CC2)=O)CCC(CC(C)NC(=O)C(c2ncccc2F)(F)F)CC1 37735,c1(C(N(CC(CC)NC(=O)CCCNC(C)=O)C)=O)nccn2cnnc12 37736,N1(C(c2cc(C)on2)=O)CCCCC1CCCNC(c1cnc(O)o1)=O 37737,C1(NC(CC2N(C(CCC(C)OCC)=O)CCCC2)=O)CCC(C)(O)CC1 37738,C1(C(N(CCOCCN(C(C(C#C)(C)C)=O)C)C)=O)COC2(CCC2)CO1 37739,C1(C(N2CC(F)C(F)C2)=O)COC2(CCN(Cc3cncc(Cl)c3)CC2)C1 37740,Cn1nc(C2CC2)cc1C(=O)NCC1CCCC(NC(=O)COC(F)F)C1 37741,c1(C(=O)NCC(=O)NCC2CCC(NC(C3(OC)CCC3)=O)C2)cccc(C)c1 37742,CCC(C)(C)CCCC(=O)N1CC(CC(C)NC(=O)C(n2ccc(C)n2)C)C1 37743,c1(C(C(=O)NC(CC)C)N(C)C(C2(C)CC2)C)csnc1OC 37744,CC(C)CC(C(=O)N1CC2CC(NC(=O)CCC(C)(C)O)CC1C2)C(N)=O 37745,C1(CC)(CC)CC(NC(c2cnccn2)=O)CN1C(C12COCC1C2(F)F)=O 37746,C(=O)(C1=C2CCCN=C2NN1)N1C2C(NC(C3CC3C(F)F)=O)CC(C2)C1 37747,C1(S(N)(=O)=O)(C(=O)NC(C)CCNC(c2cn(CCN(C)C)cn2)=O)CCC1 37748,C1(C(=O)NC2CN(C(Cc3ccc(C)cc3)=O)CC(F)C2)C(O)C(=O)N(C)C1C 37749,N1(C(C2CC(F)(F)C2)=O)CCC(CCNCC2COCCO2)CC1 37750,CCCCCC(CC)C(=O)NCCCOCCC(N1CCN(C(C)C)C(=O)C1)=O 37751,Cc1cccc(S(=O)(=O)Nc2ccnn2C2CCCCC2)c1Br 37752,C1(Cn2c(C(C)C)ncc2)CCCN(C(=O)OCCCCSc2ccccc2)C1 37753,N1(C(CCCSC)=O)CCCC(O)C1.c1(CC(=O)NCC)nc(C)sc1C 37754,c1(C(=O)NCC(CC=C)NC(C2CCN(C(=O)CC)C2)=O)ccnc(OCC)c1 37755,C1(C(C)NC(=O)C=CCN(C)C)CCN(C(c2csc(C#N)c2)=O)CC1 37756,C(=O)(CC(C(C)(C)C)NC(=O)C(C)OC(C)C)NCC1(OCC)CC1 37757,C=CCC(C)(C)CC(=O)N1CCC(NC(C2(c3oncc3C)CC2)=O)C(C)C1 37758,C1(NC(c2[nH]cc(CC)c2)=O)CC12CCC(NC(=O)C(C1CC1)SC)CC2 37759,C1(O)(CNC(C(C)OCC2CC2)=O)CCN(C(c2nnn3c2CCC3)=O)CC1 37760,C1(CNC(CC=C=C)=O)C(C)CCN1C(c1nn(C)cc1Cl)=O 37761,C(=O)(CCCC(=O)NCC(C)CNC(c1cc(C)nn1C)=O)NC 37762,Cc1cc(C(=O)NC2CN(C(=O)Cn3nc(Cl)ccc3=O)CC2O)ccc1Cl 37763,c1(C(N2C(C(=O)Nc3n(C)ncc3Br)CSCC2)=O)cc2ccoc2cn1 37764,CC(C)(CCCNC(c1nc(Br)sc1Cl)=O)NC(C1CC1Cl)=O 37765,c1(CC(=O)NCC2CC2NC(C2CC2F)=O)c(F)cc(F)cc1F 37766,Cn1cncc(C(=O)NCCCN2CCN(C(=O)CCn3cccn3)CC2)c1=O 37767,CC1(OCCC(=O)NCCCOC2(CCCCO)CC2)CCC1 37768,c1(C(N2CCC(NC(c3cccn(C4CC4)c3=O)=O)C2)=O)ccn2ncccc12 37769,c1(C(=O)NC(CCN(C(COCC(=O)NC)=O)C)C)cnc(Cl)s1 37770,C(C(=O)NCCC1(NC(C2CCCC(C)O2)=O)CC1)(C(C)C)OC 37771,C1(NC(=O)Cc2nccs2)CCC2CN(C(c3cccc(Cl)c3)=O)CC2C1 37772,C12(CN3CC(C(=O)OCC)C3)CCCC1C2 37773,C(=O)(CC(C)C(C)(C)NC(=O)C(CC)C(C)C)NCC1(OCC)CC1 37774,c1(-c2nc(-c3cc(Cl)ncc3)nn2CC2CCOC2)cc(F)cc(F)c1 37775,O=C1CN(CC(N2CC(NC(c3cc(Cl)n[nH]3)=O)C(O)C2)=O)C(=O)N1 37776,N1(CC2(C(C)C)CC2)CCN(CCc2cccs2)CC1 37777,C1(C(N2CCCC(N(C(=O)C=CBr)C)C2)=O)CC(F)(F)CCC1(C)C 37778,c1(C(=O)NC2C(C)CN(C(=O)C=C3CCCCC3(C)C)C2)cnn2c1CCCC2 37779,C(=O)(CC(C)(C)c1cccc(Br)c1)NCC1(CNC(C2(F)C(C)C2)=O)CCC1 37780,c1(C(C(=O)OC)C)ccc(S(=O)(=O)NCc2c(N(C)C)cccc2C)cc1 37781,C12(C(N3CCN(C(C4CCO4)=O)CC3C3CC3)=O)C3C4C1C1C2C3C41CO 37782,c1(C(=O)NC2(CNC(C(C)C3CC3)=O)CCC2)n[nH]c2c1COc1ccccc1-2 37783,C1(CC=C)(NC(=O)CC2CCCC2O)CN(C(=O)CCC2CCC(C)O2)C1 37784,CC(C)C(CCN(C(=O)C(C)C(F)F)C)NC(=O)Cc1ccc(Cl)cc1 37785,c1(C(C(=O)NCCOC)N(C2CCC(F)(F)C2)C)ccc(F)c(Br)n1 37786,Cc1ccc(C(N2CCC2CNC(C2CCCC2C)=O)=O)c(N)c1C 37787,c1(OC)ccnn1C(C)(C)OC(=O)NC1CC1C1CCCC1 37788,N1(C(=O)CCC2CCCO2)CC2CCC(C1)N2C(=O)CC1CC2CC2C1 37789,N1(C(c2ccsc2C(F)(F)F)=O)CC2(C1)CN(C(c1ccnc(F)c1)=O)CCO2 37790,C1(C(N2C(CN(C(C(C=C)(C)O)=O)C)CC(F)C2)=O)C2CCC1(C)C2(C)C 37791,CC1C2C(CCN2C(=O)CCc2cccs2)CN1C(C12CSCC1C2)=O 37792,C1(CNC(c2c(C)cco2)=O)CN(C)CCN1C(=O)COCCO 37793,c1(C(=O)NC2C(CNC(C(CCCC)O)=O)CC2)cc([N+](=O)[O-])ccc1O 37794,C1(NC(c2c(O)cccc2O)=O)CCCC12CCN(C(C1CS(=O)(=O)C1)=O)CC2 37795,N1(C(CC2CC(=C)C2)=O)CCN(C(=O)C(N2CCOC2=O)C)C(CC(C)(C)C)C1 37796,c1(C(=O)NCC2C(NC(c3c(C)ncc(C)c3)=O)C2)cc(Cl)cc2c1OCC2 37797,CS(=O)(=O)c1ccc(C(N2CCC(NC(=O)CO)C(CO)C2)=O)cc1Br 37798,c1(C(N2CC(CCn3cc(C4CCCO4)nn3)C2)=O)cnc(S)[nH]1 37799,C1(C(N2CC(CC(=O)NCc3nccc(OC)c3)OCC2)=O)CC(=O)OC1(C)C 37800,c1(CC(=O)NC2CC3(C(NC(C(CC#C)O)=O)C3)C2)ccc(Cl)cc1F 37801,C(=O)(C(CNC(=O)CN1CC(C)(C)C1)C(C)(C)C)NCCc1c(C)ncs1 37802,CCCCCCn1nnnc1C(c1cnn[nH]1)NCc1ccc(Br)o1 37803,CC1CN(C(=O)CC2NC(=O)NC2=O)CC(C)CN1c1nnc(-c2ccon2)s1 37804,Cc1c(C(=O)NC(C)C(C)NC(c2c(Cl)ccc(Cl)c2O)=O)sc2ccccc12 37805,C(CC(=O)Nc1cccc(C(N)=O)c1)(C(F)F)NC(CN(C(C)C)C)=O 37806,Cc1cc(C(=O)N(C)CCOCCNC(C2CC(F)C2)=O)cc(C)c1N 37807,C1(CNC(CC(C)(C)SC)=O)CC12CCN(C(=O)Cc1cccnc1C)CC2 37808,C1(C)(C(=O)NC2C(NC(c3cccc(N(CC)CC)c3)=O)C2)CCC(=O)NC1 37809,C(=O)(C(F)(CC)C(=O)OC)N(CC(C)NC(c1c(CC)occ1C(F)(F)F)=O)C 37810,c1(C(N2CCC(C)(NC(C3CCC(C)C3)=O)C2)=O)cc2c(s1)CN(C)CC2 37811,N1(C(CCCC(=C)C)=O)CCCC2(C1)CN(C(=O)CC1CCCCC1(F)F)C2 37812,c1(C(C(=O)NC(CC=C)CNC(=O)C(F)CC)(C)C)ccc(Cl)cc1F 37813,N1(C(C2CC(C#C)(O)C2)=O)CCN(C(C2(C(O)C(F)(F)F)CCC2)=O)CC1C 37814,c1(C(=O)NCc2ccc(C(NOC)=O)o2)ccc([N+](=O)[O-])[nH]1 37815,N1(C(C(CC#C)C2CC2)=O)CCC(F)(F)C(C(=O)NC(C)(C)C#CCCCCC)C1 37816,c1(OC(C)C)ccc(Cl)cc1C(=O)NCCC(C)NC(=O)CC1CC(=O)C1 37817,C1(NC(c2scc(OC)c2)=O)CN(C(c2cc(SC)cc(F)c2)=O)CCC1(C)C 37818,N1(C(C2CC(C)OCC2)=O)CCCCC2(CCOCC2)C1 37819,C1(NC(CC2(COC)CCCC2)=O)CCC(NC(c2nscc2N)=O)CC1 37820,c1(C2(NC(C3CCC(C(=O)NC(C4CCC4)C)C3)=O)CC2)cc(F)c(F)c(F)c1 37821,c1(C(N2CC(CNC(c3nc(C(C)=O)sc3)=O)C(C)C2)=O)c(C)nc(C)nc1C 37822,CC(CCC(=O)N(C)C)c1cn(-c2ccc(C(=O)Nc3cccc(F)c3)cc2)nn1 37823,C1(CNC(Cc2cc(C(C)C)no2)=O)(CNC(=O)CC2CC23CC3)CC12CCC2 37824,c1(C(=O)NC2CC(NC(C(CC)n3ccnc3)=O)C2)n[nH]c(C)c1Cl 37825,Cc1cnn(C)c1CC(=O)NCCC(C)CCNC(c1ccnn1C1CCC1)=O 37826,C1(C(N(CCC)CCO)=O)CN(C(=O)CC(C)C(C)C)CCC1(C)C 37827,C#CCC(C)C(=O)NCCC1CCCN(C(=O)C(C)(C)Oc2ccccc2)C1 37828,N1(c2cc(CC)ncn2)C2CCC1C(C)C(NC(c1c(C)noc1C)=O)C2 37829,c1(C(N2CCCN(C(C(=O)NCC)=O)CC2CO)=O)[nH]c2ccc(F)cc2c1C 37830,N1(C(C)=O)CCCCC1CC(=O)N(CCNC(=O)Cc1ccccc1)CC1CC1 37831,N1(C(C2C(OC(C)=O)C2)=O)CCN(CC(C)NC(c2cc(C)c[nH]2)=O)CC1 37832,c1(CCC(=O)NC(C(C)NC(CCOCC)=O)CO)ccccc1[N+](=O)[O-] 37833,N1(C(CCSCCCC)=O)CCC2(CCC2NC(=O)CN(C)C(N)=O)CC1 37834,C1(NC(C(C(C)C)n2ccnc2)=O)CN(C(c2csc(Cl)n2)=O)CC2(CCC2)C1 37835,c1(C(N2CCC(CCCC)C2(C)C)C(=O)NCC(=C)C)cc(Cl)c(Cl)c(Cl)c1 37836,C(=O)(C(C)(C)N1CCCC1)N(C(C)CNC(=O)CCOCCN(C)C)C 37837,C1(C)(C(=O)NCC2C(NC(c3c(CC)con3)=O)CCC2)CC(C(F)(F)F)=NO1 37838,c1(OC)cc(C(N2CCC(N(C)C(c3c[nH]c(=N)o3)=O)C2)=O)cc([N+](=O)[O-])c1Cl 37839,C1(C)(C(N2CC(C)(NC(C3C(C(C)C)(CC)C3)=O)C2)=O)CCN(C)C1=O 37840,c1(CC)ccc(C=CC(=O)NCCC(C)N(C(=O)Cn2cncn2)CCO)o1 37841,N1(C(c2c(C)cc(Br)cc2F)=O)CCC2CN(C(c3ccc(O)cn3)=O)CC2C1 37842,C1(NC(COCC(C)(C)C)=O)CN(C(C2CCOC(=O)CC2)=O)C(C)(C)C1 37843,c1(C(N2CC(C(C)NC(c3cc(O)no3)=O)OCC2)=O)cccc2oncc12 37844,c1(C(=O)NC2CN(C(CCCCC)=O)CC2C)ccc2c(c1)C(C)CO2 37845,C1(O)(C(N(CCNC(C2C(C(=O)OC)CCC2)=O)C2CC2)=O)CCC(C)(C)CC1 37846,C1(C(=O)NC(c2cnn[nH]2)C)CCCN1NC(=O)c1c(Cl)cnn1C 37847,CCCC(C)(O)C(=O)NCC(CC1CC1)C(=O)N(CC(C)C#N)C 37848,C1(CNC(C=C(C)C2CC2)=O)C2CCC(C2)N1C(=O)CC1(O)CCCC1 37849,C(CS(=O)(=O)C1CCOCC1)NC(C(N)Cc1ccccc1F)=O 37850,C(c1ccc([N+](=O)[O-])cc1)=CC(=O)NCC1C(CNC(c2[nH]c(=NC)sc2)=O)C1 37851,N1(C(CC(C)C(F)F)=O)CCN(C(=O)C(F)OC(F)(F)F)CCC1C 37852,c1(C(=O)NCCCC(C)NC(c2ccnc(C#N)c2)=O)ccn2ncnc2c1 37853,C1(C(=O)NCC2C(NC(c3ccc(CCC)[nH]3)=O)C2)CC(=O)N(CC(F)(F)F)C1 37854,N1(C(C(=O)N(C)C)=O)CC2(CCC2NC(=O)CC2CCCC23CC3)C1 37855,C(C)(c1ccccc1)=CC(N1CCC(C)(CC(N2CC(C)(CC)C2)=O)C1)=O 37856,C(=O)(CC(F)(F)F)NC(C)(C)C.C12CCC(C1)CN(C)CC(=O)N2.C1(=O)CCN1 37857,c1(C(c2n(CC)nnn2)NCc2cncc(Br)c2C)cccc2c1OC(F)(F)O2 37858,C1(NC(c2ccc3c(n2)NCC3)=O)CCN(C(C2CCCS2(=O)=O)=O)C12CCC2 37859,C1(C2CCC2)(CNC(C2C(C)OCC2)=O)CCN(C(c2cccc[n+]2[O-])=O)CC1 37860,CC1CC(CCNC(C2(C)CC2)=O)CCN1C(=O)Cn1ncnn1 37861,CCC(CC(=O)N1CCCC(CCNC(C2(C3CC3)CCCO2)=O)C1)C(C)C 37862,N1(C(CC2CC(C)(C)CN2C(C2CCC(=O)C2)=O)=O)CCOCC(C)(O)C1 37863,N1(C(c2occ(C)c2C)=O)CCOC(C)(CNC(=O)CSCCC(C)C)C1 37864,C=CCCCCCCCCNC(C1CCCCNC1=O)=O 37865,c1(CC(=O)N(CC(C)CNC(=O)C=Cc2ncco2)C)cn2cc(F)ccc2n1 37866,C(=O)(C(O)C(F)F)NCCC1CC(NC(COCC(=C)C)=O)C1 37867,c1(C(=O)NCC2CC(CNC(c3cc(Cl)no3)=O)C2)sc(F)cc1Cl 37868,C1(CN(C=O)CC)(CN(CCCCOC)C)CCCC1 37869,c1(C(=O)NCC2C(C(=O)NC3CC(COCC)C3)CCC2)cccc(C#N)c1C 37870,C1(C(=O)NCC#CC2CC2)(COC)CN(C(=O)CCC2CCCCC2)C1 37871,c1(C(N2CC(NC(c3cc(COC)[nH]n3)=O)C(F)CC2)=O)ccc2c(c1)CCC2 37872,c1(NC)c(C(=O)N(C)CCNC(=O)Cc2ccc(Cl)nc2)sc2nccnc12 37873,c1(C(N2C(C(=O)NCCCC=C)CC2)=O)nccnc1N 37874,c1(C(N2CCC(CN(C(C3C(C(C)=O)C3(C)C)=O)C)CC2)=O)ncnc(C)c1C 37875,CC(C)(C)CC(C(=O)N1CC(OCCO)C1)NC(=O)CC(C1CC1)C1CC1 37876,C(=O)(C1COc2ccccc21)NC(C1CCN(C(=O)CSC2CC2)CC1)CN 37877,c1(C(N2CCC(N(C(=O)CCOCCOCCO)CC)C2)=O)nnn(CC)c1C 37878,c1(C(=O)NC)ccc(OCC(=O)NC(C)CC(C)NC(=O)C=C(Cl)Cl)cc1 37879,Cc1ccc(C(N2CC3CC2C3CNC(C2CN(S(C)(=O)=O)C2)=O)=O)cc1CO 37880,CC1(C(N2CC(O)(CCNC(C3C4COCC34)=O)C2)=O)CCCS1 37881,C(C)(CN=c1[nH]nc(C(C)(C)C)o1)Oc1c(OC)c(OC)ncn1 37882,n1(CC(=O)N(CC)CC)nc(C)c(-c2cscn2)c1C 37883,C(C)(CC(C(=O)Nc1c(C)cccc1C)N1CCN(CC2CCC2)CC1)SC 37884,c1(CC(=O)N(C2CCCCN(C(=O)C(O)C3CC3)C2)C)ccc2occc2c1 37885,c1(-c2c(C(=O)NCC3C(NC(CC(=O)OCC)=O)C3)c[nH]n2)ccccc1Cl 37886,Cc1nc2sccn2c1C(N1CCC(NC(=O)CC2CC2(Cl)Cl)C12CC2)=O 37887,C1(CCNC(C=CC(=O)OCC)=O)CSCCN1C(=O)CS(=O)(=O)NC 37888,c1(C(=O)NCC(C(C)C)NC(=O)C(C)Cc2cccc(F)c2)ncc[nH]c1=O 37889,c1(-n2c(=O)c2=O)ccc2c(c1)CCC(C)C2.n1(CC(C)C)nccc1C1CC1 37890,Cc1cc(C(=O)N(CC(C)NC(=O)Cn2nccn2)C)c2c(Br)cccc2n1 37891,C1(OCC=C)CCC(NC(C)(C)CCCN)CC1 37892,c1cc2[nH]c(=NCC3SCCS3)nc(-c3ccccc3)c2[nH]1 37893,c1(C(=O)NCc2ccc(-c3cnc(O)nc3O)nc2)ccc(I)cc1[N+](=O)[O-] 37894,c1(OC)ccc(CC(=O)NC(C2CN(C(=O)CN3CCS(=O)CC3)C2)C)c(Cl)c1 37895,N1(C(CCCCOC)=O)CCN(C(c2cc(CC(C)C)on2)=O)C2CC12 37896,Cc1cc(C(N2CCOCC2C(N2CCOCC(O)C2)=O)=O)cnc1C 37897,c1(CC(C(=O)NCC2(CCNC(C3(OC)CC3)=O)CC2)C)c(C)nn(C)c1C 37898,c1(C(=O)NC(CNC(CCc2ccnc(C)n2)=O)C)cn(C2CC2)c(C)cc1=O 37899,CC(C)(C)C1=NOC(CNC(=O)NCc2cccc(OCCF)c2F)C1 37900,CC(C)(C)CC(=O)N1CCC1(C)C(=O)NCCOc1ccc(Cl)cc1 37901,C(C)(C(=O)N1CC(NC(c2ccc(CN(C)C)nc2)=O)C2(CC2)C1)(C(C)C)OC 37902,C(=O)(CCC(C)(C)C)N1CC(NC(CCCCOC(C)C)=O)C(n2ccnn2)C1 37903,N1(C(C2C(C)CCOCC2)=O)CCC(C(=O)NCC(C)(C)C#N)C(C)(C)C1 37904,N1(C(C(c2cnn(C)c2)OC)=O)CC(C)(CNC(=O)CCCCSC)CC1(C)C 37905,CC(C)CCC(O)C(=O)NC(CC1CCC1)C(=O)NCc1cccnc1Cl 37906,S(=O)(=O)(c1ccc(NCc2ccncn2)c(Cl)c1)NCC(C)(C)CCCO 37907,c1(C(N2CC(NC(C3C(C)OCC3)=O)C2)=O)ccc(=O)n(-c2ccccc2)n1 37908,Cc1ccc(NC(C2(CNC(=O)CCCC3CC3)CCCCC2)=O)cc1C 37909,c1(C(=O)NC2CCN(C(C(n3ccc(Br)n3)C)=O)C2)ccc2ccccc2n1 37910,CC(C)C(C)(C)C(=O)NC1CC(NC(c2c[nH]nc2[N+](=O)[O-])=O)C1 37911,c1(N(C)CC2(CC)CC2)nnc(-c2csc(C)n2)n1CCCc1ccccc1 37912,C1(=O)C(CC(C)C)NC(=O)C2CCN12.C(=O)(CCCC1CCC1)N(CC)CC 37913,c1(C(=O)NCC(CCCC)NC(C2(CC#C)CC=CCC2)=O)cc(F)ccc1N 37914,c1(C(=O)NC2C3(CC(NC(C(CCSC)O)=O)C3)C2)cc(Cl)ccc1O 37915,Cc1cnc(NC(C2CC(F)CN2Cc2cc(F)ccc2I)=O)nc1Cl 37916,C(=O)(CC(CNC(=O)N(C1CCCCC1)CCOC)C(C)C)NC 37917,c1(C(C)OC)nc(N2CCC(CNC(C3CCC(N=[N+]=[N-])C3)=O)C2)cc(Cl)n1 37918,C(=O)(CN=c1cc[nH]cc1)N1CC(CC(N2Cc3c[nH]nc3C2)=O)OCC1 37919,N1(c2ncc(C(=O)OC)c(C)n2)CCC2(CCCN(C(c3cccn3C)=O)C2)C1 37920,CCCCC(CNC(=O)COCCCOC)NC(=O)CC1CCS(=O)(=O)C1 37921,CCC(CNC(C12COCC1CN(C(=O)C1=CCN(C)C1)C2)=O)CC(C)C 37922,c1(C(N2CCC(O)(CN(C)C(c3cc(F)n[nH]3)=O)C2)=O)[nH]c2ccccc2c1Cl 37923,C=CC1(C(=O)NO)CCN(C(c2cscc2OC)=O)CC1.c1ccc(C)cc1 37924,C12(C(N(CCCNC(=O)CC3COC(=O)N3)C3CC3)=O)CC1Cc1c[nH]nc12 37925,CC1(C)CCOC(CC(=O)NCC2CCCCC2NC(=O)CCc2cocn2)C1 37926,C1(CCC)CN(C(c2cc(N)ccn2)=O)CC1NC(=O)CCCOCC 37927,N(C(=NCC1CC1)NC1CCN(CC2CCCC2)C1)Cc1nnc(C)s1 37928,c1(C(N(C)CC)=O)cccc(C(=O)NCC2CN(C(=O)C(C)COC)CCO2)c1 37929,CCCCCC(C)NC(=O)CC1CCC(NC(=O)CCCC2CCCC2)CC1 37930,C(=O)(CC(F)(F)CS(C)(=O)=O)N1CCC(C(C)NC(c2n(CC)cnn2)=O)C1 37931,c1(C(N(CCCNC(C2CC(c3ccccc3)O2)=O)C)=O)cccc2nccn12 37932,C(=O)(C1CCc2c[nH]nc21)N(C1CCCN(C(=O)CCc2cccs2)C1)CCO 37933,c1(NC(=O)CC2CC(NC(C3(O)CC3)=O)C2)cc2nccn2c(=O)[nH]1 37934,N1(C(C=CC)=O)CCN(C(=O)C(C(C)(C)C)N(C)C(=O)OC(C)(C)C)CC1C 37935,c1(C(CNC(=O)C(O)C2CC2)NC(c2c(C)n(C)nc2)=O)ccc(F)cc1F 37936,C1(C(N(CCCCNC(Cc2ccc(C)o2)=O)C)=O)CCn2nncc2C1 37937,c1(C(N2CC3(OCC(NC(CCC#C)=O)C3)C2)=O)cc(C)c2c(c1)CCC2 37938,CN1CCc2c(C(N3CCCC3C(=O)NC3CC(F)(F)C3)=O)cccc21 37939,c1(C(=O)NCC2(CNC(C3C(CC)OCCC3)=O)CC2)cn2c(n1)C(C)CCC2 37940,N1(C(CSCCN(C)C)=O)CCC(N(C)C)(CNC(C2CCCSC2)=O)C1 37941,c1(CC)ccc(C(=O)NC(C)CNC(=O)CCC2CCOCC2)cc1S(C)(=O)=O 37942,c1(C(=O)NCCN(C(C(CCC#C)O)=O)CC2CC2)cnc(O)c2cccnc12 37943,C(=O)(CC(CC)C(C)(C)C)N1CCC(CC(=O)Nc2ccc(C=C)cc2)C1(C)C 37944,c1(CC)cc(=NC(=O)C(CN(C)C(C2(C)CC2)=O)CC(C)C)[nH]n1C 37945,C(=O)(C(CCC)C(=O)OC)N1CCC(C)(CCNC(C2(CC#C)CCCC2)=O)C1 37946,N1(C(C=NOC)=O)CC2CC(NC(c3cc(O)ccc3Br)=O)C(C2)C1 37947,N1(C(CC2(C)CC2(Cl)Cl)=O)CCC(c2cccc(F)c2)C(NC(=O)C2CC2)C1 37948,c1(CC(N2CCCC(CNC(=O)CC3(O)CCOCC3)C2)=O)c(F)cccc1F 37949,c1(C(=O)NC2CCCC(C(=O)N(C3CCOCC3)CC)C2)ccc2c(c1)CCCS2 37950,c1(CC(N2CCCCC(NC(C3CCCS3)=O)C2)=O)cnc2cccnn12 37951,c1(CC)nc(C(=O)N(CC(C)(C)NC(c2csc(-c3ccco3)n2)=O)C)n[nH]1 37952,C1(C(N(CCCOC)C)=O)(NC(C2CON(C)C2=O)=O)CCCCC1 37953,c1(C(N2CC(NC(CCCC(C)=O)=O)CC2(C)C)=O)cc2ccc(F)cc2[nH]1 37954,N1(C(c2c(CC)nccn2)=O)CCC2CCC12CNC(c1cccc(Cl)c1O)=O 37955,N1(C(c2cccc(C)c2O)=O)CC(N=[N+]=[N-])CC1C(=O)NCC(O)C(N)=O 37956,c1(-c2ccc(CNC3(CO)CC4(C3)OCCO4)cc2)nccc2ccc(Br)cc12 37957,Cc1cc(Cl)c(C(=O)NNC(=O)C2CC(=O)N(c3ccc(F)cc3)C2)c(Cl)c1 37958,C(=O)(C(C)(C)CO)NC(c1n(C)ccn1)c1ccccc1 37959,CC(C(=O)NCCC1CCN(C(c2ccc(Cl)cc2)=O)C1)C(F)F 37960,C12(NC(C3(CC=C)CCC3)=O)CC1CN(C(C1(CN(C)C)CCCC1)=O)C2 37961,N1(C(CC2CC(OC)C2)=O)CCCC(F)(CNC(=O)C(C)(C)c2ccccc2)C1 37962,c1(CCNCC2CCC(C(CC)(C)C)CC2)cnc2c(Cl)cnn2c1 37963,N1(C(CC2N(C)CCC2)=O)CCC(C)(C)C1CC(=O)NOCCc1ccccc1 37964,Cc1cc(C(F)F)n(CC(N2CCCCC2C(C)NC(=O)C(C)(C)CO)=O)n1 37965,N1(C(C(C(=C)Cl)(C)C)=O)CCC2CC(C1)CN(C(=O)C#CC1CC1)C2 37966,c1(C(N2CCC(O)(CNC(c3cc(CC)c(C)s3)=O)C2)=O)ccc(N)c(Cl)c1O 37967,C1(CNC(c2nocc2Cl)=O)CCC2CN(C(=O)CCc3cncs3)CC12 37968,c12ncccc1C(=O)N(C1CCC1)C2.Cn1nccc1C(=O)NCC#N 37969,CCCCCCCC(=O)N1CC(CC(=O)NCCCCN(C)C)C2(CC2)C1 37970,C1(CCC)CCC(C(=O)NCCC2CN(C(c3ccc(C4CC4C)o3)=O)C2)CC1 37971,c1(C(=O)NCC2(O)CCN(C(C3(CSC)CC3)=O)C2)c[nH]c2cc(C#N)ccc12 37972,C1(NC(CC(C=C)C)=O)CN(C(=O)Cc2nnc(C)o2)C2(CCCC2)C1 37973,C1(C)(CC)CC(C(=O)NC(Cc2ccoc2)CO)CCO1 37974,C1(CC)CN(C(c2ccnc(C(C)(C)O)c2)=O)C(C)CO1 37975,CC(C)(C)C(C(=O)NC1CCC(Oc2ccccc2)CC1)C1CCC1 37976,C12(C(=O)NCC3C(NC(C(C)N(C)C)=O)CCC3)CC(CO1)C2 37977,c1(C(=O)NCCC2N(C(c3ncn(C)c3)=O)CCC2)cnn(C)c1S(C)(=O)=O 37978,N1(C(CC(C)O)=O)CC2CCC(C1)C(NC(C1CC(n3cccn3)C1)=O)C2 37979,c1(C(N2CCC(CNC(C3SC4C=CC3C4)=O)CC2)=O)cccnc1C(F)(F)F 37980,c1(-c2nccc(OCC3C(OC)CCN(C)C3)c2)nc2cc(Br)ccc2n1C 37981,C(C1CC1)(C1CC1)=CC(=O)NCC(C)N(C(c1cc(SC)oc1C)=O)CC 37982,C1(CNC(C2CN(C)C2)=O)CCCCC1NC(c1ccnn1C1CC1)=O 37983,c1(C(=O)NC2CC3CC(NC(CCCC=C)=O)C3C2)c(C)nn(C)c1OC 37984,C=CC1CN(C(C2(N(C)C)CC2)=O)CC1NC(=O)CNC(=O)CCC 37985,N1(C(C2(C#N)CC=CC2)=O)CCC(NC(c2ccc(Cl)s2)=O)C(CO)CC1 37986,C(=O)(CCCCC(F)(F)F)NC(CNC(C=C1CCC(C)C1)=O)C1CCC1 37987,c1(C(=O)NC2(C)CN(C(C3C(C)(C)C3(F)F)=O)C2)ccc2c(c1)OCC(=O)N2 37988,N1(C(C(C2(O)CCC2)NC(CCCCCC)=O)=O)CC(F)(F)CCC1C 37989,N1(C(CN(CCOC)C)=O)CCC(NC(c2cccc(OC)n2)=O)C2CC12 37990,c1(C(=O)NC2C(NC(C(C)(CO)OC)=O)C2)cc2c(s1)CCCNC2=O 37991,N(C(=S)N1CCN(C)CC1(C)c1ccccc1)Cc1c(C)cccc1 37992,C12(C(=O)NC(C3CCN(C(C4CCC=CO4)=O)CC3)C)CCC(CC1=O)C2 37993,N1(C(CCCC2C(C)C2)=O)CCCN(C(c2cc(O)nn2C)=O)CC1C 37994,c1(CNC(=O)NCC(F)(F)F)ccc2c(c1)CCN(C(=O)CN1CCCC1=O)C2 37995,C12(NC(=O)CCSC(F)(F)F)CCCN(C(c3ccc(F)o3)=O)CC1C2 37996,CC1CN(C(=O)Cc2ccoc2)CC(CNC(=O)Cc2cnn(C(C)(C)C)c2)O1 37997,c1(CNC2CCC(C)(C(=O)OCC)C2)c(F)cc(Cl)cc1Cl 37998,c1(N2CCOCC(NC(c3cnn(CC)n3)=O)C2)ncc(Br)cc1C#N 37999,C(=O)(C(CC)C(C)C)NCC1CC(OC)CN1C(c1ccc(CO)nc1)=O 38000,Cc1cc(Cl)cc(C(=O)NC(CNC(=O)CCS(C)=O)CO)c1N 38001,c1(C(=O)NCC(CNC(c2cn(-c3ccccc3)nn2)=O)OC)ncccc1Cl 38002,C1(CNC(CCC2(C)N(C(c3n(C)ncc3)=O)CCC2)=O)CCCCC1(C)C 38003,CCC(C)C(C)CN=c1[nH]c(=NCCCc2nncs2)c2cc(Cl)ccc2[nH]1 38004,c1(C(=O)NC2CC(C(C)NC(c3cn[nH]c3)=O)C2)ccoc1Br 38005,C1(C(C)=O)CC1(Cl)C(=O)NCCCOCCCNC(=O)CNC(=O)CN(C)C 38006,C1(C)(CNCc2nc(C)n(C)c2C)CCCC(C)(C)C1 38007,N1(C(=O)CC2CC3CC3C2)CCN(C(c2cnc(C3CCC3)o2)=O)C(CCO)C1 38008,c1(C(N(CCCNC(C2COCC(C)O2)=O)C2CC2)=O)cc(C#N)ccc1O 38009,CCCCCC(O)CC(=O)NC1CCC(CNC(=O)CCCN(C)C(=O)OC)C1 38010,CC(C)(C)C(C(=O)N1CC2(CCCO2)C1)NC(c1sccc1CO)=O 38011,C1(NC(c2c(C)cco2)=O)Cc2ccccc2C1NC(=O)CC(F)(F)Cl 38012,CCCN=C(NCCN1CCN(C)C(=O)C1)NCc1cnccc1Cl 38013,n1(CC(=O)NC2CC(N(C(CCNC(=O)OCC)=O)C)C2)cc(S(C)(=O)=O)cn1 38014,C(=O)(C1=CCCC1(C)C)NC(C(C)(C)NC(CC1(C=C)CCC1)=O)C 38015,N1(C(CC2CCN(C)C2)=O)CCC2(CCCC2CNC(=O)CC2CCC2)CC1 38016,N1(C(C2(C)CC2(F)Cl)=O)CC2CCC(C1)N2C(c1cnns1)=O 38017,N1(C(COC(C)(C)C)=O)CCC2(C1)CN(C(=O)CC(F)(F)Br)CCO2 38018,Cc1nc(C2CC2)ncc1C(N1CCOCC(NC(c2cnsc2)=O)C1)=O 38019,CC1COC(C)(C)CN1C(C12CCCC1CN(C(C13CCCC1C3(F)F)=O)C2)=O 38020,C1(C(C)C)CN(C(=O)C(C)(F)F)CCC1NC(=O)CN1CCCCCC1=O 38021,c1(N(C)C)cccc(C(c2cnc(C(F)(F)F)s2)N(CCC#N)C)c1 38022,c1(N2CC(C)C(N(C)C(=O)OC(C)(C)C)C2)nc(C(N)=O)nc2sccc12 38023,C(=O)(C(O)C(C)(C)C)NC1CC(C)(NC(c2nc(CN3CCOCC3)cs2)=O)C1 38024,C#CCCCCCCCNC(=O)CC(CC)NC(c1cc(C)cc(C)c1)=O 38025,Cc1ccnc(F)c1NC(c1ccc(Br)cc1OC(C)C)=O 38026,C12(C(=O)NCC(C)CN(C(=O)CC3OCCC3(C)C)C)CC(C)(C1)OC2C 38027,O=C(C(CO)c1ccccn1)NCC1CC(Cl)(Cl)C1 38028,N1(CC(c2cccc(Cl)c2)C)C2CCCC1CN(C(C1(C)CC1)=O)C2 38029,N#Cc1c(C(N2CC(CNC(=O)CCC3CCC(C(N)=O)O3)C2)=O)cccc1F 38030,N1(C(c2nn(C)nc2Br)C(=O)NCCCC)CCC(C2CNC(=O)C2)C1 38031,CCCCC(C)CCC(=O)N(CC(C)O)CCNC(c1cccc(C)c1N)=O 38032,c1(C(N2CCC(NC(C3(CC#C)CC3)=O)C(O)C2)=O)ccc2nc(C)[nH]c2c1 38033,Cc1c(C(N2CCCN(C(c3ccc[nH]3)=O)CC2)=O)sc2[nH]cnc(=S)c12 38034,C1(CC(C(=O)Nc2cnn(CCO)c2)NC(=O)OC(C)(C)C)CCS(=O)(=O)C1 38035,C(C)(C(C(=O)NC1CC(O)C1O)NC(C1OCCC1(C)C)=O)OC 38036,C1(C(N2C(C)C(NC(c3ccnc(CO)c3)=O)CC2)=O)CCn2nnnc2C1 38037,N1(C(C2CC(C(C)C)C2)=O)CCCC2(NC(C3CCCOC3)=O)CCCC12 38038,Cc1nn(C)nc1C(=O)NCC1(CNC(c2cc(Cl)cs2)=O)CCCC1 38039,O=S(=O)(c1cnc(Cl)c(C(=O)O)c1)N1CCN(CCC2CC2(Cl)Cl)CC1 38040,c1(OC)cccc(-c2cc(C(=O)OCc3nnn(C)n3)c(C)o2)c1 38041,Cc1[nH]c(CN2CC3CC2C3C(=O)Nc2ccc(Br)c(Cl)c2C)c(C)c1[N+](=O)[O-] 38042,CCC(C)CC(C)C(=O)NCC1CC2CCC1N(C(c1cnnc(Cl)c1)=O)C2 38043,C1(CNC(CC2C(=O)NC(=N)S2)=O)CCN(C(=O)CCc2ccsc2)CC1(F)F 38044,N1(C(Cc2c(C)occ2)=O)CCC(CNC(=O)CC(C)(C)C)C1C 38045,N1(C(c2cc(NC)ncc2)=O)CCC(C)N(C(=O)C(O)COC)CC1 38046,C1(CC(=O)NC(C)CCCNC(c2ccnn2C2CCC2)=O)CC2CCC1CC2 38047,C(C)(C(=O)NC1CCCC1NC(=O)C=CBr)(C1CC1)NC(C)=O 38048,C1(CC)(NC(=O)CC2CC=CCC2)CN(C(=O)CCOC)C1 38049,c1(CC)c(C(N2CCCC2C2CCCOC2)=O)cnn1C(C)(C)C 38050,c1(OC)cnc(C(=O)NC2(C)CC(NC(c3n[nH]c(C4CC4)n3)=O)C2)c(F)c1 38051,C1(C(=O)Nc2ccc(C(C)=O)cn2)CCN(C(=O)C=CC(CC)=C(C)C)C(C)C1 38052,C#Cc1ccc(C(=O)NCC2CC2C(=O)NC(c2ccnn2C)C)o1 38053,C(=O)(CCCCCCn1cc(C2CCS(=O)(=O)C2)nn1)N1C(C)(C(N)=O)CCC1 38054,C1(C(N2CC(NC(C=C(C)C3CC3)=O)C(CO)CC2)=O)CCc2nc[nH]c2C1 38055,c1(OC)ncc(C(=O)NCc2ccc(CNC(=O)C3=COCC3)cc2)cc1Cl 38056,c1(C(N2CCC(OCC(N3C(C)(CCC)CC3)=O)C2)=O)ccc(C)c(C)c1 38057,C(=O)(CCN=c1[nH]ccs1)N1CC(CN(C)C(c2ccc(F)c(CO)c2)=O)C1 38058,c1(C(=O)NC2(C)CC(C(N(CC(C)SC)C)=O)C2)cccc(F)c1F 38059,c1(C(=O)NC2(CNC(C(C)c3cccs3)=O)CCC2)cnc2sccc2c1 38060,C1(CNC(C2(CC)CCCO2)=O)CC(C)CN(C(=O)C(C)(C)OC(C)C)C1 38061,c1(OC)cc(NC(=O)CC2CCC2C2CC2)cc(F)c1[N+](=O)[O-] 38062,C(CCC(CO)NC(=O)CCNC(C)=O)NC(c1c(CC)nc[nH]1)=O 38063,c1(C(=O)NC(CNC(c2ccc(C)nc2O)=O)C2CCC2)c(Cl)ccc(F)c1C 38064,C1(NC(Cn2cc(C(C)O)nn2)=O)CC2CN(C(=O)CCC(F)(F)F)CC2C1 38065,C(=O)(C(O)CC(C)(C)C)NCCCC(CCC)NC(C1CS(=O)(=O)C1)=O 38066,C(N=c1cc2c(c[nH]1)C(=O)CCC2)C12CC(NC(=O)COC3CCCOC3)(C1)C2 38067,c1(C(=O)NC(C(C)(C)NC(C(CCSC)O)=O)C)ccc(C2=NOC(=O)C2)cc1 38068,CCCCC(N=c1ccn(-c2ncccn2)[nH]1)C(=O)N1CCNC2COCCC12 38069,c1(NC(C23C(CN(Cc4scc(C(=O)OC)n4)C2)C3)=O)cc(C)c(Cl)cc1Cl 38070,C(=O)(C1CCCc2n[nH]cc21)NC1(C(=O)O)CC(OC)N(C(C)=O)C1 38071,c1(C(=O)NCC2CN(C(CNC=O)=O)CC2C(F)(F)F)cc2cccc(F)c2o1 38072,C1(NC(c2cc(-c3cccnc3)no2)=O)CC(F)CN(C(C2CCCSC2)=O)C1 38073,C=CCCCC(C)(C)C(=O)Nc1cc(CC(C)(C)C(F)(F)F)n[nH]1.c1(C=O)nc(C(C)(C)C)no1 38074,CS(=O)(=O)c1cccnc1C(=O)NCC1CCC2C(C1)C2(F)F 38075,N1(C(C)=O)CCC2CN(C(=O)C(C)(C)c3cscc3Cl)CCC2C1 38076,c1(N2CC(c3ccc(OC)cc3)C(C)CC2)nc2ccc(Cl)cc2o1 38077,N1(C(=O)COC2CCOCC2)CCN(C(C23CCCCC2OCC3)=O)C2(CC2)C1 38078,c1(CC(=O)N(C2CCN(Cc3ccn(C(C)C)n3)C2)CC)cc(C)[nH]n1 38079,CCCC(C)(O)C(=O)NC1CN(C(=O)C(=O)NC2CC2)CC1CC(C)(C)C 38080,Cn1nc2c(c1NCC(F)(F)Oc1cc(C#N)ccc1C(=O)O)CCC2 38081,C1(NC(NCCc2cc(C)sc2C)=NCCCF)(C(F)(F)F)CC2(CC(F)C2)C1 38082,CCCCC(F)C(=O)NCc1occc1C(N1CCC(OC)C(F)C1)=O 38083,Cc1ccnc2c(C(=O)NC(C)CCN(C)C(C34CC(C)(CCO3)C4)=O)cnn12 38084,c1(OC)ccc2cc(C(=O)NC3CCCN(C(=O)C(C)=CC4CC4)C3)sc2c1F 38085,c1(C(N(C2CCN(C(C3COCCO3)=O)CC2)CC)=O)cccnc1N 38086,c1(N2CCC(c3scc(C)n3)CC2)ncnc(NCC=C(Cl)Cl)c1C 38087,c1(C(=O)NCCN(CCCCCC)C(c2cccc(C)n2)=O)c(C)ncnc1C 38088,C(=O)(C1=NN2CCCN=C2N1)NCC(CN(C(=O)CSc1cccs1)CC)(C)C 38089,C1(C(=O)NCCC(C)(C)NC(=O)CC2CC3CC3C2)CC2(CCCC2)CO1 38090,C1(C(=O)NC(c2cc(OC)c(F)cc2)C)CC2OC(C)CC2N1 38091,C(CC(=O)OC)(C(C)C)SCCc1n(CCOC)nc(-c2ccc(F)cc2)n1 38092,C1(NC(CNC2CC(C#N)C2)=O)CCn2nccc2C1 38093,N1(C(c2occ(C(=O)OC)c2)=O)CC2CC(NC(C3CN(CC(F)(F)F)C3)=O)C1C2 38094,N1(C(C2=NOC(CNC(c3ccc(C#N)cn3)=O)C2)=O)CCc2cncnc2C1 38095,C1(NC(C(C2CN(C(COCCN(C)C)=O)C2)O)=O)CCN(C)CC1(C)C 38096,Cc1nn(C)cc1CCNC(C1CN(C(=O)CC2(O)CCCC2)CC1C)=O 38097,N1(C(C(=Cc2ccco2)C)=O)CC2(CC2)CC1CNC(=O)C(c1nc(C)cs1)C 38098,C1(CCC)(NC(c2csnc2Cl)=O)CCN(C(c2cccc(C)n2)=O)CC1 38099,c1(-c2sc(C(=O)NC3C(NC(C=C(C)C4CC4)=O)CC3)c(C)n2)c(C)nn(C)c1C 38100,c1(C(C)OC)ccc(-c2nc(-c3cnn(C)c3)nn2-c2ccnc(O)c2)cc1 38101,C1(C(N(CCCNC(C(C(=O)OC)(C)F)=O)C)=O)CCc2nn[nH]c2C1 38102,c1(C(=O)NCC(CNC(CCN(C(CCC)C)C)=O)F)cc(O)cc(Cl)c1 38103,C1(C(=O)NCCN(C(C2(NC(=O)OCC)CCCC2)=O)C)COCCN1C 38104,C1(C(=O)NCCC=CBr)(CCOCCOCCOCC)COC1.COC 38105,Cc1ccc(C(C)NC(C2CC=CCN2C(c2cnn(C)c2Cl)=O)=O)cc1 38106,c1(CN2C(CC)CN(C(c3c(Cl)ccnc3Cl)=O)CC2)ccc2nc(O)[nH]c2c1 38107,C1(C)(C(=O)NCC#CCNC(CCc2c(C)noc2C)=O)CCCCC1C 38108,C(C(C)(C)CCl)(c1n(CC=C)nnn1)NCCCc1cccc(OCC)c1 38109,c1(C(=O)NC2CCCC(N(C(CCC(=O)NC)=O)C)C2)oc2ccccc2c1C 38110,c1(NC(=O)Nc2ccc(CC(=O)NC)cc2)c(Br)cc(F)c(F)c1F 38111,CC(N=c1[nH]c2c(c(=NCCSC3CCOCC3)[nH]1)CCCCC2)c1ccco1 38112,CC1=NS(=O)(=O)NC=C1C(=O)NC1CC(CCNC(C2(S(N)(=O)=O)CCC2)=O)C1 38113,C1(NC(c2c(C)noc2)=O)CC2CCC(C1C)N2c1ncccn1 38114,Cc1ccc2c(c1)CC(C(N1CCN(C(=O)CC3CC3)CCC1C)=O)S2(=O)=O 38115,C(=O)(CCCC(C)(C)C)NC(C(=O)N(CCCC=C)C)Cn1cncn1 38116,c1(C(=O)NCC2C3CN(C(C(C)n4cccc4)=O)C2C3)cc([N+](=O)[O-])ccc1Cl 38117,Cc1cnc2c(NC(N3CCC4(CC3)CCS4=O)=O)cccc2c1Cl 38118,c1(C(=O)NCC2N(C(c3c(C)cncn3)=O)CC(F)C2)ccnc2ccccc12 38119,Cc1ccc(Br)c(CC(=O)NC2CCC23CN(C(=O)C=CCO)C3)c1 38120,N(C1CCc2sc(Br)cc21)C(c1cnc(OC)s1)c1nnnn1C1(C)CC1 38121,C1(C(N2CCN(CC(=O)NCc3ccco3)CC2)C2N(CC(=O)OC)CCC2)CC(=O)C12CCC2 38122,C1(CC(=O)NCCCCC2C(C)C2)CCCN(C(c2nonc2N)=O)C1 38123,C1(C(=O)NC(C)(C)CCNC(=O)Cc2cnoc2)CC2(CCC2O)C1 38124,C1(O)(CNC(CC(=O)N(C)C)=O)CCN(C(c2n[nH]cc2C(C)(C)C)=O)C1 38125,C1(NC(C2(C#N)CCC2)=O)CN(C(C2CC(=O)CCO2)=O)CC(F)(F)C1 38126,C1(NC(C=CCOCCOC)=O)CC2CN(C(c3ccc(C4CC4)cn3)=O)CC12 38127,S(=O)(=O)(c1cnn2c1CCCC2)NC(C(Cc1cc(C)[nH]n1)N)=O 38128,CCC(CS(C)(=O)=O)NC(C1CC(NC(=O)OC(C)(C)C)C1)=O 38129,N1(C(C(c2ccc(Cl)cc2)C)=O)CC(C)(C)CC1CNC(C1CC1(C)C)=O 38130,N1(C(C2CCC(C)(C)C2)=O)CC2CCN(C(c3ccc4occc4n3)=O)CC2C1 38131,C1(C(=O)NC(C)CCNC(C23CC(C#N)(C2)C3)=O)CC(=O)C12CCC2 38132,N1(C(c2c(C)ccs2)=O)C(C(=O)Nc2cncc(Br)c2)CC2CC12 38133,CC(C)(C)C(C)(C)CN=c1[nH]c2c(c(=NCC3CCCC(O)C3)[nH]1)CSC2 38134,C1(CC=C)CCCC1(c1nnnn1CCC1(C)CC1)NCCOC(C)C 38135,C12(NC(CC3N(C)CCOC3)=O)CCCC1CN(C(=O)Cc1cc[nH]n1)C2 38136,C1(NC(=O)NCCC(CC)C)CCCN(C(=O)OC(C)(C)C)C1c1cnn(C)c1 38137,C1(C(N2CCC(C(C)C)C2)=O)CC2CC2N1C(=O)CC1CCC1 38138,C1(CN(C(c2c(CC)cc[nH]2)=O)C)CCC(NC(C2CC=CCC2C)=O)CC1 38139,N1(S(CCC)(=O)=O)CCCC(C(N2CCC(NC(=O)C(C)(CC)OC)CC2)=O)C1 38140,C12=CN=C3C=CC=CN1N3C(=O)C(O)(CNC(C(COC)C)=O)CC(C)NC2=O 38141,c1(C(=O)NCC2C(CNC(c3ccc(N4CCCC4)nc3)=O)C2)cccc(=O)o1 38142,c1(CNC(c2n(CCC)ncc2)=O)nnn(C)c1C(=O)NCC1CN(C2CC2)C1 38143,C1(C(=O)NC2(CO)CN(C(=O)C(c3ccccc3)C)C2)CC2CC(=O)C1C2 38144,C1(C)(CNC(C2C(C)OCCC2)=O)COCCN(C(=O)CNC(=O)CCCCO)C1 38145,c1(CCCCC)cc(C(=O)NC23CC(CNC(c4ccsc4CC)=O)(C2)C3)n[nH]1 38146,c1(C(=O)NCC(C)NC(=O)CC2CC=CCN2C)ccc2c(c1)CCC(C)(C)O2 38147,C1(NC(=O)CSC2CCCCO2)(CNC(=O)C=C2CCSCC2)CCOCC1 38148,CCCCC(CC)CC(=O)NCC(C)(C)C(=O)NCCS(C)(=O)=O 38149,C1(NC(=O)CN2C(=O)CCC2=O)CCCCN(C(C2CN3CCN2CC3)=O)C1 38150,Cn1nc(C(=O)NC(C)(CNC(C2CC(CF)C2)=O)CO)cc1Cl 38151,c1(C(=O)NC2CC3(CN(C(C4C(C)CCC4)=O)C3)C2)ccc2c(n1)OCC(=O)N2 38152,N1(C(c2ccnn2C2CC2(F)F)=O)CCCC(CO)(CO)C1 38153,c1(CC(N2CC(C)C(NC(=O)Cc3nc[nH]n3)CC2)=O)c(F)ccc(Br)c1F 38154,N1(C(CC2(C)CCCC2)=O)CCCC(n2cc(CO)nn2)CC1.C(=O)(CCCC(N)=O)N 38155,C(=O)(CCCN=[N+]=[N-])N1C(C(=O)N(CCCCN(C)C)C)(COCC)C=CC1 38156,C1(CNC(c2cc(C)oc2)=O)CN(C(=O)CSC(C)(C)C)CCC1C 38157,c1(CSC)cccc(C(=O)N(CC(O)CNC(C2CC(SC)C2)=O)C)c1 38158,c1(C(C(=O)NCCOC)N(C2CCCC(O)C2)C)nc(C)c(C)s1 38159,C1(F)(CNC(CN(C)C(N)=O)=O)CCCN(C(=O)C(F)Cc2ccccc2)CC1 38160,CC(C)(CC(F)(F)F)C(=O)NCC1CCC1NC(C1CCC(C(F)(F)F)O1)=O 38161,CC1(C)CCCN(C(c2ccc(N)c(F)c2)=O)C1CNC(=O)C#CC1CCC1 38162,C1(NC(C(CC)C2CCOC2)=O)CCC(CNC(=O)Cc2cc[nH]c2)CC1 38163,Cn1cc(C#CCNC(C2CC(C)(C)CCN2C(=O)CP(C)(C)=O)=O)cn1 38164,CC1CCCCC1C(=O)NCC1(CC(=O)NCCCC(C)(C)O)CC1 38165,c1(CNC(=O)COCCCF)ccc2c(c1)CN(C(c1cc(CO)ccn1)=O)C2 38166,C1(NC(CC(=C)C)=O)CCCOC12CCN(C(=O)C(C)C(C)C)CC2 38167,C1(C(=O)OC)(NCCC2CCCC23CC3)COc2ccccc2C1 38168,c1(CC)ccc2c(c1)C(CCOC(C)=O)C(=O)N2.c12cc(C)c(C)cc1N2CC 38169,c1(N2CC(C(=O)NCCCc3cn(CCOCC)nc3)C2)ncccc1C#N 38170,CC1CN(C(=O)CCNC(=O)C=Cc2cc[nH]c2)CCC1SCc1ccccn1 38171,c1(C(=O)NC(CC(N2CCOCC(C(C)C)C2)=O)(C)C)cc2cc[nH]c2cn1 38172,c1(C(N2CCCC(CNC(CC3(C#C)CC3)=O)C2)=O)cc(S(N)(=O)=O)cnc1C 38173,C1(C(=O)NOCCO)(CC=C)CCCN1C(C1CCC(F)CC1)=O 38174,c1(C(N2CC(C)C(C)(CO)C2)=O)ccc2c(n1)CN(C(=O)C(CO)N(C)C)CC2 38175,CCC(CC)C(C)C(=O)N(CCNC(=O)C=Cc1ccc(OC)cc1)C(C)C 38176,c1(C(N(CCCOC)C)=O)c(OC(C)C)ccnc1F.C1=CCCCN(C)C1=O 38177,N1(C(C(C=C)CC)=O)CCOC2(CCN(C(=O)Cc3ccn(CC)n3)C2)C1 38178,C(=O)(C(F)(CNC(=O)C(C#N)C(C)C)C(C)C)NCCc1cn(CC)nn1 38179,C(=O)(C(O)C(O)c1ccccc1)N1C(C2(NC(=O)CCn3cnnn3)CC2)CCC1 38180,N1(C(C(C)CNC(=O)C=CC2CCC2)=O)CCC(CN=[N+]=[N-])CC1 38181,C1(C(N2CCC3CC23)=O)COCCC1NC(C12CCN(CC1)C2)=O 38182,c1(C(N2C(C)(CNC(=O)C=CC3CC3)CCC2)=O)occ2c1CCOC2 38183,c1(NC(N2CC3C(c4onc(C)n4)(C3)C2)=O)cncc(F)c1I 38184,c1(CC)cccnc1C(=O)N(CC(C)NC(c1ccc(-c2cccs2)[nH]1)=O)C 38185,C=C(C)C1OCCC1CNC(C1CC1c1cccc(Br)c1Cl)=O 38186,CCC(C(C)(C)O)NC(=O)CC1CCN(C(=O)C(c2ccnn2C)C)CC1 38187,c1(C(N(C2CN(C(c3n(CC=C)ccc3)=O)CC2O)C)=O)nsc2ccccc12 38188,c1(SC)cc(C(N2CC3CC2CN3C(c2cn[nH]c2)=O)=O)cc(SC)c1 38189,N1(C(CCCC)=O)CC2CCC2(C(=O)NC(c2ccc(Br)cc2)C)C1 38190,C1(C(=O)NC(C2CN(C(C(CC#C)(C)C)=O)C2)C)CC2(C1)CC1(CC1)C2 38191,c1(C(=O)NC2(C(=O)NC)CCC2)coc2c1CN(C(=O)C=CCN1CCC1)C2 38192,c1(CN2CCC(C)(C(=O)NCCC)C2)cc2ccccc2s1 38193,N1(C(CCC(C)SC)=O)CC2CCC(C(N3CCCC(C)(C#N)C3)=O)(C2)C1 38194,c1(CNC(CCCNC(N)=O)=O)cncc(C(=O)NC2COC(C(F)F)C2)c1 38195,c1(C(C)=O)cccc(CC(=O)NCCC2CCN(C(=O)C=C3CCC(C)C3)C2)c1 38196,C(=O)(CCCn1cccn1)N(CC(C)NC(=O)CSCCN(C)C)C 38197,c1(N(CC)Cc2cccc3[nH]ccc23)nc(N2CCC3CC3C2)c2sccc2n1 38198,C(=O)(CC(CC(C)C)C(=O)O)N1CCC(c2cc(C)cc(C)c2)(F)CC1 38199,C1(CNC(CC(C)(O)C2CC2)=O)CN(C(C2CC2(Cl)Cl)=O)CCC1(F)F 38200,N1(C(=O)COCCF)CCC2CN(C(=O)CSCc3ccc(Cl)cc3)C2C1 38201,C1(C(=O)NCC2CC(C)C2)CCN(C(C2CCC(=O)N2C)=O)CC1 38202,N1(C(C(C)(C)C#N)=O)CCC(F)(F)C(CNC(C2(C)CNC(=O)C2)=O)C1 38203,N1(C(C=CC)=O)CCOC2(CCC(NC(C3CCCC(C(F)(F)F)C3)=O)CC2)C1 38204,c1(C(=O)NCC2N(C(CC(=O)OC)=O)CCN(C)C2)ccccc1N=S(C)(C)=O 38205,C1(C(=O)NCCCC(C)NC(C2(C)CCC(F)(F)CC2)=O)CCc2nn[nH]c2C1 38206,CC(CC(=O)NC(C)CN(C(=O)CCc1nccs1)C)c1cnn(C)c1 38207,C1(CC)(CO)CCCN1C(C1C=CCN(C(C2CC(F)(F)C2)=O)C1)=O 38208,c1(C(N2C(C(C(=O)NC3CC4(CN(C)C4)C3)(C)C)CC2)=O)ccn2cncc2c1 38209,c1(OC)cc(C(=O)NCCCc2ccc(-c3cn[nH]c3)cc2)cc(Br)c1 38210,C12(C(=O)NCC(=C)CCNC(C3COC(=O)N3C)=O)CC(CO)(C1)OC2(C)C 38211,C1(C(=O)NCC2(COC)CCCN2C(=O)CN=S(C)(C)=O)COC2(CCC2)C1 38212,c1(C(N2CC=C(CNC(=O)CN3CCOCC3)CC2)=O)ccc2c(c1)CC(=O)N2 38213,c1(C(=O)OC)c(NCCN(C)C(C2CC(C3CC3)=NO2)=O)nnc2c1CCC2 38214,N1(C(C2(CO)CCN(C(CCCC#CC)=O)C2)=O)CCC2(CCOC2)C1 38215,CC1CCN(C(C2CC(F)C2)=O)CC1CC(=O)NCC1CC[Si](C)(C)C1 38216,C(=O)(C1CCc2cccc(=O)n21)NC1C(OC)CN(C(C2(C(=O)OC)CC2)=O)C1 38217,C(=O)(C(F)CC(C)(C)C)N(C)CC1(OC)CC1.c12ccc(cn1)CNC2=O 38218,c1(C(=O)OC(C)(C)C)cccc(CN(C)C)n1.C12(C)CCN1C2=O 38219,C(=O)(C(C(C)(C)C)OC(C)(C)C)N(C)CC1CCN(C(C2(C(N)=O)CCC2)=O)C1 38220,N1(CC)C(=O)CCC1C(=O)NC(C1CCCC1)CNC(=O)C(=C1CCCCC1)F 38221,C(C1CCN(C(C2CS(=O)C2)=O)CC1)=CC(=O)NCC1(F)CCN(C)C1 38222,N1(C(c2c(NC(N)=O)cccc2)=O)CC2(CCN(C(c3cc(CO)[nH]n3)=O)C2)C1 38223,c1(C(=O)NC(C)C(CO)NC(c2cc3n(c2)CCSC3)=O)cccn2nccc12 38224,C1(CC)CC(C(=O)NCCC(C)N(C)C(c2cnc(C(N)=O)cn2)=O)CCO1 38225,Cn1cc(C(=O)NCCCNC(=O)C(F)CC2CCCCC2)ncc1=O 38226,CCC(C)CCCCC(=O)NCC(C)N(C(c1ccc(OCCF)cn1)=O)CC 38227,C1(NC(C(CCC)CC2CC2)=O)COC2(C1)CN(Cc1cncs1)C2 38228,Cc1cc(C(=O)NCC2(NC(=O)C=Cc3ccc(=N)[nH]c3)CC2)c2c(c1)CCC2 38229,Cc1cc(F)ccc1C(O)C(N1CCC(O)(CCNC(=O)C(C)(C)C2CC2)C1)=O 38230,Cc1ccnc(O)c1C(=O)NCCCCNC(c1ccnn1CC(F)F)=O 38231,C(=O)(C(CC)(CC)CC)N1CC(C(=O)NC(C(=O)OCC)CO)(SC)C1 38232,C1(N(C(=O)CCC2OCCO2)C)CN(C(=O)CN2CC(=O)N(C)C2=O)CC12CC2 38233,N1(C(CC2N(CC)CCC2)=O)CCN(C(=O)C=C2CCCC2)C2CS(=O)(=O)CC12 38234,c1(C(N(CCN(C(C(COC)C)=O)C(C)C)C)=O)ccc2c(c1)NCCNC2=O 38235,C1(C(C(=O)NCCCSC)N(c2ccc(C)cc2)CC2CC2)CC=CCC1C 38236,c1(N2CCC(N(CC(=O)NC)C)CC2)nc(=NCC2CC2C)[nH]c2c1SCC2 38237,CCC(C(=O)NC1(C(=O)N(CCO)CCOC)CCCCC1)C(C)(C)CC 38238,C1(CC)(NC2CCC(C#N)CC2)CCCN(Cc2ccccc2)C1 38239,CCC(C)CC(=O)NCC1(CNC(c2ccncc2N)=O)CC1(F)F 38240,CC(CNC(=O)CCCN1CCCC1)C(F)C(=O)NCCN1CCC2CC12 38241,CCC(C(=O)NC(CO)C(C)NC(=O)CC1CCCC1)Sc1ccccc1 38242,Cc1cc(O)c(C(N2CC(NC(=O)C=CC3CCCC3)C(C)(C)C2)=O)nn1 38243,c1(C(N2C(C)C(NC(=O)CC3CCCCC3O)CCC2)=O)c[nH]c2nccc-2c1 38244,C1(NC(CC2CC(=C)C2)=O)CC(F)CN(C(=O)Cn2cccc(C)c2=O)C1 38245,C#CCC(C)(C(=O)NC(CCO)C1CCCC1)NC(c1ncnc(C)c1C)=O 38246,N1(C(c2c(C)cc[nH]c2=N)=O)CC2(CCC2)CC1CNC(=O)C#CC1CCCO1 38247,C1(NC(C2CCC(C3CC3)O2)=O)CCN(C(C2CN3CCC2CC3)=O)CC1O 38248,c1(C(=O)NCCOC2CN(C(c3nn(CC)c(C)c3)=O)C2)sc(C)c(C)c1C 38249,c1(C(=O)NC2(C)CN(C(C3(C)CCCS3(=O)=O)=O)C2)ccc(F)c(C(F)F)c1 38250,C=CC1OCCC1C(N1CCC(CCN(C(=O)CC(O)CN(C)C)C)CC1)=O 38251,N1(C(C2C(C3C(C)C3)C2)=O)CCC(O)(CN(C)C(c2cn3ccsc3n2)=O)CC1 38252,C12(NC(C34CC(OC)C3C4)=O)CCCC1CN(C(=O)Cc1c(C)cccc1C)C2 38253,c1(C(=O)NCCC(C)(C)NC(=O)C(O)CCS(C)=O)nnc(O)c2ccccc12 38254,c1(C(=O)NC(C(=O)NC(CC)CCCO)c2ccoc2)c[nH]c(C)cc1=O 38255,Cc1cc(F)sc1C(=O)NC(C(=O)N(C)Cc1cccnc1O)C1(O)CCC1 38256,N1(C(C2(CC(C)C)CCC2)=O)CC2CC1CN2C(C1CC1(Cl)Cl)=O 38257,N1(C(COCC)=O)CC2(CCCN2C(=O)NC(c2ccccc2)C)C1 38258,CC1CCN(C(=O)C2=CCCC2)CCN1C(c1noc2c1CCCC2)=O 38259,Cc1ccc(C(=O)NC2CCC(NC(c3cnn4cccnc34)=O)C2)c(C)c1Br 38260,c1(CC(=O)NC2C(CNC(=O)COc3ccsn3)C2)ccc(O)nc1 38261,Cc1oc2ccccc2c1C(N1CCN(C(=O)CC2COC(C)(C)O2)C(C)C1)=O 38262,C1(C(N2CCC(O)(Cn3cc(C4CCCC4O)nn3)C2)=O)CCCC2(CCC2)O1 38263,N1(C(C=CC2(C)COC2)=O)CCC2CCCN(C(C3C4CC5C(C4=O)C35)=O)C2C1 38264,N1(C(C(C)NC(=O)OC)=O)CCOCC(F)(CNC(C2(C3CC3)CCC2)=O)C1 38265,C(=O)(C(F)C(=O)N(C)CC1CCCCN1C(=O)C(C)(C)OCC(F)(F)F)OCC 38266,CCCC(C)(CCC)C(=O)NC1CC(NC(=O)CN(C)CCOC)CC1O 38267,C1(N=[N+]=[N-])(C(=O)NCC(CCC)(C)C)CCN(C(C2CCOC2(C)C)=O)C1 38268,c1(OC(C2CC(OCCNC(=O)OC(C)(C)C)C2(C)C)=O)ccc2c(c1)OCO2 38269,c1(CC(=O)NC2CN(Cc3c(F)ccc(C)c3)C2)ccc2c(c1)OCCO2 38270,N1(C(c2cncc(N)c2)=O)CC2CCC1C1CN(C(c3cnc(O)o3)=O)CC21 38271,c1(C(CC)C(=O)N(CCCN2CCCC2)C)ccc2c(c1)OCO2 38272,Cc1conc1C(=O)NC(C1CN(C(c2cnn(C(C)C)n2)=O)C1)C 38273,C1(C(=O)NCC2(C(C)(C)O)CN(C(CSC(C)C)=O)C2)CCCCCC1(F)F 38274,CC(C(C)(C)C(=O)NCC1CC1)NC(c1cnc(CC2(CF)CC2)o1)=O 38275,C1(C(=O)NCc2c(CC)cncc2)CCCN1NC(=O)C(F)C(F)(F)F 38276,C1(C)(C(=O)NC)CCCN1C(c1cn(CCNC(=O)CC2(C#N)CC2)cn1)=O 38277,C(C(F)(F)C(F)(F)F)OCC(=O)N(CCCNC(C1(F)CC1)=O)C 38278,C=CC(C)(CC)C(=O)NCCC1(C(=O)NC2(c3ccccc3)CCC2)CC1 38279,n1(CCOC)ccc2cc(NC(c3cccc4c3COC4)=O)ccc12 38280,c1(CC)cccnc1C(=O)NC1CC(C)N(C(=O)CC(C)n2ccnc2)C1 38281,C#CC(C)(C)C(=O)NC(C)CN(C(c1csc(C(F)(F)C(F)(F)F)c1)=O)CC 38282,n1(C(C(=O)OC)C)nnnc1C(c1nocc1OCC1CCCO1)NC(C)(C)C 38283,C1(C(=O)NC(C2(C(N3CCCC(CC(C)C)C3)=O)CC2)C)CC(C2CC2)=NO1 38284,c1(C(=O)OCc2cccnn2)nc(Br)sc1Cl 38285,c1(C(=O)NCC(CC)NC(C2(C3CC3)CCCO2)=O)[nH]c2ccc(C)cc2c1C 38286,C#CCC(O)C(=O)N(CCC(C)NC(c1cc(COC)oc1C)=O)C 38287,C1(C(N(C2CCCC2)CCCNC(C2CCO2)=O)=O)CCS(=O)(=O)C1 38288,C1(OC)CN(C(=O)C(n2ccnc2C)C)CC1NC(=O)CN1CSCCSC1 38289,N1(C(c2c(C)csc2)=O)CCCCC1CNC(c1ccc(-c2ccco2)s1)=O 38290,N1(C(c2c(C#C)c[nH]n2)=O)CC(NC(=O)COC(C)(C)CC)C(S(C)(=O)=O)C1 38291,Cc1n[nH]cc1C(C(=O)NC(C)C)N(C)CCC1CCCCC1 38292,C1(C(=O)NC(CC=C)COC)(C(=O)OCC)CCCNC1 38293,C1(CNC(C(=O)N(C)Cc2ccn(CC)n2)=O)C2CCCCCC12 38294,N1(C(CC(CCC)C)=O)CC2CC(C1)N(C(=O)COCC1CCOCC1)C2 38295,C1(NC(c2ccn(CC(C)C)n2)=O)CC2CC(C1)CN(C(C1CC3CC3C1)=O)C2 38296,N1(C(=O)NC2(C)C(C)OCC2)CCN(S(=O)(=O)N2CCCC2)CC1 38297,C1(C(=O)NCC(CN(C)C(C2(C(F)F)CC2)=O)O)CCC=CCCC1 38298,C1(NC(=O)NCC(N2CCN(C)CC2)(C)C)C(O)C(O)CC(O)C1O 38299,CC1(C)CC(C(=O)NCCCCCC(=O)NC2CCCSC2)CCO1 38300,c1(C(=O)NC2CC(C(N3CC=CC3)=O)C2)ccc(F)cc1OC(F)F 38301,Cc1cc(C)c(C(=O)NC2CCC(CNC(c3cc(CO)[nH]n3)=O)CC2)cn1 38302,c1(C(=O)NCC(C=C)O)nc(CNC(=O)C(C)OCC)oc1C 38303,c1(-c2onc(COC(c3ccc(CC)cc3)=O)n2)c(C)oc(C)c1Br 38304,c1(C(=O)NCCCCNC(c2c(SC)cccc2F)=O)ncnc2ccsc12 38305,n1(CC(N2CC(CCNC(c3n(C=C)nnc3)=O)C2)=O)nnc2ccccc12 38306,C(CCCCC(=O)NC1CCC(C(=O)NC(C(N)=O)C(N)=O)CC1)=CC 38307,CCCC(C(=O)N1CCCC(N(C(=O)C=C(C)Cl)C)C1)c1ccccc1 38308,CC1(C)CC(C(F)(F)F)(C(=O)NCC2CCC2NC(=O)CSc2ccccn2)C1 38309,N#Cc1n[nH]c(=NC2CCCC23CN(C(c2c[nH]cc(Cl)c2=O)=O)C3)s1 38310,CC1CC=C(C(=O)NCc2cc(C(=O)NCCn3ccccc3=O)ccn2)CC1 38311,C1(C(N2CCC(OC)C(CO)C2)=O)COC2(C1)CN(C(=O)CSCC(N)=O)C2 38312,C(=O)(C(C)CCCC(C)C)N1CC(CCCCNC(C(C)=C(CC)C)=O)C1 38313,N1(C(CCCCCCNC(CCOC)=O)=O)CC23CCC2(COC3)C1 38314,CC1CN2C(C)CN1Cc1scc(n1)C2=O.c1(CO)cc(C(F)F)ccn1 38315,N(C1COc2c(Cl)cccc21)C(N(C)Cc1ccccc1I)=O 38316,C12(NC(C3CC(C)OCC3)=O)CCCC1N(C(=O)COC1CCOC1)CCC2 38317,c1(C(=O)NC2C(OC)CN(C(=O)CC(C)C3CC3)C2)cc2cc(Cl)ccn2n1 38318,CC1CN2CCN1C(C(N1CC(NC(c3nccnc3Cl)=O)C(C)(C)C1)=O)C2 38319,CC1(C)CCN(C(=O)C=C2CCC2)CC1C(=O)NCC1CC(O)C(O)C1 38320,C1(C(N(CC(CC)CC)C2CC2)=O)CCCN(C(=O)CCC(C)=O)CC1 38321,C1(C(=O)NCC(C2CCCC2)O)(COC)CN(C(C2CCCO2)=O)C1 38322,N1(CC)C(=O)CCC1CC(=O)NCc1nc(CNC(C2COCC2(C)C)=O)cs1 38323,C1(C(N(C2CC2)CC2N(C(c3ccccn3)=O)CCCC2)=O)(CF)CCOCC1 38324,N1(C(c2sc(C(F)F)nc2-c2ccccc2)=O)CCS(=O)C(F)(F)C1 38325,c1(NC(C2CN(C(N(C)C)=O)C2)=O)nc(Cl)c(Cl)nc1Cl 38326,C(C(C)C(F)C(=O)NC1COCC1CO)NC(c1noc(CC)c1C)=O 38327,C1(COC)(NC(=O)C(c2ccccc2)F)CCN(C(=O)OC(C)(C)C)CC1 38328,C(=O)(NNC(=O)C(CN)CC(C)C)c1nc(C)c(C(=O)O)cc1 38329,N1(C(C(CC(C)(C)C)NC(c2cnn(CC)c2C)=O)=O)CC(C)C12CCOCC2 38330,Cc1nc(C(C(=O)NC2(C)CC2)N(C)C(c2ccc(F)cc2)C)sc1C 38331,c1(CCNC(C(C2CCN(C(c3ccn(C)n3)=O)C2)F)=O)ccc(F)cc1 38332,CC1CN(C)CC(C(N2CCCN(C(=O)CN3C(=O)CNC3=O)CC2)=O)O1 38333,C1(OC)CC(CNC(c2cccnc2)=O)N(C(=O)CC(F)(F)Cl)C1 38334,c1(-c2onc(C)n2)ccccc1CC(=O)NCC1CCN1C(=O)CCCN(C)C 38335,C1(CNC2CN(C(=O)OC(C)(C)C)C2)(NC(N(C)C)=O)CCSCC1 38336,c1(CC(=O)NC(C2CC=CCC2)C(=O)NCC(C(C)O)O)ccccc1F 38337,C(=O)(C(O)CCCC)NCC1CCC(C(=O)NC2(CC=C)CCCCC2)CC1 38338,c1(CC(=O)NCC2CCN(C(=O)CCCc3ccsc3)CC2)ccc(O)c(Cl)c1 38339,C(C1=CCN(C(c2ccsc2)=O)CC1)NC(c1cn(C2CCC2O)nn1)=O 38340,C1(C(N2CCCN(C(CCSc3n(C)nnn3)=O)CC2)=O)CC2CCCCCC12 38341,C1(NC(c2cc(CCC)ncc2)=O)CCN(C(c2sccc2F)=O)CC1CO 38342,CC1(C)CC(=O)N(CC(=O)NC2C=CCN(C(c3cccc(F)n3)=O)C2)C1=O 38343,c1(C(=O)OC)cccc(NC(=O)NCc2ccncc2C(C)C)c1OC 38344,C=CC1CN(C(c2cnnn2CC)=O)CC1NC(c1ccc(SC)s1)=O 38345,C1(C(=O)NCC(CC=C)(F)F)CC2CCC(C1)N2C(=O)C(C)(C)C(=O)OCC.O 38346,c1(C(=O)NC2CCCCC2NC(C2(CO)CCC2)=O)ccc2c(c1)OCO2 38347,N12CC3CCC3(C1)C2=O.c1(NC(C2C(OCC=C)CC2)=O)cc(CC)cc(F)c1 38348,c1(CC)ccc(NC(C2CN(C(c3cc(F)cc(Br)c3)=O)CCN2)=O)c(O)c1 38349,C1(NC(c2c(CC)cco2)=O)CCN(C(C2(C)CCCN2C)=O)CC1O 38350,Cc1c(NCC2CC2C)ncnc1N1CCN(c2ncccn2)CC1 38351,C1(C)(C(=O)NCCCNC(c2c(COC)cco2)=O)CCOC1C 38352,c1(NC(C(COC)NC(=O)CCCN(C)C(C)=O)=O)cc(C)c(C)c(C)c1 38353,C1(NC(CC2C(C)(C)CCO2)=O)CN(C(=O)CC2=CCOCC2)C2(CCC2)C1 38354,C1(NC(C(CC=C)CNC(=O)C=C(C)C(F)F)=O)CC2CC1CC21CC1 38355,C1(C(N2CCCN(C(c3ccc4cc[nH]c4n3)=O)CC2)=O)CCc2n[nH]cc2C1 38356,N1(C(c2ccc(CO)cc2)C(=O)NCC2CCCCC2)CCC(C2CCOC2)C1 38357,c1(C(N2CCC(N(CCC)C(c3ncc[nH]c3=O)=O)C2)=O)cc2c(ccn2C)[nH]1 38358,C1(NC(C(C)Oc2ccc(Cl)cc2)=O)CCN(CCF)C1(C)C 38359,c1(C(=O)NCCN(C(=O)Cc2cc(Cl)ccc2O)CC)cnc2ncccc2c1 38360,C1(N(C)Cc2ccc(Cl)o2)CCN(C(c2onc(C(C)OCC)n2)=O)CC1 38361,N1(C(c2c(CC)nns2)=O)CCN(C(=O)Cc2ccc(C)c(C)c2)CC1C(C)C 38362,N1(C(CN(CCC)C)=O)CCC(N(C)C(c2ccc(OC)c(Cl)n2)=O)C(C)C1 38363,c1(C(N2CC(C)(C(=O)Nc3cncc(C(C)(C)C)c3)C2)=O)ccc(Br)nc1Br 38364,c1(C(N2CCCC(N(C)Cc3cc(C)no3)C2)=O)n[nH]c(C)c1[N+](=O)[O-] 38365,c1(C(=O)NC2C3(CC(NC(=O)Cn4cncn4)C3)C2)cccc2c1OCCO2 38366,N1(C(c2ncn(CC)c2)=O)C2CCC1CC(CNC(=O)C(=Cc1cscn1)F)C2 38367,CCCCCC(O)CC(=O)N1CCCC1CCNC(c1cnccc1C(F)F)=O 38368,C1(C(=O)OC)CN(C(=O)NCC2CC(C)(C)OC2(C)C)C2CCCC2O1 38369,N1(C(C2CC(C)N2C(c2ccc(C#N)[nH]2)=O)=O)CCCC(F)CC1 38370,c1(OC)ccc(OC)c(C(N2CCC(C)(CNC(C3(C)CC(C)(C)C3)=O)C2)=O)n1 38371,Cc1ccc(C2CC2C)cc1Br.N1(N(C)Cn2cc(CCO)nn2)CCOCC1 38372,c1(C(=O)NCC(CC=C)NC(=O)C(O)CC(F)F)cccc(S(=O)(=O)C2CC2)c1 38373,O(NC(=O)CC(CCCC)NC(=O)C(CC)C(C)C)CC#C 38374,C1(CNC(c2nc(CCC)sc2)=O)C(O)C(O)CN1C(C1CCCCS1(=O)=O)=O 38375,C1(NC(c2cn3c(n2)CCC3)=O)CCN(C(=O)Nc2ccccc2)CC1F 38376,c1(C(N2CCCC(=C)C2)C(=O)NCCOC)cccc(F)c1I 38377,C1(c2cccs2)(C(=O)NC(C#C)(C)C)CCN(C)C1 38378,C(=O)(CC(C1CC1)C1CC1)NC(CN(C(C(=O)NCC)=O)C)CC 38379,CC1(CNC(c2coc(Cl)n2)=O)COCCN(C(c2ccnc(O)c2)=O)C1 38380,Cc1cccc(C)c1CC(=O)NC1CC2(C1)CC(NC(C1(F)C3CCCC13)=O)C2 38381,c1(C(=O)Nc2cc(O)n[nH]2)cnc2n[nH]c(-c3cccnc3C3CC3)c2c1 38382,N1(C(COCCC#C)=O)CC2CCC2(CC(=O)NC(C)COC)C1 38383,c1(N2CC(C)CS(=O)CC2)ncc(S(=O)(=O)NCc2ccc(Br)c(F)c2)cc1Cl 38384,Cc1c(C(=O)NC2CC3CCC2N3c2cc(OC3CC3)ncn2)cncc1Cl 38385,C=CCC(CC(=O)NCCc1ncon1)NC(=O)C(C)(C)N(C)C 38386,C1(C(N(CC(C)(F)F)C)=O)CN(C(c2cc(C(N)=O)co2)=O)C(C)(C)C1 38387,c1(NC(C)C)cccc(S(=O)(=O)NC2(CO)CCC(=O)NC2=O)c1 38388,c1(C(N2CCN(C(C(C(CC)C)O)=O)C(CO)C2)=O)cc(C)c2[nH]nnc2c1 38389,c1(C(=O)NCC(CNC(c2c(C(=O)OC)cco2)=O)F)ccc2nn[nH]c2c1 38390,C1(C(C)NC(CC=C)=O)CCCCN1C(c1nc(C(F)(F)F)sc1C)=O 38391,N1(C(CC2C3CN(C(=O)NC4(C)CCCC4O)CC32)=O)CCn2cncc2C1 38392,c1(C(=O)NC2CC3(CC(NC(CCC(CC)C)=O)C3)C2)ccc2c(c1)CCN2 38393,C1(NC(C2CC(C(C)C)C2)=O)CC2CCC1CN2C(=O)CCc1nncs1 38394,C1(CC(=O)NCC(CC2CC2)CO)C2CCCC2N1C(=O)CC1CC2(CCC2)C1 38395,C1(NC(CCCC=C)=O)CCC2(CC1)CC2NC(c1c(C2CC2)cnn1C)=O 38396,n1(C2(C(=O)NC(C3CCN(C(C45CCC4C5)=O)C3)C)CC2)cc(Cl)cn1 38397,C1(C(N2CCCC(C)C2CNC(c2ccoc2Cl)=O)=O)CCCC2CCCN12 38398,C=C(C)CCC(C(=O)Nc1ccc2c(c1)OCO2)N1C2CCC1CC(O)C2 38399,CC1COC(CNC(=O)CCOCC(F)F)CN1C(c1cc(C(N)=O)c[nH]1)=O 38400,CCN=c1[nH]c(C(=O)NCC(C)(C2CC2)NC(=O)CSC(F)(F)F)cs1 38401,c1(C(=O)NCCCn2cc(C(C)(C)C)nn2)ccc(CC#N)cc1F 38402,c1(C(N2CCC(CNC(C(C=C)O)=O)CC2C)=O)c[nH]c2c(F)cccc12 38403,O=S(=O)(CCCCc1c[nH]nn1)N1CCCC1.C1(c2ccc(F)cc2)(N)CCCCC1 38404,N1(C(Cc2ncc(C)s2)=O)CC2CC(NC(c3cn(C)nc3C(F)(F)F)=O)C2C1 38405,CC1=C(C(=O)N2CCC(C)(NC(C3CC4CC4C3)=O)C2)CCCO1 38406,c1(C(N(C(C2CCOCC2)C)C)=O)ccc(CNC(C2CC3(CC3)CO2)=O)cn1 38407,c1(CC)oc(C(=O)NCCC2(O)CN(C(=O)CCC(C)OC)C2)cc1C(=O)OC 38408,c1(C(=O)NC2(CCOC)CCN(C(c3cnncc3O)=O)C2)c[nH]cc(C)c1=O 38409,Cc1cc(F)ccc1C(=O)NC(c1cc(F)cc(Br)c1)CNC(C1CC1F)=O 38410,c1(NC(C2CN(C(c3c(I)ccnc3Cl)=O)CCN2)=O)ccc(Br)cc1Cl 38411,CC1CCC(C)(NC(=O)NCC2CNCC23CCC3)C1(C)C 38412,c1(CNC2CCC3(CN(C(c4cnccc4Cl)=O)C3)C2)ccc2ncccc2c1 38413,c1(C(=O)NCC2CC(NC(C3(S(N)(=O)=O)CC3)=O)C2)cn2cc(Cl)cnc2n1 38414,C1(CC(=O)N(C)CC2CN(C(=O)Cc3cnsc3)C2)OCCC1(C)C 38415,C12(C(N(C3CCCN(C(C(CC#C)O)=O)C3)CCO)=O)CCOC(C)(C1)C2 38416,CN=c1[nH]cc(C(=O)NC2CCOCC2C(=O)NCc2cc(Cl)ccn2)s1 38417,C(CC(=O)N=c1ccn(CC(N)=O)[nH]1)OCCN(C)C(C1(C)CCC(=O)N1)=O 38418,N1(C(=O)NCc2nc(C(=O)OCC)on2)CC(C2CCC2)CCC1C 38419,C(=O)(CC(O)(c1ccccc1)C1CC1)N(CC(C)NC(c1c[nH]c(=N)s1)=O)C 38420,c1(C(=O)NC2CC(C)N(C(=O)CC3CCCCCCC3)C2)coc2c1CCCC2 38421,C1(C(N2C(CNC(c3c(C)c[nH]n3)=O)CC3CC32)=O)CCc2nc(O)[nH]c2C1 38422,C1(C(=O)NCC(CCNC(c2ccc(Cl)o2)=O)OC)CCCCC12CC2 38423,c1(C(=O)NC2CC(CNC(C3CC4CC4C3)=O)C2)cccc2ccnn12 38424,N1(CC(=O)NC2CC(C)(CNC(c3n(C)c(S)nn3)=O)C2)C(=O)NC(C)(C)C1=O 38425,N1(C(c2nn(C)c(=O)cc2)=O)CCC(NC(=O)CC2CC2C(C)C)CC(C)(C)C1 38426,N1(C(CP(C)(C)=O)=O)CC2CC1CN2C(c1[nH]cc2c1CCC2)=O 38427,c1(C(N2CCC(C3(NC(C(C)C(C)O)=O)CC3)C2)=O)coc2c(F)cccc12 38428,c1(C(=O)NC(C2CCN(C(=O)C(F)(F)C3(O)CCC3)C2)C)cnc(S)n1C 38429,O=C(CC(C(F)F)c1cccc(F)c1)NCC1CC1CNC(=O)CO 38430,N1(C(c2cc(OC)ncn2)=O)CCN(C(C2(CC3CC3)CCCO2)=O)CC1C 38431,C1(C(NNC(c2cccc(C)c2)=O)=O)C2CC3C1C3C2F 38432,N1(C(CCC(=C)Cl)=O)CCCCC(CNC(C2CCCN(CC)C2)=O)CC1 38433,C(C(C)CC(=O)NCCCC(C)(C)NC(=O)CN(S(C)(=O)=O)C)OC(C)=O 38434,C1(NC(c2ncoc2CCC(=O)OC)=O)CCC(NC(C2C=C2C)=O)CC1 38435,C(=O)(CC(O)COC)N(CC(C1CCCC1)OC)C 38436,C(CC(=O)NCC1(F)CCN(C)C1)(C(F)(F)F)NC(C1(OC)CCOC1)=O 38437,C1(NC(CNC(C(C)(C)C)=O)=O)CN(C(=O)Cn2nnc(=O)[nH]2)CC12CC2 38438,CCCC(C)(O)CC(=O)N1CC(CC(N2CCC(C)(CCO)CC2)=O)(OC)C1 38439,N1(C(C(C)C2CC2)=O)CCOC(C)(CNC(c2cc(CO)on2)=O)C1 38440,C1(C(=O)NC2C(c3cn(C)nc3)C2)N(C(=O)CC2CCC=CCC2)CCC1(C)C 38441,C(=O)(C(CC(C)CCC=C(C)C)N1CCC(C(=O)NC)CC1)NC 38442,Cc1ccc(CN2CCC(C(=O)NCc3cccnc3F)C(O)C2)cc1C#N 38443,CC(CN(C)C)N=c1[nH]c(N2CCC(C(C)(C)C)C2)nc2c(F)cccc12 38444,Cc1nc(O)ccc1C(N1CC2CC2(CNC(C2(F)CCOC2)=O)C1)=O 38445,C(CNC(c1cc(Br)no1)=O)(C(C)(C)C)NC(c1ccc(C(=O)OC)s1)=O 38446,N1(C(C(n2cc(Cc3ccc(C(C)=O)o3)nn2)C)=O)CC(=O)N2CCOCC2C1 38447,C(=O)(CCCC(C)C)NC1C(SC)CN(C(=O)C(C)Cc2ccco2)C1 38448,C(C(C)(CNC(C12CC(NC(=O)CC3CSCCO3)(C1)C2)=O)CO)OC 38449,C1(CNC(c2n[nH]c(C)c2O)=O)(NC(=O)C(C)SC(F)(F)F)CCC(C)(C)CC1 38450,CC(=O)CCCC(=O)N1C2CCC(C2)C1C(=O)Nc1cn(C)nc1C#N 38451,c1(OC)ccc2oc(C(=O)NC3(C#N)CCN(Cc4ccccc4I)C3)cc2c1 38452,C1(N(C(C(CC)O)=O)C)C2CN(C(=O)CCCNC(=O)OC)CC12 38453,c1(C(=O)N(C2CC2)CC2CCN2C(=O)CCc2ccon2)cc(C(F)(F)F)n[nH]1 38454,c1(C(=O)NC2C(CNC(CSCC(C)C)=O)CCC2)nnc(O)cc1O 38455,Cc1cc(=O)n(C)cc1NC(C1CC12CC(NC(=O)C(C)CN(C)C)C2)=O 38456,C(=O)(C(C)C(O)C(C)C)NCCCC(C(N1CCCC(C)(CC)C1)=O)O 38457,C1(C(N2CC=CC2Cn2cc(CCN3CCSCC3)nn2)=O)C2COCC12 38458,C1(C(=O)NC(c2cc(F)ccc2OC)CC)CC2(CCC(N)CC2)C1 38459,c1(OC)cc(C(N2CCC(O)(CNC(=O)CCC3(C)CC3)C2)=O)cc(F)n1 38460,S(=O)(=O)(c1ccc(N2CCC3CCCC3C2)cc1Cl)NCC1N(C)CC(O)C1 38461,c1(OC)ccc(C)cc1CNC(=O)Nc1cccc(N2CCCCC2=O)c1 38462,Cc1nc2ccc(C(N3CC(C)OC4(CCC4)C3)C(=O)NC3CCOC3)cc2s1 38463,C12(CNC(C(C)NC(=O)NC)=O)CC1CN(C(=O)C=Cc1c[nH]nc1C)C2 38464,c1(C(=O)NCc2scc(C(=O)NCCCS(N)(=O)=O)c2)cncc2[nH]ccc12 38465,N1(C(C(C)c2cccs2)=O)CCC(N(CCO)C(C2C(C)C2(F)F)=O)CC1 38466,CC1(C2CCN(CC(N)Cc3ccccc3Cl)CC2)CC1 38467,C1(C(=O)NCC(CC)OC)C=CCN(C(C2(C)CC3CC3C2)=O)C1 38468,N1(C(C(=O)NC(C(CC)C)=O)CCO)CCc2sccc2C1 38469,N1(CC(N2CCCC(C3N(C(C(CC)CC)=O)CCC3)C2)=O)C(=O)CN(C)C1=O 38470,C1(C(N(CCC(C)NC(c2cc(-c3ccns3)on2)=O)C)=O)CC(O)CN1C 38471,N1(CC(=O)NC2CC2CNC(C2(F)CC2)=O)CCCc2sccc2C1=O 38472,c1(C(=O)NCc2cn(CCCCCO)nn2)cc2c(=O)cc[nH]c2s1 38473,S(=O)(=O)(C1CC2C(C1)C2(F)F)N1CCC(N(C2CCCC2)C)C1 38474,c1(C(=O)NC(CNC(CC(CCC)C)=O)C(C)(C)C)ccc(C)c([N+](=O)[O-])c1 38475,C(CCCCNC(=O)C(C)NC(=O)C1CC1)NC(C(C1CCOCC1)OCC)=O 38476,C1(NC(c2cc([N+](=O)[O-])n[nH]2)=O)CCN(C(=O)COCC2CC2)CC1F 38477,N1(C(c2ccc(C(C)=O)o2)=O)CCC(O)(CN(C)C(C2CCNC2=O)=O)CC1 38478,C1(NC(C(C)SCC)=O)CCCN(C(C23CC(CC)(C2)C3)=O)C1 38479,N1(C(CC2(N(C)C)CCC2)=O)C(C(=O)NCCCCC)CCC1C1CC1 38480,CC1CN(C(=O)CC2CC2CNC(=O)CCc2ncccn2)CC1(F)F 38481,c1(C(=O)NC)cn(CC(N2CCC(CNC(C3CC=CCC3)=O)C2)=O)nn1 38482,N1(C(C2(C)C(C(=O)OC)C2)=O)CCOC(CCNC(=O)CCSCC(N)=O)C1 38483,c1(C(N(CC(CN(C(=O)COCCOCCO)C)O)C)=O)c(N)cccc1Cl 38484,C1(=CCNC(c2cc(CCC)on2)=O)CCN(C(=O)C(C)(COC)OC)CC1 38485,C=CC1CCCCN1C(=O)COCCC1CCN(C(=O)OC(C)(C)C)CC1 38486,N1(C(CCC2CCN(C(C3N(CCC)CCC3)=O)C2)=O)CCC(O)CC(C)C1 38487,C(C(C)(C)C(=O)NOCC1(C)CC1)N(C(c1ccc(C(C)C)o1)=O)C 38488,N1(C(C(=O)N(CC)CC)=O)CCCC(N(CC(C)C)C)CC1 38489,N1(C(c2c(CC)c(F)ccc2)=O)CCC2(CCN(C(C3CCCS3)=O)CC2)C1 38490,N1(C(C2=CC(C)(CC)C2)=O)CCN(C(c2c(C(C)C)n[nH]c2C)=O)CCC1C 38491,CCC(CC(=O)NC(CC1CCC1)C(N1CC(C2=NOC(C)C2)C1)=O)CC(C)C 38492,N1(C(C(CC2CC2)OC)=O)CCN(C(=O)Cc2cnn(C)c2C)CC(C)C1 38493,c1(C(=O)NCC(C)CNC(=O)CCc2cn(C)cn2)cccc2c[nH]nc12 38494,Cc1csc2c(C(=O)NC3(CCNC(=O)C=Cc4ccoc4)CCC3)cccc12 38495,N1(C(C2C(OC(C)(C)C)C2)=O)C2CCC1CC(O)(CNC(=O)C(F)C(F)(F)F)C2 38496,C1(CNC(CCc2c(C)ncs2)=O)CCC2CN(C(=O)Cc3cnsc3)CCC2C1 38497,C(C(=O)NCC1CCCCC1NC(c1cocc1C(=O)OC)=O)(C(C)C)OCC 38498,N1(C(C2C(C(C)(C)C)C2)=O)CCC2(CC1)CC(NC(c1ncc(F)cn1)=O)C2 38499,c1(CC(=O)NC2C3CCN(C(c4nc(C)oc4)=O)C32)c(C)cccc1C 38500,C1(COC)(NC(=O)CCC2CCCCC2)CCN(C(=O)C#CC(C)(C)C)CC1 38501,C1(COC)(CNC(C2CN3CCC2C3)=O)CCN(C(c2[nH]nnc2C2CC2)=O)C1 38502,c1(C(=O)NCC2(C(C)(C)C)CCN(C(C34CC(C)C3C4)=O)C2)cccc(CO)c1 38503,c1(C(=O)NC(CCNC(C2CCC(C(=O)OC)C2)=O)(C)C)nc(C)sc1Br 38504,S(=O)(=O)(c1ccsc1C(=O)NC1C=CCN(C(=O)CCF)C1)N1CCCC(C)C1 38505,C1(NC(CC(CNC(CC(CC)OC)=O)C)=O)CC12CCOCC2 38506,CC(CCCCNC(C1(NC(=O)CC2COC3CC2C3)CCCOC1)=O)N(C)C 38507,C1(NC(c2nnnn2CCOC2CCOC2)(CC)C2CC2)CCC2(CC1)CSC2 38508,c1(C(N2CCC(C(N3CCCN(C)CC3)=O)CC2)=O)ccc2cccc(Br)c2c1 38509,c1(OC)ncccc1CNC(=O)CCC1CCN(C(=O)C(=O)NC2CC2)C1 38510,Cc1nc(C=CC(N2CC(NC(=O)CC3CCCCCO3)C(F)C2)=O)[nH]c1C 38511,C(=O)(CCCNC(=O)C1CC1)NC(CN(C(c1cnc(Cl)[nH]1)=O)CC)C 38512,CC(C(=O)N1CCOCC(CNC(=O)CNC(C2CCOCC2)=O)C1)S(C)(=O)=O 38513,C1(C(N2CC(CCNC(C3(C)CC3(C)C)=O)(OC)C2)=O)CN2CCN1C(C)C2 38514,c1(N2CC(C)(C)N(CCO)CC2)nc(N2CC3CCC(C2)O3)c2ncsc2n1 38515,CC1CCN(C(c2ccc(O)nc2)=O)CC1NC(c1cnc(C(C)(F)F)s1)=O 38516,c1(C(=O)NC2(C3CCCCN3C(=O)C(F)=C3CCC3)CC2)cc(Cl)c(F)c(Cl)c1 38517,c1(C(N2CCC(NC(c3ncc(CC)nc3)=O)CC2)=O)c(C)oc(C)c1C 38518,C1(CNC(C(C(C)C)CO)=O)C2CCCC1N(C(c1cnc(C(C)(C)C)o1)=O)C2 38519,c1(N2CC(C)(CNCCNC(CCC(=O)NC)=O)OCC2)ncnc2scnc12 38520,N1(C(C(C(C)(C)C)OC)=O)CCC(C2(NC(c3scc4c3OCCO4)=O)CC2)C1 38521,CCC(CCC(=O)NC(CC)C(C)C)NC(c1sc(F)cc1C)=O 38522,C1(c2nnnn2CSc2ccccc2)(CC=CC)CC2c3ccccc3CCC12 38523,Cc1cc(=NCC2(O)CC3C=CC2C3)[nH]c(N(C)CCOc2cccnc2)n1 38524,CCC(CC(=O)N(CCNC(c1c(C)nnn1CC)=O)C1CC1)C(F)F 38525,C1(CCCCNC(=O)CC2COCCO2)CCN(C(=O)CC2C=CCC2)CC1 38526,c12c(cnn1C)C(=O)N2.C1(NC(C(C)OCC)=O)CCN(CC)C1 38527,N1(C(c2cc(C)oc2C)=O)CC(CO)C2(CCN(C(=O)C(C)C(C)O)CC2)C1 38528,C1(NC(c2c(C)onc2CO)=O)CC2CC1N(C(=O)C(=CC1CCCCC1)F)C2 38529,C1(C(=O)NCCc2ccccc2C)(COC)C=CCN1C(=O)C=Cc1ccsc1 38530,c1(NC(c2c(C)nco2)=O)cccc(NC(=O)C=C(Cl)Cl)c1 38531,N1(c2c(C)noc2N2CCc3c(Br)cccc3C2)Cc2cc(Br)ccc2C2CC1C2 38532,c1(CCC(=O)N(CCC)CCNC(C2CC3CC2C3)=O)ccc2c(c1)CCCO2 38533,c1(N(C2CC2)CC)nc(C(=O)OC)cs1.C1(=O)C(C)N1 38534,CC1(C)Cc2cccc(C(N3CC(C(=O)O)C(c4ccccc4)C3)=O)c2O1 38535,N1(C(C(CC)(C)O)=O)CC2(CC2)CC1C(=O)Nc1ncc(Br)nc1C 38536,C#CCC(C(=O)N1CCC1)NC(C1CC1C(F)(F)F)=O.c12cn(nn1)C2 38537,N1(C(=O)OC(C)(C)C)CC2C(NC(=O)Cc3ccc(Cl)cn3)C2C1 38538,C=CC(O)(C(=O)N1CCCCCC(NC(c2sc(C)c(C)c2C)=O)C1)C(F)(F)F 38539,C1(CN(C(CC=CC=C)=O)C)CCC(CNC(=O)CC2CCCO2)CC1 38540,C1(C)CN(C(=O)C(c2nc(C)cs2)C)CCO1.n12ccc(n1)CC(=O)N2.CC 38541,Cc1cccc(C(CNC(c2ncncc2C)=O)NC(c2cn[nH]c2)=O)c1 38542,C1(C(=O)Nc2c(CC)csc2)CCN(C(c2ccc(=O)n(C)c2)=O)C(C)(C)C1 38543,C(C(C)(CC(C)C)NC(=O)Cn1ccc([N+](=O)[O-])n1)NC(C1C(OC)CC1)=O 38544,CCC(C)CCCC(=O)NCCCC(C)(C)C(=O)N1CCC12CCCSC2 38545,c1(N2CCC(C)C2CNC(c2ccc[n+]([O-])c2)=O)nc(Cl)ncc1C(F)(F)F 38546,N1(C(c2c(C)ccs2)=O)CCCCC1C(=O)Nc1cccnc1C(N)=O 38547,c1(NC)ccc(CCC(=O)NC2CN(C(=O)CC3CCCN3C)CC2OC)cc1 38548,N1(C(CCC2CCCC(=O)N2)=O)CCCN(C(C23CSC(C2)C3)=O)CC1 38549,c1(C(=O)NC2CC(CNC(C3CCCO3)=O)C2)cscc1Cl 38550,C1(CC(=O)NCCCNC(CNC(=O)OCC=C)=O)CC2(CCC2)C1.OC 38551,Cc1csc2ncc(C(=O)NC34CCCC3N(C(=O)COCCC(C)C)CC4)n12 38552,C1(CN(C(C2CCCC(=O)N2)=O)CC)CCN(C(=O)C=CCCC(C)C)CC1 38553,n1(C(C)C)ccc(C(C)NC(=O)CC2CCN2C(=O)CCCn2cncn2)n1 38554,Cc1ccc(C)c(NC(c2ncoc2CNC(C2CCS2(=O)=O)=O)=O)c1 38555,c1(C(=O)NC(C2CN(C(c3ccsc3)=O)CCO2)C)c(O)cccc1O 38556,C1(OC)CCC(C(=O)NC(C2(O)CN(C(=O)CN3CCNC(=O)C3)C2)C)CC1 38557,C1(C)(C(=O)NCCCCN(C)C(C2CC2c2ccccc2)=O)CC(C2CC2)=NO1 38558,CC1CCN(C(=O)Cc2cnns2)CC1NC(=O)C=CC1CCCCC1 38559,c1(C(=O)NCc2c(C(N3C(C(C)C)CC3)=O)occ2)ccc2nccn2c1 38560,Cc1c(Cl)cc(CNC(=O)C(=O)N(CC(c2ccc(Br)cc2)O)C)cc1I 38561,C(CC(C)(C)C)(C(=O)N1CCC(CF)(NC(=O)CSC(F)(F)F)C1)OC 38562,C1(CNC(CC=CC)=O)COCCN(C(C2(C)CC=C(C)CC2)=O)C1 38563,C1(C(=O)NC2CN(C(c3cnc(-c4ccoc4)s3)=O)C2)CCc2nncn2CC1 38564,Cc1ccc(CC(N2CCC(C(C)NC(=O)C(C)CCO)C2)=O)cc1 38565,c1(OC)nc(Cl)c(C(N2CC=CC(NC(=O)COC3CC3)C2)=O)s1 38566,c1(NC)cccc(OC)c1C(N1CC(CO)(NC(C2CC(Cl)=NO2)=O)C1)=O 38567,C1(CN(C(=O)CCCC2OCCO2)CC)CCCN1C(=O)CCCC1CC1 38568,Cc1cc(C(=O)N(C)CCN(C(=O)CCCc2c(F)cccc2F)C)ccc1Cl 38569,C12(C(N3CCN(C(C(C)=CC)=O)C(CC(F)(F)F)C3)=O)CCC(N=[N+]=[N-])C1C2 38570,N1(C(Cc2cc(C)no2)=O)CC(CNC(=O)CCCc2cnn[nH]2)C(C(F)(F)F)C1 38571,c1(CC)cccnc1C(=O)NC1CCC1CNC(c1ccn(CC(F)(F)F)n1)=O 38572,Fc1cc(NC(=O)CCC2CCN2C(C2CC2)C2CC2)ccc1Br 38573,CCCCC(O)C(=O)NCC(CC(C)C)NC(c1cnn(C)c1OCC)=O 38574,c1(OC)ccc(NC(C2CC2C2CN(C(c3c[nH]c(C)c3)=O)C2)=O)cc1C 38575,c1(OC)cc(C(=O)NCC2(NC(C3CCN(C)C3C)=O)CCOC2)ncn1 38576,C1(C)(NC(C(C2CCOCC2)OC)=O)CCCN(C(=O)Cc2cccnc2C)C1 38577,C(C(C)(O)CCO)NC(c1c(CNC(C2C(CC)CCO2)=O)cco1)=O 38578,c1(CCC)onc(C)c1C(=O)N(C)Cc1ccc(Br)nc1 38579,CCCC(C#N)C(=O)NCCN(C(=O)C(CSC)OC)C(C)C 38580,N1(C(c2c(C)c(N)cnc2)=O)CC2CCCC2(NC(=O)Cc2ccccc2Cl)C1 38581,N1(C=O)CCC(N2CCSCC2)CC12CCC2.CC(C)(C)OC(=O)NCCCSN 38582,C1(NC(CCC=CC(C)C)=O)CC(C(=O)NCCN2CCCNC2=O)C1(C)C 38583,c1(OC)ncnc(C)c1C(N1CC2C(CNC(=O)CCCC(C)C)C2C1)=O 38584,c1(NC(C2(O)CCN(Cc3c(C)cccc3Cl)C2)=O)cc(F)cnc1C#N 38585,C=CCCCCCCCC(=O)NCC(C)NC(c1c(N)cc(F)cc1F)=O 38586,c1(C(=O)NCCCN(C(=O)CCC2CC(F)(F)C2)CCC)ccc(CC)cc1N 38587,c1(OC)cc(Cl)cc([N+](=O)[O-])c1NC(=O)CC1COCCN1c1nccc(C)n1 38588,C1(CNC(Cc2cnc(C)o2)=O)CC2(CCC2)CN1C(=O)CC(C)(F)F 38589,C(=O)(C(CC(F)F)NC(=O)CN1CCCCC1C)N(C(c1cc(C)on1)C)C 38590,c1(C(N(CCC)CCNC(C2CCC2C)=O)=O)coc2ccc(OC)cc12 38591,C1(SC)C(=O)NN2CCCC2C(=O)N1.N1(CC)Cc2cccc(F)c2C1 38592,c1(CC)c(OC)cccc1C(=O)NC(CNC(C1COCCC1(F)F)=O)C(C)C 38593,N1(CC(=O)N(CCC(=O)NCCC2CC2C)C(C)C)CC2CCC1C2 38594,N1(C(C(CC)NC)=O)CCC2(CCCN(C(=O)Cc3ccc(Br)nc3)C2)CC1 38595,N1(C(C(C2CCOC2)OCC)=O)CC2(CCCC2NC(=O)CC2CC2)C1 38596,N1(C(c2c(C)cc(N)cn2)=O)CC2COCC2(C(N2CCC(O)(C(N)=O)C2)=O)C1 38597,c1(OC)cc(OC)c(C(N2CCN(Cc3cncc(C)c3)C(C)C2)=O)cc1Br 38598,CCC(CC(F)F)C(=O)NC1CCCCN(C(C2CCCN(CC(C)C)C2)=O)C1 38599,CCCCC(C(=O)NCC1CC(OCC)C1)NC(c1ccoc1CC)=O 38600,Cc1ccc(Cl)c(O)c1C(=O)NCCCCC(C)NC(c1c[nH]nc1C)=O 38601,N1(C(c2cc(C)sc2Br)=O)CCC2C(C1)CN2C(c1nocc1C)=O 38602,c1(C(=O)NCC(C)CN(C)C(C2CC(C(C)(C)C)=NO2)=O)ccc2n[nH]cc2n1 38603,C(c1cnc(C)nc1O)=CC(=O)NC1CCN(C(CCCCC=C)=O)CC1CC 38604,c1(C(=O)NC2CCN(Cc3c(C)ccs3)CC2)cc(F)cc(Cl)c1 38605,c1(C(N2CCC(N(C(=O)CNC(C3CCC3)=O)C)C2)=O)ccnc(O)c1 38606,C12(OC)CCCCC(C(=O)N(CC(C)NC(=O)CCn3ccccc3=O)C)(C1)C2 38607,c1(C(N(C)Cc2cccc(C#N)c2)=O)cc(Br)c(F)cc1F 38608,C12(C(=O)NC3CN(C(C4CCN(S(C)(=O)=O)C4)=O)C3)CCCC(=O)N1CCC2 38609,c1(C(N2CCN(C(C(CC=C)C)=O)CC2)=O)ccc(C)c2cccnc12 38610,N1(C(CC2C(C)(C)C2)=O)CCC(NC(c2cc(N)c(O)c(F)c2)=O)C(F)(F)CC1 38611,C1(F)(C(=O)NC2CC(NC(C=CC(C)(C)C)=O)C2)CCCOC1 38612,CN1CCC2CN(C(C3CCN(C(c4cc(Cl)ncn4)=O)CC3O)=O)CC2C1 38613,Cc1nc(Cl)[nH]c(=NCC2CC(CNC(=O)CC3CCCCO3)CO2)c1Cl 38614,C1(NC(C(c2n(C)cnc2)O)=O)CC2(CCC(NC(C3OCCCO3)=O)CC2)C1 38615,c1(C(=O)NC2CC(C)(NC(CCC(C)OC)=O)C2)csc2cc(C)ccc12 38616,C(CN=c1[nH]c(=NC(C)CCN(C)C)c2ccc(OC)cc2[nH]1)NC(=O)OC 38617,c1(CC)cc(C(N2CCC(NC(c3cc(O)ncn3)=O)C2)=O)ccn1 38618,Cc1cc([N+](=O)[O-])c(Cl)cc1S(=O)(=O)NCCOC1CCC1 38619,n1(CCC)cc(Cl)c(C(=O)NCC23CC2CN(C(=O)Cc2conc2C)C3)n1 38620,c1(COC)nccc(=NC2CCC3CN(C(c4n[nH]c(C)c4O)=O)CC23)[nH]1 38621,Cc1nnc2n1CC(C(=O)NCC1CCC1NC(=O)C(C)c1cc[nH]n1)C2 38622,C(=O)(CCCC(C)(C)NC(c1n[nH]c(C)c1O)=O)N1CCC(OC)C(C)C1 38623,C(=O)(C(C)(F)CCCC)NC1CCCCN(C(c2cn(CCC=C)nn2)=O)C1 38624,N(C1CCCn2cnnc21)C(CC(C)N(C(C(C1CCCCC1)C)=O)C)=O 38625,c1(C(N2CCC(c3nc(C4CC4)no3)C2)C(=O)NCC=C)cc(Cl)cnc1OC 38626,c1(OC)ccc(C(CCO)NCC2CCC3(CC3)C2)cc1 38627,N1(CCC2CC(N(CC(=O)N3CCC3)C(C3CC(=C)C3)=O)C2)CCCOCC1 38628,C(=O)(C1Cc2ccccc21)N1CC(C)N(C(=O)CCC2CCC(=O)N2)CC1 38629,N1(C(CN(C)C2CC2)=O)CCC(CNC(c2cnnc(C3CC3)c2)=O)C(F)(F)CC1 38630,C1(C)(COC)CCCN(C(=O)Cn2cc(CNC(C3(C#N)CC3C)=O)nn2)C1 38631,C1(CN(C(CNC(C)=O)=O)C)CCCN(C(=O)C(N2CCCC(O)C2)C)C1 38632,C(=O)(CCCCC(C)(C)C)N1CCC(NC(c2c(C(C)C)onc2)=O)C1 38633,c1(OCC)cc(C(=O)NC2CCC(O)CC2)c(-c2nccs2)cn1 38634,N1(C(CCC#CC)=O)CCCC(NC(=O)Cc2c(O)ncnc2O)C(F)C1 38635,C(CCCCCC(C(=O)NC(=O)OC(C)(C)C)N1CCOCC(C)(O)C1)SC 38636,C(=O)(C1=C(C)S(=O)(=O)CC1)N1CC(NC(COC)=O)C(F)C1 38637,N1(C(COCCCOC)=O)CCC(C)(C(=O)N(C)Cc2cnccn2)C1 38638,N1(C(CCC(C)C)=O)CC(C(=O)NCC(=O)N=S(C)(C)=O)CCC1(C)C 38639,N1(C(c2nc(C)sc2C)=O)CCC(C2CCCN(C(c3ccnn3C)=O)C2)C1 38640,N1(C(c2c(C)cnnc2)=O)CC2(CC(NC(=O)C(C)CN(C)C)c3nccn32)C1 38641,C(=O)(C#CC(C)(C)C)N1CC(OC)C(NC(c2ccccc2SC(C)C)=O)C1 38642,c1(CC)nn(C)c(CC)c1CC(=O)N(CC(O)CNC(c1cnnn1CC)=O)C 38643,N#CC1CCC(N=c2cncc[nH]2)C1C1CC1 38644,C(CCCCC(=O)N1CC(O)CC1(C)C(=O)N(C)Cc1ccncn1)OCC 38645,c1(C(N2CCN(CCCNC(C3C(=C)C3)=O)CC2)=O)nn(C)cc1[N+](=O)[O-] 38646,C1(C2CCCN(C(c3ccn4ncccc34)=O)C2)(NC(c2n(C)cnc2)=O)CC1 38647,C12(NC(CC(CC)C)=O)CCCC1N(C(c1c(OC)cc(OC)cc1N)=O)CC2 38648,N1(C(C(CC)OCC)=O)CCCC(C2CN(C(c3cccc4[nH]ncc34)=O)C2)C1 38649,Cn1cc(-c2nc(C(c3nnnn3C3COC3)NC(CF)CF)cs2)cn1 38650,c1(C(C)C)conc1CC(N1CC(CCNC(c2c[nH]nc2C(C)(C)C)=O)C1)=O 38651,C12C=CCCN1C(=O)CNC2=O.CCC(=O)NCCC 38652,N1(C(=O)CO)CCC2(CCC2)C(NC(=O)CCOc2cccc(Cl)c2Cl)C1 38653,N1(C(CCCc2nnc(C)n2C)=O)CCCC(NC(=O)CC2CCCCC2)C1C 38654,c1(N(CCN2CCCC23CCC3)CC)ccc2c(c1)OCO2 38655,c1(N(C)C)nc2cc(C(=O)NC3CC(NC(=O)COC4CC4)C3)ccc2o1 38656,CCCC(CCC)CC(=O)NC(CCC1CC1)C(=O)N1CCC1CC(=O)NC 38657,N1(C(c2cc(C)c(F)cc2)=O)CCC2CCN(C(C3CCCCNC3=O)=O)C2C1 38658,c1(C(N(C2CC(C)(NC(=O)CC3CCC3)C2)C)=O)ccc(NC(=O)C2CC2)cc1 38659,N1(C(C(C(C)O)N(C)C)=O)CCOCC(C)(CNC(c2coc(CO)c2)=O)C1 38660,c1(C(N2CCC(O)(CNC(c3ccc(OC)nc3)=O)C2)=O)ccc2cc[nH]c2c1 38661,C(C)(CNC(C1(C(C)(C)C)CCCCC1)=O)(C(C)C)NC(Cc1nnc(C)o1)=O 38662,C(=O)(C(C)(C)CCCNC(=O)C(F)C1CCOC1)NC(C)Cn1cnnc1 38663,N1(C(C2CN(C(C(CC)(C)COC)=O)CC(C)C2)=O)CCOC2C(O)CC12 38664,CC(CO)CCCNC(C1CCCN(C(=O)Cc2cccc(F)c2)C1)=O 38665,C(=O)(CCCCC(C)C)N1CCC(CC)(NC(C2C(C(=O)OC)CCC2)=O)CC1 38666,C1(C(N(C(CNC(C2N(CC#C)CCC2)=O)C)C)=O)CCc2nncn2C1 38667,C(=O)(C1=NN(C)C(=O)CC1)NC1CCN(C(CC)=O)C(C2CC2)C1 38668,c1(C(N2CCC(N(C(=O)CSc3nnnn3C3CC3)CC)C2)=O)cncc(N)n1 38669,C(Cn1cncn1)(C(=O)N(C)C(C1CCOCC1)C)NC(C=CC)=O 38670,N1(C(=O)Nc2nccc(OCC)c2)CCCN(CC)CC1.C(C)(=O)O 38671,C1(CC(=O)N(CC(C)C)CC(C)NC(=O)CC=CC(C)(C)C)OCCC1(C)C 38672,N1(C(C(=O)Nc2cc(OC)ns2)=O)CCC(c2ccccc2)C(OC)C1 38673,c1(C(=O)NCC2(C)CCN(C(C(C)C3CCCC3)=O)C2)ccc(N)c(F)c1F 38674,C1(C)(C(=O)NC2CCC(C)N(C(C3C=CCCC3)=O)C2)Cc2ccccc2C1 38675,C1(C)(CNC(C(C2CC=CCC2)NC(CN(CCOC)C)=O)=O)CCCO1 38676,Cc1ccc(C(=O)NCC2CCC(C)N(C(=O)C3=NNC(=O)CC3)C2)c(Cl)c1C 38677,C1(N(C(COCCCCCC)=O)C)C2CN(C(C3CC3c3cccs3)=O)CC12 38678,c1(C(=O)NC(CNC(c2ccc(C)cn2)=O)(C)C)cc(C2CCC2)n(C)c1C 38679,Cc1nnc(N2CC=CC(NC(=O)CCC(C)(C)C)C2)nc1C 38680,C(CCCC(=O)N1CCC(C(C)NC(=O)CC2(C)CCOCC2)C1)N(C(C)C)C 38681,O1NC(=O)CC2(CCCC2)C(=O)NCC1.c1(C(=O)O)ccns1.CC=C 38682,N1(C(C2C(C)OCC2)=O)C2CCC(C(=O)NC3CCCCCC3F)C1CC2 38683,c1(OCC(=O)NC2(C)CN(C(Cc3cnc(C)[nH]3)=O)C2)ccc(Br)c(F)c1F 38684,c1(CCC(=O)NCC(C)NC(c2cc(N(C)C)ccc2N)=O)ccc(F)cc1F 38685,C(CC(O)C(=O)NC1CCCC1NC(C1(C2(C)OCCO2)CC1)=O)N(C)C 38686,c1(C(=O)Nc2ncc[nH]2)cc2ccc(-c3ccc4c(c3)CNC4=O)nc2[nH]1 38687,N1(C(COCCCC#C)=O)CCCCCC1CNC(C1CC12CC(F)(F)C2)=O 38688,c1(OC)cccc(C(O)C(N2CC(NC(c3nc(C)nn3C)=O)C(C)C2)=O)c1 38689,C1(C(N2CCC(CN(C)C(c3ncc(F)cc3N)=O)CC2)=O)CCCC(F)(F)C1 38690,CC1(C)CN(C(=O)CCCCC2CC2)CC1NC(c1cnn(CC(F)(F)F)c1)=O 38691,C(=O)(N=c1[nH][nH]c(C)c1Cl)C1CN(C(c2cnc(OC)c(Br)c2)=O)CC(F)C1 38692,c1(C(C)C)ccc(C(=O)NCC2CC(F)(CNC(C3(C)CC3(F)Cl)=O)C2)cc1 38693,C1(c2n(CCOC)nnn2)(NCc2cccc(Br)c2F)CCCC(F)(F)CC1 38694,c1(CC(=O)NS(Cc2c(CC)con2)(=O)=O)ccc(OC)nc1 38695,N1(C(Cc2ccc(C#C)cc2)=O)CC2CCC1CC2NC(c1c[nH]nc1CC)=O 38696,C1(CNC(Cc2cc(C)nn2C)=O)CCCCCN1C(C1CCC(C)(C)CC1)=O 38697,c1(C(=O)NCC(CN(C)C(C2CCC(C(F)(F)F)O2)=O)O)ccnnc1O 38698,c1(N(CC)CC)ccc(C(=O)NC(C)COC2CCOCC2)cc1 38699,CC1CCN(C(C2CCCCC2O)=O)CC1CNC(C1(c2ccccc2)CC1)=O 38700,C1(NC(C(C)=CC)=O)CC2(CCCN(C(C3CC3CCC)=O)C2)C1 38701,C1(C(N2CC(C(CC)CC)C2)=O)(NC(c2ccn(CCF)n2)=O)CCSC1 38702,Cc1ccc2sc(NC(=O)NCc3cc4cccc(C)c4o3)nc2c1 38703,C1(C=O)CC(C2CCCC2)C1.C(C(=O)NCCC1(CO)CC1)=CC=CC 38704,C1(C(N(CCCNC(c2ncoc2C2CC2)=O)C2CC2)=O)CCCC(O)C1 38705,C(=O)(CCS(C)(=O)=O)N(CCC(=O)N(C1CCCC(C)C1C)C)C(C)C 38706,N1(C(=O)Cc2cn(CC3CC3)nn2)CCC2CN(C(=O)CC3COCCO3)C2C1 38707,C1(C(N2C(C3CCN(C(C4CCCN4C4CC4)=O)C3)CCC2)=O)CC(=O)N(O)C1 38708,c1(C(=O)OC)n[nH]c2cc(-c3ccc(C(=O)Nc4ccc(Br)c(C)n4)o3)ccc12 38709,CC1(C)NC(=O)C2(CCN(C(=O)NCc3cc(C4CC4)no3)CC2)O1 38710,C(=O)(CCC(C)CN(C)C)N1CCC(O)(CCNC(C(CC=C)C)=O)C1 38711,N1(C(c2cc(CC)no2)=O)CCC(C)(C)CC1C(=O)NC1CC12CCCC2 38712,CC1(OC2(CNC(=O)CC3CC=CCC3)CCOC2)CCCC1.C1C(=O)N1 38713,c1(CN2CCN(CCSC)CC2)ccc(C(=O)NCc2cn(CCC)nc2)cc1 38714,n1(C(C)(C)C)cc(NC(C2(F)CN(C(=O)Cc3ccnnc3O)C2)=O)ccc1=O 38715,C(C(=O)N=c1ccn(CCF)[nH]1)=CC(C)NC(C1CC2(CC2)CN1C)=O 38716,Cn1ncc(CC(C(=O)N2CC(c3ccccc3)C2)NC(=O)OC(C)(C)C)c1O 38717,c1(NCc2cn(CC(C(=O)OC)O)nn2)cccc(C(=O)O)c1 38718,Cc1c(Cl)ccc(C(N2CCCC(NC(=O)C#CC(C)(C)C)C(F)C2)=O)c1N 38719,C(=O)(CCC(C)(C)[N+](=O)[O-])NCC(C)CNC(=O)CSCc1ccccn1 38720,O=C1Nc2ccc(C(N3CC4CN(C(=O)CC5(O)CCC5)C4C3)=O)cc2C1=O 38721,N1(C(C(CC)N(C)C)=O)CCN(C(=O)C(N)=O)C(c2cn[nH]c2)C1 38722,C1(C2CCN(C(=O)CN3CCCC3C)CC2)(NC(CC(CC=C)(C)C)=O)CCC1 38723,C(CCCCC(=O)N1CCC(C)(C)C1C(=O)NC(C)C(=O)NCC1CC1)SC 38724,CCC(O)C(F)(F)C(=O)N1CCC(C(C)NC(=O)CCCn2ccnc2C)CC1 38725,N1(C(c2scc(C(C)=O)c2)=O)CC(C)N(C(=O)CCOC2CCC2)CC1C 38726,C1(N2CC(N)C3(C2)COC3)CCC2(CCOCC2)C1 38727,Cc1ncc2ccc(C(N3CCC(CNC(C4(C5CC5)CC4)=O)C3)=O)cn12 38728,C1(NC(c2nnn(CC)c2C)=O)COCCN(C(=O)COCC(=O)OC(C)(C)C)C1 38729,CCCC(C(=O)Nc1cnccc1OC)NC(C1(C(=O)OCC)CC(=O)C1)=O 38730,N1(C(=O)Cn2ncccc2=O)CC2CCN(C(=O)CCc3ccncc3)C2C1 38731,C1(C(=O)NCC(C#C)NC(=O)CCCOCCOC)OCCC1(C)C 38732,n1(CCOC)cc(CC2CN(C(=O)CCc3cnc(C4CC4)o3)C2)nn1 38733,c1(C(C(=O)NC(C)(C)CCNC(C2COCC2CF)=O)OC)c(F)cccc1F 38734,CCC(CCCC(=O)N(C1CC1)CC1(O)CCC1)NC(=O)C(n1ccc(C)n1)C 38735,c1(C2(NC(=O)NCc3scc(CCOCC)n3)CC2)nnc2n1CCC2 38736,C1(OC)(CN)CN(C(=O)CNC(C2CC2C)=O)C1.C1(=O)CC1=O 38737,c1(C(=O)NCC2C(CNC(Cn3c(C)nnn3)=O)C2)ccc(NC=O)cc1 38738,C(=O)(CCCS(C)(=O)=O)N(C1CCCN(C(c2ccc(F)c(SC)c2)=O)C1)CC 38739,Cc1[nH]c2ccccc2c1C(=O)N(CCC(C)NC(=O)CC1CCCCO1)CCO 38740,N1(C(Cc2nnc(C)o2)=O)CCC2(CCCCC2NC(=O)C(C(C)C)C(C)C)C1 38741,O=C(NN1CCSCC1)C(=O)N1CCCCC1c1ncc[nH]1 38742,C1(C(N2CCS(=O)(=O)CC2)=O)CC2(CC2)CN1C(c1cccc(Br)c1)=O 38743,C(=O)(CC(C)CC(C)(C)C)NC1(CN(C(CC2(OCC)CCC2)=O)C)CC1 38744,N1(CC(=O)NC23CC(CNC(CCc4onc(CC)n4)=O)(C2)C3)CC2C=CC1C2 38745,Cc1ccc(F)cc1CC(=O)NCC1(C)CCCN(C(C2C3(CC3)C23CC3)=O)C1 38746,c1(CC)ccc(C(N2CC(NC(c3ccc(CN(C)C)[nH]3)=O)CC2C)=O)cn1 38747,C1(c2nnnn2-c2ccccc2Nc2ncccc2Cl)(COC)CCOCCC1 38748,c1(SCC)nc(C)c(CC(=O)NC(C)(C)CCCNC(C2(C)CC2(F)Cl)=O)s1 38749,c1(NC(C2CN(S(CCC(=O)OC)(=O)=O)CC(F)C2)=O)ccc2c(n1)NC(=O)CC2 38750,c1(C(C)C(=O)NCC2CC(NC(c3occc3Br)=O)C2)cccc(C#N)c1 38751,CCC(O)(CC(=O)NCc1ccc(N2CCCC2)cc1C)c1ccccc1 38752,C(CC(CNC(C1CCCN1CCC(C)C)=O)NC(=O)COCCC(C)C)OC 38753,C(=O)(C(C)C(O)CC)NCc1cc(C(=O)NCCC(=O)NCC)n[nH]1 38754,C1(C(C(=O)NC2CCOC2)N(c2ccccc2)CC2CC2)CC2CCC1O2 38755,c1(C(N2CCC(N(C(=O)C=CC3CCOC3)C)C2)=O)ccc(C(F)(F)F)nc1O 38756,C(=O)(C(F)(F)C(C)(C)O)NCC12OCC(CNC(C(C)NC(CC)=O)=O)(C1)C2 38757,C1(C(=O)NCCOC2CCN(C(C3C(OCC)C3)=O)C2)CCC(C)CC1 38758,C1(C#N)(C(=O)NC(CC)CNC(C2CC(=O)N2)=O)CC12CCCC2 38759,N1(C(C(CC(C)C)F)=O)CC2C3CCC(C2C1)N(C(c1ccc(Cl)cn1)=O)C3 38760,CC1CCC(NC(=O)CCC2CC2)CN1C(c1cc(-c2ccccc2)[nH]n1)=O 38761,c1(C(=O)NCC2C(C(=O)NC3C(OC)CC3)CCO2)cc(F)ccc1C 38762,c1(C(=O)NC2CN(C(C3C(C)OCCO3)=O)CC2F)cn(C)c(=O)cn1 38763,n1(C(C)C(=O)NC2CCCC2NC(c2cncc(O)c2)=O)cnc2ccccc12 38764,Cc1nc2cc(C(=O)NC(C)CCN(C)C(C3CCCC(=O)N3C)=O)cnc2[nH]1 38765,C1(C(=O)NC(C)C(O)CO)CCC(C(C)C)N1C(=O)CC1CCCC(=O)N1 38766,CC1CC(C(=O)N(C)CCOCCNC(=O)C(C)(C)C2CCCCC2)C1(C)C 38767,Cc1ccc(C=CC(=O)NCCC2(NC(C3CCSC3)=O)CC2)cc1C 38768,CCCC(C)CC(=O)N1CCC(C(C)CNC(C2(CF)CC2)=O)CC1 38769,c1(C2C(C(=O)NCC3(O)CN(C(C(c4ccsc4)=O)=O)C3)CC2)ccc(F)cc1 38770,C(=O)(CC(F)F)NCC1CC(NC(C=CC)=O)C1 38771,N1(C(C(C=C=C)C)=O)CC2(CC(CNC(c3c(C)cccc3Cl)=O)C2)C1 38772,c1(OC)nc(N2CCN(C(=O)CCC3(OC)CC3)CC2)cc(C)n1 38773,c12ccc(F)cc1[nH]c(=O)n2C.c1(OC)ccc(SCC2CNC(=O)CO2)cn1 38774,c1(C(N2C(C)(C(=O)NCC(=O)OCC=C)CCC2)=O)cc(F)ccc1F 38775,C(=O)(C1=CCc2ccccc21)NCC1N(C)CCN(C(C(CC)=CC)=O)C1 38776,C1(COC)CCN(C(c2nc[nH]n2)=O)C(C(=O)N(CC(C2CCC2)OC)C)C1 38777,C1(C(=O)NCCOC)COCCC1NC(C1CN(C(=O)N(C)C)C1)=O 38778,C1(NC(c2n(CC=C)ccc2)=O)CCCCC1N(C(=O)Cn1nccc1C)C 38779,c1(C2CCN(c3n(C(F)Cl)nnn3)C2)ccc(Cl)cc1 38780,C(C(CNC(=O)CC(C)(C)O)CC(=O)NCCn1nnc(-c2cccs2)n1)OC 38781,C(CC(F)F)(C(=O)NC1CC2CCC1CC2)N(C(COCC(=O)OC)=O)C 38782,c1(C(N2C(CN(C(C(CC=CC)C)=O)CC)CCC2)=O)cc(C)cc([N+](=O)[O-])c1 38783,Cc1cc(OCCC(N2CCC(C)C(CC(=O)NC3CC3)C2)=O)cc(C)c1 38784,c1(OCCC(=O)NC(C(C)NC(c2ccncc2)=O)C)ccc(CC#N)cc1 38785,C1(C)(NC(CC2CC(C(C)C)OCC2)=O)CCN(C(C2(C)COCCO2)=O)CC1 38786,c1(CC)cc(NC(=O)C(C2CCC2)NC(c2coc(C3CC3)n2)=O)cc(O)c1 38787,c1(C(N2C(C)CC(NC(c3cncc(COC)c3)=O)C2)=O)ccc(N)c(Cl)c1O 38788,c1(N2CC(C(C)NC(=O)CCC3(C)CC3)OCC2)cc(-n2ccnc2)ncn1 38789,c1(C(C)=O)ccc(C(F)(F)F)nc1N1CC(CC(C)NC(C2CC(=O)N(C)C2)=O)C1 38790,c1(C(=O)NC(CN(C(CSC)=O)C)(C)C)ccc2c(c1)OC(C)(C)O2 38791,C1(CCCC)CN2CCN1C(=O)CN(C)C2=O.C1(C(=O)NC)CC12CCCCC2 38792,C(C(F)(C(=O)NCCc1cocn1)C(C)C)NC(C(CC#C)O)=O 38793,c1(CC)cc(C(=O)NC2CCN(C(=O)CC3CC(C)=NO3)C2C(C)(C)C)n(C)n1 38794,Cc1cccc(C2C(C)CN2C(c2cnccc2C)c2ccccc2)c1 38795,C(C(=O)NCC1(F)CC(CNC(c2ccc(C#N)cn2)=O)C1)(C(C)(C)C)SC 38796,C(=O)(C(CN(C)Cc1ccccc1)NC(=O)C(C1CCOCC1)=O)OCC 38797,c1(CC)conc1C(=O)NCCC1CCC(NC(C2CN(C(=O)C3CC3)C2)=O)C1 38798,Cc1c(C(=O)NC2CC(C)N(C(=O)C(C)Sc3nncn3C)C2)noc1C1CC1 38799,Cc1c(C(=O)N(C(c2cnn(C)c2)C(=O)NC)C)cccc1Cl 38800,N1(C(C2(CC#C)CCCO2)=O)CCC(C)N(C(=O)CC2(CC)CCC2)CC1 38801,C1(N(C(=O)CC2CC2(Cl)Cl)CC#C)CCN(C(C2CCC2CC)=O)CC1 38802,N1(C(C(=O)NC(C)CCn2cncn2)=O)CC(F)(CO)C1 38803,C(=O)(C(CCC1CC1)NC(=O)OC(C)(C)C)NC1CC(CC(C)(C)C)C1 38804,CN1C(=O)CSC1=CC(=O)NCC(C)(C1CC1)NC(=O)Cc1cnccn1 38805,N1(C(C=CCC)=O)CCC2CN(C(c3cc(CC4CCC4)c[nH]3)=O)CC2CC1 38806,Cc1cc(CNC(C)C(C)OCc2ccccc2)ccc1[N+](=O)[O-] 38807,N1(S(=O)(=O)C2CC2)CCC(O)(C2(C(=O)O)CCC2)CC1.C12CC(C3CC13)N2 38808,C(C(C(=O)N(CC(=O)NC(C)C)C)C(C)C)NC(C1(CC=C)CCC1)=O 38809,Cc1ccc(C(=O)N(CCCCCC(=O)N2CCC2C(C)C)C)c(F)c1 38810,S(=O)(=O)(CCC(=O)NCC1CCN(C(c2cc(C)c(Br)o2)=O)CC1)NC 38811,CC1CN(C(=O)CN2CCN(C(C3CC3c3ccco3)=O)CC2)CC(C)(C)O1 38812,Cc1cnc(CCN2CCC(CCNC(=O)OC(C)(C)C)C(O)C2)c(C)c1 38813,c1(C(=O)NCC2C(NC(C(C3CCCC3)SC)=O)C2)cn(CCN(C)C)nn1 38814,c1(CONC(c2ccc(C(=O)NC(C(O)CO)C3CC3)s2)=O)ccccc1O 38815,c1(C(c2nnnn2CC2CCCO2)SCC=C)ccc(NCCF)cc1 38816,c1(C(C)C)cnc2cc(C(N3CCC(CNC(=O)CO)C3)=O)[nH]c2c1 38817,c1(OCCC(C)C)ccc(C(=O)NCC(C)(C)NC(C2CCCN2C=O)=O)cc1 38818,c1(NC(C)=O)ccc(C=CC(=O)NC2CCC(NC(c3cc[nH]n3)=O)C2)cc1 38819,n1(CC(=O)NCC2CCC(C(F)(F)F)O2)cc(N)c(SC(C)(C)C)n1 38820,N1(C(C(COC(C)C)NC(Cc2c(C)nsc2)=O)=O)CCC2(CC2)C1 38821,C1(NC(=O)Cc2cncnc2)CCCC12CCN(C(c1ccc(Cl)c(Cl)c1)=O)C2 38822,c1(COC2CC(C(=O)OC)C2)cccc2c1CCC2 38823,c1(C(N2CCC(NC(C(C)OC)=O)C(O)C2)=O)scc2c1CCCC2 38824,C1(CC=C)OCCC1(c1nnnn1Cc1cccs1)N(CC=C(Cl)Cl)C1CC1 38825,c1(C(N2CCN(C(=O)CC(F)F)C3CC23)=O)cc2ncc(Br)cc2o1 38826,Cc1[nH]c2ccccc2c1C(N1CC2(CC(CNC(=O)C#CC(C)(C)O)C2)C1)=O 38827,N1(C(c2c(C)n(C)nn2)=O)C2CCC(C2)C1C(=O)NC1CC(C(F)(F)F)C1 38828,C(=O)(CCCCC(=O)OC)N1C(CCNC(C(CC)C(C)O)=O)CCCC1 38829,C1(CCO)(NC(=O)CN2CC=CC2)CN(C(=O)C(CO)N(C)C)C1 38830,C(=O)(CCC(CF)CF)NC(C(=O)NC(C1C(C(=O)OC)C1)C)CC(C)C 38831,N(C(=NCC1CC1)N1CCOC(CC2CC2)C1)CCC(C(F)(F)F)N(C)C 38832,N1(C(CO)CO)CCCN(c2nccc(OC(F)(F)F)n2)CC1 38833,c1(C(=O)NCCCC(C)NC(C2CC3CCC2C3)=O)cc2sccc2s1 38834,N1(C(Cc2c(O)nc(=N)[nH]c2)=O)CCC2(CCC2)C(NC(=O)CC2(CO)CC2)C1 38835,N1(C(c2c(CC)cncc2)=O)CC(NC(c2[nH]nnc2C)=O)CCC(O)C1 38836,CCCS(=O)(=O)C(C)C(=O)NCC1CC1CNC(=O)C=Cc1nccn1CC 38837,c1(SCCC(=O)NC2(CNC(C(CC)C)=O)CCOC2)c[nH]c2ccccc12 38838,CC(c1ccco1)=CC(=O)N(C1CCC(NC(=O)CC=C(C)C)C1)C 38839,C=C(C)CC(C(=O)NCCn1ccccc1=O)NC(=O)CCC=CC(C)C 38840,Cn1ncc(C(N2CC3C(NC(C4(CO)CCC4)=O)C3C2)=O)c1C1CCCNC1 38841,c1(C(C(=O)NC(Cc2c(OC)cccc2)C(C)C)SC)ccc(C#N)cc1 38842,C1(CCOC)(NC(c2ccc(Br)o2)=O)CCN(C(c2cccc(C(C)C)c2)=O)C1 38843,c1(C(=O)NC(CNC(C2(C)COC2)=O)C2CCC2)cc(=O)cc[nH]1 38844,Cc1ncc(Cl)cc1N(C1CCCCC1)C(c1[nH]c(C)c(C(=O)OCC)c1C)=O 38845,c1(NC(C2CCN(C(C(C)n3cccn3)=O)CC2O)=O)cccc(S(N)(=O)=O)c1 38846,C=CCCCCCC(=O)NC(C)(CC#C)C(=O)N(CC)CC1CCC1 38847,N1(C(C2C(C=C)CC2)=O)CC2(CCN(C(C3(F)CCCCC3)=O)C2)C1 38848,c1(OCC)ccc(C(N2CCN(C(=O)C(C)C)CC2)C(=O)NC2CCOC2)cc1 38849,N1(C(c2c(CC)n(C)nc2)=O)CCC(C2CCN(C(=O)C3=CCCOC3)C2)C1 38850,CS(=O)(=O)C1CCN(NC(C2(N)COC2)=O)CC1 38851,c1(CC(C)NC(C(CC)OCC)=O)ccc(CNC(C2(F)CC2)=O)cc1 38852,CSC1=C(C(=O)NC2CCN(C(=O)Cn3ccnn3)C(C)C2)CCCC1 38853,CCS(=O)CC(=O)N(CC(C)CNC(C1COCCN1C)=O)C 38854,c1(CC)nonc1C(=O)NC(C)(CNC(c1ccncc1)=O)CO 38855,CC1(C(N2CCN(C(=O)Cc3cocn3)CC2)=O)C=CCCC1 38856,N1(C(c2cc(C)oc2)=O)CC(CNC(=O)Cc2ccsc2Br)C(C)(C)C1 38857,c1(OC)c(F)ccc(F)c1C(N1CC(CNC(=O)CCc2ccc(O)nc2)C1)=O 38858,C=CC1(C(N2CCC(C3CCCN3C(c3cc(COC)[nH]n3)=O)C2)=O)CCC1 38859,C(=O)(CC1CCOc2ccccc21)NCC1N(C(C2CC(OC)C2)=O)CC(F)C1 38860,c1(C(=O)NC2CC3CN(C(C(C)C#N)=O)CC32)cc2ncccn2n1 38861,Cc1cc(Cl)cc2cc(C(=O)Nc3cnn(-c4ccccc4)n3)[nH]c12 38862,C1(NC(CC(C)SC)=O)CN(C(c2cc(Cl)c(C)cn2)=O)C(C)(C)C1 38863,C1(C(=O)NCc2cc(CC)no2)CC(NC(=O)C(=O)N(C)C)C1(C)C 38864,c1(CCSCCC(N)C2COC2)c(F)cccc1Cl 38865,CC1CC(NC(=O)CCc2nnc(C3CC3)o2)CN(C(C2CC3CCC2O3)=O)C1 38866,c1(OCC)cccc(CNC(C2CC(=O)N(Cc3ccncc3)C2)=O)c1O 38867,C1(CC(NOCCC(C)O)=O)CCCN(C(=O)C(C(C)(C)C)n2ccnn2)CC1 38868,CC1(C)C2CCC1(C(N1CCC(NC(=O)Cn3cccn3)C(C(N)=O)C1)=O)C2 38869,N1(C(C(C)(C)C#N)=O)CCC(NC(=O)Cn2ccccc2=O)C(F)C1 38870,N1(C(c2cncc(CC)c2)=O)CC2CCCC2(NC(c2cnn(C(C)C)c2)=O)C1 38871,c1(C(=O)OC)cc(=NCC(C)(C2CC2)NC(C2COC(C)C2)=O)[nH]c(Cl)n1 38872,c1(C(N2CCCC2CF)C(=O)NCCCSC)cccnc1C(F)(F)F 38873,Cc1cc(CC(N2CCCC2CCCNC(=O)Cc2ccnc(F)c2)=O)nn1C 38874,c1(CC)ncccc1NC(=O)C(F)CC1CN(C(=O)C(C)OCC2CC2)C1 38875,C(c1cncnc1O)=CC(=O)NC(C)C(C)NC(=O)Cc1nn(C)cc1Cl 38876,c1(OC)ccc(N)c(C(=O)NC2CC(CNC(=O)C(C)C3CCC3)C(O)C2)c1 38877,Cn1c(C(=O)NCC2(CCNC(C3CCC3(C)C)=O)CC2)c(Cl)c2ccccc12 38878,C(=O)(C#CC1CCCCC1)N1C(C)(C(=O)NC2CC(CC)C2)CCC1 38879,O=C1CC2CC2(C(=O)NC2(c3nc[nH]n3)CC2)N1 38880,N1(C(c2[nH]ccc(=N)n2)=O)CC2CC1CC2CNC(=O)CC1CCCC1 38881,CCC(C)CCC(=O)N1CCCOC(C2CN(C(=O)C(CN(C)C)N(C)C)C2)C1 38882,CC(CC(N)=O)N(C)C(C1C(CNC(c2nccn2C)=O)C1(C)C)=O 38883,CN1CCCCC1CCC(N1CCOCC1CCNC(c1ccc(F)cc1)=O)=O 38884,c1(CC(=O)NCc2ccc(CNC(C(C)(C)SC)=O)nc2)cncc(C#N)c1 38885,CCC(CC(=O)NC1(CO)CCCN(C2C(C(=O)OC)CCCC2)C1)C(C)(C)C 38886,C12(C(=O)NCC(CN(C(=O)CN3CCCNC3=O)C)O)COC(CF)(C1)C2 38887,N1(C(C2CCC(F)(F)C2)=O)CCC2C(CCN2C(c2cnc(F)c(F)c2)=O)C1 38888,N#Cc1csc(C(=O)NC2CC(NC(C3CCN(C4CC4)CC3)=O)C2)c1 38889,C1(COC)(NC(c2ccc(O)nc2)=O)CCCN(C(=O)C(O)P(C)(C)=O)C1 38890,c1(OC)cc(C(=O)NCC(C)(C(C)C)NC(C2CCC=CCCC2)=O)ccc1C 38891,C1(CNC(C(C=C)(C)O)=O)CC2(CCN(C(=O)CCCN=[N+]=[N-])C2)CO1 38892,N1(C(c2c(SC)cn(C)n2)=O)CC(NC(C2CC(C)CCO2)=O)CC(O)C1 38893,C(=O)(C(F)(F)CCn1cccn1)NC1C(NC(c2c(N)nccc2)=O)CCC1 38894,c1(C(=O)NC2CN(C(C3CC(CC)OCC3)=O)C2)ccc(Br)c(C(F)(F)F)c1 38895,c1(CC)ncc(C(=O)N(CC(CC)NC(=O)C=CCN2CCCC2)CC)cn1 38896,c1(C(c2n(CC(=C)C)nnn2)NCC(CC)OC)snc(OC)c1Br 38897,N1(C(CCOC)=O)CCCC2(C1)CN(C(=O)C=C1CCOCC1)C2 38898,C1(F)(CNC(C2CCN(CC)C2)=O)CCC(NC(=O)Cc2c[nH]nc2C)C1 38899,Cc1nn2c(c1CNC(=O)C(O)c1ccco1)CN(C(C1CCCSC1)=O)CC2 38900,c1(C(=O)OC)cc(C(=O)NCCN(C(C2CCCC2O)=O)C(C)C)cs1 38901,CCC(C(=O)NCCC1(C)CCN(C(=O)COc2ccsn2)CC1)C(F)(F)F 38902,N1(C(C2CN(C(C(C=C)OC)=O)CC2F)=O)CCCOCC1C 38903,c1(N2CCC(CC)C2)cc(=NCc2nc(=N)n(C)[nH]2)[nH]c(C(C)C)n1 38904,C1(C2N(Cc3n[nH]c(=N)s3)CCC2)CC(c2ccc3c(c2)CCO3)=NO1 38905,N1(C(CCSc2nc(C)[nH]n2)=O)CC2CN(C(=O)Cc3nccn3C)CC2C1 38906,Cc1cc(C(N2CCC(C)(NC(c3nc(C4CC4)oc3C)=O)C2)=O)ccc1CO 38907,N1(C(c2c(Cl)cnc(CC)n2)=O)CCC(C2CCN(C(C3CC3F)=O)CC2)C1 38908,N1(C(=O)NC(COC)C(C)C)CC2CS(=N)(=O)CC2C1 38909,C1(OC(C)C(=O)NCC(C)(C)NC(=O)CC2CC3(CC3)C2)CCCCC1 38910,C1(C(=O)NCCC2CC(NC(C=CCOC)=O)C2)Cc2nccn2C1 38911,c1(NC(C2CCCC(C(=O)Nc3cccc(CO)n3)C2)=O)ccc(Br)c(F)c1F 38912,CCC(C)CC(C)c1nc(-c2occc2C)nn1-c1cccnc1C 38913,N1(C(C2(C)C(C)C2)=O)CC2CCN(C(=O)CCc3ccc(C(C)(C)C)cc3)C2C1 38914,C1(NC(c2c(C)ccnc2C)=O)CC2CCC1C(NC(C1CCC(=O)N1C)=O)C2 38915,c1(OC)cc(C)c(NC(=O)CC2CCN(C(C3(CC4CCC4)CC3)=O)CC2)cn1 38916,C1(O)(CNC(c2ccc(CNC(c3cnc(=N)[nH]c3)=O)cc2)=O)CCCCCC1 38917,C1(NC(c2c(NC)scn2)=O)CN(C(=O)C(C)SC)C(C)(C)C1 38918,c1(C(=O)NC(C2(O)CCN(C(Cc3cnc(C)o3)=O)C2)C)c(F)ccnc1F 38919,C1(C(=O)NC2CN(C(CCc3ccc(C(C)=O)nc3)=O)C2)CCC(C)NC1=O 38920,Cc1csc2ncnc(NCCCN(C(=O)CCc3cc(Cl)ccc3Cl)C)c12 38921,C1(C(=O)NC(CC=CC)C(=O)NC(C2CCCC2)CO)CCC2CC1CO2 38922,C(=O)(N=c1ccn(CC)[nH]1)C1(CC=C)CCCN1C(c1cc(C)ncc1C)=O 38923,Cc1cc(C(N2CCN(C(C34CSC(C3)C4)=O)CC2)=O)c(N)c(F)c1 38924,C1(C(N2CCC(NC(c3c(SC)nccn3)=O)CC2C)=O)CCCCC12CCC2 38925,n1(CC(N2CCN(C(c3c(C)cno3)=O)CC2CCO)=O)ncc2ncccc12 38926,Cc1ncc2n1CCN(C(=O)NC(C)CCOc1ccc(Cl)cc1)C2 38927,C1(O)(CNC(C(C)C)=O)CCCN(C(C2CCC3CC2CO3)=O)C1 38928,N1(C(c2cc(C)c(Br)cc2)=O)CC2CCN(C(c3cn(C)cn3)=O)CC(C2)C1 38929,O=S(=O)(c1ccc(Br)cc1Cl)NC(c1ccc(F)cc1)CC1CC1 38930,c1(NC(Cn2ccc(C)n2)=O)ccc(NC2(C)CN(C(=O)CCCF)C2)c(C)c1 38931,N1(C(C=C(C)Cl)=O)CCC2(CC1)CN(C(=O)Cc1cnn(C)c1)CC2CO 38932,c1(NC(CNC2C(NC(C(F)=CCC)=O)CCC2)=O)cnncc1C 38933,C1(NC(c2nn[nH]c2Cl)=O)CC2(CCN(C(=O)Cn3cccc3)C2)C1 38934,C(=O)(C1=CC2(CCOC2)C1)N(C1CCN(C(c2ccoc2Br)=O)C1)C 38935,CCCC(C)(O)C(=O)NCC(CC)(CC)NC(C1COCC(C)(C)O1)=O 38936,N1(C(CC2ON=C(C)C2)=O)CCCCC1C(N1CCN(C(=O)C(C)C)CC1)=O 38937,C1(C)(C(=O)OC)CC(C)=NO1.c12ccc(o1)C(C)(C)C(=O)N(C)CC(CC)NC2=O 38938,c1(CCNC(N2C(COC)C(C)(C)C2)=O)cnc2n1CCOC2 38939,c1(C(c2n(C)nnn2)NCc2cscc2Br)nc(F)ccc1Br 38940,C#CCCC(O)C(=O)NC1CCCN1C(=O)CCOc1ccccc1OC(C)=O 38941,N1(C(CCCC)=O)CCCC(O)(CCNC(=O)C(O)C(C)CC)C1 38942,C(=O)(C1=CC2CCCCCC12)N1CC(C)C(CNC(C2CCC3CC3C2)=O)CC1 38943,c1(CC)nn(C)cc1C(=O)NC1CCCN(C(=O)C(C)SC)C1 38944,C1(CNC(=O)C(F)C2CC2)CC2(CO1)CN(C(c1ccc3c(c1)CCC3)=O)C2 38945,C1(NC(C2(COC)CCOC2)=O)CN(C(=O)Cc2ccc(O)c(Cl)c2)C(C)(C)C1 38946,CCC(CC(=O)N1CCC(C)C1CNC(=O)CC1CCCC(=O)N1)C(C)C 38947,Cc1ccc(C(=O)NC(C)CCNC(=O)C(F)C(C)(C)O)c(N)c1Cl 38948,C1(C2CCN(C(C3CCCC3S(C)(=O)=O)=O)CC2)(NC(C(CO)N(C)C)=O)CC1 38949,C1(C)(C(=O)NC2CC(NC(C3N(C(CCC)=O)CCC3)=O)C2)CCC(=O)NC1 38950,n1(CCC)cc(C(=O)NC2CCCC2CNC(c2ccc(NC)cc2)=O)c(C)n1 38951,N1(C(C(CC)C)=O)CCc2ccc(C(N3CC(C)(C#N)C3)=O)nc21 38952,c1(C(=O)NCC2(O)CN(C(c3cc(F)cs3)=O)C2)ccc(-n2cncn2)nc1 38953,C1(C(N(C2CCCCN(C(=O)C=CSc3nc[nH]n3)C2)C)=O)CC2C(C1)C2(C)C 38954,N1(c2snc(C)n2)CC2CC(NC(C3(Br)CC3)=O)C2C1 38955,N1(C(Cc2n[nH]c(=N)s2)=O)CCC(C2(NC(c3ccn4nnnc4c3)=O)CC2)C1 38956,c1(C(=O)NCC(CC)NC(=O)CSC)cccc2oncc12 38957,O=C1CCCc2cc(C(=O)NC3CN(Cc4cc(F)cc(F)c4)CC3F)ccc21 38958,c1(C(N(C2C(C)CCN(C(=O)CO)C2)C)=O)ccc(S(C)(=O)=O)cc1 38959,c1(C(N2CCN(CCCNC(CCC=CC)=O)CC2)=O)ccc2nn[nH]c2c1O 38960,C1(NC(CC2C(C)CN(C(C3C4CC5C(C4=O)C35)=O)C2)=O)CC2CCC(C1)N2C 38961,S(=O)(=O)(c1cccnc1NCc1ccc(C)s1)NC(CC)C(O)C(C)C 38962,CCCC(CC(=O)NCC1CCC(C)CC1)NC(c1sc(C)nc1C)=O 38963,C1(C)(CNC(c2c(C)cns2)=O)CCCN(C(c2ccc(C(C)C)cc2F)=O)C1 38964,c1(C(=O)NCC(CN(C(CS(=O)(=O)NC)=O)C)O)cccc(C#CCO)c1 38965,C=C(C)C(C)(C)C(=O)NC(C1CCN(C(C2CSC3(C)CCC(=O)N23)=O)CC1)C 38966,C1(CC)CCN2C(C1)C2=O.C(=O)(CC(C)(C)CNC(N)=O)NC1CN(C)CC1O 38967,Cc1ccc(-n2ncc(C(=O)NC(c3cccnc3)C3CC3)n2)cc1 38968,N1(C(C(Cc2ccoc2)NC(c2cc(F)c[nH]2)=O)=O)CCCCC1C1CCC1 38969,N1(C2CCCN(C)C2)CCC2(CC1)CC2C(N1CCCC(CCN)C1)=O 38970,c1(C(N2CC(O)(CCNC(CNC(=O)NC)=O)C2)=O)c(C)[nH]cc([N+](=O)[O-])c1=O 38971,C1(NC(C(c2cc(C)sc2)(F)F)=O)CN(C(=O)CC(O)C2CC2)C2CCCCC12 38972,C(=O)(CC(C)F)NC1C(CNC(COC)=O)C(O)C1 38973,C1(NC(c2ccc(C#C)c(C)c2)=O)C2CCCN(C(=O)CC(F)(F)F)C2C1(C)C 38974,C1(N)CCC(C)(C)CC1.C(C(=O)NC1CCCC1)(C1CCC1)N(CC)CC 38975,C(=O)(n1ccc(C2OCCO2)n1)NCCN1C(C)CC(C(F)(F)F)C1C.CO 38976,C(=O)(CCCC(CC)CC)N1CCN(C(C(COCC)C)=O)C(C)C1 38977,C(=O)(C1=CCOCC1)N(CCNC(c1c(C)cc(C(F)(F)F)s1)=O)C 38978,c1(CC(=O)N(C(C(=O)NC(C2CCCC2)C#C)C)CC)ncccc1C 38979,C(C)(C(C(=O)NCc1ncc(F)cc1F)C(C)C)NC(C(F)=CCC)=O 38980,C(=O)(CC(C)(C(F)(F)F)N(C)C)N(C1CCN(C(c2cn(C)c(O)n2)=O)C1)CC 38981,N1(C(C2CC(C)(C(=O)OC)C2)=O)CC(NC(=O)C=CS(C)=O)C(F)C1 38982,CC1CCC(C(N2CC(N(C(=O)Cn3cncn3)CCO)C2)=O)S1 38983,c1(C(C)=O)ccc(C(=O)NCC(F)CNC(c2ncnc(C)c2C)=O)c(F)c1 38984,N1(C(c2cc(C)ns2)=O)CC2C(CN(C)C(c3cccc(C(C)C)n3)=O)C2C1 38985,c1(NC(C(C)NC(=O)COc2ccc(Br)cc2)=O)ccc(Cl)cn1 38986,c1(C(N(C)Cc2cn(CC3(C(C)(F)F)CC3)nn2)=O)onc2ccccc12 38987,N1(C(c2cc(C)on2)=O)Cc2cccn2CC(C(N2CCC23CCCCC3)=O)C1 38988,c1(OCC)cc(C(N2CCCC(CNC(=O)CC3CCC(=O)N3C)C2)=O)ccn1 38989,CCC(F)(F)CC(=O)N1CCC(F)CC1C(N1CCC(F)CC1)=O 38990,C1(n2c(-c3cc(OC)nnc3OC)nc(-c3cscn3)n2)CCN2CCCCC12 38991,N1(C(C2(Oc3cn(C)nc3)CC2)=O)CCCOC(CNC(=O)CCCSC2CC2)C1 38992,C(C)(C)(CCCCC(=O)NC(C1CN(C(C2CCO2)=O)C1)C)OC 38993,CC(C)(CN1CCOCC1)C(=O)NCCC1(NC(C2(C3CC3)CC2)=O)CC1 38994,C(C(C)(C)C(=O)NCCC1CCC(C)O1)NC(C=CCCC)=O 38995,CC(C)(CCF)C(=O)NC1C=CCN(C(c2cc(CCO)on2)=O)C1 38996,C1(C(=O)NCC(CNC(c2ncoc2C2CC2)=O)OC)CCc2nc(C)nn2C1 38997,N1(C(C23C(C)(C)OCC2C3)=O)CCCC2(C1)CN(C(c1ncc(N)cc1Cl)=O)C2 38998,c1(N(CC)CC)ccc(C(N2CC3CC2C3c2ccccc2)=O)cc1.C1(C)CN1 38999,c1(C(N2C(CC(=O)NCC3(C)CC=CCC3)CC(O)C2)=O)ccccc1C#N 39000,c1(C(N2C(COC)(CNC(=O)C(C)C(C)O)CCC2)=O)cc2[nH]nc(C)c2cn1 39001,c1(OC)ccc2[nH]c(=NCc3ncco3)nc(N3CCSC(C)C3)c2c1 39002,c1(C(N2CCC(NC(C3(Br)CCC3)=O)CC2)=O)ccc(Cl)c(F)c1F 39003,c1(C(=O)NC2C(C)C2C)cc(C#N)ccc1N 39004,Cc1ccc(CC(=O)NCCCN2CCC(NC(=O)CCc3cn[nH]c3)C2)s1 39005,C#Cc1ccc(OCC(=O)NCCC2(NC(C3CCN(C)S3(=O)=O)=O)CC2)cc1 39006,c1(C(N2CCC3CN(c4ccnc(C5CC5)n4)CC3C2)=O)cc(=O)n2[nH]nnc2n1 39007,c1(C(=O)NC2C=CC(CNC(C(C)(C3CC3)OC)=O)C2)nc(Cl)oc1C 39008,N1(C(CC(CC)OC)=O)CCOCC(C)(CNC(c2ccc(C)cc2SC)=O)C1 39009,CCCC(CCC)=CC(=O)NC(C)CC(C)NC(=O)CCc1nccn1C 39010,c1(NC(=O)Nc2c(C(N)=O)nccc2)ccc2nc(O)n(C3CC3)c2c1 39011,C1(NC(c2n[nH]cc2I)=O)CC12CCN(C(c1c(Cl)cc(F)cc1Cl)=O)CC2 39012,N#Cc1c(NC(C2CC(NC(C3CCC(O)CC3)=O)C2)=O)cccc1Br 39013,c1(CCC)cc(C(N2CC(NC(=O)C(C)COCC)CC2CO)=O)c(C)o1 39014,C(=O)(C(C(C)(C)C)N(C)C)NCC1C(CC(=O)NC(C)CN2CCCC2)C1 39015,C1(C)(CC(=O)NCC(C)N(C)C)CCN1C(=O)COCCCCN=[N+]=[N-] 39016,Cc1cnc(Cl)[nH]c1=NC(C)CC(C)NC(=O)CCc1nccn1C 39017,C1(CCNC(COCCOCCOC)=O)CCN(C(C2CCCS2)=O)C1 39018,C(=O)(CS(C)(=O)=O)NCC1(NC(C(C)Cn2ccnc2)=O)CCCC1 39019,N1(C(c2n(C)ccc2)=O)CCCN(C(=O)C(F)CC2CCCCC2)CC1CO 39020,n1(CC(=O)NCCC(C)N(C(COCc2cc(C)on2)=O)C)nc(C)c(O)c1C 39021,c1(OC)nn(C)cc1NC(=O)CC1(N(C)C(C2COCCN2C)=O)CC1 39022,c1(-c2cncc(C(C)(C)OC)c2)ccc(OC)c([N+](=O)[O-])c1 39023,C(=O)(CCC(=O)NCC1CN(C(=O)COC2CCOC2)C1)NC1C(Cl)(CC)C1 39024,C1(CNC(C(c2ccc(F)cc2)OC)=O)CCCCN1C(=O)C=CC1(C)COC1 39025,c1(C(=O)NC2CC(C)(NC(=O)C3=COCCO3)C2)ccnc(S(N)(=O)=O)c1 39026,c1(C(=O)NC(CNC(c2nc(OCC)sn2)=O)(C)C)ccc(OC)c2ccsc12 39027,c1(C(C(=O)NCCC(C)CCNC(=O)C(C)C(F)(F)F)(C)C)cccc(C#N)c1 39028,C1(CNC(COCCC=C)=O)CCCCC1NC(=O)Cc1cccc(OC)c1 39029,N1(C(CCCC2C(C)C2)=O)CCC(C2CC2)C1C(N1CC(C#N)C1)=O 39030,c1(CNC(c2cccc(-n3c(C)c(C(=O)O)cn3)c2)=O)cn2cccc(C)c2n1 39031,N1(C(C(=O)NCc2n(CC)c(C)nc2)=O)CC2CCC2(C)C1 39032,C(=O)(C(=O)N=c1cc(C)[nH][nH]1)NC(COC)C(=O)N(c1ccc2c(c1)CCC2)C 39033,C(C)(N=c1cc[nH]cc1S(=O)(=O)N1CCOCC1)CC1OCCC(C(=O)OC)C1 39034,c1(C(=O)NC(CC)CNC(C2(C)CCC(C)CC2)=O)cc(O)ccc1[N+](=O)[O-] 39035,c1(C(=O)NC2CC(NC(c3c(C)nc(CC)o3)=O)CC2O)cc2n(n1)CCOC2 39036,c1(CC(N2CCN(C(CC(=C)C)=O)CC3(C2)CC3)=O)nc2nc(C)cc(C)n2n1 39037,c1(C(N2CC(CC=C)(NC(=O)CC3CCCC3(F)F)C2)=O)ccc(CC)nc1O 39038,c1(C(=O)NCC2(O)CCN(C(C(C)OCCC#C)=O)C2)ccc(C)c(CC)c1 39039,C(=O)(C(C)(C)CCCO)NC1CC2CN(C(C(C)(C)Cc3cnn[nH]3)=O)CC21 39040,C1(C(=O)NCc2c(C)occ2)CN(C(=O)CCC(=O)C2CC2)CC12CC2 39041,C(=O)(C1=CC2CCC=CCCC12)NCC1C(C)CCN(C(C2(O)COC2)=O)C1 39042,CCC(CC)C(=O)N1CCCCC1C(=O)N(CCN1CCCC1=O)CC 39043,C(CC(C)(C)CC(=O)NCCCCC(C)NC(c1cc(C2CC2)n(C)n1)=O)OC 39044,Cc1ccnc(C)c1NC(C12CCC1CN(C(=O)Cc1cc(Br)ccc1Br)C2)=O 39045,C1(NC(=O)NCc2ccccc2C2CCNCC2)(CC2CCCC2)CCOCC1 39046,CC1CN(C(c2cccnc2CO)=O)CCN1C(C1CCS(=O)(=O)CC1)=O 39047,c1(CC(=O)NC(CNC(=O)C=CC2CCC2)C2CC2)nc([N+](=O)[O-])n[nH]1 39048,C(=O)(CCCCCCC=C)N1CC(CC=C)(C(=O)NC2CC(=O)N(CCC)C2)C1 39049,N1(C(c2ccc(CNC(N)=O)s2)=O)CC2CC1CCC2O 39050,CC(C)CN=C(NCc1ccccc1CS(C)(=O)=O)NCC1CCSC(C)C1 39051,Cc1cnc(CNC(=O)C(CN(C)C)NC(=O)CC(C)(C)C#N)c(C)c1 39052,Cc1scc(C(N2CC(NC(C3(C4CCCO4)CCCC3)=O)C(O)C2)=O)c1N 39053,c1(OCCC)ccc(CNC(=O)NC2CC(C(=O)OC)C2)cc1 39054,C1(C(=O)NC2C(=C)C2C(=O)OC)CC(CCCNC(=O)Cc2cnnn2C)CO1 39055,CC(C)C(C(=O)N1CC2CC1C2NC(=O)COCC1CC1)NC(=O)OC(C)(C)C 39056,C1(NC(C(CCC)OC)=O)CC2CN(C(c3cn(C)c(=O)n3C)=O)CC2C1 39057,Cc1cnc(C#N)c(-c2c[nH]c(=NCC3(c4cc(F)c(F)cc4Br)CC3)s2)c1 39058,CC1C(NC(C2COCCN2C)=O)CCCN1C(c1[nH]ncc1C#N)=O 39059,N1(C(c2c[nH]ccc2=O)=O)CCN(C2CCCN(C(C3CC4CC4C3)=O)C2)CC1 39060,CC1(C(=O)NC(C2CCCC2)CNC(=O)Cc2ccc(Cl)nc2)CC=CCO1 39061,c1(C(C)C)ccc(C(N2CC(N(C(=O)CC3CC=CCC3)C)C2)=O)cc1 39062,C1(C)(COC(c2c(C)ccnc2C(C)C)=O)CC(C2CC2)=NO1 39063,c1(CC)ncccc1NC(C1CC1c1ccccc1Cl)=O 39064,C12CCN(C1)C(C1CCC1)C(=O)N2.C1(CN(C(C)=O)C2CC2)CCOC1 39065,c1(C(N2CCC(C)(CCNC(C3CNC(=O)C3)=O)C2)=O)c(F)ccc(Cl)c1N 39066,c1(C(=O)NCCCN(C(C(C)SCC)=O)C2CC2)cc(O)c2[nH]c(C)nc2c1 39067,C1(O)(CNC(CC2(CSC)CC2)=O)CCCN(C(c2csc(C#N)c2)=O)C1 39068,c1(C(C(N2CCC(C(F)F)(CNC(C)=O)C2)=O)C)ccccc1S(N)(=O)=O 39069,C1(NC(CCCC(=O)OC)=O)C2CC(CN(C(C3(CF)CC3(F)F)=O)C2)C1CO 39070,C1(NC(C2(CCC)CC2)=O)CCCCC1CNC(c1cc(F)n(C)n1)=O 39071,c1(CNC(C(=O)NCC)=O)cc2n(n1)CCN(C(C1CCc3cncn3C1)=O)C2 39072,N1(C(C2C=C(C)CS2)=O)C2CCC1CC(C(=O)NC(C)C(C)F)C2 39073,C1(CNC(C2ON=C(CC)C2)=O)CC2CCC1N2C(c1cc(C)ccc1C)=O 39074,N1(C(c2ncn(CCC)c2)=O)CCC2(CCN(C(c3cnc(C)s3)=O)C2)C1 39075,C1(OC(C)C(=O)NCC(C)(C)CNC(=O)COC2CC2)CCCCCC1 39076,c1(C(N2CCC(NC(c3c(C)onc3C(F)(F)F)=O)C2C)=O)ccc([N+](=O)[O-])[nH]1 39077,C1(C(=O)NCCCC(C)NC(c2c(C(F)(F)F)ncn2O)=O)CC(=O)OC1(C)C 39078,c1(C(CC)(C)C)cn(CC2CC(NC(=O)C(F)OC(F)(F)F)C2)nn1 39079,C1(C(N2CC(C)N(C(C3CS(=O)(=O)CCO3)=O)CC2)=O)Cc2nccnc2C1 39080,CC1=NNC(=O)C1CC(=O)NCC(N1CCCCC1C(=O)NCc1ncco1)=O 39081,CS(=O)(=O)C1CCN(CC2CC3C=CC2C3)CC1 39082,C(=O)(CC(CC(C)C)NC(=O)C(CCC)=CCC)NC1(CC=C)CC1 39083,CC1CCN(C(=O)C(=O)NCC2CCCN(C(=O)CCC3CNC(=O)N3)C2)CC1 39084,c1(C(=O)NC2C(C)CN(C(c3c[nH]nc3F)=O)C2)n[nH]c2c1CCCC2 39085,n1(CC(=O)NCC2C(N(C)C)CN(C(=O)CC3CC4CC4C3)C2)ccc([N+](=O)[O-])n1 39086,c1(C(=O)NC)cccc(C(=O)NC(CO)C(C)NC(C2CCS(=O)(=O)N2)=O)c1 39087,C(=O)(CCS(=O)(=O)N(C)C)NCCOC1CN(C(c2ccc(OC)o2)=O)C1 39088,C1(C(=O)NCCCC(C)NC(c2sccc2CO)=O)CC2CC1CC2O 39089,C1(CNC(c2c(C)cc(C)[nH]2)=O)(NC(c2c(C)cnn2C)=O)CC2CCC1CC2 39090,Cn1cc2c(C(=O)NCC3(CNC(=O)C4=CCOCC4)CC3)cccc2n1 39091,C1(C(=O)Nc2cccc(NCc3ccccn3)c2)CC2CNCC(C1)C2 39092,C12(CNC(C34C(C)OC(CO)(C3)C4)=O)CC(NC(=O)CC3CC3)(C1)C(C)(C)O2 39093,Cc1cc(C(N2CC(CC(F)C(=O)N3CCC4CC34)C2)=O)sn1 39094,c1(C(=O)NC2CCN(C(CN(CCCCCC)C)=O)C2)cc(=O)c(OC)c[nH]1 39095,c1(C(N)=O)ccnc(C(=O)NCC2C3CN(C(=O)Cn4cnnc4O)CC23)c1 39096,c1(CSCC(C(C)(C)C)OC)nc2ccccc2o1 39097,C1(C(=O)NC2CN(C(c3ccc(C)cc3)=O)C(C)(C)C2)CNC(=O)CC1(C)C 39098,N1(CCC(=O)NCC(CC)(C)NC(c2cnc(C(C)O)s2)=O)CCCCC1=O 39099,C12(C(N(C(CCCC)C)C)=O)CCCC1CN(C(C1CC1CCOC)=O)C2 39100,C1(C(C=CC(=O)NCC(COCC)O)=O)CCCN(C(C)=O)C1.C(=O)(CC)N 39101,N1(C(C(Cn2ccnn2)NC(C2(CC)CC2)=O)=O)CCCN(C(C)=O)CC1 39102,Cc1cc(C(=O)N(CC(C)NC(=O)CCc2nc(C(C)C)no2)C)c(N)c(Cl)c1 39103,N1(C(CCC(C)N(C)C)=O)CCC2(CCN(C(=O)Cc3cncc(F)c3)C2)C1 39104,c1(C(N2C(CC=C)CCC2)=O)cn2c(n1)C(N)CCC2 39105,Cc1cccc(CN(C(c2ncccc2C)C(=O)NCCC2(C)CC2)C)c1Br 39106,Cc1nc(C)n(CCN(C(c2sc(NC(=O)C(C)(C)C)cc2C)=O)C(C)C)n1 39107,c1(NC(C)=O)nc(CNC(=O)C(CC)NC(c2cc(N(C)C)no2)=O)oc1C 39108,C1(C)(C(N2C(CNC(C(c3n(C)cnn3)(C)C)=O)C=CC2)=O)CCNC1=O 39109,S(=O)(=O)(c1cccc(Br)c1)NCC1(O)CN(C(c2c(F)ccc(Cl)c2F)=O)C1 39110,CC1C(NC(=O)C=Cc2ccccc2)C(C)CCN1C(C1CCC=CO1)=O 39111,Cc1nc2ccc(-c3cncc(NS(C)(=O)=O)c3)cc2n1C 39112,N1(C(C2(CC=C)CC=CC2)=O)CC2CCC(C1)C2C(=O)NCc1ncco1 39113,c1(C(=O)NC2C(CC)CN(C(=O)C#CC3(C)CC3)CC2)cc(O)cc(C#N)c1 39114,Cc1c(C(N2CCCC23CCN(C(C2CCCN2C)=O)C3)=O)nn2ccccc12 39115,N1(C(C(COC)C)=O)CC2C(CNC(=O)C(C)OC3CCCC3)C2C1 39116,N1(C(c2cc3nc[nH]c3cn2)=O)CCC2CN(C(=O)C(O)CC(F)(F)F)C2C1 39117,c1(C(=O)NCC2CN(C(CCCCSC)=O)C3C2C3)cc2cc(Cl)ccc2[nH]1 39118,C1(CNC(=O)C(=O)NC2CC2)CN(C(=O)CCC2OCCO2)CC12CCOCC2 39119,C(=O)(C(CC(F)F)C1CCC1)NC1(C)CN(C(C2(C)N(C)CCC2)=O)C1 39120,O=C1NC(=O)C(C2CN(C(=O)CC34CC3CN(C(=O)CO)C4)C2)N1 39121,N1(C(CCc2ccc(N)c(F)c2)=O)CC2ON=C(CNC(=O)C3=CCSC3)C2C1 39122,C(C(=O)N1CCC(N2CCN(C(=O)CCC=C(C)C)CC2)C1)(C(C)C)SCC 39123,O=C1CN2C(CN1)C(=O)NO2.N1CCN(C(=O)CO)CC1.CC(F)(F)F 39124,C1(C2CCN(C(=O)CC3CSCCS3)C2)(NC(C2C=CC=CC=C2)=O)CC1 39125,Cc1scc(C(=O)NCC2(F)CCN(C(=O)CCc3ccon3)C2)c1C 39126,c1(C(=O)NC2C(NC(C3CCCC(C)(C)C3)=O)C2)nc2cc(O)ccc2[nH]1 39127,CC1CCCc2ncc(C(=O)NC3CN(C(C4CC5CC4C5)=O)CC4(CC4)C3)n21 39128,N1(C(C(CC)CO)=O)CCC(NC(=O)C(C)NC(=O)CC(C)(C)C)C(C)(C)C1 39129,Cc1ccc(C=CC(N2CCCC(NC(=O)CC3C=CCC3)C2C)=O)nc1 39130,C1(NC(C(C=C)(C)C)=O)CC1C1CCN(C(c2cc3c(F)cccc3[nH]2)=O)CC1 39131,c1(C(c2nnnn2C)OC)sc(Br)cc1C(=O)SC.C(CC)(C(=O)OC(C)(C)C)N 39132,C1(C(=O)OC)CC(NCc2cc(Br)co2)C12CCC2 39133,N1(C(C(CC)CC)=O)CCC2(CC1)CN(C(C1CCCC13CC3)=O)CC(C)O2 39134,C1(OCC)CC(NC(C2COCC(C)O2)=O)C12CCC2 39135,C1(C(N2CC=CC(C(N(CCC)C)=O)C2)=O)CC(C)(C)CN1C 39136,c1(C(N(C)CC2CCCN2C(=O)C=CC2CCCO2)=O)cc(O)cc(C#N)c1 39137,C1(C(N(CCCC)CC)=O)CC(NC(=O)CCCC)C1(C)C 39138,C1(N(C)C)CCCC(N=c2[nH]c(=NC3CC(N4CCC4)C3)[nH]c3c2COC3)C1 39139,N1(C(=O)CC2CC(F)(F)C2)CCC2CCN(C(C3CC4CC3C4)=O)C2C1 39140,CCCCC(CNC(c1cc(C2CC2)no1)=O)NC(c1cnc(Cl)s1)=O 39141,C1(C(N(CCCNC(c2ccc(F)o2)=O)CC)=O)CC1C1CC(F)(F)C1 39142,c1(C(=O)NCc2scc(CNC(CC3C(C)CCO3)=O)n2)cc(O)ncn1 39143,N1(C(c2ccc(C(C)C)c(Cl)c2)=O)CCN(C(c2cnncc2O)=O)C2(CC2)C1 39144,c1(OC)ccccc1C(=O)NCC(N1CC2(CC2NC(C2CCCC2)=O)C1)=O 39145,Cc1cc(=NCCCS(=O)(=O)C(C)(C)C)[nH]c(NCc2cccc(C)c2N)n1 39146,N1(C(CS(N)(=O)=O)=O)CCC2CCCN(C(=O)Cc3cccc4[nH]ncc34)C2C1 39147,C1(CNC(C(N2CCOCC2)C)=O)CC(F)(CNC(=O)CNC=O)C1 39148,C(=O)(C(C)S(=O)(=O)C1CCOCC1)NC1COCCN(C(c2cc(C)no2)=O)C1 39149,c1(C(=O)NCC(C)NC(c2cn(CCF)nn2)=O)cn(C)nc1CCC(F)(F)F 39150,c1(OC)noc(C2CC2)c1C(=O)NCC1CCCN1C(C1CC2CC2C1)=O 39151,c1(CC)cc(CC)ccc1C(N1CCC(C2CC2)(NC(=O)C(C2CC2)OC)C1)=O 39152,CCC(C)CCCC(=O)NCC(CNC(=O)Cc1cc(O)nnc1O)OC 39153,N1(C(C(C2CN(C(CC3ON=C(C)C3)=O)C2)O)=O)CCC2(CC1)CSC2 39154,c1(C(N2CCC(C)(NC(COC(C)=O)=O)C2)=O)nn(C)c(C)c1Br 39155,c1(CC(=O)NCC2(C)OCCN(C(C(CC)C(C)C)=O)C2)cccc2ccoc12 39156,C(=O)(CC1=Cc2ccccc2C1)N(CC(CC)NC(C1CC1C(F)(F)F)=O)C 39157,Cc1nc2cc(C(N3CCCC3CCCNC(=O)C(C)N(C)C)=O)ccc2s1 39158,C1(NC(c2c(C)c(Br)ccn2)=O)CCCC2CN(C(=O)CSC(C)C)CC12 39159,C1(C(=O)NCC=CCCOC)COCCN1C(=O)C(CO)OC 39160,C1(NC(c2c(C)cn(C)n2)=O)C(C)(C)C(NC(=O)CS(=O)C(F)(F)F)C1(C)C 39161,N1(C(C=CC(CC)=CC)=O)CCC2(CCCN2C(=O)CCc2ncc(F)cn2)C1 39162,c1(C(N2CCCC2CCC#N)C(=O)NC(CC)C)cnc(C2CCC2)s1 39163,C1(C(=O)NCC2CCN(C(C3C(C)CCO3)=O)C2)CCCN(C)C1 39164,CC1(C)CC(NC(=O)CC2C=CS(=O)(=O)C2)CN1C(=O)CCCn1ccnc1 39165,N1(C(C=C)=O)CC2(C1)CN(C(C1COCCN1C1CCCC1)=O)C2 39166,c1(-c2cn(CCC(=O)NC(c3ccccc3)CC)nn2)cc[nH]c(=N)c1 39167,c1(C(=O)NC(CCNC(c2nnc(C(C)(C)C)s2)=O)(C)C)nnc(O)cc1O 39168,C(=O)(CS(=O)(=O)c1ccccc1Cl)NCC1(O)CN(C(C(CC#C)O)=O)C1 39169,c1(C(N2CC(CCC)N(C(c3cncs3)=O)CC2)=O)ccc(Cl)c(F)c1O 39170,CC1(C)CN(C(=O)C=C2CCSCC2)CC1NC(=O)CSc1ccccc1Cl 39171,c1(C(N(C(CNC(c2cnn(CC)n2)=O)C)C)=O)onc(Br)c1C 39172,C1(CNC(C2(SC)CC2)=O)CCC(C)CN1C(c1ccc(C2CC2)o1)=O 39173,c1(CN(CCN(C(C)C)C(C2CCC(C(=O)NC)C2)=O)C)cncnc1O.C1CC1 39174,C(CCN=c1nc(N2CCCC(F)(F)CC2)c2c([nH]1)CCC2)C1C(C)C1 39175,C(=O)(C(CC(C)C)NC)NCC(C1CC1)NC(CC1C(C(=O)OCC)C1)=O 39176,N1(C(CCC=C)=O)CC2C(C(F)(F)F)CC2(NC(c2ccc(C)n2C)=O)C1 39177,N1(CCCN(C(=O)CCc2ccc(Cl)s2)C2CC2)CCCCCC1 39178,c1(OCC(=O)NCC(CO)NC(c2cnc(CC)[nH]2)=O)ccc(F)c(Br)c1 39179,N1(C(COCCN(C)C)=O)CC(C)(CNC(C2CCCCCCC2)=O)CC1(C)C 39180,c1(C(=O)NC2CC(C)N(C(c3cc4cnccc4[nH]3)=O)C2)cc(Cl)c(F)cc1N 39181,Cc1nc(C2CC2)nc(S)c1C(=O)NCC1CC2CC2N1C(=O)C(C)C(C)C 39182,N1(C(C(=O)NCCCOC)C2=NOCC2)CCC(C2CCN(C)CC2)C1 39183,C1(C(N(CC(C)NC(C23CCOC(C)(C2)C3)=O)CC)=O)CC2CCCCN2C1 39184,C#CCC(C)(CC)C(=O)NCC1CCN(C(C2Cc3ccccc3C2)=O)C12CC2 39185,C1(N=c2cncc(Cl)[nH]2)(CNC(Cc2n(C)nnc2)=O)CCOCC1 39186,N1(C(C=NOC)=O)CCC2CC(NC(=O)Cc3cnn(C)c3)CCC2C1 39187,CCCCCCCCCC(O)CCC(=O)NCc1cn(CC2CCCOC2)nn1 39188,CC1CC(C(=O)NC(C)(C)CCCNC(=O)Cc2cnc[nH]2)CCS1(=O)=O 39189,CC1CC(NC(c2cnc(Cl)s2)=O)CN(C(=O)CC2OC(C)(C)OC2=O)C1 39190,CC(CF)CC(=O)N1CCCC(CN(C(=O)Cc2cccn2C)C)C1 39191,N1(C(C(=O)NCCCCCCCC)=O)CCC2CN(C(C3(C)CC3)=O)CCC2C1 39192,CCC(C)(CC)C(=O)NCC1(O)CN(C(c2cccc(C#N)c2)=O)C1 39193,c1(OC)ccnc(O)c1C(N1CC(CNC(=O)C=Cc2ccnn2C)C1)=O 39194,N1(C(CC)=O)CCN(C2CCCN(C(=O)C=CC3CCCCC3)C2)CC1 39195,c1(OC)cnc(C(=O)N(C2CCCN(C(=O)C(C3CCCCC3)O)C2)C)c(F)c1 39196,N1(C(c2c(CC)nc(C)nc2)=O)CCCC2(C1)CN(C(=O)CC1=CCCCC1)C2 39197,C1(CN(CC)Cc2c(Br)ncn2C)(CO)CCN(C(=O)OC(C)(C)C)CC1 39198,C1(C(=O)NC(C(C)NC(C2CC3CC3C2)=O)CO)CC(C)(C)CO1 39199,C(c1cccc(C#N)c1)=CC(N1C(CNC(C(NOC)=O)=O)CN(C)CC1)=O 39200,N#Cc1cccc(N2CCC2)c1.c12nnc(CCCc3ccc(Cl)cc3)n1CC2 39201,C1(C(N(CC(C(C)C)OC)C)=O)C=CCN(C(C2CCC=CCC2)=O)C1 39202,C1(C(C(=O)N(CCC=C)CCOC)C)CCN(C(=O)CC2(OC)CCC2)C1 39203,CC(C)(CCNC(C1(CO)CCCO1)=O)NC(C1CCCO1)=O 39204,CC1CC(NC(=O)CN(C2CCCC2)C)CCN1C(=O)C=Cc1ccc(F)cc1 39205,C1(C(N2CC3C(CNC(CN4CCCC(CC)C4)=O)(C3)C2)=O)CC(C2CC2)=NO1 39206,c1(NC(N(CC(C)C)CCC)=O)ccc2c(-c3ccccn3)cccc2n1 39207,C(C(C)(C)C(=O)NCCC1CCCN(C(=O)CCc2ccccc2C)C1)SC 39208,n1(C)ccc(O)nc1=O.C1(C(=O)NON2C(N)C=CC2)CCN(CC(c2ccccc2)O)C1 39209,C1(CNC(CCCCCOC)=O)CC2(CCC2)CN1C(=O)C(C)CC1CCCC1 39210,C(=O)(C1=COCCO1)NCC(CN(C)C(c1ccc(C(=O)OC(C)(C)C)cn1)=O)O 39211,c1(C(=O)NCC2(C)N(C(CCC(=O)OCC)=O)CCC2)nnc2ccccc2n1 39212,N1(C(C(C)OCCOC)=O)CCN(C)C(C(=O)NC2CC(CO)(CO)C2)C1 39213,C1(CC=C)(C(=O)NC(C=C)C2CCC2)CCCN1C(=O)C(C)CN(C)C 39214,Nc1cncc(C(=O)NC2CCCCC2CNC(c2cc(Br)no2)=O)c1 39215,S(=O)(=O)(c1cccc(Cl)c1)NCCC(=O)N(C1CCCN(C(CCSC)=O)C1)C 39216,N1(C(C(C(C)C)OCC)=O)CC2(NC(=O)C(C)SC)CCC1CC2 39217,CC1CCC(C(=O)NCC2(NC(=O)COCC3CCCC3)CC2(C)C)CC1 39218,N1(C(C(=O)NC(C)C)=O)CCN(C(=O)C(CC2CC2)C(F)(F)F)C2CCCC12 39219,C1(C(=O)NCC(=O)NCC(=O)Nc2c(OC)nccc2)CCOC(=O)CC1 39220,N1(C(C(CC#C)C)=O)CCCC(CC=C)(NC(c2cc(Cl)ccc2Cl)=O)C1 39221,C1(OCC(=O)N(CC(C)NC(=O)Cc2cc(C3CC3)no2)C)CCC(F)(F)CC1 39222,C1(C)(OC)CCCN(c2cc(NCc3nc(C)c(C)o3)nc(C(F)(F)F)n2)C1 39223,CC1CCN(C(c2n[nH]cc2Cl)=O)CCN1C(=O)CCCS(N)(=O)=O 39224,c1(N2CCC3(C(NC(c4cc(F)c[nH]4)=O)CC3)CC2)ncc2c(Br)cccc2n1 39225,c1(C(=O)NCCN(C(=O)C=Cc2ncc[nH]2)CC)ccc(-c2ccccn2)cc1 39226,c1(CNC(=O)NC(C2CN(C)CCN2C)C)cccc(F)c1Br 39227,C(=O)(C(C(C)(C)C)n1ccnn1)N(CC(C)O)CCNC(=O)COC1CCOC1 39228,C(=O)(CS(=O)(=O)CCO)N1CCC(C)(CNC(C2C(CC(C)C)C2)=O)CC1 39229,N1(C(C=C(c2n(C)ncc2)F)=O)CCCC2(CCN(C(=O)CN3CC=CC3)C2)C1 39230,C(=O)(C1=CCCCO1)NC(CCOC)C(=O)N1CC(C)=C(C)C1 39231,C1(C(=O)NCC2N(C(CN3C(C)CCC3)=O)CCC2)CC(S(C)(=O)=O)C1 39232,CC1CN(C(C2COC(C)(C)O2)=O)CC2(CCN(C(=O)CN3CCC3)C2)O1 39233,CC(C)CC(O)CC(=O)N(CC(N1CC(CO)CC(C)C1)=O)C1CC1 39234,N1(C(c2cncc(NC)c2)=O)CCN(C(=O)CC(C)(F)F)C(C(C)C)C1 39235,C1(C)(N(C(c2ccc(-c3ccccc3)o2)C(=O)NCC=C)C)CCCC1O 39236,N1(C(c2[nH]c(CC)c(Cl)n2)=O)CCC(NC(c2ccn(CC(C)C)n2)=O)C(F)C1 39237,N1(C(C(=O)NC(CC)(C)C)CC(C)SC)CCc2cc(C)cc(C)c2C1C 39238,N1(Cc2c(Br)ccc(F)c2F)CCc2ccc(Cl)cc21 39239,N1(C(=O)Cc2sccc2Cl)CCCC(N(CCO)C(C2CC(F)C(=O)N2)=O)C1 39240,CN1CCC2CC(C(=O)NC3(C4CCCC4)CCNC3=O)CCC12 39241,N1(C(C(c2ccn(C)n2)C)=O)CC=CCC1C(=O)N(C)CC1(C)CC1 39242,CC(C)CCCC(C)C(=O)NC1(C2CCCN2C(c2cnc(C(C)C)o2)=O)CC1 39243,N1(C(C2C(=C)C2)=O)CC2CC(CNC(c3ccc(C(C)(C)C)[nH]3)=O)C2C1 39244,C1(N(C(C)=O)CC2CCN(Cc3nc(C(=O)O)co3)C2)CCS(=O)(=O)C1 39245,C(=O)(C(C)(C(C)C)NC(C)=O)NC1(CNC(COCC(=O)NC)=O)CCC1 39246,N(C1CCCn2ccnc21)C(C(C(C)CC)N(C(C=C(CC)CC)=O)C)=O 39247,n1(C(C)C)ncc(C(N2CCC(CF)(NC(=O)CC3CCCC(=O)N3)C2)=O)c1Cl 39248,N=c1ccn(CC(=O)NCC2(CNC(=O)CCc3ccccc3)CCC2)[nH]1 39249,c1(C(=O)NC2C(C)CN(C(c3c[nH]nc3-c3ccoc3)=O)C2)cc(=O)cc(Cl)[nH]1 39250,c1(C(N2CCC(CC3CC3)CC2)=O)ccc(F)cc1C(F)F.N12CCN(CC1)C2=O 39251,N1(C(C2(OCC)CCCC2)=O)CCCN(C(=O)Cn2nnc(C(C)(C)C)n2)CC1 39252,C1(CNC(CN(CC)CC)=O)CCCN(C(c2ccc(F)c(Cl)c2)=O)CC1 39253,c1(C(N2C(CCNC(=O)CC3COCCO3)CSCC2)=O)cnn2ccsc12 39254,N1(C(CCN(C(C2C(=C)C2)=O)CC)=O)CC(C)OC(C)(C)C1 39255,N1(C(C(C2CCCC2)OC)=O)CCC(NC(c2cc(C(C)C)on2)=O)CC(O)C1 39256,C(=O)(NNc1nc(Cl)ccc1Br)NCCc1cc(C)on1 39257,CC1CCCC(N2CCN(C(c3ccoc3)=O)CC2)C1 39258,c1(N(CCCNC(c2cccc(OC)c2C)=O)C2CC2)nc2ccccc2o1 39259,c1(C(=O)NCC2N(C(C3N(C(C(C)=CC)=O)CSC3)=O)CC2)ccc(NC)cn1 39260,Cc1noc2ncnc(N3C4CCC3CN(C(=O)CC3CCCCC3)C4)c12 39261,c1(CN(C)C(C2(C)CC2)=O)cnn2c1CN(C(c1cc(F)ccc1F)=O)CC2 39262,C(=O)(C(O)C(F)(F)F)NC1CC(NC(CC(C)(C)CC)=O)CC1O 39263,C(=O)(C1=CCC(C)(C)CC1)N1C(CNC(C2(COC)CCCC2)=O)CCC(C)C1 39264,c1(C(N(CCC(N2C(C=C)CCC2)=O)CCO)=O)ccc2c(c1)CCC2 39265,C1(C(=O)NCC(C)(C)NC(=O)C(c2ccc(F)cc2)CO)CCCCN1N=O 39266,C(=O)(C(Cn1ccnn1)NC(c1cc(C2CC2)[nH]n1)=O)NC(CCOCC)C 39267,c1(-c2nc(CC(C(CC)O)C)n(CCC(=O)N(C)C)n2)csc2cc(C)ccc12 39268,c1(C(N2CC(CCNC(=O)C(c3ccn(C)c3)C)(OC)C2)=O)ccc([N+](=O)[O-])o1 39269,C1(O)(CC(N2CC(O)(CCNC(C(C=C)(C)O)=O)C2)=O)CCN(C)CC1 39270,C1(NC(C(=O)N(CC)CC2Cc3ccccc3CO2)=O)CC2(C1)CC1(CNC1)C2 39271,C(c1ccc(N(C)C)cc1)=CC(=O)N(CCC(C(C)C)NC(C1CC1CF)=O)C 39272,C(CCS(=O)(=O)c1ccc(C)cc1)N(CC(=O)N(C1CC1)CC)CCC 39273,N1(C(C=CCCC(C)C)=O)CCC(C)C(CNC(C2(C)CCC2)=O)C1 39274,N1(C(CCCN(C(C2C(C(=O)OC)CC2)=O)C)=O)CCC12CCCCC2 39275,CCCCCCC(F)C(=O)N1CCC(N(C)C(c2ccc(O)c(N)n2)=O)CC1 39276,c1(C(=O)NCCOCCNC(C2C(C=C)C2)=O)cccc(CC)c1N 39277,Cc1scc(C(=O)NC2CCC(n3ccnn3)CC2)c1N 39278,n1(CC)cnc2[nH]c(=NCc3ocnc3C)nc(N3CC4CC3CS4=O)c12 39279,c1(CC(=O)NC2CC(NC(c3c(COC)nn(C)c3)=O)C2)c(C)cccc1C 39280,c1(C(=O)NC(CC)C(O)C(F)F)nc2c(s1)CCCC2 39281,Cc1cccc(NC(=NCCc2ncnn2C)NC2CCCC2)c1C(C)(C)C 39282,c1(N2CCCN(CC=C)CC2)nc(NCCC2CC2)c2cnn(C)c2n1 39283,C1(C(N2CCCC(NC(=O)COC3CCCC3)CC2)=O)CC2(C1)CC(C#N)C2 39284,C(C(=O)NOCCN(C)C)=C(CNC(C1CC(=C)C1)=O)C 39285,C(=O)(C(CC(C)(C)C)OC)NC(C(N1C(C)(CCC)CC1)=O)Cn1cccn1 39286,C1(NC(c2c(OC)ccnc2)=O)CCCC2CN(C(C3(C)CCCC3C)=O)CC12 39287,n1(CCC(N2CCN(C(CSCCOC)=O)C(C)C2)=O)c(=O)oc2ccccc12 39288,c1(OC)nc(Br)ccc1C(N1CC2CC1CN2C(c1cccc(F)c1O)=O)=O 39289,c1(C(c2n(CC(=C)C)nnn2)N(CCCCOC)C2CC2)cccc2nccn12 39290,Cc1cccc(OCCC(N2CC(NC(c3ncccn3)=O)CCC2C)=O)c1C 39291,C1(C(N2CCN(C3CCC(C)CC3)CC2)=O)CC2(CC(=O)N2)C1 39292,n1(CC(=O)N(CCNC(C(N2C(=O)CCC2=O)CC)=O)C)cc(S(N)(=O)=O)cn1 39293,N1(C(Cc2ccc(C)cc2Br)=O)CC2COCCC2(NC(c2cn[nH]c2)=O)C1 39294,C(C)(CO)(CS(C)(=O)=O)C(=O)NCC(c1ccc(OC)cc1)OC 39295,C(=O)(C(F)C(C)CNC(C1CC2CCC2C1)=O)NCc1cc(OC)ncc1 39296,C1(NC(C2(S(N)(=O)=O)CC2)=O)CN(C(C2CC3(CC3)CO2)=O)CCC1CO 39297,c1(OC)ncc(C=O)cn1.c1(C(=O)NC2CN(C(=O)C3CC3)C2)[nH]nnc1C 39298,CC1(C)OCC2(CCN(C(C3CC(=O)N(c4c(F)cccc4F)C3)=O)C2)CO1 39299,C(=O)(CC1=CCCC1)N(CC(C(=O)NCC(C#C)CC1CC1)C)C 39300,CC(C)S(=O)(=O)c1ccc(C(N2CC(C(C)NC(=O)C3=CC(C)(C)C3)C2)=O)cc1 39301,CC(C)CC(CC(=O)NCC(O)C(N)=O)NC(C1CCCCC(=O)N1)=O 39302,N1(C(CCN(C(CC)CC)C)=O)CCC2CCN(C(C3CC4(C3)CC4F)=O)CC12 39303,CCCC(CCC)CC(=O)N1CCCC1CNC(C1(CC)CC(C)(C)C1)=O 39304,c1(C(C)=O)ccc(C(=O)NC2CCC(CNC(c3ccc(Br)s3)=O)C2)o1 39305,C1(NC(Cc2cc(C)[nH]n2)=O)COCCN(C(=O)Cc2ccccc2C(F)(F)F)C1 39306,C1(NC(C(CC)OCC)=O)CN(C(c2cn(C(C)(C)C)nc2C)=O)CC12CC2 39307,C1(CNC(C(COC)O)=O)N(c2ccnc(C(C)(C)C)n2)CCCC1(C)C 39308,c1(C(N(CCC(C(C)C)NC(=O)CCOCC2CC2)C)=O)cccc(N)c1O 39309,CC1CN(C(c2ccc(C(F)(F)F)[nH]2)=O)CC1CNC(C1(S(C)(=O)=O)CC1)=O 39310,N1(C(C(CCC)NC(C)=O)=O)CC(CNC(c2cc(N)ccc2C)=O)C(C)(C)C1 39311,C1(=CC(=O)N(C)CCNC(C2(n3ccnn3)CC2)=O)CCCCCC1(F)F 39312,C1(CNC(c2c(CC)ncs2)=O)CCC(C)CN1C(c1cc(C2CC2)nn1C)=O 39313,c1(CC)ccc(F)cc1C(N1CCC(NC(=O)CSC(F)F)C(CC)C1)=O 39314,n1(CCC)nc(C)cc1C(=O)NCC1CC1CNC(C1(CF)CC1)=O 39315,N1(C(CSC)=O)CCC2(CCC(NC(c3ccc(C4(C)CC4)cc3)(C)O)CC2)C1 39316,C1(C(N2C(COC)(CNC(=O)Cn3cc(C)cn3)CCC2)=O)CCC(C)(O)CC1 39317,c1(C(N(CCC(C)NC(=O)CC(C)c2cccnc2)C)=O)ncncc1Cl 39318,CCCCS(=O)(=O)NC(C)C(N1CCC(CNC(C2CCCCC2C)=O)CC1)=O 39319,c1(OCC=C)ccc(Cl)nc1C(N1CCC(C(C)CNC(=O)CCOC)CC1)=O 39320,N1(CCCNC(CC2(C)CCCC2)=O)CCN(C(=O)CCC(F)F)CC1 39321,N1(C(C2(CC=C)CCC2)=O)CCC2(C1)CN(C(=O)C(C)NC(=O)OC)CCO2 39322,C1(CCC)CN(C(c2cccnc2)=O)CC1C(=O)NOCC1CCC1 39323,C1(OC)CC(N=c2[nH]c(=NCCP(C)(C)=O)[nH]c3c(F)cccc23)C1 39324,N1(C(c2nc(OCC)oc2)=O)CC=C(CCNC(C2CCOC(C)C2)=O)CC1 39325,C(=O)(C(CCc1cccc(F)c1)C(C)(C)C)NC12C(CN(C(C=CCC)=O)C1)C2 39326,n1(CC)ccc(C(N2CCC(CNC(=O)CCc3cncs3)C23CC3)=O)cc1=O 39327,CCCCC(C(=O)N=c1ccn(Cc2ccco2)[nH]1)C(C)C 39328,C1(C#N)(C(=O)NCC(CNC(c2ccc(NC)cc2)=O)F)CCS(=O)(=O)CC1 39329,CCC(C)CC(C(=O)NCC#CC#CCO)NC(=O)CCN(CC)CC 39330,C1(NC(C(CC)(C)CNC(=O)CCc2cscn2)=O)CC12CCCCCC2 39331,C1(NC(C=CC(C)(C)NC(CC(=O)OCC)=O)=O)CCCCC1C 39332,C=CCC(CC(C)C)C(=O)NCC1(C)CCCN1C(=O)C(CC(=C)C)OC 39333,c1(C(=O)NCC2(CNC(c3c(C)scn3)=O)CC2)cnn(C2CCOCC2)c1C 39334,C1(C(=O)NC(C#C)C)(OC)CCN(C(c2cc(C)cc(F)c2)=O)CC1 39335,C(CC(O)C(=O)NC1CCOCC1NC(c1cc(-n2cnnc2)ccn1)=O)SC 39336,N1(C(c2c(CC)scc2)=O)CC2(CCN(C(=O)CCF)C2)C1 39337,C(=O)(CCCCC(C)C)NC(CCN(C(C=Cc1n(CC)ncc1)=O)C)C(C)C 39338,C1(C(=O)NCC(C)(C)NC(=O)CCc2ccc(C#N)cc2)CCS(=O)(=O)C1(C)C 39339,C1(CNC(c2c(CC)sc(=N)[nH]2)=O)COC(C(C)C)CN1C(=O)CSC(F)F 39340,c1(CCC(=O)NC2CCN(C(=O)C(F)F)C2C2CC2)ccc(Br)cc1Cl 39341,c1(C(=O)NC2COCCN(C(C(CC(C)C)(C)O)=O)C2)ccnc2c1CC(=O)N2 39342,N1(C(CCC2N(C(c3c(C#C)cnn3C)=O)CCCC2)=O)CCC2(C=CCO2)C1 39343,N1(C(CCSCCCC)=O)CCCCC1C(N(C)Cc1oc(C)nc1CC)=O 39344,c1(OC)cc(CC)ccc1O.N1(CC(C)C)CCCC(C(C)NC(C)=O)C1 39345,O=C(C1=CCC(NC(=O)CC2CC3(CC3)CO2)C1)Nc1ccc(Cl)c(O)c1 39346,C1(CCNC(=O)C(C2CCCCC2)F)CCCN(C(=O)Cc2cccnc2)C1 39347,c1(OC)cccc2cc(C(=O)COC(=O)CSCN=S(C)(C)=O)oc12 39348,CC1CCCCC1(C)NC(=O)C(c1cnn(C)c1)NC(=O)CC(=O)NC1CC1 39349,C(=O)(C(CCCCCO)N1CCC(c2nc(C)cs2)C1)NCCOCC 39350,C1(C(N(C(C2CCC2)C)CC)=O)CCCC1CNC(=O)CCCn1ccnn1 39351,C1(C(C)C)CCN(C(=O)CN(C(c2ccc(=N)[nH]c2)=O)C2CC2)CC1 39352,CCC(CC(=O)NC1(CCNC(C2C(F)(F)C23CC3)=O)CCCC1)C(C)C 39353,CCC(CC(=O)N1CC2CCN(C(c3cn(C)c(=O)n3C)=O)C(C2)C1)C(C)(C)C 39354,C(c1ccc(C)c(Cl)c1)=CC(=O)NCC1C(NC(C(n2ccc(C)n2)C)=O)CC1 39355,c12cncc(n1)N2.C(=O)(CC(=O)NCCNC(=O)COC1CCCC1)OC 39356,c1(N(C2CCCN(C(CC(CCC)O)=O)CC2)C)nc(C2CC2)nc2[nH]ccc12 39357,C(C(COC)C(=O)N1CSCC1C(=O)NCCn1cnnn1)OC 39358,N1(CC(C)(C)C)CCC(O)CC1C.c1(OC)ccc(C2C(=O)N2)cn1 39359,c1(C(N2C(COC)(CNC(C3CC(C)CO3)=O)CCC2)=O)ccc([N+](=O)[O-])n1C 39360,C(C(C)(O)C(=O)N(CC(C)N(C(=O)CCn1cncn1)C)C)OC 39361,CC(O)C(C)C(=O)N1CCN(C2CCN(C(C34CC3C4)=O)C2)CC1 39362,c1(OCC=C)ccccc1C(=O)NCCC(C)CCNC(c1cc(Cl)n(C)n1)=O 39363,N1(C(C2C(C)C2C)=O)CC(CNC(=O)CC2CC(C)OC2C)OC(C)(C)C1 39364,N1(c2cc3nnn(CC)c3cc2)CCCn2cc(Br)cc2C1 39365,c1(OCCC=C)ccc(NC(=O)C(N)Cc2ccc(F)cc2)cc1C 39366,N1(C(CONC(C#CC(C)C)=O)=O)CCC(C2CCOC2)C1 39367,N1(C(CCOCC#C)=O)CC(CNC(=O)C(CO)c2ccccc2)CC12CCC2 39368,c1(CN2CC(C)C(N3CCOCC3)C2)cc2c(Cl)nccc2s1 39369,C1(CCCNC(CCOC)=O)CCCCN1C(=O)C(N1CCC(C)CC1)=O 39370,C1(C(N2CCC(=CCNC(c3c(CC)nn[nH]3)=O)CC2)=O)CN(CP(C)(C)=O)C1 39371,C1(CNC(C2(C(C)C)CCC2)=O)CCN(C(c2cnn[nH]2)=O)C12CCC2 39372,N1(C(CCSCC)=O)CCCC1C1CCCCN1C(=O)CN(C)C 39373,c1(NC(COc2cn(C(C)C)nc2)=O)ccc(C(=O)O)c(Cl)c1C 39374,N1(C(C2N(C(C3C4CC(=O)CC43)=O)CCC2)=O)CCc2cncnc2C1 39375,CC(C)CCCCCC(=O)NCC1(O)CCCN(C(=O)C(C)CC(F)(F)F)CC1 39376,C1(C(=O)NC(CC2CN(C(Cc3onc(C(C)C)n3)=O)C2)C)CCC=CCC1 39377,c1(C(=O)NC2C(NC(c3cc(CC)on3)=O)COCC2)cc2nccn2c(O)n1 39378,c1(C(CC(=O)OC)NC(=O)CNC(N)=O)cccc(-c2cccnc2)c1 39379,CCC(C)CCC(=O)NCC(c1ccc(F)cc1)NC(=O)C=Cc1cc[nH]c1 39380,C1(NC(CN(C)C(N)=O)=O)CCOC(CNC(=O)CC2COCC2(C)C)C1 39381,C1(Cl)(C(=O)OC)CC1C(=O)N(CCC(C)NC(C1(N(C)C)CC1)=O)C 39382,C1(CCC)CN(C(=O)C(C)C#N)CC1NC(c1ccc(N(C)C)nn1)=O 39383,N#CC1CCCC1NC(C1CCCCN1c1nccs1)=O 39384,C1(NC(C=CC(CC)C)=O)CCCCCN(C(=O)Cc2ccsc2)C1 39385,C(=O)(C(C)(C)C(C)(F)F)N(C)CC1(NC(C(CCC)c2ccc(Cl)cc2)=O)CC1 39386,C(C(C)(C)C(c1nnnn1C(C)C(=O)OC)NCc1sc(Cl)nc1C)OCC 39387,c1(CCC(=O)NC2C(NC(CCCNC(C)=O)=O)CCC2)cccc(F)c1F 39388,c1(C(CNC(CCOC)=O)NC(=O)C(C)C#N)ccc(C(C)C)cc1 39389,CC(C(=O)NCC1CN(C(=O)CCn2cc([N+](=O)[O-])cn2)CCO1)C(C)(C)C 39390,Cc1ccc(F)cc1N(C(=O)C(C)N(C)C(c1cc(Cl)cs1)=O)C 39391,C(CC(=O)NC(C)CC1CN(C(=O)CC2CC2C)C1)NC(COC)=O 39392,c1(C(=O)NCC(C2CC2)NC(C2N(C)C(=O)CC2)=O)cncc2ncn(C)c12 39393,c1(C(=O)NC(C2CN(C(C(CC)N(C)C)=O)C2)C)cnn(CCO)c1N 39394,c1(C(N2CCC(NC(c3cc(OC)n[nH]3)=O)C23CC3)=O)n[nH]c2c1CC(C)CC2 39395,O=NN1CCCCC1C(N1CCCC(NC(c2cnoc2)=O)CC1)=O 39396,C1(NC(C2C(C)C2)=O)CCC12CCN(C(=O)CN(CCO)Cc1ncnn1C)CC2 39397,CCC(CCC(=O)N1CC=C(C)CC1)NC(=O)CCNC(=O)NC 39398,N(C(=NCCC(=O)N(C)C)NCC1CCN1C(C)(C)C)CC(CC)(C)C 39399,c1(C(OC)CC2CCCC2NC(c2sccc2-c2cccs2)=O)cn(CC)nn1 39400,CCC(CCCC(=O)NCC1(CC(=O)OC)CC1)NC(C1(C)COCCO1)=O 39401,C1(C(=O)NC(C)Cn2cncn2)CCN(C(=O)c2ccn(C(F)F)n2)O1 39402,C1(OC)CC(NC(C2CC(O)C2)=O)CN(C(c2cc(C)oc2C(F)(F)F)=O)C1 39403,c1(OC)ccc(Cl)cc1C(N1CCC(CCNC(C2(C)CCN(C)CC2)=O)C1)=O 39404,C(=O)(C(C)CCCC(C)=O)NC1CN(C(C(C(CC)CC)OC)=O)C2(C1)CCC2 39405,N1(c2nc(N3CCCC(CC(=O)NC)C3)nc(C)c2)CCc2nc(O)[nH]c2C1 39406,c1(SC)ncc(C(N2CCSC(C(=O)Nc3ccc(Br)nc3)C2)=O)c(Cl)n1 39407,C(c1ccsc1)=CC(=O)NC(C)CCN(C(=O)C(C)N1CCCC1)C 39408,Cc1noc(C2CC2)c1C(=O)NC(CNC(c1ccnc(C2CC2)c1)=O)C(C)C 39409,CC(C(C)NC(=O)CSc1nncs1)NC(c1csnn1)=O 39410,c1(CC(=O)NC2C(C(=O)OC)C2)ccc(Cl)c(C)c1.C(C)(C)(C)CCN1C(=O)C1 39411,C1(C)(C(=O)NC2C(CCC)C2)CCCN(CC)C1.C12(OC)CN(C1)C(=O)C2 39412,c1(N2CC(NC(CCCC)CO)(CO)C2)ncnc2sc(C(=O)OC)cc12 39413,N#CC1CCCC(C(N2CCOC(C(N3CCCC3C(N)=O)=O)CC2)=O)C1 39414,C1(CCC)CCCN1C(C1CC1C(C)C)=O 39415,C1(=O)C(CC(C)(C)C)NC(=O)C(CSC)NC(=O)COC1CCOCOC 39416,C1(C(C)NC(CCCOCC=C)=O)CCCCN1C(=O)CCc1nccn1C 39417,c1(C(=O)NC(C(C)NC(COC(CC)CC)=O)C)cc(C)c(F)cn1 39418,c1(N(CC#C)C(=O)Nc2cccc(N3CCCC3=O)c2)cccnc1OC 39419,c1(NS(=O)(=O)CC2CCN(Cc3ccc(CO)o3)C2)ccc2ncnn2c1 39420,C(=O)(CCCCNC(N)=O)N1CC(CCCCNC(C(CC)n2ccnc2)=O)C1 39421,Cn1cc(C(N2C(C)CC2(C)C)=O)c(-c2ccco2)n1 39422,c1(SC)cc(=NC(=O)C2CC(C)N2C(=O)CCC2(C)N=N2)[nH]n1C 39423,C(=O)(C(CC)CC(F)F)N1C(CN(C(c2n(C=C)ncc2)=O)C)CCCC1 39424,CN=c1[nH]cc(CSC2(CCCNC(=O)OC(C)(C)C)CC2)s1 39425,N1(C(C=CC(C)C)=O)CC(NC(=O)CCOc2c(F)cccc2Cl)CC(C)C1 39426,CCCCC(O)C(=O)NCc1cc(C(N2CCCC(C)C2CCO)=O)no1 39427,C1(C(=O)NC(C#C)CC2CCC2)C2CC3C(C2NC(=O)CCOC)C13 39428,C1(CCC(=O)NC(CNC(C(CC)C2CCC2)=O)C(C)C)NC(=O)NC1=O 39429,c1(C(=O)NC(C2CCCN(C(=O)COC(F)(F)F)C2)C)ccnc2ccccc12 39430,C1(NC(c2cnc(CC)[nH]2)=O)CCN(C(c2nc(Br)cnc2N)=O)CC1C 39431,N1(C(C(=O)NCCC)C)CCCC1C1CCCCN1C(=O)CC1CC=CCC1 39432,c1(C(N(C)CC2(NC(C3CC3(F)Cl)=O)CC2)=O)c[nH]c2ccncc2c1=O 39433,N1(C(c2c(CC)cco2)=O)CC(F)CC1CC(N1CCC(O)(COC(C)=O)C1)=O 39434,N1(CC)CC2CN(C(=O)N=c3[nH]nc(N(C)C)s3)CC2C1 39435,N1(C(c2c(C)c[nH]n2)=O)CCCC2CN(C(=O)Cc3ccc(C#N)cc3)CC12 39436,Cc1cc2ccccc2cc1C(=O)NCC(O)CNC(c1cc(Cl)ccc1N)=O 39437,Cc1nc(CNC(c2nnsc2N)=O)oc1C(=O)NCCOCC(F)F 39438,C=CC(C)(O)C(=O)N(CC(C)C(=O)NCCn1cccnc1=O)C 39439,c1(C(=O)NC(c2ccc(I)cc2)(C)C)n[nH]c2cc(N)ccc12 39440,Cc1cccc2c1CCN2C(C(=O)NCC1CCCO1)c1ccco1 39441,Cc1ccc(C#N)c(N(C)CCN(C(=O)CNC(C2CCCC2O)=O)C)n1 39442,S(=O)(=O)(c1ncc(F)cn1)NCC(C)S(C)(=O)=O 39443,c1(CSC)noc(C)c1CN=C(NCC1(C#N)CC1)NC(c1cccs1)C 39444,C(=O)(C(CC1CCCC1)N1CCC(C(=O)OCc2ccccc2)C1)NC 39445,C1(CNC(N2CC(c3nc(C(F)(F)F)no3)C2)=O)CCC12CC(F)(F)C2 39446,c1(OC)c(C(N2CCC(O)(CNC(=O)CCC(=O)N(C)C)C2)=O)ccc(Cl)c1C 39447,N1(C(C2CC(C#N)C2)=O)CCC(O)(CNC(C2CC(=O)N(CC(F)(F)F)C2)=O)C1 39448,c1(NC(C2(C)CN(c3ncncc3I)C2)=O)cc(C#N)cn1C(C)(C)C 39449,Cc1ccc2nc(N3CC4CC3(CNC(=O)CC3C=CCC3)C4)sc2n1 39450,N1(C(C2C(O)CCN(C(C3N(C(C)=O)CSC3)=O)C2)=O)CCCC2CNCC12 39451,Cc1cc(C(F)(F)F)c2cc(C(=O)NC(C)CCN(C)C)oc2n1 39452,CCC(CC)C(O)CNC(=O)CC1CN(C(=O)CCc2ccco2)CC1C 39453,N1(C(C2(CC)COC2)=O)CC(N(C)C(C2CCCC2)=O)C(C)(C)C1 39454,N1(C(c2cnc(C(C)O)s2)=O)CCC(C2CCCN(C(C3(C)CC3(F)F)=O)C2)C1 39455,CON(C)C1CN(C(C2CCN(C(c3ccc(C)o3)=O)CC2C)=O)C1 39456,c1(N(CCCCO)C)nc(=NCc2cc(F)ccc2Cl)[nH]c2c1COCC2 39457,Cn1nnc(Cn2nnnc2C(COCC(F)(F)F)NCc2ccco2)n1 39458,C1(C(=O)NC)CCCN(C(C2CC3CCC2O3)C(=O)NCC(F)F)C1 39459,C1(SC)CCC(N=c2nc(N(C)CC3CCSCC3)c3c([nH]2)CCCC3)CC1 39460,C(=O)(C(F)(F)C(O)C1CC1)N1CCC(NC(C(C(C)C)NC(N)=O)=O)C1C 39461,C(CNC(=O)C=Cc1cncc(F)c1)(C(C)C(C)C)NC(CNC(COC)=O)=O 39462,c1(OC)cc(CN(C(=O)C(=O)NC2CCCNC2)C)ccc1OCCCC#N 39463,N1(C(=O)OC(C)(C)C)CCN(C(c2cccc3oncc23)=O)CCCC1CCO 39464,CC1CC(=O)CCC1C(N1CCC(C(=O)NCCOCC(F)F)C1)=O 39465,N(C)(S(N)(=O)=O)CC(=O)NC1CC(N(CC(=O)Nc2ccco2)C)C1 39466,C(=O)(C(O)CC(F)(F)F)N(c1ccccc1)CCNC(C(CC)NC(C)=O)=O 39467,CC(CS(C)(=O)=O)C(=O)NCC1(C)CCCN1C(=O)CCC(C)(F)F 39468,C1(NC(c2c(OCC)scc2)=O)(CO)CCN(C(c2ccc(C)nn2)=O)C1 39469,CC1(C(=O)NC2CCC(F)(CN3CCCC3)C2)Cc2ccccc2N1.C1(=O)CCN1 39470,c1(CC)ccc(C(N2CCCC2CN(C(=O)Cc2cc(C3CC3)no2)C)=O)o1 39471,N1(C(CS(CCOC)(=O)=O)=O)CCOC2(C1)CN(C(c1ccc(N)c(F)c1)=O)C2 39472,C1(NC(c2c(C)nc(CCC)o2)=O)CC2CC(NC(C3(C)CC=CC3)=O)C2C1 39473,c1(C(N2CCC(NC(C(CC#C)(C)C)=O)C2)=O)cc2c(C)[nH]nc2s1 39474,c1(C(N2CC(CC(C)NC(CCSC)=O)C2)=O)ccncc1Cl 39475,C(=O)(C(O)CC(F)(F)F)NCC1CC(C(=O)NC2C3(CC(OC)C3)C2)C1 39476,CCCC(C)(C)C(=O)NCC1CCC(C(N2CCC(CCN(C)C)C2)=O)CC1 39477,C1(C)(C(=O)NC)CCN(C(=O)C(=O)Nc2cnn(-c3nccs3)c2)CC1 39478,c1(COC)nc(=N)[nH]cc1C(N1CC(NC(=O)C(O)C2CC2)C1)=O 39479,C1(NC(c2c(C)con2)=O)CC2(C(=O)NC3CC(CO)(CO)C3)COC1C2 39480,C12(C(=O)NC(C)CC3CN(C(C4CCCC(C)(C)C4)=O)C3)CC=CCN1CCC2 39481,C1(C(=O)NC2CCN(C(c3nccc(CC)c3)=O)CC2F)Cc2ccccc2C1 39482,C1(NC(COCC)=O)CCCCC12CCN(C(c1cc(O)c(O)c(O)c1)=O)C2 39483,Cc1cc(C(=O)N(CCCCC(=O)N2CCOC(C3CC3)C2)C)oc1C 39484,c1(CC)cc(C(=O)NC2(CO)CN(C(C3CCCC3O)=O)C2)sc1C 39485,C1(=O)CC(C)(C)CC(=O)N1.c1(CC(N2CCCS2(=O)=O)C)cccc(Br)c1 39486,c1(CNC(=O)NC(c2ccc(OC)c(F)c2)C)c(C)cc(Cl)nc1Cl 39487,c1(OC)c(F)cc(C(=O)NCC2CCN(C(=O)CCCSC)CC2)cc1F 39488,N1(C(CCCOC)=O)CCC2CCCC12CNC(c1cc(Cl)ccc1F)=O 39489,c1(OC)cc(CNc2nc(C(=O)Nc3cc(Cl)c(O)c(Cl)c3)cs2)cc(O)c1O 39490,C(=O)(C(F)C(C)(C)O)NC1CC(C(C)NC(c2cncc(CC)c2)=O)C1 39491,C(=O)(C1CCCc2n[nH]cc21)N1C2C(NC(=O)CCn3cnnn3)(CCC2)CC1 39492,C1(C(=O)NCCS(CC)=O)(CNC(=O)OC(C)(C)C)CCC(C)(C)CC1 39493,C1(N(CC(N2CC(C)(NC(=O)Cn3nccn3)C2)=O)C)CCCC(C)(C)CC1 39494,c1(CN(C2CCCC23CCNCC3)C(COC)=O)c(O)c(Cl)cc(Cl)c1Cl 39495,C(=O)(NNc1cc(C(=O)O)ccc1Br)c1onc(OC)c1I 39496,N1(C(C=C(CC)C)=O)CCC(N2CCN(C(C3CCOC(=O)N3)=O)CC2)CC1 39497,N1(C(C(C)OCCN(C)C)=O)CC2CC(C1)N(C(C1(C)CC1(F)F)=O)C2 39498,CC1=CC(C)CN(C(C2CCC(NC(=O)CCc3cccn3C)CC2)=O)C1 39499,C(C)(C(C(=O)N1CC(c2ccccc2)C1)C(C)C)ONC(c1c(C)c(Cl)ccc1)=O 39500,Cc1ncc(Cl)cc1C(=O)NCC1(C(F)F)CCN(C(=O)C(C)N2CCC2)C1 39501,N1(C(c2ccc3occ(C(=O)OC)c3c2)=O)CCCCC(C2CCOC2)C1 39502,C1(C2CCC2)(C(=O)NCC2CN(C(C3(Cl)CC3)=O)CC2O)CC1(F)F 39503,C1(NC(CCOCC)=O)CCCC12CCN(C(=O)CN1CCCC1CO)CC2 39504,N1(C(=O)NC(N2CCCC2)CC)CCCCCC(S(C)(=O)=O)C1 39505,N1(S(C2C(C)CCc3sccc32)(=O)=O)CCC2C1CCCN2CC(=O)O 39506,c1(C(=O)NC(C(C)NC(c2cc(CC(C)C)on2)=O)C)cc2c(nn1)CCOC2 39507,c1(C2(C(=O)OC)CCC2)cc(NCC(O)CNC(C)=O)ncn1 39508,C1(N(CCNC(CCN(C)C=O)=O)C)CC2(C1)CC21CC1.N(S(N)(=O)=O)CC 39509,C1(NC(CCSC)=O)C2CN(C(=O)CCn3cccnc3=O)CC12 39510,C=CC(CCC)CC(=O)NCC1CCCC(NC(=O)Cn2nnnc2C(C)C)C1 39511,C(=O)(CC(F)(F)CC(=O)NCC1CCN(C(C2(C)CCCO2)=O)C1)OC 39512,C1(C(=O)NCC(C)N(C(=O)C(C2CCOC2)OC)C)(CC)CCOCC1 39513,C1(CCCNC(C2C(Cl)(Cl)C23CC3)=O)CCCCN1C(=O)Cn1nccn1 39514,N1(C(C(C)CC(N)=O)=O)CC2(CC(C(=O)NC(C)(C)C(C)(C)O)CO2)C1 39515,N1(C(C(CC(C)(C)C)NC(c2c(CC)nc(C)o2)=O)=O)CCN2CC(F)CC2C1 39516,Cc1cc(C(C)(C)C(=O)NC2CC(CCNC(c3cc[nH]c3C3CC3)=O)C2)cs1 39517,c1(C(=O)NC(C)CCCNC(C2(C)CC2Br)=O)ccc2ccnc(O)c2n1 39518,CCC(CC)C(C(=O)N1CC(OC)C(NC(=O)C(O)C2CCC2)C1)OC 39519,CCC(O)C(F)(F)C(=O)NCC1CCCCN1C(=O)C(CCC)NC(C)=O 39520,C1(CNC(C2OCC(C)C2)=O)(NC(=O)C=Cc2cncn2C)CCCCCC1 39521,n1(CC)ccc(C(=O)N(CC(CC)NC(c2c(C)n[nH]c2C)=O)C)c1C 39522,Cc1nc(O)nc(C)c1C(N1CCC(NC(=O)CN2C(=O)CCC2=O)C(F)C1)=O 39523,C1(SC)CN(C(=O)CCn2cc(Cl)cn2)CC1NC(C1CCNC1=O)=O 39524,C(C)(N=c1cc[nH]cc1S(=O)(=O)NCc1ccncc1)c1c(C)nccn1 39525,c1(NC(C2CCCC(NC(C(C=C)(F)F)=O)C2)=O)cccc(F)c1C 39526,C1(n2cc(CNC(C(C)=CC(C)(C)C)=O)nn2)CCN(C(C2CCCO2)=O)CC1 39527,c1(C(=O)NC(CN(C(c2c[nH]c3nccc-3c2)=O)CC)C)sc2cncn2c1C 39528,c1(C(=O)NCC2(NC(CCCOC)=O)CCCCC2C)cnc2c(c1)COCC2 39529,N1(C(=O)NCc2nnsc2CO)CCC(CO)C(O)CC1 39530,c1(CC(N2CCC(N(C(CCNC(N)=O)=O)CCO)CC2)=O)c(F)cncc1Cl 39531,N1(C(c2cc(OC)c(C)c(OC)c2)=O)CCC2CN(C(=O)C(C)(C)C)CCC2C1 39532,c1(NC(CNC(C2(CC#C)CC=CCC2)=O)C2CC2)ncn(C)c(=O)c1Br 39533,c1(SC)cccc(-c2cc(C3CC3)ccn2)c1.N1CCCCC1c1ccccc1F 39534,C1(Nc2nccc(OCC)n2)CCN(C(C2CCCC(C)C2)=O)C12CC2 39535,C1(CNC(Cc2n(C)cnc2)=O)CCCN(C(=O)Cc2ccn(C(F)F)n2)CC1 39536,C(CCCCC(=O)NCc1nc(C(=O)NCC2COC(C)(C)C2)co1)=CC 39537,C(=O)(CCCC(=O)N(C)C)NC1CC(NC(c2c(C(F)(F)F)cn(C)n2)=O)C1 39538,C1(C(=O)NCCC2CCCN(C(C3(C(N)=O)CC3)=O)CC2)OCCOC12CCC2 39539,c1(C(N(C2CCN(C(C34CCC3C4)=O)CC2)CC)=O)ccc(SC2CC2)cc1 39540,Cc1cc(C)n2ncc(CNC(=O)C(N3CC(C(F)(F)F)C(F)C3)=O)c2n1 39541,c1(CC2CCN(C(C=CC3C(CC(=O)OC)CCC3)=O)CC2)ccc(N)cc1F 39542,N(C1CC(C)(C)CCc2ccccc21)C(NNc1ccc(C)cc1)=O.C(CCO)O 39543,N1(C(C(CC)O)=O)CCN(C(=O)Cc2cncc(F)c2)C(CC(F)F)C1 39544,Cc1cc(C(=O)N(C)C)n[nH]1.n12cc(cn1)C(=O)NCC2 39545,CCCC(O)C(=O)N1CCCC1(C)CNC(c1onc(C)c1C)=O 39546,c1(C(N2CCCC(N(C(CC3N(C)CCC3)=O)C)CC2)=O)ccn2ccccc12 39547,N1(C(C(c2ccc(C)cc2)=O)=O)CC(NC(C2CC2C(C)C)=O)CC(C)(C)C1 39548,C(C(C)CC(=O)N1CCC(C)(CO)C1)NC(C(OCC)OCC)=O 39549,c1(C(N(C)C)=O)ccc2c(c1)CN(C(=O)C=Cc1cnccn1)C2 39550,Cn1c(I)cc2c(N(C(c3cnnc(Cl)c3)=O)CC3(O)CCCNC3)ncnc12 39551,N1(C(c2cnc(O)[nH]2)=O)CCCC12CCN(C(c1cccc(C3CC3)n1)=O)CC2 39552,C1(CC)CCN(C(=S)Nc2ccc(OC(F)(F)F)cc2)C1 39553,C12(C(=O)NCC3N(C(CCOc4ccc(C)cc4)=O)CC3)COC(CCO1)C2 39554,c1(CC(=O)NC2(CO)CCN(C(C=Cc3cn(C)nc3)=O)C2)cc(F)cc(Cl)c1 39555,CC1CC(CCNC(c2cnn(C)n2)=O)CCN1C(=O)CCNC(=O)CO 39556,C1(C(C)C)CCn2cc(nn2)C2(CNC2)NC1=O.c1(OC(C)=O)c(C)csc1C 39557,c1(OC)cc(C(=O)NC(C2CN(C(C3C4CC5C(C4)C35)=O)CCO2)C)ccn1 39558,N1(C(C(CC)O)=O)CC(C2CN(C(c3ccc(C)c(O)c3)=O)C2)C1 39559,C1(COC)(CNC(=O)CCF)CN(C(c2cnc(-c3ccccc3)[nH]2)=O)C1 39560,C(=O)(C(C)(O)CCc1ccccc1)NCCC(C)NC(CCCOC)=O 39561,c1(CC(=O)OCc2noc(CCC)c2CC)ccc(Br)cc1Cl 39562,C1(NC(CCC#C)=O)CC(CNC(=O)CCc2nc(-c3ccoc3)no2)C(O)C1 39563,N12CCC(F)(F)C(C1)CSCC2=O.c12ccc(Cl)cc1O2.N(CCOC)(CC)CC 39564,N1(C(CC2(NC(C(n3c(C)ncc3)C)=O)CCC2)=O)CCCC(CO)CC1 39565,C1(C(=O)NC2CCC(NC(C(CC)OCC)=O)CC2)CCC2CC2CC1 39566,c1(OC(C)C)ccc(C(=O)NCCCCN(C)C(C2CCC2C)=O)cc1 39567,C1(CNC(=O)C=C2CCC2)CCCCN(C(C2CN3CCCC2C3)=O)C1 39568,N1(C(C2C(C)(Br)C2)=O)Cc2ccccc2CC1CNC(C1CC(F)(F)C1)=O 39569,N1(C(C(C2CCN(C(C3(C4CC4)CC3)=O)C2)C)=O)CCC2CN(C)CC2C1 39570,c1(CC)ncc(Cl)c(C(=O)N(CC(C)CNC(C2(C)CCCN2)=O)C)n1 39571,Cc1nc2c(s1)CCCC2C(=O)NC1CCOCC1NC(=O)Cn1cncn1 39572,C1(NC(C2(C(C)(C)OC)CC2)=O)CC2CC1N(C(C1(C(F)F)CCCO1)=O)C2 39573,CC(C)(CCCCNC(C1CC=CC(O)C1)=O)NC(=O)CC1CC1C1CC1 39574,C(=O)(C(CCN(C)C)n1cccc1)NCCOCCNC(C(C)C1CC1)=O 39575,c1(C(N(C2CC(NC(=O)C(C)(Cl)Cl)C2)C)=O)ccc(N)c(F)c1F 39576,CC1(C(=O)NCC2CC(O)CN2C(C2COCCN2C=O)=O)CCCNC1=O 39577,N1(C(CCC(=O)NC)=O)CCC(C)C(CNC(C2CCC(=O)N2C)=O)C1 39578,C1(CNC(CCOC(C)C)=O)CN(C(C23CCC(C2)C3)=O)CCC1C(F)(F)F 39579,C1(O)(CN)CN(C(c2csc(C)n2)=O)C1.C(=O)(CC=CC(C)(C)C)N(C)C1CC1 39580,C(C1CN(C(=O)C(C)(C)C2CCOC2)CC1C(=O)NCC(C)CC(F)(F)F)=CC 39581,N1(C(Cc2cccc(C)c2)=O)CCC2CCC12CNC(=O)C=Cc1cncs1 39582,C1(NC(c2cccc(C)c2)C2CCCC2)COC2(c3ccccc3)CC1C2 39583,CC1CCCc2ncc(C(N3CCCC(C)(NC(c4cc(=O)cc[nH]4)=O)C3)=O)n21 39584,CCCCCCC(C(=O)NCC1CN(C(c2scnc2Cl)=O)CC1O)NC(C)=O 39585,c1(COC)cc(=NCCC2(NC(=O)CC3CC4CC4C3)COC2)[nH]cn1 39586,C(=O)(C(CC1CCC1)OC(C)C)NC1CC(CCNC(CCNC(C)=O)=O)C1 39587,N1(C(C=CC)=O)CCc2ccccc2C1CNC(C1CCc2ncncc2C1)=O 39588,C(=O)(C(CNC(C12CC(F)(C1)C2)=O)CC(C)C)Nc1c(COC)ncs1 39589,C1(NC(C2CCSCC2)=O)C2CCC(C2)C1C(=O)NC1CC2CC3C(C2)C13 39590,c1(OC)cc(C)ccc1CC(=O)OCCOOC(=O)CSCCC(F)(F)F 39591,CCC(C)(CCC(C)C)C(=O)N(CC(C)(C)NC(c1n[nH]c2c1CC1CC21)=O)C 39592,Cc1cn2cccc(C(N3CCSC4CCC34)C(=O)NCC3CC3)c2n1 39593,c1(C(=O)NCc2cccc(OC)c2OC)c(C)c(O)nc2ccccc12 39594,C1(C)(C(=O)OC)CN(C(C2CCC2)=O)C1.C12(CC1)C(=O)N2 39595,C(=O)(C(=O)CCC(C)C)N1CCCCC(C(N2CC(C)C=C(C)C2)=O)C1 39596,c1(C(N2CCC(O)(C(=O)Nc3c(OC)nccn3)C2)=O)cccc2c1CCC2 39597,N1(C(=O)CCCC2CCOCC2)CCC2(CCCN2C(=O)CCOC2CC2)C1 39598,c1(C(=O)NC(CC=C)CNC(C2CC(OC)C2)=O)cccc([N+](=O)[O-])c1Cl 39599,C1(C)(CCC)CCN1C(=O)CCCN(C(=O)C(CC)OC)C 39600,C1(C2(O)CN(C(=O)CCC(F)(F)F)C2)(CNC(c2ccn3c2CCCC3)=O)CC1 39601,Cc1nc(=NN2CCC(C#N)CC2)c(C#N)c[nH]1 39602,c1(C(C(=O)NC2CCN(C(c3nncs3)=O)CC2F)O)ccc2ccccc2c1 39603,c1(C(N2CCCC(N(C(=O)CCc3nc(O)n[nH]3)C)C2)=O)n[nH]cc1[N+](=O)[O-] 39604,c1(OC)nn(C)cc1NC(=O)CC1CCN1C(=O)OC(C)(C)C.C12CC(C1)N2 39605,c1(OCCC(N2CCC(NC(c3c(C)scn3)=O)C2)=O)ccc(Cl)cc1 39606,C(=O)(C(C)(C)C(C)NC(=O)CCC(C)OC)NC(CCC=C)(C)C 39607,c1(C(=O)NC23C(CN(C(C4C(C)C4)=O)C2)C3)nccc2ccccc12 39608,C1(N(C)C(C2CNC(=O)C2)=O)CCCN(C(c2ccnc(O)c2)=O)CC1 39609,C1(C(C)C(N2CCCCC2)=O)(CO)CCN(C(=O)C=CC2CCCC2)C1 39610,Cc1cc(Cl)ncc1NC(C1CC2CC2N1C(c1c(C(F)(F)F)coc1C)=O)=O 39611,C#CC1COCCN1C(c1ccc(OC(C)C)cc1)C(=O)NC(C)C(=O)OC 39612,CCCCCCC(F)C(=O)NC1CC2CCC(C1)N2C(c1ccc(Cl)o1)=O 39613,NC(=O)CCCC(=O)NCC1CC1CNC(C1NC(=O)CC1C(F)(F)F)=O 39614,CN1CC2CC2(NC(=O)C(Cn2cncn2)NC(C2CCC=CCC2)=O)C1 39615,C1(C(=O)NC2C(NC(Cc3cccc(C)c3)=O)COCC2)CC2CCC1CC2 39616,C=Cn1nccc1C(=O)NC(Cc1cn[nH]c1)C(=O)NCC1CC(F)(F)C1 39617,c1(OC)ccc(C2CC2CC(N2CCC(N(C)C(c3[nH]ccc3C)=O)C2)=O)cc1 39618,C1(C(=O)NC2C(CNC(c3coc(-c4ccccn4)n3)=O)COC2)CCCCO1 39619,C1(C(N2CCC(C(C(C)C)NC(=O)C(=O)Nc3nccs3)CC2)=O)C2CCN1CC2 39620,Cc1cccc(-n2nc(CCN(C)C)nc2-c2cnn3ccsc23)c1C 39621,C1(NC(C2(OC)CCCOC2)=O)CCCN(C(=O)C=Cc2ccn(C)c2)C1C 39622,c1(NC2CCN(CC)C2=O)nccc(=NC(C)Cc2cccc(OCCNC)c2)[nH]1 39623,C1(C(N2CC(O)(CCC)C2)=O)(NC(=O)C(C)N(C)C(C)=O)CCCC1C 39624,CC1(C)CCCC(NC(=O)CSCCNC(=O)CC2CC=CCC2)C1 39625,C(=O)(C(CN(C)C)C(C)C)N1CC(O)(C(CNC(C(C)C)=O)(C)C)C1 39626,c1(C(=O)NC2(CO)CN(C(=O)Nc3ccccc3O)C2)ccc(O)cc1.C1(=O)CN1 39627,N1(C(C2=CC(C)(C)C2)=O)CCC(C2CC2)(CNC(c2cnn(C3CCC3)n2)=O)C1 39628,N1(C(C2(CC#C)CCCO2)=O)C2CCC(C2)C1C(=O)NC1C(O)CC1O 39629,c1(-c2nc(Cc3scc(CF)n3)on2)cc(F)cc(F)c1 39630,Cc1cncc(CC(=O)N(C(C)CN(C(=O)CC2CCCC(=O)C2)C)C)c1 39631,C1(CC(=O)NCC(CNC(C(COCC)C)=O)F)CCCCC1(C)C 39632,c1(C(N2CCC(NC(C(C)=C3CCC3)=O)C(C)C2)=O)cc([N+](=O)[O-])c(C)cc1C 39633,C12(C(=O)NC(c3ccccc3)CNC(CN(C)C(N)=O)=O)CC(C)(C1)OC2(C)C 39634,N1(C(c2c(C(=O)OC)nccc2)=O)CC2CC1CCN2C(C1(F)CCCCC1)=O 39635,C1(NC(c2ccc(CNC(CC(C)F)=O)cc2)=O)CNC(=O)C1(C)C 39636,C1(F)(CNC(c2ccccn2)=O)COCCN(C(C2OCCCO2)=O)C1 39637,CCCC(C)(O)CC(=O)N1CC(NC(c2cnc(C(C)C)s2)=O)C(CC2CC2)C1 39638,c1(C(=O)NC(C)CNC(=O)C(F)(F)c2cnccn2)ccc(N)cn1 39639,c1(C(=O)NC2CC(CCn3cc(CC4CCC4)nn3)C2)cn2ncccc2n1 39640,CC(O)C(F)(F)C(=O)NCCC(C)(C)CNC(=O)CCOCc1ccncc1 39641,N1(CCNC(c2cc(CNC(c3coc(C(F)F)c3)=O)on2)=O)CCCOCC1 39642,C12(NC(c3c(CC)c[nH]c3)=O)CCN(C(C3(CC4CC4)CC3)=O)CC1C2 39643,C1(CC)CCCC1(C)C(=O)NC(C1CCN(C(=O)CSCCC(C)C)CC1)CO 39644,N1(C(Cc2cc(C(C)C)no2)=O)CCC(NC(=O)C(F)C(C)(C)O)C(CO)CC1 39645,C=CCC(F)(F)C(=O)NCC(O)C(=O)NC1CC2CCC(C1)O2 39646,C(=O)(C(F)CC(C)(C)NC(C1CC(=O)CC12CCC2)=O)NCC(=O)OCC=C 39647,C(=O)(C(F)CCC(C)C)N1CCC2C(C1)C(=O)NO2.C(C(C)CC(F)(F)F)OC 39648,c1(OC)c[nH]c(C)cc1=NC1CCc2ncc(OC(F)(F)C(F)(F)F)cc21 39649,c1(OC)ccc(CCNC(=O)Cc2cc(Cl)ccc2Cl)c(F)c1F 39650,CCC(CC(=O)N1CCC(CF)(NC(c2c[nH]nc2C)=O)C1)C(C)(C)C 39651,O=C(CCCCC(F)F)NCCC1CSCCN1C(=O)C(O)Cc1cnc[nH]1 39652,C1(NC(c2c(COC(C)=O)cccc2)=O)CCN(C(=O)CCc2ccc[nH]2)CC1F 39653,N1(C(C(CCF)NC(CC(C)n2cccn2)=O)=O)CCC12CCN(C)C2 39654,c1(COC)cc(Cl)nc(NC(=O)C(N2CCCC(OC)C2C(=O)OC)=O)n1 39655,C(CNC(=O)CC1(C)CCOC1)(CCNC(c1[nH]cnc1C)=O)OC 39656,C1(CNC(C=CCC)=O)CCC12CCN(C(=O)C=CS(F)(F)(F)(F)F)CC2 39657,N1(C(CNC(c2cc(C(=O)OCC)sc2)=O)C)CCN(C(=O)CC(C)CF)CC1 39658,C(c1cncc(O)c1)=CC(=O)NCC1N(C)CCN1C(=O)CCC(N)=O 39659,N#CC1CC2(CC(NC(C3CC(NC(=O)Cn4cccn4)CCO3)=O)C2)C1 39660,c12cc[nH]c1C(=O)NOC2.c1(C2CN(C(=O)CN3CC4CC4C3)C2)ccccc1 39661,CCCC(O)(CCC)CC(=O)N1CCN(c2cc(NCCOC)ncn2)CC1 39662,CC1CCN(C(=O)CNC(c2ccccn2)=O)CC1CNC(=O)Cc1n[nH]c(=N)s1 39663,C1(NC(C(C)NC(N)=O)=O)C2CC3C(C2)C13C(=O)N(CCC[Si](C)(C)C)C1CC1 39664,C1(C(=O)NCCC(C(C)C)NC(C2CNC(=O)CC2C)=O)CCc2nnnn2C1 39665,N1(CC)CCC(N(C(=O)C(C2CCOC2)NC(=O)C=CC(C)(C)C)C)C1 39666,CC1C(CO)NC(=O)NC2(CC(=O)N1)CC2.C1(CC(F)F)(C(=O)N(C)C)CCC1 39667,N1(C(C(C=C)(C)C)=O)CC2(C1)C(NC(=O)C1Cc3ccc(F)cc31)CCS2(=O)=O 39668,Cn1nc2c(c1C(N1CCN(C(C3(Cl)CC3(C)C)=O)CC1)=O)CCC2 39669,C1(N(CC(C(=O)NC)C)C)CCCN(C(c2ccc(CN3CCCCC3)s2)=O)C1 39670,C1(C(C)=O)CCCN(CCC(=O)N(Cc2ccccc2)Cc2ncn(C)n2)C1 39671,c1(CNC(C2CCC(C)O2)=O)ncc(C(=O)NCc2nn(C)c(=O)o2)cn1 39672,c1(OC)cnnc(C(=O)NC(C)CCCNC(=O)C(C)OCC2CC2)c1 39673,C(C1=CCN(C(C2CCC(N(C)C)C2)=O)CC1)NC(C(C=C)(C)C)=O 39674,C(CCCCC(=O)N1CCC(C(=O)NCC2CC2(Cl)Cl)C1(C)C)OC 39675,Cc1ncc(C=CC(=O)NC2(CNC(C3CC(C)(C(C)(C)C)C3)=O)CC2)s1 39676,c1(C(C(=O)NC2CC(NC(c3cn(CC=C)nn3)=O)C2)(C)OC)ccccc1F 39677,C1(CC(N)=O)CCCCC1C(=O)NCC1CCCC1NC(C1CC(CC2CC2)C1)=O 39678,Cc1[nH]c2ccccc2c1C(N1CCCCC(CNC(c2cnns2)=O)C1)=O 39679,C1(CNC(CC2CNC(=O)O2)=O)CC1C1CCN(C(=O)C2=CCCOC2)CC1 39680,N1(C(CNC(C)=O)=O)CCC(NC(c2cnn3c2C(C)CCC3)=O)CC(C)(C)C1 39681,C1(CNC(CCC(=O)OC)=O)COC(C)(C)CN1C(C1CC2CCC(C1)N2C)=O 39682,N1(C(c2cc3nnn(C)c3s2)=O)CCC2CCN(C(=O)CS(C)(=O)=O)CC12 39683,c1(C(N2CC(NC(C(C(C)C)O)=O)C(C)C2)=O)nc(C(F)(F)F)n2ccncc12 39684,N1(C(CC(C)C)=O)CCC2(CCCCN(C(C3CN4CCN3CC4C)=O)C2)C1 39685,c1(NC2CC(CNC(C3CCCCC3O)=O)C2)ncnc(Cl)c1F 39686,C12(CNC(c3cc4sccc4[nH]3)=O)CN(C(C3CCCS3)=O)CC1(C(F)(F)F)C2 39687,C1(C(=O)NC2CCN(C(C)=O)C2)CN(C(=O)CC2CCSC2)CC1N(C)C 39688,c1(OC)cnccc1C(=O)NCCC1CCCCN1C(c1cc(C(C)=O)c[nH]1)=O 39689,c1(C(=O)NCCNC(CCCC2CCC(C)C2(C)C)=O)c2ccccc2nn1C 39690,C#Cc1cc(F)c(C(N2CC3CC3(NC(C3COC3)=O)C2)=O)cc1F 39691,O=C1COc2cc(C(N3C4CCC3CN(C(C35CCCC3C5)=O)C4)=O)ncc2N1 39692,N1(C(CC2C=CC(NC(C(C=C)(C)O)=O)C2)=O)CCC2(CCC2)C(O)C1 39693,C1(C(=O)NCC23CC(NC(c4ccn(C)n4)=O)(C2)C3)CCC(F)CC1 39694,c1(C(=O)NCC(CCC)C(=O)N(CCC(F)(F)F)C)ncn2ccccc12 39695,CC(C)CCCC(C)C(=O)N1CCC(CCNC(c2cc3occc3[nH]2)=O)C1 39696,C1(CNC(c2c(C)occ2C(F)(F)F)=O)CC(F)(F)CN1C(c1cc(Br)c[nH]1)=O 39697,Cc1nc(C2CCCCC2)sc1C(=O)NCC#CCNC(=O)CC#N 39698,c1(C(N(c2ccn(C)n2)CC)=O)occc1CNC(C1CCO1)=O 39699,C1(C)(NC(C(c2cccc(I)c2)C)=O)CCN(C(=O)CNC(=O)C(C)(C)C)C1 39700,C1(NC(C2C(NC(Cc3c(C)cnn3C)=O)COC2)=O)Cc2cscc2C1 39701,C1(N(CC(C)C)C(=O)COC2CCCC2)CCN(C(C2CC(F)C2)=O)C1 39702,C(c1cc(C)ccc1OC)=CC(=O)N(CCCCNC(CC(COC)C)=O)C 39703,N1(C(C#CC(C)C)=O)CCCCC(CCC(N2CCOCC2CCO)=O)C1 39704,Cc1ccc(C(N2CCCC2C(C)(C)CNC(C2OCC2(C)C)=O)=O)n1C 39705,c12ccccc1N2.c1(C(C)C)ccccc1C1CCCNC1 39706,c1(C(=O)OC)ccn(CCNC(=O)NCC2CC(O)CN2C)c1C 39707,C(C)(CCCCNC(=O)CCc1nnc(C2CCCC2)o1)NC(C1C(C)C1C)=O 39708,Brc1c(N2CCC3(C=CCO3)C2)nc2nc[nH]n12 39709,N1(c2ncc(C)c(O)n2)CCC(C)C(NC(=O)C=Cc2cc[nH]n2)C1C 39710,C1(O)(CNC(CCC)=O)CCCN(C(=O)CC(O)C(C)C)C1 39711,c1(SC)cncc(NC(=O)NC(C2(C)CC2(F)F)C2CC2)c1 39712,CCCCCS(=O)(=O)CC(=O)NCC1(OC)CN(C(C2OCCC2C)=O)C1 39713,c1(CCC)c(C(N2CCCC(CCc3ccccc3Cl)C2)=O)nnn1CC 39714,c1(NCC2C3CN(C(CN4CCC(C)CC4)=O)CC32)nc(Cl)ncc1[N+](=O)[O-] 39715,c1(CCNC(C2N(C(C(C)(C)C)=O)CCC(O)C2)=O)ccc(S(=O)(=O)F)cc1 39716,C(C1=CCN(C)CC1)NC(C1C(CC)CN(C(=O)CC2CC2CC)C1)=O 39717,N1(C(c2cnc(CCC)s2)=O)CCC(C)C(CNC(=O)C#CC(C)(C)C)C1 39718,N1(C(C)=O)CC(O)CC1C(=O)N(CC(F)F)Cc1ccccn1 39719,c1(C(=O)NC2CCCC(OC)C2)ccc(P(C)(C)=O)s1 39720,c1(C(=O)OC)ccc2c(c1)OCCN(C(c1cc(Br)c(F)cc1OC)=O)C2 39721,n1(C(C(=O)N(CCNC(=O)CN(CC(C)(C)C)C)CC)C)ccc(C)n1 39722,c1(OCC=C)ccccc1C(=O)NCC1CCCN1Cc1cccnc1OC 39723,C(=O)(C1=C(C#N)CCC1)NCC1CC(C)(C)CN1C(=O)COC(F)F 39724,C1(C(=O)NC2C(n3cc(CCC(C)O)nn3)CCC2)CCc2nncn2CC1 39725,Cc1ccncc1CC(=O)N(CCCNC(=O)CC1CSCCO1)CC1CCCC1 39726,C1(C(=O)NCC(C=C)O)CC12CC(NC(c1c[nH]nc1C(F)F)=O)C2 39727,CC(C)CC(C(=O)NC1CC2C1CCN2C(C1CN2CCC1CC2)=O)C(N)=O 39728,c1(OC)cccc(NC(=O)NCC2(CSc3cc(Cl)ccn3)CC2)c1 39729,C1(CN(C(CSc2n(C)ccn2)=O)C(C)=O)CCCCN1CC(c1cnsn1)=O 39730,N1(C(C2CCC(=O)O2)=O)C2CCC1(CNC(c1cn(CCO)nn1)=O)CC2 39731,c1(OC)nn(C)cc1Cl.C1(=O)CCCn2cc(nn2)C2CN1C2 39732,N1(C(c2cccc(Cl)c2)C(C2CCCCC2)OC)CCC2(CSC2)C1 39733,Cc1ccc(F)c(O)c1C(=O)NC1CCCCN(C(=O)CCc2cscn2)C1 39734,N1(C(CC=CC)=O)CCC(C)(C)C(CNC(=O)C(C(C)CC)N(C)C)C1 39735,C1(NC(CC(C)=C(C)C)=O)CCCC(NC(c2c[nH]nc2Cl)=O)C1 39736,C1(CCCNC(C2(C)CC2C(F)(F)F)=O)CCCN1C(=O)CC1CCOC1=O 39737,Cc1cc(C(=O)NCC(C)CCCO)ccc1[N+](=O)[O-] 39738,c1(NC(C(C)N(C(c2cscn2)CO)C(N)=O)=O)cccc(F)c1 39739,C1(CNCc2ccccc2)CCCCCC(=O)N1.CC1(C)CC=CC(=O)NOC1 39740,C1(CC(N2CC(CC=C)(NC(CCCC#C)=O)C2)=O)NC(=O)CN(C)C1=O 39741,C1(CC(=O)NCC(O)(CO)SC)CC2CCC1O2.C(CC(=O)C1CC1)NC(C)=O.C1C(=O)N1 39742,C(CCCCC(=O)N1CCOC(CNC(C2CC2C(C)(C)C)=O)C1)NC(C)=O 39743,C(=O)(C(C)(C)CCC#N)NCC(CC(C)C)NC(C1OCCN(C)C1=O)=O 39744,C(C)(CCCC(=O)N1CCOCC1C1CC1)NC(COCCCC(C)C)=O 39745,Cc1cc(CN2CC(CN(C(=O)C(c3cnn(C)c3)O)CCl)CC2=O)c(O)c(Br)c1 39746,c1(C(=O)NC(CCN(C(C(C)OCC=C)=O)C)(C)C)cc(Cl)c(Cl)cc1O 39747,C=CCCCCCC(=O)NC(C(=O)NC1CC(C)(C)OC1(C)C)C1CC1 39748,Cc1ccc2n[nH]cc2c1C(N1CCNCC1c1ccc(Br)cc1)=O 39749,N1(C(=O)C=C2CCC2)CCCC2(C1)CN(C(=O)C1=CCCCCC1)CCO2 39750,N1(C(C(CC=C)NC(C)=O)=O)CCC(C(=O)NCc2nccs2)C1(C)C 39751,C1(F)(C(=O)NCCC2(CNC(C(C)C3CCOC3)=O)CC2)C(C)(C)C1(C)C 39752,CC1CCCC(OCC(=O)NC2CC(c3ccccc3)(NC(=O)COCF)C2)C1 39753,c1(C(=O)NCC(C)(O)C(=O)O)cc2cc(F)ccc2cn1 39754,C12(C(=O)NCCN(CCCC)C)CCC(CC1NC(c1cncc(O)c1)=O)C2 39755,CC1OC(C)C(C(=O)N(C)CC2CN(C(C3(C(F)(F)F)CCCC3)=O)C2)C1C 39756,Cc1cc(N(C2CCN(C(=O)C(C3(O)CCOCC3)(F)F)C2)C)c(C#N)cn1 39757,C(=O)(C(F)CC(C)(C)C)N1C(CC(=O)NC(C(=O)OC)C2CCC2)CCC1 39758,c1(C(N2CCC(CN(C(CCc3c(C)noc3)=O)C)C2)=O)cc(Cl)nn1C 39759,C(=O)(C1=NOC(C)C1)N1CCC(C)(CCNC(c2c(CCC)nns2)=O)C1 39760,c1(OC)c(-c2nc(C3CCOC3)nn2CCC(C)C)ccc([N+](=O)[O-])c1O 39761,N1(C(c2c(OC)cncn2)=O)CCC(C=CC(=O)NCCC(O)C(F)(F)F)CC1 39762,Cc1cc(C2CC2)ncc1C(=O)NC(C1CN(C(c2ccncc2Cl)=O)C1)C 39763,c1(CN2CC3C(C(N4C(CC(=O)OC)CCC4)=O)(C3)C2)cncc(Cl)c1Cl 39764,O=C(NN1CCCC1C(=O)NC1(c2nc[nH]n2)CC1)C1CC(=O)C1 39765,N1(C(=O)OC(C)(C)C)CCCCC1C(=O)N(O)Cc1cn(-c2ccncc2F)nn1 39766,c1(CC(N2CCC(NC(C3N(CC)CC3)=O)C2)=O)cc(C2CC2)nn1C 39767,C#CC(Cn1cccn1)NC(=O)CC1CC(N)C1 39768,c1(CC)cc(C(F)(F)F)nc(N(C)CCN(C(=O)C(F)=CC2CC2)C)n1 39769,C1(CC(=O)NCCCNC(C(C)c2ccon2)=O)CSc2ccccc2O1 39770,N12CC(C(C)C1)C2=O.c1(CNC(C2N(C(CCC)=O)CCC2)=O)cc(O)nn1C 39771,C(=O)(C(F)(F)C(F)F)NCC1(NC(C(C(C)C)F)=O)CCCCC1 39772,c1(NC(=O)NC(C(c2cc(C)c(F)cc2)O)C)cc(Br)cc(F)c1F 39773,CN1CCN(C(C2CCOC(C)(C)C2)=O)C(C(=O)NCCc2ccc(O)nc2)C1 39774,c1(-c2cc(C)c(Cl)cc2)cc(NC(=O)C(C)S)cc2[nH]ccc12 39775,C1CCC(=O)NCC2CC(CO2)CNC1=O.C1(C)CCCC1.CS 39776,c1(CCC)cc(-c2ccccc2C(=O)N(c2cccc(C)c2C)C)ccc1O 39777,c1(OC)cc(C=CC(=O)NC2CC(NC(=O)C(O)C3CCC3)C2)ccc1O 39778,C=C=CCCC(=O)NCC(=O)NC1CCCC1.c12noc-1n2 39779,c1(CC)[nH]nc(C(=O)NC2(C(=O)N(CCCN=[N+]=[N-])C)CCCC2C)c1C 39780,N1(C(CC2C(C)(C)CCN2C(=O)Cn2c(O)nnc2O)=O)CCC2(C=CCO2)C1 39781,c1(C(C(=O)NC(C)Cc2ccccc2Br)N)c(F)cccc1F 39782,c1(CCC(=O)NC(CCCNC(c2c(C)n[nH]c2C)=O)C)ccc(Cl)cc1Cl 39783,n1(CC(=O)NC2(C3CN(C(C4(C)CC=CCC4)=O)C3)CC2)ncc2ccccc12 39784,C1(C(=O)NC2CON(CC)C2=O)CN(C(C2C3CC(=O)CC23)=O)CC1(C)C 39785,N1(C(c2cc(C)n(CCO)n2)=O)CC(CNC(c2n[nH]cc2Cl)=O)OC(C)(C)C1 39786,NS(=O)(=O)C1(C(=O)NCC2CC3CCC2N3C(=O)C2=CCCO2)CCCC1 39787,c1(OC)cc2oc(=O)n(-c3ccccc3F)c2cc1CC(N1CC=C(Br)CC1)=O 39788,Cc1cccc(C(=O)NCC2CCCC2NC(c2c(F)cccc2F)=O)c1C 39789,c1(NC(c2cc(CNC(C3C(C(=O)OC)C3)=O)ncc2)=O)cnc(Br)c(I)c1 39790,C(=O)(C(C)(C)CS(C)(=O)=O)N(CCC1N(C(C(COC)COC)=O)CCCC1)C 39791,n1(CC(=O)OC)cc(CNC(=O)NC2(c3cccnc3)CCC2)nn1 39792,Cc1ccn2c(C(=O)NCC(C)(C)CNC(=O)C(C)OCCN(C)C)cnc2c1 39793,c1(C(=O)NCC2(F)CC(NC(c3nn(CC)nc3C)=O)C2)cccc(F)c1OC 39794,c1(NCc2ccc(OCC(=O)NCC)c(OC)c2)cc2c(s1)CCOC2 39795,C1(C(=O)NCc2cn(CC=C)nn2)C=CCCN1C(=O)CCCCOC 39796,C1(NC(C2(C#C)CCCC2)=O)CC2CC1N(C(=O)C(CC)=CC)C2 39797,C(CN=C(NCCF)NCc1cc(C2CCC2)on1)NC(=O)OC(C)(C)C 39798,C1(c2n(C)cnc2)CN(C(=O)CC2(C#N)CC2)CC1CNC(=O)C=CBr 39799,Cc1nc(CO)ncc1C(N1CCC(NC(C2CN(C(C)C)C2)=O)C12CC2)=O 39800,Cc1cc(NC(=O)Nc2c[nH]nc2C2CC2)n2ncnc2n1 39801,N1(C(C2N(C(C(C=C)CC)=O)CC3(CC3)C2)=O)CC2(CC(CO)CO2)C1 39802,N#Cc1ccc(CNc2ccnc(C(N3CCC(CO)C(O)C3)=O)c2)c(O)c1 39803,C1(C(=O)NC2(C(=O)NC3CC(N(C)C)C3)CCCCC2)CCCCC(=O)C1 39804,c1(C(=O)NCC=CCNC(C2C(C)C2)=O)ccc(N2CCC(C)CC2)nc1 39805,c1(C(N2CC(C(=O)C(CCCNC(c3cnns3)=O)=O)C2)=O)ccncc1C1CC1 39806,Cc1cccc(C)c1C(O)C(=O)NC1CCC(NC(C2CCC(C)S2)=O)CC1 39807,C(N=c1nc(COC)cc(C)[nH]1)c1ccc(CNC(C2N(CC)CC2)=O)c(F)c1 39808,N1(C(C(C2CC2)OC)=O)CC(NC(c2cc(Cl)c(F)cc2F)=O)C(N=[N+]=[N-])C1 39809,N1(C(=O)NCc2c(CC)cncc2)CCCCCC1Nc1ccnc(F)c1 39810,c1(C(=O)NCC2(NC(C3CCN(C)CC3)=O)CCOCC2)cc(F)ccc1N 39811,N1(C(c2[nH]cc(CC)c2)=O)CCC(N(C(c2ccc(CN(C)C)s2)=O)CC)CC1 39812,C(=O)(CCC(C)(C)O)NC(C1CN(C(=O)C2=CCCCC2)C1)C 39813,c1(C(=O)NCCCNC(C2(C(=O)OCC)CC2)=O)ccc(F)cc1NC(C)=O 39814,N1(C(CCCc2n[nH]c(=N)s2)=O)CCN(C(c2cc3c[nH]nc3s2)=O)C2CC12 39815,C(=O)(C(=O)CC(C)CC)N(C(C)C(=O)NCC1CCCCCCC1)CCC 39816,c1(CSc2nnc(-c3nnsc3C3CCC(CC)CC3)o2)cc2c[nH]cnc-2n1 39817,n1(CC)c(=O)c(C)nc2cc(C(=O)NC3CC3NC(=O)C=C3CCCC3)ccc12 39818,Cc1cc(CC(=O)N(C(C)C(=O)NC(C2(O)CCCCC2)C)C)c(C)s1 39819,CC1(C)CCC2(CN(C(c3cn(CC(F)(F)F)nn3)=O)C2)O1 39820,C(=O)(C1OCCc2ccccc21)NC1(CC=C)CN(C(=O)C(C)(F)C(F)(F)F)C1 39821,S(=O)(=O)(c1[nH]c(=NC(C)Cn2ccnn2)ccc1Br)N(C)Cc1c(C)cccc1 39822,c1(C(N2C(CNC(C(C)(C)Br)=O)CCC2)=O)cccc2cc[nH]c12 39823,CCC(C)(C#N)C(=O)N1CCCC(O)(CCNC(c2ccc(F)s2)=O)C1 39824,C(=O)(C(C(C)C)C1CCC1)NC1(CCC)CN(C(c2ccccc2C(N)=O)=O)C1 39825,c1(C(C)=O)cc(C(N2CCCC2CCNC(=O)Cc2cccnc2F)=O)c(C)o1 39826,C1(C2CCOCC2)(C(N2CCN(CC(C)NC(CCSC)=O)CC2)=O)CC1 39827,C1(NC(C=CC=CC)=O)CC(O)CN(C(=O)C(C)(C)CC#N)C1 39828,C1(C(N(CCNC(C(C)NS(CC)(=O)=O)=O)CC2CC2)=O)CCCSC1 39829,C(=O)(CC(C(=C)C)OCC)N1C(CN(C(CCNC(=O)NC)=O)C)CC(F)C1 39830,c1(C(=O)NC(C2CCN(C(C(CC)OCC)=O)C2)(C)C)cc2n(n1)CCCN2 39831,C1(NC(C2N(C(C)=O)CCC2)=O)CC2(C1)CN(C(=O)CC1C(=O)N(C)N=C1C)C2 39832,C(=O)(C(F)C(=O)NC(C)CNC(c1cc(=O)n(-c2ccccc2)[nH]1)=O)OCC 39833,Cc1ccc(CCNC(C2(CNC(C3(c4cc[nH]n4)CC3)=O)CCC2)=O)cn1 39834,N1(C(c2cccc(OC)n2)=O)CCC2(CNC(c3cnc(S)n3C)=O)CCCC12 39835,C1(C(N(CCNC(C2CCCC(C)(C)C2)=O)CC)=O)CC12CCCCCC2 39836,C(=O)(CCCCC(F)F)NCC1N(C(c2ccc(N)cc2F)=O)C2C(C1)C2 39837,n1(CC)cc(Br)cc1C(=O)NCCOCCNC(C1(CF)CC(F)(F)C1)=O 39838,C1(CNC(c2cscc2F)=O)CCCCC1NC(C1CCC(O)C1)=O 39839,C=C=CCCNC(=O)C(C)NC(=O)C(C)c1cccs1 39840,Cc1cc(CCNC(=O)Cc2cnc(NS(=O)(=O)CC#N)s2)c(O)c(Br)c1 39841,c1(C(=O)NCCOCC(=C)C)cccnc1CNC(=O)CN1CCCCCC1 39842,c1(NC(CC(=O)NC2C(CSC)CCCC2)=O)ccc2nc(N(C)C)sc2c1 39843,C1(N(C(Cc2c(C)scc2)=O)C)CCCC(NC(=O)C=CBr)C1 39844,c1(C(=O)NC(CC=C)CNC(c2cn(C)nc2C)=O)cc(N)c(F)c(O)c1F 39845,C(=O)(CC(F)(F)F)N(CC(C(=O)NCCC(=O)OC(C)C)C)C 39846,CC1=C(C(=O)NC(C2CCCN2C(C2OCCCO2)=O)C)CCO1 39847,C1(Cn2c(C)ncc2)CCCN(CC23CNCC2C3)CC1 39848,N1(C(CC(=O)OC)=O)CCOC2CN(C(c3n[nH]c4cc(C)ccc34)=O)CC12 39849,c1(C(N2C(C)CCC(CNC(C(CC)N(C)C)=O)C2)=O)cccc2ccsc12 39850,N1(C(Cc2ccc(NC(c3ccccc3Cl)=O)cc2Cl)=O)CCc2[nH]ccc2C1 39851,C(=O)(C(C(C)CCC=C(C)C)N1CC2CC(N(C)C)C2C1)NCC=C 39852,c1(OC)ncc(C(N2CC(N(C(=O)CNC=O)CC3CC3)C(O)C2)=O)cc1F 39853,c1(N2C(C)CC(NC(c3cc(O)cc(C#N)c3)=O)CC2)nc2ccccc2s1 39854,N1(C(c2c(C)nc(C)[nH]2)=O)CCN2CCOCC2(CNC(=O)CC(C)F)C1 39855,c1(C(=O)NCC(CC)(CC)NC(=O)C(F)CC(C)C)snc2ccccc12 39856,C1(CC)CN(C)CCN1c1cc(CC)ncn1.C1(N2CC2=O)CCCC(C#N)C1 39857,c1(CC)cccc(F)c1C(N1CC2(C1)CN(C(=O)C(F)CC1CC1)C2)=O 39858,Cn1cnc2[nH]c(C(N3CCN(C(=O)CC4=CCCC4)C4CC34)=O)cc12 39859,N1(C(C2(C)C=CCCC2)=O)CC2CC1CC2CNC(=O)CCc1ccc(Cl)nc1 39860,N1(c2cc(C)ncn2)CCCC12CCN(C(c1cccc3c1ncn3C)=O)C2 39861,C1(C(N2CC(c3n(C)ccn3)C(NC(=O)C3=CCC3)C2)=O)Cc2cscc2C1 39862,N1(C(C=CC(=O)OCC)=O)Cc2ccccc2CC1CNC(=O)Cc1csnn1 39863,C(c1ccccc1F)=CC(=O)NC(C)CC(C)NC(=O)C1=C(Cl)CC1 39864,C1(C(N(CCN(C(=O)CC2CC=CCC2)C)C)=O)CCN(CC(F)(F)F)C1 39865,CC1CCC(=CC(=O)NC(C)CNC(=O)C(C)N2CC(C)C2)CC1 39866,C1(C(N2CCOC(CCNC(c3cccc(Cl)c3)=O)C2)=O)(CSC)CCOCC1 39867,N1(C(c2nc(CC(C)C)sc2)=O)CC2(C1)CN(C(=O)CC1(C)CC1(F)Cl)C2 39868,C1(C(N(CCCN(C)C(C2(C(F)F)CCCCC2)=O)C)=O)CCC2(CCC2)OC1 39869,CCC(C)C(O)C(C)C(=O)NCCn1cc(C(=O)NCC2(SC)CCC2)nn1 39870,C1(NC(c2ncn(C(C)C)c2)=O)CN(C(C2(O)CCOC2)=O)CC1C 39871,N1(C(C(F)=CCC)=O)CC(NC(=O)Cc2c(C)ncn2C)CC12CCCCC2 39872,CC(CCC(=O)N(CC(C)(C)NC(c1cncc(N(C)C)c1)=O)C)c1ccc[nH]1 39873,c1(OC)c(C(=O)NC2(C)CN(C(c3c(N)cccc3Cl)=O)C2)oc2ccccc12 39874,C1(CC)C(C(=O)NCc2ccc(C)cc2)CCN1C(=O)C(C)O 39875,N1(C(CCC(=O)NC)=O)CCC(C2CC2)C1CNC(c1cnc(C)c(OC)c1)=O 39876,c1(OC)ccc(C#N)cc1Cc1noc(-c2nc(OCC)ccc2Cl)n1 39877,N1(C(c2cccc(CNC(CCCCC#C)=O)n2)=O)CCC2C(CCN2C)C1 39878,c1(C(=O)NCCC2(NC(c3cncc(N(C)C)c3)=O)CC2)nc[nH]c2nccc1-2 39879,c1(C(=O)NC(C)C(c2ccncc2)O)ccnc(C(F)(F)F)c1F 39880,C(=O)(C1CCc2cccc(F)c21)N1CC(COC)OC(C)C1 39881,C(CC1=CCOCC1)NC(C(CC)N(C)C(c1cn(C)c(=O)n1C)=O)=O 39882,C1(NC(C(CC)C)=O)CCC12CCN(C(c1cc(Cl)c(F)cc1N)=O)CC2 39883,N1(C(Cc2nc(C)sc2C)=O)CCCN(C(=O)CCc2cscn2)C(CO)C1 39884,N(C(=NCCC)NC1CC(CC)C1)C(C#C)CC 39885,C1(CNC(=O)NCC(C(C)C)(F)F)CCC2(CCOCC2)C1 39886,Cc1ccc(C(=O)NCC(C(C)(C)C)NC(C2CCOC2)=O)c(C)c1 39887,N1(C(Cc2scc(C)c2)=O)CC(C)CN(C(=O)C(N2CCCCC2)C)C(C)C1 39888,C(C)(C)(CC(=O)NCCc1nc[nH]n1)N(C(=O)CCc1cn(C)nn1)C 39889,c1(C(N2CCC(CNC(C3(C)CCC(=O)NC3)=O)C2)=O)cc2cc(Cl)ccc2o1 39890,C(=O)(CC(C)C(C)(C)NC(c1cnc(N(C)C)o1)=O)N1CCC(C)(CCC)C1 39891,c1(CC(=O)NC(CCNC(C2(OC)CC2)=O)C)csc2ccccc12 39892,c1(C(=O)NCC2CCN(C(c3csc(C)c3N)=O)CC2)ccn2nnnc2c1 39893,c1(C(=O)NC2CCN(C(C(COC)(C)OC)=O)CC2CO)cn2cnnc2cn1 39894,C1(NC(c2cnn(C(C)C)c2F)=O)CCN(C(=O)C(C)Cc2cnc[nH]2)C1(C)C 39895,CCC(C(=O)NCC(C)(CO)NC(=O)C(=O)N(C)C)C(C)(C)CC 39896,C(=O)(CCC(C)(F)F)NCCN(CCC)C(c1c(Cl)cncc1Br)=O 39897,CC1Cc2ccccc2N1C(=O)NCC1C(c2ccccc2)C1(F)F 39898,CC(C)(CC(=O)NCC1(NC(C2CCCC3CCCN23)=O)CC1)C(F)F 39899,C1(C#N)(C(=O)NCC2CCC(NC(c3scc(C)c3Cl)=O)CC2)CC12CCCC2 39900,C1(C(N2CCC(OCC(N)=O)C2)=O)CCC(C)(C)N(C(C2CC2(Cl)Cl)=O)C1 39901,c1(CC(=O)N(C)CC2CCCN2C(C23CC(F)C2C3)=O)cc(Cl)sc1Cl 39902,CC(Cl)(Cl)C(=O)N1CCC(CCNC(C2CCC(C(=O)OC)O2)=O)C1 39903,N1(C(c2cnc(C3(CC)OCCO3)s2)=O)CCN(C(=O)C(N)=O)CC1C1CC1 39904,C1(OC)(CNC(c2c[nH]cc2C2CC2)=O)CCN(C(C2C3CN(C)CC23)=O)C1 39905,C#CCCC(C(=O)NCC(c1ccco1)O)NC(=O)C=C1CCC(C)CC1 39906,c1(C(=O)NCc2c(C(=O)NC(C3CCC3)CO)scc2)cn2ccccc2n1 39907,c1(OC)ccc(C#N)cc1NC1CC(C(C(=O)OC(C)(C)C)F)C1 39908,C(=O)(C(F)C(F)(F)F)NCCSCC(N1CC(OCC#C)C1)=O 39909,C1(C(=O)NCCC2(CNC(c3ccc(C#N)o3)=O)CC2)C2(CCC2)C12CCC2 39910,N1(C(C(C(COC)C)C)=O)CCCC2(NC(C3CCCCC3C)=O)CCCC12 39911,O=C(C1=C(Cl)CCCC1)NC1CC(NC(c2cc(C(F)(F)F)nn2C2CC2)=O)C1 39912,c1(-n2cc(C(C=C)(C)O)nn2)ccccc1C(=O)NC1CCOCC1OCC 39913,N1(C(C(C)NS(C)(=O)=O)=O)CCC(F)(CNC(=O)CN(C)C(=O)C2CC2)C1 39914,N1(C(C2=CCCCC2C)=O)CC2(C1)CN(C(C1(CCN(C)C)CCC1)=O)CCO2 39915,C(=O)(C1CCCc2ncnn21)NC1CCCN(Cc2cccc(OC)c2)C1 39916,C12(CNC(C(N3CCOCC3)C)=O)CCCCC1CN(C(=O)C(C)(C)CO)C2 39917,C(=O)(C(C)S(N)(=O)=O)N(CCNC(c1c(C)onc1)=O)CC1CC1 39918,C1(C#CC(=O)NCCN(C(=O)C(C)N(C)C(C)=O)C2CC2)(CC)CC1 39919,C(CC)(C(=O)NC1CCC1C(=O)N(C(C)CC1CC1)C)=CCCC 39920,O=C(CC1=CCCCC1)N1CCC2(CC2C(N2CCCC2CCO)=O)C1 39921,Cc1nc(C(=O)NCC23CC2CN(C(c2ccc(-c4cc[nH]n4)s2)=O)C3)sc1C 39922,N1(C(c2ccc(C)s2)=O)CC2CCCCC2(NC(c2occ(C)c2C)=O)C1 39923,C1(O)(CNC(c2cc(C3CC3)no2)=O)CCCN(C(C2SCCS2)=O)CC1 39924,C1(=O)C(F)(C(C)C)CN1CC(C)(C)C.C1(C(C(=O)OC)F)CCCCC1 39925,N1(C(C2CC(C)OCC2)=O)CC2CN(C(c3ccc4nccn4c3)=O)CC(C1)O2 39926,N1(C(Cc2nc(COC)sc2)=O)CC2CC1CN2C(c1sccc1F)=O 39927,C1(C(=O)Nc2cn(CC)nc2)CC12CCN(C(=O)COC(C)=O)CC2 39928,C1(C(=O)NC2(CNC(CC(CCC)O)=O)CC2)Cc2ccccc2N1 39929,N1(C(C(n2cc(Cl)cn2)C)=O)CC2CN(C(=O)CCC3CCCCC3)C2C1 39930,Cc1ccnc(O)c1C(=O)NCCC1(CNC(C2(C(N)=O)CC2)=O)CC1 39931,c1(OCC)ccc(CCC(=O)NC(C2CCN(C(=O)C3CC3)CC2)C)cc1.CS 39932,CC1CCCN(Cc2ncccc2CNC(C2CN(C(C)C(=O)N(C)C)C2)=O)C1 39933,C12(C(N(CCC(C(C)C)NC(=O)CCCCCO)C)=O)CC3CC(CC(C3)O1)C2 39934,c1(C(N(CC(C)NC(CCN(CCC)C)=O)C)=O)noc2c1CCCCC2 39935,C1(C)(C(N2CC(O)(CN(C(=O)CNC(c3cscn3)=O)C)C2)=O)C=CCCC1 39936,C(=O)(CCCNC(C1CCC1)=O)NC(CN(C(C1(C#C)CC1)=O)C)(C)C 39937,c1(C(N2CC(C3CN(C(C(C)(C)CF)=O)C3)C2)=O)cc2ccsc2c(O)n1 39938,C1(NC(CCCC=C)=O)CCCC12CN(C(C1CCN(C)C(=O)C1)=O)C2 39939,C1(C)(CNC(c2c(C)cno2)=O)CCCN1C(=O)CN(C(=O)C(C)C)C 39940,Cc1ccc(C(=O)O)c2c1N(C(c1cncc(OC(C)C)c1)=O)CC(C)C2 39941,C(C)(CN=c1nc(C2CC2)[nH]cc1OC)N(C(c1ncc(OCC)nc1)=O)C 39942,C1(CC(=O)NCCc2ccc(CO)cc2)CCC2(CCC2)O1.CC(O)C(=O)NC 39943,C1(n2cc(C(C=C)(C)O)nn2)CC2CCC(C1)N2C(c1cc(F)cc(Br)c1F)=O 39944,N1(C(CCCCCOC)=O)CC(C)N(C(c2ccc(C(F)(F)F)cn2)=O)CC1C 39945,C(C(O)C(=O)N1CC(O)(C2CCCN2C(=O)CCc2nc(=N)[nH][nH]2)C1)SC 39946,N(C1CCCc2c(F)cc(F)cc21)C(=O)C(C1CCCCO1)F 39947,N1(C(C(C)NC(CC)=O)=O)CC(CO)C2(C1)CN(C(=O)CC(C)(C)CCOC)C2 39948,N1(C(C2C(CC)OCC2)=O)CC(N(C)C(c2cc(C)c(C)[nH]2)=O)C(C)(C)C1 39949,N1(C(C(C2CCC2)OC)=O)CCC2CN(C(=O)Cc3cc[nH]n3)C(C)C12 39950,N1(C(CC(=C)Br)=O)CCC2(CCCN(C(=O)CCOC3CCCC3)C2)CC1 39951,C1(CC(=O)OC)CC(Nc2cn(CC)nn2)CCO1.c1(C=O)ccccc1 39952,Cc1c(-c2cscc2C(=O)Nc2nc3sccc3s2)cc(Br)cc1F 39953,S(=O)(=O)(c1ccc(NC2CC2C2CC2C(=O)O)c(F)c1)N1C(C)CCCCC1 39954,c1(CC)ccc(O)c(C(N2CC(CNCC)C3CC23)=O)c1.C(C)(C(C)C)=CC=O 39955,Cc1ccc(C(=O)NCCC2(NC(c3ccn(C4CC4)c3C)=O)CC2)nc1O 39956,c1(C(CN(C2CC(C)(C)C2)Cc2ccccc2)O)ccc(F)cc1 39957,N1(C(=O)NC2CCN(C(C)=O)CC2)CC2CCN(C(=O)Cc3cnccn3)C2C1 39958,N1(CC(=O)NCC2(CCCC)CCC2)C(=O)c2ccccc2C1=O 39959,N1(C(C=C2CCC(C)CC2)=O)CC2CC(NC(c3ccc4c(c3)OCO4)=O)C(C2)C1 39960,c12cc(ccc1C)NC2=O.CCCC(C(=O)N(CCOC)CCOCC)OC 39961,c1(C(N2CC(C)CC(NC(CCC=CCC=C)=O)C2)=O)ncc(P(C)(C)=O)cn1 39962,c1(OCCCC)ccc(C(=O)NC2CCCC2NC(c2n[nH]cc2Cl)=O)c(O)c1 39963,C1(C(N2CC(CC)(CC)C2)=O)CCN(C(c2cc(C3CC3)no2)=O)C(C)(C)C1 39964,c1(C(=O)OC)sc(C(=O)NC2CCCCC2CNC(C2CC2F)=O)cc1N 39965,O=C1NCC2CN(C(c3ccccc3OC(F)(F)F)=O)CC12 39966,c1(C(=O)NCC2N(C(CC34CCC(C)(OC3)C4)=O)CC=C2)cnc2[nH]cncc1-2 39967,Cc1ccc([N+](=O)[O-])c(C)c1C(=O)NC1CCC1NC(=O)CC1CC=CCN1C 39968,N1(C(c2noc(CC)c2C)=O)CC(NC(c2ccc(C#N)[nH]2)=O)CC(O)C1 39969,C12(NC(COC)=O)CCOCC1CN(C(c1ccccc1S(=O)CC)=O)C2 39970,c1(NC(C2CC(O)CN2Cc2ccc(CO)cc2)=O)cccc(CC(F)(F)F)c1 39971,C1(C(=O)NCC2(C)CCCC2O)C2CCC(C2)C1NC(C1(C)COCCO1)=O 39972,c1(CCCCCNC(c2c(C)cccc2)c2nnnn2C2CC2)ccccc1Br 39973,Cc1ccccc1N1CCC(NC(c2ccn(C)n2)c2nnnn2C(C)C)CC1 39974,c1(CCNC(C2C(OC)CCC2)=O)ccc(CNC(=O)Cc2ccns2)cc1 39975,C1(NC(CSc2c(C)cccc2)=O)CN(C(=O)CCCC(C)N(C)C)CC1(C)C 39976,CC(CC(=O)N1CC(F)(C(N2CCCC(NC(N)=O)C2)=O)C1)C(F)(F)F 39977,c1(C(=O)NC2CC(CNC(CC(COC)C)=O)C2)ccc(Br)cc1O 39978,c1(C(=O)NC(CNC(C(CCCOC)C)=O)C(C)C)nccn2nc(C)cc12 39979,N1(C(C)=O)CC(C)(C)OC2(C1)CN(c1nnc(-c3cccc4ccccc34)o1)C2 39980,CC1(CC(=O)NCC2(C)CCC(NC(c3cncc(Cl)c3)=O)C2)CS(=O)(=O)C1 39981,C1(N(C(COCC#C)=O)C)CN(C(C2CCCCN2S(C)(=O)=O)=O)CC1(C)C 39982,O=C1CNC(=O)C(CCn2cc(CNC3CC(=O)C34CCC4)nn2)N1 39983,CCCC(CC(C)C)C(=O)N1CCCC1CNC(=O)CCC(=O)N(C)C(C)C 39984,C(=O)(CCC(C)(F)F)NC1C(OC)CN(C(=O)CC2CCCCC2)C1 39985,N1(C(CN(C(C)C)C)=O)CCCC2CN(C(=O)C(C)c3cncs3)CC12 39986,CCCCCC(C)(CC)C(=O)NCC1CC2(CC2)CN1c1ccnc2ncnn12 39987,c1(C(=O)Nc2scc(CC(=O)NC3C(C(N)=O)C3)n2)ccc(F)c(Cl)c1 39988,N1(C(c2c(CCC)nns2)=O)CC2CC2(CNC(=O)CCSCC(=O)OC)C1 39989,c1(C(=O)NCCCN(C(C(CC)=CC)=O)Cc2ccccc2)cncc(OC)c1 39990,N1(C(C(C)(CO)NC(C2CCN(CC)CC2)=O)=O)CCCC2(CC(O)C2)C1 39991,N1(C(C2CC3(CC(C)C3)C2)=O)CC2CCN(C(=O)CCC3CCCCO3)C(C2)C1 39992,c1(C(=O)NCC2(F)CCC(NC(C(CCOC)C)=O)C2)cc(OC)c(O)c(N)c1 39993,N1(C(C2C(COC)CC2)=O)CCC2CN(C(=O)CC3(CO)CC3)C2C1 39994,S(=O)(=O)(c1ccc(NCC2(C(C)C)CCOC2)c(Cl)c1)N1C(C)CC2(CCC2)C1 39995,C1(CNC(c2cn(CCC)nn2)=O)C(C)CCCN1C(C1CCC(CO)CC1)=O 39996,CCC(C)CCC(=O)N1CCOCC1C(=O)NC(C)CSC(F)F 39997,c1(C(=O)NC2CC3(C(=O)NC(CO)CCCO)COC2C3)c[nH]c2ccncc12 39998,C1(NC(c2cc(COC)oc2C)=O)(CO)CCN(C(=O)C(C)CC(F)F)CC1 39999,c1(CCC(=O)OCC)cccnc1F.C1CCCN(C(=O)CC2CN(C(C)=O)C2)C1 40000,N1(C(c2nc(CCC)oc2)=O)C(CNC(=O)C(C)(C)CO)CC2CCCC12 40001,N1(C(CSCC(=O)OC)=O)CCC(C(C)(C)NC(=O)CC2CSCCS2)C1 40002,C(C)(C1CCCc2ccccc21)NC(c1ccc(Cl)cc1F)C 40003,N1(C(=O)CN2CCCC2)CCC2(CC1)CC2C(N1CCC2(C=CCO2)C1)=O 40004,C1(C(=O)NCC(C)(C)CNC(C2CC3(CCCC3)C2)=O)C2Cc3ccccc3C12 40005,CCCCC(CNC(C1C=C(C)CS1)=O)NC(=O)C(C)OCc1ccccc1 40006,c1(CC(=O)NC(CN(C(CN(CCOC)C)=O)C)C)ccc(Br)c(F)c1 40007,c1(C(C(N2CCCC(N(C(CC(=C)C)=O)CCO)C2)=O)C)c[nH]c2ccccc12 40008,C(CC(C)C)(C(=O)N1CCCC(CNC(c2c(C)noc2C)=O)C1)OC 40009,C=C(C)C(O)CC(=O)NCc1cnn(C2CN(C(=O)CCC3CC3)C2)c1 40010,C12(CNC(c3cccc(C)c3)=O)CCC1CN(C(C1CCCCNC1=O)=O)C2 40011,CC(C#N)CCC(=O)N1CCOC(CNC(=O)Cn2cnc(Br)n2)C1 40012,C(C(C)C)(C(O)C(=O)N1CCCCCC1C(=O)N(C(C)CC1CC1)C)OC 40013,C(=O)(C#CC1CCOCC1)NC1CC(NC(CCCNC(C)=O)=O)C12CCC2 40014,C1(C(=O)NCC(C)NC(C23CCC(F)(CC2)C3)=O)CC2C=CC1CCC2 40015,C1(NC(c2ccc(C)nc2)=O)CN(C(c2ccc(SC(F)(F)F)s2)=O)CCC1C 40016,C=CCC(C)(C(F)F)NC(=O)CCN.C(=O)(CC(C)COC)N(CCN(C)CC)CC 40017,Cc1nc(C)c(CCC(=O)NCC2CN(C(C3CC(N(C)C)C3)=O)C2)c(O)n1 40018,CCCC(C(=O)NCCCCCN1CCN(C(C2COC(=O)C2)=O)CC1)N(C)C 40019,C12(CNC(C3CC4(CSC4)C3)=O)CCN(C1)C2=O.C1(CO)CCCC12CC2 40020,C1(C(=O)NCC(C)(C)NC(c2ncoc2Br)=O)CCOCC1(C)C 40021,C(=O)(C(F)CC(C)(C)C)N1C(C(=O)NC(c2c(C)nccn2)C)COCC1 40022,c1(C(=O)NCCCN(C(C(C)C2CCCC2)=O)C)cc(F)cc(S(N)(=O)=O)c1 40023,C(CCC(C)CC(=O)N1CC(O)(CCNC(C2CCCOC2)=O)C1)=C(C)C 40024,N1(C(c2cc(C)c(=N)[nH]c2)=O)C2CCC(C(=O)NC3(CC(C)C)CC3)C1CC2 40025,C1(C(=O)NCC2(CNC(C3C(SC)CCC3)=O)CC2)CCCN(C(=O)C(C)C)C1 40026,c1(NC(C2(C(=O)NCC(C(=O)OCC)(F)F)CC2)=O)cc(Br)cnc1C#N 40027,N1(C(c2c(C(C)C)occ2)=O)CCCCC12CN(C(C1SC3C=CC1C3)=O)C2 40028,C1(C(=O)NC(c2ccccc2)C(F)F)CCC(=O)N1 40029,C1(c2n(CCCSCC)nnn2)(NCC2CCC=CCC2)CCN(C(C)C)C1 40030,C1(C(N2CC3C(CNC(C(c4cccnc4)C)=O)C3C2)=O)CCCCC12CCC2 40031,CS(=O)(=O)c1cc(C(N2CCC3CN(S(=O)(=O)C4CC4)CCC23)=O)ccc1F 40032,C1(NC(C(c2n(C)ncc2)O)=O)(COC)CCN(C(=O)CSc2nncn2C)C1 40033,Cc1cc(Cl)c(C(N2CC(C)(C)C2Cn2cc(C3CCCCO3)nn2)=O)s1 40034,C1(CNC(c2nnnn2CCCF)(C)CN2CCCC2=O)CCS(=O)(=O)C1 40035,C(=O)(C1=NOC(C)C1)NCCN(C(C1C(C=C)OCC1)=O)C 40036,C1(NC(CC(=O)OC)=O)CC(O)CN(C(=O)Cc2ccc(OC(F)(F)F)cc2)C1 40037,C(CCCCC(=O)N1CC2CC1(CNC(C)=O)C2)OCC 40038,c1(C(=O)NC2CCCN(C(C3C4COCC34)=O)C2)cc2oc(Br)cc2s1 40039,c1(CC(=O)NC2(COC)CN(C(c3cc(C#N)cs3)=O)C2)cnccc1Cl 40040,C(=O)(C(CC(F)F)NC(=O)NC(C)(C)C)NC(c1c(C)nn[nH]1)=O 40041,C1(CC)CCCN(C(c2cncs2)=O)C1C(=O)NCC1CC(=O)N(C)C1=O 40042,c1(C(C)NC(=O)NC2(C(C)C)C(OC)CC2N(C)C)csc2ccccc12 40043,O=S(=O)(c1cccnc1NCCC1CCC2CC12)NCc1cc(C(F)F)on1 40044,c1(C(=O)NC2C(C)N(C(=O)CCc3cnoc3)CC2)nccc2[nH]ccc12 40045,Cc1c(C(N2CCN(C(=O)C(F)C(C)C)CC2CS(C)(=O)=O)=O)cccc1C#N 40046,C(C(CC(C)C)C(=O)NC1CC(CNC(=O)C(C2CCCC2)SC)C1)OC 40047,C(C(C)(F)F)N(C(C=CC(C)NC(C1(C(N)=O)CC1)=O)=O)C 40048,c1(NC2C3OCC(N4CCC(C(=O)OCC)CC4)C2C3)cc(Cl)c(F)cc1C 40049,c1(C(C)NC(=O)CSC(C)(C)C)ccc(CNC(C2(F)CC2)=O)cc1 40050,N1(CC(=O)NC2CN(C(C(C)=C3CC3)=O)CC2C(F)F)CCSC2CCCCC12 40051,C1(NC(c2c(C)cco2)c2nnnn2CC2CC2)C2CC2C2CC12.c1ccccc1 40052,N1(C(c2cccc(CC)c2)=O)CCC2(CC1)CC2NC(C1(C)CC(C)=NO1)=O 40053,N1(CC#C)CCCC2(CCN2C(=O)CCN(C)C(C)=O)C1 40054,CC1OC2(CO)CC1(C(N1CC3(C1)CN(C(=O)C(O)(C1CC1)C1CC1)C3)=O)C2 40055,C1(C(F)F)(CNC(CC(=O)NCC)=O)CCN(C(c2cnn(C)c2OC)=O)C1 40056,c1(CC)nc[nH]c1C(N1CCCC1CNC(=O)CC1CCSCC1)=O 40057,C1(C)(C(=O)NCC(C)NC(=O)CCCCN2CCOCC2)CCC12CCC2 40058,c1(CN2CCC(C(=O)NCC3(N(C)C)CCCC3)C2)cc(Cl)ccc1N 40059,C1(CSc2ccc(C(=O)OCC)cc2)Cc2ccccc2O1 40060,N1(C(CC2OCC(C)(C)C2)=O)CC2CC(C1)N(C(c1ccc(F)cc1)=O)C2 40061,C1(NC(c2cccc(C)c2Cl)=O)CC(N=c2[nH]cnc3cccc([N+](=O)[O-])c23)C1 40062,C1(N(C(C(C)N(CC(F)(F)F)C)=O)C)CN(C(=O)CCc2nccs2)CC1(C)C 40063,c1(C2C(C(=O)NCCN(C(=O)Cc3cnn(C(F)F)c3)CC)C2)ccccc1Cl 40064,C1(C(=O)NC2(CO)CN(C(=O)C(C3CCOCC3)O)C2)COC2(CCC2)CO1 40065,c1(C(=O)NC(C)C(C2CCCCC2)NC(N)=O)ccc(Cl)c(N)c1Cl 40066,N1(C(c2c(C)nsc2C)=O)CC(NC(=O)CC(O)CN(C)C)CC2(CC2)C1 40067,C(C)(CCN=c1cc(CC2CC2)nc[nH]1)NC(c1cnn(CC)c1C1CC1)=O 40068,c1(CCC(=O)NCCC2CCN(C(C3N(CC)CCC3)=O)C2)ccc(C)cc1C 40069,C1(C(=O)NCCNS(CC)(=O)=O)CN(C(C2(CC)CCCC2O)=O)CC1(F)F 40070,c1(C(N(CCNC(CC(C)OC)=O)C)=O)cnc2ncnn2c1C(C)C 40071,C1(CNC(CCC=CCC=C)=O)CC(NC(c2coc(Br)n2)=O)C12CCC2 40072,C1(CC#C)(C(=O)NCC(C)(CNC(=O)C=CCN(C)C)OC)CCOC1 40073,c1(C(N(CCCOCCN(C(C(CC=C)C)=O)C)C)=O)c(C)cc(C)nc1O 40074,CCC(C(=O)NCCc1cnc(C)s1)N(C(=O)CNC(=O)CNC(C)=O)C 40075,N1(C(C(C(C)(C)C)NC(=O)C(=O)NC2CC2)=O)CC2C3CCC(O3)C2C1 40076,C(C(C(=O)NC1CC(C)CC(C)(C)C1)C(C)(C)C)NC(c1c(C)ncnc1)=O 40077,CN(C1CCCc2n[nH]cc21)CC1COCCC12CCC2 40078,c1(C(C)=O)cc(C(=O)NCC2(CO)CCCO2)n[nH]1.C1=CCNC1=O 40079,Cc1cc(C(N2CC3C(NC(c4cccnc4)=O)C3C2)=O)c2cc[nH]c2c1 40080,c1(NC(C2(N(C)C)CC2)=O)cccn(C)c1=O.N12CCC1(C)CC2=O 40081,C=C(C)CC(C(=O)NCCC1CC(F)(F)CN1C(C1CCCOC1C)=O)OC 40082,N1(C(c2n(CC)nnc2)=O)CCC(NC(=O)C(C)(C2CC2)OC)C1C 40083,c1(SC(CNC(C2(F)CC(NC(C)=O)C2)=O)(C)CO)nnnn1CC(F)(F)F 40084,Cn1cncc1C(c1nnnn1Cc1cccs1)NCCC(O)CO 40085,c1(C(N2C(CNC(C3C(C#N)C3)=O)CCCCC2)=O)noc2cc(F)ccc12 40086,O=C(N=c1[nH]c(Cl)ncc1O)C1CN(C(C2CC2(F)F)=O)CCC1O 40087,C1(N=[N+]=[N-])(C(=O)NC(C(C(=O)OC)C)C)CCN(C(C2CCCC2C(C)C)=O)C1 40088,N1(C(CC(C)N2CCCC2=O)=O)CCC(C(F)F)(CNC(C2(Cl)CC2)=O)C1 40089,c1(C(=O)NC2C(CNC(c3scc(COC)c3)=O)CCC2)cccn2nncc12 40090,C#CC1CCN(C(=O)C(COC(C)C)NC(c2cccn(C)c2=O)=O)CC1 40091,c1(C(=O)NC2CCN(C(CC(C)C(F)(F)F)=O)C(C)C2)c(N)c(F)cc(F)c1F 40092,CCC(Cc1ccccc1)C(=O)NC(C)CNC(c1cc(C(F)(F)F)no1)=O 40093,S(=O)(=O)(c1ccoc1)N1C2CCC21.c1(NC=O)cccc(F)c1 40094,Cc1cc(C(C)(C)C)ccc1C(=O)NCCC1=CCCC1 40095,C=C(C)C(C)(C)C(=O)NCCC1CCN(C(C2CCC(C(=O)OC)O2)=O)C1 40096,c1(C(=O)NC(CC)CNC(C2(O)CC(C)(C)C2)=O)ncc2ccccn12 40097,C1(NC(c2n(CC)ncc2)=O)CCC(C(=O)NCC2CC3C=CC2O3)CC1 40098,N1(C(CC(C)(C)OC)=O)CCC(CO)C(NC(=O)CC2(C(=O)OC)CC2)C1 40099,c1(C(=O)NCC2CCCC(NC(CCC)=O)C2)cc(C)c(C)c2ncccc12 40100,N1(CCNC(C2CCC(CNC)CC2)=O)CCCOC(C)C1 40101,N1(C(CCNC(COC)=O)=O)CCC(C(=O)Nc2cnnn2C)C1 40102,S(=O)(=O)(c1cnc(NC(C2CCCO2)C)c(Cl)c1)NCCc1cccc(C)c1C 40103,n1(CC(=O)NCC2N(C(C3C(CCOC)C3)=O)CCCC2)ccc([N+](=O)[O-])n1 40104,C1(Cl)(C(=O)OCC)CC12CCN(Cc1cnn(Cc3ccccc3)c1)CC2 40105,CCC(O)C(C)C(=O)N1CC(CCn2cc(-c3ccc(C)cc3C)nn2)C1 40106,C(=O)(C(O)CCCNC(=O)C(O)CNC(C)=O)NCCC(CC)C 40107,C(C(CNC(=O)CCc1cnoc1)NC(=O)CC1CC(C(C)(C)C)C1)OC 40108,CC1(C)C(NC(c2cc(C3CCC3)no2)=O)CCN1C(=O)Cn1cccc1 40109,C=CC(C)C(C)C(=O)N(CC(CO)(CO)NC(c1cc(CCC)[nH]n1)=O)C 40110,N1(C(C2CC(=C)C2)=O)CC2CCC1C1CN(C(c3ccsc3S(N)(=O)=O)=O)CC21 40111,C(=O)(CCN(OC)C(=O)C(C)(O)C(F)(F)F)NCC(C#C)CC 40112,C1(S(C)(=O)=O)(C(N(C)CCNC(C2CCC2C(F)F)=O)=O)CC(O)C1 40113,C1(NC(Cc2cncc(C)c2)=O)CC2CCC(C1F)N2C(c1csc(S)n1)=O 40114,N1(C(CCN(C(c2ncn(C)n2)=O)C2CC2)=O)CCOCC(CO)C1 40115,C(=O)(C(O)CC(N)=O)NCC1(OC)CN(C(=O)CCNC(C2CCCO2)=O)C1 40116,c1(C(=O)NC(CN(C(=O)COC2CC(F)(F)C2)CC)C)cccc(OC)c1F 40117,N1(C(CC)=O)Cc2ccccc2CC1CNC(C1CCC2CC2C1)=O 40118,N1(C(C(C)Oc2ccc(C)cc2)=O)CCN(C(C2CCCCN2C)=O)CC1C 40119,c1(C(=O)NCC2CCCC(C)C2)cccc(S(C)=O)c1 40120,c1(-n2c(CCc3cnn(C)c3)nc(C(C3CC3)OC)n2)ccc2c(c1)OCCO2 40121,c1(C(=O)NC(C(C)NC(c2c(CCC)nco2)=O)CO)cc2cccc(C)n2n1 40122,CC1CN(C(C)C(=O)N(CC(=O)NC(C(N)=O)C2CCCC2)C2CC2)C1 40123,C1(NC(c2csc(-c3ccco3)n2)=O)CC(O)CN(C(C2CC(O)C2)=O)C1 40124,C(C(CC=C)NC(c1conc1C1(C)COC1)=O)NC(COCCOC)=O 40125,C(=O)(CCC(=O)NN(C)C)N(C(C)C(C)CC)CC.C12(CCC1)C(=O)NC2 40126,c1(C(=O)NCC2(OC)CN(C(=O)COCCF)C2)cc(Br)ccc1Cl 40127,c1(-c2onc(C(CC)(C3CC3)Nc3cccc(C)c3)n2)cc(SC)c(C)nc1O 40128,C1(SC)CN(C(=O)C(C)(C)C2CC2)CC1NC(c1cc(F)n(C)n1)=O 40129,c1(OC)cc(N)c(Cl)cc1C(=O)NCC1(NC(C2CC23CC(O)C3)=O)CCOC1 40130,CC(O)(Cn1cc(Br)cn1)C(=O)N1CCC(CC(N2CCSCC2)=O)C1 40131,N1(C(c2cc(C)c(N)cc2C)=O)CCC2CCCNC2C1 40132,C1(C(=O)NC(C)C(C)(C)C)CN(C(C2(c3ccccc3)CC2)=O)CCC1(C)C 40133,c1(C(c2n(CC=C)nnn2)NCC2(n3cccn3)CC2)cc(Cl)cc(C)c1OC 40134,c1(CN(C(Cc2cc(C)no2)=O)C)cccc(CNC(C2CCCC(O)C2)=O)c1 40135,C1(C(N(CCN(CC)CC)C)=O)CC12CCN(C(c1cncc(NC)c1)=O)C2 40136,N1(C(c2c(C(N)=O)cccc2)=O)CCC(F)C(NC(C2CCC(F)CC2)=O)C1 40137,c1(C(C2CCN(C(=O)C(F)C(C)(C)O)C2)C)cc([N+](=O)[O-])ccc1NC(C)(C)C 40138,CC1OCCC1(F)C(=O)NC1CC(C(=O)N(C)CCC2CCCCC2)C1 40139,C12(CNC(c3n(CC)ccn3)=O)CCC(C1)N(C(=O)C=Cc1ccc(C)cn1)C2 40140,c1(CN(C(C(=O)N(C(c2ccco2)C)C)=O)C)cc2c(s1)CCCC2 40141,C(=O)(C(CCC(C)C)NC(=O)C1=CC2C=CC1C2)NC1(C=C)CCOCC1 40142,n1(COC)nccc1NC(=O)C(N)CC1CC(Cl)=NO1 40143,C1(C2CCCCO2)(C(=O)NCCCCNC(c2c(CC)cncc2)=O)CCCO1 40144,C1(C(N2CCOCC(O)C2)C(=O)NCC2CCCO2)CC2(CCC2)CO1 40145,C1(NCC(C(C)C)C)CC2(COC(C)C2)C1 40146,N1(C(c2c(C)onc2)=O)CCN(C(C2C(C)C2C)=O)C2(CCC2)C1 40147,c1(CC(=O)NC(CCNC(CCCOCC)=O)C)cccc(Br)c1 40148,c1(C(=O)NC2CCC(NC(Cc3ncc(C)s3)=O)CC2)ccc(C(C)=O)nc1O 40149,C(=O)(C(O)CC[S+](C)C)NCC1(C)CCN(C(c2cn(CCOC)nn2)=O)C1 40150,c1(C(N2CCN(C(c3cnsn3)=O)C(C3CCC3)C2)=O)nccc2[nH]ccc12 40151,[N-]=[N+]=NCCC(=O)NCCC(O)C(=O)N1CCOC(C2CCC2)C1 40152,C(=O)(C(F)C(CC)CC)NCCOCCC(=O)NC(c1nccn1C)CC 40153,N1(C(=O)CCCC2CCC2)CC2(CCCCN2C(=O)CCN2CCOC2=O)C1 40154,Cc1ncc([N+](=O)[O-])cc1C(N1CCOC(C(C)Nc2ncccn2)C1)=O 40155,C(CN=c1ccnc(N2CCNC(=O)C2)[nH]1)N1C(=O)NC(C)(C)C1=O 40156,c1(C(=O)NC(CCNC(Cc2ccn(CC)n2)=O)C)cc(C)cc(O)c1 40157,c1(C(=O)NC2CC(C)(C)CN(C(=O)C#CC3CC3)C2)c[nH]c2ccncc2c1=O 40158,C1(NC(CCNC(CC(C)C)=O)=O)CN(C(=O)C(C)(C)C(F)F)CCC1O 40159,CC(C)C(C)CC(=O)NCC(C(=O)N1CC(O)(C(C)C)C1)N(C)C 40160,c1(C(=O)Nc2c(C)cccc2C#N)c[nH]c2cc(C#N)ccc12.C12CC1C(=O)N2 40161,N1(C(CCCC(=C)C)=O)CC=C(CCNC(=O)CCc2ccsc2)CC1 40162,c1(-n2cc(CCC(=O)NCC3CC4CCC3(CO)C4)nn2)ccc([N+](=O)[O-])cn1 40163,C1(C(N(C(CCNC(c2c(C)ncnc2)=O)C)C)=O)COc2ccc(F)cc2C1 40164,c1(NC2CC(C)N(C(=O)CCCc3cnccn3)C2)ncc([N+](=O)[O-])cc1Cl 40165,O=C1CN(CC(=O)NCC2C3CN(CC(=O)Nc4ccc(Cl)nn4)CC23)C(=O)N1 40166,c1(C(=O)NC2CC(CNC(C3C=CCC3)=O)C2)c(Cl)ccc2ncccc12 40167,c1(C(N2C(C(C)NC(CC3(C=C)CCC3)=O)CCCC2)=O)cccn2cncc12 40168,C12(C(=O)NCc3ccnc(C)n3)CCC1CN(C(C1CCCC1F)=O)C2 40169,C(=O)(CC(C(C)OC)NC(=O)C(F)C(C)C)N(CCC#C)C1CC1 40170,C(C(C(=O)NC1CCOC1)N(C)Cc1cn(-c2ccccc2)nn1)(C1CC1)OC 40171,c1(C(N(C(C)CCNC(=O)CC2CCC(O)C2)C)=O)cccc2c1CCC2=O 40172,C(C(COC)C(=O)N1CC(CCCCNC(C2(OC)CCC(C)C2)=O)C1)OC 40173,C#Cc1c[nH]nc1C(N1C(C(N2CC(C(CC)CC)C2)=O)CC1C)=O 40174,C1(NC(C2(COC)CCCC2)=O)COCCN(C(=O)Cn2ccnn2)C1 40175,C(=O)(C1=CCCCO1)NCC(CCOC)NC(C1CC(=O)NC(C)C1)=O 40176,C1(NC(c2cnc(CC)s2)=O)(CF)CCN(C(=O)C(c2cccs2)SC)C1 40177,c1(C(N2C(CNC(C3CCN(OC)CC3)=O)CC2)=O)cnc(O)c2c1NCCC2 40178,c1(OC)ccc(Cl)cc1CC(=O)NCC(C)(C1CC1)NC(=O)CCc1ccsc1 40179,N1(C(C(c2ccnn2C)NC(c2nc(CC)sc2)=O)=O)CC(C2CCCCC2)C1 40180,C12(C(=O)NC3CCCN(C(c4c(CC)c[nH]n4)=O)CC3)CC3CC(CC1C3)C2 40181,C12(NC(C(=O)NC(c3ccc(F)cc3Cl)(C)C)=O)CCC(CO)(C1)OC2 40182,C(CCC)(C(=O)NCCC1(NC(=O)COc2ccsc2)CCCC1)=CCC 40183,C1(C(=O)NC2CC(NC(CC(C=C)(C)C)=O)C2)COc2ccc(OC)cc2C1 40184,Cc1nc(=N)[nH]cc1C(N1CCCC1C1(O)CN(C(=O)CC2CCCN2C)C1)=O 40185,C1(CCC(=O)NCCC(C)NC(=O)C(c2ccc(F)cc2)(F)F)CCCCN1C 40186,C1(NC(C=CC(C)NC(C2(CN(C)C)COC2)=O)=O)CNC(=O)C1 40187,c1(C(C)(C)C)nc(C(=O)NCCCC2CCCN2C(=O)CN2CCOC2=O)co1 40188,Cc1nn(C)cc1C(O)C(=O)NCc1cccc(NC(c2coc(O)n2)=O)c1 40189,c1(C(=O)Nc2ccnc(N3CCOC(C(F)(F)F)C3)c2)cc2c(cc1O)CCCC2 40190,CC(C)CC(O)C(=O)NC(C)CNC(c1cc(C(F)(F)F)cc(N)c1)=O 40191,C(=O)(C1CCCn2nccc21)N1CC2(CCN(C(c3ccccn3)C)CC2)C1 40192,N1(C(C=CCNC(C2CC(C)(O)C2)=O)=O)CCc2ncccc2C1 40193,C1(C(=O)NCCCN2CCC2)(CC)C=CCN1C(=O)CNC(N)=O 40194,C(C(COC)CC(=O)NC1CCC(NC(=O)CC=C(Cl)Cl)CC1)OC 40195,c1(NC(CNC(=O)Nc2nn(CCOC)c(C)c2)=O)ccc2ncsc2c1Br 40196,N#Cc1cncc(CN2CCC(O)C(C(N3CCC(O)C3)=O)C2)c1 40197,N1(C(c2nc(CC)sc2)=O)CC(NC(=O)C(c2ccccc2OC)(C)C)CC1C 40198,C12(CC)CC1CN(C(C1CCCCC1NC(=O)C(C)c1ccsc1)=O)C2 40199,c1(C(=O)NC(C2CN(C(C(=O)NCC)=O)C2)C)ccc2nnc(O)n2c1 40200,c1(C(N(CCCCCC)CCNC(c2ncsc2CC)=O)=O)cccc(=O)o1 40201,c1(CC(N2CC(C)N(C(C3CCN3C(C)(C)C)=O)CC2)=O)cccc([N+](=O)[O-])c1 40202,Cc1ccc(C(C)C)cc1C(=O)NC1CCN(C(=O)C(O)P(C)(C)=O)CC1O 40203,O=C(C(O)Cn1cncn1)NC1CN(C(C2CC2(Cl)Cl)=O)C1 40204,Cc1nc(CC2CCC2)sc1C(=O)NC1CN(C(c2ccccc2C(C)C)=O)C1 40205,c1(C(=O)NC2CC3C(NC(C(=O)N(CC(F)F)C4CC4)=O)C3C2)ncccc1Cl 40206,C1(C(=O)NCC2C(CNC(CC=CC)=O)C2)CCc2ncsc2C1 40207,c1(C(=O)NC(C)CC(C)NC(=O)Cc2ccc(C#N)cc2)cnc2[nH]ccc2n1 40208,Cn1nc(C2CC2)nc1CNC(=O)C(=O)NC1CC(N2CCCC2)C1(C)C 40209,N1(C(c2cnc(C)s2)=O)CCC(NC(c2cc(=O)n(C)o2)=O)CC1C 40210,C1(C(=O)NCCc2ccc(CC(C)C)cc2)CCCC12CCN(C(=O)C(C)C)C2 40211,c1(C(N2CC3(NC=O)CC2C3)=O)ccc2n[nH]cc2c1.C1(NC(=O)C2CC2)CC1 40212,c1(C(N2CC(NC(C=Cc3c(C)ccs3)=O)C2)=O)cccc(P(C)(C)=O)c1 40213,c1(C(N(CCNC(C2(O)CCSC2)=O)CC)=O)ccc(S(=O)(=O)NC(C)C)cc1 40214,Cc1ccsc1-c1cn(CC2C=CCN2C(=O)CC2CCOC2=O)nn1 40215,CCCC(CC(C)C)C(=O)NCC(C)CNC(c1cc(N)cc2c1OCCO2)=O 40216,NS(=O)(=O)C1CN(C(=O)Cn2nnc(-c3ccc(Cl)cc3)n2)C2(CCC2)C1 40217,c1(CC(=O)NCCOCCCNC(C(C)(C)n2cnnn2)=O)ccc2c(c1)CC2 40218,c1(C(N2CC(NC(C(CCC)NC(C)=O)=O)C(C)C2)=O)cn(C)c(C)cc1=O 40219,CC1(C)C(CC(=O)NC(CCO)c2ccsc2)CCN1C(=O)CCCC1CCC1 40220,Cc1nc(CSC)ncc1C(=O)N(CCCNC(c1ccco1)=O)CCO 40221,CC(CNC(C1COCCC1C)=O)C(F)C(=O)NC1(CC2CCC2)CC1 40222,n1(CC=C)c(SCC2NCCC2C)nc2sc3c(c2c1=O)CCC3 40223,C=C1CC2CCCC(C1)N2C(=O)C(c1ccoc1)NC(=O)C(O)CC(C)C 40224,N1(C(C=C(C)Cl)=O)CCCN(C(=O)CCOC2CCC2)C(c2ccccc2)C1 40225,CC(C)C(O)C(F)(F)C(=O)NCC1C(C)CCCN1C(=O)CCc1cnc[nH]1 40226,c1(C(=O)NC(CNC(C2C(=C)CC2)=O)CCOC)c(C)cc(C)oc1=O 40227,C1(C(N2CC(N(C)C(C3CCS3(=O)=O)=O)C3(C2)CC3)=O)CC2(C1)CC(C)(C)C2 40228,C1(N(C(CNC(CC)=O)=O)C)CCN(CCSc2cc(C)c(C)s2)CC1 40229,CCCCCC(C)CC(=O)NCCC(O)CNC(c1ncoc1C1CC1)=O 40230,CC(C)CC(C(=O)N(C)CC1(CO)CC1)NC(C1CCC(=O)N(C)C1)=O 40231,C(CCSC)(C(=O)NCc1cn(CC(C)NC(=O)Cc2ccccn2)nn1)OC 40232,C1(C(N(CCC)CC)=O)CCC(O)CN1C(=O)CC(Cl)Cl 40233,C1(C(N2C(CC(=O)OC)COCC2)=O)CC2OCCC2N(C(=O)CCCCCl)C1 40234,c1(C(N2C3C(NC(C(C(=C)C)(C)C)=O)C(C3)C2)=O)cc2c(s1)CCS(=O)(=O)C2 40235,Cc1nn(C2CCC2)cc1C(N1CC(CNC(=O)CCC(=O)C2CC2)C(O)C1)=O 40236,CCCC(CCC)C(=O)Nc1cccc(CC)c1.n12cnc(c1)C(=O)NOCC2 40237,Cc1nc(N2CC3CN(C(c4cc(Cl)c(Br)c(Cl)c4)=O)C3C2)c2c(n1)CCC2 40238,Cc1cc2sc(CC3CN(C(c4ccccc4)C(=O)NCC(F)F)CCO3)cc2s1 40239,C(=O)(C(C)(C)C(C)(F)F)NC(C1CC(NC(C2CC2C2(O)CCC2)=O)C1)C 40240,N1(C(C(=Cc2ccncc2)C)=O)CCC(C2CCN(C(C3CC3(C)C)=O)C2)CC1 40241,c1(C(=O)NCC2CCN(C(C3C(C)CCC3)=O)C2)ncccc1NC(=O)C(C)(C)C 40242,N1(C(C(CC2CCOC2)NC(=O)OC(C)(C)C)=O)CC2(CNC(=O)OC2)C1 40243,C1(NC(C(CC)O)=O)(COC)CCCN(C(C2CCC2C(=O)OC)=O)C1 40244,c1(C(=O)NCCC2CC(NC(C3CC3Cl)=O)C2)cc2c[nH]cnc-2n1 40245,Cc1ccc(F)c(C(N2CCCC(C)(CNC(c3c[nH]c(C#N)c3)=O)C2)=O)c1F 40246,O=C1CCC2(C(=O)NCC3(O)CCN(C(c4cnsc4)=O)CC3)CCCCC2N1 40247,C1(C(=O)NCCCC(C)C)CN(C(=O)C(C)C(C)C)CC1(C)C 40248,N1(C(c2cc(C)ncc2)=O)CC(C(=O)NCC2CC(=O)N(C)C2)CC(F)C1 40249,c1(C(N(C2CCCN(C(c3csnc3Cl)=O)C2)CCO)=O)ccc2[nH]ccc2c1 40250,c1(C(C)NC(c2nnn(-c3ccccc3)c2C(F)(F)F)=O)c(F)cccc1F 40251,n1(C(C)C)cc(C(=O)NCC2COC(CN)C2)c(O)nc1=O 40252,N1(C(c2ccc(SC)o2)=O)CCCC(C2CN(C(c3scc(C)c3Cl)=O)C2)C1 40253,N1(C(C(C)=CC2CC2)=O)CCC2CC2(C(=O)Nc2cccc(CO)c2)CC1 40254,CC(CCNC(=O)C=Cc1ccco1)CCNC(C1COCCN1C)=O 40255,c1(CCC(N2CCC(NC(Cc3c(C)scc3)=O)C2)=O)cnc2ccccn12 40256,C1(OC2(CC(=O)N(CC(=O)OC(C)(C)C)C)CCC2)CCCCCC1 40257,c1(C(N2C3C(CNC(CC=CC=C)=O)C(CCC3)C2)=O)nc2n(c1Cl)CCCC2 40258,N1(C(C(CC)(C)OC)=O)CCc2nc(CNC(=O)CCCN3CCCC3)sc2C1 40259,C=C(C)CCCC(=O)NCC(CCOC)NC(c1nc(OC)cc(OC)n1)=O 40260,c1(C(C)C)ccc(C2CCCN(C(=O)C(C(C)O)N3CCNCC3)C2)cc1 40261,C12(CNC(=O)Cc3ccsc3Br)CCC1CCN2C(c1c[nH]nc1F)=O 40262,C(=O)(C(C#N)CC)N(C(=O)CN1CCOCC1)NCCC(=O)N(C1CCSC1)C 40263,C1(c2nnnn2C(C)(C)C)(CNCCC2(OC)CCC2)CC2CCOC12 40264,c1(-c2ccc(C(F)F)cn2)cc(F)ccc1F 40265,CC(C)(C)CC(C)(C)C(=O)N1CCC(C)(CC(=O)NCCCOCC(F)F)C1 40266,C1(O)(C(=O)NC2C(NC(CCNC(COC)=O)=O)COCC2)CC(C)(C)C1 40267,c1(OCCCNC(=O)C(N2CC(CO)C3(CC3)C2)=O)ccc(Cl)c(Cl)c1 40268,c1(CNC(C(c2cc(C)n(C)n2)N(C(C)CC(N)=O)C)=O)ccc2ccccc2c1 40269,c1(N(CCC)C)ccc(C(=O)NC23CC2CN(C(=O)C(C)n2cccc2)C3)cc1 40270,CCC(C)C(O)CC(=O)NCC(C)(C)OCCNC(c1cnc2ccccn12)=O 40271,C1(NC2CCN(C(=O)NCc3cn(CC)nc3)CC2)CCCC(C)(C)C1 40272,c1(CN(C(c2c(COC)noc2)C(=O)NC(C)C)C)ccc(Cl)c(Cl)c1 40273,N1(C(CCN(CCCCC)CC)=O)CCC(N(C(=O)Cc2scnc2C)C)C1 40274,c1(C(=O)NCC2(CCNC(CC3N(C)CCC3)=O)CC2)csc(C#N)c1 40275,Cn1ccc2sc(C(N3CCC3CNC(c3nccn4cnnc34)=O)=O)cc12 40276,N1(C(C(C)CC2CC2)=O)CC2CCC(C1)N2C1CCN(C(=O)C(O)C2CC2)CC1 40277,c1(C(C(=O)NC2CCCC2)N(C(C)C2CC2)CC)cnc2n1CCC2 40278,N1(C(C(C)SC)=O)CC2=C(C1)CN(C(c1cnc(C(F)F)c(C)c1)=O)C2 40279,c1(C(N(C2CN(C(C(CC)(F)F)=O)CC2O)C)=O)cc(F)c(C(C)C)cc1F 40280,c1(C(N(CCNC(CC2CN(C)C2)=O)CC2CCCO2)=O)ccc2nccn2c1 40281,c1(C(=O)NCC2C(NC(=O)Cc3cc(Cl)ccc3O)CC2)cccc2c[nH]nc12 40282,C(=O)(C1=CCC(C)(C)CC1)NCC1(F)CCCN(C(CSCC=C)=O)C1 40283,c1(NCC2CC(NC(C(C(=O)OC)C)=O)C2)cc(C(F)(F)F)c(C)c([N+](=O)[O-])c1 40284,C(CC(C)C(=O)NC12CC(NC(=O)Cc3ccc(CO)cc3)(C1)C2)=CC 40285,CC(C)C(CC(=O)NC1CCCCNC1=O)NC(C1CCSCC1)=O 40286,C(=O)(CN1C(=O)CCc2ccccc21)NCC1C(NC(CC2CN(C)C2)=O)CC1 40287,c1(-c2c(NC(N(C(CC(CC)C)C)C)=O)c[nH]n2)ccc(Br)cc1F 40288,CC1(C)COCCC1NC(C1CC(NC(c2cccnc2CO)=O)C1)=O 40289,C1(NC(=O)NCCCN(C(CC)C)C(C)C)CCC1C(=O)OC(C)(C)C 40290,N1(C(Cc2c(C)cnn2C)=O)CCN(C(=O)COc2ccsn2)CC(O)C1 40291,C(=O)(C(C)C(C)NC(C1(COCC)CC1)=O)NCC1CCOC1 40292,c1(-n2c(CC(N3CCOCC3)C)nc(CC3(C)CC3)n2)ccnc2ccccc12 40293,N1(C(C(C)(C)F)=O)CCC2(CCN(C(C3CC(c4ccc(F)cc4)C3)=O)C2)C1 40294,c1(OCC)ncc(-c2cnc(CNC(c3ccc(C(C)(C)C)cc3)=O)nc2)cn1 40295,c1(C(=O)NC2CC(CS(N)(=O)=O)C2)cccc(C(=O)O)c1 40296,Cc1ncc(C(=O)NC(C)(CO)C(=O)N(C)CC2(N(C)C)CCC2)c(C)n1 40297,C1(NC(C2C(c3c(C)occ3)C2)=O)CC(C)N(C(c2ccc(C(C)C)nc2)=O)C1 40298,N1(C(COCCOC)=O)CCN(C)C(CNC(C2CN(C)CCO2)=O)C1 40299,C1(NC(C2(C)COC2)=O)CCC2(CC1)CCN(C(=O)CC1CCCC1(F)F)CC2 40300,C1(NC(=O)C(CC(F)F)N2CCOCC2)CCN(C(=O)C(Cl)=CCl)CCC1(F)F 40301,Cc1csc2ncnc(NC(C)CC(C)NC(c3ccc4nccn4c3)=O)c12 40302,c1(C(N2CCC(CNC(CC)=O)c3c2cccc3)=O)ccc2c(c1)C(=O)NC2=O 40303,c1(CC)nc(N2CCCC(NC(c3sc(SC)cc3C)=O)C2)c(CC)c(Cl)n1 40304,O=C1Cc2cc(NC(C34CC(C(=O)Nc5scc(Br)c5Br)(C3)C4)=O)cnc2N1 40305,c1(N2CCCC(NC(c3c(C)nn[nH]3)=O)CC2)cc2ncnn2cn1 40306,c1(C(=O)NCC2(OCC)CN(C(C(C=C)CC)=O)C2)ccc2c(c1)OCC2 40307,Cc1no[nH]c1=NC(=O)C1(C)CCN(C(=O)CCc2ccccc2)CC1 40308,c1(C(=O)NCCC2CC(NC(=O)C(F)F)C2)ccc2c(Br)cnn2c1 40309,N1(C(C(C=C)OC)=O)CC(CC(=O)NCC(C)(O)CCC)C2(CC2)C1 40310,CN1CCN(C(=O)CC2CCN2C(C2CC3CC3C2)=O)CC(O)C1 40311,C1(C(=O)NC2CN(C(c3ccc(CCC(C)O)cc3)=O)C2)CCC(N=[N+]=[N-])CC1 40312,c1(OCCCC(=O)NCCC2CC(NC(CC=CC=C)=O)C2)ccc(F)c(F)c1 40313,c1(CC(C)C(=O)Nc2nc(-c3ccc(Cl)s3)cs2)ccc(F)c(F)c1 40314,CCCCC(COC)NC(=O)CCN(C(=O)CC(OC)OC)CC1CC1 40315,N1(C(CC2(CC(=O)OC)CC2)=O)CCN(C(c2cn(C)nn2)=O)CC(CO)C1 40316,CC1CCC(Cl)=C(C(=O)NC2C=CCN(C(=O)C(C)(C)N(C)C)C2)C1 40317,c1(OC(C(=O)NCC(CNC(C(C)(C)OC(C)C)=O)C)C)ccc(Cl)cc1 40318,C1(CCC)CN(C(c2cc(Cl)ccc2F)=O)CCN1C(=O)CC(O)C1CCCC1 40319,Cc1[nH]c2ccccc2c1C(=O)NC1(CF)CCN(c2nccc(C(C)C)n2)C1 40320,C=CC1CN(C(=O)C(CN(C)C)NC(=O)CCSCC)CCO1 40321,c1(C(N2C(C)CC(NC(C3CCC(=O)NC3)=O)C2)=O)cc(F)cnc1Cl 40322,C(=O)(CCCCC(C)CC)N1C(CC)CN(C(c2nn(CC)cc2Br)=O)CC1 40323,C1(CNC(c2cn(C)nc2C(C)(C)C)=O)CC2COCC2N1C(=O)C(C)(C)CO 40324,C(=O)(N=c1nn[nH]n1CCC(C)C)NC(c1ccc(Cl)cc1)CCC 40325,C(=O)(C(C)(C)C(=O)NC1CCC(NC(c2ncc[nH]c2=O)=O)CC1)OC 40326,C12(COC)COC(C(N3CCCC(C(C)NC(=O)C(Br)=C(C)C)C3)=O)(C1)C2 40327,c1(CC)cc(NCC(C2CC2)N(C)C(C2CCC(C(C)C)CC2)=O)ncn1 40328,C(C(=O)NC(C1CCN(C(C2CCCC(C)(C)C2)=O)C1)(C)C)(C(C)(C)C)SC 40329,c1(C(=O)OCc2cn(CC3CC(OC(C4C(C)C4C)=O)C3)nc2)csc(Cl)c1Cl 40330,c1(C(N2CCC(OC)C2)=O)ccc(Br)c(CCC(=O)N2CCCC2)c1F 40331,c12cn(C)nc1NC2=O.c1(CCSCC)cn(CCCC(=O)O)nn1 40332,c1(C(N(CC(CNC(Cc2c(C)noc2)=O)O)C)=O)cncc(-n2cccn2)n1 40333,N1(C(c2nccc(OC)c2F)=O)CCC2CCCN(C(c3cnc(O)o3)=O)C2C1 40334,C1(C2CCN(C(COCC(c3ccncc3)C)=O)C2)CCCCN1C(=O)C(N)=O 40335,C(CCCCCCC(=O)NC(CNC(=O)CC(C)C(C)C)C1CC1)SC 40336,c1(SC)nccnc1C(=O)NCCCOC1CCN(C(=O)C(F)F)CC1 40337,CC(O)(CCNC(N1CC2(CCC2)C1CO)=O)C(F)(F)F 40338,c1(C(N2CCCC(CN(C(=O)C#CC3CC3)C)C2)=O)ccc(N)c(N)c1 40339,N1(C(CCOC(C)=O)=O)CC(C2CC2C(=O)N(C2CCOCC2C)C)C1 40340,N1(C(C(C)=O)=O)CCN(C(c2cnc(CC(C)C)s2)=O)CC1C 40341,C1(NC(CC=CC)=O)CC2CN(C(=O)CCCCC(C)(C)C)CCN2C1=O 40342,CC1=C(C(=O)NC2CCC(NC(c3cn(C)nc3Cl)=O)C2)C=C2CCCN=C2N1 40343,CCCCCCOC(C)C(=O)NCC(CC)NC(c1ccnn1C1CCCC1)=O 40344,C1(C)(C(=O)NCC2CCN(C(COCC)=O)C2)CNC(=O)C1 40345,N1(C(C2(OC)CC2)=O)CCC(O)(CNC(=O)CC2CCN(C)C2=O)CC1 40346,N1(C(C2(CC=C)CCN(C(=O)C=CCN3CCC3)C2)=O)CCCCC(OC)C1 40347,C1(C2CCN(C(C3CC4CC3C4)=O)CC2)(NC(CCC(CCCC)C)=O)CCC1 40348,C(c1ccc(C2CC2C)o1)=CC(=O)N(C(=O)C(C)=C1CCC1)CC 40349,C1(C(=O)OC)CC=CCN1C(C1CC2CCCC12)C(=O)NC(C)C 40350,C1(CNC(C(CC#C)C2CC2)=O)(NC(c2nccnc2C)=O)CC2CCC1CC2 40351,C1(C2(NC(=O)CSc3cscn3)CC2)CCCCN1C(C1CC12CCC2)=O 40352,n1(CCC)cccc1C(=O)NCC1C(CNC(C2(N(C)C)CC2)=O)C1(F)F 40353,C(C(C)C(=O)NC1CC1NC(c1cc(C2(C)COC2)no1)=O)OCC 40354,N1(C(C=CC(=O)OC)=O)CC(CO)C1(C)C.c12cc[nH]c1C(=O)NC2 40355,C1(C#N)(C(N(CCCNC(=O)C=CCCC(C)C)CC)=O)CC2CC2C1 40356,Cc1[nH][nH]c(=N)c1C(=O)NCCCCCCN(C)C(c1coc(C(F)(F)F)c1)=O 40357,C1(CC(=O)N(CC)CC2CCCN2C(C2CC=CC2)=O)CCC(C)(C)O1 40358,CC1CN(C(=O)CN(C(=O)C2=CCOCC2)C)CCC1N(C)C 40359,C=CCCCC(C(=O)Nc1cccc(NC=O)c1)NC(=O)CCC(=O)CC 40360,n1(CC(=O)NC2C(NC(C(F)=CCC)=O)CC2)cc(Cl)c(C)n1 40361,N1(C(c2ccc(C)c(F)c2)=O)CCN(C(c2cncc(F)c2F)=O)CC2(CC2)C1 40362,C(c1cnn(C)c1)=CC(=O)NC(CC=CC(=O)N(C1C(C)CCC1)C)(C)C 40363,C1(NC(CC#CCN(C(C)C2CC2)C(=O)OC(C)(C)C)=O)CC1 40364,C1(C(N(C(CC)C)CCO)=O)COCCN(C(C2(C#N)CC2)=O)C1 40365,C(CCCCC(=O)NC1CC2(C1)CC(NC(C1SCC=C1C)=O)C2)SC 40366,N1(C(CNS(CC)(=O)=O)=O)CCCC(C)C1CCNC(c1cc(Cl)c[nH]1)=O 40367,C#CC1(C(=O)N(CCC(N2CC(O)(c3cc[nH]n3)C2)=O)CCO)CC(=O)C1 40368,CCCC(C(=O)NCC1C2CN(C(c3cnn(C(C)C)c3F)=O)CC12)OC 40369,N1(C(C=C(C)C2CC2)=O)CC(C(=O)NCC(n2ccnn2)C)C(C)(C)C1 40370,C(=O)(CCCCC#N)NC1CCCN(C(C(CC#C)O)=O)C1 40371,N1(C(C2(CC=C)CC=CC2)=O)CC2(CCC2NC(=O)CSS(C)(=O)=O)C1 40372,C1(CC(=O)NCCC(C)OC)CN(C(=O)CC2CC(C)=NO2)CC1C 40373,C1(CNC(C(N2C(=O)CCC2=O)CC)=O)CC(C)(C)CN1C(=O)CCOC1CC1 40374,C1(NC(Cc2c(SCC)cccc2)=O)CC(C)CN(C(c2n[nH]cc2OC)=O)C1 40375,C(CCCC(=O)NCC(c1ccco1)O)NC(c1cc(OC)n[nH]1)=O 40376,CN=c1cc(C(=O)NC(C2CCCC2)CNC(=O)COC(C)C)cc[nH]1 40377,Cc1nc(C(C)C)ccc1C(=O)NCC1CCCC(NC(=O)CNS(N)(=O)=O)C1 40378,N1(C(COCCCC)=O)CCC(C)(C)C(NC(=O)CCN(CC(F)(F)F)C)C1 40379,C1(OC)COC2(COC2)C1.n12cc(nn1)CCC1CN(C1)C(=O)C2 40380,C1(CNC(c2ncn(C(C)C)c2)=O)CC(C)N(C(C2CCC(=O)N2C)=O)C1 40381,Cc1ccccc1C(=O)NC(C)CCNC(=O)CCCc1cncs1 40382,C(C(C)(C)C(C)NCCCN)OC.C1(OC(N)=O)(C)CC(C(C2(C(=O)OC)CC2)=O)C1 40383,c1(N2CCN(CC(C)(F)F)CC2)nc(N2CCC(CCF)CC2)nc2scnc12 40384,c1(OC)ccc2cc(-c3ccc(C(N4CCC5(CCOC5)C4)=O)s3)c(O)nc2c1 40385,C1(NC(c2cc(=N)[nH]cc2)=O)CCC2CCN(C(c3csc(C(N)=O)n3)=O)C12 40386,c1(OCCC)cccnc1NC(N1CCC(CC)(CC)C1)=O 40387,N1(C(C2CN(C)C(=O)C2)=O)CCC(C)(C)C1CC(=O)NCCc1cnn[nH]1 40388,C1(C2CCOCC2)(C(N2CC(N(C(C(C(=O)OCC)C3CC3)=O)C)C2)=O)CC1 40389,c1(C(=O)NC(c2ccccc2)C(C)NC(C2CCNC2=O)=O)cc(Cl)ncc1N 40390,C1(NC(=O)Cc2cccnc2O)C2CC3CN(C(C4CCCS4)=O)C1C3C2 40391,N1(C(=O)OC(C)(C)C)CCC2(CNC(c3ncn4c3COCC4)=O)C(F)(F)C12 40392,C1(NS(C)(=O)=O)CCN(C(C2CC(F)CN2CCCC(=O)O)=O)CC1 40393,c1(C(=O)NC(CCOC)CNC(=O)CC(C)CF)ccc(S(N)(=O)=O)c(F)c1 40394,C(=O)(C1SCCc2ccccc21)NCCN(C(CC(CC(C)C)O)=O)CCOC 40395,N1(C(c2cccc(C)c2C)=O)CC(NC(c2cnc(C)c(N)c2)=O)CC(F)(F)C1 40396,C12(C(=O)NCC(CC)(CC)NC(=O)Cc3csc(S)n3)CCCC1CC(=O)C2 40397,CC1(C)CCC(CNC(=O)C(C2CCCCC2)F)N(C(=O)CN2CCSCC2)C1 40398,c1(C(=O)NC2C(C)CN(C(c3ccoc3)=O)C2)cccc(C(N)=O)c1N 40399,N1(C(C(CC)CCOC)=O)CC2CCN(C(=O)CC3CC3C3CC3)CC12 40400,N1(C(C(CNC(c2c(C)[nH]cc2)=O)CC2CC2)=O)CCC(CO)C12CC2 40401,C1(C(N2C(C(C)(C)NC(c3scc(OC)c3)=O)CCC2)=O)(OC)CS(=O)(=O)C1 40402,C1(C(=O)NCC2CCC(CNC(CNC(C)=O)=O)CC2)CCCCC1(F)F 40403,c1(CN(c2snc(C(=O)OC)n2)C)cc(C#N)ccc1F.C12CCN(C1)C2=O 40404,C1(C(=O)NCCC(C)(C)O)C2CCN(C(c3ccccc3C#N)=O)CC12 40405,CCC(C)(CCC(C)C)C(=O)NC1CC(CC(N2CCC(O)C(O)C2)=O)C1 40406,c1(-c2cc(C)cc(Br)c2)csc(=Nc2ccc(C)c(F)c2)n1CCC1CCSC1 40407,C(c1cccc(Cl)c1)=C(C(=O)NC1(COC)CN(C(=O)COC2CCC2)C1)C 40408,C=CC1CN(C(c2cnn(C3CC3)c2)=O)CC1NC(C1(C)CCCS1(=O)=O)=O 40409,C=CCC(CC(=O)N(CCC(F)(F)F)CC)NC(=O)C(COC)CC 40410,c1(NC2(c3nnnn3C(C)(C)C)CC(C(=O)OC)C2)nc2cc(Cl)cnc2[nH]1 40411,C(=O)(C(C)(C)C1=CCN(C(C2CCCC2C)=O)C1)NC1CC(CC)C1 40412,N1(C(COC2CC(C(C)C)OCC2)=O)CC(C2(NC(=O)Cc3cccs3)CC2)C1 40413,c1(OC)ncc(C(=O)NCC2(O)CCN(C(c3n[nH]cc3C)=O)C2)c(C)n1 40414,c1(N2CCC3(C(C(=O)Nc4cccnc4O)C3)C2)ncc2ccsc2n1 40415,C12(C(N(CC(C3CCCC3)O)C)=O)COCC1CN(C(=O)CCc1cscn1)C2 40416,C(=O)(CC(C)CC(C)C)N1CCC(CC(=O)N(CCC(CCC)O)CC)CC1 40417,c1(C(=O)NC2CC(N(C(=O)CNC(N)=O)C)C2)c(F)ccc2[nH]ccc12 40418,c1(CNC(c2n(CC)ccc2)=O)ccc(F)c(CC(=O)OC)c1 40419,CC1CN(c2nnnn2CCC2CSc3ccccc3O2)CCS(=O)(=O)C1 40420,Cc1cn2cc(CC(=O)NCC(C)CNC(=O)CC(C)CF)nc2s1 40421,c1(C(=O)NC(CC(C)NC(CCC(=O)NCCC)=O)C)nccc(Cl)c1Cl 40422,n1(CC(C)NC(C(C)OCCC(C)C)=O)cc(CNC(=O)C(F)(F)F)nn1 40423,C1(NC(CCc2c(C)noc2)=O)CC=C(C(=O)N2CCC(CCO)C2)C1 40424,c1(C(=O)NC2C(CNC(=O)COc3ccsc3)C2)ccc(C2CC2)s1 40425,CC1=C(C(=O)N2CCC(O)(C(C)NC(=O)C(C)NC=O)C2)CCO1 40426,Cc1ccc([N+](=O)[O-])cc1C(N1CCC(F)(F)C(NCc2cnn(C)c2C)C1)=O 40427,N1(C(C(C)=NOCC#N)=O)CCC2(C=C(C(=O)N(C3CCOC(C)C3)C)C2)C1 40428,C1(C(=O)NCC2CCCC(CC)C2)C2CCC(C2)C1NC(C1(Cl)CCC1)=O 40429,c1(CC)sc(C(=O)NCCC2CN(C(c3cc(CC(C)C)[nH]n3)=O)C2)cc1C 40430,C(CCCC(=O)N1CC(C(=O)NC2CCS(=O)(=O)C2)OC(C)C1)(OC)OC 40431,CCCCC(CC)C(=O)N1CC(C(=O)NCCN2CCC2)CC1(C)C 40432,C1(C(=O)NCC(CNC(c2ccn(CCCC)n2)=O)(C)C)C2CCC(=O)C12 40433,c1(C(=O)NCC2N(C(CCCC#CC)=O)CC(OC)C2)cnc2[nH]nnc2c1 40434,C(=O)(C1CCCn2ccnc21)NC1CCN(C(COC)=O)CCC1(F)F 40435,c1(N2CCCCC(SC)C2)ccc(Br)c(S(=O)(=O)NC(C)Cc2ccc(C)o2)n1 40436,CC1(NC(=O)Cc2ccc(F)cn2)CCN(C(=O)C=CBr)C1 40437,Cc1occc1C(=O)NC(C1CCCN1C(c1cc(CCO)on1)=O)(C)C 40438,C#Cc1cncc(C(=O)NCC(CNC(=O)Cc2ccc(Br)cc2)OC)c1 40439,c12[nH]c(C)c(c1C)CNC2.C1(SC)CN(C(C2CC2C(=O)O)=O)C1 40440,C(=O)(C(Cc1ccco1)NC(C1CNC(=O)N1)=O)N(CCCC)CCO 40441,c1(C(=O)NC2CC=CCC2C(=O)NCc2ccccc2F)cnc(O)c(F)c1 40442,C1(C(=O)NCC(CNC(Cc2c(C)ncnc2C)=O)C)OCC2CCCCC12 40443,CCC(CC(=O)NC1CCC(C)(NC(c2cnn(C)c(=O)c2)=O)CC1)CC(C)C 40444,c1(C2(C(=O)NCCC3CCN(C(c4c(C)cco4)=O)C3)CC2)ccc(F)c(Cl)c1 40445,CCCCC(CC)C(=O)NC1CC(CO)N(C(=O)C=CCN2CCCC2)C1 40446,C(=O)(C1=CC2(CN(C(=O)C(O)CN3CCCC3)C2)OC1)NCC(COC)(C)CO 40447,c1(C(N2CC(C)NC(=O)C2)=O)ccc2c(n1)CCN(C(c1cccc(Br)c1)=O)C2 40448,CCCCCC(C(=O)NC1CCC(NC(=O)Cc2cn(C)nc2Cl)CC1)C(C)C 40449,c1(C(=O)NCC(CNC(C(COCC)C)=O)C)oc2ccccc2c1CC 40450,c1(CNC(C2(NC(CCC=CC(C)C)=O)CCC2)=O)ccc(F)c(F)c1 40451,C1(C(N(C2CCN(C(=O)C(C)O)CC2)CCC)=O)C2CCC1(c1ccccc1)C2 40452,N1(C(CC2CC(OC)C2)=O)CCCC1(C)CNC(=O)CC1CCC=CCC1 40453,C1(CC(=O)NCC2CCC(NC(c3n(C)cnc3)=O)CC2)CCCCC1(C)C 40454,C(C(F)(F)C(N)=O)NC(C1(CC=C)CN(C(C2COCCO2)=O)C1)=O 40455,Nc1cc2c(cc1C(=O)NC1CCC(NC(C3CC3(Cl)Cl)=O)CC1)CCC2 40456,C(=O)(CCCC(F)(F)CO)N1CC(C(C)NC(C23CCC(CC2)CC3)=O)C1 40457,C1(F)(CNC(C(SC)SC)=O)CCN(C(=O)C(=Cc2cn(C)cn2)F)CC1 40458,c1(C(=O)NC(Cc2c[nH]c(=NC)s2)C(=O)O)ccc(OC)cc1S(C)(=O)=O 40459,Cc1nc(C=CC(=O)N(C2CCCN(C(C3CC3CF)=O)C2)C)cs1 40460,c1(SC)ccc(NC(=O)NCCOc2cccc(F)n2)cc1C#N 40461,N1(C(C(C)N2CCCC2)=O)CCC(CCC(=O)N(C)Cc2nncs2)C1 40462,c1(C(=O)NCC2(NC(COC(CC)(C)C)=O)CCC2)ccc(Cl)c(Cl)c1 40463,c1(C(N2CC(C(=O)Nc3ccc(O)nc3)SCC2)=O)cn2ccc(Cl)cc2n1 40464,c1(OC)cc([N+](=O)[O-])c(NC(C2CCCCN2C(=O)C(C)S)=O)cc1F 40465,C1(O)(CNC(C2(C#C)CN(C(=O)CC3CCCN(C)C3)C2)=O)CC2CCC1O2 40466,N1(C(Cc2ccc(CC)s2)=O)CCCN(C(c2cc(C)ncn2)=O)CC1C(C)C 40467,C(=O)(CCCCc1ccc(Cl)cc1)NCC(CN(C(Cc1cc(C)sc1)=O)C)O 40468,C(C)(C)(CCCCC(=O)N(CC(C)CNC(=O)C1=CCC1)C)OC 40469,C1(C(=O)NCC(C(C)C)NC(=O)C2CC2)CCN(C(C2CC2F)=O)CC1 40470,Cc1cc(N2Cc3ncsc3C2)nc(=NCCCc2ncc[nH]2)[nH]1 40471,N1(C(c2c(C)nco2)=O)CCC2(CC(NC(=O)C(C)(C)c3ccn(C)n3)CO2)C1 40472,c1(C(=O)NC(C)CN(C(=O)CC(=O)OC(C)(C)C)C)nnc(S)n1C 40473,C#CCCCCC(=O)N1CCCC(C)(NC(=O)C(CCC)OCC)C1 40474,C1(C(N2C(C#C)CCCC2)=O)CN(C(=O)Cc2nccn2C)CCC1(C)C 40475,N1(C(c2cc(OC)no2)=O)CC2CC(NC(=O)CC3CC(=O)NC3=O)CC1C2 40476,c1(CC)cc(NC(=O)CC2CCCN(C(C3CCCSC3C)=O)CC2)cc(O)c1 40477,Cc1cc(F)c(C(N2CCC(C)(CCNC(=O)C(C)n3cncn3)C2)=O)c(F)c1 40478,Cc1cc(C(C)NC(c2ccc(CC3(C)CCCCC3)cc2)=O)cnc1C 40479,CC1CN(C(c2ccncc2F)=O)CC1CC(=O)NCCCCC1CC1 40480,CC1CC(C(=O)N(CCNC(c2ccsc2)=O)CCc2ccccc2)CC(C)C1 40481,N1(C(c2c(C)nsc2C)=O)CCC(C2(O)CCN(C(=O)C#CC3CC3)C2)CC1 40482,C1(NC(C(C)OC)=O)CCC(NC(c2cnn(C)c2C)=O)CC1 40483,c1(C(C(=O)NCCOC)N(C)Cc2cnn(C3CCCCC3)c2)cccc(Cl)c1C 40484,N(C)(S(=O)(=O)N(C)C)CC(=O)NCCCN(C(c1c(NC(C)=O)cncc1)=O)C 40485,C1(NCC)CCC(C)(C(C2(CC)CN(C(=O)N(C)C)C2)c2nnnn2C(C)C)C1 40486,C=C(C)CC(C(=O)N(C(C)C(=O)N(CCCCOC)C)C)OC 40487,C1(C#N)(C(=O)NCC(c2n(C)ccn2)=O)C(C#N)C1(C)C 40488,N1(C(C(CCF)NC(C(C=C=C)C)=O)=O)CCOC(C)(C)C1 40489,c1(OC(C(=O)N(CC(CNC(C2N(C(C)=O)CSC2)=O)O)C)C)ccc(C)cc1 40490,N1(C(c2c(CC)n(CC)nc2)=O)CCCN(C(=O)CC2(OC)CC2)C(C)C1 40491,c1(C(=O)NC2C(NC(C3(COC)CCCC3)=O)C2)cc(F)c(N)c(F)c1 40492,c1(OC)cc(NC(c2cccc(N3CCNC(=O)C3)c2)=O)ccc1O 40493,N1(C(C(CC)OCC)=O)CCCC12CCN(C(c1ccc(C)cc1)=O)C2 40494,c1(CC(=O)NCC2N(C(C(C(C)C)OC)=O)CCCC2)cc(F)ccc1Cl 40495,c1(C(=O)NCC(CC)NC(=O)C(C)(C)C(N)=O)ccc([N+](=O)[O-])cc1 40496,N1(C(C2C(C)(C)C2C(F)F)=O)CC(CNC(c2cc[nH]c(=N)c2Cl)=O)CC1(C)C 40497,Cc1nc(C(=O)NC2(CN(C)C(C3(C)CC=CCO3)=O)CC2)ccc1C#N 40498,Cc1occ(C(F)(F)F)c1C(=O)NC1C=CCN(C(=O)C2=COCC2)C1 40499,CCCC(C(=O)N1CCC1Cn1cc(-c2cn(CCO)nn2)cn1)OC 40500,C1(NC(C=NOC)=O)CCOC(C(=O)NCc2csc(C)c2C)C1 40501,C(=O)(C=CCNC(=O)CNC(C)=O)N(CC=C)CCO 40502,N1(CC2(O)CCN(Cc3c(OC)cccn3)CC2)CCC2(CCCC2)C1 40503,C1(C)CCN(C(=O)C=C(C)Cl)CC1.C1(C(C)N)CCC(c2nn[nH]n2)O1.C12CC(C1)CC(=O)C2=O 40504,c1(CC(=O)NC(CC)CNC(C23CCC2C3)=O)nnn(-c2cccc(Cl)c2)c1C 40505,C1(C(N(C2CN(C(CC3CCCN(C)C3)=O)C2)C)=O)CNC(=O)CC1(C)C 40506,N1(C(c2c(C)cns2)=O)CCOCCC1C(=O)NCCc1cncs1 40507,C1(C2CCN(C(=O)C=Cc3ccccc3)CC2)(NC(c2c(C)cnnc2)=O)CC1 40508,C(=O)(C(C)(C)CC(C)C)NCC1(O)CCCN(C(c2cccc(C)n2)=O)C1 40509,c1(C(=O)NC(C(C(C)C)C)CNC(c2cccnc2S)=O)noc2c1CCCC2 40510,CC1(C)CCC(C(N2CC=CC2CNC(c2ccon2)=O)=O)C1 40511,N1(C(=O)C=Cc2cccs2)CCC(C2CCN(C(C3(F)CCCCC3)=O)CC2)C1 40512,C1(NC(c2cc(CCC)on2)=O)CCCN(C(=O)C=C(C)Cl)C1C 40513,C1(O)(C(=O)NCCC(C)N(C(CC2CC(OC)C2)=O)C)CCC(C)(C)CC1 40514,c1(C(N2CC(CNC(CCC3CC(C)C3)=O)OCC2)=O)ccc(F)c(Cl)c1N 40515,Cc1c(Br)csc1C(N1CC(CC(C)NC(=O)C(C)C2CCC2)C1)=O 40516,C(C(=O)N1CC(O)C(O)CO1)C1C(C)(C)CCN(C(C(CO)N(C)C)=O)C1 40517,C1(C=O)CCC(C)(O)CC1.C1(OC)CN2CC1NC(=O)CC1CCN2C1.C(C)=O 40518,C1(CNC(C2CCCC(NC(CC(C)F)=O)C2)=O)CC12CCOCC2 40519,C1(C)(C(N(CC(CC)NC(=O)CCOCC(F)F)C)=O)CCC(=O)N1 40520,C(=O)(C(C)CC(C)(C)C)N1CCCC(N(C(c2cnn3ccn(C)c23)=O)CC)C1 40521,c1(NC2C(C(C)NC(C3CC(Cl)(Cl)C3)=O)C2)ncc(S(=O)(=O)N(C)C)cc1Cl 40522,CCCCCCC(C)C(=O)N1CCCC1CN.C1(NC(C)C)CCCCN1N=O 40523,N1(CC(N2CC(NC(=O)CSc3ccncc3)C2)=O)CCCCCCC1=O 40524,C(=O)(C1=CCOCC1)NC1(CO)CN(C(c2c(C(C)C)n(C)nc2)=O)C1 40525,Cc1cc(NC(=O)C(=O)NCCc2ccc(Br)s2)ncn1 40526,C(c1ccncn1)=CC(=O)NC(CNC(C1(CC=C)CCC1)=O)(C)C1CC1 40527,Cc1cccc([N+](=O)[O-])c1C(N1CC(N(C(=O)CC2OCCC2C)C)C1)=O 40528,c1(C(=O)NCC(CNC(C2CCN(C)C2)=O)(C)O)c[nH]c2cccc(Cl)c12 40529,C(=O)(CS(=O)C(F)(F)F)NC1C(CO)CCN(C(CCCOC(C)=O)=O)C1 40530,CC1CCc2ncc(C(N3CCC(NC(c4cnc(C(C)(F)F)s4)=O)C3)=O)n2C1 40531,N1(C(C2(CC(=O)OC)CCC2)=O)CCCN(C(C2(CN(C)C)CC2)=O)CC1CO 40532,N1(C(C2CC(N(C)C)C2)=O)CCC(C)(CNC(C2CC3C=CC2C3)=O)CC1 40533,N1(C(c2oc(C)c(CO)c2)=O)CCN(C(C2CCC(=O)N2C)=O)CC1CF 40534,N1(C(COCC(=O)OC)=O)CCCC1CN(C(c1coc(C2CCC2)n1)=O)C1CC1 40535,N1(C(c2c(N)nccc2)=O)CCC=C(CNC(=O)CCN2CCCC2)C1 40536,CCCCC(C)C(=O)N1CC(C(=O)N(CC)CC2CCOC2)C(F)C1 40537,c1(C(N2CC(C#N)OCC2)=O)cc(-c2cccc(OC(F)F)c2)c2[nH]ccc2c1 40538,C[S+](C)CCC(O)C(=O)N1CC2CC1C2NC(c1cc([N+](=O)[O-])n[nH]1)=O 40539,c1(C(=O)NCC2CN(C(C=CCOC)=O)C(C)C2)cc(C(C)C)nc(O)c1 40540,c1(CN(C(=O)C(CC2CCC(F)(F)CC2)CN)C)ccc2c(c1F)CCC2 40541,c1(C(=O)NCC(CNC(C(CC)(C)OC)=O)CO)ccnc2ncccc12 40542,c1(C(N(C(CCNC(C(C(=C)C)(C)O)=O)C)C)=O)ccc2c(C)nn(C)c2n1 40543,N1(C(c2c(CC)ncs2)=O)CC2CN(C(c3cnc(C(C)(C)C)o3)=O)CC(C1)O2 40544,c1(N2CC3OCCN(CCN(CC)CC)C3C2)cc(C)c(S(=O)(=O)NCC)cn1 40545,C12(NC(=O)Cc3ccccc3Cl)CCN(C(=O)CCN3CCC(O)CC3)CC1C2 40546,Cc1ccc(CC(=O)NCCC(C)(C)NC(c2ccnc(CC(C)C)n2)=O)cn1 40547,c1(OCC)cncc(C(=O)NC(C2CN(C(=O)Cn3[nH]cnc3=N)CCO2)C)c1 40548,N1(C(Cc2c(C)occ2)=O)C(C)C2CC1C2NC(c1cccnc1O)=O 40549,N1(C(COCC#C)=O)CCC(NC(=O)CCc2cccs2)C1C1CC1 40550,c1(OC)cc(N)ccc1C(=O)NCCN1CCC(NC(=O)C=CCO)CC1 40551,C1(C(=O)NC(CC)CC(F)(F)F)(NC(CCC#CC)=O)CCC(C)(C)C1 40552,C(N=c1ccc(-c2ccc(F)cc2F)n[nH]1)c1ccc(C)cc1 40553,c1(C(=O)OCC2(NC(C)(C)C)CCN(CC3C(C)C3)C2)cccc2c1CCCC2 40554,c1(NC(C2N(Cc3ccn(CC)n3)CC(O)C2)=O)cc(F)c(C)c(F)c1 40555,c1(C(N2CCC(NC(c3cc(C#N)sc3)=O)CC2)=O)cc(S(N)(=O)=O)ccn1 40556,N#Cc1cc(C(=O)NCC2CC2NC(c2c(Cl)ccc(F)c2F)=O)c(N)nc1O 40557,C1(NC(=O)CC=C(Cl)Cl)CCC2CN(C(c3cnn4cccnc34)=O)CCC2C1 40558,c1(NC(c2cc(-c3ccc(C)o3)[nH]n2)=O)nccnc1C(=O)Nc1ccccc1 40559,CC1CCCCC1(CNC(c1ccc(O)c(O)c1)=O)NC(c1c[nH]ccc1=O)=O 40560,CC1CN(C(=O)C(c2ccc(Cl)cc2)O)CCN1C(=O)CC1(n2cnnc2O)CC1 40561,C1(CNC(c2scc(C)c2)=O)CC(NC(C2CN(C(N)=O)C2)=O)C12CCC2 40562,C(=O)(C(O)CCNC(C1COCC(C)O1)=O)NC(c1nnc(C)s1)C 40563,C1(CNC(c2c(CC)cncc2)=O)N(C(=O)CCNS(C)(=O)=O)CCCC1(C)C 40564,C(=O)(CCCNC)N.C(=O)(C(C)CC1CC1)N(CC(=O)OC)CC(F)F 40565,c1(CC)nc(C)[nH]c1C(=O)NCC1C2CC1N(C(=O)CCC(=O)NC)C2 40566,CC1(CNC(C2CC2F)=O)CCCN(C(=O)Cc2c(Cl)cccc2Cl)C1 40567,c1(CC(=O)NCC2(CNC(=O)CC3OCCO3)CC2)ccc(Cl)s1 40568,C1(C(C)C)N(C(c2cncn2C)=O)CC12CCN(C(C1CC1F)=O)CC2 40569,N1(C(C2(n3cc(-c4ccc(C)cc4C)nn3)CC2)=O)CCCCNC(C)C1 40570,CC(C)(C)C(CC(=O)NCC1CCN(C(=O)CN2CSCCSC2)C1)C(F)F 40571,c1(C(N2CC(NC(=O)CN3CCOCC3)(CF)C2)=O)ccc(CC2CCC2)cc1 40572,CN1CCOCC1C(=O)NCC1(C(N2CC=CC2CF)=O)CC1 40573,Cc1c(C(=O)NC(C)CNC(=O)CCc2ccon2)ccn1C 40574,c1(-c2nc(CC(C)OC)nn2-c2ccnnc2)cc(S(=O)(=O)N(C)C)cn1C 40575,C(=O)(C1=NOC2(CCN(C(=O)Cc3cccs3)C2)C1)NCc1cccc(C#N)n1 40576,N1(C(COCCOC)=O)CCC2(CCCCN(C(c3coc(COC)n3)=O)C2)C1 40577,C12(C(=O)Nc3cccc(NC(COCCC=C)=O)c3)CCCC(C1)C(=O)NC2 40578,Cc1cc(C(N2CC(C)C2C(N2CCCC2C2CCOC2)=O)=O)no1 40579,c1(N2CC(NC(C3CCC4CC34)=O)(CO)C2)ncncc1Br 40580,N1(C(C2C(C)(C)CC2)=O)CCCCC1C1CCN(C(c2cc(Br)no2)=O)CC1 40581,N1(C(C2OCCN(CC)C2)=O)CCCC(CCNC(c2ccnn2CC)=O)CC1 40582,N1(C(C(C2CCN(C(c3ccnn3C3CC3)=O)C2)C)=O)CCC(O)C(C)C1 40583,C1(C(N2CCC(C(=O)OC)C2(C)C)=O)CC2C=CC1N(C(=O)C(C)n1ccnn1)C2 40584,Cc1sc(C)c(C(N2CC3(CC(NC(=O)C(C)CC(N)=O)CO3)C2)=O)c1C#N 40585,C1(C(=O)OCC)CCC(C)(C(=O)NCCN(C(=O)Cn2nccn2)C)C1 40586,CC(c1ccccc1)=CC(=O)NC1(C(=O)NC(N)=O)CC1.C12CCC1C2 40587,N1(C(C(C)CC(F)(F)F)=O)CCCC2(NC(=O)CN3CCC3)CCCC12 40588,C1(CC(=O)NCC(C(C)C)(C)C)C2CCC(C2)N1C(=O)CCCn1cncn1 40589,c1(C(N2CCCC(CN(C(c3n(CC)ccc3)=O)C)C2)=O)c(OC)ccnc1F 40590,N1(C(C2C(C)CC2)=O)CCN(C)CC1CNC(=O)CCc1ncc[nH]1 40591,c1(-c2scc(COC(C3CC(O)(C(F)(F)F)C3)=O)n2)ccc(O)cc1 40592,N1(C(C=C(C)Cl)=O)CCC2(NC(=O)COc3cccc(C)c3)CCCC12 40593,Cc1ccsc1C(=O)N(CCC(=O)NC(C)(C)CO)C 40594,C(=O)(CCCS(=O)(=O)N1CCCC1)NC(CNC(COCCC#C)=O)C 40595,c1(OC)cccc(Cl)c1CC(=O)NC1CCN(C(C2CCNC2=O)=O)C(C)C1 40596,c1(CC(=O)NCC(CNC(CNC(=O)OCC)=O)F)ccnc(O)c1 40597,N1(C(CC(C)C)=O)CC2CCCC1CN(C(=O)Cc1ccc3nc(O)[nH]c3c1)C2 40598,C(=O)(CCCC(C)(C)C)N(C(CC(C)C)C(N)=O)C.c12coc(n1)C(=O)N2 40599,N1(C(C(C)S(N)(=O)=O)=O)CCC2(CCCC2NC(c2cc(Cl)cn2C)=O)CC1 40600,C(CCCC(=O)NCC1(O)CN(C(c2cn(C(C)(C)C)nc2C)=O)C1)NC(C)=O 40601,N1(C(c2cn(CC=C)nc2)=O)CCC(C(=O)Nc2cnc(OC)nc2)=C(F)C1 40602,O=C(C1=CC2CCCC12)NCC1CC(NC(c2ncnc(O)c2Br)=O)C1 40603,CCC(C)C(O)C(=O)NCC(CO)NC(c1ccc(F)c(C(F)(F)F)c1)=O 40604,CCC(C(=O)NCCCNC(=O)CC12CCC(CC1)C2)C(C)(C)CC 40605,C#CC1(C(=O)OCC)CCN(C(=O)C(N2CCOC(C)CC2)C)CC1 40606,c1(C(C2CC(C(c3nnnn3C3CC3)N)C2)OC)ccc(F)c(Cl)c1.c1(C)cn[nH]c1 40607,c1(C(=O)NC(C)CC2CN(C(c3ccco3)=O)C2)cnc(F)c(F)c1 40608,Cc1[nH][nH]c(=N)c1C(=O)N(C)CC1(O)CCN(C(=O)CCC2CNC(=O)N2)C1 40609,C1(NC(N(C(CNC(C(CC)C)=O)C)CC)=O)CCN(C(=O)NC)CC1(C)C 40610,c12ncnc3c1ncn3C(CC(C)C)N2CCOC.c1cn(-c2nccs2)nn1.OC 40611,c1(C(N(C2CCCN(C(CC(C)F)=O)C2)C)=O)ccc2oc(S)nc2c1 40612,C1(NC(CSCC(N)=O)=O)CCCN(C(=O)C(=O)NCc2ccc(Cl)cc2)C1 40613,C1(CN(C(CC(C)NC(C2CCC(C(=O)OC)C2)=O)=O)C)CCCC2CC12 40614,N1(S(CCC)(=O)=O)CCC2(CCOCC2)C(NS(=O)(=O)CC)C1 40615,N1(C(CC=C=C)=O)CCC(NC(c2ccn(-c3ccccc3)n2)=O)C1C(C)C 40616,c1(C(C)C)cc(C(N2CCOCC2CNC(C2(CF)CC2)=O)=O)ccc1F 40617,c1(CC)cc2oc1CNCC(=O)N(C)CC(C)CNC2=O.C1(OCC)CC1 40618,c1(C(=O)NCC(CC)NC(c2cnn(CCO)c2C)=O)cccc(F)c1OC 40619,C(=O)(C1=CC2CCC=CCCC12)N1CC(C(C)NC(c2cn(C)c(=O)n2C)=O)C1 40620,C1(CNC(C=C(C)Cl)=O)CN(C(=O)C(C)C2(O)CCC2)CC2(CCC2)O1 40621,C1(NC(CCC)=O)(CNC(=O)Cc2ccc(O)c(OCC)c2)CC2CCC1CC2 40622,C=C(F)C1(C(=O)NCCCN(C(=O)CCC(C)OCC)CC(C)C)CCOCC1 40623,c1(OC)cc(C(=O)NC23CCN(C(=O)CN4CCCCC4)CC2C3)c(N)c(C)c1 40624,O=C(N=c1[nH]ccc2cc(Cl)ccc12)C1CC1N.c1c(Cl)cc(F)cc1Cl 40625,C(=O)(C1=C(C)CCOC1)NCC(CC(=O)NC1C(C)(CC)COCC1)OC 40626,C1(C(=O)NC(c2cnccn2)C)CCCN1NC(=O)c1cn2ccccc2n1 40627,N1(C(c2ccc(CSC(F)F)o2)=O)CCN(C(=O)CCF)C2CCCCC2C1 40628,c1(CNC(=O)NCc2n[nH]c(=N)o2)cc2n(n1)CCC2 40629,c1(C(N2CCN(c3cc(Cl)ncn3)CC2)C(=O)NCCC#N)cccc(F)c1Br 40630,C12(CCNC(CCCC#C)=O)CCC(C1)N(C(C1CCC(=O)N1C(=O)NC)=O)C2 40631,C1(OC)CN(C(=O)CCN(CC(F)(F)F)C)CC1NC(=O)Cc1cccn1C 40632,Cc1ncnc(C)c1CC(=O)NCC(O)CN(C)C(C1CC1C)=O 40633,CC1CCN(C(C2CC(=O)NC(=O)C2)=O)CCN1C(=O)C=CC=C(Cl)Cl 40634,C1(C)(CC)CCN(C(=O)CC2(NC(=O)COC)CCC2)CC1 40635,C1(C(N2C(CCNC(=O)Cc3ncc(Cl)s3)COCC2)=O)CC2CCC(C1)C2 40636,C1(CNC(c2c(C)ncs2)=O)CN(C(c2ccc(F)cn2)=O)CC1C(F)(F)F 40637,Cc1nnc(NC(CNC(c2nccc(Cl)c2F)=O)C2CCC2)c(C#N)c1C 40638,C#CC1CC2(CC2)CN1C(C1CCCC(NC(=O)CC(F)(F)C(F)F)CC1)=O 40639,c1(CC(=O)NCCC(=C)CNC(=O)CCCc2ccsc2)nn(C)cc1Br 40640,C(=O)(C(CC1CCC1)NC(=O)COC1CC=CC1)NCC(C)SC 40641,c1(OC)cccc2c1OCCC2NC(c1c(Br)ccc(C)c1F)=O 40642,N1(C(=O)C(c2ccccc2)Oc2ccc(F)cc2)CCC(O)C(O)CC1 40643,N1(C(C2(C(=O)NC)CC2)=O)CC2=C(C1)CN(C(C1COCC1(C)C)=O)C2 40644,C(=O)(C1CC(C)S(=O)(=O)c2ccccc21)NCC(C)NC(C=CC(CC)(C)C)=O 40645,C1(N(C(=O)CCCc2ccsc2)CC)CCN(C(=O)C=Cc2nnn(C)n2)CC1 40646,c1(C(=O)NCC2N(C(C(C)S(N)(=O)=O)=O)CC3(CC3)C2)coc2ccc(O)cc12 40647,N1(C(C(CC)C)=O)CCCC(N(C(=O)Cc2c(C)n[nH]c2C)CCO)C1 40648,N1(C(CC(CC#C)NC(=O)CC(=O)N(C)C)=O)CC(C)CCC(C)C1 40649,CN1CC2(CCN(C(=O)CNC3=NCCN3)CC2)c2ccccc21 40650,N1(C(C2C(C(=O)OC)C=C2)=O)C(C(=O)NCc2cnn(C)c2OC)CC2CC12 40651,c1(OCC(=O)Nc2c(C(=O)OCC)cncn2)cc(C)ccc1C(C)C 40652,c1(NCC(C)(C)NC(c2cnc(OC)nc2C)=O)ncc2c(ncn2C)n1 40653,C1(CC(=O)NC)SC(=Nc2ccccc2CO)N(Cc2cc(Br)ccc2Cl)C1=O 40654,N1(C(C(C)N(C(c2ccn(CC)n2)=O)C2CC2)=O)CCC(C)(COC)CC1 40655,CC1(SCC(F)(F)F)CCOCC1.C12COCC1C(=O)N(CC(F)(F)F)CC(=O)N2 40656,c1(C(N(CCCCCCNC(C(F)=CC)=O)C)=O)cc(=O)n(C)cc1Br 40657,CCC(CC(=O)N(C(C)C(=O)NC1(CC)CCCCC1)CC)OC 40658,C1(C(=O)NC(CC)(C)CCNC(=O)C(C)N=[N+]=[N-])CCc2nc[nH]c2C1 40659,C1(CC(=O)NCC(CNC(CCOCC=C)=O)(C)C)CCC(=O)N1CC 40660,C(C)(C)(C(=O)N1CCCCO1)C1CCN(C(c2ccn(CCC)n2)=O)C1 40661,Cc1ccsc1C(N1CCC(NC(C2(CC3CC3)CCCO2)=O)C1)=O 40662,C=CCC(C)(C)CC(=O)NCC(O)CC(=O)NCc1cscc1C 40663,C1(C(C)NC(=O)Nc2ccccc2F)CCCCN1C(=O)CSc1nncn1C 40664,N1(C(=O)COC2CCCC2)CCC2(CCCN2C(=O)C2=CCCC2)C1 40665,c1(-c2[nH]c(=NCc3c(OC)c(F)ccc3)sc2)cc(F)c(C#N)cc1C 40666,N1(C(C2C(CC)CCCN2C(=O)CCC(C)N(C)C)=O)CC2CCC1CN2CC 40667,C1(C(N2C(CCN(C(=O)CCC#N)C)CCCC2)=O)CCC2CCC1O2 40668,CCC(O)C(C)(C)C(=O)NC1CCC(C(N2CCC(C)(C)C2C)=O)CC1 40669,C(=O)(CCC(F)(F)Cn1cc(-c2cccc(CNC3CCC(=O)N(C)C3)c2)nn1)OC 40670,N1(C(c2c(OC)cncc2)=O)CCC(C)(C)C1C(=O)NCCCSCCO 40671,c1(OC)cc(Cl)c(CN2CCCN(C(=O)CC3CCCCO3)CC2)cc1OC 40672,c1(N(S(N)(=O)=O)CCN(C(c2n(CC)nnn2)CC)Cc2ccccc2)ccc(Cl)cc1 40673,C1(N(C(c2ncn(CCNC(C(C3CC3)OC)=O)c2)=O)C)CCC(C)(C)C1 40674,C(=O)(C(O)CC(C)(C)C)N(C1CN(C(C2(C)CCC(C)C2)=O)C1)C 40675,CCC(C)(C)C(=O)NCc1nc(C(=O)Nc2ccc(C(N)=O)cc2)c(C)o1 40676,c1(NC(C)=O)ccc(CC(=O)N(C2C3CN(C(=O)C(F)=C(C)C)CC23)C)cc1 40677,C1(C(=O)NCC(CC)C#N)CC12CCN(C(=O)CN(C1CC1)CC)C2 40678,Cn1nnc(CNC(=O)C(c2csc(Cl)n2)N2CCC2c2ccccc2)n1 40679,C1(C(=O)NCC2CN(C(CC(=C)C)=O)CC2C(F)(F)F)Cc2nccn2C1 40680,n1(CC)c(C(=O)NCCC(F)Cn2cc(C3(C)CCCC3O)nn2)cnc1O 40681,c1(C(N2CC(CNC(CC(CC)C)=O)C3(C2)CC3)=O)cnc2c(c1)nnn2C 40682,N1(c2oc(C)c(C(=O)N(C)C)n2)CC(C)CC(C)(C)C1 40683,c1(NC(c2c(NCc3ccc(OC)nc3Br)c[nH]n2)=O)cccc2cn(C)nc12 40684,C1(CC=C)(NC(=O)Cc2c[nH]nc2C)CCN(C(=O)C(C)(C)COC(C)C)C1 40685,S(=O)(=O)(c1ccc(=NCC(C)(COC)OC)[nH]c1)N1CCC(OC)C1C 40686,c1(C(N2CCC(CNC(CCCSC)=O)C2)=O)ccc(Cc2ccsc2)cc1 40687,CC1(C(N2CCC3CCC23)=O)CNCC1(F)F 40688,C(C1CCCN1C(=O)Cc1cc(C)sc1C)=CC(N1CCC(CN(C)CC)C1)=O 40689,c1(OC)ccc(F)cc1C(=O)C(=O)NCC1COCC1NC(C12CC(F)(C1)C2)=O 40690,C#Cc1cncc(C(=O)NC2CCCCC2CNC(=O)C(F)C(C)(C)O)c1 40691,C1(N(C(c2c(COC)cc[nH]2)=O)C)CN(C(C2CCCC(=O)N2C)=O)CC1(C)C 40692,c1(C(N2C(C(=O)NCCN(C(=O)OC)C)COCC2)=O)cc(C)c(F)cn1 40693,CN1CCN(C(c2ccccn2)=O)C(C(=O)N(C2CCN(C)CC2)C)C1 40694,N1(C(CC(CC)C)=O)CCCCCC(NC(C2OCCC2(C)C)=O)C1 40695,c1(C(=O)NC2CCN(C(c3c(C)nn[nH]3)=O)CC2C)cc2c(s1)CCSC2 40696,Cc1cc(F)c(Cl)cc1C(=O)NCC(F)CNC(=O)CC(O)C(C)C 40697,C1(N(c2ccsc2)CC)C2CN(Cc3cc[nH]c3)CC12 40698,C(=O)(CC1=CCCCC1)NCC1CCCN(C(CCCOC(C)=O)=O)C1 40699,c1(CC(C(=O)Nc2n(CCN(C)CCO)ncc2)NC=O)ccc(Cl)c(Cl)c1 40700,CCC(C(C)O)NC(=O)CCN(C)C(c1c[nH]c(C(=O)OC)c1)=O 40701,C1(CC(=O)NCC2CC(NC(=O)C=CC3CCCCCC3)C2)CCC(F)(F)CO1 40702,c1(CCC)cc(C(=O)N(C(C)C(=O)NCC(O)CN(C)C(C)C)C)n[nH]1 40703,C=CCC(CC(=O)N1CCCC(N(C)C)CC1)NC(c1ccc(C)c(C)c1)=O 40704,C(CCN(C(=O)CC1(OC)CCC1)CC)(C(C)C)NC(C(CC)n1cncn1)=O 40705,c1(C(N2CC(NC(c3ccc(C)cn3)=O)C3C2C3)=O)cnc(C2CC2)nc1C 40706,CC(C)CC(C)(C)C(=O)NC1CCOCC1NC(C1CN(CC(F)(F)F)C1)=O 40707,Cc1nn(C)c(C)c1CNC(=O)C(C(C)O)NC(=O)OC(C)(C)C 40708,C(=O)(C1=CCCS1)NCC1(OC)CN(C(C2CCCC2(C)C)=O)C1 40709,c1(CC(=O)NS(CC2(C)COC(=O)N2)(=O)=O)cccc(Cl)c1Cl 40710,C(C(C)NC(c1ccn(C(F)F)n1)=O)(C(C)C)NC(c1c(OC)n[nH]c1)=O 40711,C(=O)(C(C)C(O)C(C)CC)N1CCC(C(C)NC(C(CCC)=CCC)=O)CC1 40712,C1(C(C(=O)NCC(F)(F)CO)NC(=O)CC2(CC3CC3)CCC2)CC=CCC1 40713,C1(C)(CC(=O)NCCSCC#C)CCN(C(C2(O)CCCC2)=O)C1 40714,c1(C(=O)NC(CCN(C(C(CCC)CCC)=O)C)C)ccc(=O)n2c1COCC2 40715,c1(C(=O)NCC2CCN(C(=O)CCc3ccnc(Br)c3)C2)cc2n(n1)CCO2 40716,CCC(CCC(=O)N(C)CCOCCCO)NC(=O)CCCC(=O)OC 40717,C(=O)(C(C)(F)C(C)(C)F)N(C)CC1(NC(CCc2cccc(OC)c2)=O)CC1 40718,C1(NC(C(CSC)C)=O)CC2CCC1N2C(=O)Cn1nc(O)ccc1=O 40719,c1(C(=O)NCC(COC)(C)OC)cc2c(cc1O)CCCC2 40720,C(Cn1cccn1)(C(=O)NC(C)(CC)C1CC1)NCC1(CCC)CC1.C1(=O)CN1 40721,N1(C(Cc2ccc(CC)cc2)=O)CCC(C(C)C)CC1CNC(=O)C(CC)OC 40722,C1(NC(c2ccc[n+]([O-])c2)=O)CC(O)CN(C(=O)CSc2cccc(F)c2)C1 40723,C1(CNC(C2(CCC)CCC2)=O)C2CCCC1N(C(=O)C(C)(C)F)C2 40724,CC1=C(C)CC(C(=O)N(C(C)(C)CC(N2CC(CO)CC(C)C2)=O)C)CC1 40725,c1(CC(=O)N(C2CCN(C(C3(C)CCCC3C)=O)C2)CC)ccccc1O 40726,C1(C(=O)NCCC=C=C)CCN(C(C2OCCOC2C)=O)CC1(C)C 40727,C=CC(C)(CCOC)C(=O)NC1CCC(C)N(CC(=O)NC2CC2)C1 40728,C1(C(N2CC(C)N(C(c3nnc(Cl)cc3N)=O)CC2)=O)COc2ccccc2O1 40729,CC1(C(=O)NCC=CCNC(c2ncoc2-c2ccccc2)=O)CC2(CCC2)C1 40730,c1(OC)nc(=Nc2cccc(C(=O)Nc3ncc(CCO)s3)n2)[nH]cc1C#N 40731,c1(N(c2n(CCC#C)c(Cc3cc(C)[nH]n3)nn2)C)nc2c(F)cccc2o1 40732,C1(CNC(CCOCCCNC(c2cc(C)sn2)=O)=O)CC2(C1)CC(O)C2 40733,c1(C(N2CCC(NC(C(C(C)C)F)=O)C2C)=O)cccn2nccc12 40734,c1(C2(NC(C=CCC)=O)CN(C(=O)C(C)C#N)C2)ccc(Br)cc1 40735,c1(CC(N2CCC(=CCNC(C3CC4CC4C3)=O)CC2)=O)cccc2c1CCC2 40736,N1(C(C2C(NC(=O)COc3ccc(F)cc3)CCC2)=O)CCN2CCC1CC2 40737,C(=O)(C(C)(O)C(C)C)NCC#CCNC(c1c(C)[nH]nc1C(F)(F)F)=O 40738,N1(C(CCCCNC(C=CCOCCOC)=O)=O)Cc2cncnc2C1 40739,C1(C(N2CC(CNC(C(C)N(C)Cc3ccccc3)=O)C2)=O)CCS1(=O)=O 40740,C12(CNC(C3(F)C4CCCCC34)=O)CCC(CC1)N2C(c1cc(C(N)=O)[nH]c1)=O 40741,C1(C2CCC(=O)NC2)(C(N(C2CCCN(C(=O)C#CC3CCC3)C2)C)=O)CCC1 40742,C1(NC(c2cccc(C(F)(F)F)n2)=O)CN(C(C2(n3cncn3)CC2)=O)CC1F 40743,C1(NC(C2CCC(C)C2)=O)(CNC(c2ccc(F)o2)=O)CCOCC1 40744,c1(C(N2CC(CC=C)(NC(C3CC3F)=O)C2)=O)ccc2[nH]c(=N)[nH]c2c1 40745,Cc1ncc(C(=O)NC(C(=O)N(CC(N)=O)C)c2ccoc2)s1 40746,C1(C(N2CC=CC(NC(C3CCC(C)(CC)O3)=O)C2)=O)CCC(F)(F)C1O 40747,c1(C(N(CCCN(C(CC2(CSC)CC2)=O)C)C)=O)nc(C)ncc1Cl 40748,CC#CCCC(=O)N1CCC(N2CCN(C(c3cnn(C)c3N)=O)CC2)CC1 40749,N1(C(C(C)CSc2ccccc2)=O)CCC2CC1CN(C(C1(Cl)CC1)=O)C2 40750,c1(C(=O)NCCN(CC(C)O)C(c2cnc(O)c(F)c2)=O)ccnc2c1CCC2 40751,c1(-n2cc(C(C)NC(c3cc(Br)c(Br)[nH]3)=O)nn2)cccc(OCCO)c1 40752,C1(C)(C(=O)NCC(CC=C)NC(=O)COc2cc(C)on2)CCCCNC1=O 40753,C1(C)(C)CCCN(C)Cc2occ(n2)CC(=O)N1CC.C1(CC)CC(C(F)F)C1 40754,N1(C(Cn2ncc(NC(C(=O)NC(C)C)=O)c2)=O)CC2CCC1C(O)C2.C1CS1 40755,CC(CC(F)(F)F)C(=O)N(CCNC(=O)CN1CCCCCC1)C1CC1 40756,c1(C(=O)NCC(C)N(C(CCNC(C)=O)=O)C2CC2)c(Br)ccc2n[nH]cc12 40757,C(=O)(CC(CC)C(C)(C)C)N1CCC(O)(CNC(CNC(=O)OCC=C)=O)CC1 40758,C1(CNC(c2c(C)ncnc2)=O)CC(C(=O)NOC2CCOC2)=NO1 40759,O=C(C1=C2CCCN=C2NN1)C1N(C(c2ccc3c(c2)CCCS3)=O)CCOC1 40760,C1(NC(c2cc(C)sn2)=O)CCC2(CC1)CCN(C(=O)CCc1cnn[nH]1)CC2 40761,C(=O)(CCC(=O)NC1CCC(CNC(c2ccn(C(C)C)n2)=O)C1)NC 40762,C1(COC)(NC(C2CC(n3cc(C4(C)CSC4)nn3)C2)=O)CCCC1 40763,c1(NC)snc(C)c1C(N1CC(CNC(c2cncn2C(C)C)=O)C(O)C1)=O 40764,C1(NC(Cc2cccc(C(C)C)c2)=O)CN(C(=O)C(C)n2cncn2)CC1(C)C 40765,CC1CN(C(=O)CC(C)C(F)(F)F)CCCN1C(c1cncc(C(F)(F)F)c1)=O 40766,C1(C(=O)NCC(C2CC2)NC(C(C#N)=CC2CC2)=O)CCCCCC1 40767,c1(C(C(=O)NCC)N(C)C(c2ccco2)C)cc2n(n1)CC(C)(C)CO2 40768,C1(C(=O)NC2C(NC(c3c(CCC)n[nH]c3)=O)CCC2)C(F)(F)C12CC2 40769,C1(CC)CC(C)(C)CCC1C(N1CCC1CCCNc1ncoc1CN)=O 40770,C1(NC(c2nc(C)[nH]n2)=O)CCC2CN(C(=O)COC(F)F)CC2C1 40771,c1(C(=O)NCCC(C)NC(c2cc(C)nnc2O)=O)c2c(nn1C)CCC2 40772,C=C(F)C1(CC(=O)NCC=CCC(=O)NCC2CC(CC)=NO2)CCC1 40773,CC1(C)COCC(NC(N2CCC(CC3CC3)CC2)=O)CN1 40774,C1(OC)(CO)CCN(C(=O)C(CO)NC(C2SCCS2)=O)CC1 40775,c1(C(c2n(CC)nnn2)NC2CN(c3nncs3)C2)cc(C)nnc1C 40776,C1(NC(c2ccc(N(C(C)=O)C)cc2)=O)CCCN(C(=O)C(F)CC2CC2)CC1 40777,N1(C(C(CC=CCC)C)=O)CC2CC(NC(=O)C3=C(C)CCC3)C1C2 40778,C1(NC(N(CC(N2CCN(C(=O)CNC3CC3)CC2)=O)C)=O)CCC2CC2CC1 40779,c1(C(CC(=O)NCC(CCNC(C=CCC)=O)O)C)ccccc1OC(F)(F)F 40780,C#Cc1cn(C)nc1C(=O)NCC1CC(NC(=O)C2=COCCC2)CC1O 40781,c1(C(N2CC(c3cn(CC(COC)O)nn3)OCC2)=O)ccc(C)c(C(F)F)c1 40782,CC(C)C(CCNC(C1(C(F)(F)F)CCCCC1)=O)NC(=O)CC1CCOC1C 40783,N1(C(C(CCC)OCC)=O)CC(CNC(c2cn(C)cn2)=O)OC2(CCC2)C1 40784,CC(C)(C)C1=CCN(C(=O)COC2CCN(C(c3ccc(C(N)=O)[nH]3)=O)C2)CC1 40785,c1(C(N(C2CCN(C(C3CNC(=O)C3)=O)CC2)CC)=O)n[nH]c(C2CC2)c1Cl 40786,N1(C(C(C(C)C)O)=O)CCN(C(=O)CCCCCC#N)CC(CO)C1 40787,C1(CNC(C(CN(C(C2(CCC)CC(=O)C2)=O)C)C)=O)C(O)C2CCOC12 40788,C(=O)(C1=CCC12CCOC2)NCCC(CC)(CC)NC(=O)Cc1ccsc1 40789,c1(OC)ccc(C(N2CCC(N(C)C(c3cc(F)ccc3N)=O)C2)=O)c(F)c1Cl 40790,c1(CC)c(C(=O)NC2CC(C(=O)N(C(C)C(=O)OC)C)C2)ccn1C 40791,C1(CN(C(CNC(C(CC)C)=O)=O)C)CCN(C(c2cc(F)c[nH]2)=O)CC1 40792,c1(CCNC(C=C(C)CNC(=O)C(C)CN(C)C)=O)ccc(C)s1 40793,N1(C(C2Cc3cscc3C2)=O)CCCC2(NC3CN(CC=C)C(=O)C3)CCCC12 40794,c1(C(N(C(CNC(c2ccc(CC)cc2)=O)C)C)=O)cc2oc(Br)cc2[nH]1 40795,C(C)(C)(CN=c1nc(N2CCOC(COC)C2)c2c(ncn2C)[nH]1)OC 40796,CC(Cc1cccs1)C(=O)NNC(=O)c1cc2c(cn1)OCO2 40797,c1(CCCC(=O)NCC(C)N(C(=O)C(C)=CC(C)(C)C)C)ccc(C#N)cc1 40798,C(=O)(CCCC(C)(C)C#N)NCC1CCCN(C(c2c(Cl)ccc(OC)n2)=O)C1 40799,N1(C(c2cc(N)c(Cl)cc2)=O)C2CCC1CN(C(c1cn(C3CCC3)nn1)=O)C2 40800,n1(C(CN(CC(=O)OCC)C(c2ccc(F)cc2)=O)C)c(=O)oc2ccccc12 40801,N1(C(C2CC(C)=C(C)CC2)=O)CC2CN(C(C3(CCF)CC3)=O)CC2(C)C1 40802,c1(CC)ncc(C(=O)NC2(CCCNC(c3ccc(CC)s3)=O)CC2)[nH]1 40803,c1(C(N2CC(O)(CN(C)C(c3nsnc3O)=O)C2)=O)ccc(Cl)c2c1OCCO2 40804,c1(SC)ccc(CCNC(C)C(=O)N(CC(F)(F)F)C(C)C)c(Br)c1 40805,N1(C(C(C)=C2CCC2)=O)CCSCC1CCNC(C1NC(=O)CC1C)=O 40806,CC1CC(NC(=O)Cn2cc(C3CC3)nn2)CCN1C(C1CCC(C)(C)OC1)=O 40807,C1(CNC(=O)C=CC2CC2)CC2COCC2N1C(=O)Cn1ccc([N+](=O)[O-])n1 40808,N1(C(c2csc(Br)c2)C(=O)NCC)CCC(C2(C)CC2)CC1 40809,CCCCCCCN(C(c1cc(F)ccn1)C(=O)NCc1cccc(OC)c1)C 40810,C(C(=O)N1CCOC(Cn2cc(CC3CCOC3=O)nn2)C1)(C(C)C)SCC 40811,c1(C(N2CCC(N(C(=O)C(F)F)CC#C)CC2)=O)noc2c1COCC2 40812,C#Cc1cccc(C(N2CCC3(NC(c4nn(C)cc4C)=O)CC3C2)=O)c1 40813,C1(C)(C(=O)NC(C2CN(C(c3cc(O)ncn3)=O)CCO2)C)COC(=O)N1 40814,C1(NC(c2occ(C)c2C)=O)CCC(C)N(Cc2ccc(F)cc2Cl)C1 40815,C=C(C)C1CCC(C)=CC1CC(N1CCN(C(=O)CN(CCO)CCO)CC1)=O 40816,Cc1cc(C#N)cc(C(=O)NCC(C2CC2)NC(=O)C(O)C(C)(C)C)n1 40817,c1(CC(=O)NCCN(C(C)C)C(c2cc(C3CC3)on2)=O)cc(C2CC2)no1 40818,n1(CC(C)O)cc(-c2ccc(CSc3ccccc3)cn2)ccc1=O 40819,C1(C(=O)NC2CCC(CCC)CC2)CCCCCCN1C(C1C(C#N)C1(C)C)=O 40820,C1(NC(c2cnc(C)nc2O)=O)COC2(C1)CN(C(=O)CCC(C)CN(C)C)C2 40821,c1(CCC(=O)N(C)CCNC(=O)Cc2cn[nH]c2)ccncc1Br 40822,C(=O)(C1=NOCC1)N(C(c1cn(C)nn1)C(=O)NCCc1ccn(C)n1)C 40823,c1(C2C(C(N(C3CCC3)C(c3csc(Cl)c3)C)=O)C2)ccc(F)c(Br)c1 40824,N1(C(CCCCC)=O)CCC(NC(c2cccnc2O)=O)C(CO)C1 40825,C(CNC(=O)C=Cc1cncnc1O)(C(C)C(C)C)Nc1cc(OCC)ncn1 40826,N1(C(c2cccc(C)n2)C(=O)NCC2CCOCC2)C2CCC1CC(CO)C2 40827,C1(C(N2CC(Cc3cn(C(CC)C)nn3)C2)=O)CCc2ncc(C)n2C1 40828,CN1CCN(C(=O)CC2CC(=O)C2)C(C(=O)NC2CCCC(C(N)=O)C2)C1 40829,C(C(CN=c1cc(C)nc(N2CCC(C(C)CO)CC2)[nH]1)OC)OC 40830,C1(C(=O)NCC(c2cc(OC)c(Cl)cc2)F)CC2COCC(C1)C2(F)F 40831,C1(CNC(Cc2ccn(C(C)C)n2)=O)CC(C)(C)CN1C(C1CC(C)C1)=O 40832,C1(C(=O)NCCCC(C)NC(C(C=CC)O)=O)CN(C)CC(C)O1 40833,N1(C(C(c2cn(C)nc2)=O)=O)CCCC(CC(=O)NCCCOC2CCC2)CC1 40834,Cc1cc(C(=O)NC2CCCC(NC(=O)C3=NOCC3)C2)cc2c1NCCC2 40835,c1(C(N2CCCC(N(c3ccno3)C)C2)=O)cc(S(N)(=O)=O)ccc1O 40836,c1(C(N2CC(N(C)C(C3CC3(Cl)Cl)=O)C(F)C2)=O)n[nH]c2c1CCC2 40837,c1(NC(=O)NC2CC(CCNC(=O)OC)C2)ccnnc1O 40838,CC1CCOC(C(=O)NCCc2n[nH]cc2C(N2CC=CC2)=O)C1 40839,CCC(C(=O)NCC1CCN(Cc2csc(-c3ccco3)n2)CC1)C(C)C 40840,N1(CCCCN(S(CCCC)(=O)=O)C(C)=O)CCCc2cc(C)cc(F)c21 40841,c1(C(CNC(c2cnco2)=O)NC(CCC2CCN(C)C2)=O)cccc(Cl)c1 40842,C1(OC)(NCCC(=O)NCCC(=O)OC)CCC(C)(C)C1 40843,C1(NC(CN(CC)CC)=O)CCCCC1NC(=O)CC1(OC)CCCC1 40844,c1(CC)nn(C)cc1C(=O)NC(C1(O)CN(C(c2onc(C)c2C)=O)C1)C 40845,C(=O)(C1CN(C)C(=O)c2ccccc21)NCC1N(C(C(COC)O)=O)CCCC1 40846,c1(SC2(CNC(c3nc(C)c(C)o3)(c3n(CC)nnn3)C)CC2)ccccc1C 40847,C1(C(N2CCC(CC=C)(NC(c3coc(Cl)n3)=O)C2)=O)CCC12CCOCC2 40848,N1(C(CCCC#C)=O)CCCC(O)(C(=O)NCC2CC2CSc2ccccc2)C1 40849,c1(C(=O)NCC2N(C(C(C)(C)NC)=O)CCC2)cc(C(=O)OC)ccc1Cl 40850,Cc1cc(C(C(=O)NC2CCC2)N(C2CC(C)CC(C)C2)C)cc([N+](=O)[O-])c1 40851,c1(C(=O)NC(C2CN(C(c3onc(CC)n3)=O)C2)C)nc(C)sc1C 40852,C1(C(=O)NCC2CCCN(C(=O)CCC3CCCC3)C2)(NC(N)=O)CCCCC1 40853,C(=O)(C1=CCCN(C(=O)COCC2CC2)C1)N(C1C(C)CC1)C 40854,Cc1ccc2cc(C(N3CCC(C(C)NC(C4CCCC4F)=O)CC3)=O)cn2c1 40855,c1(C(N2CCN(C)CC2CNC(=O)CCCCO)=O)cnc2n1CCOC2 40856,C1(C(=O)N(C)Cc2ncc[nH]2)(COC)CCCN1C(=O)CC(O)CN(C)C 40857,C(C(CC(F)(F)F)NC(=O)CCOC(C)=O)NC(c1ccc(C(CC)=O)cc1)=O 40858,c1(C(N2C(CNC(c3ncn(CC)c3)=O)CCC2)=O)cc2scnc2[nH]1 40859,CN1CCN(C(c2ncccn2)=O)C(C(=O)NC2CN(C)CC2O)C1 40860,c1(C(=O)NCC=C)oc(CNC(C2(Cl)CC2)=O)nc1C 40861,N1(C(C(C#C)(C)C)=O)CC2(CCN(C(C)(C)C)CC2)C1.C1(C(=O)NCC)CC1C(=O)O 40862,N1(CCOCCOC)CCC2(CCN(C(c3c(C)nn(C)c3C)=O)C2)C1 40863,C#CC1(C(=O)N(C)CC2C3CN(C(C4(CC)COC4)=O)CC23)CCCC1 40864,N1(C(C(c2ccccc2)OC)=O)CCOC(c2cn(CCN(C)C)nn2)C1 40865,c1(C(=O)NCCNC(=O)CCC2CCC2)cccc(F)c1 40866,N1(C(C(C)=C(CC)C)=O)CC2CC(C1)C2NC(=O)CC1CC(OC)C1 40867,CC1CC2CC(C(=O)NCCC3CCCN(C(=O)C4=COCCO4)C3)(C2)O1 40868,c1(C(C)NCC2(NC(=O)OC(C)(C)C)CCCCC2)ccc(Cl)c(F)c1 40869,N1(C(C2C(C(=O)OC)CC2)=O)CCC(C(=O)NC(c2nc(C)no2)C)C12CC2 40870,C1(NC(CC2(C(=O)OC(C)(C)C)CCC2)=O)CCOC(c2ccc(F)cc2)C1 40871,n1(CC(=O)NC2CC2CNC(C23CCN(CC2)C3)=O)cc(F)cc([N+](=O)[O-])c1=O 40872,CC1Oc2ccccc2OC1C(=O)NC1CCC2CN(C(C3CCC3)=O)CC2C1 40873,N1(C(C2(C(C)(C)C)CCCC2)=O)CC2CN(C(C3CCCS3(=O)=O)=O)CC2(C)C1 40874,CCCC(CCC)CC(=O)N1CCN(C(=O)CN(CC)CC)C(CS(C)(=O)=O)C1 40875,C1(C(=O)NCCNC(C(C(C)C)NC(=O)C(C)(C)C)=O)CCC(F)(F)CO1 40876,C(=O)(C(C)(C#N)CC)NCc1c(CNC(c2c(CC)nn(C)c2)=O)cccc1 40877,N1(C(c2cc(C)c(Cl)cn2)=O)CCCC(C2CCN(C(=O)CCCC#N)C2)C1 40878,C(c1cncnc1O)=CC(=O)NCC1(NC(Cc2nn(C)c(Cl)c2)=O)CCOC1 40879,CC(C1CCCCC1)=CC(N1CCC(N(C)Cc2ccnc(C)c2N)C1)=O 40880,NC(=O)CC(C(=O)Nc1ccc(F)cc1)NC(=O)CN1CCNC1=O 40881,CCC(C(=O)NCCC1CCN(C(=O)C(N2CCC(C)CC2)=O)CC1)C(C)O 40882,c1(C(N2CCC(NC(C(C(C)C)OCC)=O)C2)=O)cnc(C)nc1C1CC1 40883,N1(C(CC(C)F)=O)CCC(CNC(=O)CN(S(C)(=O)=O)C)C(F)(F)CC1 40884,N1(CCOCCCC)CCCC(CO)(NC(c2cnc(COC)s2)=O)C1 40885,CC(C)(C)CCCCC(=O)NC1CC(CNC(c2ccccc2OC(F)F)=O)C1 40886,C(C)(C)(C(=O)N(CCCNC(C1(C)CCCC1)=O)CC1CCC1)N(C)C 40887,N1(CC(=O)NCC(=O)N(CCCCCOc2ccccc2)CC)CCCC(C)C1 40888,CCCC(C)(C)C(=O)N1CC(C(=O)Nc2ccc(Cl)cc2C(F)(F)F)CC(C)C1 40889,O=C(C1CNc2ccccc21)N1CCN(C(=O)Cc2cccc(Cl)n2)C(CO)C1 40890,CS(=O)(=O)C(C(=O)NCCCCNC(C1(F)CCS(=O)(=O)C1)=O)C1CC1 40891,Cc1c(C(=O)NCCCOCCCNC(C2CCC(O)C2)=O)ncn1C 40892,Cc1nc(Cl)[nH]c(=NC(C)CC(C)NC(C2CCCC(F)C2)=O)c1F 40893,CCCCC(CNC(=O)C1=CCSC1)NC(c1cnn(CC2CCC2)c1)=O 40894,C1(C(N2CCC(C(CC)CC)C2)=O)C2CC3C(C2NC(=O)C(C)(O)CCSC)C13 40895,N1(C(C(CC#C)C2CC2)=O)CCN(C(=O)C(C)(F)F)CC1C1CC1.ONC 40896,c1(C(N(C(C)CN(C)C(c2n[nH]cc2Br)=O)C)=O)cc2c(cc1O)CCC2 40897,C1(CNC(CC2(CNC(CCCOC)=O)CC2)=O)CCOC(C)(C)C1 40898,c1(C(N2CCC(C)(NC(CCOCCOC)=O)CC2)=O)ccc2occc2n1 40899,CN1CC(C(=O)NCC(C)(C)CN(C(=O)Cn2cnnn2)C)C(C(F)(F)F)C1 40900,c1(NC(C2C3(CCN(Cc4ccn(C)n4)C3)C2)=O)ccc2nc[nH]c2c1 40901,c1(C(C)NC(CC)C(C)C)cc(C(F)(F)F)ccc1F 40902,c1(C(=O)NC(CCNC(c2c(COC)nn[nH]2)=O)(C)C)cn2c(n1)CCCC2 40903,c1(C(C2CC3CC3C2)OC(C)(C)C)nnnn1C(C)(C)C.C(C1CN1)OCC 40904,c1(C(=O)NCCN2CCN(C(C3C(C(=O)OC)C3)=O)CC2)ccc2ncsc2c1 40905,c1(C(=O)NC(CNC(C=NOC)=O)CO)cc(Br)c([N+](=O)[O-])[nH]1 40906,C1(NC(CC2CC(OCC)C2)=O)CCCC(N=c2[nH]c(Cl)nc(C)c2[N+](=O)[O-])C1 40907,C(=O)(CC1CCOc2ccccc21)NCC1C(NC(c2cnc(C)s2)=O)CC1 40908,c1(C(C)C)ncc(NC(=O)C(C)NC(=O)CC2CC2C2CC2)cn1 40909,CC(C)(C)C(C)(O)C(=O)NCCNC(=O)COc1ccc(C(N)=O)cc1 40910,N1(C(CSCC(=O)OC)=O)CC(NC(=O)C(C2CCC2)OC)CC2(CCC2)C1 40911,c1(C(N2CCCC(CCNC(CC(=O)N(C)C)=O)C2)=O)cc(Cl)ncc1N 40912,CC1(C)CCC(C(=O)NC2(CNC(C3(C(F)F)CC3)=O)CCOC2)C1 40913,C1(C(=O)OC)CC(C)CN(C(=O)C(=O)NCc2c(NC(C)C)cccc2Cl)C1 40914,CCN=C(NCC1CCCC1C(=O)NC(C)(C)C)NC(C1CCOC1)C 40915,C1(CC(=O)N(CCOCCNC(C(CCC)C)=O)C)COC(C)(C)CO1 40916,C(=O)(CC1OCCc2ccccc21)NC1CC(NC(C2COCC(C)(C)O2)=O)C1 40917,C12(CNC(=O)NC3(C(F)(F)F)CCC(OC)C3)CCN(CC1)CC2 40918,C12(C(N3C(CNC(c4c(C)onc4CO)=O)CCC3)=O)CCC(CC1)C(C)O2 40919,C1(C(N2C(CNC(C(CCSC)O)=O)CC3CC32)=O)CCC(=O)N(C2CC2)C1 40920,CCC(C)CC(C(=O)NC1CN(C(C)C)CC1C)NC(=O)Cn1cccc1 40921,N1(C(C23CC(CNC(C)=O)(C2)C3)=O)CCCN(C(c2cc3sccc3[nH]2)=O)CC1 40922,C1(F)(CNC(C2(CN(C)C)CC2)=O)CC(NC(=O)C(C)(C)c2cncs2)C1 40923,c1(C(N2CC(C(C)NC(Cc3c(C)noc3)=O)OCC2)=O)ccn2nnnc2c1 40924,N1(C(C(C2CC2)OC)C(=O)NC2CCC2)CCN(C2CCOC2)C(=O)C1 40925,c1(C(N2CC3(C(NC(c4ccc(F)s4)=O)CC3)C2)=O)coc2ccccc12 40926,c1(C(N(CC(C)NC(Cn2cc(C(C)O)nn2)=O)C)=O)cnc2[nH]c(O)nc2c1 40927,CC(CN(C(=O)NC(CC(=O)OC(C)(C)C)C1CCOCC1)C1CC1)S(C)(=O)=O 40928,c1(C(=O)NCCOCCN(C(CC(COC)(C)C)=O)C)cc(N)c2ncccc2c1 40929,c1(CCC(=O)NCCOCCNC(C(C)(C)F)=O)ccc(F)cc1F 40930,C(C(CC(C)C)NC(=O)C(O)C(F)F)NC(CCCN(C(=O)OC)C)=O 40931,N1(C(CCCOC)=O)CCC2C(C1)NC(=O)N2C1CCN(C(=O)CC(C)(C)C)CC1 40932,C=CCCC(O)CN(C(=O)C(C1CCCN(C(c2ccc(CO)o2)=O)C1)(C)C)C 40933,C1(NC(CC2C(C)C2)=O)CCOCC1C(=O)NCC(C)N(C)C1CC1 40934,CC(C)CC(O)C(=O)NCC1OCCC1C(=O)NC1(CO)CC(F)(F)C1 40935,c1(C(=O)NC(C(CO)NC(COc2cccc(OC)c2)=O)C)ccc(C)nc1O 40936,C(=O)(C1=NOC2COCC12)NC1(C(=O)Nc2c(OC(C)C)cccn2)CC1 40937,N1(C(CC(=O)N(C)C)=O)CC(C2(NC(=O)CCc3ccoc3)CC2)C1 40938,CC1CN(C(=O)Cn2cnnc2)CCC1C(=O)NCc1ccnc(C#N)c1 40939,c1(C(=O)NCC(C)N(C)C(c2ccc(F)cc2Cl)=O)ccc2cnsc2c1 40940,CC(C)C(O)C(F)(F)C(=O)NC1CN(C(c2onc3ccccc23)=O)CC1C 40941,c1(C(=O)OCC2Cc3ccccc3CO2)n[nH]c2c1CCCCC2 40942,CC#CC1CN(C(C2(NC(=O)Cc3ccc[nH]3)CCCC2C)=O)C1 40943,N1(C(c2c(C#C)c[nH]n2)=O)CCC(C=C)(C(N2CCCC(OC)C2C)=O)CC1 40944,Cc1cc(C)n(CCCNCc2ccccc2-c2ccc(F)cc2)n1 40945,C(c1cc(Cl)ccc1Cl)=CC(=O)NC1C(NC(Cc2ccc(C)s2)=O)CC1 40946,C1(CN=[N+]=[N-])CCc2ccccc2N1C(=O)NCc1ccc(OC2CC2)cc1 40947,N1(C(CC(C2(O)CCCOC2)(C)C)=O)CCc2cccc(O)c21 40948,CCCC(CNC(=O)CSC(F)F)NC(=O)CCOCC 40949,c1(C(=O)NC2(CF)CCN(C(Cc3c(C)nc(C)s3)=O)C2)cc(C)c(F)cc1F 40950,C1(NC(C(C)SC)=O)CCN(C(C23CCC(CO)(CC2)C3)=O)CCC1CO 40951,Cc1c(C(=O)NC2CCCN(Cc3ncsn3)C2)cnn1C(C)(C)C 40952,N(C1c2ccccc2CC12CCNCC2)CC1N(C(N)=O)CCC1 40953,N1(C(COCC=C)=O)CC(NC(=O)CC2CC2)C2CC12 40954,N1(C(CC2CN(C)C2)=O)Cc2ccccc2CC1CNC(C1CC2C=CC1C2)=O 40955,N1(C(Cc2cnc(C)[nH]2)=O)CCOCC(C)(CNC(=O)C(C)NC(=O)C2CC2)C1 40956,CC1(C)C=C(C(=O)N2CCN(C(c3cnc(C4CC4)o3)=O)C(C3CCC3)C2)C1 40957,N1(C(CC2CCCC(C)C2)=O)CC2CC(C1)N2C(=O)CN1CCN(C)C(=O)C1 40958,N1(C(C=C(C)C)=O)CCC2CN(C(c3cc4sc(C)cc4s3)=O)CCC12 40959,c1(C(N2CC3CN(C(C4(F)CNC4)=O)CC(C2)O3)=O)cc(Cl)cc(Cl)c1[N+](=O)[O-] 40960,CC(C)(CS(N)(=O)=O)C(=O)NCC1CN(C(C2(O)CCOCC2)=O)CC12CC2 40961,CN1CCC(F)(C(=O)N(C2CC2)CC2CCCN2C(=O)CCC2CCC2)CC1 40962,C1(C(=O)NCC2CCC(C(=O)NCc3cnc(CC)s3)O2)CC2CCC1O2 40963,CC(c1cccnc1)=CC(N1CC(NC(c2nccc(C)c2N)=O)C2(CC2)C1)=O 40964,Cc1cc(NC(=O)C(Cc2cn[nH]c2)NC(C2COCCC2C)=O)cc(CO)c1 40965,CCC(CC(=O)N1CCN(S(C)(=O)=O)CC1)NC1CN(C(=O)CCOC)C1 40966,Cc1nc(F)ccc1CNC(C1CC(NC(=O)CCCN(C)C)C1(C)C)=O 40967,c1(NC(C2(NC(c3ccc(C)cn3)=O)CCCCC2)=O)ccc2occc2c1 40968,c1(C(=O)NC(CN(C(=O)C2=CSCCO2)CC)C)c[nH]c2c(OC)nccc12 40969,C(=O)(CC(C)CC(C)C)NC(CC=CC)C(=O)NCCc1cccnc1F 40970,c1(CNC(C2CCN(C(c3c(C)coc3)=O)C2)=O)cccc(CO)n1 40971,C#CC#CC(C)(C)NC(=O)CN(CC#C)C(C1CC2CCC1C2)=O 40972,O=C(C1=Cc2cc(F)ccc2OC1)NCC1CCCC1NC(c1ccccn1)=O 40973,c1(OC)cc(NC(=O)CC2CCCN(C(C3CCC3)=O)C2)ccc1Cl 40974,C12(C(NOCCCC#C)=O)CCN(C(=O)COCC(=O)NCC)CCC1C2 40975,c1(C(=O)N)cc(C(C)C)on1.C(C(=O)NCC1CC1C)OCCOCCOCC#C 40976,CC1CCCC(C)C1NC(c1ccc(CNC(=O)CN2CCC(F)CC2)nc1)=O 40977,c1(CN(CC(CC)(C)OC)C)[nH]cnc1C#N 40978,C=CC(CC)C(=O)NC1CCCCC1C(=O)N(C(C)C(=O)NC)CC 40979,N1(C(c2c(NCC)scn2)=O)CC2C(CNC(c3ncoc3C(C)(C)C)=O)C2C1 40980,C(CC(C)C(=O)NCCCOCCNC(=O)CC(c1cccs1)OC)OC 40981,c1(C(=O)NCCCCC(C)NC(=O)C(F)(F)C(F)F)cnc2c[nH]nc2c1 40982,CC1(CC(=O)NC2(CCO)CCCCC2)CCCN1C(c1ccoc1)=O 40983,N1(C(CCCC#N)=O)CCC2(CCC2)C(CNC(C2CC3CC3C2)=O)C1 40984,C1(CNC(c2cc(C(C)=O)oc2)=O)CN(C(c2ccc(O)nn2)=O)CC1C 40985,Cc1nc(C(=O)NC2CCCC(NC(c3cc(O)cs3)=O)CC2)c2ccccn12 40986,N1(C(C(C)OCC2CC2)=O)CCCC(CCNC(c2cn(C)nc2Cl)=O)CC1 40987,C=Cn1nncc1C(=O)NCCCCCNC(c1c(Br)n[nH]c1C)=O 40988,C(=O)(CC(CC(C)C)NC(c1ncccc1CC)=O)N(C(C=C)C)C 40989,C(C)(CC(=O)N(C1CCN(C(C2(N(C)C)CC2)=O)C1)C)=C(C)C 40990,C(=O)(C(CCC(=O)NCCCCOC)NC(=O)Cc1cc(C)on1)NC 40991,c1(C(=O)NC2C(NC(CCN(S(C)(=O)=O)C)=O)CC2)cccc(N)c1 40992,c1(CC(=O)N(CCCCCNC(C2(C#C)CCC2)=O)C)cccc(F)c1F 40993,C12(C(N3CCC(N(C(c4ccc(Cl)cc4)=O)CC)C3)=O)C3C4C1C1C2C3C41CO 40994,N1(C(C(C)NC(=O)NCC)=O)CC2CC3CC2C1C3NC(c1cn(CC)nn1)=O 40995,Cc1cc(C#N)c[nH]c1=NC(=O)C12CC(NC(C34CC3C4)=O)(C1)C1(CCC1)CC2 40996,c1(C(=O)NCC(CC)NC(=O)C(N2CCC(C)CC2)=O)cc(N)c(Br)cc1C 40997,c1(C(=O)NC(C2CCN(C(C3CCC(=O)N3C)=O)C2)C)ccc2nc(O)[nH]c2n1 40998,Cc1[nH]nc2ncnc(N3CCOCC3CN(C(=O)CCC3CCC(C)O3)C)c12 40999,S(=O)(=O)(c1cccnc1NCCCC=C)NC1(CC=C)CCOC1 41000,C1(COC)(NC(c2nocc2Br)=O)CCN(C(=O)OC(C)(C)C)CC1 41001,C1(C)(CNC(CC)=O)CN(C2CCN(C(c3ccsn3)=O)CC2)C1=O 41002,c1(C(C(=O)NC(C(CO)NC(C(CC)C)=O)C)(C)C)cccc(F)c1 41003,c1(C(N(CCC)CCNC(=O)CC(C)n2ccnc2)=O)nccnc1CC 41004,C1(CC)CN(C(c2cnn(C)c2CC(C)C)=O)CCN1C(=O)CS(=O)(=O)N(C)C 41005,c1(CC)oc(C)cc1C(=O)NCCC(C)N(C(=O)Cc1cc(C)cs1)C 41006,CC(C)CC(O)C(=O)NC1CCCN(C(c2cccc(C3(F)COC3)c2)=O)C1 41007,N1(C(c2ccc(C)cc2O)=O)CCC2CN(C(C3(C#N)CC3(C)C)=O)CC2CC1 41008,C1(N(C(C(C)CC2CC2)=O)C)CCCN(C(=O)Cc2cncc(Br)c2)C1 41009,N1(C(C2C(NC(=O)CC3CSCCO3)COC2)=O)CCC2(CC1)CC(O)C2 41010,c1(C(=O)OCC)ccccc1CC(CCc1ccc(OC(F)(F)F)cc1)C(C)C 41011,c1(C(N2CC(N(C)CCO)C2)=O)cc(CCNC(c2c[nH]c(=N)o2)=O)on1 41012,C1(NC(c2n(CC)ncc2)=O)CC2(CCN(C(C3CC(N4CC(O)C4)C3)=O)C2)C1 41013,C(=O)(C1=C=CCCC1C)N1CCC(CNC(c2c(C)sc(Cl)n2)=O)C(O)C1 41014,c1(OC(C)C)ccc(CNC(=O)CC2CCCCN2C)nc1 41015,Cc1ccc(OCCCC(N2CC(NC(=O)C(C)N(C)C)C(C)C2)=O)cc1 41016,N1(c2ncc(C)c(O)n2)CC(CNC(=O)CCCn2cccn2)OC(C)(C)C1 41017,N1(C(=O)COCC2CCCO2)CCC2C(C1)CN2C(c1cc(CC(=O)O)c[nH]1)=O 41018,c1(OC)nccc(CNC(=O)CC2(OC)CN(C(=O)CC3CCOC3C)C2)n1 41019,N1(C(C(C#C)C2CC2)C2CCCO2)CCCC1(C)C 41020,c1(CNC(C2C(CC)CC2)=O)nnn(C)c1C(N1CCC(OC2CC2)C1)=O 41021,Cc1cc(F)c(C(N2CCC(NC(c3ncccn3)=O)C(C)C2)=O)cc1F 41022,C1(C#N)(C(N2CC(SC)C(NC(c3cnn4c3CCC4)=O)C2)=O)CCN(C)CC1 41023,CCC(C)CCCCC(=O)N(C)CC1C2CN(C(=O)C=C(C)C(F)F)CC12 41024,c1(C(=O)NC2CC(C)(NC(C3CC3c3cccs3)=O)C2)cccc2nc(O)oc12 41025,C1(C(=O)NC(C#C)(C)C2CCC2)CN(C(=O)CC2CCC(=O)C2)CC12CC2 41026,c1(CCCC)ncc(C(N2CC(C(N)=O)(CNC(=O)CC3CN(C)C3)C2)=O)s1 41027,c1(C(=O)NCC2CCCN(C(c3n(CC)ncc3)=O)CC2)cc2n(n1)CC(F)C2 41028,c1(C(=O)NC2C(NC(c3cc(CCCO)on3)=O)CCC2)ccn2c1CCCC2 41029,c1(C(=O)OCCCN(C(C)C)C)cnc(O)c2cncn12 41030,c1(C(N(CC(COCC)(C)C)C)=O)ccnnc1C.C12(CCC1)C(=O)N2 41031,C=C(CNC(=O)C(CCC1CC1)NC(C1CC(=O)CS1)=O)C(F)(F)F 41032,Cc1ccccc1C1(C(=O)NCC2CC(NC(c3n[nH]cc3Cl)=O)C2)CC1 41033,C1(CNC(COCCCC)=O)CN(C)CCN1C(c1cc(C2CC2)nc(O)c1)=O 41034,N1(C(C2(F)CN(C(c3cc(C)no3)=O)C2)=O)CC2CCC2(C)C1 41035,c1(C(=O)NCC2C3CN(C(CC(=O)NC4CC4)=O)CC32)ccc2scnc2c1 41036,N#Cc1ccc(S(=O)(=O)NCC2(F)CCCNC2)o1 41037,c1(C(=O)NC2CC(CNC(=O)CC3CCC4CC34)C2)cccn2nncc12 41038,Cc1[nH]c(C#N)cc1C(N1CCC(C)(CNC(=O)CCN2CCCCCC2)C1)=O 41039,C1(CC)CN(C(C2CCC3CC3C2)=O)CCC1Nc1nc(C)cc(C)n1 41040,C(CN=c1nc(C(F)(F)F)cc[nH]1)C1CCN(C(Cn2c(=O)cccn2)=O)CC1 41041,c1(C(=O)NCC(CC)NC(=O)CSC(F)(F)F)cn(C)c2ccc(F)cc12 41042,c1(CNC(=O)CCC(F)Cl)cccc2c1OCCC2 41043,c1(C(=O)NCCC2(C(=O)NCc3c(C)occ3)CCC2)cn(C)c(C)n1 41044,c1(C(=O)NCCCCNC(C(C)(C)OC(C)=O)=O)snc(Cl)c1Cl 41045,C1(NC(c2c(CC)c(C)sc2)=O)CCCN(C(c2ccc(=N)[nH]c2)=O)CC1 41046,C(=O)(N=c1[nH]nc(-c2ccc(OC)cc2)s1)N1C(CC(C(=O)OC)F)CC1 41047,C1(O)(CNC(c2c(CNC(C=NOC)=O)ccs2)=O)CCCC1C 41048,O=C(O)CCCCC(=O)NCc1cn(CC2CCCC2)nn1 41049,C(CC1=CCCCCC1)NC(C1(F)CN(C(c2cccc(C)c2O)=O)C1)=O 41050,C1(NC(C2(COC)CC2CO)=O)CCN(c2ccc(-n3ccnc3)cc2)C1=O 41051,Cc1nc(C(=O)NCC2(C)CCC(NC(=O)CNS(N)(=O)=O)CC2)c(C)n1C 41052,C1(CNC(=O)NC2C(CC)COC2)(NC(=O)OC(C)(C)C)CC2CCC1CC2 41053,CC1(C(=O)NC2(C(=O)NC3CCOCC3CO)CC2)CC2C=CC1C2 41054,C#CCC(CC#C)C(=O)N1CC(NC(=O)COc2cncc(C)n2)C2CC12 41055,C1(CC=C)(NC(=O)C(C)SC(F)(F)F)CCCN(C(C2CN(C(C)C)C2)=O)C1 41056,C1(NC(CCCCNC(C(c2ccn(C)n2)C)=O)=O)CCN2CCCCC12 41057,C(C)(C)(CCCNC(c1ccnc(CN(C)C)c1)=O)NC(C(CC)NC(C)=O)=O 41058,N1(C(C2(NC(C)=O)CC2)=O)CCC2(CCC2)C(CNC(c2ccco2)=O)C1 41059,N1(C(COC(C)C)=O)CCN(C(=O)CSc2cccs2)C(C)CC1C 41060,c1(NC(C2OCCC(NCc3ccn(C)n3)C2)=O)cc(Cl)ccc1NS(C)(=O)=O 41061,c1(C(C(=O)N(C(C)C)Cc2ccccn2)C)c[nH]c2ccccc12 41062,c1(OC)ccccc1-c1nc(CN(C)C(=O)N(C2CC2)Cc2cscn2)cs1 41063,C1(NC(c2c(C)oc(C(C)C)c2)=O)CCCN(C(c2[nH]nnc2C2CC2)=O)C1C 41064,CC(C)(C)C(CC(=O)NC1CCCC(NC(C23CCOC(C)(C2)C3)=O)C1)C(F)F 41065,Cc1cc(C)cc(C=CC(=O)NCC(CNC(C2C(C#N)C2(C)C)=O)CO)c1 41066,C(=O)(C1=CCCC1(C)C)N1CC(C(C)C)N(C(c2cc(F)cnc2O)=O)CC1 41067,c1(C(=O)NC(C)CN(C)C(C2CCN(C)C2)=O)cnc2ncc(Br)cc2c1 41068,N1(C(C2CN(CC)C(=O)C2)=O)CC(NC(=O)CCOCC2CC2)CCC1C 41069,CC(C)(C)C(C#N)C(=O)NCC1CC(C(=O)NC2(C3CC3)CCC2)=NO1 41070,N1(C(C2C(C=C)C2)=O)CCC2(CC1)CN(C(=O)CCCCCSC)C2C(C)C 41071,C1(OC)CCN(N2CCCCC2c2ccc(OC3CCC3)nc2)CC1 41072,c1(C(N(C)CC2OCCN(C(CCc3ncc(C)[nH]3)=O)C2)=O)cc(Cl)ccc1Cl 41073,c1(C(N2CC(N3CC(O)C3)C2)=O)cc(CNC(C2CC2(Cl)Cl)=O)no1 41074,CCC(C)CC(=O)C(=O)NCC(C(=O)NCCn1cncn1)C(C)C 41075,C(c1cccc(F)c1F)=CC(=O)NC1CCCN(C(C(C)SC(C)C)=O)C1 41076,N1(C(CCOc2c(C(C)C)cccc2)=O)CC(NC(C2CC2F)=O)CCC1C 41077,c1(C(N2C(CNC(c3cc(C(=O)OC)on3)=O)CC(O)C2)=O)ccc([N+](=O)[O-])[nH]1 41078,C1(COCC(=O)NC2CN(Cc3cocn3)C2)CCCC1 41079,c1(Cn2ncc(C(N(CCN(C)C(C3CC3Cl)=O)C)=O)c2)ccccc1Cl 41080,CC1CCN(C(C2CCCN(C(N)=O)C2)=O)CC1NC(=O)C(F)n1cccn1 41081,c1(C(=O)NC(C(=O)NCC#CC)Cn2ccnn2)oc(C)nc1C 41082,C1(NC(COCC#C)=O)CCOC(C(=O)N(C)Cc2cccn2CC)C1 41083,N1(C(C)=O)CCCC(N=c2nc(N3CCC(C)(C)C3)c3c([nH]2)CCC(C)C3)C1 41084,c1(C(=O)NC2COCCC2NC(C2(C3CCCO3)CC2)=O)cc2n(c1)CCCC2 41085,CC(CC1CCCO1)C(=O)NCC1(NC(c2cc[nH]n2)=O)CCCC1 41086,CC(C(=O)NCC1CC1CNC(C1(c2cccc(Cl)n2)CC1)=O)C(F)(F)C(F)F 41087,C(=O)(C1CS(=O)(=O)c2ccccc21)NC1C(C)(C)CCN(C(c2cnco2)=O)C1 41088,c1(C(C(=O)N(CC(C)C#N)C)NC(=O)C(F)C2CCC2)cn(C)nn1 41089,C1(C(N2CC(COC)(NC(=O)CC#N)C2)=O)CC2CCC1CC2(F)F 41090,N1(C(Cn2cc(CN3N(C)C(=O)C3)nn2)=O)CC(O)(C2(COC(C)(C)C)CC2)C1 41091,C1(CNC(C2CN(C)C2)=O)CCC2(CN(C(c3cc(=N)[nH]cc3Br)=O)C2)O1 41092,c1(C(N(C(CCNC(C2C(C)C2C)=O)C)C)=O)cc(C(N)=O)ccc1N 41093,Cc1ccc2c(c1)CCC2C(=O)NCC(O)CCNC(=O)CCOCC(C)C 41094,C(CC(C)C)(C(=O)NCC(F)C(C)(C)O)NC(C)=O.N12CC(C1)CC2=O 41095,c1(C(=O)NC2C(CNC(Cc3ccc(C)s3)=O)CC2)ccc2nccn2c1 41096,C1(CC=C)(C(=O)N(CC)Cc2ccccc2)CCCN1C(=O)CC1CSCCO1 41097,c1(C(N(C2CN(C(=O)COC(C)=O)CC2O)CC)=O)nc(C)sc1Br 41098,c1(CC(=O)N(C)N(C2CCNCC23CC3)C)cc(OC)c(NC)cc1OC.CO 41099,n1(CC)ncc(CNC(C2(OC)CCN(C(=O)Cc3cncnc3)C2)=O)c1C 41100,C=CC1(C(N2CCC(N(C)C)C2)=O)CCN(C(C2CC(N(C)C)C2)=O)C1 41101,c1(OC)nc(C)ncc1C(=O)N(CC(C)N(C)C(C1CCC2CC12)=O)C 41102,C1(CNC(C2CCC(F)(F)CC2)=O)C2CCC1CN(C(C1CC1(Cl)Cl)=O)C2 41103,C1(NC(c2n(C(C)C)ncn2)=O)CCCCC1CNC(c1cncnc1C1CC1)=O 41104,N1(C(c2cncc(OC)c2)=O)CC2CCC1C2NC(=O)CS(=O)(=O)N(C)C 41105,Cc1cc(F)cc(NC(C2CC2NC(=O)CCCn2ccnc2)=O)c1Br 41106,C1(Cn2c(C3C(NC(C)=O)C3)ccc2)CN(C(c2ccc(C)cc2)=O)CC1N=[N+]=[N-] 41107,C(=O)(CC(C)CC(C)C)N1C(CNC(c2n(C(CC)CC)ncc2)=O)CC1 41108,C1(NC(CCCc2n(C)cnn2)=O)CCCC12CN(C(=O)Cn1cccn1)C2 41109,c1(N(C)C)ccc(F)c(C(=O)NC2CN(C(=O)CCC3CC3(C)C)C(C)(C)C2)c1 41110,CCCC(CC1CCCC1)C(=O)NCC(C(C)(C)C)NC(=O)CSCC(N)=O 41111,Cc1ocnc1C(=O)N(CC(C)N(C)C(C1CC(CF)C1)=O)C 41112,C1(C(=O)NC(C)C=CC(=O)N(C)CC2CCCOC2)CCSCC1 41113,C1(C(C)NC(c2nnc(CC)s2)=O)CCN(C(c2c(C)ncn2O)=O)CC1 41114,CC1C(CNC(C2CC3(CC3)CO2)=O)CCCN1C(=O)CC(=O)N(C)C 41115,C#Cc1cnc(C(=O)NCC2(NC(=O)CC3CCCC(C)O3)CC2)c(C)c1 41116,C1(C(N2CC(OC3CCN(C(C(C4CC4)OC)=O)C3)C2)=O)COC(C)(C)O1 41117,Cn1ncc2nc(Cl)nc(N3CC(NC(=O)COC(F)F)CC4(CCC4)C3)c12 41118,C1(C(N)=O)CCN(C(c2cccnc2CNC(=O)COc2cccnc2)=O)CC1 41119,C(CN=c1[nH]c2c(c(=NC3CCCc4sccc43)[nH]1)CCC2)NC(=O)NC 41120,C(CC(C)(C)C(=O)NCCC(C)CCNC(=O)CCCCN1CCCC1)OC 41121,Cc1[nH]nc(C(=O)NC2CC(CNC(c3nscc3Br)=O)C2)c1C 41122,Cc1ncnc(C(=O)NCc2ccc(CNC(=O)C(C)C(C)O)c(F)c2)c1C 41123,c1(CCC(=O)NC23CN(C(C4CCN(C)C4)=O)C(C2)C3)ccc(Cl)cc1Cl 41124,N1(C(C2CC(NCc3ccc(F)c(C(F)(F)F)c3)C2)=O)CCC2COCC2C1 41125,N1(C(CC2(N(C(=O)CCc3cncs3)C)CC2)=O)CCCC(F)(C(N)=O)C1 41126,C1(C(N2CC(NC(c3cccc(C(=O)NC)c3)=O)C2)=O)CCCCC12CC2(F)F 41127,N1(C(C(c2ccc(Cl)s2)C)=O)CCN(C(=O)COCC(C)(C)C)C(CC2CC2)C1 41128,C1(C(=O)NCC(CC)(C)NC(c2cc([N+](=O)[O-])n[nH]2)=O)CC2CC1CC2(F)F 41129,C1(NCCN(C(C)CCCCCC=O)CC)CCc2ccccc2C1.OC 41130,C(CN=c1[nH]c(=NCCOC(F)F)[nH]c2c1COC2)(c1ccccc1Cl)N(C)C 41131,CC1CNC(=O)CN1C(C1(NC(c2coc(C(N)=O)c2)=O)CC(F)(F)C1)=O 41132,C1(CN(C)C(C2CCOCC2)=O)CCN(C(=O)CCCc2cncs2)C1 41133,C1(C(=O)NC2CCN(C(CCOC)=O)C2C(C)(C)C)CN(C)C(=O)CCO1 41134,C1(SC)CN(C(c2ccnc(S)c2)=O)CC1NC(c1cn(C)c(C)n1)=O 41135,CCC(CC)(CCNC(=O)C(F)C(C)C)NC(c1ccc(C2CCC2)cc1)=O 41136,Cc1ccnc(O)c1C(=O)NCC1C(C)CCCN1C(=O)C(C)OC1COC1 41137,C1(C(=O)NCCn2cc(-c3cn[nH]c3)nn2)CCCN1CC(F)F 41138,c1(CC)ccc(C(=O)C(=O)NC23CC(CNC(c4ncsc4C)=O)(C2)C3)s1 41139,Cc1coc(C)c1C=CC(=O)NC1(CCNC(=O)CCCN(CCO)C(C)C)CC1 41140,C1(OCC#C)CCCN(C(C2CCC(CNC(=O)C(C)O)C2)=O)C1 41141,Cn1nccc1CC(N1CSCC1C(=O)NOC1CCOC1)=O 41142,c1(NC(=O)C(C)CNC(C2(CC=C)CN(CC)C2)=O)cc(N)c(C)cc1C 41143,CCC(C)C(C(=O)N(C)Cc1ncn(C)n1)N(C)C(C1CCC(OC)CC1)=O 41144,CN1CCC(C(N2CCN(C(=O)CCc3cncc(O)c3)C(C3CC3)C2)=O)CC1=O 41145,c1(C(=O)NCc2c(OC)c(F)ccc2F)cnc2ccc(Br)cc2c1 41146,Cc1c(CC(=O)NC(CNC(=O)CC2CC(=O)NC2=O)C2CC2)cnn1C 41147,C(CCCCC(=O)NCC(C)(C(C)C)NC(c1c(C)nn(C2CC2)c1Cl)=O)OC 41148,C1(NC(C2(COC)C=CCN2C(=O)CC(C)C2CC2)=O)CC2CC1C(O)C2O 41149,CC1(C)CCC(C(N2CC(C(N)=O)(CNC(=O)CCC3CCCCO3)C2)=O)OC1 41150,c1(N(C)C)cc(Br)ccc1CN1CC(C(=O)NCc2ccccc2Br)CC(F)C1 41151,C(=O)(CC1=CCCCC1)N1C(C(C)NC(=O)C2=CSCS2)CCCC1 41152,c1(C2CC(C(N3CCC(C(=O)C4CC4)CC3)=O)C2)cc(Cl)c(O)c(Cl)c1 41153,CC1C(NC(=O)Cc2csc(Cl)c2)CCN1C(=O)CCc1cccs1 41154,c1(CC)ncc(C(N2CCC(CCN(C)C(c3ncccn3)=O)CC2)=O)c(C)n1 41155,C1(CNC(c2c(C)ncn2C)=O)CC2(CCN(C(=O)C(C#N)C(C)C)CC2)CO1 41156,C(=O)(C(C(C)C)n1cnnn1)NCC(CCNC(C1CCN(C2COC2)C1)=O)OC 41157,N1(C(c2cc(CCC)[nH]n2)=O)CCC(C)(NC(=O)CCCOC(C)(C)C)C1 41158,c1(OC)ccc(Br)cc1S(=O)(=O)Nc1ccc(C(=O)NCC2COCCO2)cn1 41159,c1(N(C)CC2CCCO2)nnc(-c2ccccc2Br)n1CCN1CCCS1(=O)=O 41160,C1(C(=O)NC2CCN(c3ncccn3)C2)CCS(=O)(=O)C12CCC2 41161,C(=O)(CCCC(=O)OC(C)(C)C)NCCC(C)CCNC(C1CC(=O)N(O)C1)=O 41162,C(=O)(C1=C(Cl)CC1)N(C1CN(C(C(C)CC2CC2)=O)C1)C 41163,C1(C(=O)NCCC(C)(C)NC(=O)C=C(Cl)Cl)CC(C(C)(C)C)=NO1 41164,c1(N(CCC(C)O)C)nc(=NCCc2ccns2)[nH]c2c1SCC2 41165,C1(C(C)C)N(C(=O)N(c2ccncc2Br)C)CC12CCC2 41166,c1(SCC2N(C(C=COCC)=O)CCC2)ccc(F)cc1O 41167,CC1CC(=O)NC1C(=O)NCCCNC(=O)CCOc1cccc(Cl)c1 41168,c1(C(=O)NCC2CCN(C(C3(C)ON=C(C)C3)=O)CC2O)cc(F)c(F)cc1O 41169,c1(OC)cc(C(=O)NC2CCC2NC(=O)COC(c2nccn2C)C)cc(C)n1 41170,C12(C(=O)NCC(CNC(CCCOC(C)C)=O)F)CC3CC(F)(C1)CC(F)(C3)C2 41171,C(=O)(C1=C(C)OCC1)NC1(COC)CN(C(=O)CC2CCOC2=O)C1 41172,CC1CCCC(C(=O)OC(=O)C2CC2)C1.N12CCN(CC1)CC(=O)NC1CN2C1 41173,N1(C(C(C2CC2)OC)=O)CC(O)(CNC(C2(CO)CCC2)=O)C1 41174,c1(OC)nc(C(N2CC(F)(CNC(=O)C(C)(CO)NC(C)=O)C2)=O)sc1C 41175,Cn1ncc([N+](=O)[O-])c1-c1nc2ccccc2n1CCCCC(=O)O 41176,C1(C(=O)NCCN(C(=O)CN(c2ccc(Br)cn2)C)CC)COCC(C)(C)O1 41177,c1(C(N(CCN(C(C(C=C)O)=O)C)C)=O)ccc(F)cc1C#N 41178,N1(C(c2cc(C)c(F)cc2F)=O)CCC2C(CCN2C(C2COCCO2)=O)C1 41179,C1(NC(C(C)SC)=O)CC(C(=O)NOCC(F)F)C1(C)C 41180,c1(CC=C)ccc(SCc2cncn2C(C)C)cc1 41181,N1(C(c2c(C)con2)=O)CC2COCC2(C(=O)NC(C)CC2CCC2)C1 41182,C(=O)(CCCCCS(N)(=O)=O)N1C(C(C)(C)NC(C(C)O)=O)CCC1 41183,c1(C(=O)NC2CC(CNC(C(CC)SC)=O)C2)oc2c(C)ccc(C)c2c1C 41184,C(CC(O)C(=O)Nc1cccc(NC(C2CCC(=O)N2C(C)C)=O)c1)SC 41185,CC(C)CC(C)(CNC(c1cn(C2CC2)nn1)=O)NC(=O)CC1CCC(=O)NC1 41186,C1(C(=O)NC(CNC(c2cn(CC=C)nn2)=O)C(C)(C)C)CC2(C)CC1CO2 41187,c1(OC)ccc(CCC(=O)NC2CCC2NC(=O)COc2ccc(F)cc2)cn1 41188,N1(C(c2nn(CC)c(=O)cc2)=O)CCOC2CCN(C(C3(O)CCCC3)=O)CC12 41189,N1(C(C2C(C)OC(=O)N2)=O)CC2CCN(C(C34CC(CO)(C3)C4)=O)CC12 41190,CC1C(=O)CCC1CC(=O)NCC1CC(NC(c2coc(C3CCC3)n2)=O)C1 41191,N1(C(C=CCN(CC(F)(F)F)C)=O)CC(F)(c2ccncc2)C1 41192,C1(CNC(CC2(CC(=O)OC)CCCC2)=O)CC(F)CN1C(c1cc(F)c[nH]1)=O 41193,C1(C(N2CCCC(C)(NC(c3cc[nH]n3)=O)C2)=O)CC2(C1)CC21CCC1 41194,C1(NC(c2ccc(C(F)(F)F)cn2)=O)CC(CNC(C2CC(O)C2)=O)C(O)C1 41195,c1(CC(N2C(CO)CC(NC(C3CC(Cl)(Cl)C3)=O)C2)=O)c[nH]c2cccnc12 41196,c1(CNc2ccc(-c3c(OC)cccc3)cn2)ccc(Cl)cc1O 41197,Cc1cc(=NC(=O)c2cc(CNC(=O)CCc3ccnn3C)on2)[nH]n1C 41198,N1(C(C(C)=C(CC)C)=O)CCN(C(C2CCN(CCC)CC2)=O)C(C(C)C)C1 41199,c1(CC)cc(F)ccc1CC(=O)NCCC(O)CNC(=O)C1=COCCO1 41200,Nc1cc(C(=O)NCCNC(=O)CC2CC3CC3C2)cc(C(F)(F)F)c1 41201,CCC1=C(C(=O)N2CCCCC2C2(NC(=O)CCCOC)CC2)CCCO1 41202,C(C(CC1CC1)C(=O)Nc1cscc1C1CC1)NC(C(C)Cn1ccnc1)=O 41203,CCC(CC)C(C)C(=O)NCCOC1CCN(C(C2(c3cc(C)on3)CC2)=O)C1 41204,N1(C(C(C)=C(CC)C)=O)CC2(NC(=O)CCc3cccc(Cl)c3)CC1C2 41205,Cn1ccc2ccc(C(N3CCC4(CCCC4NC(=O)CC(C)(C)C)C3)=O)cc12 41206,c1(NC2(c3n(CCOC)nnn3)CCCC2)cnc(Cl)c(Br)c1C 41207,C1(NC(C2C(C)(CC)C2)=O)CCC2CN(C(C3CC3(F)F)=O)CC2C1 41208,N1(C(C(C(C)C)S)=O)CCCC2(C1)CN(C(=O)C(c1ccccn1)C)CCO2 41209,C(=O)(C(C)S(=O)(=O)CCC)N1CCC2CN(C(CC3CC(=C)C3)=O)CC21 41210,CC(=O)CCCCCCC(=O)NC1CCCC(NC(=O)C(C)C(C)O)C1 41211,c1(C(=O)NC2(CO)CN(C(CSc3n(C)cnn3)=O)C2)cccc(C2COC2)c1 41212,CC1(C)CN(N2CCCC(CCF)C2)CCS1=O 41213,N=c1[nH]c2c(s1)CCCC2C(=O)N1CCCC(F)(CNC(=O)Cc2ccsc2)CC1 41214,c1(-c2cc(NC(C3CC(C(=O)OC)C3)=O)sc2)ccc(OC(C)C)nc1 41215,C1(C(N(C2CCN(CCCSC3CCC(C)O3)C2)CC)=O)CC=CCC1 41216,C1(C(=O)NCC(CC(F)(F)F)NC(C2(CC)CC2)=O)CCCC2(CCC2)C1 41217,C#Cc1ccccc1CC(=O)NCC1CCCCN1C(c1c[nH]ccc1=O)=O 41218,CC1CN(C(c2cn(CCNC(C3CNC(=O)N3)=O)cn2)=O)CCO1 41219,C1(OC)CCCN(C(=O)Cn2cc(CNC(c3cn(C)nc3OC)=O)nn2)C1 41220,c1(C(N2CCCC(O)(CNC(C3CC34CCCC4)=O)C2)=O)cc2n(n1)CCOC2 41221,Cn1cc2cccc(NC(C3CCC4(CN(C(=O)CCC(N)=O)C4)O3)=O)c2n1 41222,n1(CC)cc(-c2noc(C3CC3OC(C)C)n2)cn1 41223,C(=O)(C(C)S(=O)(=O)c1ccc(F)cc1)NC12CN(C(CC(C=C)C)=O)C(C1)C2 41224,c1(C(=O)NCC(C)(C)NC(=O)CSC2CCOC2=O)cnc2ncnn2c1O 41225,N1(CCC(=O)NCC(CN(C(=O)C(c2nc(=N)[nH][nH]2)(C)C)C)O)CCN(C)CC1 41226,C1(C)(C(=O)NCC(C)=CC(=O)NCC(C)C)CCCO1 41227,N1(c2c(OC)cncn2)CCC(C2CC2)(CNC(c2ncoc2C(F)(F)F)=O)C1 41228,C1(OC)CCC2(C(=O)NC(C)(C)C(=O)NC(Cc3ccco3)CO)CC12 41229,N1(C(c2ccc(C)o2)=O)CCN(C(c2c(F)cccc2I)=O)C(C#N)C1 41230,N1(C(c2cccc(Cl)c2C(F)F)=O)CC2(CCC(CNC(C3CC34CC4)=O)O2)C1 41231,N1(C(c2c(CC)onc2)=O)CC2CC(C1)N(C(c1cccc3cnsc13)=O)C2 41232,c1(NC(C(=O)NC(c2ccc(OC)cc2)CC#N)=O)cc(C)ccc1C 41233,c1(C(=O)NC2CN(C(C(C(C)C)OC)=O)CC2C)cncc2c(O)nccc12 41234,C1(N(C(=O)CSCC2CCCCO2)CC)CCCN(C(=O)C(C)(C)O)CC1 41235,N1(C(CS(N)(=O)=O)=O)CCC([SH](CCN2CCCC2=O)C2CC2)CC12CC2 41236,C1(O)(CN(C(C(CCC)O)=O)C)CCN(C(c2cc(C)c(CC)s2)=O)CC1 41237,c1(C(N(C2CC(NC(c3c[nH]ccc3=N)=O)C2)C)=O)ccc2c(c1)CCO2 41238,N(C(=NCCN1CCCC1)NCC1CCCC1C)Cc1c(OCF)ccc(Cl)c1 41239,c1(C(=O)NCCC2(OC)CN(C(=O)Cc3ncc(Cl)s3)C2)cccc2c1NCC2 41240,C1(CNC(C(=O)N(C)Cc2ccc(CO)cc2)=O)CCC(C)(C)CC1 41241,CC1CCN(C(=O)C(C)N(C)C)C(CNC(c2cc(=O)c(Br)c[nH]2)=O)C1 41242,C(CCC(=O)NCc1nocc1C(=O)NC1CCCSC1)OC(C)=O 41243,c1(C(=O)NCC2N(C(CCCCOC(C)C)=O)CCCC2)nc2c(s1)COCC2 41244,c1(C2C(C(=O)NC3(C)CN(C(c4cn(CC)nn4)=O)C3)C2)cccc2[nH]ncc12 41245,C(=O)(C1=CC2CCCCCC12)N(CCNC(CS(C(C)(C)C)(=O)=O)=O)C1CC1 41246,N1(C(C23N(C(c4ccc(OC)o4)=O)CC(CO)(C2)C3)=O)CCC2(CC2)CC1C 41247,N1(C(=O)Nc2cnn(-c3cccc(C)c3)c2C)CCN(C(=O)C2CC2)CC(O)C1 41248,c1(OC)ncc(-c2nc(C)c(NC(c3nccc(Cl)c3Cl)=O)s2)cc1C 41249,C1(C(=O)NC2CC(NC(CN3CCC(C)CC3)=O)CC2O)SC2C=CC1CC2 41250,N12CCOCC1(C)c1cn(nn1)SC(C)C2=O.C1(NC(N)=O)CCOC1 41251,C(=O)(N=c1[nH][nH]c2cc(C#N)ccc12)C1(C)CNC1.c1(C)ccnc(Cl)c1Br 41252,c1(NC(C2CCN(Cc3c(Cl)cccc3Br)C2)=O)cc(Br)cc(F)c1O 41253,C12(NC(C(COC)C)=O)CC1CN(C(=O)C(c1ccnn1C)O)C2 41254,N1(C(C=Cc2n(C)cnc2)=O)CCN(C(=O)C(O)CF)C(c2ccccc2)C1 41255,c1(C(=O)NCCC(C)N(C(=O)CC2CCCC(=O)N2)C)cccc2[nH]nc(O)c12 41256,C(CCC(=O)N1CCCC1CCCNC)N(C=O)CCO.C1(C)(SC)CSC1 41257,CCC(CCC(=O)NC1C2CN(C(c3cncn(C)c3=O)=O)CC12)NC(C)=O 41258,C(c1cc2ccccc2o1)=CC(N1CC(CNC(C(C=C)(C)C)=O)C(O)C1)=O 41259,C(CCCC(CO)NC(C1(N2CCCC2)CC1)=O)NC(CC(CC)SC)=O 41260,CCCCCC(F)C(=O)NCCC(C)(C)C(=O)N(C)Cc1ccsc1 41261,C=CCC(C)(C)C(=O)N1CCCOC(CNC(C2CC2C(C)O)=O)C1 41262,C1(C(=O)NCCC(C)NC(CCN(CCC)C)=O)CCCSC1 41263,c1(CC)sc(C(=O)NC(C)CCNC(c2nnsc2C)=O)cc1Br 41264,C1(NC(CCOCC#C)=O)CC(NC(=O)C(C)Cc2cccc(Cl)c2)C(O)C1 41265,CC1(C(=O)NCc2cc(Br)cs2)CC(NC(=O)Cc2ccon2)C1 41266,N1(C(C(C)CC(N)=O)=O)CC2CC(NC(=O)C=Cc3cnn(C)c3)CC1C2 41267,C(CC1CC1)(C(=O)NC(c1ccccc1)CCNC(C1(OC)CC1)=O)OC 41268,C1(NC(=O)NC(CN(C)C)C2(c3cc(C)c(O)nn3)CC2)CCc2ncsc2C1 41269,C(=O)(CS(=O)CCC(F)(F)F)NCC(C1CC1)NC(CCC(N)=O)=O 41270,C=CCCCCCNC(c1csc(COC)n1)c1nnnn1C1COC1 41271,O(NC(=O)CC(CC=C)NC(=O)CC1CCOCC1)CC(=O)OCC#C 41272,c1(C(c2ccco2)NC(C(C)(C2CC2)OC)C)ccc(S(N)(=O)=O)cc1 41273,CC1CN(C(=O)CCOc2ccc(F)cc2)CCCN1C(=O)C(N)=O 41274,c1(CC)ncsc1C(=O)NC(C)(CNC(C1CCCC1CC)=O)CO 41275,C1(S(N)(=O)=O)(C(=O)NC(C(C)NC(c2cccc(C(F)F)c2)=O)C)CCCC1 41276,C12(CNC(CC3N(C)CCC3)=O)CCC(CC1)CN2C(c1cnc(S)[nH]1)=O 41277,C(=O)(C1=C(Cl)CCOC1)NC1CCN(C(C(c2ccncc2)C)=O)C(C)C1 41278,CC(C)C(C(=O)NCC1CN(C(C23CCC(C2)OC3)=O)C1)n1cccc1 41279,C1(CNC(C=C(CCC)C)=O)OCCC1C(N1CC(N2CC(F)C2)C1)=O 41280,C1(C(=O)NCCn2c(C)cnn2)CCN(C(=O)CCc2cccn2C)C1C 41281,N1(C(=O)OC(C)(C)C)CC2CCC1C2C(N1CC(CNC(=O)C(N)=O)C(C)C1)=O 41282,C1(C(=O)NCCCc2cc[nH]n2)CC2CC1CN(C(=O)Cn1cnnc1)C2 41283,C=CCCC(C(=O)N(CC(C)(C)OC)C)NC(c1cnc(OC)s1)=O 41284,C1(CNC(CN(C)C)=O)CN(C(c2ncc3ccccn23)=O)CCC12CCOC2 41285,CC1(C)CC(NC(=O)C(N)=O)CCN(C(c2ccnc(F)c2O)=O)C1 41286,C1(C(=O)NC(CC=C)CNC(C2CC(=O)OC2(C)C)=O)CC2(CCCC2)CO1 41287,C(=O)(C1CCCc2c[nH]nc21)NC(C)CNC(=O)CNC(=O)C(F)(F)F 41288,N1(C(C)C(N2CCN(c3ccc4nncn4n3)CC2)=O)CC(SC)CC(C)(C)C1 41289,CC1(CCC(=O)NCC2CCC2NC(=O)CCCc2csc(=N)[nH]2)CCC(=O)N1 41290,CC1(OC(F)F)CCN(C(=O)NCC2(C)CCCOC2)CC1 41291,c1(C(N2CCCC(n3cc(C(C)OC)nn3)C2)=O)cc(O)nc(Cl)c1 41292,C=CCC(CNC(C1CCSCC1)=O)NC(=O)C(C1CC1)SC 41293,C1(NC(C2C(C)=C2)=O)CN(C(c2ccnc(OCCOC)c2)=O)CC1C 41294,C(=O)(N1CC(n2cc(CCCC#N)nn2)CO1)C1CCC(CC)O1 41295,c1(C(=O)NCCOC2CCN(C(c3ccc(CC)o3)=O)C2)cccc(CO)c1C 41296,N1(CC(=O)NC(CNC(C(c2cn(C)nc2)O)=O)(C)C)CCC(C)(C)C1 41297,CC1(C)Cc2ccsc2CN1C(c1c(O)cccc1O)=O 41298,C1(O)(C(C)NC(=O)CCC2CCCO2)CCN(C(=O)COCc2nccn2C)C1 41299,CN(CCCC(=O)N1CCCCC(NC(C2CCCN2CC(F)(F)F)=O)C1)N=O 41300,c1(C(C(=O)NC(C)C(CO)NC(=O)C=CCN2CCCC2)O)ccccc1F 41301,N1(Cc2c3ccc(OC)cc3ccc2)CCC(N=c2[nH]cnc3cc(I)sc23)C1 41302,c1(C(N(C(C)CNC(=O)C(C2CCCC2)N(C2CCCC2)C)C)=O)ccccn1 41303,C(=O)(C1=CC2(CCOC2)C1)NC1(C(=O)NCC=CC)CCC(C)(C)C1 41304,c1(C(=O)NCC2(F)CN(C(C3(CC(C)C)CC3)=O)C2)ncccc1F 41305,C1(CNC(CC2(C)CC2(F)Cl)=O)CCC(CNC(C2(F)CCCCC2)=O)CC1 41306,c1(C(=O)NCC2CCC(C(=O)NCC(C)(C)CO)O2)ncn2ccccc12 41307,c1(C(N2CCCN(C(N)=O)CC2)C(=O)Nc2c(C)cccc2)cc(F)ccn1 41308,C(=O)(C(CC(C)C)N(C)C(c1cc(CO)on1)=O)N1CCC(C(CC)C)CC1 41309,Cc1cc(C(=O)NC2CN(C(=O)CC3CCCN3C)CC2F)c(O)nn1 41310,N1(C(C(C)OCC=C)=O)CC2CC(O)C1C2NC(c1cc(C)sn1)=O 41311,C1(OC2CN(C(=O)OC(C)(C)C)C2)CCC(CC(=O)NCC2C3CCC23)CC1 41312,C12(CNC(CCOCC)=O)CCC(C1)N(C(c1ccc(C(F)F)nc1O)=O)C2 41313,N1(C(c2ccc(OC)c(O)c2)=O)CC2OCCN(C(=O)COCCF)C2C1 41314,c1(CC(N2CC(C(=O)Nc3n(C)nc(C)c3Cl)NCC2)=O)ccc2c(c1)CCO2 41315,c1(CCCCCC)ccc(C(N2CC3CC2C3C(=O)Nc2ccncn2)=O)cc1 41316,C1(C)(NC(C2C(NC(CCCNC(C)=O)=O)COC2)=O)C=CCCC1 41317,N1(C(CC(=O)OCC)=O)CCC=C(CNC(=O)C(C)CC2CCC2)C1 41318,N1(C(c2c(C)n[nH]c2)=O)CC2CCCCN2CC1CNC(c1cc(O)ncn1)=O 41319,C1(C(=O)NCc2nc(C(N3CC(n4ccnc4)C3)=O)co2)COCCOC1 41320,C1(CNC(c2nccc(C)c2)=O)CCC(C)(C)CN1C(C1CCOC(C)(C)C1)=O 41321,C(C)(C(=O)NC1COCCN(C(=O)Cc2cc(F)ccc2Cl)C1)(C(C)C)OC 41322,N1(C(c2cc(C)ncc2)=O)CCN(C(=O)C(C2CCCCC2)O)C(CC2CC2)C1 41323,c1(N2CC3N(c4nc(C)cc(OCC)n4)C3C2)ncc2cc(Br)cc(F)c2n1 41324,c1(C(N2CC(CC(C)NC(=O)C=Cc3cn[nH]c3)C2)=O)c(F)cccc1F 41325,c1(OC(C(=O)OC)(C)CNc2ccccc2OC)ccc(S(C)(=O)=O)cc1 41326,N1(CC(C)CC2CCCO2)CC2(C1)CC(C)(C)C2 41327,CC(O)(C(=O)NC1C=CC(C(=O)Nc2cc(C(F)(F)F)cc(I)c2)C1)C(F)(F)F 41328,N1(C(CCNC(=O)OCC)=O)CC(OC)CC(NC(=O)CC2CCC(C)CC2)C1 41329,C(=O)(CCCCCc1ccc(OC)cc1)NC1CC(C)(NC(C(C=C=C)C)=O)C1 41330,c1(C(=O)NC2C(NC(C3(C(C)=O)CC3)=O)CCCC2)ccc(F)c(C#N)c1 41331,C1(Cl)(C(=O)NCC2C(CNC(C3CCCC3)=O)C2)CC12CCOCC2 41332,CC(C(C)C(=O)N1CC(C(C)NC(C23CCCCN2CCC3)=O)C1)S(C)(=O)=O 41333,O=C1Nc2ccc(C(N3CCCC3(C)CNC(=O)CC3CC=CC3)=O)cc2CO1 41334,C(CCN=c1[nH]c(N2CCOCC3(CCCCC3)C2)nc2ccccc12)OC=C 41335,CN1CCN(C(C2(C3CC3)CC(=O)C2)=O)CC1C(N1CCC(C(=O)NC2CC2)C1)=O 41336,c1(C(=O)NC2C(NC(c3n(OC)cnc3C)=O)COC2)cnc(O)n(C)c1=O 41337,c1(C(=O)NCC#CCNC(CN(C)CC)=O)cc(F)c(C(F)(F)F)cc1F 41338,C1(CC=C)(C(=O)NCC2(F)CC(NC(c3coc(C(F)F)n3)=O)C2)CC=CC1 41339,c1(C(N2CC3C(CNC(c4cn(CC)nn4)=O)(C3)C2)=O)ncc(F)cc1F 41340,N1(C(c2cnn(C)c2Cl)=O)CC2=C(C1)CN(C(=O)CP(C)(C)=O)C2 41341,C1(NC(c2c(C)nc(C)o2)=O)CCN(C(=O)Cc2cc[nH]n2)C12CCC2 41342,C1(N(C)C)CC(NC(=O)CNC(C2(C)CCCO2)=O)CN(C(=O)OC(C)(C)C)C1 41343,C1(NC(CC2CC(=C)C2)=O)CC2CCCC(C1)N2C(C1CCN(CC(C)C)C1)=O 41344,N1(C(C=CC)=O)CCN(C(c2cc(C)c(C(F)F)cn2)=O)CC(CO)C1 41345,Cc1cc(CC(=O)NC(C)(C)CNC(C2CCCC(C)(C)O2)=O)ccc1O 41346,c1(OC)cc(F)ccc1CC(=O)NC1CC1NC(c1nccnc1C(N)=O)=O 41347,c1(C(N2CCC(NC(C(C)c3ccsn3)=O)C2)=O)c(N)cc(F)cc1Cl 41348,C1(CC(=O)NCC2CC(NC(CN(CCC#C)C)=O)C2)CCCCC12CC2 41349,c1(C(N2CC(CC)C(NC(C)=O)CC2)=O)ccc2cnn(CCO)c2c1 41350,C(=O)(C1CC(=O)Nc2ncccc21)NCCCN(C(C1CC(C)(CC)C1)=O)C 41351,N1(C(Cc2c(C)cccn2)=O)CCOC(C)(CNC(C2CCC(F)(F)CC2)=O)C1 41352,N1(C(c2c(CC)c[nH]n2)=O)CCN(C(=O)C(C(C)O)N(C)C)C2(CC2)C1 41353,c1(OC)cccc(Br)c1C(=O)NC12CC1CN(C(=O)C(=O)Nc1ccccc1)C2 41354,CC1C(=O)CCC(C(=O)N(CCCC(=O)O)Cc2ccc(F)cc2)C1(C)C 41355,C=C1CC(CC(=O)NCCC2(CNC(=O)C=C(C)C(F)F)CC2)C1 41356,CC1=CCC(CNC(c2cc(CNC(c3cc(C#N)cs3)=O)ccn2)=O)CC1 41357,C#CCCC(C(=O)NCC1(CSC)CC1)NC(=O)C=CC(C)C 41358,c1(C(=O)NC(CNC(C2(C(=O)NC)CC2)=O)C)ccc2c(c1)C(=O)CCN2 41359,c1(CN(C2CCN(c3ccnc(N4CCCCC4)n3)C2C)C)ccccc1I 41360,CCC(C)C(O)C(=O)NCC1CCN(C(=O)Cc2ccccc2CC(N)=O)CC1 41361,c1(CNC(=O)NC(C)CC#N)ccccc1OCCc1cccnc1 41362,c1(C(=O)NCC(CC)NC(C(C)OCC)=O)[nH]c2c(c1C)C(=O)CC(C)(C)C2 41363,CC(C)CC(C(=O)NCc1ccc(C(=O)NCC(=O)N(C)C)cc1)C(N)=O 41364,CCCC(C(=O)NCC1(NC(=O)C(C)NC(N)=O)CCCC1)OCC 41365,Cc1c(Cl)ccc(C(N2CCOCC2C2(C(=O)O)CCC2)=O)c1N 41366,N1(C(c2cccc(NC)n2)=O)CCC2CCN(C(=O)Cc3sccc3Cl)C2C1 41367,CCCC(CO)NC(=O)NCC(n1ccnn1)C 41368,C(=O)(CC(F)(F)C(F)F)NC(CCN(C(C(CC#C)O)=O)C)(C)C 41369,C12(C(=O)NCC3(O)CCOC3)CC(NC(=O)C=CCN3CCC3)(C1)C2 41370,C1(NC(C(C)SCC)=O)CC2CC1CN(C(c1cc(C#N)cc(C)n1)=O)C2 41371,C1(C(=O)NCCCN(C(C)C)C(C2CCCCCCC2)=O)CC2(CCC2)C(=O)O1 41372,c1(C(=O)NC2CN(C(C3(O)C(C)(C)C3)=O)CC(F)C2)cc(F)c(F)cc1F 41373,C1(NC(=O)COc2cccc(C(F)(F)F)c2)CC2CCC1N(C(C1CC(O)C1)=O)C2 41374,C12(C(=O)NC(CCNC(C(C=C=C)C)=O)C)CC3CC(CC1C3)C2 41375,CC(CC(=O)NCc1ncccc1CNC(=O)C=CCOCC(F)(F)F)C(F)F 41376,C(=O)(CC(O)CNC(=O)C(CC)OCC)N1CC(N(CC=C)C)C1 41377,CC1CC(C(N2CCC(C(=O)NCCCOC(=N)O)CC2)=O)CCO1 41378,C1(C(N(CCN(C(C(CC=CCC)C)=O)C(C)C)C)=O)CCC(C)=C(C)C1 41379,C12(CNC(=O)CC3CNC(=O)C3)CC1CN(C(C13CC(C1)C(C(F)(F)F)O3)=O)C2 41380,N1(C(C(C)=C(C)C)=O)CCN(C(C2CC3CC3C2)=O)C(c2ccc(F)c(F)c2)C1 41381,C=C=CC(C)C(=O)NC1CC1CNC(=O)Cc1cc(Cl)sc1Cl 41382,C1(NC(CN(C)C2CC2)=O)CCC(N(C)C(c2cnc(-c3ccsc3)s2)=O)C1 41383,c1(COC(C)C(=O)NC2(CN(C)C(C3CS(=O)C3)=O)CC2)ccccc1 41384,S(=O)(=O)(c1ccnc(C(=O)OCCCC(F)F)c1)NC 41385,C(=O)(C1=NOC2(CCCN(C(=O)C(O)Cc3cccc(Cl)c3)C2)C1)NCCSC 41386,Cc1cccc(N(C)C(C2CSCN2C(=O)CC2OCCC2(C)C)=O)c1C 41387,C(=O)(C1CCc2ccc(Cl)nc21)NC1(CCO)CN(C(C(CCC)C)=O)C1 41388,c1(C(N2CC3C(NC(C4C(C)(C)CO4)=O)C3C2)=O)ccc2c(c1)CCCC2 41389,c1(C(N2CCC(Cc3ccccc3)C(O)C2)=O)cc(Br)ccc1C1CNC1 41390,CCCCC(CNC(c1c(C2CC2)noc1C)=O)NC(=O)C(C)OCC1CC1 41391,Cc1cc(S(N)(=O)=O)oc1C(=O)NC1CCC(NC(=O)C2=CCOCC2)CC1 41392,c1(OC)cc(N)ccc1C(=O)NC1CC(C)(NC(C2CCCCC2O)=O)C1 41393,CCC(CC(=O)NC1CC(CCC(=O)NCCOC2CCCC2)C1)C1CCC1 41394,C#Cc1ccc(F)c(C(=O)NCC2CC(OC)CN2C(c2cnn(C)c2N)=O)c1 41395,CCC(CCOC)C(=O)NC1C=CCN(C(=O)CC(C)(F)F)C1 41396,C1(C(N2CCC(NC(CCc3nc(C)sc3)=O)C2C)=O)CCc2nc[nH]c2C1 41397,c1(CN(CCCNC(=O)OC(C)(C)C)C(=O)C2CC2)ccccc1.c1(=O)c(=O)[nH]1 41398,N1(C(c2cc(C)c(F)nc2)=O)CCc2ccccc2C1CNC(=O)C1=COCC1 41399,C(=O)(C#CC1(C)CCCO1)NC(C)CCCNC(c1coc(C2CCCC2)n1)=O 41400,CC1(C)CCN(C(C2CCC(F)C2)=O)CC1CNC(c1cc(C2CC2)on1)=O 41401,c1(C(N(CC(C)O)CC)=O)c(CNC(=O)COCCCF)nnn1C 41402,c1(C(=O)NC(CC)(C)CNC(=O)COCC2CCOC2)ccc(CO)c(Cl)c1 41403,N1(C(C(C)(c2ccccc2)OC)=O)CCC2(CCC(=O)NC2)C1 41404,Cc1ccc(F)c(C(N2CCCC2CNC(C2CCS(=O)(=O)N2C)=O)=O)c1F 41405,C(=O)(C1OCCc2c(O)cccc21)N1C2CN(C(C3CCC(=O)N3)=O)C(CC2)C1 41406,C1(CC)CCN(C(=O)C(c2ccoc2)NC(c2ccc(COC(C)=O)o2)=O)CC1 41407,C#CC1(NC(=O)C=Cc2c(F)cccc2F)CC2(CCCC2)C1 41408,c1(NC(CCSCCCC)=O)cccc(NC(c2cc(Br)sn2)=O)c1 41409,Cc1ncc2n1CCN(C(C1CCCC1CNC(C1(C3CC3)CC(=O)C1)=O)=O)C2 41410,C(=O)(CC(C)(C)CC(F)F)N1CCCCC(NC(c2c(C)cc(C)nc2O)=O)C1 41411,C1(C(N(C)CC2N(C(c3c(C)nc(C4CC4)o3)=O)CCC2)=O)CCN(C)S1(=O)=O 41412,N1(C(=O)CCc2ccccc2O)CCCC(C2CC2NC(C2(C3CC3)CC2)=O)C1 41413,CN1CC=C(CC(=O)N2CCC(CN(C)C(C3Cc4ccncc4N3)=O)C2)CC1 41414,C12(C(NOCCOCC)=O)CC1CCN2C(C1(CO)CC1)=O 41415,N1(C(C2(CCOCC)CCCC2)=O)CCN(C(C2CCC23CCC3)=O)CC1C 41416,C(CCCCCNC(C1CCCCN1C(C)C)=O)NC(C1(COCC)CCC1)=O 41417,Cc1cc(C)c(C(N2CC(N3CCN(C(=O)C(F)(F)CN(C)C)CC3)C2)=O)o1 41418,C1(N(C(C(C)n2cccn2)=O)C)CC2CCC(C1)N2C(C1(O)CCOCC1)=O 41419,C1(NC(c2c(CNC(CCC3CC(C)C3)=O)ocn2)=O)CCC(C#N)CC1 41420,Cc1ccc(F)c(CC(N2CC(CNC(=O)Cc3nncn3C)C3(CC3)C2)=O)c1 41421,N1(C(=O)OC(C)(C)C)CCC(n2cc(CCNC(C(N)=O)c3ccc[nH]3)nn2)C1 41422,C1(CNC(=NC)NC2COCC2OC)CC2(CCOCC2)O1 41423,CC(N=[N+]=[N-])C(=O)NC(CNC(=O)CC1COCCOC1)C1CC1 41424,CCCCCCC(F)C(=O)NC(C)CN(C(=O)Cc1nc2ncccn2n1)CC 41425,C1(C(N(CC(C)CNC(c2csc(S)n2)=O)C)=O)COC(C)(C)C1 41426,CCC(CNC(c1cn(C)nc1OC)=O)(CC)NC(=O)C(C)C(=O)OC 41427,N1(C(CC(CC)O)=O)CCCC2(CCCCN2C(C2CCCN(C)C2)=O)C1 41428,Cc1ncc(C(=O)NC(CC(C)C)C(=O)NCCN(C2CCOC2)C)c(=N)[nH]1 41429,C12(CNC(=O)CCNC(C3CCOCC3)=O)CC1CN(C(=O)C1=CCSC1)C2 41430,c1(CN=C(NC(CC)CC)N(C)Cc2cc(Cl)cn2C)cccc2cc[nH]c12 41431,C1(CC(N2CCC(CC(=O)NC(C3CCCC3O)C)C2)=O)CCCC2CC12 41432,c1(NC(c2c(CCC)occ2)=O)cccc(NC(=O)C(C(=O)OC)OC)c1 41433,N1(C(C(CC#C)O)=O)CC2CCC(CNC(c3cc(C4CC4)ncn3)=O)(C2)C1 41434,C1(NC(CC(CN(C)C)O)=O)CN(C(=O)COCc2ccccn2)CC12CCC2 41435,CC1C(C(=O)N2CCC(C)(C)C2C(=O)Nc2cc(CO)cc(F)c2)=NOC1C 41436,C1(NC(C(C(CC)C)N(C)C(C2C3(CC3)C23CC3)=O)=O)CC12CCCCCC2 41437,CCC(CC)C(=O)NCC1(COC(=O)COc2ccccc2C(C)C)CC1 41438,c1(C(C)NC(C)C)cccc(N(C(C(=O)NCCN)=O)S(C)(=O)=O)c1 41439,Cc1cc(N)c(C(=O)NCC2(CNC(c3cnc(N(C)C)o3)=O)CC2)cc1C 41440,C(=O)(CC(CCCC(C)C)NC(C1CCOC(C)(c2ccccc2)C1)=O)OCC 41441,CC1(NC(=O)CCCNC(C2(C(F)(F)F)CC2)=O)CCCOC1 41442,N1(C(C=CC)=O)CCC(NC(c2cccn(C)c2=O)=O)C(c2ccccc2)CC1 41443,c1(CCC)nc(C)c(C(=O)NCC2CC(NC(C3CCOC3(C)C)=O)C2)o1 41444,CCCCC(C)C(=O)N1CCC(C2CCCN2C(c2ccc(Cl)nc2C)=O)C1 41445,N1(CC)CCN(C(C23CC(CO)(CN2C(=O)CCc2nc(O)n[nH]2)C3)=O)C(C)C1 41446,N1(C(C2CCC(COC)C2)=O)CC(C)(C)OCC1CNC(=O)CS(C)(=O)=O 41447,C1(CC(=O)OC)CN(C(=O)NC2COCCN2CC(F)F)C2(CCC2)CO1 41448,N1(C(CCC(C)C)=O)CCC2COC(CNC(=O)C(c3ccc(Cl)cc3)=O)C2C1 41449,N1(C(C(c2cccnc2)C)=O)CCCC1c1cncn1C 41450,N1(C(C2CC(OC)C2)=O)CCC2(CC1)CC2CNC(c1cccc(F)c1O)=O 41451,N1(C(c2nc(NC)nc(O)c2)=O)CCOC2CN(C(C3CC=CCN3C)=O)CC12 41452,c1(CC)ccc(C(=O)N(C2CCN(C(=O)C#CC3CC3)CC23CC3)C)cc1OC 41453,C(=O)(C(C)(O)Cn1ccccc1=O)NC1C(NC(c2ccc(OC)s2)=O)C1 41454,C=C(Br)CC(C)(C)C(=O)N1CC(C)(NC(=O)CCOCC(C)(C)C)C1 41455,C1(O)(CC(=O)NCc2cc(C(F)(F)F)cc(F)c2)CCN(Cc2cc[nH]n2)CC1 41456,C1(C(=O)NC(CC)(C)CN(C)C)C=CCCN1C(C1CC1OC)=O 41457,C(=O)(C(O)CCCNC(=O)Cn1[nH]cnc1=N)N(CC(N)=O)C 41458,n1(C2C(C(=O)NC3CC3)C2)cnc2c(N3CCC(S(N)(=O)=O)CC3)ncnc12 41459,Cn1cc(S(N)(=O)=O)c(C(N2CC(NC(=O)CC3COCC4(CCC4)O3)C2)=O)n1 41460,c1(C(=O)NCC2COCCN2C(=O)C(F)CC2CC2)nc[nH]c2nccc1-2 41461,C1(c2nc(-c3ccccc3Cl)no2)COCCN1C.Cc1conc1NC(=O)CSS 41462,C1(C(N2C(C(=O)O)CC(OC)C2)=O)CC2CC(=O)C1C2 41463,C1(C(=O)NCc2snnc2C2CC2)CSCCN1C(=O)CCCCC1CC1 41464,CC1CC(NC(=O)COc2ccccc2)CN1C(c1cc(F)cs1)=O 41465,c1(C(=O)NCC(CN(C(c2cnc(C)n2C)=O)C)(C)C)cnc2ccc(F)cn12 41466,c1(NC(c2c(Br)cc(C)o2)c2nnnn2C(C)C)cc(Cl)cc(Cl)c1[N+](=O)[O-] 41467,C(=O)(CCCCN1CCCC1)NCCCCN(C(CCOCC#C)=O)C(C)C 41468,CC1=CCC(C(=O)NC2CC(C)(NC(=O)CC(C)(C)O)C2)CC1 41469,c1(CN(C2(O)CCNCC2)C(=O)NCC(C)(C)[N+](=O)[O-])c(Br)cncc1Br 41470,c12ccnc(c1)C(=O)NC2.C1(CNC(C2(OC)CCOC2)=O)CCOC(C)C1 41471,C(C)(CN=c1ccnc(NCc2nnc(O)n2C)[nH]1)(C1CC1)OC 41472,Cn1c(C(N2CCC(NC(C3(C4CCCO4)CC3)=O)C2C2CC2)=O)cccc1=O 41473,C1(CNC(c2cccc(F)c2F)=O)CN(C(=O)Cn2cnnc2O)CC12CC2 41474,c1(OC)ccc(F)c(F)c1C(N1CCN(Cc2cc(C(N)=O)nn2C)CC1C)=O 41475,C(=O)(CCCCC(N)=O)NCC(C)NC(c1cnc(OCC(F)F)c(Cl)c1)=O 41476,C#CCCCCCCCC(=O)N1CCC(O)(CNC(=O)CCc2cc(C)[nH]n2)C1 41477,c1(C(=O)NCC(CO)NC(C2CC23CCC3)=O)nnc2c(F)cccc2c1O 41478,C(=O)(C(C)(O)COC)N(C)CC1N(C(CC(=O)NC)=O)CCC1 41479,CCCCC(O)CCC(=O)NCC(C)(C1CC1)NC(C1CCCCN1N=O)=O 41480,C1(C)(C(=O)NCC2C(NC(CCC(C)(C)C)=O)CCC2)CC2CCC(C1)S2(=O)=O 41481,CCCCCCCCC1C(C(N2CCC(c3cccc(C)c3)C2C)=O)CCCC1 41482,C(=O)(CC1=CCN(C)CC1)N1C(CNC(C2(C(=O)OCC)CCC2)=O)COCC1 41483,C1(C#N)(C(=O)NCc2c(C(=O)NCCSCCOC)cccn2)CCCCC1 41484,c1(NC(N2CCOC(c3cn(CC(F)(F)C(F)F)nn3)C2)=O)ncc(Br)cc1F 41485,C12(CNC(COCCOC)=O)CC(CO1)N(C(c1cnn(C)c1SC)=O)C2 41486,C1(CC(=O)NCC2OCCN(C(c3c(C)cn(C)c3)=O)C2)COCC(C)(C)O1 41487,CCCC(C)C(=O)N1CCC(C(C)(O)CNC(=O)C=C(C)c2ccco2)CC1 41488,c1(N(CCCNC(c2c(Cl)cnc(C(C)(C)OC)n2)=O)C)cc(SC)nc(C)n1 41489,C1(NC(COCC)=O)CCCN(C(=O)CC(CC#N)c2ccccc2)CC1 41490,CCC(CC(=O)NC1(CCO)CCC1)NC(=O)C(O)C1CCC1 41491,C1(COC)(CNC(C2CCCC23CC3)=O)CCN(C(c2cc(C)cc(C)n2)=O)CC1 41492,c1(OCC)cc(CNC(c2nc(C(=O)O)c(C)s2)C)ccc1S(C)(=O)=O 41493,c1(SC)ccsc1C(=O)NCCN(C(=O)C(C)SC1CCOCC1)C 41494,c1(NCCCN(C)C(c2ccc([N+](=O)[O-])o2)=O)cccc(F)c1[N+](=O)[O-] 41495,C=CC1CCCCN1C(C12CC1CN(C(=O)CC(C)(C)CC1CC1)C2)=O 41496,c1(CNC2(C(=O)NCC)CCCC2)ccc(-n2cccn2)cc1.C12(CC1)C(=O)N2 41497,c1(NC(C(N2CCC(c3cn(C)nc3)C(C)(C)C2)=O)=O)cccc2c1CC(=O)N2 41498,C12(CNC(c3cnc(Cl)s3)=O)CCCCC1N(C(=O)CC1CC(F)C1)CCC2 41499,c1(C(=O)NC2C(NC(Cc3c(C)ccs3)=O)CC2)cnn(C(C)C(C)C)c1C 41500,n1(CCC)nnnc1C(c1c[nH]nc1-c1ccncc1)NC(COC)C1CC1 41501,S(=O)(=O)(c1c(Cl)ccc(C)c1F)NCC(COCC)O 41502,CC1(F)CC2(CN(C(C3CCCCCN3C(c3cccn4cncc34)=O)=O)C2)C1 41503,C1(C(=O)NC(C)C(=O)NCCc2ccccn2)CC(=O)CCO1 41504,CCC(CC(=O)NCC(CC)(CC)NC(c1ccc(CC(N)=O)cc1)=O)C1CC1 41505,CC1CC(NC(C2(COc3cccc(C4CC4)c3)CC(F)(F)C2)=O)CCO1 41506,C#CCC(C)C(=O)NCC(C)(C)CN(C)C(c1cc(Br)n[nH]1)=O 41507,C1(CNC(CC2ON=C(C)C2)=O)CCC(NC(C2CCN(C)C2)=O)CC1 41508,CC(CCCc1cn(CC(=O)O)nn1)C(=O)NC1CCN(C2CCC2)C1 41509,c1(CN(C(=O)COC2CCN(C(=O)C=C3CCN(C)C3)C2)C)cccnc1 41510,CCC(C(=O)NC1CCN(C(c2oc(C)cc2C)=O)CC1O)C(F)(F)F 41511,CC1(C)CCN(CCNC(=O)C(c2ccoc2)NC(=O)CNC=O)C1 41512,c1(CC)ccc(N)c(C(=O)NCCN(C(=O)C=Cc2cc(Br)cs2)C)c1 41513,Cc1ccc(F)c(N)c1C(=O)NCC1(F)CC(NC(=O)CN(C)C2CC2)C1 41514,N1(C(=O)Nc2c(C)nc(CC)s2)CC(CC(=O)O)C(C2CC2)C1 41515,c1(CC)nnc2c(C(N3CCC(NC(C4(O)CC4)=O)CC3C)=O)cccn12 41516,C(=O)(C(C)(C)C(C)O)NC1(CC=C)CN(C(=O)Cc2c(Cl)c(CC)nn2C)C1.CC 41517,c1(NC2CC3CN(C(CC(CCC)(C)O)=O)CC32)ncnc(N(C)C)c1[N+](=O)[O-] 41518,C1(CC)(NC(=O)CN2CCOCC2=O)CCCN(C(=O)C(CC)n2ccnc2)C1 41519,N1(C(C(c2cccc(Br)c2)(C)N)=O)Cc2ccccc2C2(CCC2)C1 41520,C(=O)(CCCCNC(N)=O)NC1(CC=CC(=O)NCC(C=C)O)CCC1 41521,c1(C(=O)NC2C3(C)CN(C(C(=O)N(C)C)=O)C2C3)cn2cccc(F)c2n1 41522,C12(CNC(C=CC=CC)=O)CCC(NC(=O)CN3CCCCCC3)(CO1)C2 41523,n1(C(C)C)cc(C(=O)NC2CC(O)CN(C(c3cn(C)[nH]c3=N)=O)C2)ccc1=O 41524,N1(C(COC2CCCC(C)C2)=O)CC2CC(C1)C2NC(c1ccnc(O)c1)=O 41525,c1(NCC)ccc(C)cc1C(=O)NCCCNC(c1cccc(C(=O)NC)c1)=O 41526,CCC(C)C(O)C(=O)NC1(C(=O)N(C(C)CC(N)=O)C)CCCCC1 41527,N1(C(C2(C)CCCO2)=O)CCCCCC(NC(=O)C(c2ccc(O)cc2)=O)C1 41528,N1(C(C(C)CBr)=O)CCC2(CCN(C(c3cc(C4CC4)nn3C)=O)C2)C1 41529,c1(CN(c2ccc(=O)oc2)OC)c(C(F)(F)F)cccc1F.O=C1CNCCO1 41530,CC12CC(NC(=O)CC3CC4CC4C3)(C1)C1(CCN(C(c3nncs3)=O)CC1)O2 41531,N1(C(CC(c2ccc(Cl)cc2)NC(C)=O)=O)CC2CCC1CO2 41532,c1(C(=O)NC2(C3N(C(C(CC)O)=O)CCC3)CC2)cc(F)c(Cl)c([N+](=O)[O-])c1 41533,c1(-c2cc(C(N(CC(C)NC(C(C)=CC)=O)CC)=O)no2)ccc(Cl)cc1 41534,CC1(CNC(C2CCOC(=O)N2)=O)CCCN(C(c2cn(CCO)nn2)=O)C1 41535,c1(CC(N2C(C(N3CCCOCC3)=O)CC(=C)C2)=O)cccc(Cl)c1F 41536,CC1(CNC(c2ncn3c2CCC3)=O)CN(C(c2cccc(Cl)c2)=O)CCO1 41537,C1CCCC(N=c2nc(N3CCC4(CCCCO4)C3)c3c([nH]2)CCC3)CO1 41538,c1(C2C(C)C2)ccc(NC2(CNC(=O)OC(C)(C)C)CCCCCC2)c(F)c1 41539,N1(C(C=C(C)c2cccs2)=O)CCCC1C1CCCN1C(=O)C1=NOCC1 41540,c1(C(C(=O)OC)N(CCOC)CCCC2CC2)csc(C)c1 41541,N1(C(C)CNC(=O)CCn2cccc2)CCN(C(=O)Cc2cnsc2)CC1 41542,C(c1ccc(C(N)=O)cc1)=CC(=O)N(CC(C)NC(C(C)OCC#C)=O)C 41543,C1(C(N(C)Cc2ccsc2)=O)CCN(C(=O)CCOC2CCC2)O1 41544,Cc1[nH]c(C)c(C(=O)NC2CC(C)(NC(c3ccn(C(C)(C)C)n3)=O)C2)c1C 41545,CN1CC(NC(c2occc2CNC(C2C3CCCC23)=O)=O)C(F)(F)C1 41546,C12(C(=O)NC3C(C)(C)C(CNC(=O)Cn4cccn4)C3)C3C4C1C1C2C3C41C#N 41547,N(C(=NCCOc1ccc(Cl)cn1)NCC1CCC(F)CC1)CCOC 41548,N1(C(C2C3CN(C(C4N(CC)CCC4)=O)C2C3)=O)CC2C(C1)C2(F)F 41549,C1(CC(=O)NC2C3C(OC)C4C(C3)C24)CN(C(=O)OC(C)(C)C)CC(C)O1 41550,c1(C(=O)NC2CCC(CCC(=O)NCCOCC=C)C2)nc(C)ccc1C 41551,C1(NC(=O)COc2cccnc2)CN(C(=O)Cc2ccc(Cl)cc2)CC1F 41552,C1(CC=C)(NC(c2cnccc2C)=O)CCN(C(C2(C)CCC2C(=O)OC)=O)C1 41553,C1(C#N)(C(=O)NC2(CCCCNC(C=Cc3n(C)cnc3)=O)CC2)CCOCC1 41554,c1(CN(C)CC2CCN(C(=O)Cc3ccco3)C2)cc(Cl)ccc1Cl 41555,c1(C(N)=O)cc(CC(=O)NCC2(O)CN(C(C3(n4nccn4)CC3)=O)C2)on1 41556,c1(C(N2CC(CC(=O)NC3CCC(CCCC)CC3)C2)=O)c(OC)cccc1C 41557,CCCC(C)CC(=O)NCC1CCCN(C(c2ccnc(Cl)c2F)=O)C1 41558,CCCC(C)CN=c1cccc(S(=O)(=O)NCCn2ccnc2C(C)C)[nH]1 41559,c1(OC)ccc(C)cc1C(=O)NCC#CCNC(c1ncccc1OC)=O 41560,C12(CNC(C3CC(=O)NC3)=O)CCN(CC1)CC2 41561,C1(C(N(CC(=O)NCCC2CC=CCC2)CC)=O)C(C(C)=O)C1(C)C 41562,c1(CC)[nH]nc(C(=O)NCCOCCNC(=O)C(O)CC2CC2)c1Cl 41563,C=CCC(C)C(=O)N1CCC(n2cc(CNC(C3CC(C(=O)OC)C3)=O)nn2)C1 41564,N1(C(C(CC)N(C)C)=O)CCC2(C=C(C(=O)N3CCCN(C)CC3)C2)C1 41565,c1(C(N2C(CNC(c3ccc(Br)nc3Br)=O)COCC2)=O)cc2cccnn2n1 41566,C(=O)(C(CC(C)C)NC1(CCF)CC1)N(CC(COC)O)C 41567,C1(C)(COC)CC(NC(=O)Cc2c[nH]nc2C)CN1C(c1cc(C)ccc1C)=O 41568,N1(C(CCC(C)OC)=O)CC2CCC1CN2C(=O)COC1CCS(=O)(=O)CC1 41569,c1(C(=O)NC2CC(F)(CNC(C3CC(C)OC3)=O)C2)ccc(-n2cncn2)c(N)c1 41570,N1(C(c2c(C)nc(CC)o2)=O)CCCC12CCN(C(C1(C(N)=O)CC1)=O)C2 41571,CN1N=C(CC(=O)N2C3CCCC2CC(NC(=O)C(O)C2CCCC2)C3)CC1=O 41572,N1(C(C2(CC)CC2(F)F)=O)CCC(CF)(NC(c2ncoc2-c2ccon2)=O)C1 41573,N1(CC)CCN(C(c2ccnc(C3CC3)c2)=O)CC1=O 41574,CCCC(C)(O)CC(=O)NC1CCCC1NC(c1cnc(C)c(N)c1)=O 41575,C(CN=C(NCCc1ccco1)N(C)CCn1ncc(O)nc1=O)c1cnc(C)s1 41576,c1(OC)c(NC(C2(NC(=O)OC(C)(C)C)CC3CCC2C3)=O)c(C)nn1C 41577,c1(NCCN(CCCC(=O)OCC=C)C)c([N+](=O)[O-])c(C)nn1CC 41578,CC1(C)CCCC(CC(N2CC(CNC(c3cncc(N)c3)=O)C2)=O)O1 41579,CC1CC(C(=O)NCCC2CCN(c3cc(C(N)=O)ncn3)CC2)CC(C)C1 41580,C(CO)(CC(C)(C)C)NC(C(CC=C)NC(c1cc(CO)on1)=O)=O 41581,CC1CN(C(c2cnn(CCF)c2)=O)CC1CNC(c1cscc1Cl)=O 41582,c1(CCN(C(C)C)CC)nc(-c2cccnc2OC)nn1CCCO 41583,Cn1c(C(=O)NC2CN(C(=O)CCC3CCCCO3)CCC2F)cc(Cl)c1Cl 41584,N1(C(CC=C)=O)CCOCC(CNC(=O)CC2CC(F)(F)C2)C1 41585,C1(NC(c2cnc(OC)nc2)=O)(CNC(=O)CN2CSCC2=O)CCCCC1C 41586,CC(C)CC(O)C(C)C(=O)NC(CC1CC1)C(N1CCCC(C=C)C1)=O 41587,C1(C(=O)NC2CC(CCNC(C3N(CC(C)C)CCC3)=O)C2)C2CCCCCC12 41588,N1(C(c2nn(C)c(Cl)c2)=O)CCC2CN(C(c3cc(Cl)sc3Cl)=O)CC12 41589,Cn1ncnc1C.c1(CC2N(NC(=O)NC(C)(C)C)CCC2)ccccc1 41590,CC#CCC(C(=O)NCC#CCCO)NC(C1CN2CCN1CC2)=O 41591,N1(C(CCCCC)=O)CC2(C1)SCCC2NC(c1ccccc1OC)=O 41592,c1(SCc2n(CC(=O)OC)ncc2)nc(N(C)C)nc(N)c1Cl 41593,c1(C(=O)NC(c2c(C(N3CC(=CC)C3)=O)con2)C)cc(CC)oc1C 41594,N1(C(CC(CC)OC)=O)CCCCC(N(C)C(c2cc(-c3ccco3)on2)=O)C1 41595,C1(O)(C(N)=O)CCCN(C(c2ccc(CNC(C3CCNC3=O)=O)cn2)=O)C1 41596,C1(NC(C=COCC)=O)CS(=O)(=O)CC1NC(c1cc(Br)sn1)=O 41597,C1(NC(CCN(C)CC)=O)CCN(C(=O)CC2CC23CC3)C1C 41598,C(CN=c1nc(C2CC2)[nH]s1)C1CCCN(C(c2cc(C(N)=O)[nH]n2)=O)C1 41599,C1(N(C(=O)COc2cn[nH]c2)C)CCCCN(C(=O)C=Cc2cccc(O)c2)C1 41600,c1(C(N(C(=O)CN2CCC(C)CC2)CC)=O)cccc(SCC)n1 41601,N1(C(c2c(C(C)=O)ccs2)=O)CCC2CN(C(C3(C)CCCS3(=O)=O)=O)CC12 41602,CCC(C)(CNC(=O)CCc1ccccc1Br)C(N)=O 41603,c1(COC)nn(C)cc1C(=O)NCC#CCNC(=O)Cc1cncc(O)c1 41604,C1(C(=O)NCC2C(CNC(=O)CCCn3cccn3)C2(F)F)CC2C=CC1O2 41605,C(=O)(C(C(F)(F)F)C(F)(F)F)NC(CNC(C(C(C(CC)C)O)C)=O)C(C)C 41606,C(=O)(CC(C)C(C)(C)CC)NCCCOCCN(C(CCC=CC)=O)C 41607,Cn1c(C(N2C3CN(C(c4ccc(Br)s4)=O)CC23)=O)cc2ccccc12 41608,Cc1ccc2oc(C(=O)NC3C4CCN(C(C5(C)CCCOCC5)=O)C34)cc2n1 41609,c1(C(c2nnnn2C)NCC2(CC(=O)OC)CCC2)cc(OC)c(F)c(F)c1 41610,c1(CC(=O)NCC(CN(C(C(C)SC)=O)C)C)cncc(C)c1 41611,c1(C(N2CC(C(C)NC(C3CCCCC3C)=O)C2)=O)cn(C)c2ccccc12 41612,C1(F)(CNC(C2N(CCC)CCC2)=O)CCN(C(c2nc(O)c(C)s2)=O)C1 41613,CC(=O)CCCC(=O)NC1C2CN(C(c3cc(C)c(C)s3)=O)CC12 41614,C(=O)(C(F)(F)CCC=C)NCCCC(C(=O)N1CCC(C#C)C1)O 41615,CC(C(=O)N(CC(C)NC(c1ccc(-n2cccc2)cc1)=O)C)C(C)(C)C 41616,Cc1cccc(C(N2CC(F)CC2C(=O)Nc2cc(Br)cnc2F)=O)c1O 41617,CC(C)(C)CC(O)C(=O)N1CCCCCC1C(N1CCCCCCCC1)=O 41618,c1(C(=O)NCC(CN(C(C(C)OC)=O)C)C)cn(-c2ccccc2Cl)nc1C 41619,CCC(CC(=O)N(CCC(C)NC(=O)COC1(C(F)(F)F)COC1)C)OC 41620,c1(CNC(C2N(C(Cc3cn(CC)nn3)=O)CCCC2)=O)n[nH]c2ccccc12 41621,C1(C)(C(=O)NC(C(=O)N(CCC(O)CO)C)CCN(C)C)CCC(=O)NC1 41622,N1(C(CCOCCOCC)=O)CC(NC(c2sccc2F)=O)C2CCCCC12 41623,C1(C(=O)NC(C)CCO)(CF)CCN(C(=O)C=CC2CCCN2C)C1 41624,C(=O)(CC(C)(F)F)N(CC(C)O)CCNC(C1C(C)C1C)=O 41625,C=CCCCC(C(=O)N1CCC(n2ccnn2)C1)NC(c1cn(C)cn1)=O 41626,N1(C(CCc2[nH]c(=N)sc2)=O)CCC2(NC(c3ncccc3Cl)=O)CCCC12 41627,c1(NC(C(CC=CC)NC(=O)Cc2ncoc2C)=O)cc(C)ccc1CO 41628,c1(CNC(C(C)NC(=O)NC)=O)cccc2c1CN(C(=O)C(C#N)C(C)(C)C)C2 41629,CCC(C)CCNC(=O)CC1(CNC(C2CC(OC)C2)=O)CC1 41630,N1(C(C(C(CC)C)O)=O)CC(NC(c2cnc(C(C)(C)C)nc2)=O)C2(COC2)C1 41631,n1(CC(=O)NC2CCCC(NC(=O)Cc3cncs3)C2)cc2ccccc2n1 41632,C(=O)(C(CC)CC(C)C)NCCCC(C)NC(c1c(CC)c(F)ccc1)=O 41633,C1(C(N(CC(CNC(CN(c2ccccc2)CC)=O)C)C)=O)CCCN(CC)C1 41634,N1(C(CC(CC)OC)=O)C2CCC1CN(C(C1CC3(CCC3)C1)=O)CC2 41635,Cc1nn(C)c(Cl)c1C(N1CCOCC(NC(=O)COC2CC(F)(F)C2)C1)=O 41636,CCC(C(=O)N1CCC(N(CCO)C(c2csc(C(C)=O)c2)=O)C1)C(C)(C)CC 41637,c1(C(=O)NC(CC)CNC(c2ncccc2Cl)=O)cc(Cl)sc1S(N)(=O)=O 41638,c1(C(=O)NC(CCN(C(C(C)NC(CC)(C)C)=O)C)C)nccc2nn[nH]c12 41639,Cc1nc(CNC(C2CCN(c3cc(-n4cncn4)ncn3)CC2)=O)sc1C 41640,CCN=C(NCC1CCCC(F)C1)NCc1ccn(-c2ccc(COC)cc2)n1 41641,CC(O)(C(=O)NCCCN(C(=O)Cc1cnc(C2CC2)[nH]1)CCO)C1CCC1 41642,C1(NC(Cc2c(OC)cccc2)=O)CCSC12CN(C(C1CCCOC1)=O)C2 41643,c1(C(=O)NCC(C)N(C(=O)CO)C)cc[nH]c1C1CCCC1 41644,CCCCC(CNC(C(CCC(=O)O)OC)c1nnnn1C(C)(C)CC)CCC 41645,CC(C)CC(CNC(C1COC(=O)O1)=O)NC(=O)CSc1ccccc1 41646,C12(CCNC(c3c(OC)nsc3)=O)CCC1CN(C(C1CC(O)CN1C)=O)C2 41647,C1(NC(C2CC3(CC(OC)C3)C2)=O)CCN(C(=O)C(O)C2CC2)CC1(C)C 41648,N1(C(COCCCC#C)=O)CCCC(O)(CNC(c2c(Cl)csc2Cl)=O)C1 41649,Cc1c[nH]cc(C(=O)NC2CC(CNC(c3cnns3)=O)C2(C)C)c1=O 41650,c1(NC2C(C)CN(C(=O)CC3(O)CCOC3)CC2)ncc2c(n1)COC2 41651,C(=O)(C(C)(C)C(N)=O)NCC(C)(C)NC(=O)C(C(C)(C)C)N1C(=O)CCC1=O 41652,N1(C(C=C(CC)CC)=O)CCC(O)(CN(C(=O)Cc2cnn(C)c2)C)C1 41653,O=C1CC(C(=O)NCC23CC2CN(Cc2cnn(C4CC4)c2)C3)NC(=O)N1 41654,c1(C(=O)NC2CC2CNC(C2COCC3(CCC3)O2)=O)cc2cc(F)ccc2s1 41655,CC1(C(=O)NCCC2CCCC2)CCCN1C(c1ccsc1Br)=O 41656,CC1CCCC=C1C(=O)N(C(C)CNC(c1cc2ncccc2[nH]1)=O)C 41657,C(=O)(CCCC(C)(F)F)NC(C1OCCN(C(c2c(C)csc2)=O)C1)C 41658,C1(NC(C(Cn2ccnn2)NC(=O)CC2C=CCC2)=O)CC2CCCC2C1 41659,N1(C(CSCCC)=O)CCOC2CN(C(c3ccsc3-n3cnnn3)=O)CC12 41660,C1(CC(=O)NC(c2cc(C)on2)C)COCCN1C(=O)CSCC(F)F 41661,Cc1ncc2n1CC(C(=O)NCCN(C)C(C1CC3(CCCC3)CO1)=O)CC2 41662,N1(C(CCN(C)CCO)=O)CC(C)(C)CC1CNC(=O)C(C)(C)C1CCCC1 41663,N1(c2c(C)c(N3CCCC(NC(C)C)C3)ncn2)CCC2(CC1)CC(C)NC2=O 41664,N1(C(CC(=O)N(C2(CCC=C)CC2)C)=O)CC(O)(SCC#C)C1 41665,N12CCCC(C1)CNC2=O.N1(CCCc2cn(C)nn2)CCCCCC1 41666,N1(C(C(CC)N(C)C)=O)C2CCC1CN(C(=O)C(C)Oc1ccccn1)C2 41667,CC(C)CCC(C)NC(C1(CC2CC2)CCCN1C(=O)CCC(=O)N(C)C)=O 41668,C1(CNC(c2ccc(OC(CC)C)cc2)=O)CN(C(=O)C2=CCSC2)CCC1C 41669,C1(CNC(C(C=C)O)=O)CCN(C(C2(C3CCCCO3)CC2)=O)C12CC2 41670,C(=O)(C(C)(CC(C)C)NC(=O)Cc1cc(C(F)(F)F)c(O)nn1)OC 41671,N1(CC(C)O)CCC(C2CCCN(C(c3cnc(C4CC4)o3)=O)C2)C1 41672,c1(CCCC(=O)NCC2COCCN2C(=O)CCCCC2CC2)ccc(F)cc1 41673,c1(C(N2CC3C(CNC(c4cnc(CCC)s4)=O)C3C2)=O)cc2nc[nH]c2cn1 41674,C1(COC)OC(c2nc(Cc3ccoc3)no2)CC1C 41675,C1(COC)CN(C(C2COCCOC2)=O)CCN1C(C12CC(O)C1C2)=O 41676,c1(C(=O)NCC(CNC(C(CCCC)N(C)C)=O)F)oc2ccccc2c1CO 41677,c1(C(=O)NCCC(=C)CNC(=O)C(O)C(C)CC)ccc(Cl)c(OC)c1 41678,C1(C(=O)NCC2(C)CCN(C(c3c(C)c(C4CC4)on3)=O)C2)CCCCNC1=O 41679,c1(C(=O)NC2(CNC(C(CC)CC3CCCC3)=O)CCC2)cc2cccnn2n1 41680,N1(C(C2(C=C)CC2)=O)CCN(C(c2cnc(Cc3ccc(Cl)cc3)s2)=O)CC1C 41681,N1(C(CC(C)F)=O)CC2CCOC2(CNC(c2cc(=O)cc(Cl)[nH]2)=O)C1 41682,C1(NC(=O)C2=CCSC2)CC2CN(C(=O)CCc3cscc3Br)CC2C1 41683,c1(-c2c(C(N3CCCC(C(=O)O)C3)=O)c[nH]c2)ccc(-c2ccncn2)cc1 41684,CN1CCC(F)(C(=O)NCCCCCCNC(c2cccc(O)n2)=O)CC1 41685,CCC(C)(CNC(C1(F)CCN(C(c2ccc(CO)cn2)=O)C1)=O)C(N)=O 41686,C(=O)(C(C)C(CC)CC)N1CCCC(C(C(=O)NCc2c(CC)nco2)(C)C)C1 41687,c1(C(C)(C)C(N)=O)ccc(NC(C2CC2c2cncc(Br)c2)=O)cc1 41688,C(=O)(C1=CC(O)C(O)C(O)C1)N1C(C(N2CCC(OC)C2)=O)CC1 41689,C(=O)(CC(F)(F)CS(C)(=O)=O)N1CCC(O)(C(C)NC(c2c(C)nccn2)=O)C1 41690,C1CCC(=O)N1.c12nocc1C(=O)NC2C.N1(CC)CC(C)(C)C1 41691,c1(OC)ccnc(C(C(=O)NC2CCOC2)N(C2CCCCC2C)C)c1C 41692,N1(C(C2N(CC)CCC2)=O)CCC(C(=O)NC(CC2CC2)C(=O)NC)C1(C)C 41693,c1(OC)cc(SC)ccc1C(N1CC(O)(C(C)NC(c2nccnc2C)=O)C1)=O 41694,C1(NC(C(C(CC)C)C)=O)CC2(CCC(CNC(c3ccnnc3C)=O)OC2)C1 41695,Cc1cccc(CN(C(=O)C(c2cccs2)NC(=O)C(C)n2ccnn2)C)c1 41696,c1(C(=O)NC2CC(N(C)C(C3CCC4(CCC4)C3)=O)C2)ccncc1N=[N+]=[N-] 41697,c1(CC)nc2ccc(F)cn2c1C(=O)Nc1ncn(Cc2ccccn2)n1 41698,C1([SH](c2nnnn2C)C(C(N2CC(CCC(=O)OC)C2)=O)=O)CCn2nccc2C1 41699,C1(C(=O)NC(CC2CCC2)CO)CCN1C(=O)C=C1CCC1 41700,C1(CN(C(c2nc(COCC)sc2)=O)C)CCCC(CNC(=O)C=CCO)C1 41701,C(=O)(CCCC(=O)NCC)OCCN1CCC(NC(C2C(OCC)C2)=O)C1 41702,C1(NC(C2(CC#C)CCC2)=O)CCCC(NC(c2cc(C)n(C)c2)=O)C1 41703,Cc1nc2cc(C(=O)NCCCNC(=O)C(C)c3cccs3)ccc2n1C 41704,c1(C(N(C2CCN(C(CCC(C)SC)=O)CC2)C)=O)ccc(F)c(F)c1F 41705,C1(CC)CCC(C(=O)NC23CC(C(=O)NCC(F)(F)CO)(C2)C3)CC1 41706,C1(CCNC(C(C2CCOC2)OC)=O)CN(c2nc(C(C)C)ns2)CCS1(=O)=O 41707,c1(OCC)ccc([N+](=O)[O-])c(C(=O)NCCC2(CNC(=O)C(C)=C(C)C)CC2)c1 41708,c1(C(N2CCC(N(C(CS(CCC)(=O)=O)=O)CC)C2)=O)ccc(C=NOC)cc1 41709,C1(NC(C(C(C)(C)O)NC(c2nc(C)sc2C)=O)=O)CCOC(C)(C)C1 41710,C1(C(N2CC(CNC(CC(C)F)=O)C2)=O)CC(C2CC2)=NO1 41711,C(C(=O)NC12CC(NC(c3csc(Cl)c3)=O)(C1)C2)(C(C)(C)C)NC(C)=O 41712,c1(C(=O)NCC2C(C)CCN2C(=O)C(F)=CCCF)cnn2c1OCC2 41713,CCC(CC)C(CNC(=NCCOC(C)C)NC(c1csc(C)n1)C)OC 41714,N1(C(C(CC)C)=O)CCCC(OC(C2N(C(c3ccccc3)=O)CCC2)=O)C1 41715,N1(c2n(C)c(-c3cc4ccccc4cn3)nn2)Cc2ncn(C)c(=O)c2C1 41716,C=CCCCCCC(=O)NC(C)C(CO)NC(=O)COC1CCN(C)CC1 41717,C1(C(=O)NCCC(C)N(CCC)C)COCCN(C(=O)OC(C)(C)C)C1 41718,N1(C(C=C(C)C2CC2)=O)CC2C(NC(c3ccc(-n4cnnn4)cn3)=O)C2C1 41719,CCCCCC(F)C(=O)NC1C(C(=O)NCCC(O)CCC)C1(C)C 41720,n1(CCOC)nccc1NC(C1CC1NC(=O)C(=O)NCC1CC1)=O 41721,c1(NCC)cccc(C(=O)NC2CCCCC2CNC(C2CCCCN2C)=O)c1 41722,CC1(C)Cc2occc2C(NC(=O)NC2CCN(c3ccc(Cl)c(F)c3)C2)C1 41723,c1(COC)ccc(S(N)(=O)=O)cc1.C12CN(CCC1(F)F)C(=O)C1(CC1)C(=O)N2 41724,C1(C(=O)NC(C(C(C)C)NC(CN(C2CC2)CC)=O)C)CC2(C1)CC21CCC1 41725,c1(CCC(=O)NC(C2(O)CCN(C(CCOC(C)=O)=O)C2)C)c(F)cccc1F 41726,C1(CC)CCCC(C(=O)NCCn2cc(SCCSC(C)(C)C)nn2)CC1 41727,C(CC(O)CNCC1C(c2ccccc2)C1(F)F)OC 41728,c1(N(C(CNC(CCC#CC)=O)C)C)nccc(S(C)(=O)=O)n1 41729,N1(C(CCn2c(C)cc(C)n2)=O)CC(C)(C)CC1CNC(c1cc(Cl)sc1Cl)=O 41730,N1(C(CC=C)=O)CCC(O)(CN(C)C(C2CN(C3CCOC3)C2)=O)C1 41731,c1(C(=O)NCC(C)NC(CC)=O)cc(-c2ccccc2)n[nH]1 41732,C(=O)(CS(=O)(=O)CCC(F)(F)F)N1C(C(C)NC(c2cscn2)=O)CCCC1 41733,Cc1nc(C)c(C(N2CSCC2C(=O)NC(C2CCC2)C)=O)o1 41734,C1(NC(CNC(CC)=O)=O)(CNC(c2nn[nH]c2Cl)=O)CCOCC1 41735,Cc1ncncc1C(N1CCCC(CC(=O)NCC2(CF)CCC2)C1)=O 41736,C1(NC(CONC(=O)CC2(O)CCCC2)=O)CCCN(CCF)C1 41737,C#Cc1ccc(OC)c(NCC2(C)CC2C)c1.OC 41738,C1(=O)C(CCNC(c2ccoc2)=O)OC2CC(C2)N1C.CC=CC 41739,N1(C(C2(NC(C=Cc3ccc(C)o3)=O)CC(F)C2)=O)CC(C)OC2(CCC2)C1 41740,CC(C)C(O)C(F)(F)C(=O)NCC1CC1NC(=O)CN(C1CCCCC1)C 41741,CC1(CCNC(=O)Cn2cnnn2)CCN(C(c2ncncc2F)=O)CC1 41742,CC1CC(CO)CN(C(=O)C(C)NC(c2ncccc2Cl)=O)C1 41743,C(=O)(C(C)CC(N)=O)N1CCC(N(C(CCCCC)=O)CCOC)CC1 41744,CCN=c1ccc(C(=O)NC2CCC2NC(c2cccc(F)c2F)=O)c[nH]1 41745,c1(N2CCN(C(C(=O)NC(C)CC(C)(C)O)=O)CC2)ccc2cnccc2c1 41746,CC1CN(C)CC(C(N2CCSCC2CCNC(=O)Cc2ccco2)=O)O1 41747,c12coc(c1)CNC2=O.C(=O)(C(O)CN(C)C)NCC1CN(C(=O)OC)C1 41748,Cc1nn(C)c2ccc(C(=O)NCC3CN(C(=O)Cc4ccco4)CC3O)cc12 41749,c1(C(N2CCC(C(C)NC(CCCC)=O)CC2)=O)c(C)sc(C)c1C#N 41750,c1(CNC(C(c2cccnc2)NC(CN(C)C(N)=O)=O)=O)cnn2ccccc12 41751,c1(C(N(CCCCNC(c2ccc(C(N)=O)cc2)=O)C)=O)cccc2c1NCC2 41752,N1(C(c2ccc(CCC)cc2)=O)CC(C)(C)OC2(C1)CN(C(C1(O)CCC1)=O)C2 41753,Cc1cncc(CC(=O)NC(C2CCCN2C(C2COCCO2)=O)C)c1 41754,N1(C(CC(CC)C)=O)CC2CN(C(c3cccc(C)c3Br)=O)CCC12 41755,CC(C)CC(CNC(C1Cc2nccn2C1)=O)C(=O)NCCC(C)C(F)F 41756,C(=O)(C(CNC(c1cnsc1)=O)(CC)CC)N(c1ccccc1)CC=C 41757,CCC(C)C(C)CNC(C1CC=CC(NC(c2cnncc2O)=O)C1)=O 41758,C(=O)(C#CC1CC1)NCC#CCNC(c1nc(CS(C)(=O)=O)sc1)=O 41759,C1(NC(C2CC(CC)C2)=O)CC12CC(NC(=O)CCCc1ccc(C)cc1)C2 41760,N1(C(C=C(C)C(C)C)=O)CCCC(C)C1CNC(c1cn(CC(F)(F)F)nn1)=O 41761,C1(NC(CC(=O)NC2CC2)=O)CCC2CN(C(c3ccnc4[nH]ncc34)=O)CC12 41762,C1(NC(C(COC)N(C)C)=O)CC(OC)CN(C(=O)CSC(F)(F)F)C1 41763,c1(OC)cccc2c(CC(=O)NCC(O)CCNC(=O)CO)c[nH]c12 41764,c1(CC(CC2CC2)NC(C2(C(=O)OC)CCNCC2)=O)cc(OC)cc(OC)c1 41765,C1(NC(c2c(CC)nccn2)=O)CN(C(C2C(C)C2C)=O)CC1N=[N+]=[N-] 41766,N1(C(C2(OC)CCC2)=O)CC2(CCC2NC(=O)C(C)(C)CSc2ccccc2)C1 41767,C(=O)(C(F)(F)C(F)F)N1C(CN(C(C(c2ccc(C)cc2)(F)F)=O)C)CCCC1 41768,c1(C(C(C)NC(c2cc[nH]n2)=O)NC(=O)C(N)=O)ccccc1 41769,c1(C(=O)NCCCC(C)NC(=O)C2=NNC(=O)C2)cc2cc(Cl)cnc2o1 41770,N1(C(c2c[nH]nc2F)=O)CCC2(CC1)CCN(C(C1CC13CCCC3)=O)C2 41771,C1(C(F)(F)F)(C(N2CCC(NC(C(N(C)C)C3CC3)=O)CC2)=O)CC2C=CC1C2 41772,CC1OC2(CNC(C3(N(C)C)CCOCC3)=O)CC1(C(=O)Nc1n[nH]cc1Cl)C2 41773,N1(C(COCC)=O)CC2CN(Cc3ccc(OC)c(Br)c3)CC2C1 41774,N1(C(CCC(CC)C)=O)CC(CNC(C2CC(=C3CC3)C2)=O)C2CCCCC12 41775,C1(NC(c2coc(O)n2)=O)CCC2CN(C(=O)Cn3cc(Cl)cn3)CC2C1 41776,CC1=NOC(CCNC(c2csc(C)c2)=O)C1.C12(CC(O)C1)C(=O)N2 41777,Cc1csc(C(N2CCCC2C(C)(C)NC(=O)CCn2ccnc2C)=O)c1 41778,c1(C(N2CC3CC2CS3=O)C(=O)NCCCOC)noc2c(Cl)cccc12 41779,C(CN=c1[nH]c(=NCc2cccc(Br)c2Br)[nH]c2c1COCC2)N(C)C 41780,C(=O)(C(C#N)(CC)CC)N(CCNC(C1CC(C(C)C)=NO1)=O)CC 41781,C1(OC)CC(NC(C2CC(F)(F)C2)=O)CN(C(C2CCN(C3CC3)C2=O)=O)C1 41782,CC1CCCC(C)N(C(C2CC3CCC(C2)N3C(c2ccncc2Cl)=O)=O)C1 41783,C(=O)(C#CC1CCOC1)N1CC(CNC(CCc2cc(C)cc(C)c2)=O)C1 41784,C1(CC(=O)NC(C(O)CO)C2CC2)CC(F)CN1C(=O)C=CC1CCCC1 41785,Cc1ccc2occ(C(=O)N(C)CC3(O)CN(C(C4CC4C)=O)C3)c2c1 41786,Cc1nc(C)c(C(=O)NC2CCN(C(c3cn(CC4(C)COC4)nn3)=O)C2)s1 41787,C(=O)(C(C(C)(C)C)C1CCC1)NCC(C)NC(=O)C(C)S(C)(=O)=O 41788,N1(C(C(c2cnn(C)c2)OC)=O)CCCC(O)(CCNC(=O)CC(F)(F)Cl)C1 41789,O=C(N=c1[nH]oc2cccnc12)C1CCN(Cc2cnc(Cl)c(Cl)c2)CC1O 41790,Cc1c(Cl)ccnc1C(N1CCCCC1CNC(C1(S(N)(=O)=O)CC1)=O)=O 41791,N1(C(c2cc(CCC)n[nH]2)=O)CCCC(NC(=O)Cc2ccnc(O)c2)C1 41792,C1(N(CCCCC)CCC(=O)NC)CCN(C(=O)C(F)C(C)C)CC1 41793,Cc1cccnc1C(=O)NC1CC(F)(CNC(=O)CC2(CS(C)(=O)=O)CC2)C1 41794,C1(NC(CCc2cccc(NC)c2)=O)CS(=O)(=O)C2CN(C(=O)CC3CC3)CC12 41795,c1(C(=O)NCCC(C)NC(=O)CCC2(C)CC2)cc2ncc(Br)cn2n1 41796,CCC(C)C(O)C(=O)NNC(=O)C(C)(C)CCCCNC(=O)C(CC)CC(C)C 41797,C(=O)(CCCCC(=O)c1ccccc1)NC(C1OCCN(C(C(C)OC)=O)C1)C 41798,C#CC1CCCCN1C(C1CN(C(=O)CCC(=O)NCCC)CC1CCC)=O 41799,c1(CNC2CC(C(N3CCCC(CO)C3)=O)C2)cc(Br)ccc1Cl 41800,CCCCCCCC(=O)NC(CCCOC)C(=O)NCc1cn(C(C)C)nn1 41801,CCCCC(C)CCC(=O)N1C(C(=O)NOCCOCCOC)CCC1C1CC1 41802,c1(C2C(=O)SCCC(COC)N2C(C)C(=O)OC)cnn(CCOC)c1.CC 41803,N1(C(C(CC=C)(C)C)=O)CC2CC(NC(=O)CCc3cnc(C)nc3O)CC1C2 41804,C1(CNC(N(c2ccc(F)c(Br)c2)CC)=O)CCC2(CC1)NC(=O)N(C)C2=O 41805,c1(SCC)ccc(CC(=O)NC(CCNC(c2ccsc2SC)=O)C(C)C)cc1 41806,c1(C(N2CCCC(C(CNC(CCC=C)=O)(F)F)C2)=O)ccc(F)c(C(C)C)c1 41807,C(c1ccc(Cl)s1)=CC(=O)NC(CN(C(c1c[nH]nc1OC)=O)CC)C 41808,N1(CCC(=O)NC2(CO)CCOC2)CCC(O)CC1.C(C1CCCO1)=CC=O 41809,N1(C(CC(C)C)=O)CCC(C)(NC(=O)CC2(C)CC2(F)F)CC1 41810,CC(F)(F)C(C)(C)C(=O)N1CC(C(N2CCCC(CO)C2)=O)C(C2CC2)C1 41811,c1(SC)ccc(C(=O)NC2CC(CCNC(C3CC(C)(C)C3)=O)C2)cc1 41812,N1(C(C(C)Cc2ccc(O)cc2)=O)CCC2(CC1)CN(C(C1(C)CCCO1)=O)C2 41813,C(=O)(C(C)C(C)C)OCCCOC(COC(CC)(C)C)=O 41814,N1(C2CCN(C(C(C)n3ccnn3)=O)CC2)CCN(S(N)(=O)=O)CC1 41815,N1(C(CC2(NC(Cn3nnc(C)n3)=O)CC2)=O)CCOC(C)C1 41816,C1(C(N2CC(N3CCCC3)C2)=O)CCCCCCN1C(C1CCCOC1)=O 41817,c1(C(=O)NCC(C)(C2CC2)NC(CCCCOC)=O)ncnc(O)c1Cl 41818,C#CCC(C)(C)C(=O)NC1CC1NC(=O)C(C)Oc1ccccc1C 41819,C1(NC(C(CC2CC(F)(F)C2)NC(=O)NC)=O)CCC(CSc2ccccc2)O1 41820,N1(C(CSCC=C)=O)CC(CNC(=O)COC(F)F)OC2(CCC2)C1 41821,c1(C(=O)NC(c2nc(C)[nH]n2)(C)C)nsc2cc(Br)ccc12 41822,C12(NC(=O)CSc3cn[nH]c3)CCC1CN(C(=O)CC1CCNC(=O)C1)C2 41823,Cc1cccc(C(C)C(=O)N2CC(NC(=O)C=CCN(CC(F)(F)F)C)C2)c1 41824,c1(C(N2C(CNC(CCCCOCCC=C)=O)CC2)=O)ccnc(C)c1O 41825,N1(C(C2C(OCC)C2)=O)CC2CC(NC(=O)CCCc3ncc(C)o3)C1C2 41826,c1(C(N2CCCN(CCNC(C(CC)F)=O)CC2)=O)cccc2c1CCCN2 41827,CC1CN(C(C2CNC(=O)N2)=O)CC1(C)C(=O)NC1CCNC(=O)CC1 41828,Cc1scc(C(=O)NCC(O)CNC(c2csc(CC(F)F)n2)=O)c1C 41829,C1(C(=O)NCCN(C(=O)Cc2csnc2C)CCC)CC12CCC(C)(C)CC2 41830,CC1(C(N2CC(OC3CCCN(C(=O)CC(F)F)C3)C2)=O)CCNC1=O 41831,N1(C(C(COCC)C)=O)CCC(CNC(=O)CCc2n[nH]c(=N)s2)(COC)CC1 41832,C(=O)(CCCCC(N)=O)N1C(C)(CNC(=O)COc2ccc(F)nc2)CCC1 41833,CCCC(CC(C)C)C(=O)N(C(C)CNC(=O)CSc1cc(C)ccc1C)CC 41834,N1(C(CCC(C)N(C)C)=O)CCC2(C=C(C(=O)NC(CCO)c3ccco3)C2)C1 41835,C#CC1(C(=O)NCC2(C)CCCN(C(C3(O)CCC3)=O)C2)CCOCC1 41836,N1(C(C2C=CCN(C(c3ccc(F)c(F)c3)=O)C2)=O)CC2C3CCC(C3)C12 41837,C1(CC#C)(C(=O)NCCOCCOCCNC(C2(C(F)F)CCOC2)=O)CC(O)C1 41838,N1(C(C(CC)N(C)C)=O)CC2CN(C(=O)C(C)CSC)CC2C1 41839,Cc1cc(C(N2CCCC(N(C(=O)C(=O)NC(C)C)C)CC2)=O)c(F)cc1F 41840,CCC(C)CC(=O)C(=O)NC(CC(=O)NCC1OCCC1(C)C)C(C)C 41841,N1(C(C=C(C)C(C)(C)C)=O)CCOC(C)(CNC(c2cc3sccc3s2)=O)C1 41842,C(CCCC(C)(C)C(=O)NNC(=O)C1(F)CC1)NC(C(CC)CC)=O 41843,Cc1cnnc(O)c1C(=O)NCc1nc(C(=O)NOCC2CCCO2)c(C)o1 41844,Nc1cc(C(=O)NC2CCCN(C(C34CCC3C4)=O)CC2)ccc1C(F)(F)F 41845,C1(NC(c2c(Cl)cn(CCC)n2)=O)CCN(C(=O)CCC(F)F)CC1C 41846,c1(C(C(N2CCC(CCNC(c3c(SC)snn3)=O)C2)=O)C)ccc(O)cc1 41847,Cc1cc(NC(=O)CC2CC(NC(c3cc(O)ncc3Br)=O)C2)cc(Br)n1 41848,c1(C(C(=O)NC(CNC(c2c(CC)con2)=O)C)(C)C)ccc(F)cc1F 41849,c1(CN2CC3C(C(N4C(C)C(O)CCC4)=O)C3C2)cc(F)c(Cl)c(F)c1 41850,CC(C)CC(O)CNC(C1(C)CCCN1C(=O)C1CC1)=O 41851,C1(NC(COC2CCC(C)CC2)=O)CCCN(C(c2ccc([N+](=O)[O-])o2)=O)CC1 41852,C1(CC(=O)N(C2C(C)CC2)C)CCN(C(C2CCCCS2)=O)C1 41853,N1(C(CNC(C)=O)=O)CCC2CN(C(c3ccc(C)nn3)=O)CC2C1.C1CO1.CCO 41854,C(=O)(C(F)C(C)CNC(=O)CN1CCNC1=O)Nc1cnc(COC)nc1 41855,C12(COC)CCC(C(=O)NC3COCC3NC(c3cc[nH]c3C)=O)(CC1)CO2 41856,c1(C(=O)OC)c[nH]c(=NC2CN(C(=O)COC3CCCCC3)CC2C)cn1 41857,c1(CN(C2CC=CC(n3cc(C4CCC4)nn3)C2)C(CCC#C)=O)ccc(Br)cc1 41858,N1(C(CC(=O)NCC)=O)CC2CC(C(N3CCC(F)C3)=O)CC2C1 41859,N1(C(=O)NC(c2ccnc(NC3CCC3)c2)C)CCC(C2CC2)C(O)C1 41860,N1(C(C2C(C)C2C)=O)CC2CCCC(NC(c3ccc(C4CC4)c(Cl)c3)=O)C2C1 41861,CC(C)C#CC(=O)NC(C)(CO)C(=O)N1CC(CO)C1(C)C 41862,C1(C(=O)NC2CC(CC(=O)NC3CC(C(C)O)C3)C2)CCCC12CCC2 41863,C1(C(=O)NC2CN(C(C)=O)C2)CCC2(CC2)N1C(C1(c2ccccc2F)CC1)=O 41864,N1(C(CC2(C=C)CCCCC2)=O)CCCC2(C1)CN(C(=O)Cc1ccn(C)n1)C2 41865,C1(C)(C(=O)NCCCN(C(=O)C(C)(C)C2(C)CC2(F)F)CC)CCCCO1 41866,N1(C(c2c(C)sc(C(F)(F)F)n2)=O)CCCN(C(=O)CC2CCC2)C(C)C1 41867,C1(C(=O)NC(C(=O)OC(C)C)C)CC(C)CCN1C(C1CC2(CCC2O)C1)=O 41868,N1(C(c2cn(C)nn2)=O)CC2C(NC(=O)CNC(=O)Cc3ccccc3)C2C1 41869,c1(C(N2CC(OC)(CNC(=O)COc3ccsn3)C2)=O)cc2scnc2[nH]1 41870,C(=O)(C1CCc2cccnc21)NC1(C)CC(c2nn[nH]n2)C1 41871,CC(C)CC(F)C(=O)NC1COCC1CNC(c1coc(C(C)(C)C)n1)=O 41872,N1(C(CC=CC)=O)CC(NC(=O)C(CC)Oc2ccccc2CC)CC2(CC2)C1 41873,CC(C)CCCC(=O)N1CCN(C(=O)C(CO)N(C)C)CC1CCO 41874,C1(CNC(C(C)(C)OCC)=O)CC(C)N(C(c2cccc(-n3cccc3)n2)=O)C1 41875,c1(OCC)ccc(OCCC2CCCN2C)c2ccccc12.C1C(=O)N1 41876,N1(C(C2N(C(C)C)CCCC2)=O)CC2(CCN(C(=O)CC3(CO)CCC3)CC2)C1 41877,C1(C(=O)NCC(Cc2ccccc2)NC(c2cc[nH]n2)=O)CCC=CCC1 41878,C1(CNC(c2cc(OCC)n[nH]2)=O)CC2(CC2)CN1C(=O)CC1CC(C)C1 41879,N1(C(c2cnc(OC)s2)=O)CCC(NC(=O)CC(C)n2ccnc2)C(O)C1 41880,C(C(=O)NC(C(=O)NCC(=O)NCCO)c1ccco1)(C(C)C)OC 41881,c1(C(=O)NC2CCN(C(=O)C=C3CCC3)C2)ccc2cnnc(O)c2c1 41882,c1(C(=O)NCC2N(C(C(C(C)(C)O)F)=O)CC2)cc2c(O)cccc2[nH]1 41883,C#CC(C)(C)C(=O)N1CC(=O)CC1C(N1CCC(CC)C1)=O 41884,c1(C(=O)NC2CC(C)(NC(CC(C)(C)OC)=O)C2)ccc(S(=O)(=O)N(C)C)o1 41885,n1(CC=C)cc(C(=O)N(C2CCCC2)CCNC(=O)CSCCC(F)(F)F)nn1 41886,c1(Nc2ccc(OC)cc2)cn2c(n1)CN(C(=O)CCCNS(C)(=O)=O)CC2 41887,c1(CC(C(=O)NCC2CN(C(CCC=CC)=O)C2)O)cccc(C(F)(F)F)c1 41888,C1(NC(C=COCC)=O)CCC2CCN(C(=O)CC(C)C3CC3)C1C2 41889,N1(C(c2cnc(C)s2)=O)CC(NC(C2(C)COC2)=O)CC(O)C1 41890,c1(C(=O)NCC(CCCC)NC(=O)C(F)C(C)C)coc2ccccc12 41891,N1(C(C2CCCC(C)C2)=O)CC2(NC(=O)Cc3nc([N+](=O)[O-])n[nH]3)CCC1CC2 41892,C12(C(=O)NC3CCC(NC(c4cc(C)no4)=O)CC3)CC(C)(C1)OC2(C)C 41893,c1(OC)ccc(OCCC(=O)N2CC(C(C)NC(=O)CC=CC(C)(C)C)C2)cc1 41894,N1(C(C(CC2CC2)OC)=O)CCC(NC(c2cc(N)c(C(=O)OC)s2)=O)CC1 41895,c1(C(N2CC(F)CC(NC(=O)CC3CC=CC3)C2)=O)cc2cc(Cl)ccc2o1 41896,C1(=O)C(CC(C)C)N1.c1(CC(=O)N(CCNC(=O)NCC)C)sc(O)nc1O 41897,N1(C(c2cc(C)nc(C)c2)=O)CCOC2(C1)CN(C(=O)C(C)OC1CCOC1)C2 41898,N1(C(CC(CCC)C)=O)CCC2(C1)CN(C(=O)COC1(C)CCC1)C2 41899,C1(C(N(CC(C(C)C)C)C)=O)C(C)OCCN1C(c1c[nH]c(=O)cn1)=O 41900,C1(NC(C2C(C)CCO2)=O)(CNC(=O)CN(C2CCCCC2)C)CCCCC1 41901,c1(CC)nccnc1C(N1CCN(C(C)CNC(=O)C(O)CC2CC2)CC1)=O 41902,C1(CC)CN(C(C2(C(C)(F)F)CCOCC2)=O)CCC1NC(c1ns[nH]c1=O)=O 41903,c1(C(N(C)CCN(C)C(C2CC2Cc2ccccc2)=O)=O)cccc2nc[nH]c12 41904,C(=O)(CC(C)CC(=O)N1CCCN(C(c2ncc(Cl)cc2F)=O)CC1C)OC 41905,c1(CC(=O)NCC2CCCC2NC(=O)CNC(c2cccs2)=O)cncc(F)c1 41906,c1(OC)c(C(=O)NC2CCC2NC(c2cc(Cl)cnn2)=O)cc(Cl)cc1Cl 41907,N1(C(C2CC(NC(c3c(CC)ncs3)=O)C(O)C2)=O)CCS(=O)C(C)C1 41908,C12CC(F)CN(C1)C(=O)c1ccc(Cl)cc1OC2=O.c1(CON)cnco1 41909,C1(NC(CCC(C)(C)F)=O)CN(C(C2CC3CCCC(C2)C3)=O)CCC1(C)C 41910,N1(C(CC2OCCN(C(c3c(C)ccnn3)=O)C2)=O)CC(O)CC(C)(C)C1 41911,C1(NC(=O)Nc2cc(C)c(-n3cccn3)cc2)C2Cc3ccc(Br)cc3C12 41912,c1(OC)ncc(Br)cc1C(N1CCCC(CO)C1)C(=O)Nc1ccc(C)cc1OC 41913,c1(C(=O)NCC2(NC(=O)CC3CCCS3(=O)=O)CC2)coc2c1COC2 41914,N1(C(=O)C=CC2CCC2)CCC(NC(c2sccc2C2CC2)=O)C(CO)C1 41915,c1(C(=O)NC2CN(Cc3ccc(C)[nH]3)C2)ccc(Br)c2cc[nH]c12 41916,C1(CNC(c2nccc(C(=O)OC)c2)=O)CCC(C)CN1C(=O)CCCN(C)C 41917,N(C1CN(C(c2cnc(C3CCC3)s2)=O)CCc2ccccc21)C(C(C)(C)F)=O 41918,Cc1nc(=NCC2CCCCN2C(c2ccc(C3CC3)cc2)=O)[nH]cc1[N+](=O)[O-] 41919,CC(CC(=O)NCC1CC(C(=O)NC(c2nc(=O)o[nH]2)C)C1)CC(C)(C)C 41920,CCCC(CC)CCC(=O)NCc1cc(C(N2CCC2(C)COC)=O)n(C)n1 41921,N1(C(C2N(C(CC)=O)CCCC2)=O)CC(NC(=O)CC(C)(C)O)C2CCCCC12 41922,c1(C(=O)NCC2(C)CCCN(C(CCC(C)(C)F)=O)C2)ccc2nc(O)oc2c1 41923,C(C)(CNC(=O)COc1ccc(COC)cc1)(C(C)C)NC(C=C(CC)C)=O 41924,N#CC1(CNC(=O)C(C(N)=O)NC(c2cc(F)ccc2F)=O)CCCCC1 41925,CC(C)CC(C)CN=c1[nH]c(=NCc2ccsc2Cl)c2ccccc2[nH]1 41926,C(=O)(CCC(C)(C)[N+](=O)[O-])N1CCN(C)CC1CNC(c1cc(=O)cc(Cl)[nH]1)=O 41927,CC1COC(C)(C(=O)NCCc2cccnc2Br)C1 41928,N1(CC(C)(C)OC)CCN(CC(F)(F)F)C(Cc2cn(C3C=CCCC3)nn2)C1 41929,N1(C(c2c(OC)ccs2)=O)CCN(C)C(C(=O)NC2CCNC(=O)C2)C1 41930,C1(NC(C2C(C)(C)C2)=O)CCCN(C(c2cc(Cl)nnc2Cl)=O)CC1 41931,Cc1ccc2c(c1)CC(C(=O)NC(CNC(=O)CCc1cnoc1)C1CCC1)O2 41932,Cc1c(C(=O)NCC(C)(C)CNC(=O)CC(C)N(C)C)ccc(Br)c1F 41933,C1(CC(=O)N(C)C2CC2)CCCCN(C(=O)C(C)(C)C2CCCC2)C1 41934,N1(c2cccc(S(=O)(=O)N3CCC(C(C)O)C3)n2)CCCC2(CN(C)CC2)C1 41935,N1(C(C(C(C)C)N(C)C)=O)CC2(CCN(C(C3CC3(C)C)=O)CC2)C1 41936,c1(NC(C)=O)cccc(C(=O)NCc2nc(CNC(C3COC(C)C3)=O)cs2)c1 41937,C1(C(=O)NCC2C3CN(C(c4coc(Br)c4)=O)CC23)CC2CCCCC12 41938,N1(C(C(=O)NCC)=O)CCC(C2CC2)(CNC(c2cccc3nonc23)=O)C1 41939,c1(CC(=O)NCC2(NC(C(C)C)=O)CCCC2)cnc2c(=O)[nH]ccn12 41940,C(CC)(C(=O)N1CC(NC(=O)CCc2scnc2C)C1)=CC 41941,Cc1ccc(C(N2CC(C)C2C(=O)NC2CC(C)(C)C23CC3)=O)c(O)c1 41942,c1(C(=O)NCC(C)O)ccc(NC(=O)CC2CCC(N(C)C)C2)cc1 41943,c1(CN(c2cc3ccccc3[nH]2)C)ccc2nccn2c1 41944,N1(C(c2sc(C)c(Br)c2)=O)CCN(C(=O)CCc2cncnc2)C(CO)C1 41945,N1(CC)OCC(NC(=O)CC2CCN2C(c2cocc2C(N)=O)=O)C1=O 41946,N1(C(COCC(=O)NC)=O)CC(C)(C)OCC1CNC(C1CCCCCCC1)=O 41947,N1(C(C(C)CN(C)C)=O)CCN(C(C2(n3cncn3)CC2)=O)CC1CCN(C)C 41948,C1(C(=O)NCC2CC2CNC(c2coc(C)n2)=O)(OC)CCCOC1 41949,Cc1cn2c(n1)CCC(C(N1CCC(Nc3cc(C)nc(C4CC4)n3)C(C)C1)=O)C2 41950,O=C(CS(=O)(=O)CCO)NCC1CCCC1NC(=O)CC1CNC(=O)O1 41951,N1(C(C2C(NC(c3ccnc(C(C)(C)C)n3)=O)CCC2)=O)CC(F)(F)C(F)(F)C1 41952,c1(OC)ncc(C(=O)NC2CC(NC(=O)CC3CCOC(C(C)C)C3)C2)c(C)n1 41953,CC(C)CC(C)CC(=O)N(CC(N1CC(c2ccncc2)C1)=O)C(C)C 41954,N1(C(C2N(C)C(=O)CC2)=O)CC2(C1)CN(c1ccnc(C#N)n1)C2 41955,CC(C)(CC(=O)NC1CCN(C(c2cnc(S)nc2)=O)C(C2CC2)C1)CC(F)F 41956,c1(OC)cc(N2CCC3CCC(C2)N3C(C2CCCO2)=O)ccc1[N+](=O)[O-] 41957,C(=O)(C1=CCC(F)(F)CC1)NC(CNC(C(CCC)C(=O)OC)=O)C1CC1 41958,N1(C(c2cnc(C(C)(C)C)nc2)C(=O)NCCC)CCn2c(cnc2C(F)F)C1 41959,c1(OC(=O)NC2C(NC(CC)=O)C2)ncc(C)cc1C 41960,c1(CNC(C(c2ccoc2)N(C(c2nnc(C)s2)C)C)=O)ccccc1Cl 41961,C=CC(C)(CC)C(=O)NCC1(C)CCN(C(C2(Sc3ccccc3)CC2)=O)C1 41962,N1(C(C(CC)Oc2ccccc2)=O)CCC(NC(=O)C(C)(C)c2cnsc2)CC1 41963,C1(C#N)(C(N2CC(CNC(C3(C(=O)OC)CC3)=O)C2)=O)CC1C(F)(F)F 41964,C(=O)(C1=C(C)CCOC1)NC(C(=O)NCC(C)OCC#C)C1CC1 41965,c1(C(=O)NCC(C)(C)NC(=O)CCc2ccsc2)cc(F)c2ccccc2c1 41966,CC1(C)CC(N=c2cc(C(F)(F)F)nc(Cl)[nH]2)CN(C(=O)CCC2CC2(F)F)C1 41967,c1(N2CCC(CNC(C3C(CC)OCC3)=O)C2)nc(Cl)c(C#N)s1 41968,N1(C(COC(c2nccn2C)C)=O)CCC(C(C)NC(c2ccns2)=O)CC1 41969,C1(CNC(C2CCN(CCC)C2)=O)CC2CCC1N2C(=O)CCCCOC 41970,c1(C2(c3nc(C4CN(C(c5ccccc5)=O)C4)on3)CC2)ccc(Cl)cc1 41971,CC(C)(CCCNC(=O)C#CC1CCCC1)C(=O)NC1CC(=O)N(C2CC2)C1 41972,c1(C(=O)NC2C(C)(CNC(CCC)=O)CCC2)cc(C#N)[nH]c1C 41973,c1(N2CCCC(C3CC(=O)NN3)C2)nc2c(c(=NCc3ccc(Br)cc3)[nH]1)COC2 41974,C1(O)(C(c2ncnn2CCC)N(C(C#CCNC(C#CC)=O)=O)C)CCCOC1 41975,c1(CN(C(=O)C(=O)NCC2CC2)CCOC)c(C)nn(C)c1C 41976,N12CCCC3CN(CCC13)C2=O.CCC1C(=O)N1.c1ccccc1.C(C)(C)(C)O 41977,c1(SCC)cccc(C(N2CC(O)(C(C)NC(c3cnoc3CC)=O)C2)=O)c1 41978,c1(N2C3(CCC(CO)CC3)CCC2)ccnc2c(Br)cc(F)cc12 41979,c1(-n2c(N3CCCC4(CCC(=O)NC4)C3)nnn2)ccc(S(F)(F)(F)(F)F)cc1 41980,CC1(C)CC(NC(=O)C=Cc2ccc(F)cc2)CN(C(c2cc3ccsc3s2)=O)C1 41981,N1(C(C(c2ccccc2)=O)=O)CC2CC(NC(C3(C4CCCO4)CC3)=O)CC1C2 41982,C(=O)(C(C)(C)C(=O)N(C(C)COC)C)NC1C(CC)CCN1C(C)=O 41983,c1(C(C)C)nnnn1CC(=O)NCC1CCN1C(=O)CNC(C1(C)CC1(C)C)=O 41984,C#CCC(CC#C)C(=O)N(C1CN(C(c2ccc(S(C)(=O)=O)o2)=O)CC1(C)C)C 41985,C1(NC(c2c(F)cncc2Br)=O)CC2(C1)CN(C(=O)CC1CC1)C2 41986,n1(CC(=O)NC(C2CCCN2C(=O)CNC(=O)CC(C)(C)C)C)cccc(N)c1=O 41987,CC1(C)CN(C(C2CCCCO2)=O)C1C1CCN(C(c2ccon2)=O)CC1 41988,N1(C(C2CCCN(C(C)=O)C2)=O)C2CCC1CC(C(=O)NC1CC1C(N)=O)C2 41989,c1(OC)ncc(Cl)cc1C(N1CC(CNC(C2CCC(C)(O)CC2)=O)C(C)C1)=O 41990,O=C(O)CCCCCCCCCNC(=O)CCNCCCO 41991,c1(NC(C(c2n(CCC)ncn2)N(CCC#N)C(C)C)=O)cc(OC)ccn1 41992,CC1CN(C(c2ccnc(O)c2F)=O)CCC1N(C(=O)C=C(Cl)Cl)C 41993,c1(C(N2CC(CC=C)(NC(c3ccnnc3C)=O)C2)=O)nnc(O)cc1O 41994,c1(CC(N2CCOCC(NC(C(C(C)C)O)=O)C2)=O)ccc(C#N)cc1F 41995,c1(C(=O)NCC(C)(C2CC2)NC(c2cncnc2)=O)cnc2c(F)cccc2c1 41996,C1(NC(CC2(C)CCN(C(COCCCC(C)C)=O)C2)=O)CCC=CCCC1 41997,CCC(C)(CNC(=O)CCc1cccs1)NC(C1CC=CCC1)=O 41998,c1(C(=O)NC(C(=O)N(CCCC)CC)CO)cnncc1OC 41999,c1(C(N(CC(CC)NC(c2ccc(N)cc2Cl)=O)C)=O)cc(P(C)(C)=O)ccn1 42000,Nc1ccc(C(=O)NC2(C3CN(C(C4CCN4S(C)(=O)=O)=O)C3)CC2)cc1F 42001,Cc1n[nH]cc1CC(=O)NC1CC(C)(NC(=O)C(C)OCCC(C)C)C1 42002,CC(C)(CN=c1nc(N2CCC(C(N)=O)C2)c2sccc2[nH]1)C(F)(F)F 42003,C1(C(=O)NC2(C3CN(C(C4C(CC(C)(C)C)C4)=O)C3)CC2)CS(=O)(=O)CC12CC2 42004,C1(OC)CCn2cc(C(=O)NC3CCCC(CNC(c4cscn4)=O)C3)nc2C1 42005,C1(NC(=O)CN(C)CCO)CCOCC1C.C12(C(F)(F)F)CC(C1)C(=O)NCC2.CO 42006,C(=O)(CC(C(=O)O)C1CCCC1)NCCCCc1ccc(OC)cc1 42007,CCCS(=O)(=O)CC(=O)NCC1CN(C(c2sc(C)c(C)c2C)=O)CC1O 42008,Cc1cccc(C)c1C(=O)NCC(=O)NCC1COCCN1C(=O)CSC1CC1 42009,C1(CNC(=O)CC2CC23CC3)CN(C(=O)Cc2ccc(O)c(Cl)c2)CCCO1 42010,N1(C(C(C(C)C)O)=O)CC(C)OC2(CCN(C(c3ccc(F)cc3O)=O)C2)C1 42011,c1(C(=O)NC(C2(O)CCN(C(=O)C(F)(F)C(C)(C)O)C2)C)ccc2c(c1)CNC2=O 42012,c1(CC(=O)NCCN(C(c2scc(COC)c2)=O)C2CC2)cnn2ccccc12 42013,CC(C(F)F)=CC(=O)Nc1cnsc1 42014,N1(C(C2(c3ccc(C)cc3)CC2)=O)CCC(NC(=O)CCCCBr)C(F)C1 42015,c12ccc3c(c1)CCN3C2C(=O)NCCCSC.C(CS(C)(=O)=O)CC 42016,C1(NC(=O)CCCC2CC2)CCC12CN(C(=O)CSCc1ccncc1)C2 42017,C1(CC(=O)N(CC(O)CNC(c2coc(C(F)(F)F)c2)=O)C)CCCC12CC2 42018,c1(OC)nccc(C(N2CC(NC(c3cc(OC)no3)=O)C(C)C2)=O)c1Br 42019,CC1C(NC(=O)C#CC2CCCC2)C(C)CCN1C(=O)CNC(N1CCCC1)=O 42020,N1(CC(=O)NCC(c2ccccc2)NC(c2ccc(OC)s2)=O)CCC(F)CC1 42021,C1(O)(CCNC(c2cc(-c3ccoc3)on2)=O)CCN(C(C2CCOC2=O)=O)C1 42022,C1(CCNC(c2cn(CC=C)nc2)=O)CCCCN1C(C1CCCC1(C)C)=O 42023,C1(C(=O)NCC2(O)CCN(C(C3CC4(C3)CC4F)=O)C2)Cc2cncn2C(=O)N1 42024,C(=O)(C#CC1(CC)COC1)NC(CC=C)C(=O)NCC(C)(C)n1cccn1 42025,C(=O)(C(CCC)NC(C)=O)NCC1(C(=O)NC(CC#C)CC)CC=CC1 42026,C1(NC(CCOC)=O)CCN(C(c2cnc(S)n2C)=O)CCC1(F)F 42027,c1(C(=O)NC(CC)CNC(=O)C=Cc2ncc[nH]2)cnc(O)n1CC 42028,C1(C)(C(=O)OCC(N2CCN(c3c(C)cccc3C)CC2)=O)CC(C(C)C)=NO1 42029,CC1(C)CCC=C(C(=O)N2CCOC(CCCNC(=O)C=CC=C(Cl)Cl)C2)C1 42030,N1(C(c2ccc(NC(C)=O)s2)=O)CCC(CNC(=O)CCN2CCC2)CC1 42031,C1(C(N(C)CC2CCN(C(=O)CC#N)C2)=O)C2CCC1(c1cncs1)C2 42032,C1(C(N(C(C(CC)C)C)C2CC2)=O)CCCC(NC(=O)C(C)=C(C)C)C1 42033,CCC(CC(=O)NCCc1cnc(C)cn1)N(C(=O)CCCCSC)C 42034,C(C)(C(C)(C)O)NC(CN(C(=O)C(C)(C)O)CCOC)=O 42035,c1(C2(C(N3CCCN(C4CCOCC4)CC3)=O)CC2)ccc(F)c(OC(F)F)c1 42036,C1(F)(CNC(c2nc(OCC)sn2)=O)CCCN(C(=O)C(C)=CC2CC2)C1 42037,c1(C(=O)NCC2(OC)CN(C(c3cc(C#N)c[nH]3)=O)C2)ccc2ccccc2n1 42038,C12(C(N(CC(C)(C)C)CCO)=O)CC(NC(=O)OC(C)(C)C)(C1)C2 42039,C1(CC(=O)NC2CCC(CCNC(c3nc(C)n(C)n3)=O)C2)(OC)CCCCC1 42040,c1(CCC(=O)NC(C)CCN(C(=O)COC2CCOCC2)C)cncc(O)c1 42041,N1(C(C=CCOC)=O)CC(NC(=O)COc2cc(C)on2)CC(C)C1 42042,c1(C(=O)NCC(C)C#N)c(CNC(=O)C(C)(C)c2cncs2)cnn1C 42043,C12(CNC(C(C)OCCC(C)C)=O)CC(CN1C(=O)C=Cc1cnccn1)C2 42044,CC1(C)CCC(CC(N2CC(CNC(C3COCCN3C)=O)C(O)C2)=O)C1 42045,C1(CNC(C=C(C)C(C)C)=O)C(C)CCCN1C(c1cccnc1)=O 42046,C=C(C)C1OCCC1C(N1CC(OCC(=O)NC2(C)CC(C)C2)C1)=O 42047,N1(C(CC2C(CC)C2)=O)CCC(CNC(c2c[nH]cc2CC)=O)C1 42048,C1(F)(C(N(C2CCN(C(c3cnc(C(N)=O)s3)=O)CC2)CCC)=O)CCOCC1 42049,C1(CC=C)(C(=O)NC2(c3ncco3)CC2)CCN(C(=O)CCn2cnnn2)C1 42050,c1(CNC(CC2C(CNC(CCC3CC(OC(C)=O)C3)=O)C2)=O)nn(C)cc1C#C 42051,C(c1ccc(F)c(F)c1)=CC(=O)NC(C1CCCCN1C(=O)C1=CCCSC1)C 42052,Cn1ncc(C(=O)NC2CCC2CNC(C2CC3C=CC2C3)=O)c1Br 42053,C1(C(=O)NCc2scc(C)c2)C=CCCN1C(C1CCSC1)=O 42054,c1(CNC(c2c(C(C)NC(C(CSC)OC)=O)noc2)=O)ccnc(F)c1F 42055,c1(CC)c(C(=O)NC2CCCCC2CNC(C2(C)CC2)=O)ccn1C 42056,N1(C(C(C2CCCCC2)OC)=O)CCC(C)(NC(=O)C(N2CCN(C)CC2)C)C1 42057,Cc1c(F)cc(CN2CCCC(CNC(c3cnn4ccccc34)=O)C2)cc1Br 42058,c1(C(=O)NCC(CNC(C2(C#N)CC2)=O)O)nn2c(c1Br)OCCC2 42059,CCC(C)(C(=O)Nc1cccc(C(N2C(CO)CC2CO)=O)c1)OC 42060,C1(CCC2N(C(CC3(C)CC3)=O)CCC2)CCCCN1C(=O)C=CC=C(Cl)Cl 42061,C(=O)(C(C)(C)CF)NC(CCN(C(CC1C(OC)CC1)=O)C)(C)C 42062,Cn1ncnc1C(c1nnnn1C)NCC1(C2CC2)CCCO1 42063,C(=O)(CC(C)C(F)(F)F)N1C2C(NC(CN(C3CC3)CC)=O)C(CC2)C1 42064,Cc1ccoc1C(=O)N(CC(=O)NC1CCC(CO)C1)CC(C)C 42065,c1(CC(=O)NCC(CC=C)NC(=O)CCCSC(C)(C)C)cnn(C)c1C 42066,CC1(C)CN(C(=O)C(=O)NCCCSC2CCCC2)CCS1(=O)=O 42067,c1(OC)ccc2cc(-c3cc(CC(=O)N(C(C)C(N)=O)C)ccc3F)ccc2n1 42068,CC(C)C(C(C)NC(=O)C=CCF)NC(c1cc(C2(C)CC2)on1)=O 42069,C1(C(=O)NC(COCCCNC(Cc2ncc(C)[nH]2)=O)(C)C)CC2CCC1C2 42070,O=C1CC(C(=O)NCC2(C3CC3)CCCO2)N(C(C2CCCCC2)=O)C1 42071,c12ccc(cc1)s2.C(=O)(C(F)(F)C1CC1)NCCN(C(c1sncc1C)=O)CC 42072,C1(NC(C2CC(OCC)C2)=O)CC(NC(=O)C(c2ncccc2F)(F)F)C(O)C1 42073,C1(NC(C2(CC)CCCC2)=O)CN(C(=O)COCc2cccnc2)C2(CCC2)C1 42074,O=S(=O)(c1cccc(N2CCn3c(cnc3Cl)C2)n1)NCCC1CCCO1 42075,c1(CCC(=O)N(CC(C)O)CCNC(=O)CP(C)(C)=O)ccc(Cl)cc1F 42076,c1(CC(N2CC(CCNC(C(CCC)(C)C)=O)C2)=O)coc2cc(Cl)ccc12 42077,C=CC(C)CC(=O)N(C1(C(=O)NCc2ccc(Cl)cn2)CCC1)C1CC1 42078,C12(CNC(c3cccc[n+]3[O-])=O)CCCC(CN1C(C1CCCCC1)=O)C2 42079,C(C(CC(C)C)C(=O)N1CCCC(C2(C)CC2)C1)NC(COCCC)=O 42080,N1(C(CC=CC)=O)CCC2(CCCC2NC(c2ccc(CO)cn2)=O)CC1 42081,c1(C(=O)NC2(C)CCN(C(C(CCC)N(C)C)=O)C2)c[nH]c2ncccc12 42082,c1(C(=O)NC(CNC(CC(C=C)c2ccco2)=O)CC=C)cc([N+](=O)[O-])oc1C 42083,C1(CCCCCNC(C(C=C)O)=O)CCN(C(=O)C(c2c(C)n[nH]c2C)C)CC1 42084,c1(C(=O)NCCC2(O)CCN(C(CC3(OC)CCC3)=O)C2)cncc(OC)c1C 42085,C1(NC(C(CC)O)=O)CC(NC(=O)CNC(=O)CCCNC(C)=O)CC1O 42086,C1(c2n(-c3cccc(OC)c3)nnn2)(NCCC2CCCO2)CCCSCC1 42087,c1(C(=O)NCC2N(C(CN(C)CC)=O)CCCC2(C)C)ccc2c(c1)CCCC2 42088,N1(Cc2cnn(CC)n2)CCC(SC)C1C(=O)O 42089,C(=O)(C(O)CC(C)(C)C)NCC1(C(N2CCC(N3CC(O)C3)C2)=O)CC(C)(C)C1 42090,C1(CNC(C2CC3CC3C2)=O)CC2(CCOCC2)CN1C(c1coc(O)n1)=O 42091,N1(C(C(CC)OC)=O)CC(N(C)C(c2sc(C)nc2C)=O)C2(CC2)C1 42092,c1(C(=O)NCC2CN(C(c3c(OC)n[nH]c3)=O)C(C)C2)nccc2[nH]ccc12 42093,c1(CNC(C2ON=C(C)C2)=O)c(C)nn2c1CN(C(=O)C1=CCCC1)CC2 42094,Cc1ccc(Cl)c(C(N2CC(N(C(=O)Cc3cnc[nH]3)C)C(F)C2)=O)c1 42095,c1(C(=O)NCC2(C(N(C(C)(COC)C3CC3)CC)=O)CCC2)cnnn1C 42096,c1(CC)ccccc1C(=O)NC(CCF)C(=O)N(CCC1CC1)CC 42097,C1(CC(=O)NC2C(CNC(=O)CNC(=O)Cn3cncn3)C2)CN2CCN1CC2 42098,C1(C(=O)NCC#CCNC(c2ccc(NCC(N)=O)cc2)=O)CCCCC(=O)N1 42099,C(=O)(CCCCCCC(C)C)C.C(=O)(CCN(C)C(C)=O)N(CC(C)O)CC 42100,C=CC1(C(=O)NCCC(O)C(=O)Nc2cccc(CCO)c2)CCCCC1 42101,CCCCC(O)C(=O)NC1COCCN(C(C2CCCCN2C)=O)C1 42102,C1(NC(=O)CCCn2c(O)nnc2O)COCCN(C(c2ccsn2)=O)C1 42103,c1(C(N2CC(OC)(CF)C2)C(=O)NCCC2CC2)ccc2cccnc2n1 42104,N1(c2nc(N3CCC(C(OC)OC)CC3)nc(C)c2)CCC2(CCCCC2)C1 42105,Cc1ccc(C(=O)NCCCCCCNC(=O)C(C)CC2CC2)nc1C 42106,N1(C(CS(N)(=O)=O)=O)CCC2(CC2)CC1c1cn(CCCCCCCO)nn1 42107,O=C1CN(S(=O)(=O)c2ccc3nc(O)oc3c2)c2ccc(F)cc2N1 42108,c1(C(=O)NCC2N(C(C3CC(OC)C3)=O)C3CCC2C3)ccc2ncnn2c1 42109,N1(C(c2cn(CC)nc2)=O)CCC2CCCC12C(=O)NC(C)Cc1nncn1C 42110,C(=O)(C1=CCCCC1C)N1CC(C(=O)NCc2cccc(OC)c2)C(F)C1 42111,c1(C(N2C(CNC(Cc3cc(C)[nH]n3)=O)CC(F)C2)=O)c(F)c(F)cc(F)c1F 42112,C(=O)(C(C#N)(CC)CC)NCCC(C)NC(C1(CCC)CC1)=O 42113,c1(CNC(=O)CN(C2CCNC2)CCc2nn[nH]n2)ccccc1 42114,C1(NC(C(=O)NCCOc2cccc(O)c2)=O)CCC2(CC1)OCCO2 42115,c1(CC(C)C(=O)NC2CCN(C(c3ncn(C(C)C)n3)=O)CC2)ccccc1Cl 42116,CC1CCCCC1C(=O)NC(C1CN(C(C2(C)CC(F)C2)=O)C1)C 42117,Cc1nc(C(=O)NC2CCC2CNC(=O)Cc2cn(C)nn2)cc(O)n1 42118,c1(CC)ncccc1C(=O)N(C(=O)C(F)(F)F)CC1(C)CC(NC(=O)C2CC2)C1 42119,N1(C(c2ccccc2)C(=O)NCCCN)CCC(F)(F)C2(CC1)NC(=O)NC2=O 42120,c1(C(N(C2CCC(NC(=O)CCc3ccco3)C2)C)=O)ccnnc1O 42121,c1(C(=O)NCCN(C(c2n(C=C)nnc2)=O)C(C)C)cc(Cl)cc(C)c1C 42122,c1(CO)ccc2occ(-c3nc(CN4CCOCC4)nn3C3CCOC3)c2c1 42123,N1(C(c2c(C)csc2)=O)CC(NC(c2cc(C(C)(C)C)no2)=O)CCC(O)C1 42124,CC1(C(N2CCN(C3CN(C(=O)CCc4cc[nH]n4)C3)CC2)=O)CC=CCC1 42125,Cc1c(CN(c2ccn(C)n2)CCN2CCCC2)c(=O)oc2cc(N)ccc12 42126,C1(OC)CN(C(=O)CC(O)CNC(C2CC23CCCCC3)=O)CC12CC2 42127,N1(C(c2c(CC)nn[nH]2)=O)CC(CNC(=O)Cc2c[nH]nc2O)CCC1C 42128,N1(C(C2OCC(C)(C)C2)=O)CC2(CC2)CC1CNC(c1cc2n(n1)CCC2)=O 42129,C1(NC(C2(C)CCC(=O)N2)=O)CCN(C(c2cnc(C3CC3)nc2)=O)CC(O)C1 42130,c1(C(N(CCCCC)CCCC)=O)sc2ccccc2c1C 42131,CC1(C)CNc2ccc(C(=O)NC3CCCC3NC(C3CC4CCC3O4)=O)cc21 42132,C1(OC)CCCC(NCC(c2cccc(I)c2)OC)C1 42133,C1(NC(CCc2cc(C)on2)=O)CCOC(C(=O)NCc2ccc(Cl)cn2)C1 42134,CC(C)C(C(=O)NCC(C)CN(C)C(C1CN(C)C1)=O)n1ccnc1 42135,C1(OCC)CS(=O)(=O)CC1NC(Cc1ccc(Cl)nc1)C(=O)OC 42136,c1(C(=O)NC2CN(C(C3(CC#C)CCCCO3)=O)CC2F)cncc(C)c1Cl 42137,C(=O)(CC(C)(O)C(F)(F)F)NC1CCC(CNC(CCN(C)CCO)=O)C1 42138,N1(C(c2cc(C)nc(O)c2)=O)CC2CCC(C1CO)N2C(c1ccoc1C)=O 42139,C(CC)(CCC(=O)NCC1(C)CSC1)NC(CCC#C)=O 42140,C1(C(=O)NCCCCN(C(CCCCCC#C)=O)C)CCc2ccc(F)cc2O1 42141,C(N=c1ccnc(N2CCC=C(Br)C2)[nH]1)c1n(C)ccn1 42142,c1(OC)c(NC(=O)C=C2CCN(Cc3c(Cl)cc(O)cc3Cl)CC2)cccc1C#N 42143,C1(C)(C(=O)NC(C)CCCNC(c2n[nH]cc2Cl)=O)CC(C(C)(C)C)=NO1 42144,C(c1ccccc1F)=CCC(=O)N(C1CN(C(C2(CC#C)CC2)=O)CC1F)C 42145,CCC(C)(C)C(c1nnnn1Cc1cccs1)NCCCCC(=O)OC 42146,c1(C(=O)NCC(c2cc(OC)c(C)cc2)=O)cnc2onc(C(C)(C)C)c2c1 42147,c1(C(N2CC(O)(CN(C(CC=CC)=O)C)C2)=O)ccc2c(c1)CCCS2(=O)=O 42148,C1(CC)CCC(C(=O)NCCN2CCC(NC(C3(C)CCN(C)C3)=O)CC2)CC1 42149,N1(C(CCC2(C(=O)OC)CCCC2)=O)CC(C2(NC(C3(F)CCOC3)=O)CC2)C1 42150,CON1CCC(NC(=O)C(c2cn(C)nn2)NC(c2ccc(Cl)cn2)=O)CC1 42151,C1(CNC(CSC)=O)(CNC(C2CNC(=O)O2)=O)CCOCC1 42152,C1(NC(c2cc(SC)oc2C)=O)CCN(C(=O)C(C)NC(=O)C(C)(C)C)CC1F 42153,Cc1c(C(=O)NCCC2CC(NC(=O)C(C)c3cccs3)C2)cnn1CC(F)F 42154,N1(C(N2C(CCCOC)CCCC2)=O)CCCc2ccc(F)cc21 42155,C1(OC)CC(C)N1C(=O)Cc1cn(C(C)(C)C(=O)O)nn1 42156,N1(C(c2nc(CC)sc2)=O)CCC(C2CCCN(C(C3(O)CC3(C)C)=O)C2)CC1 42157,C(=O)(C(C)C(C)(C)C)NC(C)CNC(c1cn(C)nc1C(C)(F)F)=O 42158,N1(CC(=O)N(CC(C)NC(c2cc(C(N)=O)no2)=O)CC)CCCCC1=O 42159,Cc1cn2c(C(=O)NCC(C)NC(=O)COc3cccc(C)c3F)c(C)nc2s1 42160,c1(C(N2CCN(c3nc(COC)nc(Cl)c3)CC2)=O)cc2cc(C)ccc2cn1 42161,c1(NC(C(C2CN(C(=O)CCC3(C#N)CCC3)C2)OC)=O)cnc2ncnn2c1 42162,C1(C(=O)NC(C)Cc2nn[nH]n2)CC(NC(=O)CSC(F)(F)F)CCO1 42163,N1(C(C(CO)NC(=O)NC2CC3(C2)CC32CCC2)=O)CCCc2ccccc21 42164,Cc1cc(CNC(C2CC(NC(C3(N(C)C)CCC3)=O)CCO2)=O)ncn1 42165,C1(CC)(CC)CNC(=O)C1NC(c1cc(OC)c(Br)s1)=O 42166,c1(OC)ccc(C(C)NCC2CC(F)(F)C2(C)C)c(OC)c1 42167,C(c1cc(C)ccc1OC)=C(C(=O)NCC(CCOC)NC(=O)CCF)C 42168,CC(C)C(CN(C)C)C(=O)NC(C)(CNC(=O)CCC=CC(C)C)C1CC1 42169,N1(C(c2cccc(CCC)c2)=O)CCC(F)C(NC(C2CCCCC2CC)=O)C1 42170,CCCC(O)CC(=O)NC(CNC(C1CCCS1)=O)(CC)CC 42171,c1(CC)ccc(N(C)C(C2C3COCC23)=O)c(C)c1 42172,CC(C)CCCCC(=O)NC1(CNC(=O)C(C)C2CC2)CCCC1 42173,Nc1c(Cl)cc(C(=O)NCC2(F)CC(NC(C3CC3[N+](=O)[O-])=O)C2)cc1[N+](=O)[O-] 42174,N1(C(CC2(OC)CC2)=O)CCC(C(C)NC(=O)C(c2ccc(F)cc2)(C)C)CC1 42175,Cc1nc(C)c(F)c(=NCC(C(C)(C)C)NC(c2cccc3c2CNC3=O)=O)[nH]1 42176,c1(C(N(CC(C)NC(=O)Cn2cc(CN)nn2)C)=O)csc(CO)n1 42177,C1(NC(C2(COC)CCCC2)=O)CC(NC(=O)C(C)(C)Cn2cccn2)C12CCC2 42178,C1(C(C(=O)NCC)N(C2CC(C)CC(C)C2)C)OCCOC1(C)C 42179,CN1CCOC(C(N2CCOC(CNC(c3cnn(C4CC4(F)F)c3)=O)C2)=O)C1 42180,N1(C(C2C(C)(C)OCC2)=O)CC2(CNC(=O)CC3(O)CCOCC3)CC1CCO2 42181,c1(C(C(=O)NCC(O)CN(C(=O)CCOCC2CCC2)C)OC)cnn(C)c1 42182,N1(C(C2(CC)CCCO2)=O)CCC(O)(CNC(c2cc(O)n(C)n2)=O)C1 42183,C(CN=c1[nH]c(=NC(C)c2ncc[nH]2)c2sccc2[nH]1)c1c(C)nc[nH]1 42184,n1(CC)cc(Cl)c(C(=O)N(CC(C)NC(=O)CC(c2ccccc2F)C)CC)n1 42185,C1(CNC(c2c(C#C)c[nH]n2)=O)CC(NC(c2cn[nH]c2)=O)C12CCC2 42186,C(CCCCCCCO)=CC(=O)NC1C(CNC(C(COC)(C)O)=O)CC1 42187,CC1C(NC(=O)CC2CCCC2)CC2CCC1N2C(c1ccc(F)o1)=O 42188,c1(C(=O)NCC(CCC)NC(C2CCCC2F)=O)cc(C)c(C)o1 42189,c1(OC)cc(F)c(F)cc1S(=O)(=O)N1CC(C)(C)CC1C 42190,C(CC(C)C)(C(=O)NC1(CO)CN(C(c2cccc(OC(C)C)n2)=O)C1)OC 42191,N1(C(CN(C)C2CC2)=O)CCc2ccc(C(=O)NC3COC(C(F)F)C3)nc2C1 42192,c1(CNC)cccc(OC)n1.C12CCC(CC1)CC(=O)N2CCO.C1CC1.CO 42193,C1(NC(c2c(C)nsc2C)=O)CC12CCN(C(c1cnn3ccn(C)c13)=O)CC2 42194,N1(C(CC2CCCN(C(C(CC)(C)COC)=O)C2)=O)CC(C)N(C)C(C)C1 42195,C(C(C)(C(=O)N(CC(C)(C)CO)C)NC(c1cc(=N)[nH][nH]1)=O)SC 42196,C1(C(=O)NC(C)CCCO)CCCC(NC(=O)Cn2ccnc2)CC1 42197,N1(C(C(C)NC(CC)=O)=O)CC2CC(NC(c3coc(C(C)C)n3)=O)CC1C2 42198,c1(N(C)C(c2cc3c([nH]2)CNCC3)=O)cc2c(cc1Cl)NC(=O)C2 42199,N1(C(C2CC(C)(C#N)C2)=O)CC2CCCC2(CNC(c2ccsc2Cl)=O)C1 42200,CCC(O)C(F)(F)C(=O)NCCN(C(c1cccc(=O)o1)=O)C1CC1 42201,c1(NC(C(=O)NC(CC)CNC(=O)CCCn2cncn2)=O)c(C)cccc1C 42202,C1(O)(CNC(C(CC)(C)F)=O)CCCN(C(=O)CN2CCCCC2=O)CC1 42203,N1(C(C=CC2(C)CCOCC2)=O)C2CCC(C2)C1CNC(=O)Cc1nc[nH]n1 42204,C(CNC(=O)CCCC1CC1C)(CC(=O)NCc1cnn(C)c1O)OC 42205,C1(COC)(NC(C2CC(C)(C)CO2)=O)CCN(C(c2ccc(C3CC3)s2)=O)CC1 42206,CCCC(C)(C)CC(=O)N1CCC(N(C(=O)CCOCC2CCC2)C)C(C)C1 42207,CCCCC(CC)CC(=O)N(C1CC(NC(c2csnn2)=O)C1)C 42208,CC1C(C)N(C(=O)C=Cc2cocn2)CCN1C(=O)C=Cc1ccco1 42209,N1(C(c2c(CC)non2)=O)CC(NC(=O)Cc2ccc(C)cc2)C(C)C1 42210,C1(CC(=O)NC(C(C)NC(CC2C(CC)C2)=O)CO)(CC)CCCCC1 42211,Nc1ccc(C(=O)NC(CNC(=O)C(O)C2CC2)CC(F)(F)F)c(Br)c1 42212,c1(OC)ccc(Br)c(C(N2CCC(C)(CNC(=O)Cn3ncnn3)C2)=O)c1 42213,CCC(CC)C(=O)NCC(N1CCOCC1CCNC(=O)Cc1ccc(C)s1)=O 42214,C12(CNC(C=C3CCC(C)C3)=O)CC1CN(C(c1c[nH]c(C(N)=O)c1)=O)C2 42215,C12(C(N3CC(C(=O)OC)C3)=O)CC1CCN2C(c1ccc(C(C)=O)o1)=O 42216,C(c1ccc(C)cc1)=C(C(=O)N(CCn1cc(C2CC(NCC)C2)nn1)CC)C 42217,N1(C(C2C(C#C)C2)=O)CCC(NC(c2c[nH]cc(Cl)c2=O)=O)C(C)(C)C1 42218,c1(C(=O)NCC(C)N(C(c2ncn(C(C)C)c2)=O)C)ccc2c(c1)COC2(C)C 42219,CC(C)C(CCNC(C1(c2ccccc2)CC1(F)F)=O)NC(c1cncc(O)c1)=O 42220,Cc1cc(C(=O)NCC=CCNC(c2ccc(CC#N)cc2)=O)nc(O)n1.C1(C)CC1 42221,C1(c2n(CC=C)nnn2)(NCc2ncnn2C(C)C)CCCN(CC)C1 42222,c1(NC(C2CC(NC(c3cc(Br)cnc3F)=O)C2)=O)cc2ccccc2cc1O 42223,c1(CNC(C2(N(C)C)CCC2)=O)ncccc1CNC(=O)CCc1ccsc1Cl 42224,C1(NC(c2n(CC)ccc2)=O)CCCN(C(=O)CCc2n[nH]c(=N)s2)CC1 42225,CC(CC(=O)N(C1CC(NC(c2sc(Br)cc2Cl)=O)C1)C)C(F)F 42226,C1(C(C(=O)N(CC(C)NC(=O)CSC(F)F)C)OC)CCOCC1 42227,C(C(=O)C(C)=O)N(C1CCN(C(CC)=O)C1)c1cnccn1 42228,N1(C(c2c(COC)con2)=O)CCC2CN(C(C3(C(=O)OC)CC3)=O)CC2CC1 42229,C(CN=c1[nH]c(=NCC2(S(C)=O)CC2)[nH]c2c1CC(C)CC2)c1c(C)noc1C 42230,c1(C(=O)NCC2CC(NC(c3cc(COC)sc3)=O)C2)cnc(O)c(Cl)c1 42231,c1(OC)cnnc(C(=O)N(C)CCOC2(N)CC2)c1 42232,N1(C(C2(F)CCCN(C(c3c(CC)cno3)=O)C2)=O)CCN(C)CC(O)C1 42233,c1(C(C(=O)NCCC2(C)CC2)N(C2(C#C)CC2)C)cc(Br)c(Cl)cc1OC 42234,Cc1ccnc(C)c1C(=O)NC(C)CNC(C1CC1c1cnn(CCO)c1)=O 42235,c1(C(=O)NC2C=CCN(C(C(C)OCCC=C)=O)C2)nc2c(s1)COCC2 42236,c1(C(C(=O)NC(COC)C)NC(=O)OC(C)(C)C)cnc(O)nc1O.C1CC1 42237,C(=O)(NNC(=O)Cc1ccccc1)c1cn(CC2C(C)CCCC2)nn1 42238,N1(C(CCCn2cc(C(C=C)O)nn2)=O)CCCC(n2ccnn2)CC1 42239,c1(CC)cc(C(=O)NCC2CC2NC(=O)CC2CC(C)(C)CO2)ccc1F 42240,C(=O)(C(C)S(C)(=O)=O)N1C(C2CCCN(C(c3c(C)noc3C)=O)C2)CCCC1 42241,C1(C(N2CC(NC(C3C(C)(C)C3)=O)C(F)C2)=O)CC2(CCCO2)C1 42242,c1(CC(=O)NCC2=CCCN(C(C3CCN(C)CC3)=O)C2)n[nH]c2ccccc12 42243,CCS(=O)(=O)C=CC(=O)NCC1CCN(C(=O)C(C)c2cccs2)CC1C 42244,C1(NC(c2cc(CC)on2)=O)CC2(C1)CC2NC(=O)C(O)C(C)C 42245,CCC(C)C(C(=O)N(CCN1CCCC1)CC1CCCO1)NC(=O)NC 42246,Cn1cc(OCC(N2CC(C)(NC(=O)CCc3cscn3)C2)=O)cn1 42247,CS(=O)(=O)C1CN(C(=O)C(F)CC2CC2)CC1NC(c1cccc2c1CCC2)=O 42248,c1(CN(C)C)ccc(C(N2CCCC(CNC(=O)C=CBr)C2)=O)cc1 42249,c1(OC)cnc(C(N2CC3C(CNC(=O)C=Cc4ccc(Cl)s4)C3C2)=O)c(F)c1 42250,c1(NC(C2CC(=C)CN2Cc2cnc(OC)nc2)=O)cc2cn[nH]c2cc1OC 42251,c1(C(N2C(CNC(c3c(OC)ccs3)=O)CC2)=O)cc(C(F)(F)F)cc(O)c1 42252,C(C1CN(C(=O)CN2CC3CC3C2)CC1C(=O)NC1C2CCCCCC12)=CC 42253,c1(C(=O)NCC2CC(COC)CN2C(=O)Cc2cncnc2)cccn(C)c1=O 42254,CCCCCCCCCCS(=O)(=O)N1CCCC(CNCCNS(C)(=O)=O)CC1 42255,N1(C(CCC(=C)Cl)=O)CC(NC(c2n[nH]c3c2CC2CC32)=O)CC12CCCCC2 42256,C1(=CC(=O)NC2(CCCNC(C3CC3(F)Cl)=O)CC2)CCOCC1 42257,N1(C(c2cc(COC)sc2)=O)CCCC1(C)CNC(=O)C#CC1CC1 42258,C1(C2CCCCC2)(C(=O)NC(CC(C)NC(c2cc(OC)no2)=O)C)CC1 42259,N1(CC(C)(C)N(CC(C)C)C(=O)OC(C)(C)C)CCC(NC2CCCO2)CC1 42260,C1(CNC(C2CCC(NC(CC)=O)C2)=O)CCN(C(c2cncnc2C)=O)CC1 42261,c1(C(c2nnnn2CC(F)F)NCC(C)(C)SC)cnn(C)c1C 42262,C1(OCC(=O)NC(C2CCCN2C(=O)C(=Cc2c[nH]cn2)F)(C)C)CC(F)(F)C1 42263,N1(C(COC)=O)CC2CCC(C1)N(C(=O)CCCCC(=O)OC(C)(C)C)C2 42264,c1(CC(=O)NCC(CNC(=O)C(=CC2CCCC2)C)OC)ccccc1SC 42265,Cc1c(-c2cn(CCCC(=O)N(CC(N)=O)C)nn2)c(=O)oc2ccc(O)cc12 42266,C(=O)(CCCCCCN=[N+]=[N-])N1CCC(OC)(CNC(C2CCS(=O)(=O)N2)=O)C1 42267,N1(C(CS(=O)(=O)N(C)C)=O)CCC2(CCCCC2NC(c2ccoc2Cl)=O)CC1 42268,c1(CCNC(C(=O)N(C(c2c(C)cccc2)C)C)=O)ccc2c(c1)CC(C)O2 42269,c1(C(=O)NCc2cccc(NC(C3CC(=O)NCC3)=O)c2)ncnc2[nH]cnc12 42270,N(C1CCCc2ccc(Br)cc21)C(C(C)CN(C)C)=O 42271,C#CC1(NC(=O)C(O)CCNC(c2cccc(=O)o2)=O)CCOC1 42272,N1(C(C(C(CC)C)NS(=O)(=O)CC)=O)CCN(C(=O)C=CCO)CC12CCC2 42273,C1(Cc2ccc(OC)cc2)CCCN(C(C2N(S(CCOC)(=O)=O)CCC2)=O)C1 42274,C1(C)(C(=O)NCC(CN(C(=O)COC2(C)CCC2)C)(C)C)CCC(=O)NC1 42275,c1(C(N2CCCN(C(C(C(C)C)F)=O)CC2)=O)coc2cc(F)ccc12 42276,C(=O)(C1=CC2CC(C1)CC2O)N1CCC(C)(NC(c2n(C)ncc2C2CC2)=O)C1 42277,CCC(O)C(=O)N1CCC(N(C)C(c2cc(C(=O)OC)cs2)=O)C1 42278,Cc1ccc(F)cc1C(N1CC2(CNC(c3cc(Cl)c(Cl)s3)=O)CCC1C2)=O 42279,C1(NC(C2C(CNC(C(CC)(C)C)=O)CC2)=O)CCCOC12CCC2 42280,C1(CCNC(=O)OC(C)=O)CC(Cn2ccnn2)C1 42281,c1(NC(c2nnc3ccccn23)CCC)nccc(=NCCCNC(C)(C)C)[nH]1 42282,C1(C(N2CCC(N(C(CCCC)=O)CC3CCCO3)CC2)=O)CN(C)CC(C)O1 42283,CN1CC(O)CC1C(=O)NCCN(CCOCCO)C(C1C(CO)C1(F)F)=O 42284,C1(C2(O)CCN(Cc3ccccc3)CC2)(NCC2Cn3c(C)nnc3CC2)CC1 42285,C1(c2ncc(C)s2)CCCCN1CC#CC(C)(C)C 42286,C1(NC(c2c(C(C)C)c[nH]n2)=O)CN(C(=O)CCc2ccnn2C)CC2CC12 42287,c1(C(=O)NCC2CCCN(C(CC3C(C)(C)C3)=O)CC2)cc(O)cc(F)c1F 42288,N1(C(C(C)OCOC)=O)CCC(C(=O)NCCc2cnnn2C)C(C)(C)C1 42289,N1(C(c2cc(F)c(F)cc2F)C(=O)NCCC#N)CCc2cccc(Br)c2C1 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42308,CC1(C)CC(NC(=O)C(C)(F)C(C)(C)F)CCN(C(c2c(O)cccc2F)=O)C1 42309,Cc1nc(C(=O)NCC2(C)CCN(C(c3cnc(C)s3)=O)C2)c2ccnc-2[nH]1 42310,c1(N2CCN(C(=O)Nc3cccc(F)c3)C3C2C3)ncnc2sccc12 42311,C1(NC(C(CSC)OC)=O)CN(C(c2ccccc2OC(F)(F)F)=O)CCC1O 42312,C12(C(N(C)CC3N(C(C4C(CC)N(C)CC4)=O)CCCC3)=O)CCC(CC1)OC2 42313,c1(C(=O)NC2CC(CNC(C(CCC)C)=O)C2)ccc2nc(O)cn2c1 42314,c1(C(=O)NCC(C)(C(C)C)NC(C=CSC)=O)cc2c(cn1)COCC2 42315,c12cc(OC)c(c(CC3(O)CCOCC3)c1)CN1CC3CC(C1)N23.CO 42316,C1(C(=O)NCCCN(C)C(c2cn(C)nc2C(C)(F)F)=O)CCOC(=O)CC1 42317,CC(C(=O)NCC1(F)CN(C(c2ccc(SC(F)(F)F)s2)=O)C1)S(N)(=O)=O 42318,c1(C(N2CC(COC)(NC(=O)CC(C)SC)C2)=O)cccc2c1COC2 42319,N1(C(C(=O)N(C)C)=O)C2CCCC1CC(NC(C13CSCC1C3)=O)C2 42320,c1(C(N2CCC(OC3CCC3)C2)C(=O)NCCOC)nccc(Br)c1C 42321,C1(NC(CNC(C(c2ccccc2)C)=O)=O)CC(C)(C)C12CC2 42322,CCCCC(O)CC(=O)NC1CCCC(NC(=O)COc2c(F)cccc2F)C1 42323,C1(CCNC(CCC#C)=O)CC(F)(F)CN1C(=O)C=Cc1scnc1C 42324,C(CCCCCNC(c1scnc1Cl)=O)NC(C(=O)NCC)=O 42325,N1(C(C2CCC(CC)CC2)=O)CC(C)N(C(c2nnn3c2CSCC3)=O)CC1C 42326,C(=O)(C#CC1CCCCC1)NC(CC=C)CC(=O)N1CCC2C(O)CC12 42327,C1(NC(CC2(COC)CC2)=O)CCC12CN(C(=O)C=Cc1ncc(C)[nH]1)C2 42328,C1(C(=O)NCCCN(C)C(c2ncoc2Cn2cccn2)=O)(CC)CCCC1O 42329,n1(CCC)ccc(C(=O)NN(C(C)=O)CC2CCCN2C(=O)C(N)=O)n1 42330,Cc1ccc(C(=O)NC2(C(=O)NCc3cc(O)ns3)CCCC2C)c(O)n1 42331,C1(C(=O)NCC(C)C#N)CCN(C(=O)C=CC2CCCCC2)C12CC2 42332,NS(=O)(=O)C1CN(C(=O)N(C2CC2)CC2CNC(=O)O2)C2(CCC2)C1 42333,CC1(NC(=O)C(C#N)Cn2cc(CN3CCCC3)nn2)CCc2ccccc2C1 42334,C1(C)(C(=O)NC(C#C)CCC)CCN(C(C2CCC=CCC2)=O)C1 42335,c1(C(N(S(=O)(=O)CCC2CCCOC2)C)=O)cccc(C(C)(C)O)c1 42336,c1(C(=O)NC2C(NC(c3ccc(OC)c(O)c3)=O)C2)c(F)cc(Br)cc1F 42337,c1(C(=O)NC(CC2CCN(C(CC(CC)C)=O)CC2)C)ccc2cc(C)oc2c1 42338,C(CC(=O)NCCN1CCCC1=O)(C(F)(F)F)NC(C(CC)N(CC)CC)=O 42339,c1(CC)cccc(CC)c1S(=O)(=O)NC(=O)C(O)CCN(C)C 42340,C1(N(C(c2ccnn2C)C(=O)N(CC)CC)C)CCN(C(=O)C=CCOC)CC1 42341,C(=O)(CCCC(F)(F)CO)N(C)CC1(O)CN(C(C2C(C)OC(=O)N2)=O)C1 42342,CCC(CNC(=O)C(C(C)C)NC(C)=O)(CC)NC(=O)Cn1cccc1 42343,c1(SC)cc(C(=O)NC2CC23CCN(C(=O)CSC2CCCCO2)C3)ccc1F 42344,C(C1c2ccsc2CCN1C(C1CCSCC1)=O)NC(C1C(OCC)C1)=O 42345,c1(OC)ccc(CN2CCN(C(C3CC3C)=O)C(C)C2)nc1Cl 42346,c1(C(N2C(C)CC(NC(C3CC34CCC4)=O)C2)=O)cccc2cc(O)ccc12 42347,C1(CC(=O)NC2CC=C(C)CC2)N(C(c2csc(F)c2)=O)CCC1(C)C 42348,N1(C(c2c(C)n[nH]c2)=O)Cc2cccc(CNC(c3cc(F)ccc3Cl)=O)c2C1 42349,Cc1c(CN2CCC(SCCC(=O)O)C2)occc1=O 42350,C(=O)(C(c1cccs1)NC(=O)C(C)N1CC(C)C1)NCC(=O)OCC 42351,N1(C(c2sccc2Cl)C(=O)NC2(C)CC2)CCCCCC1C(C)(C)CO 42352,C1(NC(N2CCC(C)C2c2cccc(F)c2)=O)CC2(C1)CC(C)(C)C2 42353,C(C(F)(F)CCC(=O)NC(C)(C)C)n1cc(Cn2c(C)nc(C)n2)nn1 42354,c1(C(=O)NCC(C2CCC2)NC(c2c(C(C)(C)C)ncs2)=O)cc[n+]([O-])cc1 42355,N1(C(c2cnn(CC)c2Br)=O)CCC(NC(=O)Cn2ccc(C)n2)CC1C 42356,C12(C(=O)NC3(SCC)CC3)COCC1CN(C(=O)C(C1CC1)OCC)C2 42357,C(CCCCCNC(c1c[nH]nc1C(C)(F)F)=O)NC(c1cc(C)sc1)=O 42358,c1(C(=O)NCC(C2CCOC2)NC(c2ccon2)=O)snnc1-c1ccccc1 42359,C(=O)(C(C)(C)C(C)C)NC(CCOC)CNC(c1sc(COC)nc1C)=O 42360,c1(C(=O)NCC2CCN(C(CS(=O)(=O)NC)=O)C(C)C2)cnn2c(N)ccnc12 42361,C1(C(=O)OC)CC1C1CCN(C(=O)Nc2cccc(NC(C)=O)c2)C1 42362,C(=O)(C(O)CCCNC(c1cnn(C)c1N)=O)NCC1C(OC)CCC1 42363,N1(C(c2cc(C)sc2C)=O)CC(C)C(C(=O)O)C(C)C1 42364,N1(C(c2n(C)nc(C3CCC3)c2)=O)CCCC(CNC(c2c[nH]c(=N)s2)=O)CC1 42365,c1(-c2nnc(N(C(CCC)C)C)n2CC(C)C)cc(Cl)ccc1OCCOC 42366,Cc1c(C(N2CC3CC(C2)N(C(=O)C(C)C#N)C3)=O)cc(Br)cc1Cl 42367,N1(C(C(CCC#C)O)=O)CCCN(C(=O)CCCc2ccsc2)CC1CO 42368,C(=O)(C1=CC2(CCOC2)C1)N(C1CN(C(c2c(C)nc(O)cc2)=O)CC1(C)C)C 42369,C(=O)(C1=CCCOCC1)N1CCCC(CC=C)(NC(=O)Cc2cnn(C)c2C)C1 42370,c1(-c2nc(CS(CC)(=O)=O)nn2C)cc(C)cc(F)c1 42371,C=CC1(CC(=O)N(CCO)CC2CC2)CN(C(=O)C(C)(C)n2cncn2)C1 42372,C1(CC)CN(C(c2cc(Cl)cnc2C)=O)CCN1C(c1ccc(C)o1)=O 42373,Cn1nc(C2CC2)cc1C(=O)Nc1cccc(NC(c2cc(C3CC3)no2)=O)c1 42374,CC(CC1CC(N(C)C(=O)NCC2OCCC2C)C1)C(=O)OC(C)(C)C 42375,N1(C(C(N(C(=O)CCCC2CCCO2)C)C2CC2)=O)CCC12CCCC2 42376,N1(C(c2n(C)nc(C3CC3)c2)=O)CCC2(CCC2)C(NC(C2(CF)CCC2)=O)C1 42377,C1(C(=O)NCC2NCCC(C)C2)Cc2ccccc2C1C 42378,Cc1cc(C)c2cc(C(N3CC(F)CC3CN(C(=O)C(C)N(C)C)C)=O)sc2n1 42379,C=CC(C)(CCOC)C(=O)N(CCNC(=O)C(C)C1=CCCC1)CC 42380,c1(OC)cc(F)c(C(=O)NCC2CC(C)N(C(C3CC(CF)C3)=O)C2)cc1N 42381,C1(C)(C(N2CCCC(C(C)NC(=O)CN(C)C3CC3)C2)=O)CCC(C)C1(C)C 42382,c1(C(=O)NC(CCC)C(=O)NC(c2nccnc2C)C)nccc(C)c1N 42383,C1(n2cc(-c3c(C)cncc3)nn2)CC(C)CN(C(C2CCCC(C)CC2)=O)C1 42384,O=C1COc2ncc(C(=O)NCC3CN(C(C4CN(S(C)(=O)=O)C4)=O)C3)cc2N1 42385,Cc1nc(O)nc(O)c1CCC(N1CCN(c2ccc(C#N)nn2)CC(O)C1)=O 42386,c1(CC)cc(C)c(C(=O)NCC2(Cn3cc(CSC)nn3)CCC2)o1 42387,Cc1nocc1CC(=O)N(CCCNC(C1CCCN1C(=O)NC1CC1)=O)C(C)C 42388,C1(CNC(CCSCCC)=O)CC2CCC1N2C(=O)CC1CCCCC1(C)C 42389,C(=O)(C(C(C)(C)C)C1CCC1)NC1CCC(NC(c2nn(CC)nc2C)=O)CC1 42390,C1(NC(C(C)=C(C)C)=O)CCN(C(=O)CCOCC2CC2)CC12CCC2 42391,S(=O)(=O)(c1cccnc1NC1(CC)CC1)NC(C)CCCS(C)(=O)=O 42392,c1(CC)ccc(F)c(C(=O)NCC2CN(C(=O)CC3CCCC3)CCCO2)c1F 42393,C=CC1(C(=O)NCCOCC(C)(C)O)CCN(C(c2ccc(F)s2)=O)C1 42394,C(CC1=CCN(C(C23CC(C(=O)OC)(CO2)C3)=O)CC1)NC(C(C(=C)Cl)(C)C)=O 42395,C(=O)(C(C)C(C)NC(=O)C(N)CC#N)OC(C)C 42396,C1(C)(C(N(CC(CC)NC(=O)COCc2ccccc2C)CC)=O)CCC(=O)N1 42397,c1(C(N(CCN(C(c2nnn(C)n2)=O)CC)CC)=O)cc([N+](=O)[O-])n[nH]1 42398,C1(C(=O)NCC2CC(OC)CN2C(=O)COC2CCC2)C2CCC1(C)C2(C)C 42399,c1(C(N2CC(SC)C(NC(=O)C(O)Cc3cnc[nH]3)C2)=O)cc(C)cc(C)c1 42400,N1(C(CS)=O)CC2CC(NC(C3(CCCCC)CCCC3)=O)C(C2)C1 42401,N1(C(C(N2CCOC2=O)C)=O)CCOCC1CC(N1CCCC(F)C1)=O 42402,CCC(CC(=O)N1CCN(C)C(C(=O)NCC2(C)CC(C)C2)C1)C(C)(C)C 42403,c1(C(N2CCCC(Cn3cc(C(CC)(C)O)nn3)C2)=O)c(C)[nH]c2ncccc12 42404,C1(CNC(C(C=C)(F)F)=O)CC2CC1CN(C(=O)CCc1cnn(C)c1)C2 42405,CC1CN(C(c2csc(F)c2)=O)C(C)CN1C(c1ccnn1CCF)=O 42406,CCCC(CNC(=O)CCCCNC(C)=O)C(=O)NC(c1cc(C)on1)C 42407,C1(NC(C(COC)OC)=O)CC(C)CN(C(=O)CCCOc2cc(C)cc(C)c2)C1 42408,N1(CC(=O)NC(C(=O)NCCC(=O)OC)(C)C)CCC(F)CC1 42409,CCC(C)(C)CCNC(=O)CC1CCC(NC(=O)CC2(OC)CCC2)C1 42410,CN1CCCC(CNC(=O)C(Cc2cn[nH]c2)NC(=O)COc2cccnc2)C1 42411,C(=O)(CCCCCCCSC)NC1C(NC(c2cccc(CC)n2)=O)CCC1 42412,N1(C(c2c(C)cco2)=O)Cc2occ(C(=O)NCC3CC4CCC3C4)c2C1 42413,c1(CNC(c2cc(F)cc(Cl)c2)=O)nc2c(s1)CCN(C(=O)C(O)C(F)(F)F)C2 42414,N1(C(c2c(=O)ccn(C)c2)=O)CC2CCC(C1)C2CNC(c1ccn(C)c1)=O 42415,c1(NC(=O)Nc2ncn(C)n2)cc(F)ccc1C(N1CCC(CO)C1)=O 42416,N1(C(C=CCOC)=O)CC(C)(NC(=O)COCC2CCCO2)C1 42417,c1(C(=O)NC(C(C)NC(CCc2c(C)ncs2)=O)CO)ccn2ccccc12 42418,C1(C2(O)CN(C(C3(C)CC3(C)C)=O)C2)(CNC(C2CN(C)C(=O)C2)=O)CC1 42419,C#Cc1cccc(CC(=O)NC2CN(C(C3COCC3C(N)=O)=O)CC2OC)c1 42420,N1(C(c2c(C)nc(O)cc2)=O)CC2(C(=O)NC(C)C(F)F)CC1CCO2 42421,C1(C(=O)Nc2cn(CCOC)nc2)CC2CC2N1C(c1cc(O)n(CC)n1)=O 42422,N1(C(COCC)=O)CC(NC(=O)CN(CP(C)(C)=O)CC)CC1(C)COC 42423,CC#CCCC(=O)NC(c1ccccc1)CNC(c1[nH]cnc1C)=O 42424,C(=O)(C(C)C(O)CCCC)NCC1CCC(N(C(CCCCC#C)=O)C)CC1 42425,n1(C(CC)CC)nc(C)cc1C(N1CC2C(C1)N2C(=O)Cc1csc(C)n1)=O 42426,Cc1ccc(CC(=O)NCC(O)CCNC(C2(N3CCOCC3=O)CC2)=O)cc1 42427,C1(C(=O)NC(CC(=O)N(C2CCN(CC)CC2)C)(C)C)CC2(CCCO2)C1 42428,C1(C(=O)OC)C(F)(F)C12CC(C(=O)NCCNC(=O)C(C(C)(C)C)NC(C)=O)C2 42429,C1(C)(C(=O)NCc2cncc(CC)c2)CCCN(C(C2CCC=CCCC2)=O)C1 42430,c1(NC(C2N(C(c3c(CCC)nco3)=O)CCC2)=O)c(C)cc(C)cc1C 42431,C1(CN(C)C(c2cncc(I)c2)=O)CCCN(C(=O)CC(C)(C)C)C1 42432,S(=O)(=O)(c1ccc(C#N)cc1Cl)N(CC(C(=O)Nc1c(C)cc(Br)c(I)c1)C)C 42433,C(=O)(C(CC)C(C)O)NC1(CO)CC(C(=O)OC)(OC)C1 42434,c1(C(c2nnnn2CC2CC2)NC(C(=O)NC)C2(C)CC2)nn(C)c(C)c1Cl 42435,C1(C(=O)NCC2C(C)(C)COC2)CCC2(CC2)N1C(c1cc(C2CC2)no1)=O 42436,N1(C(=O)COC2CC2)CCC2(CCN(C(c3cc(Cl)c[nH]3)=O)C2)C1 42437,n1(CC)c(C(N2CC(C)C2C(=O)N(C2CN(C(C)C)C2)C)=O)cnc1O 42438,C1(C(=O)NCC2CCN2C(c2csc(Cl)n2)=O)CC1C1CCC1 42439,c1(NCc2cnc(CC)[nH]c2=N)cc(=NC2CCCN(C)C2)[nH]c(CC)n1 42440,N1(C(c2c(C)ocn2)=O)CCC(C)C(NC(c2occc2C(C)C)=O)C1 42441,n1(CC(=O)NC2C(NC(C(C)OCCOC)=O)CCC2)ncccc1=O 42442,C(=O)(C#CC1CCCO1)N1CC(CNC(CC2(C#N)CCC2)=O)C(C(F)(F)F)C1 42443,Cc1ncn(C)c(=O)c1C(=O)NCCN(C(=O)CN(C1CCC1)C)CC1CC1 42444,C(=O)(C(CC(C)(C)C)Nc1ccccn1)Nc1c(C(=O)OC)c(C)c(C)s1 42445,N1(C(C(C)C(C)(C)C)=O)CC(NC(=O)CN2CCCNC2=O)C(S(C)(=O)=O)C1 42446,Cc1nn(C)cc1OCC(=O)OC(c1cccc(C(F)(F)F)n1)C 42447,c1(C(=O)NCC2(OC)CN(C(C3C(=C)CC3)=O)C2)cc(OC)nc(Cl)c1 42448,c1(CNC(C(CNC(C2CCCN2C)=O)OC)=O)cnccc1Cl 42449,CCC(C)C(C)C(=O)NC1CCN(C(=O)C(C)(C)COC)CC1C 42450,C(=O)(C(CN(C)C)NC(C1CCCN1C1CC1)=O)N(CCNC(C)=O)C 42451,C1(C(N(CCC)CCNC(=O)CCc2cncn2C)=O)CC(C)CCO1 42452,Cc1ncccc1C=CC(=O)NC1CCC(C)N(C(c2cccc(N)n2)=O)C1 42453,CCN=C(NCc1nccn1CC(F)F)N1CCOC(C(F)(F)F)C1 42454,C1(NC(COc2cn(C)nc2)=O)CCN(C(=O)C(C)(C)C2CCC2)CC1F 42455,C(=O)(C(CCN(C)C)NC(=O)CC1OCCC1C)N(C1CC(SC)C1)C 42456,c1(-c2ccc(CC(=O)OC)c(F)c2)cccc2c(NCCC#N)cccc12 42457,N1(C(C)=O)CCC2CN(C(=O)C=Cc3ccc(OC(F)F)cc3)CC12 42458,c1(CC)nc(=N)[nH]c(=NC(C)C2CN(C(C3CC(n4ccnc4)C3)=O)CCO2)[nH]1 42459,C#CC1CCCCN1C(C1(C#C)CN(C(=O)CC23CCC(CC2)C3)C1)=O 42460,C=C(Br)CN=C(NC)NC1CC1C.c1(C2CCC2)ccco1 42461,c1(CNC(C(C)Cc2ccco2)=O)cccc(NC(C2(Cl)CCCCC2)=O)c1 42462,C1(CCN(C(CCN(C)CC)=O)C)CCCCN1C(c1csc(Cl)n1)=O 42463,c1(C(=O)NCC2(CNC(COC3(C#C)COC3)=O)CCC2)nc[nH]c2ncnc1-2 42464,CC(=O)CCCCCCC(=O)N1CCN(C(C2CC3CC3C2)=O)CCC1C 42465,CC12CSCC1CN(C(c1cnc(OCC(F)(F)F)c(Cl)c1)=O)C2 42466,N1(CC)C(=O)CCC1C(=O)N(C(C)CCNC(=O)CC1CCCCO1)C 42467,C1(CC(=O)NC)CN(C(=O)CCCN(C)C)CCN1C(c1cccc(=O)n1C)=O 42468,C1(NC(CCC=CC(C)C)=O)CC2C1CCN2C(=O)CC(C1CCC1)C1CCC1 42469,N1(C(CC(CC)(F)F)=O)CC2(CCN(C(=O)CC3OCCO3)CC2)C2COCC12 42470,C1(C)(C(N2C(C(=O)NCc3snc(CC)n3)CCC2)=O)CCC(O)CC1 42471,C1(C(N(CCCC)C2CC2)=O)CN(C(C2CC23CCCC3)=O)CC1C1CC1 42472,Cc1nsc(C)c1C(=O)NCc1cc(C(N2CCCC2CC2CCC2)=O)n[nH]1 42473,C(c1cc(F)cc(F)c1)=CC(N1CCN(C(C2CC2F)=O)C(CC2CC2)C1)=O 42474,CN1CC(CCNC(c2ccc(CNC(=O)CSC3CC3)o2)=O)CC1=O 42475,C1(C)(CC)C=C(C(=O)NC(C2(O)CCN(C(c3c[nH]nc3F)=O)CC2)C)C1 42476,c1(C(=O)NCC(C)(C2CCC2)NC(CNC(=O)OC)=O)cc2ccnn2cn1 42477,c1(OC)cc(C(C(=O)NCC(F)F)N(C)CC2CCCO2)cc(F)c1OCSC 42478,N1(C(c2c(C)nc[nH]2)=O)CCCCC1CC(C)NC(=O)CCNC(=O)OC(C)(C)C 42479,N1(C(c2n(CC)nnc2)=O)CCC2(CCC2NC(c2cccc(F)c2C)=O)CC1 42480,C1(SCC(=O)NCC2(NC(C3CC(F)C3)=O)CCCC2)CCS(=O)(=O)C1 42481,C=C=CC(C)C(=O)NCCOCCOCCNC(C1(C#N)CC(C)C1)=O 42482,N1(CC(=O)N(CC(CC)NC(=O)Cc2nccs2)CC)CCCCCC1=O 42483,c1(C2(C)CC(NC(C(c3ccccc3F)OC)=O)C2)cccc(Cl)c1 42484,c1(SC2(CNC(NC(CC)CC)=NCC3CC3)CC2)c(F)cccc1F 42485,C1(CC)CCCCC1OCC(=O)NC(C1CCN(C(=O)C(=O)NC)C1)C 42486,C12(C(=O)NCC(CC(=O)OC)O)CCCC1CCN2C(=O)C(C)C(C)(C)C 42487,c1(CC(N2C(C)C(C(=O)NCC3CN(C)C3)CC2)=O)ccc(C#N)cc1 42488,C1(C(N2CC(C(C(=O)NC3CCOCC3)OC)C2)=O)Cc2nccn2C1 42489,n1(CC(=O)Nc2c(C)cc(C(F)(F)F)cc2)nc(C(F)(F)F)c2c1CCC2 42490,c1(C(N2C3C(NC(C4C(C)(C)C4)=O)(CCC3)CC2)=O)nc(Br)c2ccccn12 42491,C1(NC(c2cccc(C#C)c2)=O)CN(C(=O)C(C)SC(F)(F)F)CC12CCC2 42492,c1(C(=O)NCCC(CNC(c2nc(OC)c(F)cn2)=O)O)c(F)cc(N)cc1F 42493,N1(C(C2(NC(C(COC)C)=O)CCC2)=O)CC(O)(C2CCC2)C1 42494,N1(C(C(C2CCCCC2)C)=O)CCC(CNC(=O)CCc2cnoc2)C1(C)C 42495,C=C1CN2C(=O)CCC2(C(=O)NCC=CCNC(C2CC(OC(F)(F)F)C2)=O)C1 42496,Cc1cccc2c(C(N3CC4CC4(NC(c4c(Cl)cnn4C)=O)C3)=O)cccc12 42497,N1(C(Cc2c(C)cnn2C)=O)CC2(CC(CC(=O)NCC(C)(O)CCO)C2)C1 42498,c1(C(NOCC(=O)NC(CC#C)C(=O)OC)=O)cc(C)ccc1F 42499,c1(C(=O)NC(C2CCCCC2)CNC(C(CC)(C)CO)=O)onc2ccccc12 42500,N1(C(CCc2nc(C)sc2)=O)CCC(C(C)(C)CNC(c2cn(C)nn2)=O)CC1 42501,C1(NC(c2ccc(OC)o2)=O)CCCC(NC(=O)CCc2cnc[nH]2)CC1 42502,CCCC(CC1CCCC1)C(=O)N1CCC(O)(CNC(c2[nH]ncc2C#N)=O)CC1 42503,CC12CCN(CC1)CC2C(N1CC(F)(CNC(=O)Cc2c(F)cncc2Cl)C1)=O 42504,C1(S(C)(=O)=O)(C(=O)NCC(CO)NC(Cc2c(C)ccc(C)c2)=O)CC(O)C1 42505,N1(CC(=O)NCCNC(=O)Nc2c(C(=O)OC)cncc2)CCCCS1(=O)=O 42506,N1(C(C=CC=CC)=O)CCC2CC12C(=O)N(CC)Cc1cnn[nH]1 42507,c1(NC(C)=O)cccc(C(N2CCC(Cc3ccc(C(C)C)cc3)CC2)=O)c1 42508,N1(C(COCCC=C)=O)CCC(C)(CCNC(c2ccc(OCCF)cc2)=O)C1 42509,C12CCCN(CC1)C2=O.c1(CN2CCC(N(CC)CC)C2)cccnc1C 42510,C(=O)(CC(C(F)F)c1ccccc1F)NCC1C(NC(C(C)(C)NS(C)(=O)=O)=O)C1 42511,c1(C2(C)CC2)nc(N2CCCC(NC(=O)Cc3ccc(O)nc3)CC2)cc(Cl)n1 42512,N1(C(C(F)=CCC)=O)CC(C)CCC1CNC(=O)COC1(C)CCC1 42513,c1(C(=O)NC(CC=C)CNC(c2c(Cl)sc(Cl)c2C)=O)cccc2nonc12 42514,c1(C(=O)NCC=CCNC(C2(OCC)CCSC2)=O)ccc(C)c2cccnc12 42515,c1(CCC(=O)NCC(CNC(C2(CCOC)CC2)=O)C)cccc(F)c1Cl 42516,c1(C(=O)NCC(C)(C)NC(C(C(=O)OCC)F)=O)ccc2c(c1)COCCN2 42517,C=CC1(C(N2CC(CCNC(C3(CCF)CC3)=O)C2)=O)CCCCC1 42518,COn1cnc(C)c1C(=O)NCCCN(C)C(c1sc(Br)cc1C)=O 42519,C1(CC(=O)N(CC(=O)NC(C)CN(C)C)C)(NC(C)=O)CC1 42520,c1(C(=O)NC(CC)(CNC(C2(CO)CC2(F)F)=O)CC)cnc2c[nH]nc2c1 42521,Cc1nc(C(C)(C)C)sc1CNCC1(CNC(=O)Cc2ccsc2)CC1.C1CC1 42522,c1(C(=O)NC(CN(C(=O)C(O)Cn2cncn2)CC)C)csc(COC)n1 42523,N1(C(c2ccc(C(=O)OC)s2)=O)C2CCC1CC(NC(C1CC13CCOC3)=O)C2 42524,C1(C(=O)NCC2CN(C(C)=O)C2)CCOC1NC(C1C=C(C)CS1)=O 42525,Cc1ncc(C(N2CCC(CCNC(=O)C(F)C(F)(F)F)CC2)=O)cc1N 42526,Cc1cc(C(=O)NC2CC(O)CN(C(=O)COc3cccnc3)C2)c(F)cc1N 42527,c1(C(=O)NC2C(CC)N(C(C3CCOCC3)=O)CCC2)cc(F)c(C)cc1N 42528,C12(CNC(C3N(CC)CCOC3)=O)CCCC1CN(C(=O)CSCC=C(C)C)C2 42529,n1(C(C)C)nc2c(c1NC(N1CCCC(C)(O)CC1)=O)CCC2 42530,C(C(=O)NCCNC(=O)C(c1ccc(F)cc1)(C)C)(C(C)C)NC(C)=O 42531,C(=O)(C(C)(C)CC(C)C)NCCCCN(CCCNC(CC(CC)C1CC1)=O)C 42532,N1(C(C=COCC)=O)CCC(CNC(=O)C(n2nccc2C)C)(OCC)CC1 42533,CC1(NC(C2CCC(P(C)(C)=O)C2)=O)CCCc2ccccc21 42534,c1(C2(OC)CCC2)ccc(C(=O)Nc2cnn(C3CCC(=O)CC3)c2)cc1 42535,Cc1cc(O)cc(=O)n1CC(=O)NCC1CC(NC(=O)CCC2CCC(=O)N2)C1 42536,C(CC(=O)NCC1CCOC1C)(CC(C)C)NC(C1C(CCC)C1)=O 42537,CCC(CC(=O)NCCCC(C)(C)NC(=O)C(CO)C(C)(C)C)C(C)(C)C 42538,C1(OC)(OC)CC(C)(CNC(c2cnn(CCN)c2)=O)C1 42539,N1(C(CN2CCN(C)CC2)=O)CCC2CN(C(=O)C(C)(C)C3CCCCC3)CC12 42540,c1(C(N2C(C)(CNC(C(C=C)(C)C)=O)CCC2)=O)cccc2oc(C)nc12 42541,Cc1ccccc1COC(C)C(=O)NC1C2CC1N(C(C1(C)CC(C)C1)=O)C2 42542,N1(C(C2(OC)CCC2)=O)CCC2C(CCN2C(c2cc(C)ncc2Cl)=O)C1 42543,Cc1cc(C(N2CC(C(=O)NCCSC(F)F)CCC2C)=O)nnc1C 42544,Cc1c(C(=O)NC2C=CC(C(N3Cc4c[nH]nc4C3)=O)C2)cccc1F 42545,c1(SC)cc(N2CCC(C)(CNC(=O)Cc3ccoc3)CC2)nc(SC)n1 42546,N1(C(C2(C)CCOCC2)=O)CCCC(NC(=O)CCC2(O)CCC2)CC1 42547,C(=O)(N=c1cc(C)n(CCC#N)[nH]1)N(CC=C)CC1CCCCO1 42548,c1(C(N2CC3C(C(=O)Nc4c(OC)ccs4)C3C2)=O)ccc2ncnn2c1 42549,CCCCC(CNC(=O)C(CC)OC1CCCC1)NC(C1CC(F)C(=O)N1)=O 42550,c1(C(=O)NCCCCCN(C(C(CSC)C)=O)C)ccn2cccc2c1 42551,N(C1CN(C(=O)Cc2ccsc2)CCc2ccccc21)C(=O)Cc1nc[nH]n1 42552,C1(NC(c2c(C)nc(CC)o2)=O)CCCC(C(N2CCSCC(C)C2)=O)CC1 42553,N1(C(CCC(=C)Cl)=O)CCC2(CC1)CC2CNC(c1cc(COC)on1)=O 42554,C1(NC(c2ccc(CO)cc2F)=O)CCN(C(=O)CSC(F)(F)F)CCC1(F)F 42555,N(C1CN(C(C2(C)CC=CC2)=O)Cc2ccccc21)C(c1cc(C)[nH]n1)=O 42556,C1(CC(N2CC(NC(c3ccncc3F)=O)(CF)C2)=O)CC2CCC1O2 42557,c1(C(=O)NC(CCN(C(C(CC)SC)=O)C)C(C)(C)C)cc(C)cc2nc[nH]c12 42558,CC1CN(C(C2CCCOC2)=O)CCC1C(=O)NCc1ccnc(C#N)c1 42559,C1(N(C(C=CC(CC)=CC)=O)CC)CCCN(C(c2ccncc2C2CC2)=O)C1 42560,CC1CC(C)(C(=O)NCC(C2CC2)N(C(=O)CC2CCCCC2O)C)CC(C)O1 42561,CC(C)(C(=O)NCCC1CN(C(=O)COc2ccsc2Cl)C1)C(F)F 42562,c1(C(=O)NCC(=O)NCC(=O)NCc2nc(C)sc2)ccnnc1O 42563,c1(OC)ccc(C(N2CCC(CNC(=O)CC(C)OC)(OC)C2)=O)cc1F 42564,c1(NC(CCOCC)=O)cccc(NC(c2snnc2C(C)C)=O)c1 42565,N1(C(CC(C)(C)OC)=O)C2CCC1CN(C(c1cnoc1C)=O)CC2 42566,C1(CNC(CC2CC(=C)C2)=O)CC(NC(c2coc(SC)c2)=O)C1(C)C 42567,C(=O)(C(C)CC(N)=O)NC1(C)CCN(C(Cc2cccc(C)c2)=O)C1 42568,N1(C(CNS(CC)(=O)=O)=O)CC2CC1CC2NC(=O)C(C)(C)c1cnn(C)c1 42569,c1(C(=O)NCC23OCC(NC(C=Cc4ccc(C)o4)=O)(C2)C3)cc(F)cnc1O 42570,N1(C(C2(Cl)C(C)(C)C2)=O)CC2CCOC2(CNC(=O)CCC2OCCO2)C1 42571,c1(OC)cc(C)nc(N(C)CC2CCN(C(=O)CC(C)SC)CC2)n1 42572,C1(CC)C(C(=O)NCc2nc(CO)n[nH]2)CCN1C(=O)C(c1cncnc1)C 42573,C1(NC2C(CC(=O)OC)CC2)CCC(O)CNC1 42574,Cc1cccc2cc(C(=O)NC3(CNC(C45CC(F)(C4)C5)=O)CCOC3)nn12 42575,c1(C(=O)NCC2(C)CCC(NC(C=C(CC)C)=O)C2)n[nH]c2c1CCC(C)(C)C2 42576,c1(NC)ccccc1C(=O)NC(C)CCC(=O)NCc1ccnc(Cl)c1 42577,CC(=O)CCCC(=O)N(C(C)CCNC(C1CCC2(CCC2)O1)=O)C 42578,c1(OC)nc(C(=O)N(C(C)CN(C(=O)C(C2CCCC2)OC)C)C)cc(O)n1 42579,CCC(C)C(O)C(=O)NC1CC(CCNC(=O)C(F)C(F)(F)F)C1 42580,C1(N(C2CC3CCC2O3)S(CCCOCC)(=O)=O)CCNCCC1C 42581,S(=O)(=O)(c1ccc(N2CC(C)C(O)C(C)C2)nc1)NCC(=C)CC 42582,N1(C(C2(C)CCN(C)C2)=O)CC2CCC(C1)N2C(c1cnn2ccccc12)=O 42583,C1(C)(N(C(=O)COc2ccn(C)n2)C)CCN(C(=O)CCc2cccs2)C1 42584,c1(C(=O)NCCC2(CNC(C(CC#C)C)=O)CC2)ccc2c(Br)n[nH]c2c1 42585,C#CC1(C(N2CCC2CC)=O)CCN(C(c2cccc(C)c2F)=O)CC1 42586,C1(C(=O)NC(CCSC)CO)N(C(C23CC(F)(C2)C3)=O)CC12CCCC2 42587,C1(NC(c2n(C)nnn2)c2ncc(-c3ccccc3)s2)C(=O)OC2CCCC12 42588,C(C)(C)(CC(C)NC(=O)CC1CN(C(=O)Cc2cccnc2F)CCO1)OC 42589,c1(NC)n[nH]c(C(=O)NCCN(C(c2cc(CS(C)(=O)=O)[nH]n2)=O)C2CC2)c1Cl 42590,CCC1=C(C(=O)NCC2CCN2C(c2c(Br)noc2C2CC2)=O)CCCO1 42591,c1(CNC(C(=O)NC(c2cc(C)ccn2)CC)=O)ccc(N2CCOCC2)cc1 42592,N1(C(C(CCOC)C)=O)CCC2(C=C(C(=O)Nc3ccc(C)cc3OC)C2)C1 42593,C(C(=O)N=c1ccn(C(C)C)[nH]1)(c1ccnn1C)NC(c1cc(C)cc(F)c1)=O 42594,Cc1cnn(CC(N2CC(NC(=O)CC3CCC(C(F)(F)F)O3)C2)=O)c1 42595,C#Cc1cn(C)nc1C(=O)NC(C(=O)NCC(F)(F)C(N)=O)C(C)C 42596,N1(C(C)=O)CCN(CCCNC(=O)C(F)CN(C)C)CC1.C1CO1 42597,N1(C(c2nc(CC)sc2)=O)CCCC(CC(=O)NCCc2cnc(C)o2)C1 42598,c1(C(N2C(C)CN(C(=O)Cc3nocc3C3CC3)CC2)=O)cc2c(nc1N)CCC2 42599,c1(-c2n(C(CC)C)nc(CCC(F)(F)F)n2)ccc2c(c1)C(C)(C)CO2 42600,Cc1ccc2oc(C(=O)NCCN(CC(C)O)Cc3ccsn3)c(C)c2c1 42601,C1(NC(c2cn(C)nn2)=O)CCOC12CCN(C(C1CC(CC3CC3)C1)=O)CC2 42602,C1(NC(c2nccn3ccnc23)=O)CCC12CCN(C(=O)Cc1cn[nH]c1)CC2 42603,CC(C)(C)CC(=O)NCC(c1ccccc1)NC(c1ccc(C(C)(C)C)s1)=O 42604,C(=O)(CC(C)CCC=C(C)C)NCC1CC(NC(c2cncc(OC)n2)=O)C1 42605,N1(C(c2ncc(OC)cn2)=O)CCC(C2CC2)C1CNC(=O)C=C1CCCC1 42606,N1(C(CN(c2ncccc2O)C)=O)CC(C2CCCCN(C(=O)CCCF)C2)C1 42607,c1(CC)ccc(Cl)c(Br)c1.C12CCN(C1C(C)C)c1nnc2n1C 42608,Cc1cccn2c(C(=O)NC34CCCC(NC(C5CCCO5)=O)(C3)C4)cnc12 42609,c1(CC(=O)NCC=CCNC(=O)CCc2cncs2)ccccc1C(=O)O 42610,C1(NC(c2c(C)cccc2Cl)=O)COC2C(NC(C3CC(F)(CO)C3)=O)COC12 42611,c1(CN2C(C(=O)NC(CC=C)CNC(C3(CC)CC3)=O)COCC2)ccc(F)cc1 42612,C(=O)(C1=C(Cl)CCCC1)N1CC(COC)(NC(C2CN(C)NC2=O)=O)C1 42613,N1(CC(N2CCC(C(=O)NCCC(=O)OCC)C2)=O)CCCCC1C 42614,c1(N2CC3(OCC(C)C3)C2)nc(N2CC(CO)C(CCO)C2)nc2c1CCOC2 42615,C1(CC(C)C)CC1N=c1[nH]c(N2CC3CC(O)CC3C2)nc2c1CCC2 42616,CCC(CC(=O)N1CC2CCC(C(=O)N(C)CCC3CCCCC3)(C2)C1)C(C)C 42617,C1(C(=O)NCC(C)(C(C)C)NC(Cc2c(C)noc2C)=O)C(O)C(=O)N(C)C1C 42618,c1(C(N2CC(NC(C3C(C)(C(F)F)C3)=O)C2)=O)c(C2CC2)nc2sccn12 42619,N1(C(c2c(Nc3c(CC)cccc3)ccs2)=O)CC2=C(C1)CN(CC)C2 42620,Cc1ccc2[nH]cc(C#N)c(=NCC3CCOCC3(C)C)c2c1 42621,Cc1c(F)cc(C(N2CC3CN(Cc4ccc(O)c(I)c4)C3C2)=O)cc1Br 42622,c1(N2CC(=C(CNC(c3c(C)csc3)=O)F)C2)ncnc2onc(C)c12 42623,Cc1n[nH]c(C)c1C(C)CC(=O)NCC(F)CNC(=O)CCC(F)F 42624,S(=O)(=O)(CCC(=O)NC(CNC(C1CC1c1cncn1C)=O)CO)NC 42625,C(c1ccc(Cl)c(Cl)c1)=CC(=O)N(C(C)CNC(c1cnnn1C)=O)C 42626,C12(CNC(=O)CCNC(c3ccsc3)=O)CC(CO1)N(c1ncccn1)C2 42627,CC(CN(C)C)CCC(=O)N(CC(C)(C)NC(=O)Cc1csnn1)C 42628,CC1(C)CN(C(c2ccsc2Cl)=O)CCC1NC(=O)CCCC1CC1 42629,C1(C)(CNC(Cc2c(CN(C)C)con2)=O)CCCN(C(c2ccnnc2)=O)C1 42630,CCCCC#CC(C)(C)NC(=O)C(C(C)C)NC(=O)CC1=CCOCC1 42631,c1(CC(=O)NC2CCC(CNC(CC=CC)=O)C2)ccc2nn[nH]c2c1 42632,C1(C(=O)NCCCNC(=O)COC2CCCCCC2)CCc2ccccc2C1 42633,N1(C(=O)NCC(C2COC(C)(C)O2)O)CCC(=C(Br)Br)CC1 42634,Cc1cccc2[nH]c(-c3ccnc(NC(c4ccccc4[N+](=O)[O-])=O)c3)cc12 42635,C(=O)(C(C)(F)C(=O)NC1(CCC(=O)NCC2CCCC3(CC3)C2)CCC1)OC 42636,N1(C(=O)OC(C)(C)C)CCCC(NC(=O)CCc2nnc(C(F)F)o2)CC1 42637,C(c1nc2ccccc2s1)=CC(N1CCN(C(CCCC=C)=O)CC1)=O 42638,CC1(F)CC(C(=O)NC(C(=O)NCc2nn[nH]c2C2CC2)c2ccoc2)C1 42639,N1(C(CS(=O)(=O)N(CC)CC)=O)CC(OC)CC(NC(c2cc[nH]n2)=O)C1 42640,c1(N2CCC(N(C(C3CC(=O)CC(=O)N3)=O)CC)C2)[nH]c(=O)n(C)c(=O)c1C#N 42641,N1(C(CCOCC)=O)CCN(C(=O)C(N2CCOCC2)C)CC1COC 42642,C(=O)(C(C(F)(F)F)C(F)(F)F)NC1CCC(NC(C23C4C5C6C4C2C6C35)=O)C1 42643,C1(COC)CCN(C(c2csc(CNC(c3ccc(Cl)s3)=O)c2)=O)CC1 42644,c1(OC)ccc(C(=O)NC(C)CCNC(C2CCN(C)C2=O)=O)c(F)c1F 42645,C(CC1=CCCCCC1)NC(C(C)N(C(=O)C(O)C(C)(C)c1ccccc1)CO)=O 42646,O(NC(=O)CCN1CCSCC1)CC(=O)N(C(C(=O)OC)C)C1CC1 42647,c1(C(=O)NC(CC=C)CNC(=O)CC(C)C)ccn2cnc(C)c2c1 42648,C(=O)(CCCCCn1cc(-c2ccnn2C2CC2(F)F)nn1)N(CCCC)CC 42649,C(=O)(C1=CCN(C(c2csc(CO)n2)=O)CC1)NC1(CC)CCCC1 42650,N1(CCC)CCCCC1C(=O)NC1CCC1NC(c1ccn(C2CC2)n1)=O 42651,C1(C(N(CC(C)NC(=O)Cc2ccon2)CC)=O)COc2cc(Cl)ccc2C1 42652,N1(C(C(C=C)(C)CC)=O)CCC2(CCCN2C(C2CC(F)(F)C2)=O)C1 42653,c1(C(=O)NC(CNC(CN(C)CC)=O)CC(C)C)cnc2n1CCS2 42654,c1(C(=O)OC)ccc2ccccc2c1C(=O)OC.c12ccc(cc1Br)NC(=O)C2 42655,C1(c2cn(CC3N(C(=O)CCOC4CCC4)CCC3)nn2)CC2CCC1CC2 42656,C12(C(N3CC(CNC(CC=C(C)C)=O)C4C3C4)=O)CCN(CC1)S(=O)(=O)C2 42657,CC(C)(Cc1cnn[nH]1)C(=O)N1CCC(CNC(c2ccc(C(F)F)cc2)=O)C1 42658,n1(C(C2CC2)NC2CCC2)cnnc1C(=O)NCC1(C(N(C)C)=O)CCCO1 42659,c1(C(N2C(CNC(CCC#C)=O)C(C)(C)CC2)=O)ccc2c(c1)OCCC2 42660,N1(C(C(CO)OC)=O)CCC(C(F)F)(CNC(=O)CCc2ccncc2)C1 42661,c1(C(=O)NC2(CC)CCN(c3nnc(C(N)=O)s3)CC2)cccc2c1nnn2C 42662,C(=O)(C1CCc2ccc(OC)cc21)NC1CC(CNC(C(CC)(C)C(N)=O)=O)C1 42663,c1(NCC(C(C)C)(C)C)nc(N2CCC3C(C2)C3(F)F)c2ccsc2n1 42664,C1(C(=O)NCCC(C)NC(C2CCC3CC2C3(C)C)=O)CCC2CCCCC2C1 42665,c1(OC)ccc(C(N2CCN(C(=O)C=Cc3cc(Br)cs3)CC2C)=O)c(OC)c1 42666,S(=O)(=O)(CCC(=O)N(C1CN(C(c2ccc(C(=O)N(C)C)cc2F)=O)C1)C)NC 42667,C1(OC)CC(NC(c2cc(C)ns2)=O)C12CCN(C(c1cnc(O)o1)=O)CC2 42668,C(=O)(CC(C)(C)CNC(=O)C(C)CO)NCCn1c(C)cc(C)n1 42669,C1(CC(=O)NCCCOCCCNC(=O)CCSCCO)CCCCO1 42670,C1(C(=O)NCc2nc(C)c(C)o2)N(C(=O)C(Cl)Cl)CC12CCCC2 42671,CC(C)C(C(=O)NCC(=O)NCC(N1CCOCC1)=O)NC(N)=O 42672,N1(C(C2CC(O)C2)=O)CCC(S(=O)(=O)N2CCCCC2)C1 42673,N1(C(c2c(C)ccc(C)c2)=O)CC(c2ccccc2C(F)(F)F)C2(CCC2)C1 42674,c1(C(=O)NCCN(CCC)C(c2cnc(C(C)C)o2)=O)c(C)coc1C1CC1 42675,c1(CC(=O)NCC(=O)NC(CNC(CSCCCC)=O)C2CC2)cccc(C)c1 42676,c1(NC(C(CN(C)C)NC(=O)CC2CC3C=CC2C3)=O)ccc(Cl)cc1O 42677,c1(CC(C)NC(c2cc(Cl)nnc2O)=O)ccc2ccccc2c1 42678,C1(CC)(NC(C2CCC(=O)N2)=O)CCCN(C(=O)CCCN(C)C)C1 42679,Cc1nncc(C(=O)NC(CCN(C)C)C(=O)NCC(O)C2CCC2)c1C 42680,N1(C(C2ON=C(CC)C2)=O)CCN(C(=O)Cc2ccc3c(c2)CC3)C(C2CC2)C1 42681,C1(NC(C2(SC)CC2)=O)COC2(CCN(C(c3ccc4ccccc4c3)=O)C2)C1 42682,c1(C(=O)CN2CCC(c3nnc(C4CCOCC4)o3)CC2)ccc(Br)c(Cl)c1 42683,C1(C(=O)NC(CC(C)NC(C2(C#N)CC3(CCC3)C2)=O)C)CCc2n[nH]cc2C1 42684,C1(C(=O)NC2CC3CC(NC(C(C(C)C)O)=O)CC32)CCC2(CC1)CNC(=O)C2 42685,c1(CC(=O)NCC2(F)CCN(C(C3(O)CCSC3)=O)C2)cnn2ccccc12 42686,CCCCCCCC(=O)N(C)CC1CN(C(=O)CC2CC(SC)C2)CCO1 42687,Cc1cocc1CNC(C1(NC(=O)COC2CCOC2)CCSC1)=O 42688,c1(OC)ccc(C=CC(=O)NCC(C)(C)CNC(=O)CCCS(N)(=O)=O)cc1O 42689,N1(C(CC2CC(=C)C2)=O)C2CCC1C(C(=O)Nc1ccc(F)c(CC)c1)C2 42690,C1(CNC(C2CC(OC)C2)=O)(NC(c2sncc2C)=O)CCCCC1C 42691,c1(CCC(=O)NC(C)CNC(C23CCCC2C3)=O)ccc2ccccc2n1 42692,C(C(C)CN(C(=O)CCNC(=O)C=CCl)C)NC(C1(SC)CC1)=O.C1CC1 42693,C1(NC(=O)CSc2cnco2)CCCCC1Nc1ncccn1 42694,C(=O)(C(CCC)C1CC1)NCC(CC=C)NC(c1cc(-c2ccns2)on1)=O 42695,c1(C(=O)NC(CNC(C(CC=C)(C)CC)=O)CO)cc(S(N)(=O)=O)sc1C 42696,C1(C(N(C2CCCC2)CC=C)=O)CCC(C)(C)N(C(C2CC2(F)Cl)=O)C1 42697,C(=O)(C(C(C)(C)NC(C)=O)c1ccccc1)N1CCN(CCCOCC)CC1 42698,c1(C(=O)NC(CC(=O)NCCCN(C)C)CC2CC2)ccc(F)cc1F 42699,C1(CNC(CCCC=C)=O)CC2CCC1N(C(=O)CCCc1n[nH]c(=N)s1)C2 42700,c1(C(=O)NC2CN(C(c3cccc(OC)c3)=O)C(CO)C2)cccc2nn[nH]c12 42701,N1(C(CCCn2cc(-c3nc(C(=O)O)sc3)nn2)=O)CCC2C(C1)C2(Br)Br 42702,c1(C(=O)OC)cc(C(=O)NCC2(NC(c3cscc3F)=O)CC2)n2c1COCC2 42703,c1(C(N2C(CNC(C(C)Oc3ccccn3)=O)CC2)=O)cccc(C(N)=O)n1 42704,c1(C(CC)(C)O)cn(CCCNC(c2coc(C(C)C)n2)=O)nn1 42705,CC1(C)CC(O)CN(C(=O)Cc2ccc(SCC(F)(F)F)cc2)C1 42706,CCC(C)(C)C(O)C(=O)N1CCCCC(CNC(C2CN3CCN2CC3)=O)C1 42707,c1(N2CCC(CCNC(C(C(C)C)(C)O)=O)CC2)ncc([N+](=O)[O-])cc1C(N)=O 42708,c1(C(=O)NCC(C)NC(=O)C(C)(C)CS(N)(=O)=O)cc2c(cc1Cl)NC(=O)C2 42709,c1(C(=O)NC(CNC(C(CC)CC)=O)(C)CO)ccnc2ncnn12 42710,c1(COC)ccc(-c2nc(CCC(C)C)nn2C)cc1OC.c12cc(C)cnc1S2 42711,Cc1n[nH]c(C)c1CC(N1CC2C(CN(C(=O)C(C)(C)C)C)C2C1)=O 42712,C1(C(=O)NCC2(NC(CCc3onc(CC)n3)=O)CCC2)CC(F)(F)C12CCC2 42713,Cn1ncc2cc(CN3CC4(CC4C(=O)Nc4cc(Cl)c(Cl)cc4Br)C3)ccc12 42714,CC1CCC(C(=O)C(=O)N)CN1C(=O)CN(C1CCCCC1)C.C1(C)(N)CCCC1 42715,c1(C(=O)NC(CNC(C(C)(C)OCC)=O)C)cccc(C)n1 42716,c1(CC)ncc(Cl)cc1C(=O)N(C(C)CO)NCC(C(C)C)N1CCCC1 42717,C1(NC(C=CC)=O)CCN(CCN(C(=O)CC2SC(=N)NC2=O)C(C)C)CC1 42718,C12(NC(C(CC#C)CC#C)=O)CCCC1(F)CN(C(=O)C(C)COCC)C2 42719,Cc1nnc2c(C(=O)NCCC(C)NC(c3ccncc3N=[N+]=[N-])=O)cccn12 42720,c1(C(c2nnnn2C2COC2)OCC=C)cccc(CCCC#N)c1.C1(C)CN1 42721,n1(CCN(C(CC2(CSC)CC2)=O)C)cc(CC(=O)CCCn2cc(C)cn2)nn1 42722,C1(CN(C)C)COCCN1C(=O)CC(C1CC1)NC(=O)C(C)(C)C1CCOC1 42723,C(=O)(C1=CC2CC(C1)CC2O)NC(CNC(Cn1nc(C)oc1=O)=O)C(C)(C)C 42724,S(=O)(=O)(c1ccc(F)cc1Cl)NCC(N1CCOCC2(COCCN2)C1)=O 42725,C1(C2CC2)(C(=O)OC)CCN(C(=O)NCCN2CCCCC2C)C1 42726,c1(OCC)ccc(C(C)NC(=O)CCC2(C)CC2)cc1F 42727,CC(CC(F)(F)F)C(=O)NC1CCN(C(=O)C=C2CCSCC2)CC1O 42728,c1(NC(C2N(Cc3ccc(C)s3)CCCC2)=O)cnc(Br)c(Cl)c1 42729,CCCC(C)(CCC)C(=O)N1CCC(CNC(=O)CSC(F)F)(OC)C1 42730,c1(NCC#CC)cc(=NCC(C(C)C)c2ccnn2C)[nH]cn1 42731,C1(NC(c2ccc(COC)o2)=O)CCN(C)CC1.C12(CCC1)CC(=O)N2C1CC1 42732,c1(C(=O)NC2CCN(C(C(Br)=C(C)C)=O)CC2C)ccc2[nH]ccc2c1 42733,CCC(CC1CC1)C(=O)N1CC(NC(=O)CCN(C)CCO)C(F)C1 42734,Cc1nc(CCCC(=O)NCCCC2(NC(c3cscc3C(F)F)=O)CC2)cs1 42735,C1(CC)C(C(NCP(C)(C)=O)=O)CCCN1C(c1ccccc1F)=O 42736,N1(C(CN(CC)CC)=O)CCC2(CCCN2C(=O)CC(F)(F)c2ccccc2)CC1 42737,C1(C(=O)NC2C(C(=O)NCc3c(C)csc3)CC=CC2)CC(=O)CC(=O)C1 42738,N1(C(c2n(C)cnc2)=O)CCc2sc(CNC(=O)CCc3cnc(O)[nH]3)nc2C1 42739,c1(C(N2CCC(NC(C(COCC)O)=O)(CO)C2)=O)cc2occc2n1C 42740,C1(CC(=O)NC(C(=O)NC(C#C)C(C)OC)C2(C)CC2)CCCCN1C 42741,CC1CN(C(=O)CC2(C(F)F)CC2)CC(CCNC(c2cc(C(N)=O)cs2)=O)O1 42742,C1(CC)CC(C)CN(C(=O)CC(C)(C)NC(=O)CCCN=[N+]=[N-])C1 42743,c1(C(=O)NCC(CC(=O)N(CC(=C)C)C)OC)cnn2c1OCC2 42744,C1(c2nnnn2-c2ccccc2)(NCC2COCC(C)(C)O2)CSC2CCCC12 42745,N1(C(CSS(C)(=O)=O)=O)CC(NC(=O)Cc2cc(-c3ccccc3)on2)C(F)C1 42746,c1(C(=O)NC2C(NC(c3ccc(OC4CC4(F)F)cc3)=O)C2)ccc[n+]([O-])c1 42747,C1(CC)CN(C(=O)C(=O)N(C)C)c2ccccc2O1.c12cc(n[nH]1)C(=O)NC2 42748,c1(C(N(CCCN(C(CCNC(C2C(C)C2)=O)=O)C)C)=O)scc2c1CCCC2 42749,C(=O)(CC(C(C)C)C(C)C)NCCC(C)(C)C(C1CC(F)(F)C1)C(=O)OC 42750,Cc1cnn(C)c1CC(N1CC(N(C)C(C2C3COCC23)=O)C1)=O 42751,C1(C(C)C)C(NC(=O)CNC(=O)CC(C)(C)C)CCN1C(=O)CC1CC(C)C1 42752,C1(C)CC(C)(C)CN1N(CCC(C)C)C(=O)NC(CC(C)C)C.c1(N)cc[n+]([O-])cc1 42753,c1(OC)c[nH]c(C(N2CC(C)(C)CC2CNC(C2CC=CCO2)=O)=O)cc1=O 42754,CCC(C)C(O)C(C)C(=O)N1CC(NC(=O)CCCCCC(C)C)C(O)C1 42755,N1(C(C(C)Cc2ccc(F)cc2)=O)CC(CO)CC(C)C1 42756,CC12CC1CN(C(=O)C(N1CCC(c3cnccn3)CC1)=O)C2 42757,c1(C(=O)NCCCNC(C(CC)O)=O)ccc(CC2CC2(Cl)Cl)cc1 42758,N1(C(C(CC)OCC)=O)CCC(CC(=O)NCC(C)(O)CC)C1(C)C 42759,C1(O)(CNC(=NCC=C)NCCc2nc(C)cc(C)n2)CCC2(CC1)OCCO2 42760,O=C(CCCc1ccsc1)NCc1nccn1C(F)F 42761,C=C=CCCC(=O)NCCNC(c1ccccc1)CNC(=O)CCC1CC1(C)C 42762,C(C(C(=O)N(C)CCN(C)C1CC1)C(C)C)NC(c1c(C)n(C)cn1)=O 42763,c1(C(=O)NC(C(=O)NCCc2n(CC)cnn2)C2CCOC2)nnc(S)n1C 42764,S(=O)(=O)(CCC(=O)NC1CN(C(C2CCSC2)=O)CC1CC1CC1)NC 42765,C(C(O)CS(C)(=O)=O)NC(=O)NCc1sc(C)c(-c2ccccc2)n1 42766,C(=O)(CC(C)(C)CCC)NCC(CC=C)C(=O)NC1COCC1O 42767,C(=O)(CCCC(C)=O)N1CC(NC(C(C)=CC)=O)C(c2nccn2C)C1 42768,C1(C(=O)NCCCN(C(c2cc(O)nn2C)=O)CC)OCCOC12CCC2 42769,N1(C(C(C)(C)NC(=O)OC)=O)CCC(CNC(c2cc(CO)n(C)n2)=O)CC1 42770,C1(C(=O)NC(C)CNC(C2CC(F)(CO)C2)=O)COCCN1CC(F)F 42771,C=CC(C)CC(=O)NC1CC(NC(c2ccccc2SCCO)=O)CC1O 42772,O=C(C1=CCN(C(C2CC2C2CC2)=O)C1)NCCCF 42773,C(=O)(C(F)(F)C1=CCOCC1)N(C)CC1(NC(=O)C(F)(F)CC2CCCO2)CC1 42774,c1(NC(c2cccc(I)c2)CC)ncc(C)cc1[N+](=O)[O-] 42775,C1(C(=O)NC2C(C)CCN(C(C=C(C)C)=O)C2C)CCc2nc(O)[nH]c2C1 42776,c1(C(=O)NC2CC(CNC(=O)CC3CCCCC3O)C2)ncc(F)cc1F 42777,C1(C(N2CCC(CNc3cc(Cl)ncn3)C2)=O)CCCCC1n1cccn1 42778,C(=O)(C(F)(F)C(F)(F)N(C)C)N1CCN(C(=O)OC)C(c2ccccn2)C1 42779,C1(CC(N2CCC(C(=O)OCC)C2)=O)CCN(S(=O)(=O)Cc2ccccc2)C1 42780,c1(C(N2CCC(C#N)(NC(c3ncc[nH]c3=O)=O)C2)=O)cc2cc(Cl)cnc2[nH]1 42781,C(CCCC(=O)NCC1CCCCN1C(c1cccc(F)c1SC)=O)(OC)OC 42782,N1(C(C(CCSC)OC)=O)CC2CC3CC2C1C3NC(=O)C(c1ccc(Cl)s1)C 42783,c1(CN2CC(NC(c3c(O)cccc3F)=O)(CO)C2)c(O)ccc(Cl)c1Cl 42784,N1(C(c2c[nH]cc2Br)=O)CCN(C(c2cc(Cl)c[nH]2)=O)C(C2CCCC2)C1 42785,c1(-c2ccc(-c3n(CC(CC)CO)ccn3)s2)cc(-c2ccccc2)n(C(C)C)n1 42786,Cc1cc(C(N2CC3CC3(CNC(C3CC34CCCC4)=O)C2)=O)cnc1C 42787,Cc1ccc(C(=O)NCC2COC(CNC(=O)Cc3csc(Cl)c3)C2)cc1CO 42788,C(C(C(=O)N1CCC(C)(NC(c2ccc(F)s2)=O)C1)C(C)(C)C)OCC=C 42789,c1(C(=O)NC(CC)CN(C(=O)C(CO)NC(N)=O)C)ccc2c(c1)NC(=O)CC2 42790,C1(C)(CNC(C2CN(C)C(C(F)(F)F)C2)=O)CCS(=O)(=O)N1 42791,C(=O)(C(C)(C)C(=O)OC(C)(C)C)N1C(C)CC1C(=O)NC(c1ncc[nH]1)(C)C 42792,Cn1ncc2cc(C(=O)NCC=CCNC(c3c(Cl)nsc3Cl)=O)cc(O)c12 42793,CCCC(CCC)CCCC(=O)N(C)CCNC(c1cc2c(cn1)CCCC2)=O 42794,CC(C)=C=CC(C)(C)C(c1nnnn1C1COC1)NCCc1cccc(Br)c1 42795,c1(OC)ccc(C(N2CC(CNC(c3cc(C#N)c[nH]3)=O)C3CC23)=O)cc1Cl 42796,CCS(=O)(=O)c1ccc(S(=O)(=O)NC(c2csc(C)c2C)=O)cc1 42797,C1(CC(=O)NCc2cnn(C3CCC3)n2)CCCN(C(c2ccc(F)cc2)=O)C1 42798,C(CC(=O)NCC1(CN(C(=O)CCC2CC2(Cl)Cl)C)CC1)SC 42799,c1(CCS(N2CCC(Oc3ccc(C)cc3)CC2)(=O)=O)nc2ccccc2[nH]1 42800,N1(CC)CCC(NC(=O)CCN(C(C2(C(C)(C)O)CCC2)=O)CC)CC1 42801,N1(C(C2(C#C)CCC2)=O)CCCC(NC(=O)CSCc2ccncc2)C(F)C1 42802,C1(C(N2C(CCC)CN(C(=O)CC(C)(C)C)CC2)=O)Cc2cncn2C(=O)N1 42803,C#Cc1c[nH]nc1C(=O)NC1CN(C(=O)Cc2csnc2C)CC1O 42804,c1(C(=O)NCC2C(NC(c3ccc(CN(C)C)nc3)=O)CC2)cc2ccsc2s1 42805,N1(C(CN2CCC(C)(O)C2)=O)CC2CC(NC(=O)CNC=O)C(C2)C1 42806,C1(C(N(CC(CC)(C)OC)C)=O)CC(C2CCCCC2)CN1C 42807,C(=O)(CC(C)(C)CC(F)(F)F)NCC(CNC(CCOCCCOC)=O)OC 42808,C(=O)(CCCC(C)(C)C)NCCNC1(CC=C)CCN(C(=O)C(=O)NC)C1 42809,c1(C(N2C(CC(=O)Nc3csc(Br)c3)CCC2)=O)ccnc2ccc(O)cc12 42810,C1(C(=O)NCC2(CCOC)CCC2)CCN(C(c2cc(C)[nH]n2)=O)C1C 42811,C1(CNC(CC(C)(C)C2CC2)=O)CC(F)(F)CN1C(=O)CC1(CO)CCCCC1 42812,c1(CC(=O)N(CC(C)NC(C(CC#C)(C)CC)=O)C)ccc2ccccc2c1 42813,c1(OC)cc(C(=O)NC2CC2NC(C2CC(C)(O)C2)=O)ccc1O 42814,C#CCCC(C(=O)NC1CCCC(O)C1O)NC(C1COCC(C)O1)=O 42815,C(C(=O)N1CC(NC(=O)C(C)(C)C#N)C(c2ccnn2C)C1)(C(C)C)SCC 42816,CCC(C(=O)N(C)C)NC(=O)COC(C1OCCC1CNC(N)=O)=O 42817,C=CC(C)(CC)C(=O)NC1CC(CCNC(c2ccc(C)c(C)c2)=O)C1 42818,c1(C(=O)NC(C2N(C(C(COC)OC)=O)CCC2)C)n[nH]c2ccc(OC)nc12 42819,C1(CC=C)(NC(c2ccnn2C)=O)CN(C(c2cc(C(C)(C)C)c[nH]2)=O)C1 42820,N1(C(C2CCC(C)S2)=O)CC2=C(C1)CN(C(C1(NC(C)C)CC1)=O)C2 42821,c1(C(=O)NCC2(O)CC(NC(CCS(C)=O)=O)C2)c(F)cccc1Cl 42822,c1(CC)ccc(N)c(C(=O)N(CCCN(C)C(c2cscc2C2CC2)=O)C)c1 42823,C(=O)(C(C)C(O)C(C)CC)N1CCC(C(=O)NC(C#C)C(C)OC)C12CC2 42824,n1(CC(=O)NCC2CC(F)(CNC(C3CC(=C)C3)=O)C2)cc(C#N)cn1 42825,C1(O)(CNC(C(C=CC)O)=O)CCN(C(=O)Cc2ccccc2C)C1 42826,N1(C(C=Cc2c(C)n[nH]c2)=O)CC2CN(C(=O)CC3CCCN(C)C3)CCC12 42827,C1(NC(c2c(C(C)C)con2)=O)CN(C(c2cc(C#N)c[nH]2)=O)CC2(CCC2)C1 42828,N1(C(C(C)NC(=O)NC)=O)CC(CNC(=O)CCn2cc(Cl)cn2)C(C)C1 42829,N1(C(Cn2cc(CCOC)nn2)=O)CCN(C(c2cncnc2C)=O)CC(O)C1 42830,CC(C)S(=O)(=O)c1cccc(C(CNC(=O)CO)NC(=O)C(C(C)C)N(C)C)c1 42831,N1(C(c2c(C)nsc2)=O)CCN(C(C2CC(C(F)(F)F)C2)=O)CC(CO)C1 42832,CC(C)C(C)CC(=O)N1CC(N(C(=O)CCc2cc(Br)ccc2F)C)C1 42833,N1(C(CC2C(C)(C)OCCO2)=O)CCC2CN(C(=O)CCC#N)CC2C1 42834,Cc1cc(C(=O)NCC(CC(C)C)NC(C2CCC(F)CC2)=O)cnn1 42835,c1(NC(C)=O)ccc(NC2CCN(C(=O)N(C3CCN(C)CC3)C)CC2)cc1Cl 42836,c1(C(c2nnnn2CCCOC)NC(CCC)CCC)nn(C)c(C)c1Cl 42837,N1(C(c2cnn(C(C)C)c2F)C(=O)NCC)CC(C(C)C)c2ccccc21 42838,C1(C(=O)NCC(CC(C)C)NC(C2C=CCS2)=O)CC(C2CCCC2)C1 42839,C1(C)(C(N(CCC)CCNC(C2CC2c2nncn2CC)=O)=O)CC(F)(F)C1 42840,C12CCCCC1C2.N1(C(C(=O)C(O)C2CCCC2)=O)CCOCC1.C1C(=O)NO1 42841,C1(C(=O)NCC2C(C)(C)CCCN2)CCc2ccccc2N1 42842,N1(C(c2scc(C)n2)=O)CCC(O)CC1.N1(C(C)=O)CCC(c2nn[nH]n2)C1 42843,N1(C(C(COC(C)C)NC(=O)CC(=O)N(C)C)=O)CCC(C)C(N(C)C)C1 42844,c1ccc(Cl)cc1Br.C1(C(C)C)CN(C(=O)NC2CN(C(=O)N(C)C)C2)C1C(C)C 42845,CCCCCCC(CC)(CC)C(=O)NCC(CNC(=O)CN(C)CCOC)OC 42846,C1(C(C(=O)NCC(O)CNC(c2coc(C(C)C)n2)=O)OC)CCC(F)(F)CC1 42847,C(C)(C(C)S(C)(=O)=O)N(C(C(=O)NC1CN(C(C)C)C(=O)C1)=O)C 42848,N1(C(=O)OC(C)(C)C)CCCC1C(C)(C)CO.c12cnc(o1)[nH]c2=O 42849,c1(CNC(Cc2c(C)nn(C)c2)=O)n[nH]c2c1CN(C(=O)C(C)S(N)(=O)=O)CC2 42850,c1(C(N2CC3CCCC(C2)N3C(C23CC(C2)C3)=O)=O)ccc2ncccc2c1 42851,C1(O)(C(=O)NCC2(CC)CN(C(=O)CCCC(C)(C)C)C2)CCCC(C)CC1 42852,c1(CCC(=O)OCC2CC(C)(OC(F)F)C2)cncc(F)c1 42853,c1(C(=O)NC2CC(F)(CNC(C3(C)CCN(C)C3)=O)C2)cccc2nc(O)[nH]c12 42854,c1(OCC)cc(C)[nH]c(=NCC2CC3CCC2N(C(c2csc(CO)n2)=O)C3)n1 42855,N1(C(CNC(=O)OC)=O)CCCC(O)(CNC(=O)CSc2ccc(C)cc2)C1 42856,c1(C(=O)NC(C(=O)NCCc2ccc(C)s2)C2CC2)cnc(C)c(C)c1 42857,c1(C(=O)NC2(CNC(c3cccc4ncnn34)=O)CCC2)ccc(O)c(F)c1F 42858,c1(CC)ccc(C(=O)N(C)CC2CCN(C(C3CC(=O)NC3(C)C)=O)C2)c(C)n1 42859,N1(C(C2CC(C)(C)C2)=O)Cc2ccnn2CC(NC(C2CCCCC(=O)N2)=O)C1 42860,c1(OC2(CC)CC2)ccc(C(=O)NC2CCC(Oc3ccncc3)C2)cc1 42861,C(C(C)C(=O)NC1COCC1NC(c1cc(C(N)=O)c[nH]1)=O)OCC 42862,C1(C(=O)NCCCCN(C)C(C2(C)CCCN2C)=O)CCC(O)CC1 42863,c1(C(CC)C(=O)N(CC(O)CN(C(=O)C=CC(=O)NC2CC2)C)C)ccc(F)cc1 42864,C12(CNC(c3nc(CC)cs3)=O)CCCC1N(C(=O)C(CCOC)OC)CCC2 42865,N1(CCN(C)C(c2cccc(F)c2)=O)CCN(C(=O)Cc2ccncc2Cl)CC1 42866,c1(C(C)OC(C2CCC(NC(=O)C3CC3)CC2)=O)ccc(Br)c(F)c1 42867,c1(C(C)(C)NC(CC(CC)(C)C)=O)ccc2c(c1)OCCO2 42868,c1(C(=O)NC2CCCC(NC(c3nsnc3O)=O)C2)ccc2nc(Cl)nn2c1 42869,N1(C(c2cn(CC)nc2)=O)CCC2(CCC(CNC(c3csnn3)=O)OC2)CC1 42870,Nc1c(CNC(=O)NC2CCCC2c2cccc(Br)c2)cccc1F 42871,c1(C(=O)NCCC2(C)CCCO2)ccc2c(N)nccc2c1 42872,c1(C(=O)NCC2(C)CCN(C(CCC(C)OCC)=O)C2)cc(Cl)c(F)cc1F 42873,c1(NCCC(=O)NCC2(F)CN(C(CCNS(C)(=O)=O)=O)C2)ccc(C)cc1 42874,C1(NC(=O)CC2(CO)CC2)CCOC(C(N2CC(O)(c3cc[nH]n3)C2)=O)C1 42875,C(C(=O)NC1CCC1CNC(C12CCC(CC1)CC2)=O)(C(C)(C)C)SC 42876,c1(NC(=O)NCC(C(C)C)C)nc(-c2ccccc2)c(Cl)s1 42877,c1(OC)cc(CN2CC(C(=O)N3CCCCO3)CC(N)C2)cc(Br)c1OC 42878,CC(C)(CC1CCOC1)C(=O)N(C1CCN(C(=O)CCc2cnoc2)CC1)CCO 42879,CCC(C(=O)N1CCOCC(CNC(c2cnn(CC3CC3)c2)=O)C1)C(C)(F)F 42880,C(CCC(F)(F)F)N(C(CC1N(C(Cc2c(C)con2)=O)CC1)=O)C 42881,c1(C(N(CCCCCC)CCNC(=O)C(C)C#N)=O)ccc2nonc2c1 42882,CC(C)CC(C)(CNC(=O)C(O)C(F)F)NC(c1ccc(Cl)o1)=O 42883,c1(C(N2C(CNC(CCC=C(C)C)=O)C=CC2)=O)cnc2ccnn2c1C 42884,Cc1ccc2oc(C(=O)NC(C)(C)CCCNC(C3(CF)CCC3)=O)cc2c1 42885,CC(C(=O)NCCSCC(=O)NC(C)COC(C)C)=CC1CC1 42886,c1(CN(C)CCn2cc(C(C)NC(C3COC(C)C3)=O)nn2)ccccc1F 42887,C1(N(C(C(CNC(c2nc(C(C)C)oc2)=O)O)=O)C)CCCC1(C)O 42888,Cc1cc(Cl)cc(C(=O)NCCCNC(c2n[nH]c3c2CSCC3)=O)c1C 42889,CN1CC(C(=O)NCCC(O)CNC(C2(C(F)(F)F)CCCC2)=O)CCC1=O 42890,c1(C(=O)NCC2N(C(C3C(CC)CCC3)=O)CC2)cccnc1C(F)(F)F 42891,N1(C(C2C(C)(Br)C2)=O)CCCC(C2CC2NC(c2cnn(CC3CC3)c2)=O)C1 42892,c1(C(=O)NCC2C(NC(C=CC(C)C)=O)C2)cccc(C2CC2)n1 42893,Cn1nc(-c2ccccc2)cc1C(=O)OC1COCC1C(=O)NC1CCCO1 42894,C(=O)(C(C)CC(F)(F)F)N(CC(C)NC(c1coc(C(F)F)n1)=O)CC 42895,C(=O)(CCn1ccnc1)NCC1(CC(=O)N(CC(C)O)CCO)CC1 42896,c1(SC(C)C(N)=O)ccc(C(=O)NC2(C)CN(C(c3ccncc3)=O)C2)cc1 42897,c1(-c2n(-c3c(C)cccc3C)nc(C(C)C3CC3)n2)sc2cccc(F)c2c1C 42898,c1(C(N2CC(NC(=O)C(F)(F)CO)CC(C)C2)=O)nc2cccnc2s1 42899,CCCCC(CNC(C1CCCN1C)=O)NC(c1snc(Cl)c1Cl)=O 42900,N1(CC#C)CCC(NC(c2cnc(C(C)O)s2)=O)C1 42901,c1(C(=O)OC)ccc(C(=O)OC(C)C(=O)NC2CCOCC2C)nc1 42902,N1(C(CC2C(C(C)(C)C)C2)=O)CCCC(CNC(=O)CCn2cnnn2)CC1 42903,C(=O)(CC(CNC=O)CC(C)C)NC1(CNC(CCN(CC)CC)=O)CCCC1 42904,c1(CNC(=O)NC(c2ccc3cc(Br)ccc3c2)C)ccc2c(c1)NC(=O)CO2 42905,c1(OCC(N)=O)ccc(C(=O)NCC(C)NC(=O)C=CSc2ccccc2)cc1 42906,c1(C(=O)NC2(C(=O)NCc3ncccc3F)CCSC2)ccc(O)cn1 42907,C1(OC)CCN(C(=O)CCCC2(NC(c3cccc(F)c3)=O)CCC2)CC1(C)C 42908,C(=O)(C1COc2ccccc21)N1CC(C)(C)OC(CNC(C2CC=CCC2)=O)C1 42909,c1(C2(NC(=O)CCn3cc(C4CCC(=O)NC4)nn3)CC2)nc(C)cc(C)n1 42910,N1(C(C2N(Cc3c(N(C)C)cccc3)C3C(C2)C3)=O)Cc2ccc(Cl)cc2C1 42911,Cn1cc(C(=O)NC2CC2CNC(c2ccc(-n3cncn3)cn2)=O)n(C)c1=O 42912,N1(C(c2cncc(SCC)n2)=O)CCN(C(=O)CC=C(C)C)C(C)C1C 42913,c1(C(=O)NCC(CNC(C(CCCC)C)=O)F)ccc(S(N)(=O)=O)cc1Cl 42914,c1(C(=O)NC(C2(O)CN(C(CCC#C)=O)C2)C)cncc(C)c1Cl 42915,N1(C(C(COCC)NC(=O)C=CC(=O)NC)=O)CCCC(N(C)C)CC1 42916,c1(C(=O)OC)nc(Br)cnc1NC(C1CCC(C)N1Cc1ncc(Cl)cc1C)=O 42917,C(=O)(CS(=O)(=O)C1CC1)NCC(CC1CN(C(C(CCC)OC)=O)C1)(C)C 42918,C1(C)(C(N(CCCNC(c2c(C)occ2)=O)C2CC2)=O)CCOC(C)C1 42919,C1(C(N(CCCCN(C(C(=Cc2cccs2)C)=O)C)C)=O)COC2COCC2O1 42920,c1(C(=O)NC(CCNC(c2c(C)n(C)nn2)=O)(C)C)ccc2[nH]c(=N)[nH]c2c1 42921,CCCN=C(NCn1c(CC)nnc1O)NC1CCC(c2ccccc2C2CC2)C1 42922,c1(CC)cc(C(=O)NCC2CC(CNC(=O)C(N)=O)CO2)on1 42923,C(=O)(C(C#N)C(C)(C)C)N1C(C(C)NC(=O)CCCn2ccnc2)C2CCC1C2 42924,C(=O)(C1=CS(=O)CCC1)NCC1(F)CCC(NC(C(CC)(C)C)=O)C1 42925,N1(C(c2cc(C)sc2)=O)CC(NC(C2(Cc3cnn[nH]3)CCC2)=O)C(C)C1 42926,c1(CC)ccc(Br)cc1NC(=O)C(N1CCC(O)CC1C(F)F)CC1CC1(Cl)Cl 42927,C(C)(C(=O)NC1CC(NC(=O)CCc2nc[nH]n2)C1)=CC 42928,N1(C(C2C(C)(Br)C2)=O)C(CNC(=O)Cn2cnnn2)CC2COCC12 42929,C1(NC(CC2(COC)CCCC2)=O)CCC(C)(C)CC1CNC(=O)C=CBr 42930,c1(OC)cc(C=CC(=O)NCc2ccc(CNC(C3CCNC3=O)=O)cc2)sn1 42931,Cc1ccncc1C(=O)NCCC1CCC(NC(c2c(C)coc2C2CC2)=O)C1 42932,c1(C(N2CCCC(NC(C(C3CCC3)OC)=O)C2C)=O)ccc(C)cc1[N+](=O)[O-] 42933,C(C(=O)NCC(C)(CO)NC(C1CN(C2CCC2)C1)=O)(C(C)C)OC(C)C 42934,c1(CN(C(CCC)C(N)=O)C=O)ccc2c(c1)OC(C)(C)O2 42935,C(=O)(C(C)(C)C(C)O)N(CCCCC(=O)NCc1cc(CC)[nH]n1)C 42936,c1(CC(N2CC(CC(=O)OC)(SC)C2)=O)cccc(OC)c1 42937,c1(C(N(C)CC2OCCN(C)C2)=O)cnn2c1NCCC2 42938,c1(OC)cc(C)ncc1NC(c1cccc(CN2CCN(C)CC2)c1)=O 42939,c1(CNC(=O)NCC2CCN(C(=O)OC)CC2)ccc2cccnc2c1 42940,CC1CC(NC(=O)CNc2cccnc2)CN1C(=O)CCCF 42941,CC1Cn2nc(C(=O)N(C(C)(C)C)C)cc2CN1C(=O)NC1CC1 42942,C#CC1CN(C(=O)C(C(C)OC)NC(=O)C(O)CN2CCCC2)CCO1 42943,N1(C(C(C)Cn2ccnc2)=O)CC(NC(c2cncc(F)c2)=O)CC12CCCC2 42944,C1(NC(c2ccc(C)nc2)=O)CC2(CCC(NC(C3C(C)CC3C)=O)CC2)C1 42945,N1(C(CC(C)OC)=O)CCCC(C)(NC(c2ccc(O)cc2C(F)(F)F)=O)C1 42946,N1(C(Cc2c(C)nsc2)=O)CC=CC(C(=O)NC2CCCCC2CCO)C1 42947,Cc1ccc(O)c(CNC(=O)CC=CCNC(c2cn(C)cn2)=O)n1 42948,Cc1c(CC(=O)NCC2(C)CCCN(C(=O)C=CS(C)=O)C2)oc2ccccc12 42949,N1(C(CC2CN(C(C(C)NC(C)=O)=O)C(C)(C)C2)=O)CC2(C1)CC(C)(C)C2 42950,CC1(C(=O)NCCCCNC(=O)Cc2ccc(O)cc2Cl)CCC12CCC2 42951,Cc1ccc(CC(=O)NC2CC(CNC(=O)C(C)CN(C)C)C(O)C2)c(Cl)n1 42952,C=CCC(CC=C)C(=O)N1CC(O)CC1(C)C(=O)N(C1CCCCCC1O)C 42953,Cc1cnc(C(=O)NC(c2ccccc2)CNC(=O)CN2CCC(C)C2)cn1 42954,c1(OCC)nc(C)ccc1C(=O)NCC(O)CNC(=O)CCc1ccnc(C)n1 42955,c1(C(=O)NC(C)CN(C(=O)C=CCF)C)ncccc1Br 42956,C1(C(N2C(C)C(NC(c3ccc(CC#N)cc3)=O)CC2)=O)CCCC(F)(F)C1 42957,c1(C(C(=O)N(C2CN(C(C3CCCN3C)=O)C2)C)OC)ccc(F)cc1 42958,c1(CC(=O)NCC(C2CC2)NC(C2CNC(=O)C2)=O)cnccc1O 42959,CCCCC(O)C(=O)N1CC(NC(=O)CCCCCC)C(c2cccc(F)c2)C1 42960,C1(OC)CC(NC(C2CCCC2(F)F)=O)CN(C(=O)CCn2c(C)ccc2C)C1 42961,C1(C(C)C)CN(C(=O)C(O)C(F)(F)F)CCN1C(=O)CC=CCc1ccccc1 42962,c1(C(C)C)cnc(O)c(C(=O)NC2CCN(C(C3CC(C)(C)CO3)=O)C2)c1 42963,C1(NC(CCN(C)C)=O)CC(F)CN(C(c2ccc(O)cn2)=O)C1 42964,N1(C(C(CCC)N(C)C)=O)CCCC2(NC(c3ccoc3Cl)=O)CC2C1 42965,c1(NC(CC2(C)CN(C(=O)CC#N)C2)=O)cccc(Nc2cc(O)n[nH]2)c1 42966,C(C(=O)N=S(C)(=O)N(C)C)NC(=O)NCC(CC)(C)OC 42967,c1(OC)cc(N2CCOCC2)ccc1C(F)F.S1(=O)(=O)CCNC(=O)C=CC(=O)N1 42968,C1(C(C)C(=O)NCCNS(N)(=O)=O)CCN(C(C2CCN(C)CC2)=O)CC1 42969,N1(C(CCCCSC)=O)CC(C)C(C)(CNC(=O)C(C2CC(F)(F)C2)OC)C1 42970,C#CC1CC2(CC2)CN1C(=O)CCC(C)NC(C1(C#N)CCC1)=O 42971,c1(OC)ccc(CC(N)C(=O)NCCO)c(OC)c1.c12cccc(c1)OC2 42972,N1(C(C2CCN(C(C(=O)NCC)=O)C(C)C2)=O)CC(C#N)C2(CCC2)C1 42973,N1(C(CC(C=C)C)=O)CCCN(C(=O)Cc2ccc(Cl)c(Cl)c2)C(CO)C1 42974,c1(OC)ccc(F)c(CN2CC(NC(C3C4COCC34)=O)C(F)C2)c1Br 42975,C1(C(=O)NC(C=CC(=O)NC(C(C)F)C)C)OCC2CCCC12 42976,C1(c2noc(CC(=O)OC(C)(C)C)n2)(NC(C)=O)CCC(C)CC1 42977,N1(C(C(C)(C)OC)=O)C2CCC1C(CNC(c1nccnc1C(N)=O)=O)C2 42978,CC1=C(C(=O)NC2CCCC2C(=O)Nc2ccc(Br)nc2)CCO1 42979,c1(CNc2c(C)nc(-c3c(OC)cccc3)s2)c(C)nn(C)c1C 42980,c1(NC(C2N(Cc3cnc(C(C)C)[nH]3)CC(F)C2)=O)nc(Br)c(Br)cc1Br 42981,C1(CNC(Cn2c(C)c(Cl)cn2)=O)CN(C(=O)C=C2CCC2)C(C)(C)C1 42982,C(=O)(CC(C=C)CC)NCC(C(=O)N(CC#C)C)CC1CCCC1 42983,c1(CC(N2CCC(O)(CN(C(C(C)n3cncn3)=O)C)C2)=O)c(O)ncnc1O 42984,C1(OC)CC2CC(C(=O)NCCCC(C)(C)NC(=O)Cc3ccco3)CC12 42985,C1(NC(=O)CCC=CBr)C2CCC1N(C(c1ccc(CF)cc1)=O)C2 42986,c1(C(N(C)CC2CCN(C(c3ccc(F)cc3N)=O)C2)=O)cnc2[nH]ccc2n1 42987,C1(CC(N2CC(O)(CNC(C(CN(C)C)N(C)C)=O)C2)=O)COCC2(CCC2)O1 42988,CCCCC(O)C(=O)NCCC(C)NC(=O)CC(F)(F)c1ccccc1 42989,N1(C(C=C(COC)C)=O)CC(O)(C(C)NC(C2(c3ccccc3)CC(C)C2)=O)C1 42990,c1(CNC(c2n(CC=C)nnn2)c2ncc(Cl)s2)cc(Br)cc(Cl)c1F 42991,C(=O)(C1=CCCCC1C)N1CCC2C(C(=O)NC(COC)C(C)C)C2C1 42992,N1(C(C(C)=O)=O)CCOCC(NC(C2(C(F)F)CCCO2)=O)C1 42993,C1(NC(C(C)O)=O)COC2(C1)CN(C(=O)Cc1cc(Cl)sc1Cl)C2 42994,c1(C(=O)NCC2CC(NC(C(C)C3CCCO3)=O)C2)cc(F)c(N)c(F)c1 42995,N(C1CS(=O)(=O)Cc2ccccc21)C(NC1CCc2c(Cl)nccc21)=O 42996,C1(NC(CSCC=C)=O)CC2CC(NC(C3CCC4CC34)=O)C1C2 42997,C1(P(C)(C)=O)(C(=O)OCc2cnc(C)s2)CC1 42998,C1(CNC(C2(OC)CCCC2)=O)CC2(CC2)CN1C(c1cc[nH]c1)=O 42999,C(C)(CN=c1nc2ncccc2c[nH]1)NC(Cc1c(C)nc(C)s1)=O 43000,C(C(O)CO)N(CCCO)N(CC(C)CC)C(C)=O 43001,C1(NC(C(CC)C)=O)CCN(C(C2COCCN2Cc2ccccn2)=O)C1(C)C 43002,CC(C)CC(C(=O)N1CCCC(NC(=O)CN(C)C(c2ccccc2)=O)C1)N(C)C 43003,C1(NC(CCCOCC)=O)CC2CC(C1)N(C(=O)CCNS(=O)(=O)C(F)(F)F)C2 43004,C1(C(C)NC(=O)CN(C)CCO)CCCN(C(=O)CCCn2cccn2)C1 43005,C12(CC=CCC1)C(=O)N2.O=C(C(=O)NCC(F)(F)F)NCCCOCCCl 43006,Cc1ncc(C(=O)NC2CC(OCC(=O)N(CC(C)(C)C)C(C)C)C2)c(=N)[nH]1 43007,Cc1noc(C)c1CSCC(=O)N(C1CCCN(C(c2cc[nH]n2)=O)C1)C 43008,c1ccc(C2CC(NCC3(C4CCCO4)CNC3)C2)cc1 43009,CC1CC(C(N2CC(O)(CNC(=O)CSCC(F)F)C2)=O)CN1C 43010,c1(NC(C)=O)ncc(S(=O)(=O)N2CCCC(N3CCCCC3)C2)s1 43011,Cc1ccc(SCCC(=O)NCC2(F)CCC(CNC(C3CC3(C)C)=O)C2)cc1 43012,c1(C(=O)NCCC2CC(C(=O)NCCC3CCC4CC34)C2)ccccc1Cl 43013,C1(NC(c2n(C)nnn2)(C)CCBr)CC2(CCCC2)C1 43014,C(C(CC(C)C)C(=O)NC12CC1CN(C(c1ccnc(C3CCC3)c1)=O)C2)OC 43015,CC1(C)CCCC(O)(C(N2CC(NC(=O)C(C)(C)F)C(CC(F)F)C2)=O)CC1 43016,C1(C(=O)N(C2CC3CCC(C2)N3C(=O)C(O)C2CC2)C)(OC)CCC(F)(F)CC1 43017,C(C(CC(C)C)NC(=O)Cc1ccc(F)cn1)NC(C1CC(C)(CC)C1)=O 43018,C(C)(CC(C)NC(c1sccc1COC)=O)NC(COC(C)C)=O 43019,N1(C(CC(CC(=O)OC)C)=O)CCN(C(C2CC(=O)N2)=O)CC(C)(F)C1 43020,CC1CCN(c2nnc(C(F)(F)F)s2)C(C)C1NC(C1CSC1)=O 43021,C1(NC(C(CC)O)=O)CCC12CCN(C(c1noc3cc(F)ccc13)=O)CC2 43022,c1(C(=O)NCCN(C(=O)C=CS(C)=O)C)cc2cc(F)ccc2o1 43023,c1(C(N2CC(NC(c3nccc(C)n3)=O)C3C2C3)=O)cc2cccnc2s1 43024,C(=O)(C(=O)C(C)(C)CC)NC(CC(N1CC(C)(OC)C1)=O)C1CC1 43025,C#Cc1cc(C(=O)NCCC(C)NC(C2(C)CCCS2(=O)=O)=O)ccc1C 43026,c1(C(N2CCC3(CC3C(N3CCC(O)CC3)=O)C2)=O)cc(Cl)cc(Cl)c1O 43027,CCCC(CC)CC(=O)NCc1cccc(NC(c2c(N)cc(F)cc2F)=O)c1 43028,C1(NC(c2c(C)ccnn2)=O)COC2C(NC(=O)CCCC(F)F)COC12 43029,c1(C(N2CCCC(CNC(C=NOC)=O)CC2)=O)cc(C)nc2c1c(C)nn2C 43030,c1(NC(C23CC2CN(Cc2ccc(O)c(F)c2)C3)=O)nc(Cl)cc(Cl)c1[N+](=O)[O-] 43031,Cc1cc(S(N)(=O)=O)sc1C(N1C(CNC(C2CC(F)C2)=O)CC2CC12)=O 43032,N1(C(CC#N)=O)CCC(c2ccccc2)(NC(c2cccc(C3CC3)c2)=O)CC1 43033,Cc1nc(C(N2CC3(NC(c4ncoc4C)=O)CC2C3)=O)n(C)n1 43034,N1(CCC=C)CCC2(CC1)CC2C(N(CC)Cc1ccc(C(=O)OC)nc1)=O 43035,C123CCOCC1CN(C2)C3=O.CC(CC(F)F)C(=O)Nc1cnc(N(C)C)nc1 43036,C1(CNC2CC(C)S(=O)(=O)CC2)CCc2n[nH]cc2C1 43037,c1(CC(=O)NC2C(CNC(C(CC)F)=O)C2)ccc(Cl)cc1Cl 43038,Cc1ccc2cc(CNC3CCCCN(C(=O)C(C)(C)F)C3)ccc2n1 43039,C1(NC(C(C(=O)OC)C)=O)CN(Cc2cc(C)ccc2Cl)CCC1(F)F 43040,c1(C(=O)NC(C2CCN(C(C3CC4CC3CC4O)=O)C2)C)ccc(C#N)cc1F 43041,c1(C(=O)OC(C)(C)C)cc(NC(=O)NCCCC(N)=S)c(Br)cc1F 43042,C12(C(N3CC(OC)C(NC(=O)C(F)(F)C(C)O)C3)=O)CCCN1CCC2 43043,N1(C(c2n(CCC)ncc2)=O)CCC(C(=O)NCC(C)C)C1(C)C 43044,N1(C(C(CCC#C)O)=O)C(CNC(c2cnc(CC(C)C)[nH]2)=O)CC2CCCC12 43045,CCCCC(CNC(=O)C(C)NC(=O)COC)NC(c1cocc1C)=O 43046,CCCC(C#N)C(=O)NCC1OCCC1C(=O)NCC(C1CCCC1)OC 43047,c1(C(=O)NCC2N(C(CCP(C)C)=O)CCCC2)ccc(N)c(Cl)c1O 43048,CC(N=c1[nH]c(=NC2CCOC2)[nH]c2c1COCC2)c1cc(NC2CC2)n(C)n1 43049,C1(C(N2CCCC(OC)C2)=O)COCCN(C(C2CC2(C)C(F)F)=O)C1 43050,Cc1nc(N2CCOCC2)nc(O)c1CC(N1CCCC(O)(C(C)C)C1)=O 43051,N1(C(CCCC(=C)C)=O)CC2COCCC2(NC(C2CCOCC2(C)C)=O)C1 43052,Cc1cc(N)c(C(=O)NC2CC(N(C(=O)CC3CC4(CC4)CO3)C)C2)nc1C 43053,C1(C(C)CN(Cc2cccnc2)CC2CC2)CCC(C)(C)CC1 43054,CC(C)CC(C(=O)NC(C)CNC(c1ccncc1Cl)=O)N1CCCCC1=O 43055,c1(C(=O)NC2CC(OCC(=O)NC3C(C)CN(C)C3)C2)cccc(F)c1O 43056,c1(COCCN(C(C2CC(OC)C2)C(=O)Nc2ncn(C)n2)C)ccc(F)cc1 43057,C1(N(C(=O)CCc2ncco2)CC)CCCN(C(=O)CCC2CCCO2)CC1 43058,c1(CC)n[nH]c(CC)c1CC(N1CC(NC(C2CCO2)=O)C(C)C1)=O 43059,Cc1ccc(CC(N2CCN(C3CCN(C(C4CC(C)(F)C4)=O)C3)CC2)=O)cn1 43060,CC(C)S(=O)(=O)CC(=O)NC1CCCCCN(C(=O)CCc2cnoc2)C1 43061,C(=O)(C(C#N)CC1CC1)NCC(CCC)NC(=O)Cc1ncsc1Cl 43062,CCC(C(=O)O)(CCO)NC(c1ccc(COC(C)(C)C)cc1)C 43063,c1(C(=O)NC2C(CNC(c3cc(OC)ncc3)=O)CC2)noc2c1COCC2 43064,N1(C(CC(C)C)=O)CCC(N(C)C(c2cc(-c3cccnc3)[nH]n2)=O)C(C)C1 43065,N1(C(c2c(CC)c[nH]n2)=O)CCC2(NC(c3c(F)cccc3Br)=O)CC2C1 43066,C1(C(=O)NCc2cc(C)[nH]c2)CCC2(CN(C(=O)NCc3cccnc3)C2)O1 43067,C1(CC(=O)NC2CC(F)(F)CC2NC(C2SCCCS2)=O)CN2CCC1CC2 43068,N1(C(Cc2c(C)con2)=O)CC2(CCN(C(=O)C(C)(c3cccs3)N(C)C)C2)C1 43069,c1(C(N2C(CNC(C3(C(C)(F)F)CC3)=O)CCC(C)C2)=O)cnn2c1OCCC2 43070,c1(C(=O)NCC(C2CCCC2)NC(C2(C#C)CC2)=O)cnn2c1CC(F)(F)C2 43071,Cc1cccc(C(N2CCC(C(C)NC(=O)CSCCC(C)C)C2)=O)c1Cl 43072,N1(C(C)CNC(=O)NCCn2cccnc2=O)CCN(C)C(=O)C1 43073,N1(C(c2c(C)scn2)=O)CCC(OCCNC(=O)CC2CCS(=O)(=O)C2)CC1 43074,CC1=CCC(C(=O)NCCCN(C(=O)CC(C)NC(=O)OC(C)(C)C)C)CC1 43075,CCCC(O)C(CO)NC(C1(CSC)CCC1)=O.C12(CC1)N(C)C2=O 43076,N1(C(c2n(C)ncc2)=O)CC(C(N2CCCC3C(O)CC23)=O)CCC1(C)C 43077,C1(C(N2CC(NC(C3CC(C)OC3=O)=O)C2)=O)(CC)CC(C)(C)C1 43078,N1(C(COC)=O)CCC(CNC(C2CC3CCCCN3C2)=O)C(F)(F)CC1 43079,C(=O)(CC(O)CCCC)N(CCCCC(N1C(CC#C)CCCC1)=O)C(C)C 43080,Cc1cc(CCC(=O)NCCC(O)CNC(C2(C)CCN(C)C2=O)=O)cc(C)c1 43081,C#Cc1cncc(C(=O)NCCC2CC(F)(F)CN2C(c2nocc2Cl)=O)c1 43082,CC1CN(C(C2(c3ccon3)CC2)=O)CCN1C(=O)C(C)c1cc[nH]n1 43083,C(CC(C)CC)(C(=O)N1C2COCC1C2)NC(c1c(CCC)n[nH]c1)=O 43084,n1(CC(N2CCC(CNC(C(C(C)C)OC)=O)CC2C)=O)cc([N+](=O)[O-])nc1C 43085,N(C1CC2(CN(C(=O)OC(C)(C)C)C2)n2ccnc21)C(C#C)(C)C1(C(=O)O)CC1 43086,N1(C(c2c(N)nc(Br)cc2)=O)CCC2(C1)CN(C(c1ncncc1F)=O)C2 43087,N1(C(CC2(COC)CCCC2)=O)CCC(C)(C)C(NC(=O)C(C)OC)C1 43088,c1(CNC(C(C(C)C)F)=O)nnc2n1CCN(C(C1(C)CCOC1)=O)C2 43089,C1(NC(C2(CCCC)CCC2)=O)CN(C(C2CN(C)C2)=O)C2(CCOC2)C1 43090,C1(C(=O)NC(C)CCCCNC(c2cnc(C(C)(C)C)[nH]2)=O)CC2(CC2)CN1C 43091,CCC(C)(C)CCCC(=O)NCCN(c1nc(C)ncc1F)CC1CC1 43092,CC(C)(CC(=O)N1CCC(O)(CNC(=O)CCCC(F)(F)CO)C1)CC(F)(F)F 43093,c1(C(=O)NCC#CCNC(=O)CCc2cnccn2)cc(Cl)c2c(c1)OCO2 43094,C(=O)(C(F)(CNC(=O)C(C)=CC1CC1)C(C)C)N(C1CCCOC1)CCOC 43095,c1(C(N2CC(C)OC(C3CC3)C2)=O)cc(Br)cc(F)c1N 43096,N1(C(Cc2cc(C)[nH]n2)=O)CC(C)(C(=O)N(CC2=CCSC2)C)CC1(C)C 43097,C(=O)(CC(C)(C)C(F)F)N(CC(C)(C)CNC(=O)Cc1ccon1)C 43098,N1(C(C(CCOC)OC)=O)CCN(C(c2ccc(C)c(O)c2)=O)CC12CCC2 43099,c1(CCNC(C(=CC2CCC(C)CC2)C)=O)cnn2ccccc12 43100,C1(CC(N2C(CN(C(c3ccon3)=O)CC)CCC2)=O)COCC(C)(C)O1 43101,N1(CC(C(=O)CC(C)(C)C)=O)CCC(F)(F)C(CNCC(C)O)C1 43102,N1(C(c2c(C)cnn2C)=O)CC(C)N(C(c2cc(C#N)c[nH]2)=O)C(C)C1 43103,O(NC(=O)C(CNC(C1CC2CCC(C1)O2)=O)CC(C)C)CC(CC)C 43104,N1(C(CC(C)SC)=O)CCC(C)(NC(=O)C(C2(O)CCCCC2)(F)F)CC1 43105,C1(NC(CCCCSC)=O)CCC2(CC1)CC2NC(=O)C(=O)N(C)C 43106,CC1CCN(C(c2cccc(SC(F)(F)F)n2)=O)CC1NC(=O)CC1CN(C)C1 43107,N12CCC(C13CCC3)C2=O.N=c1[nH]cc(C(=O)NCC2CN(CC(F)F)C2)s1 43108,C1(C(C(=O)NCCOC)NC(C)(C)C)CC(C2CC2)C1.C12(CC=CC1)C(=O)OC2 43109,C(=O)(C(CCSC)NC(=O)CCc1nncs1)N1CCC(C(CC)CC)C1 43110,c1(CC(=O)NCCC(C)NC(=O)C=CC(C)(C)C)ccn2ncnc2c1 43111,CC1CN(C(=O)CC2CC3CCC2O3)CCC1CNC(C1(O)CCCCCC1)=O 43112,c1(C(C(=O)NC2(C)CC2)N(C(c2ccccc2)C(=O)OC)C)c(SC)cccc1F 43113,C12(NC(=O)Cc3cc(Cl)cs3)CN(C(c3cnc[nH]3)=O)CC1CS(=O)(=O)C2 43114,c1(C(N2CCC3CN(C(C4ON=C(C)C4)=O)C3C2)=O)cnc2sc(C)cn2c1=O 43115,c1(CC(N2C(CNC(CC(C)O)=O)CN(C)CC2)=O)cc(F)c(F)cc1F 43116,C1(NC(C=NOC)=O)CC2CC1CN(C(c1ccc(C(F)(F)F)cc1)=O)C2 43117,C1(N(C)C(C2(C(N)=O)CCC2)=O)CCC(NC(c2c[nH]nc2C2CCCO2)=O)C1 43118,c1(CNCC2CCC(C)(C)O2)ccc(Br)nc1F 43119,C1(C(=O)Nn2cc(C#N)cn2)Cc2c([nH]c3ccccc23)CN1CC.C1(=O)CN1 43120,c1(C(=O)Oc2ccc(NC(C(C)OC)=O)cc2)cc(F)ccc1NC(=O)C(C)(C)C 43121,c1(SCC(=O)NC2COCCN(C(CC(=O)OC)=O)C2)ccc2c(c1)CCC2 43122,N1(C(CC(=O)N(C)C)=O)CCN(C2CCCN(C(=O)CCC(C)(F)F)C2)C(=O)C1 43123,N12CCCN(CC1)C(c1cscn1)C2=O.CCC(CC=O)C1CCC1.CCO 43124,C1(C(=O)NCC(c2cccc(Cl)c2)NC(c2nnc(C)s2)=O)CN(C)CCO1 43125,N1(C(=O)Cc2cc(-c3ccccc3)on2)CC(CNC(c2cncs2)=O)C2CC12 43126,N1(C(C2(COC3CCC3)CCCCC2)=O)CCCCC(n2cc(C)nn2)C1.CCS 43127,c1(C(=O)NCCN(C(C2C(C(=O)OC)C2)=O)C)nnn2c1CSCC2 43128,C(CCCCC(=O)NC(C)CCC(=O)NCCc1ccncc1)=CC 43129,C(C)(CCCN=c1nc(N2CCNC(=O)CC2)c2ncccc2[nH]1)OC 43130,C=CC(C)C(C)C(=O)NCC1(NC(=O)CC2CN(C)C2)CCCC1 43131,c1(C(c2n(CCCC)nnn2)NC2(CCF)CC2)cc(Br)cc2c1OCC2 43132,CC1CN(C(c2ccc(CO)o2)=O)CCCN1C(C1(C(F)F)CCCC1)=O 43133,c1(C(N2C3CC(NC(c4nc(C)n(C)n4)=O)C(C3)C2)=O)nnc2n1CCCCC2 43134,C#Cc1cc(C(=O)NC2C3CC(NC(C4CCC(OC)C4)=O)CC23)ccc1C 43135,c1(C(N2CCC(NC(C3(CC)CCC3)=O)C2)=O)ccccc1NCc1ccsc1 43136,C(=O)(N=c1cc[nH]cc1-n1ccnc1)C1CCC2(CN(C(C(CCC)O)=O)C2)O1 43137,c1(OC(C)C)cnc(NC(C)(C)CN2CCN(C(C3CC(C)C3)=O)CC2)nc1 43138,N1(C(c2n(CC#C)ccc2)=O)CC(NC(=O)C(C)c2cc[nH]n2)CCC1C 43139,C(c1c(Br)c(Br)cc2c1OCC2)=CN1CCCC(CO)C1.C(=O)(C=C)OCC 43140,c1(C(=O)NCC(CN(C)C(c2ccc(N)c(F)c2)=O)(C)C)nn(C)c2c1CCC2 43141,Cc1oc(C(=O)NC2CN(C(C3C(C)C3(F)F)=O)CC2O)cc1S(N)(=O)=O 43142,CC(C)C(C)C(C)CC(=O)NCC12CC(NC(c3cnn(CC(F)F)c3)=O)(C1)C2 43143,c1(N2CC(C)S(=O)CC2)ccc(S(=O)(=O)NCCc2cnoc2)cc1Cl 43144,CC(C)CC(O)C(C)C(=O)NCc1ccc2ccccc2c1 43145,N1(C(C2C(CC)OCC2)=O)CCC(CCNC(C2(OC(C)=O)CCCC2)=O)CC1 43146,c1(CC)cccnc1C(=O)NCC1(O)CCN(C(=O)C(CSC)OC)C1 43147,c1(COC(c2nccc(C)c2O)=O)cccc(C#N)c1Br 43148,O=S(=O)(c1c[nH]ccc1=NCC1(Br)CC1)NC1CCCCC2(C1)OCCO2 43149,c1(-n2cc(CCN3C(C(C)O)CCC3)nn2)nnc(O)nc1O 43150,c1(OCC)cc(C(=O)N(CCC(N2CCC2C=C)=O)C2CC2)sn1 43151,C(CNC(=O)CCc1nnc(S)n1C)(CC(F)(F)F)NC(C(C)SCC)=O 43152,c1(CNC2CCC(C(=O)Nc3cc(OC)n[nH]3)C2)c(F)cc(Br)c(F)c1F 43153,CCCS(=O)(=O)C(C)C(=O)NCc1cc2ccccc2s1 43154,c1(C(=O)NC2C(NC(C3ON=C(C)C3)=O)CCC2)c(C)nn2c1CCCC2 43155,c1(OC)ccc(C(=O)NCCN(C)C(C2CC3CC23)=O)c(C(F)(F)F)c1 43156,CCCN(OC)C(=O)CC1CCN(C(C2C3CC4C(C3)C24)=O)C1 43157,C1(OC)CN(C(c2ccc(NC(=O)Cc3cccs3)cc2)=O)CC1OCC1CC1 43158,N1(C(c2c(OC)ncc(C)c2)=O)CCc2cc(-c3ccccc3OC)ccc2C1 43159,C1(C(=O)NC(C2CCN(C(=O)CCc3cccnc3)CC2)C)CCCCC(=O)C1 43160,c1(C(=O)NCC(CNC(C=CC(=O)NC2CC2)=O)F)ncoc1C1CCCO1 43161,C1(C(N(C)Cc2cn[nH]c2)=O)CCC(n2cc(C3(O)CCC3)nn2)C1 43162,CCCC(C)CC(=O)N(C)CCOCCCN(C(=O)CC=C(Cl)Cl)C 43163,CC1CC(NC(c2ccc(Cl)nc2O)=O)c2nccn21 43164,N1(C(CC2N(C(C3=CC(C)(C)C3)=O)CC(O)C2)=O)CCCC2(CCC2)C1 43165,CC(C)C(C(C)NC(C1C2CCC1CC2)=O)NC(C1CC2(CSC2)C1)=O 43166,C12(CNC(C3C(C)(C)C3)=O)CCC1CN(C(=O)Cn1nnnc1C1CC1)C2 43167,C(=O)(C(F)C(C)C(F)(F)F)N1CC(C(C)NC(C2(C#C)CC2)=O)OCC1 43168,Cc1cncc(C(=O)NC2CC(NC(c3cn(C4CC4)cn3)=O)C2)c1 43169,c1(C(=O)NC2CCCCC2CNC(C2CC=CC2)=O)cc(C(F)F)cc(Br)c1 43170,c1(C(=O)NC(CN(C)C)C(=O)NCC#CC(F)(F)F)ccc(C#N)n1C 43171,C1(NC(C(C2CCCC2)OC)=O)C=CCN(C(c2cc(C)c(C)s2)=O)C1 43172,Cc1ncc(C(=O)N(CCCNC(=O)Cn2ncc(Br)c2C)C)c(C2CC2)n1 43173,c1(C(=O)NCC2N(C(C(CCOC)OC)=O)CC(OC)C2)scc2c1CCCC2 43174,C(C(C)(C)Cc1ccccc1)CN(C(C(=O)OCC)=O)CCOCCO 43175,C1(C(=O)NCC#CCCO)(CC)CCN(C(=O)C(C2(O)CCCC2)F)CC1 43176,C1(NC(c2c(CC)ncnc2)=O)CN(C(=O)Cc2cccc(F)c2)C2CCCC12 43177,C1(c2n(CCSC)nnn2)(NCC2CC2(C)C)CCOCCC1C 43178,N=c1[nH]c(=NCC2CCC3CC23)[nH]c(=NCCN2CCCc3ccccc3C2)[nH]1 43179,c1(C(=O)NC(CN(C(=O)C(Cl)=CCl)C)(C)C)cc(N)c(Cl)cn1 43180,C1(CN(C2CC(C)CCO2)CC)CCCN(C(=O)CCCc2cnccn2)C1 43181,CC1CC(O)CCN(C(=O)CC(C2CC2)NC(c2cnn[nH]2)=O)C1 43182,C1(C(=O)Nc2cnn(CC)c2C)CC(C)(C)CN1C(=O)CC(C)COC 43183,c1(C(=O)NCc2cscn2)cc(OCC2CC2)ccc1F 43184,C1(CCCC)CCCCN1N1CCC(C(F)(F)F)(C(=O)OCOC)CC1 43185,N1(C(c2c(CNC(C(N3CCNC3=O)C)=O)nnn2C)=O)CCC12CC(C)(CO)C2 43186,c1(C(=O)Nc2c(C#N)ncc(Br)c2)ccc2cccc(-c3cnoc3)c2n1 43187,C1(C(=O)NC(C)CO)(NC(CNC(CC(C)C)=O)=O)CCN(C)C1 43188,N(C(=NCCOCc1ccc(Br)cc1)NC1CCOCC1)C1CCC(CO)C1 43189,c1(C(N2C(CCNC(c3ccc(C)s3)=O)CC(OC)C2)=O)cccn2cnnc12 43190,c1(C(=O)NCC2(CNC3(C(CC)=O)CC3)CN(C(C)=O)C2)ccc(=O)n(CC)n1 43191,C(=O)(CC(C)C(F)(F)F)NCCCC(C)NC(C(C(C)C)C)=O 43192,C1(NC(C(C)OCC)=O)CS(=O)(=O)C12CCN(C(c1cc(Cl)nc(=N)[nH]1)=O)CC2 43193,FCCCN=C(NCC1(c2ccc(F)cc2)CCC1)NC1CC1C(F)(F)F 43194,C(=O)(CCC(=O)N1CC=CC1CNC(=O)C(O)CC1CCCC1)OC 43195,C1(C(=O)NCCOCCNC(=O)C(C)n2cnnn2)(OCC)CCOC1 43196,N1(C(CC(C)c2ccccc2)=O)CCN(C(=O)COCCOCCO)C2CCC12 43197,c1(C(N2CCC2Cn2cc(CC3CCOCC3)nn2)=O)cc2n(c1)CCCC2 43198,c1(CN2C3(c4nnc(C)o4)CCC3CC2)nc2ccc(C)cc2s1 43199,C1(C(N(C(C)CNC(c2ccccc2SC)=O)CC)=O)NC(=O)OC1C 43200,N1(C(c2occ(C)c2)=O)CCC2(CC1)C(NC(C1(C3CCC3)CC1)=O)CS2(=O)=O 43201,Cc1cc(C(=O)NC2CC2NC(=O)C(C2CCCCC2)C)cnc1C 43202,c1(SC(C)C(N2CC=CC2CNC(C2CCCN2C)=O)=O)ccc(F)c(F)c1 43203,Cc1cc(C)c(C(=O)N(CCCNC(=O)C=C2CCSCC2)C)c(=O)o1 43204,c1(CNC(C2N(S(C)(=O)=O)CC2)=O)cnn2c1CN(C(C1CC1C(N)=O)=O)CC2 43205,c1(CC(C(=O)NC2C(NC(c3ccncc3O)=O)CC2)O)cccc(Cl)c1 43206,N1(C(C(N2C(CC)CCC2)=O)=O)CCOCC1CNC(=O)Cn1nc(C)cc1C 43207,c1(C(N2CC(NC(C(C)=C(CC)C)=O)C(C3CC3)C2)=O)cccc([N+](=O)[O-])c1Cl 43208,N1(C(C(n2cc(-c3ccc(N)cc3Cl)nn2)C)=O)CCc2cnccc2C1 43209,c1(C(=O)Nc2c(C(=O)NC(CC=C)C(=O)O)nccc2)c(F)ccc(Cl)c1F 43210,C(CS(=O)(=O)CC(=O)N1CC2(CC(NC(=O)CCCCC(C)C)C2)C1)OC 43211,c1(C(N2C(CN(C)C(C3CCS(=O)(=O)CC3)=O)CCC2)=O)ccc2ocnc2c1 43212,N1(C(CC=C)=O)Cc2[nH]nc(C(=O)NCC(COC)C(C)C)c2C1 43213,N1(C(c2c(C)n[nH]c2C)=O)CCCC1C1CCCN1C(c1csc(C#N)c1)=O 43214,Cc1c(NC(=O)CN(c2ccc(C#N)cn2)C)cc(F)cc1[N+](=O)[O-] 43215,N1(C(c2c(CC)csc2)=O)CCC2(CCN(C(=O)COC)C2)C1 43216,C(=O)(C(C)(C)CC(C)(C)C)NC1CC(C)N(C(C2CCSC(C)C2)=O)C1 43217,Cc1cc(C(=O)NC2C3CC2CN(C(=O)C(C)C(C)C)C3)c(Br)c(C)c1 43218,c1(C(N2CC(CC)N(C(=O)C(O)CC(F)F)CC2)=O)ccc2ocnc2n1 43219,CC(C)CC(C)(O)C(=O)N(C1CCCC1)CCCNC(=O)C(C)N(C)C 43220,C1(C(=O)NCCN(C(C2(C(F)(F)F)CCN(C)C2)=O)CC)CNC(=O)CC1(C)C 43221,c1(NC(C(CCN(C)C)NC(=O)C(O)C2CC2)=O)ccc2nccn2c1 43222,C1(CC)CN(C(c2nccn2C)=O)CCN1Cc1ccc(SC)cc1 43223,C1(NC(=NC)NCCCc2ccco2)CCOC2(CCCC2)C1 43224,C(CCC(C)(C)C(=O)NCc1nonc1C)NC(C(=Cc1ccco1)C)=O 43225,C=CCC(CC(=O)Nc1cnc(Cl)cc1C)NC(=O)CCC1OCCO1 43226,c1(C(N2C(CN(C(=O)CC#N)C)CCC2)=O)cnn2c1CCC2 43227,N1(C(CC(C)(C)O)=O)CCCC2CN(C(=O)CC3CCC(=O)CC3)CC12 43228,C1(C(N2CC3C(C(=O)NC(CC(=O)NC)C)C3C2)=O)CC(=O)NC(C)C1 43229,C#CCC(CC(=O)NC(c1nnc(C)o1)C)NC(C1CCCN1C(C)=O)=O 43230,c1(C(=O)NCCCC(C)(C)NC(CC2N(C)CCOC2)=O)cn(C)ccc1=O 43231,C(C(C)C(C)C(=O)NCCN(C(c1ccnc(C(F)(F)F)c1)=O)CC1CC1)OC 43232,c1(C(=O)NCC(C)CNC(c2ccc(C#N)s2)=O)n[nH]c2ccccc12 43233,N1(C(c2ccc(C(=O)OC)o2)=O)CCCC1(C)CNC(=O)Cc1n[nH]c(C)n1 43234,C(=O)(NN1CCCC1C(=O)NCC(C)(CO)OC)c1cc(CC)nn1C 43235,Cc1sc(Cl)nc1C(N1CC(NC(c2cc(C(N)=O)c[nH]2)=O)CC1C)=O 43236,C1(C(=O)NCC(=O)NCC#C)N(C(=O)C(C)NS(C)(=O)=O)CCC1(C)C 43237,Cc1ncnc(C)c1NC(C1CCCCN(C(C2C3CCC(F)C23)=O)C1)=O 43238,N1(C(C(C)CS(C)(=O)=O)=O)CCN(C(=O)CNC(n2cncn2)=O)C2(CCC2)C1 43239,N1(C(C=C(CC)CC)=O)CCC(O)(CCNC(c2csc(Cl)n2)=O)CC1 43240,c1(C(=O)NC(C2(O)CN(C(C3(O)COC3)=O)C2)C)ccc(F)cn1 43241,c1(C2C(=O)N2)ccc(OC(F)(F)F)cc1.N1(CC=C)CCC1C1CCC1 43242,CCCC(CCC)C(=O)NCC(C1CCOC1)NC(c1ccc2cncn2c1)=O 43243,c1(C(N2CCC(NC(C3(C)CCC(C)CC3)=O)C(O)C2)=O)c(F)cc(Cl)cc1F 43244,c1(C(=O)NC2CN(C(c3c(OCCC)cccc3)=O)CC2O)cc(Cl)ccc1Cl 43245,c1(C(C)=O)cc(CC(=O)N(C2CCN(C(=O)C(n3cc(Cl)cn3)C)C2)C)cs1 43246,C1(C(N2C(CC=C)CCCC2)=O)CN(C(=O)CC(C)C2CC2)CCN1C 43247,c1(CC(N2CCN(C(CC3(C=C)CC3)=O)CC2)=O)ccc(S(N)(=O)=O)s1.C1CC1Cl 43248,C1(O)(CCNC(c2cc(C)n(C)c2)=O)CCCN(C(=O)C2=CCC2)C1 43249,N1(C(CC(C(C)C)OCC)=O)CCN(C(c2c(C)cccc2Cl)=O)CC(C)(C)C1 43250,C(=O)(CCC(C)(F)F)NCC(C)C(=O)NCCN1CC(C)(O)C1 43251,N1(C(C(C=C)(C)CC)=O)CC(C2CN(C(c3[nH]c(=N)ccc3C)=O)C2)C1 43252,c1(N2C3C(NC(=O)CC4CCOC4)(CCC3)CC2)ncnc2[nH]ccc12 43253,N1(C(Cn2ncc(C)c2)=O)CCCCC1c1cn(CC(N2CCC2CO)=O)nn1 43254,C(CC)(CCCC(=O)NCc1cc(C#N)cs1)NC(C1(CC#C)CC1)=O 43255,C(CCC(N)=O)(C(=O)NCCCN=S(C)(C)=O)n1cc(CCCC(C)C)nn1 43256,CCCCC(CC)C(=O)NCC(c1ccc(F)cc1)NC(C1(C)CCC1)=O 43257,C1(C)(CNC(CCN(CC=C)C(c2cc(N)cc(F)c2)=O)=O)CCCCC1O 43258,C(CCC(C)C(=O)NCC1(F)CCN(C(C2(C)CC3CCC2O3)=O)CC1)OC 43259,C(=O)(C1Cc2ccccc21)N1CCCC(CCCCNC(c2occ(C)c2)=O)C1 43260,c1(C(N2CC(CNC(C3CC3F)=O)CC23CCC3)=O)cc2cc(F)ccc2s1 43261,c1(CN(C2CN(C(=O)Cc3n[nH]cc3Br)C2)C)csc(Cl)n1 43262,Cc1nc(N2CCC(C)C2CNC(C2COCCN2CC(F)F)=O)[nH]c(=N)n1 43263,c1(C(=O)OCC)cccc(-c2cn(CC(=O)NC(CCSC)C(=O)O)nn2)c1 43264,C1(C(=O)NCC2CCN(C(c3c[nH]c(=NC)o3)=O)C2)CCN(C2CC2)S1(=O)=O 43265,c1(C(N2CCC(C)C(NC(C3(C)CC(C#N)C3)=O)C2)=O)ccc(Cl)c2occc12 43266,C(=O)(C1=CCCC(C)(C)C1)NC(CNC(CCSCC(=O)OC)=O)(C)C1CCC1 43267,c1(C(CNC(CNC(CCOCCC)=O)=O)O)ccc(F)cc1 43268,C1(N(CCC)C(C2CC2OC(C)(C)C)=O)CCN(C(c2cc(O)n(C)n2)=O)CC1 43269,c1(OCC)cccc(CNC(=O)NCc2c(-c3ccccc3)coc2C)c1CC 43270,N1(C(C2(CC)CCCO2)=O)CCCC(N(C(=O)CCC2OCCO2)CCF)C1 43271,C(=O)(C(C)C(O)CC(C)C)NCCC1(CNC(c2c(C)cc(CC)o2)=O)CC1 43272,C(C)(C)(CC(=O)NCC(O)CC(=O)NCC(N1CCCC1)C)OC 43273,N1(C(c2c(CC)occ2)=O)CC(C(N2CCC3C(OC)CC23)=O)C(F)(F)C1 43274,C(C(C)(C)C(=O)NCCC1CN(C(=O)C(C)Cn2ccnc2)C1)OC 43275,c1(OC)ccc(CC(=O)CN2CCN(C3CC(O)C3)CC2)cc1 43276,C1(CNC(c2cc(-c3ccc(C)s3)[nH]n2)=O)CCC(C)CN1C(=O)C(C)C 43277,Cc1cc(O)cc(C)c1CC(=O)NCC1(O)CC(NC(c2cc(CO)[nH]n2)=O)C1 43278,c1(CC(=O)NC2CN(C(C(COC)C)=O)C2)ccc(N2CCOCC2)cc1 43279,Cc1ccc(C(N2CCCCC2C(C)NC(=O)C(C)(C)C(N)=O)=O)c(O)n1 43280,c1(C(N2CCC(C(=O)NCC=C3CCSCC3)(OC)C2)=O)cc(C#N)oc1C 43281,C1(C(=O)NCCOCCN(C)C(c2cccs2)=O)CCCC1S(C)(=O)=O 43282,C1(CNC(c2ccc(NS(C)(=O)=O)cc2)=O)CC(F)(F)CN1C(C1CCCS1)=O 43283,N1(C(COC2CN(C(CC3CCC(C)CC3)=O)C2)=O)CCCNC(=O)C1C 43284,C1(C(=O)NC2C3CN(C(C(COC)N(C)C)=O)C2C3)CCn2cnnc2C1 43285,C=CCC(C)C(=O)N1CCC(OC2CN(C(=O)CCN3CCN(C)CC3)C2)CC1 43286,c1(CC(N2C(CN(C(CNC(CNC(C)=O)=O)=O)C)CCC2)=O)ccnc(O)c1 43287,N1(C(c2c(C(=O)OCC)con2)=O)CC(C2CCCN(C(=O)C(C)C(C)O)C2)C1 43288,C1(C)(CNC(Cn2c(C)c(Cl)cn2)=O)CN(C(c2cncnc2)=O)CCO1 43289,Cc1cccnc1C=CC(N1CCN(C(=O)CC(C)C(F)F)C(CO)C1)=O 43290,c1(C(N2CCCC(CCC)(NC(=O)C(O)C3CCC3)C2)=O)ccc2nncn2c1 43291,C1(F)(C(=O)NC(C(=O)NC(C)CCC2CCCC2)CNS(C)(=O)=O)CCCCC1 43292,C12(CNC(C(CC)c3ccccc3)=O)CC(NC(c3cc(C)[nH]n3)=O)(CCO1)C2 43293,c1(C(C)(C)C)ccc(C(=O)NC2CC(NC(C3CC3(F)F)=O)C2)o1 43294,C1(CNC(C(C)(C)c2ccno2)=O)CN(C(C2CCCC2)=O)C2CCCC2O1 43295,c1(C(N(CCCCNC(CC2CCN(C)C2)=O)C)=O)cncc2nc[nH]c12 43296,c1(C(N2CC(NC(C(n3ncc(C)c3)C)=O)C(F)C2)=O)c(F)cccc1Br 43297,c1(N2CCCC(C(C)C)C2)nc(N2CCS(=O)C3(CCC3)C2)nc2cccnc12 43298,C1(NC(c2c(C)cc(C)s2)=O)CN(C(C2CC3(C2)CC3F)=O)CC2(CCC2)C1 43299,c1(N(c2ccccc2)C(C2CCN(C(C)=O)C2)=O)nc(C)cc(O)n1 43300,C1(CC(=O)NCC2CCC(O)C2)C2CN(C(c3cnccc3Cl)=O)CC12 43301,c1(C(=O)NC23CC(NC(CNC(C4C(C)C4)=O)=O)(C2)C3)cc(N)cc([N+](=O)[O-])c1 43302,c1(C(=O)NCC(C)CNC(C2CN3CCN2CC3)=O)cc2cc(F)cc(F)c2[nH]1 43303,c1(C(N(C2CN(C(c3nc(C)sc3)=O)C2)C)=O)cc(Br)cn2ccnc12 43304,n1(CC(N2C(CN(C(C3C(=C)C3)=O)C)CCC2)=O)nc(C)cc1C(F)F 43305,CS(=O)(=O)c1ncccc1NC(=O)CC12CCCC1C2 43306,C1(NC(C(CC)(F)F)=O)CC2CCC1N(C(=O)C(COC(C)C)NC(C)=O)C2 43307,CC(C)(CNC(=O)CC(O)CNC(=O)CS(C)(=O)=O)C(N)=O 43308,C(=O)(C1=C(C)CCCC1)NC1C(SC)CN(C(=O)C(=Cc2ccc(F)cc2)C)C1 43309,C(C(CNC(=O)CCCOC)C(F)(F)F)NC(C1CCN(CC)C1)=O 43310,c1(OC)c(C(=O)NCC23CC2CN(C(C2(C#N)CCC2)=O)C3)cc(Cl)cc1Cl 43311,c1(CC)cc(C(=O)NC(CC(=O)N(CC(=O)OC)C)C2CC2)n[nH]1 43312,c1(NC(C(C)SCc2nncn2C)=O)ccc(CNC(=O)C2=C(Cl)CC2)cc1 43313,n1(CC)nc(C(=O)NC(C)(CSC)C(=O)NCC(=O)OC(C)C)c(C)n1 43314,c1(OC)ccccc1CCCNC(=O)C(=O)NC1CCCNCC1 43315,c1(N(C)C)ccc(NC(C2CCN(C(C3(N(C)C)CCC3)=O)C2)=O)cc1 43316,N1(C(C=CC(C)(C)C)=O)CCN(C(=O)CCc2ccc(Br)cc2)CC12CC2 43317,N(C(=NCCCF)NCC(c1ccc(OC(F)F)cc1)O)C(c1ccncc1)C 43318,CCC(O)(C(=O)N(CC(O)CNC(=O)CN(C)C1CC1)C)c1ccccc1 43319,C1(C(=O)NCC2CC(NC(c3c(Cl)nc(OC)s3)=O)C2)CCCC2(CCC2)C1 43320,C1(CNC(C(C)OCCC(C)C)=O)CCC(NC(=O)COCCCF)C1 43321,CC(C)(CC(F)F)C(=O)NC1CC2CC1N(C(=O)CCc1ccc[nH]1)C2 43322,c1(OC)c(C(=O)NC2CCC(C)(CNC(c3nncs3)=O)CC2)cc(F)cc1F 43323,C1(CS(=O)(=O)Nc2ccc(C(=O)OCCOC)cn2)(OC)CCOCC1 43324,N1(C(c2ccn(CC)c(=O)c2)=O)CCCC2CN(C(C3(CC4CC4)CC3)=O)CC12 43325,c1(NC(C2CN(C(c3ccc(Cl)cc3I)=O)C2)=O)cccc2c(I)n[nH]c12 43326,Cc1cccnc1CCNC(C1CCN1C(C1(c2ccno2)CCC1)=O)=O 43327,C1(C(NOCC(=O)NC(CCOC)C(N)=O)=O)CCC(=O)C(C)C1 43328,C12(C(=O)NC(CN(C(C(C)=C3CC3)=O)C)(CO)CO)CC3CC1C2C3(F)F 43329,Cc1cc(C(=O)NCC2(NC(C3(C)CCCN3C)=O)CC2)nn1C1CCCCC1 43330,C1(C(N2CCC(N(C(=O)Cn3cc(Cl)cn3)C)C2)=O)(OC)CCCOC1 43331,c1(C(=O)NC2C3(NC(=O)Cc4ccsc4)CCC(C2)C3)nnn2c1CCCC2 43332,Cc1cc(NC(C2CC(F)CN(C(c3cc(Cl)cnc3Br)=O)C2)=O)cnc1C#N 43333,Cc1c(NC(c2csc(CC3CC3)n2)C)ncnc1N1CCOC(CF)C1 43334,Cc1cccc(OCC(N2CCC2CNC(C2(N(C)C)CCCC2)=O)=O)c1F 43335,Cc1c(NCC2CC23CCC3)ncnc1N1CCOC(C(F)(F)F)CC1 43336,c1(C(=O)NCCCN(C(=O)CN2CCOCC2)CCO)cnc2sccn12 43337,N1(S(c2ccn(C(C)C)n2)(=O)=O)CCCC2(CNC2)C1 43338,c1(OCC)ccccc1C(=O)N(C1CCN(C(=O)C(C)c2cccs2)CC1)C 43339,CC(C)CC(O)C(C)C(=O)N1CCC(CNC(c2coc(CO)c2)=O)CC1 43340,C1(C(=O)NC2C(NC(COC3(C#C)COC3)=O)C2)CN2CCCC2CO1 43341,CC(N=c1[nH]c(=NCCCF)[nH]c2c1COC2)c1snnc1C1CC1 43342,c1(OC)cc(CC(N2CC3CC(NC(=O)CCC(N)=O)C2C3)=O)cc(OC)c1O 43343,C1(CNC(=O)COc2ccccc2)CCN(C(=O)C=C2CC2)C12CC2 43344,c1(OCC)ccc(C)c(C)c1.C12CC(C)N(C1)C(=O)C(=O)NC1(CC1)C(=O)N2 43345,CCCC(C(=O)N1CC(NC(C2CCC2n2ccnc2)=O)C1)OCC 43346,Cc1cc(C(=O)NCCN2CCC(NC(=O)CC3CCCOC3)CC2)nn1C 43347,C1(C(N(CCC(=O)NCc2c[nH]nc2C(C)C)CC)=O)CNC(=O)CC1C 43348,c1(OC)ccccc1C1CC1C(=O)N(CC(C)(C)NC(c1nn(C)cc1C)=O)C 43349,N1(CC(=O)NC(c2ccc(C)s2)c2ccccc2)CCOCC12CNC(=O)OC2 43350,n1(CC)nc(C(=O)N(CCCC(=O)NCC(C2CCCC2)C)C)c(C)n1 43351,c1(OC)ccc(F)c(C(N2CCOCC(NC(=O)COCC(C)C)C2)=O)c1 43352,C1(C(N2CC(C)(NC(c3cc(OCC)n[nH]3)=O)C2)=O)(CC)CC1S(C)(=O)=O 43353,c1(OC)cc2[nH]ncc2cc1NC1CN(C(c2[nH]nc3cc(C)ncc23)=O)C1 43354,C1(CC(N2CCC(CNC(CCN(CCCCC)C)=O)C2)=O)CC2CCC1CC2 43355,C1(C(N2CC3C(NC(Cc4c(C)cc(F)cc4)=O)(C3)C2)=O)CN(CP(C)(C)=O)C1 43356,n1(CCC)cc(C(N2CC(OC)C(NC(=O)C3=CC(C)(C)C3)C2)=O)cc(Cl)c1=O 43357,C1(N(C(CCC)C(=O)NC(C)C)C)CC2CCC(C1)N2C(=O)C(C)c1cccs1 43358,C1(NC(C)(C)C)CC2(CC(S(CC(=O)OC)(=O)=O)C2)C1.C12CN(C1)C(=O)N2 43359,c1(C(=O)NCCC2N(C(CCCN=[N+]=[N-])=O)CC(F)(F)C2)ccc2c(c1)COC2 43360,N1(C(C2CCN(CC(C)C)CC2)=O)CC(NC(=O)Cc2cnns2)CC12CCC2 43361,Cc1cc(C(=O)NC2CC3CC2N(C(C2(C(F)F)CC(F)(F)C2)=O)C3)cnc1O 43362,c1(OC)cnc2ccccc2c1C(N1CC2CC(NC(=O)CC3CC3)C(C2)C1)=O 43363,c1(CCC(=O)NC(C)CN(C(=O)C(C2CCCN(C)C2)C)C)cccc(F)c1F 43364,C12(CC(=O)NC(CC(C)NC(c3nccc(NC)c3)=O)C)CCCCC1C2(F)F 43365,C1(CNC(COc2cccc(C(C)C)c2)=O)Cc2ccccc2CO1 43366,N1(C(C(C=C=C)C)=O)CCCC(C2CCN(C(=O)CCC(=O)OC)CC2)CC1 43367,c1(OC)cccc(C(=O)NC2CC(NC(C3CCC(C(F)(F)F)C3)=O)C(O)C2)c1 43368,Cc1cn(C)nc1C(N1CCCCC1CC(N1CCCC1(C)C1CCC1)=O)=O 43369,c1(OC)ccc(Cl)c(C(=O)NC2CCC(NC(c3cnc(Cl)n3C)=O)CC2)n1 43370,C(=O)(C(C)(C)CN(C(=O)CCc1cncs1)C)NC1CC(COC)C1 43371,Cn1cnc2sc(C(=O)NC3CN(C(=O)CC4CC5(CC5)CO4)CC3O)cc12 43372,N1(C(C(C2CCC2)OCC)=O)CCN(C)C(CNC(C2CC3(CC(=O)N3)C2)=O)C1 43373,c1(C(=O)NCC(CN(C(Cc2c(C)cccc2)=O)C)O)ccc2c[nH]nc2c1 43374,C1(NC(C=CCCC(C)C)=O)CCCN(C(c2cnn(C3CC3)c2)=O)CC1 43375,c1(C(=O)NCc2cn(CC(CC)O)nn2)cc2c(C)cc(C)cc2[nH]1 43376,c1(CNC(C2N(C(C(C)CN(C)C)=O)CSC2)=O)ccc(O)cc1 43377,CC(C)(CN=c1[nH]c(=NCc2ccc(F)cc2Br)[nH]c2ccccc12)C1CCC1 43378,N1(C(c2c(C)oc(C(C)C)c2)=O)CC(NC(C2CCC2C)=O)C2(CCCC2)C1 43379,Cc1cc2c(C(=O)NC3COCC3NC(c3cc(CO)[nH]n3)=O)nccn2n1 43380,C1(NC(C2CN(C)C(=O)CC2)=O)CCC2CN(C(=O)COCC(F)(F)F)CC2C1 43381,CCCCC(C)CCC(=O)NCC1COCCN1C(c1ccc2nccn2n1)=O 43382,N1(C(C(C)C#N)=O)CC(CNC(c2c(C3CC3)cnn2C)=O)CC1(C)C 43383,N1(C(C=CC2COC(C)(C)O2)=O)CC(NC(=O)CC2CC2)CC2(CCC2)C1 43384,c1(C(=O)NCCCCCN(C)C(c2ccc(Cl)cn2)=O)cc2n(c1)CCOC2 43385,c1(CNC(C2CCN(C(c3ncc(C(C)=O)s3)=O)C2)=O)ccc(F)c(C)c1 43386,C(=O)(C1=C(F)CN(C(c2csc(C)c2)=O)CC1)N1CC(C)CC(OC)C1 43387,C1(C(=O)Nc2c(C(C)=O)ccc(Br)c2)CC2(CCN(C(C3(C#N)CC3)=O)CC2)C1 43388,n1(C(C)C)cc(C(N2CCC3(CC3NC(=O)C(C)n3cncn3)C2)=O)ccc1=O 43389,c1(C(N(C2CCCC(NC(C3(C)C=CCCC3)=O)C2)C)=O)cnc2[nH]ccc2n1 43390,Cc1cnc(S(C)(=O)=O)nc1N1CCC2(C(N3CC(CO)C(O)C3)=O)CC2C1 43391,N1(CCC)CCC(C(=O)NC2CN(C(=O)OC(C)(C)C)C2)C(O)C1 43392,CC1Cn2nc(C(=O)N(CCCCCNC(=O)COCCF)C)cc2C(=O)N1 43393,c1(CC(C)NC(=O)NCC2COCCN2)ccc(F)cc1Cl 43394,C(=O)(CCCN(CC)C(=O)Cc1sc(-c2nc[nH]n2)nc1-c1ccccc1)OC 43395,c1(N(C)C)ncnc(NC(C2COCCN2C(=O)OC(C)(C)C)=O)n1 43396,c1(N2CC(NC(C(C3CCOCC3)C)=O)C(C)(C)C2)ncc(Br)cc1C#N 43397,C(N=c1[nH]c(=NCCc2nccc(O)n2)c2[nH]ccc2[nH]1)c1c(N)cc(F)cc1 43398,O=C(CC1(C(=O)O)CCc2ccccc21)NC(c1cc(Br)ccc1F)C1CCOC1 43399,CC(C)CC(O)CC(=O)NCCN(C(=O)Cn1cccnc1=O)C(C)C 43400,c1(C(CNC(C2(C(C)C)CCC2)=O)NC(c2cc(CC)on2)=O)cccc(C)c1 43401,c1(OC)cc(NC(c2cnc(CNC(=O)CC3CCC(C)O3)nc2)=O)ccc1O 43402,c1(OC)ccccc1NC(=O)C(C1CN(C(=O)CC2(SC)CCC2)C1)OC 43403,C1(c2nnnn2C2CCCCC2)(NCCC2(C)CC2)CCC(=O)NC1 43404,N1(C(c2cc(CNC(C(C)N=[N+]=[N-])=O)no2)=O)CCOC2CCCCC12 43405,N1(C(c2c(CC)cco2)=O)C2CCC1CN(C(=O)C(c1cccc(Br)c1)O)C2 43406,C1(C(=O)Nc2c(C)cc(Sc3nncs3)cc2)CCc2ccnn2C1 43407,C1(C(N(CC(=O)NC)CC)=O)CC12CCN(C(=O)Cc1ccc(C)nc1)CC2 43408,C1(C(N2CCC(c3cc(O)no3)C2)=O)CCCC2CCCN12 43409,C(=O)(CCCC(F)F)N.N1(C(c2nc(C(=O)NCC#C)sc2)=O)CCN(CC)CC1 43410,N1(C(c2n(CC)nc(C)c2)=O)CC2CN(C(=O)CCc3cccnc3C)CC12 43411,N(C(=NCC)N1CCc2ccccc2C1)C(CC=C)CC 43412,Cn1ncc2c(C(=O)NC3CN(C(=O)Cn4cc(Cl)cn4)CCC3F)ccnc12 43413,CC1(C)CC(OC(N2CCCCC2OC2CCCN2)=O)CO1 43414,CC12CN(C(=O)C3=COCC3)C(C(=O)NC(c3cscn3)CO)(C1)C2 43415,N1(C(c2c(C)n(C3CC3)cc2)=O)CCOCCC1C(F)(F)F 43416,C1(NC(C2(C)N(C(C(CC(C)C)O)=O)CCC2)=O)CCn2nnnc2C1 43417,C12(NC(CCCSC)=O)CCN(C(c3cc(O)nn3C)=O)CCC1C2 43418,Cc1cccc(C(=O)C=CC(N2CC(NC(c3scnc3Cl)=O)C(C)C2)=O)c1 43419,C(C(S(C)(=O)=O)C1CC1)NC(c1ncccc1F)c1n(CCCOC)nnn1 43420,C1(C)(C(=O)NCC2C(C)CN(C(c3ccc(F)cn3)=O)CC2)CCC(C)(C)CC1 43421,CCC(C)CC(C)C(=O)N(C)CCOCCNC(=O)CCc1cccc(Cl)c1 43422,N1(C(CSCCN(C(C(C)=CCC)=O)CCC)=O)CCCC1C(C)(C)O 43423,N1(C(c2c(OCC(C)C)nccc2)=O)CCCC(C2CCN(CC(N)=O)C2)C1 43424,N1(C(C(C)SC)=O)CCC(NC(=O)COc2ccc(F)cc2F)C(F)(F)CC1 43425,C1(NC(c2n[nH]c(CC)c2Cl)=O)CCN(C(=O)CSCC(=O)OC)CC1C 43426,Cc1ccccc1CN1CCCC1CN(C(=O)CCCOCCN(C)C)C 43427,N1(C(=O)Nc2c(CC)nn(C)c2)CCN(C)C(CC(=O)NC)C1.n12cc(nn1)C2 43428,N1(C(CSc2c(C)n[nH]c2C)=O)CCC(NC(=O)CN2CCCNC2=O)CC1C 43429,N1(c2nnc(C)s2)CCC(CNC(c2ncnc3c(C)csc23)=O)C(F)(F)CC1 43430,N1(C(=O)Cn2cccc2)CCC2CCCC12C(N1CC(CCO)C1)=O 43431,C1(O)(CC(N2CCC2Cn2cc(CC3(O)CCSC3)nn2)=O)CCCCC1 43432,CC1(CCCO)CCCN1C(=O)Cn1cc(I)nn1 43433,c1(C(N2CC(NC(c3cc(C)sn3)=O)C(F)C2)=O)cc(F)c(C)cc1F 43434,C(C(CC(C)C)C(=O)NCc1ccoc1)NC(CC1(OCC)CC1)=O 43435,c1(C(=O)NCC(C(C)C)NC(C(COC)(C)OC)=O)c(C)cc(Cl)cc1[N+](=O)[O-] 43436,C(=O)(C(C)(F)C(F)(F)F)NCC1CCN(C(C=Cc2ccc(C)cc2)=O)C1(C)C 43437,C1(C)(CNC(C(CC)SC)=O)CN(C(C2(CO)CC(F)(F)C2)=O)CCO1 43438,C1(NC(C(CC)N(C)C)=O)CCOC(C(N2CCOC(C(C)C)C2)=O)C1 43439,C(=O)(CC(F)(F)CC)N(C(C)C(=O)NCCC#CC(C)(C)C)CC 43440,C12(NC(C(C=C)O)=O)CC(CNC(C3CCS(=O)(=O)C3(C)C)=O)(C1)OC2(C)C 43441,CCCCCC(C(=O)N1CCC(C)(NC(c2onc(C)c2C)=O)CC1)C(C)C 43442,C(=O)(C(CCC(=O)OCC)N1CCCC(c2ccncn2)C1)NCC=C 43443,c1(C(=O)NCCCC(C)NC(c2cn(C)cn2)=O)nc(Cl)sc1Cl 43444,C1(NC(C(CCSC)Nc2ccccc2)=O)COC2(C1)CN(C(=O)CC#N)C2 43445,CC(C)(C(=O)N1CC(NC(c2cccc(Br)c2)=O)CC(F)C1)C(N)=O 43446,C12(C(=O)NC(C)Cc3ccc(CNC(=O)CO)cc3)CCC(F)C1CC2 43447,CN1CCN(C(C2CCOC2CNC(=O)C(F)C(C)(F)F)=O)CC1CO 43448,C1(NC(C2(CC)COC2)=O)CC(NC(=O)C(C)OCC(C)C)CC1O 43449,C1(NC(C(C)NC(C)(C)C)=O)CCN(C(c2cc(C3CC3)ns2)=O)CC1 43450,Cc1nc(C)c(C(=O)NCC2CC(F)(CNC(C3CCC(C)O3)=O)C2)nc1C 43451,CC1CC(c2nn[nH]n2)CCN1C(C1CCCN1Cc1ccccc1)=O 43452,C=C(CNC(C)=O)CCNC(=O)COCCCOCCC(=O)N.O(C(F)(F)F)C(=O)C 43453,c1(CCN2CCC(CNC(c3c(C)n[nH]c3)=O)CC2C)cn(C)c2ccccc12 43454,C1(NC(C(C)C2CCC2)=O)C(C)CCN(C(c2ncc(C(F)(F)F)n2C)=O)C1C 43455,C1(C)(CNC(C(C(C)C)O)=O)CCCN(C(c2cccc(Cl)c2F)=O)C1 43456,C(CN(C)C)(CN=c1nc(N(C)Cc2nc(CO)n[nH]2)cc(C)[nH]1)OCC 43457,c1(C(=O)NC2C(C)CCN(C(c3cc(Cl)cnn3)=O)C2)ccc2nc(O)oc2c1 43458,C1(C(=O)O)(OC)CCS(=O)(=O)C1.c12cc(no1)C(=O)NCC2 43459,C1(C(N2CCCC(F)(C(=O)NCc3snc(C)n3)C2)=O)CC(=O)CC12CCC2 43460,N1(C(C)=O)CC(O)CC1C(N1CC(CO)(NC(=O)Cn2nc(C)nc2C)C1)=O 43461,c1(OCCOC)ncccc1C(=O)NCCCNC(=O)CC1CCC(C)(C)C1 43462,N1(C(CN(S(CC)(=O)=O)C)=O)CC2CC1C2CNC(=O)C(C)CN1CCC1 43463,c1(OCCC(N2CCC(C(C)NC(CCC#C)=O)CC2)=O)cc(C)cc(C)c1 43464,C(=O)(CC(C)(C)C1CC1)NC(C1(O)CN(C(=O)C=C2CCSCC2)C1)C 43465,C1(CNC(CCC(C)SC)=O)CN(C(c2ccc(C(C)C)cc2N)=O)CC1(F)F 43466,C1(C(C)NC(CCN(CCC)C)=O)CCCN1C(=O)CC1(CC)CC1 43467,c1(C(N(CCC(C)NC(C2C(C=C)C2)=O)C)=O)cc2ncccc2[nH]1 43468,C1(CC(=O)NCC(C)CNC(=O)C(C2CCCCC2)C2CC2)CCCC(C)(C)O1 43469,C(=O)(C(CO)C(F)(F)F)N(C1CCCN(C(c2[nH]cc(C)c2C)=O)C1)CC 43470,N1(C(C=Cc2c(C)nccc2)=O)CC(C)CN(C(=O)C(=O)NC2CC2)CC1C 43471,c1(N(c2ccccc2)C)nc(=NCN)[nH]c2c1CC(C)CC2.C12CCCC1OC2.SC 43472,C1(C(N2CCN(C(C3CN(C(C(C)(C)O)=O)C3)=O)CC2)=O)CC2(C1)CS(=O)(=O)C2 43473,N1(C2CCN(C(CC=C)=O)CC2)CCN(C(=O)CC2CC=CCC2)CC1=O 43474,C1(NC(c2c(C)nc(CCC)o2)=O)COCCN(C(c2ccc(C#N)s2)=O)C1 43475,O=C(N=c1ccn(CCCO)[nH]1)C(F)=CC1CC1.n1(CC(=O)N)ncnn1 43476,C1(CC)CN(C(c2occc2F)=O)CCC1NC(c1ccc(=O)n(C)n1)=O 43477,C1(CNC(C2CC(C)(F)C2)=O)CN(C(c2ccc(N)cc2F)=O)CCC1(F)F 43478,c1(OC)ccc(C(=O)NC2CCC(NC(=O)CCC3CCOC3)CC2)nn1 43479,C12(C(N3CCC(CCC(=O)NCC4(C)CC4)C3)=O)CC(C)(CCO1)C2 43480,C(C(CCC(=O)O)CC(F)(F)F)OC(C1(c2ccc(OC)cc2)COC1)=O 43481,c1(C(N2C3CCN(C(c4ncccc4Br)=O)C3CC2)=O)cn2cccnc2n1 43482,C12(NC(CCCC#C)=O)CCCCC1N(C(c1ncccc1F)=O)CC2 43483,Cc1cccnc1CC(=O)NC1(CCC(=O)NOCCC2CC2)CCCC1 43484,C1(C(N(CCCNC(=O)CCc2cccc(O)n2)C)=O)CCC2CCCCN12 43485,C(=O)(C(C)(C)Cc1ccccc1)N1CC(CNC(C(CN(C)CC)F)=O)C1 43486,N1(C(CN(C)C)=O)CCC2CN(C(c3cc(C4CCOCC4)[nH]n3)=O)CCC12 43487,N1(C(C2(CC#C)CCCO2)=O)CCC(NC(=O)C(CCO)N(C)C)CC1 43488,CC(C)(CC(F)F)C(=O)N1C2CCC1CC(CNC(c1cnc(C3CC3)[nH]1)=O)C2 43489,CCC(CCCC(=O)NCC1(CF)CCC1)NC(c1cc(OC)n(C)n1)=O 43490,c1(-c2cc(C)[nH]c2)nn(-c2ccccc2)cc1CNCc1ccon1 43491,C1(NC(=O)CC23CC(C2)C3)CN(C(=O)Cc2ccccc2)Cc2nccn2C1 43492,N1(C(C(CC)N(C)C)=O)CCC(NC(C2CN3CCC2CC3)=O)C12CCCC2 43493,N1(C(C(C)OCCC=C)=O)CCC2CN(C(c3ccc(F)c(Cl)c3F)=O)C2C1 43494,O=C1CCC(CNC(c2ccc(CNC(=O)CC3CCCO3)s2)=O)O1 43495,C1(NC(=O)Cn2cccn2)CN(C(c2cccc(C(F)(F)F)c2F)=O)CC1(F)F 43496,N1(C(C2(CN(C)C)CC2)=O)CC(C)(CNC(C2(C(N)=O)CCC2)=O)CC1(C)C 43497,c1(CNC(=O)NCCCOCC#C)c(Cl)nc(C)nc1Cl 43498,C12(C)CCC(C1)C2.C1(C(=O)NC(C)C)CCN(NC(CN(CCC#C)C)=O)CC1 43499,C1(CNC(C2CCCOC2)=O)CC12CCN(C(=O)CC1CC3CC(=O)C1C3)CC2 43500,N1(C(C(C)=C2CC2)=O)CC(C)CN(C(c2nc[nH]c3ncnc2-3)=O)C(C)C1 43501,c1(CCC(=O)N(C2CCC(SC)CC2)C)c([N+](=O)[O-])ccc(F)c1F 43502,n1(CC=C)cc(C(=O)N(CC(CC)NC(=O)CC23CCCC2C3)C)cn1 43503,C(CCCC(F)(F)F)OC.N1(c2n3c(nn2)CCC3)CC2CCC2(OC)C1 43504,C1(C(C)(C)C)(C(=O)NCc2c(N)cccc2F)CCS(=O)(=O)CC1 43505,CCCC(O)C(=O)N1CCC(N(C(=O)CC(C)SC)CCO)C1 43506,c1(C(N2CC3(CCN3C(=O)C=Cc3cccnc3)C2)=O)c(F)ccc(F)c1F 43507,CC(C)(C)CCCNC(=O)NCCS(N1CCCC(C(F)(F)F)C1)(=O)=O 43508,C1(C(C(=O)NCC)N(C)CC2CC2)CCS(=O)(=O)C1 43509,C(CCC(=O)N1CCCC(O)CC1)(C(C)C)NC(c1c(CCC)nco1)=O 43510,C12(C(=O)NCC3N(C(C(=Cc4ccccn4)C)=O)CC(F)C3)CCC(C1)C(C)(C)O2 43511,C(=O)(CC(C)(C)C(F)F)N1CC(CC)C(NC(=O)CN2CCOCC2)CC1 43512,Cc1ccccc1CC(=O)NC1COCCC1C(=O)NC(c1ccc(O)cc1)C 43513,N1(C(COCCC)=O)CC(CNC(c2cc(C(N)=O)co2)=O)OC2CCCC12 43514,C1(C)(CNC(C2C=CC(NC(C(C)n3cccc3)=O)C2)=O)NC(=O)NC1=O 43515,c1(C(=O)NC(CNC(CC(C)C(C)(C)C)=O)CO)ccnc2c1CC(=O)N2 43516,N1(C(c2c(C)occ2)=O)CCC(NC(c2cnc(N(C)C)cn2)=O)C(O)C1 43517,CC(C)C(O)CC(=O)NCC1CC(F)CN1C(=O)C=Cc1cc[nH]c1 43518,C1(C(=O)NCc2cnco2)(NC(=O)Cc2ccsc2)CCCCC1 43519,CC(C(=O)NC1CN(C(c2ncccc2N)=O)CCC1c1ccccc1)C(C)(C)C 43520,C(=O)(C(F)C(F)(F)F)N(CCC)CCNC(C1CCC1C(C)(C)C)=O 43521,C(=O)(C1CCc2ccc(C)cc21)N1CC2C(CNC(C3(NC(C)=O)CCC3)=O)(C2)C1 43522,N1(C(CSCCCC)=O)CC(CNC(c2cc(OC)cnn2)=O)CC1C 43523,c1(C(=O)NCc2nccn2C(F)(F)F)cccc(Cl)c1Br 43524,c1(C(=O)Nc2ncc(-c3cccc(CCO)c3)s2)cc(Br)cnc1O 43525,C1(C(=O)NC2CCC(NC(c3c(C(C)C)c[nH]c3)=O)C2)CCCN(C)C1 43526,Cn1c(C(N2CCC(NC(=O)CCCC(C)(C)C)C2)=O)c(Cl)c2ccccc12 43527,CCC(CC)C(=O)N1C(C(=O)N(C2CCN(C(C)C)C2)C)CCC1C1CC1 43528,c1(C(N2CC(C(=O)NCCC(=C)CNC(=O)OC(C)(C)C)C2)=O)cc(C)ccc1Cl 43529,Nc1cc2ccccc2cc1C(=O)NCC1CCN(C(=O)C(F)CC2CCC2)C1 43530,C1(C(=O)NC2C(CNC(c3c(C)[nH][nH]c3=N)=O)CC2)COCC(=O)N1C(C)C 43531,C1(CC(=O)NC(C2CCN(C(=O)CCCF)C2)C)CCN(Cc2ccccc2)C1 43532,C(=O)(C1=NNC(=O)C1)NCC(C)(C)NC(C1CN(C2CCOC2)C1)=O 43533,C1(C(=O)NCC(CNC(CCCOCC)=O)C)CCCC12OCCO2 43534,c1(OC)cccnc1CNC(C1(CNC(=O)Cc2ccc(O)cc2)CC1)=O 43535,c1(C(=O)NCCN(CCC(F)(F)F)C(CC2CCCCC2)=O)ccc(F)c(F)c1Br 43536,C1(C(N(CC(C)(C)CO)C)=O)C(C2CC2)CCN1C(c1ncccc1Cl)=O 43537,Cc1nc(C)c(C(N2CCC(OCCNC(=O)Cc3cccc(F)n3)C2)=O)[nH]1 43538,C1(NC(c2c(C)nn[nH]2)=O)CCCCCN(C(C2CCCCS2)=O)C1 43539,Cc1nn(CC(=O)NCCCN(C)C(C2CCC(C3CC3)C2)=O)c(=O)n1C 43540,c1(CN(C(=O)C(F)n2ccnc2)CCNC(CSC)=O)ncnn1C 43541,C1(CCNC(=O)C(C2CC2)OC)(OC)CN(C(C2(c3ccnn3C)CC2)=O)C1 43542,c1(NCCCc2n(C)ncn2)[nH]c(=NCCc2ncc[nH]2)nc2c1cnn2C 43543,Cc1c(C(N2CCCC(C)C2CCNC(C2OCCO2)=O)=O)nc2sccn12 43544,CCCCC(C(=O)N(CC(=O)NC1(OC)CCC1CC)CCOC)N(C)C 43545,c1(N(C(CC)C)C)cc(N(C)CCN(C)C)nc(CCCn2cccn2)n1 43546,Cc1oc(C(C)(C)C)cc1C(N1CCC(=CCNC(=O)C(C)CO)CC1)=O 43547,c1(SCCCOCC(=O)NC(CNC(C(C)c2cncs2)=O)CO)ccnn1C 43548,Cc1cc(C(=O)NC(C)(C(=O)NCCc2cc(C)ns2)C2CCC2)ccc1C#N 43549,c1(C(=O)NCC23N(C(c4cc(C)c(C)o4)=O)CC(C2)C3)cccc(C=C(F)F)c1 43550,C1(CC(=O)N(CC(C)O)C(C)C)C2CCCC2N1C(=O)C=Cc1ccsc1 43551,C1(CNC(C(C=C)(C)CC)=O)CN(C(C2OCCO2)=O)CCC1(F)F 43552,c1(C(=O)NC2CC(CNC(c3sc(C)c(O)n3)=O)C2)ccc(=NCC2CC2)[nH]c1 43553,C1(NC(=O)Cc2ccc(O)nc2)CN(C(=O)C2=CCCSC2)C2(CCCOC2)C1 43554,N1(CC)CCN(C(C2CCN(C(c3cc[nH]c(=N)n3)=O)C23CC3)=O)CC1=O 43555,c1(CCNC2CC(C)N(c3ccccc3)C2)cc(O)nc(O)n1 43556,Cc1ccnc(CC(=O)NC(C2CCCN2C(=O)CCc2ncc(F)cn2)C)n1 43557,c1(SCCC)ncc(C(N2CCC(C)(N3CCCC3)C2)=O)cn1 43558,CC(C(=O)N1CCN(CCCNC(C2CCCN(C(N)=O)C2)=O)CC1)C(F)F 43559,N1(C(C=C(C)C(F)F)=O)CC(NC(c2ccncc2-c2ccccc2)=O)CC(O)C1 43560,C1(C)(C(=O)NCC2N(C(c3c(CC)nc(C)o3)=O)CCOC2)CCC12CCC2 43561,N1(C(c2cc(CCC)on2)=O)CCC(C(F)CNC(C2CC2C#C)=O)CC1 43562,c1(NC)cnc(C(N2CC(CNC(c3n[nH]cc3Br)=O)C(C(F)(F)F)C2)=O)cn1 43563,Cn1c(C(=O)N(CCCN2CCc3ccccc32)C(C)(C)C)cc2ccsc12 43564,C=CC(C)(C)CCCNC(=O)CCCC(C)NC(C1CC(C)(F)C1)=O 43565,Cn1c(=O)n(CC(N2CC3(C2)CN(C(=O)CCOC2CC2)C3)=O)c2ccccc12 43566,c1(C(=O)NCC(C)N(C(=O)Cc2csc(C3CC3)n2)C)cc(C(F)(F)F)no1 43567,CC1(C(N2CC(C#N)C2)=O)CCN(C(=O)CSc2nc[nH]n2)C1 43568,Cc1ccccc1C1(COC(C2C3CC2N(C(=O)NC(C)(C)C)C3)=O)CC1 43569,C12(C(=O)OC)CCC(C(N3CCC(C)C(NC(=O)C(C)SC)C3C)=O)(CC1)CC2 43570,N1(C(c2n(CC)nnc2C)=O)CCC2CCCC12CNC(=O)CCC(C)(C)C#N 43571,C1(C(N(CC(CNC(c2c(C)nc(O)cc2)=O)(C)C)C)=O)CC2CCCCC2O1 43572,C1(CC)C(=O)NCCCN1C(C1C2CCC(C2)N1C(c1cc(C#N)cs1)=O)=O 43573,n1(CC(=O)NCCC(=O)N(C)C)cc(C2CC2c2ccccc2)nn1 43574,N1(C(CC2C(C)(C)C2)=O)CCCC(NC(c2ccc(C(F)F)cc2)=O)C1 43575,c1(C(N2CCC(CNC(=O)C(O)Cn3cncn3)C2)=O)cc2sc(Cl)cc2s1 43576,N1(CCC)CC(NC2(CNC(=O)OC(C)(C)C)CCCC2)CC1=O 43577,N1(c2snc(C(C)C)n2)CCN(C(=O)NC(C)C(C)n2cccn2)CC1 43578,C1(C(=O)NCCc2nc(CC)[nH]n2)CCN(C(=O)c2cnn[nH]2)O1 43579,c1(SC)cc(=NC(=O)Cc2csc(NC(=O)Nc3ccccn3)n2)[nH]n1C 43580,CN1CC(C)(C)CC1C(N1CC(NC(=O)C2=C(Cl)CC2)C(O)C1)=O 43581,C1(C(=O)NCC(CC(=O)NC(C)C(C)C)OC)CC2(CCC2O)C1 43582,C(CCN=c1nc(N2CC3CCC2CC3)c2ccc(Cl)cc2[nH]1)n1c(C)ncc1 43583,N1(C(CC=C)=O)CC(NC(C2(C(=O)OCC)CCCO2)=O)C(c2cnn(C)c2)C1 43584,C1(NC(C=CCCC=C(C)C)=O)CCOCC1NC(c1ccc(C(F)F)nc1)=O 43585,N1(C(C=C(CC)CC)=O)Cc2ccccc2C(NC(c2cccc(CC)n2)=O)C1 43586,CS(=O)(=O)CCC(=O)NCC12CCC(CC1)N2C(c1cncc(OC2CC2)c1)=O 43587,C1(CC(=O)NCCC2CN(C(=O)CCc3cccs3)C2)CC(F)(F)C1 43588,c1(CNC(=O)Nc2c(SC)cccc2)cccc2[nH]c(C)cc12 43589,N1(C(c2ccc(F)nn2)=O)CCOC2(CCN(c3nccnc3F)CC2)C1 43590,CCCC(C)(O)CC(=O)N1CCCCC(CNC(=O)CCNC(C2CCC2)=O)C1 43591,c1(OC)cccc(C(=O)NC2CC(CCNC(C3CCC(=O)NC3)=O)C2)n1 43592,Cc1nc(CC(=O)N(C)CCN(C(=O)C2=CCCC2)C)c(Cl)s1 43593,c1(OC)ccc(Cl)c(F)c1C(=O)NC(C1CCOC1)CNC(c1occc1C)=O 43594,c1(OC)cc(C(N2CC(C(C)NC(c3occc3C)=O)C2)=O)cc(N)c1O 43595,c1(C(=O)OC)nc(NC(=O)NC2(CO)CC(C(C)(C)C)C2)cs1.C(C)(C)C 43596,Cc1occc1S(C)(=O)=NC(=O)CC1(C)CC1 43597,C(CCCCC(=O)NCc1n[nH]cc1C(=O)NC1CN(C)CC1(F)F)OC 43598,C(=O)(CC(C(F)(F)F)NC(c1ccc2ccoc2c1)=O)NC(CCC)C1CCC1 43599,N1(C(C2(Cl)C(C)(C)C2)=O)CCC2(CCC2NC(=O)CCP(C)(C)=O)CC1 43600,C1(CNC(c2cncc(C)c2)=O)CCC(C)N(C(=O)CCc2cncnc2O)C1 43601,C1(CC(=O)N(CCN(C)C)CCO)CCCCC1NC(=O)CC1(N(C)C)CC1 43602,N1(C(CC2CC(C)C2)=O)CCC(C(N2CCC(c3ncco3)C2)=O)C1(C)C 43603,CN1CCC(C(N2CCC2C2CCCCC2)=O)(NC(C2CC3(CC3)CO2)=O)C1 43604,Cc1cc2sc(C(N3CC(F)(CNC(=O)CCn4ccnc4)C3)=O)cc2s1 43605,N1(C(C2(C#C)CN(C(c3ccc(C4CC4)o3)=O)C2)=O)CCC(C2CCC2)C1 43606,c1(C(N2CCC(C3N(C(c4cc(C)no4)=O)CCC3)C2)=O)cn(C)c(=O)nc1O 43607,c1(C(C)C)cccc(C(=O)N(CC(C)(C)NC(=O)C=CC2CCCC2)C)c1F 43608,c1(C(=O)NCCCCCN(C(CC2(CC)CC2)=O)C)c(C(C)C)cccc1C 43609,c1(C(N(C)CC2(NC(C3CCCC3c3nc[nH]n3)=O)CC2)=O)cccc(=O)n1C 43610,CS(=O)(=O)C(CNC(=O)CCc1cocn1)CNC(=O)CC1CCCOCC1 43611,C1(NC(C2CCN(CC(C)C)C2)=O)C2CC1CN(C(=O)CC1CSC1)C2 43612,C(=O)(CC(C(C)(C)C)NC(=O)Cc1cncs1)NCC(CN(C)C)O 43613,Cc1cncc(C(=O)NCC2CCN(C(=O)Cn3ccc(=N)[nH]3)C2)c1 43614,C1(C(=O)OC)CCc2cc(OC)ccc2N1C(=O)CCc1ccc(C)cn1 43615,c1(C(N2CCCC(C(=O)NC3C(OC)CC3O)C2)=O)c(F)cccc1[N+](=O)[O-] 43616,N1(C(C2C(C)C2C)=O)CCN(C(=O)Cc2nc(-c3ccco3)no2)C(CO)C1 43617,C(=O)(C(CNC(c1cc(N2CCCC2)ccn1)=O)CC(C)C)OC 43618,C(=O)(C(C)(C)C(C)NC(c1c[nH]c(C)cc1=O)=O)N(c1c(OC)cccc1)C 43619,c1(C(N(CCNC(C2(CC=C)CC2)=O)C)=O)cccc2ncnc(O)c12 43620,N1(C(CC2CCCC(NC(CCCCC=CC)=O)C2)=O)CC(C)CCCC1C 43621,C1(NC(CCc2onc(C)n2)=O)CCN(C(=O)CCc2scnc2C)CC1(C)C 43622,CS(C)(=O)=NC(=O)C(=O)NC1CN(C(C2CCCN2C(C2CCCC2)=O)=O)C1 43623,c1(C(=O)NCCC(C)NC(C(C)=C2CCC2)=O)ccc(-n2cccc2)cc1 43624,N1(c2cc(NCCN(CCOC)C)nc(C)n2)C2CCC1CC(CCO)C2 43625,CC1CC2(CCN(C(=O)CCN3CCCC3=O)CC2)CN1C(C1CCC1(C)C)=O 43626,c1(OC)ccc(O)cc1C(=O)NCC1(NC(c2nnn(C)c2C)=O)CCOC1 43627,N1(C(COC(C)=O)=O)CCCC12CCN(C(=O)Cn1cc3ccccc3n1)C2 43628,C1(CC)CN(C(c2ncc(F)cn2)=O)CC1NC(=O)C(C1CC1)SC 43629,C1(CNC(C(CC)CC)=O)CCC(C)(C)CN1C(c1cccc(C2CC2)c1)=O 43630,CC(C)C(F)C(=O)NC1(C(=O)NCC2CN(C3CC3)C2)CCC1 43631,C1(C(=O)NCc2cccc(OC(F)F)n2)CCc2nc[nH]c2C1 43632,C=C(C)CCCC(=O)N(C)CCOCCN(C(=O)CC1C(C)C1(F)F)C 43633,C12(C(=O)OC(C(=O)NCC)C)CCC(CC1)C2(C)C 43634,C1(C(C)C)OCCC1NC(c1ncc(I)s1)(C)C 43635,c1(C(=O)NCC2CCN(C(C(CCC)O)=O)C2(C)C)ccc2cc(Cl)ccc2n1 43636,c1(C(=O)NCC(C2CCCN(C(C3CS(=O)(=O)C3)=O)C2)(C)O)cnc2sccn12 43637,c1(C(=O)OC)cnc(Cl)[nH]c1=NC(CNc1ccc(C)c(Cl)c1)C1CC1 43638,C1(CNC(C(CC)N(C)C)=O)CCCN(C(C2(C3CCCO3)CCC2)=O)CC1 43639,C1(CNC(CCCc2ccc(C)s2)=O)CCN(C(C2CCC2CF)=O)CC1 43640,CC1C(C(=O)N(C)CC2CCCN2C(C2CC3C=CC2C32CC2)=O)=NOC1C 43641,c1(C(N(C2CCN(C(c3cnnc(O)c3)=O)C2)CC)=O)cnn2ccn(C)c12 43642,C#CCCC(O)CCNC(=O)CN(C(=O)C(C1CCC1)OC)CCC 43643,N1(C(c2nccc(CC)c2)=O)CC2CCC2(NC(c2cnc(C3CC3)s2)=O)C1 43644,N12CC(F)(F)CC1C(=O)N1C(CC(OC)C1)C2=O.c1(CO)ccccc1C 43645,C1(CC(=O)N(CCCCN(C(c2cc(C)sc2)=O)C)C)CCOC(C(C)C)C1 43646,c1(CCN(C(c2occc2F)=O)C2CC2)cccc(F)n1 43647,C(=O)(C(O)CC(C)C)N1CC(NC(C(=C(C)C2CC2)F)=O)C(C)C1 43648,CCCC(CC)C(=O)N1CCN(C(=O)CCCOc2ccc(F)c(F)c2)C(C)C1 43649,C(N=c1[nH]oc2cc(Br)ccc12)c1ccc(OC)c(OC(F)F)c1 43650,C(CC(CC)C(=O)N1CCOC(CC(N2CC(C)CCC2COC)=O)C1)=CC 43651,Cc1ncc(C(N2CC(C)(CCC(=O)N(C3CCOC3)C)C2)=O)cc1C#N 43652,c1(C(N2CCN(C(C3C(C(N)=O)C3)=O)CC2)=O)ccc2c(c1)COCC2 43653,c1(CC)csc(C(F)(F)C(=O)N(C)CCNC(c2cc(C3CC3)on2)=O)n1 43654,c1(NC(c2c(OCC)cc(C)cc2)=O)cc(Cl)c(F)cc1C 43655,c1(C(=O)OC)ccc(NC(=O)NC2(C(N)=O)CCCCCC2)nc1C(F)(F)F 43656,C1(NC(c2cc(OC)ncc2)=O)CCN(c2ccnc(C(F)(F)F)n2)CC1C 43657,C(C(C)C)(C(O)C(=O)NCC1CN(C(=O)C(C)(C)OC(C)C)CC(C)(C)O1)OC 43658,C1(CNC(CCN(C(CC(C)C)=O)C2CC2)=O)CC(C)(C)CO1 43659,C(C(C(C)C)NC(c1cn(CCNC(c2ccc(Cl)s2)=O)nn1)=O)OC 43660,N1(C(CCC(=O)N(C)C)=O)CCC2(CC1)CC2(C)C(=O)NC(C)C(C)(C)C 43661,Cc1cc(C(=O)NC2CC(O)(CNC(=O)CC3CCC(C)CC3)C2)cc(N)c1 43662,C1(NC(=O)CCc2cnc[nH]2)CC12CCN(C(=O)C=CC=C(Cl)Cl)C2 43663,C1(NC(C(C)OCCOCC)=O)CCN(C(=O)C(C)CC(C)C)CC1F 43664,N1(C(=O)Nc2cccc(C)c2C)CC(C2CN(C(=O)CN3CCCC3=O)C2)C1 43665,c1(CC)c(C(=O)Nc2cccc(-c3cn(CCC(C)C)nn3)c2)cnn1C 43666,CC1CCN(C(c2ccc(Cl)c(N)c2)=O)CC1NC(=O)CC1CC(O)C12CCC2 43667,C1(C(N(C2CN(C(C3CCCCCC3)=O)C2)C)=O)CN(S(N)(=O)=O)C1 43668,C1(NC2(c3nnnn3CCCSC)C(CC)CC2)CCCCC1(C)C 43669,c1(N)ccccc1.C12CN(C1)C(=O)CO2.CC(C)C=CC(=O)N(C)CCNC 43670,N1(C(c2c(CNC(C(CSC)(C)C)=O)cnn2C)=O)CC(C)CCC1CO 43671,C1(C(=O)NCC(C)NC(c2c[nH]nc2C(C)(F)F)=O)CCc2nnc(O)cc2C1 43672,c1(CNC(C(C)N(C=O)Cc2cccnc2)=O)cccc(C(=O)NC(N)=O)n1 43673,N1(C(CNC(C(C)(C)C)=O)=O)CCCN(C(=O)CCc2ncco2)CC1COCO 43674,C1(C)(C(N2C(CN(C)C(C3CCCN3C)=O)CCC2)=O)CCOCC1 43675,C1(CNC(CCC(=C)C)=O)CC2COCC2N1C(c1ocnc1C(F)F)=O 43676,c1(C(=O)NCC(CNC(c2c[nH]c(=NC)o2)=O)F)ccc2nccnc2c1 43677,c1(CC(=O)NC(CNC(C2N(CC)CCCC2)=O)(C)C)ccc(OC)c(Cl)c1 43678,C1(CCC)CN(C(c2cc(C)[nH]n2)=O)CC1C(=O)NCCn1cncn1 43679,c1(C(N(CCN(C)CC2(COC)C=CCC2)C)=O)nccnc1SC 43680,C#Cc1ccc(CCC(=O)NCC(C)NC(=O)CN2CCOCC2)cc1 43681,N1(C(CCCC)=O)CC(C(=O)NC(CCC)C(=O)NC)C2(CCC2)C1 43682,c1(CNC(c2n(C(CC)C)nnn2)CCCOC)ccc(N(C)C)cc1 43683,C1(C2CCCN(C(=O)C=Cc3nccs3)C2)(NC(c2c(C)ncnc2C)=O)CC1 43684,N1(C(C(CCC)OCc2ccccn2)=O)CC2(NC(=O)CC(F)(F)F)CCC1C2 43685,Cc1ccnc(C)c1NC(C1CCN(C(c2cc(Br)cnc2Br)=O)C1)=O 43686,c1(CC(=O)NCCC2N(C(c3c(CC)cco3)=O)CCSC2)c(C)nn(C)c1C 43687,O=C1CCC(C(N2CCC(CNC(=O)C(O)CCc3ccccc3)C2)=O)CCO1 43688,c1(COC)cc[nH]c1C(=O)NC(CNC(CCN(CCC)C)=O)CC 43689,c1(CNC2CCC(NC(=O)CC3CCCCO3)C2)cc(F)cc([N+](=O)[O-])c1 43690,C#Cc1cncc(C(=O)NC2CCC2NC(=O)Cc2ccc(F)c(Cl)c2)c1 43691,c1(C(=O)NC2CCS(=O)(=O)C2)ccc(S(=O)(=O)N2CC3CC3(CO)C2)cn1 43692,n1(CC(=O)NCC(C)(C)CNC(=O)C(C)(C)CF)ccc2cc(F)ccc12 43693,C(c1ccncc1C)=CC(=O)NCCC(C)NC(C(c1ccccc1)OCC)=O 43694,c1(C(=O)NC2C(NC(C(n3cc(C)nc3)(C)C)=O)CC2)cc2nc[nH]c2cn1 43695,Cc1ccc(C(=O)NCC2CC(F)(CNC(C3(C(C)(C)C)CCCC3)=O)C2)nc1 43696,c1(C(=O)NCC(CCOCC)NC(=O)CCC=C(C)C)cc(Cl)c(OC)c(Cl)c1 43697,N1(C(CC2C(C)(C)CC2)=O)CC2(CCOCC2)CC1CNC(c1csc(S)n1)=O 43698,c1(C(N2CCC(NC(CC3(C)CCCCC3)=O)C2)=O)cc(=O)c2ccccc2o1 43699,C1(C(=O)NC2(C(N(CC#C)CC3CCCO3)=O)CC2)CC1C1(C)COC1 43700,c1(C(=O)OC)cnccc1CN1CCCC1CNC(=O)C(c1ccccc1)O 43701,C(=O)(CCCCC(F)F)NC1(C)CCCN(C(c2cccc(CCC)c2)=O)C1 43702,c1(CC(=O)N(CC(O)CN(C)C(C2CC2C(C)(F)F)=O)C)ccnn1C 43703,C(=O)(CCN=c1[nH]ccs1)N(c1ccccc1)Cc1c(OC)ccc(F)c1 43704,c1(C(=O)NCC(CNC(=O)CC2CCCC2O)CO)nccc2ccncc12 43705,N1(C(CNC(CC)=O)=O)CCN2CCN(C(=O)CC3CCCC(=O)N3)CC2C1 43706,C=CCC(C)(C(=O)NC1CC(NC(=O)CCc2cc(C)n(C)n2)C1)N(C)C 43707,C(=O)(C(CC)N(C)C(c1ocnc1C)=O)NC1CN(C(CC)=O)C1 43708,C(CC(C)(C)C(=O)NCC1COCCN1C(=O)C=CC(=O)NC1CC1)OC 43709,C1(NC(C(CC=CCC)C)=O)CC2CCC(C1F)N2C(=O)C(C)(C)F 43710,C(=O)(C(C)S(C)(=O)=O)N1CCC(N(CC#C)C(c2cccs2)=O)C1 43711,C1(CNC(C(C)C2CCCC2)=O)CCCN(C(c2cnoc2)=O)CC1 43712,c1(C(=O)NC2C(NC(CCOC(C)C)=O)CC2)cnc(Cl)c(N)c1 43713,C1(NC(CCCCC=CC)=O)CN(C(C2NC(=O)OC2(C)C)=O)CC2(CC2)C1 43714,C1(C(=O)NCCCNC(CC2CCC(C)C2)=O)CC=CC(O)C1 43715,C(CNC(=O)CCCC1CCCCC1)(CC(F)(F)F)NC(CCC(C)OCC)=O 43716,C(CCC(O)C(=O)NCCCCn1ccnc1)NC(=O)CN1CC2CC2C1 43717,c1(C(=O)NC(CC)CNC(c2cnc(C)n2C)=O)cc2ccc(F)cc2nc1O 43718,c1(CC)nc(CC(=O)NC2CCCN2C(=O)C(C)NC(=O)C(F)(F)F)cs1 43719,C1(CC)CCN(C(=O)C(C)=CC(C)(C)C)C1C(N1CC(OC(=O)N(C)C)C1)=O 43720,c1(-n2cc(C(=O)NCCCCNC(C3(CC)CCOC3)=O)nn2)ccccc1F 43721,c1(OC)ccc(CNC2CCC(C(=O)O)C2)c(O)c1 43722,CON(CC1CCCCC1)C(=O)C(F)(CNC(=O)CC(C)C)C(C)C 43723,N1(C(CCC2N(C)CCCC2)=O)CC(F)(F)CC1CNC(C1CCCN1N=O)=O 43724,Cc1cc2onc(C)c2cc1NC(c1cc(C)c2c(c1)CCC2)=O 43725,O=C(C(F)C(F)(F)C(F)(F)F)NC1CCCN(C(=O)CCc2ccoc2)CC1 43726,C1(NC(c2ccc(CNC(C3OCC(C)C3)=O)cc2)=O)CCC(=O)NC1C 43727,c1(Cc2nc(CC(C(O)C(N)=O)Nc3ccc(CC)s3)on2)c(C)cccc1C 43728,N1(C(c2cn(CC)nn2)=O)CC2CCCN(C(C3CC(OC)C(OC)C3)=O)C2C1 43729,C#CCCCC(C)C(=O)NC(C)Cc1nccs1 43730,C1(NC(c2n(CCC)nc(C)c2)=O)CC2CN(C(=O)CCC(C)(C)F)CC2C1 43731,S(=O)(=O)(c1cc(C)c(Br)cc1F)N(C)CC1CCCN(C(C=C(C)C(=O)O)=O)C1 43732,C1(NC(CC2CCN(C(CC(C)(F)F)=O)CC2)=O)CCCCCC1O 43733,N1(CC(=O)NC(CC)(C2CC2)C2CC2)CCC(N2CCC(O)CC2)CC1 43734,c1(C(=O)NC23CC(CNC(CCC(C)SC)=O)(OCC2)C3)ccn2cnnc2c1 43735,N(C(=NCCC(=O)NC)NCC1CC2C=CC1CC2)C1CC(C#C)C1 43736,C(=O)(CCCCC(C)(C)OC)NC(C)C(C)NC(c1c(OC)c(F)ncc1)=O 43737,C(c1cc(F)cc(F)c1)=CC(=O)NCC(C(C)C)NC(C(C1CC1)SC)=O 43738,N1(C(c2ccn(CCC)n2)=O)CCC2(CCN(C(c3cc(N)ccc3C)=O)C2)C1 43739,c1(-n2ccnn2)c(C(F)(F)F)nc2ncccn12.N1(CCN(C)CCO)CCNCC1 43740,c1(NC2(CNC(CSc3c(C)cccc3)=O)CCCC2)c(Cl)cccc1[N+](=O)[O-] 43741,N1(C(CCC2CC(NC(c3c(C)n(C)nn3)=O)C2)=O)CCC(N(C)C)C(C)C1 43742,C(=O)(C(F)(F)CN)NCC(Cc1ccccc1)OCC 43743,c1(C(=O)NCC(CC)(CC)NC(CCC#CC)=O)ccc2c(O)ncnc2c1 43744,c1(C(NOCC(=O)N(C)CC2CC(=C)C2)=O)ccc(F)cc1C 43745,c1(CNc2cccc(P(C)(C)=O)n2)ccc2cc(Cl)ccc2c1 43746,C1(CNC(C(C=CCCC)O)=O)(NC(c2cc(O)cs2)=O)CCCCC1C 43747,N1(C(c2c(CNC(CN3C(C)CCC3)=O)cnn2C)=O)CC(CO)C2(CC2)C1 43748,N1(C(C(CNC(C(C(C)C)OC)=O)(C)C)=O)CC(=O)N2CCCC2C1 43749,C(=O)(CC(CNC(=O)CC1(C)OCCO1)C1CCC1)N(CC(C)C)C 43750,C=CCC(CNC(=O)C(=O)C1CC1)CC(C)C(C)(C)C 43751,Cc1ccc(O)cc1C(N1CCN(C(=O)Cc2ccon2)C(C)C1)=O 43752,CC1(C)CCN(C(=O)C(=O)NCCCOC)CC1.C(CCO)NC(C1CC1)=O 43753,C=CCCCCCCCC(=O)NCC(C1CC1)NC(=O)Cn1cc(C(C)=O)nn1 43754,C1(CNC(CSCC(=O)OC)=O)CN(C(=O)CC2CCCN(C)C2)CC1C 43755,c1(C(N2CC(CNC(CC=CCC)=O)C(F)(F)C2)=O)cccc2nc(Cl)cn12 43756,S(=O)(=O)(c1ccc(NC(C)C)cc1)N(C(=O)Nc1ccc(C(C)CC)nc1)CC 43757,N1(C(C2(CC)CCOCC2)=O)C(C(=O)NC2CCC(OC)C2)C2CC(O)C1C2 43758,c1(CC(N2CCN(C(c3c(C)ccnc3)=O)C(CF)C2)=O)cccc([N+](=O)[O-])c1 43759,c1(CC(N2CC(C)(NC(CS(=O)(=O)NCC)=O)C2)=O)ccc2c(c1)ncn2C 43760,c1(C(CNC(=O)NCc2c(C)nc(CC)o2)(C)C)cccc(Br)c1F 43761,c1(OC)nc(C(=O)Nc2cccc(OCc3ccncc3)c2)ncc1F 43762,C1(O)(CN(C(CC=C=C)=O)C)CCN(C(=O)CC2(C)CCOCC2)C1 43763,C1(O)(C(=O)NCCN(C(=O)C(c2cccc(C(F)(F)F)c2)(C)C)CC)CC(F)(F)C1 43764,N1(C(c2n(CC(C)C)ncc2)=O)CCCCCC(NC(=O)C(C)n2ccnc2)C1 43765,N#Cc1ccc(F)c(C(N2CCC3CCC23CNC(c2csnc2Cl)=O)=O)c1 43766,CC1CCN(C(=O)C(n2cc(C(O)C(C)(C)C)nn2)C)CC1 43767,c1(C(=O)NC2(CNC(=O)CC3(C(F)F)CC3)CCOC2)cc(O)cc(Cl)c1 43768,c1(CC(=O)NC2CCC(NC(C3C(C)OC(=O)N3)=O)CC2)nc2ncccn2n1 43769,C1(CNC(COC(CC)C)=O)CCCC1NC(=O)C=Cc1cncs1 43770,CC1CN(C(c2cncn(C)c2=O)=O)CCC1NC(c1cc(C2CCC2)[nH]n1)=O 43771,c1(OCC)nccc(C)c1NC(=O)CCC(C)NC(C1CCC(=O)NC1)=O 43772,c1(C(=O)NC2CCCC(NC(C(CC)SC)=O)C2)cccc2oc(C)nc12 43773,C(CC(C)C(=O)N(C(C)CNC(C1(C)SCCCS1)=O)C)=CC 43774,C1(NC(C(C)C)=O)CCC2(CC1)CCN(C(C13C=CC(CC1)C3)=O)C2 43775,c1(C(N2CC(CNC(COCC)=O)(CO)C2)=O)ccc(C)cc1C 43776,C(=O)(CC(C)C(F)F)N1CCCC(NC(c2nc(COC)sc2)=O)C1 43777,c1(CCC)cc(C(=O)NC2COCC2CNC(C2CC2OC)=O)n(C)n1 43778,c1(C(=O)NC2(C)CCN(C(=O)Cc3ccc(O)c(O)c3)C2)ccc2nn[nH]c2c1 43779,Cc1c(C(=O)N(C)CC2CCN(C)C2=O)sc2nc(C(F)(F)F)ccc12 43780,N1(C(CC=CC)=O)CC2CC2(CNC(=O)NC)C1 43781,c1(NC(C(CC)SC)=O)nc(C(=O)OCC(=O)OC)nc2ccccc12 43782,c1(CN2CCC(C(=O)Nc3ncc(F)s3)C(O)C2)c(F)cc(Br)cc1Br 43783,C(CCO)(C(=O)O)NC(c1ccc(Cn2cc(-c3ccsc3)nn2)o1)=O 43784,n1(CC)cnc2nc(N(C)CC3CCCN(C)C3)nc(NCCc3cn[nH]c3)c12 43785,Cc1cc(C(N2CCC(CCNC(C3CC(F)(F)C3)=O)C2)=O)cnc1C(F)(F)F 43786,C12(CC(=O)NCC(CC=C)NC(=O)COC3CCCC(C)C3)COC(CF)(C1)C2 43787,Cc1cc(Cl)c(C(=O)NCC2C=CCN2C(=O)CNS(C)(=O)=O)s1 43788,CC(N=c1ccnc(NCCOc2ccc(F)cc2Cl)[nH]1)c1nncs1 43789,CC1=NOC(CC(=O)N(C(C)C(=O)NCCCN=[N+]=[N-])CC)C1 43790,c1(C(C)NC(N(C2CCNCC2)CCCC)=O)cc(C)ccn1 43791,c1(C(C)NC(C(C2CCCC2)NC(c2c(C)cco2)=O)=O)nccc(O)n1 43792,c1(C(N2CCC(COC)(NC(C3CC=CCC3)=O)C2)=O)ccc(OC)c(Cl)n1 43793,C1(C(N2CCOC(C3CN(C(=O)C=C4CCCCC4)C3)C2)=O)(CC)CC(C)(C)C1 43794,N1(C(c2ncc(C)cc2F)=O)CC2CCC(N(C)C(C3CCCC3O)=O)C2C1 43795,C1(CNC(C2(OC)CCC2)=O)CC(C)(C)CN1C(=O)CC1CC(OC)C1 43796,C(=O)(CCS(C)=O)NCCN(C(C(C)N(C(C)=O)C)=O)CCc1ccccc1 43797,C1(NC(C2C(CNC(C(COCC)C)=O)C2)=O)CNC(=O)C1(C)C 43798,C(CCCCC(=O)N(C)CCOCCNC(C1CCC(C2CC2)C1)=O)SC 43799,c1(OC2CCN(C(=O)NCc3cc(Cl)nc(Cl)c3)C2)ccc(C)c(COC)n1 43800,C(=O)(CC(C(F)F)c1ccccc1)N(C)CCNC(c1cc(F)n[nH]1)=O 43801,CC1(C)C(CNC(=O)NCC2(c3nn[nH]n3)CC2)CC1O 43802,c1(CCC(N2CC3CCC(C2)N3C(=O)COCCF)=O)cccc2ccccc12 43803,N1(C(C(C(C)C)OCC)=O)CC2CCC1C(NC(=O)Cc1n[nH]c(C)n1)C2 43804,N1(C(c2c(C(C)C)onc2)=O)CCC2(CC(C(=O)NCCN(C)C)C2)C1 43805,C1(OCC(N2CCC(C(C)(C)NC(c3cc(F)c[nH]3)=O)C2)=O)CCCCCC1 43806,C1(NC(Cn2nnc(=N)[nH]2)=O)CCCCCN(C(C23CCN(CC2)CC3)=O)C1 43807,c1(OC)c(C(=O)NCC=CCNC(=O)C(CN(C)C)N(C)C)cc(Cl)cc1C 43808,N1(C(c2ccc(C)cc2)C(=O)NC(CC)(C)C)C2CCC1CC(F)C2 43809,c1(NC(C2CCCN2C(c2cc(Cl)c(Cl)cn2)=O)=O)cc(F)cc(Br)c1 43810,CC1CN(C(=O)COC2CCN(C(=O)C=CC3CCC3)C2)CC(C)(C)O1 43811,Cn1nc(C2CCOCC2)cc1C(=O)NC1CN(C(C2COC(=O)O2)=O)CC1F 43812,c1(C(=O)NC2CC(CNC(CN3CC(C)C3)=O)C2)ccnc2c1cnn2C 43813,N1(C(CC(=O)OC)=O)CCC2(CCC2CNC(=O)C(O)C2CCC2)CC1 43814,N1(C(=O)Cc2cc(F)cc(Cl)c2)CCC2OCCN(C(=O)C=CCO)C2C1 43815,C1(CNC(CC2N(C(C)=O)CCCC2)=O)CC2CCC(C1)N2C(=O)COC1CC1 43816,C1(C(N(C)CCC2OCCO2)=O)CCN(C(c2cc(Cl)cnc2F)=O)CC1O 43817,c1(C(CC(CNC(C(C)(C2CC2)OCC)=O)(C)C)=O)cc(SC)nn1C 43818,C1(C(N(CC)CC2CCCCN2C(C2CC2COC)=O)=O)OCCOC1(C)C 43819,CS(=N)(=O)CCNC(=O)C(Cc1cc[nH]n1)NC(=O)CC1CCCOC1 43820,N1(C(C=C(CCC)C)=O)C2CCC1CN(C(c1sc(Cl)cc1Cl)=O)C2 43821,CC1CN(C)C(=O)C2=C1N(c1ccccc1)C(=S)NC2c1ccc2c(c1)CC=C2 43822,C(=O)(C(CCC)OCC)N1CCC(C(N2CC(C(CC)C)C2)=O)C1 43823,C1(CC(=O)NC2C(NC(CSCC=C)=O)C2)OCCCC1(C)C 43824,C(=O)(C(O)C(F)(F)F)NC1CC2(C(C(N3CC(C)(OCC)C3)=O)C2)C1 43825,N1(C(C)=O)CC2CC1CN2C(C12CC1CCN2C(=O)C(N1CCCCC1)C)=O 43826,C1(C(=O)NCC#CCNC(c2cc(C)n(C)c2)=O)CC(c2cccc(F)c2)=NO1 43827,c1(C(=O)NCC2C(C(N3CCC(CC#C)C3)=O)C2)cccc2nccn12 43828,c1(CC)ccc(C(=O)NC2CCC2NC(c2cnc(O)cc2OC)=O)c(Cl)c1 43829,c1(C(=O)NC(c2ccccc2)CCC)ccc(N2CCC(N)CC2)cc1 43830,O(NC(=O)C(C)(C)S(C)(=O)=O)C(CC(C)C)C(=O)N1CCC(C(C)C#N)CC1 43831,n1(CC(=O)NCCN(C2CCCC2)C(=O)CNc2ccccn2)cnnc1O 43832,c1(OC)ccc(NC(=O)NC2CC2c2ccncc2)cc1Br 43833,N1(C(CC(CC)OC)=O)CCCC2(CCN(C(=O)Cc3ncn4c3CCC4)C2)C1 43834,C1(C(N(CC#C)C)=O)CC12CCN(C(=O)CN1CC(C)(C)C1)C2 43835,C(c1cccnc1)=C(C)C(=O)NC1C=CCCC1C(=O)NC12CC(C1)C2 43836,C1(NC(CC2(C=C)CC2)=O)CN(C(=O)CC2CC=CCC2)Cc2nccn2C1 43837,CCCCCC(F)C(=O)N(CC(N1CC(O)CC1COC)=O)CC1CC1 43838,c1(C(N2CC3C(NC(c4ncn(C)c4)=O)(C3)C2)=O)ccc2[nH]nc(O)c2c1 43839,C1(F)(CNC(C2C(CC(C)(C)C)C2)=O)CCN(C(=O)CS(N)(=O)=O)C1 43840,CC(=O)CCN=C(NCC(C)(C)Cc1cccs1)NCC1(OC)CCCC1 43841,Cc1nn(CC(N2CCC(C(C)NC(c3ccoc3Br)=O)CC2)=O)cc1Cl 43842,N1(C(C=CC)=O)CCC2(CC1)CN(C(=O)C(C)n1cccn1)CC2CO 43843,c1(C(N2CCC(CNC(C3C(=C)C3)=O)CC2C)=O)ccc2nnc(O)n2c1 43844,C1(CNC(CC2C(OCC)COCC2)=O)CN(C)CCN1C(C1CNC(=O)N1)=O 43845,C(=O)(C(C)(C)C1CCN(C(=O)C(Cl)Cl)C1)NC(c1cn(C)cn1)C 43846,C(=O)(C(S(C)(=O)=O)C1CC1)NCC(C)CNC(C1(C)CCSCC1)=O 43847,CC1COC2(CCC2)CN1C(=O)Nc1ccc(C2CCN3CCCCC23)cc1 43848,N1(C(CC(C=C)(C)O)=O)CCC2(C1)CN(C(=O)COC(C)(C)C(F)(F)F)CCO2 43849,C(=O)(C(CC(C)C)NC(=O)OC)NCC(C1(OC)CCOCC1)(F)F 43850,C1(C(N2CC(NC(Cc3cc(C)n(C)n3)=O)C(C(F)F)C2)=O)CN2CCN1CC2 43851,c1(CCC(=O)NC2CCN(C(CCC(=C)C)=O)C2C)ccc(Br)cc1OC 43852,CCCC(C(=O)N1CCC(C)C1CNC(c1ccc(C)cc1)=O)S(N)(=O)=O 43853,c1(C(C)C)nnc2cc(N3CCC(C(C)NC(=O)C(C)C(C)O)C3)ncn12 43854,C1(O)(CCNC(CC2(C=C)CC2)=O)CCN(C(c2cnc(C3CC3)s2)=O)C1 43855,c1(C(C(=O)OCC2CCC(F)(F)C2)OC)cccc(CC(F)(F)F)c1 43856,C(=O)(C1=CCC(C)(C)CC1)N(CCCNC(=O)Cc1nocc1C)CC 43857,c1(CNCC(O)CC(F)(F)F)c(O)ccc(F)c1F 43858,CCC(=O)CCC(=O)N1CCOCC(CNC(c2scnc2COC)=O)C1 43859,C(CCCCC(=O)NCC1CCN1C(c1sccc1Br)=O)OCC 43860,C1(N(C(=O)NC(CC)Cc2ccc(Cl)cc2)C)CCNCC1O 43861,N1(c2cc(NCC(CC)N(C)C)ncn2)CCc2c(F)cc(F)cc2C1 43862,C1(C)(NC(CCCNC(C)=O)=O)CCC(NC(C2(O)CCSCC2)=O)CC1 43863,C(=O)(C1CC(=O)c2ccccc21)N1CC(N(C(=O)C2=CCOC2)C)C(O)C1 43864,CN1CCC(N(C)C(C2CCN(C(=O)CCC3CCCN3C)C2)=O)C1 43865,CCC(C)C(C(=O)NC1CCN(C)CC1C)N(C(=O)CCc1ccc[nH]1)C 43866,Cc1ccc(C)c2[nH]c(C(=O)NCC3CCC3NC(C3CCS(=O)CC3)=O)cc12 43867,c1(C(=O)NCCCCNC(=O)CCc2cncnc2)c(Cl)ccc2c1OCO2 43868,C1(CC2CC(NC(CCNC(C)=O)=O)C2)CCCN(C(=O)C(=Cc2cn[nH]c2)C)C1 43869,c1(C(=O)NC2(CC=C)CN(C(=O)C=CCC)C2)cc2c(s1)COCC2 43870,C1(C)(C(=O)OC)CC(C(=O)NCC(C)N(C)C(c2coc(Cl)c2)=O)C1 43871,c1(C(N2CC(N(C)C(C3(c4cccs4)CCC3)=O)C2)=O)cnn(C)c1N 43872,C(CCCCCNC(C1CCNC12CC2)=O)N(c1ccccc1)C 43873,c1(OC)ccc(CN(C)CC2CCCN(C(C3CCCC(C)C3)=O)C2)cc1C 43874,C1(C)(CC)CC(C(=O)NC(c2cccnc2)c2ccccn2)CCO1 43875,CCCCCC(F)C(=O)NC(C1CCCCCC1)CNC(c1cncn1C)=O 43876,c1(C(=O)OCC)ccc(C(C)(F)F)nc1O.c12cccc(c1)CS(=O)(=O)NC2=O 43877,C1(C(=O)NCCC2(C)CCN(C(c3ccc(C)nn3)=O)C2)CCCC(C)(C)C1 43878,c1(C(=O)NC2C(C(C)C)CN(C(c3nn[nH]c3Cl)=O)CC2)cccc2nccn12 43879,c1(C(=O)NCC2(C(N3CC(n4cnnc4)C3)=O)CCC2)ccnnc1 43880,c1(C(=O)NC23CC(NC(CC(CCC)C)=O)(C2)C3)cc2ccc(O)nc2s1 43881,C(=O)(C(F)(F)C(O)C(C)C)NCCC1=CCN(C(c2cccc(SC)n2)=O)CC1 43882,c1(-c2ccc(OC)cc2)cnc(N2CCS(=O)C(C)C2)cc1C 43883,C1(NC(C=CC(C)C)=O)CC(NC(=O)Cc2ccccc2)CC1O 43884,N1(C(CNC(CCC(C)C)=O)=O)CCC2(NC(=O)CC(C)(C)N(C)C)CC2C1 43885,C1(OC)CC(CNC(c2nnc(C)s2)=O)N(C(C2CCC(C)S2)=O)C1 43886,C1(C(=O)Nc2cccc(-n3ccnc3)c2)CC2CN1CC2 43887,N1(c2nnc(C)o2)CCC(C(C)NC(C2C3COCC23)=O)CC1 43888,c1(OC(=O)CN2CCCC2C(=O)NCC2CC2)cncc(Br)c1 43889,CC(C(=O)NC1C2CCC1N(C(C1(c3cccc(Cl)c3)CC1)=O)C2)S(C)(=O)=O 43890,c1(C(N2C3CC(NC(C(=O)N(C)C)=O)C(C3)C2)=O)n[nH]c2ccc(Cl)cc12 43891,Cc1cnc2cccc(C(N3CCC(NC(=O)CCc4cccnc4)C3)=O)c2c1 43892,C12COCCN1C2=O.C1(NCc2ccc(C(=O)OC)s2)CC(=O)N(C)C1 43893,C(=O)(C(C)(CO)CO)N1CCCC(C(=O)Nc2c(C(C)=O)cccn2)C1 43894,c1(C(N2CCC(CC)(NC(c3cc(O)n(C)n3)=O)C2)=O)ccc2nccnc2n1 43895,C(CCC(N)=O)(C(=O)NCC1CCCCN1C(=O)C(O)C(F)F)NC(C)=O 43896,Cc1cccn(CC(=O)NCCC2CN(C(C3CC(O)C3)=O)CCO2)c1=O 43897,C1(NC(=O)NC2C(OC)CCCC2)CCS(=O)(=O)C(C)(C)C1 43898,N1(C(CN(CCC#C)C)=O)CC(NC(C2CC(n3ccnn3)C2)=O)CCC1C 43899,N1(C(c2cncnc2)C(=O)NCCOCC)CCC(O)(CN(C)C(C)C)CC1 43900,c1(C(N2CCC(CNC(C=CC=CCC)=O)C(C)C2)=O)cc2c(cn1)CCCC2 43901,O=S(=O)(c1cnccc1N1C2CCCC1COC2)NCc1nc(CO)cs1 43902,C1(F)(CNC(C(CC2CC2)OC)=O)CCN(C(=O)CC2CC(=O)C2)C1 43903,C1(c2n(C)ccc2)COCCN1C(=O)CCC1CCCCO1 43904,c1(C(N2CCN(CC3CN(C(CCC#C)=O)C3)CC2)=O)cc(C)cc(Cl)c1N 43905,CC(CC(=O)NCC1CC12CC2(F)F)C(C)(C)NC(C12CC(F)(C1)C2)=O 43906,c1(C(=O)NCC(C)(C)NC(=O)Cc2ccoc2)ccc(-c2ccccc2)s1 43907,N1(C(N)=O)CCCC(CC(=O)NC(CC)Cc2ccc(I)cc2)C1 43908,c1(C(=O)NC2CC(C)N(C(c3cc4cccnn4c3)=O)C2)ccc2nonc2c1 43909,c1(C(N(CC(=O)NC(C)(C)C)C)=O)ccc(NCC2(CO)CC(F)(F)C2)cc1Cl 43910,CC1(C)C(CC(=O)NC2CCC(NC(c3coc(Cl)c3)=O)CC2)CC1O 43911,Cn1cc(S(=O)(=O)CCNC(=O)C(c2ccn(C)c2)N)cn1 43912,C(C(C)(C)C#CC(=O)NCC1CSCCO1)NC(CN1C(C)CCCC1C)=O 43913,C=Cc1cncc(C(c2nnnn2C2CCCC2)NS(=O)(=O)C(C)C)c1 43914,C1(C#CC(=O)NCC2CC2CNC(=O)CCCCN(C)C)(CC)CC1 43915,C1(C(=O)NCC(S(C)(=O)=O)CNC(C2CCCCC2O)=O)OCC2COCCC12 43916,C(C(C)(CC(C)C)NC(=O)CC1(CSC)CCCCC1)NC(CCNC(=O)NC)=O 43917,C(=O)(C(F)C(=O)NCC1CCC(NC(=O)C(C)(C)OCCOC)CC1)OCC 43918,N(C(=NCCC(C)=O)NCC1CC(C)(C)C1)Cc1cccc(OCC#C)c1 43919,C1(NC(CC2N(C(Cc3cnc(C)o3)=O)CC2)=O)CCCC(O)CC1 43920,c1(C(=O)NC2CN(C(CCOCCOCC)=O)C(CO)C2)n[nH]c(C)c1[N+](=O)[O-] 43921,c1(C(=O)NC(CNC(CSC)=O)C2CCC2)cnns1 43922,C(C(C(=O)NNC(=O)CC1(OCC)CCC1(C)C)n1cc(C2CC2)nn1)OCC 43923,C1(O)(CCNC(c2n(C)nnc2)=O)CCN(C(c2c(Br)ncn2C)=O)C1 43924,Cc1cc(C(=O)NCC(C(C)(C)C)NC(=O)Cc2cccc[n+]2[O-])ccn1 43925,C(=O)(C1CCCc2c1ncn2C)N1CC(NC(c2c(C(C)C)occ2)=O)C(O)C1 43926,C1(N(CC(=O)NC(CNC(=O)COC2CCCC2)C2CC2)C)C=CCCC1 43927,C1(OCC(=O)NCC(CNC(c2ccccc2Br)=O)OC)CCCOCC1 43928,N1(C(C2(C(C)(C)OC)CCCC2)=O)CC(C)CN(C(=O)CCN(C)C)C(C)C1 43929,c1(C(N2C(C(=O)NC(C3CCCCC3)CC)C(O)CC2)=O)ccccc1[N+](=O)[O-] 43930,Cn1c(C(=O)NC2C=CCC2)ccc1C1COCCN1C(c1cnc(Cl)s1)=O 43931,c1(C(=O)NC2CCN(C(c3cn(CC)nc3)=O)C23CC3)cn2c(C)cccc2n1 43932,C1(CNC(CC2CCCN(C(C)=O)C2)=O)CN(C(c2cnn[nH]2)=O)CC(C)(C)O1 43933,c1(SCC(N2CCC(NC(C(CC)(C)F)=O)C2)=O)ccc(Cl)cc1Cl 43934,c1(N2CC3CC(NC(C4=C(C)OCCS4)=O)C3C2)nc(Cl)nc(C(C)C)c1C#N 43935,N1(C(C(CCCC)CC)=O)CC2CCC(C1)C(NC(c1n[nH]c3c1COC3)=O)C2 43936,C1(CC(=O)NCC2CCN(C(C3CC4(CSC4)C3)=O)C2)CC2CCC1C2 43937,Cc1cccc(C(=O)NCC2CCC2C(=O)NC(C)(C)CNC(N)=O)c1 43938,C1(CN(C(C=CC(=O)N(CC(C)N(C)C)C)=O)C)CCCC1C 43939,CCC(CCC(=O)N1CCCCC1CC(N)=O)NC(c1cc(C)ncn1)=O 43940,C1(CNC(COC(CC)C)=O)C2CN(C(C3(COC)CC3(F)F)=O)CC12 43941,C=Cc1ccc(C(N2CCCC(C)(CNC(c3c(Cl)noc3C)=O)C2)=O)cc1 43942,CC1(C)C2CC(C(N3CC(C(C)(C)O)(CNC(C4CCS(=O)CC4)=O)C3)=O)CC12 43943,CCC(C)C(C(=O)NCCN1CCN(C(C2CC(OC)C2)=O)CC1)NC(=O)OC 43944,c1(C(N(C2CC2)CC2N(C(c3c(CC)c[nH]n3)=O)CCC2)=O)cc(O)nc(C)n1 43945,CC(CNC(C1CC1Cl)=O)C(F)C(=O)NCCN1CCOCC1 43946,c1(C(=O)NC(C2CN(C(=O)Cn3ncccc3=O)C2)C)ccnc(S)c1 43947,C1(CNC(CCC=C)=O)CN(C(=O)C(CCC)OCC)CCCO1 43948,c1(C(=O)NCC2CN(C(c3c(C)coc3)=O)C(C)(C)C2)cc(P(C)(C)=O)cs1 43949,C(C(N=c1cnc(F)c[nH]1)C1CCCC1)Oc1c(Cl)cccc1F 43950,N1(C(CCCCCSC)=O)CCC(C2CC2)C1C(n1cnnn1)C.C1(O)CC2(CCC2)C1 43951,C(C(CC(=O)N1CC(O)CC1CNC(c1ccn(C)c1)=O)CC(C)C)NC(C)=O 43952,CS(=O)C1(CNCC2CCCC(Nc3ccnn3-c3ccc(F)cc3)C2)CCC1 43953,c1(C2(C)CN(C(=O)Nc3nccc(N4CCCC4)n3)C2)ccccc1Br 43954,C1(CC(=O)NCC(CC)N(C)C(c2cccc(CCO)c2)=O)CCCC(=O)C1 43955,c1(C(=O)NC2(C(N3CC(c4ccccc4)C3)=O)CCN(C)C2)ncc(F)cc1F 43956,C1(C(=O)NCC2CC2NC(=O)C(F)CC2CCC2)(OC)CCSCC1 43957,c1(C(=O)N(C2CCCCCC2)Cc2ccnnc2S)c(F)cccc1F 43958,c1(CC(=O)NC2CCN(C(COCCC)=O)C2)ccccc1CS(N)(=O)=O 43959,Cc1cc(C(N2CC3(CC(NC(c4cnn(C)c4Br)=O)C3)C2)=O)ccc1F 43960,C1(COC)CN(C(c2nccc(Br)c2C)=O)CCN1C(C1CC1CF)=O 43961,c1(C(=O)NC2C(NC(c3c(C)cc(C(F)F)o3)=O)CC2)n[nH]c2c1COC2 43962,Cc1nc2ccccc2n1CC(=O)NC1(C)CC(NC(=O)C2=CCCC2)C1 43963,C1(CC#CC)NC(=O)N(C(c2nn(C)cc2O)C)C1=O 43964,C1(C(N2CCC(C#N)C2)=O)(CC)CCN(C(=O)COC(C)=O)C1 43965,c1(C(C(=O)NC2CCC2)N(C23CC(C2)C3)CC)cncc(Cl)c1 43966,CC1C(NC(=O)CS(N)(=O)=O)CCCN1C(c1cncc(C(C)(F)F)c1)=O 43967,C1(C(C)C)(C(N2CCC(C)(F)C2)=O)CCCN1C(=O)CCn1cccc1 43968,N1(C(C2(NC(=O)C3=CCCC3)CC(CO)C2)=O)CCn2nncc2C1 43969,c1(CSC)cc(C(=O)NCC=CCNC(C2CCN(CC(C)C)C2)=O)ccc1F 43970,N1(C(CCN(C(C(CC=C)CC)=O)C(C)C)=O)CC(C2CC2(F)F)C1 43971,C(CC1CCC1)(C(=O)N(CC(C)NC(=O)Cn1cnnc1O)C)NC(C)=O 43972,NS(=O)(=O)c1ccc(C(=O)NCC2CCCCC2NC(=O)CC2NC(=O)NC2=O)o1 43973,Fc1cc(OC(F)(F)F)ccc1Nc1cncnc1 43974,C12(CNC(C(CNC(=O)C#CC(C)C)OC)=O)CCC(F)(CC1)C2 43975,C(=O)(C(C)P(C)(C)=O)NCC(CCOC)NC(c1ncccc1CSC)=O 43976,C1(C(C)NC(=O)C(OC)OC2CC2)CCCN(C(=O)OC(C)(C)C)CC1 43977,C(CC(C(=O)N1CC(C)(CO)C1)NC(=O)CCC1OCCO1)OCC 43978,c1(C(N2CCC(NC(C(CCSC)(C)C)=O)C(C)C2)=O)cc([N+](=O)[O-])cc(C)n1 43979,C(CC1=CCN(C(c2cnc(OC(C)=O)s2)=O)CC1)N(C(c1cnn(C)n1)=O)CC 43980,C1(NC(c2cc(CC)cc(F)c2)=O)CS(=O)(=O)CC1N1CCOCC1 43981,c1(C(=O)NCC2(F)CCC(NC(CC(CC)OC)=O)C2)c(C)nc(O)nc1C 43982,Cc1c(C(=O)NCCNC(C2OCCC2C(F)(F)F)=O)c(=O)oc2ccccc12 43983,Cc1cc(C#N)ccc1C(N1CCC(NC(=O)CCCc2ccc3c(c2)OCO3)C1)=O 43984,c1(CC(N2CCC(NC(CNS(NC)(=O)=O)=O)(CF)C2)=O)cc(F)cc(Cl)c1 43985,N1(C(C(C)(C)NS(C)(=O)=O)=O)CC(CNC(c2cnc(Cl)cc2N)=O)C(C)(C)C1 43986,C12(CNC(=O)CC3CC=CCC3)CCCC1N(C(=O)C=Cc1cccnc1)CC2 43987,C1(C(N2CCC(CCNC(C=CC(=O)N(C)C)=O)C2)=O)CC1C1CCCC1 43988,N1(CC(=O)OC(C(c2ccc(CC)cc2)=O)C)C(=O)c2cccnc2C1=O 43989,N1(C(C2(C)CC2Br)=O)CC2(CCCC(CNC(C3CCCO3)=O)O2)C1 43990,S(=O)(=O)(c1ccc(Br)cc1NCc1ccc2c(c1)CN(C)C2)NC1CC(CC)C1 43991,C1(C(C(=O)NCCCN(C(=O)C(c2cccnc2)OC)C)OC)CCCCCC1 43992,c1(C(=O)NC(CNC(c2c(C)ccc(SC)c2)=O)C2CC2)ccc2c(c1)CCO2 43993,C1(C(N2C(CNC(CSCC=C)=O)C(CC)CC2)=O)CCN2CCC1C2 43994,N1(C(=O)NCC)CCCN(C(CC2CCCC2)C(=O)NC2(C)CC2)CC1 43995,C1(NC(C(C)=C(C)C)=O)CC(NC(c2cnn(C)c2N)=O)CC1O 43996,C1(CN(C(CSCC(C)=O)=O)C)CCCCN1C(=O)Cc1csc(S)n1 43997,C1(NC(c2cn(CCC)nn2)=O)CCN(C(=O)C(c2ccc(F)cc2)CC)CC1 43998,C(=O)(C1COc2ccccc21)N(C1CCCN(C(C2(CF)COC2)=O)C1)C 43999,c1(C(C)NC(c2n(CCCOC)nnn2)c2cc(OC)ns2)cccc(OC)c1 44000,CC(C)(C)C(CNC(C1CCC(O)C1)=O)NC(c1occc1-c1ccccc1)=O 44001,C(=O)(CCC(=O)NC1CC(CNC(C2CSCN2C(C)=O)=O)C1)NCC 44002,c1(CN=C(NC(C2CCOCC2)C)NCc2cccs2)cnn2cccnc12 44003,C(=O)(C1=NN(C)C(=O)CC1)N1CCCC(CNC(c2c(C)cccc2C)=O)CC1 44004,C(C(=O)N1OC2C=CC1CC2)(C1CCOC1)NC(C1C=CCS1)=O 44005,c1(OC)ccc(CC(=O)NCCOCCNC(c2cc(Cl)ccn2)=O)nc1 44006,NC1C2CCC1N(C(c1ccc(C(F)C(F)(F)F)cn1)=O)C2 44007,c1(C(CNCC23OCC(C(C)C)(C2)C3)O)ccc(S(C)(=O)=O)cc1 44008,c1(C(=O)NCC(C)(C)NC(c2c(CC)n(C)cc2)=O)oc2ccc(C)cc2c1C 44009,c1(C(N(C2CN(C(c3ccc(CO)o3)=O)C2)C)=O)n[nH]c2c1CC1CC21 44010,C(=O)(C(CCc1ccc(F)cc1)C(C)(C)C)OC.C12CC1C(=O)N2CC=C(C)C 44011,c1(SC)ccc(C(=O)NCC(C(C)(C)C)NC(C2CCCCC2)=O)c(Cl)c1 44012,c1(CC(=O)NCC(CN(C(c2cncnc2)=O)CC)(C)C)ccc2ccoc2c1 44013,c1(C(N2C3C(CNC(C(C(=C)C)(C)C)=O)C(C3)C2)=O)c([N+](=O)[O-])cnn1CC 44014,CC1=C(C)CC(C)(C(=O)NC(C2CCCC2)CNC(c2cc(O)cs2)=O)CC1 44015,O=C(C1=CCCCC1)N(CCC(=O)NCC(c1cccnc1)O)C1CC1 44016,S(=O)(=O)(c1ccc(N2CCn3ncnc3C2)c(C#N)c1)NCC(=C)c1ccccc1 44017,C1(C)(NC(COCCCOC)=O)CCC(NC(=O)Cc2ccc(F)c(Cl)c2)CC1 44018,C=CC(C)CC(=O)NC1CC(CNC(c2ccsc2-n2cnnn2)=O)C1 44019,CC(C)C(CNC(c1cnn2c1OCC2)=O)C(=O)NCCCc1cnccn1 44020,n1(CCCC)nc(C)c(C(=O)N(CCCNC(=O)COCCF)CC)c1Cl 44021,C1(NC(C2(CCCC)CCC2)=O)CCN(C(=O)C(C)(C)c2ccns2)CC1CO 44022,c1(C(N2CCC(CC(=O)Nc3n[nH]c(O)n3)CC2)=O)cnn2c1CCC2 44023,C1(C(=O)NCCSCC(=O)NC(C#C)CC2CCC2)CN(C)CC(C)O1 44024,N1(C(c2cc(C)sc2)=O)CCN(C2CCCN(C(=O)CCNC(N)=O)C2)C(=O)C1 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44042,Cc1nc(-c2cc(N(C)C)cc(F)c2)ccc1C(=O)NCc1cc(F)cc(F)c1 44043,CC1CCN(C(=O)C2=CCCCC2)CC1CNC(=O)C=Cc1ccoc1 44044,Cc1cc(N(C)Cc2ccccc2C)nc(NC2CC2F)n1 44045,C#CCC(C)(C)C(=O)NCCCN(C)C(C1CC1C#N)=O 44046,N1(C(c2c(C)nns2)=O)CCCC(C(=O)NCc2ccc(N(C)C)cc2)C1 44047,c1(C(=O)NCC(CNC(c2ccn(CCC)n2)=O)OC)nnn(CC)c1C 44048,c1(-c2ccc(C(=O)OCC)cc2)ccc2c(n1)CCC2=O 44049,c1(C(=O)NC2CN(C(C3CC3(Cl)Cl)=O)CC2C(F)F)oc2ccccc2c1CO 44050,n1(CC)c2ccccc2c2cc(CN3CC(C)C3(C)C)ccc12 44051,Cn1ncc2c1CCN(C(=O)OC(C)(C)C)C2C(N)=O 44052,C1(O)(C(=O)NC2CC3(C(NC(c4c(C)c(N)ccc4)=O)C3)C2)CCCC(C)(C)C1 44053,C1(N=c2cc(Br)n(C)[nH]2)(c2n(CC(=C)C)nnn2)CC1OC 44054,c1(C(=O)NCC(C)O)cc2cc(-c3cn(C)c4ncccc34)ccc2oc1=O 44055,C1(NC(Cc2cccc(N(C(C)=O)C)c2)=O)CC(C)CN(C(=O)C=C2CC2)C1 44056,C(=O)(C(C)C(=O)N1CCN(CCCNC(=O)C(C)(C)n2cnnn2)CC1)OC 44057,c1(C(=O)NCCC2N(C(c3c(C)con3)=O)CCOC2)c(Cl)cc(Cl)cc1Cl 44058,C1(C)(CNC(c2c(C)cc(CNC(=O)C=CCF)o2)=O)CCCC(=O)N1 44059,C1(C(N(C(C)C)CCc2ccco2)=O)CCN(C2CCOC2C)CC1 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44078,C(=O)(C1CCc2nccn21)NCC(C1CCN(C(C2(C(C)C)CCC2)=O)CC1)F 44079,C1(NC(=O)CCCF)CN(C(c2cccc(F)c2)=O)CC1CC1CC1 44080,N1(C(Cc2c(C)n[nH]c2C)=O)CC(NC(c2cc(CO)ccc2O)=O)C(C#N)C1 44081,C(c1cccc(CO)c1)=CC(N1C(CCNC(C2CSCCS2)=O)CSCC1)=O 44082,N1(C(c2c(C(C)C)nns2)=O)CCC2OC(CNC(=O)CSc3nc[nH]n3)C2C1 44083,c1(C(c2cccnc2)C)noc(COC(=O)CCCN)n1 44084,c1(C(N(C(C)C)CCNC(=O)CCC2CCC(=O)N2)=O)cc(C(F)(F)F)nn1C 44085,C12CN(CCO1)C2=O.c1(CN(C(C)=O)C)scnc1C 44086,c1(C(=O)NCCCNC(C(C)C2CC2)=O)ccnn1-c1cccnc1 44087,C(=O)(CCC(=O)C(C)(C)C)C(CN1CCCC(C)C1)=O.c1(CC)cn2c(n1)CCC2 44088,CC1CC(C)N(C(c2oc(S(N)(=O)=O)cc2Cl)=O)CCN1C(=O)CCF 44089,C(=O)(CCCCCCN(C)C)N1CCCC(NC(c2c(C)cns2)=O)C1 44090,n1(CCNC(C2C(C(=O)NCC3CC(OC)C3)C2)=O)cc(C)cn1 44091,Cc1cc2ncnc(N3CCC4(CCN(C(c5ccc(F)c(F)c5)=O)C4)C3)c2[nH]1 44092,C12(C(=O)Nc3cc(N)c(C(N4CCCCC4)=O)cc3)CCCCC(=O)N1CCC2 44093,c1(OC)ccc(CN2CCC(C(N3CCOCC3C)=O)C(O)C2)c(Br)c1 44094,c1(C(=O)NC2C(CNC(=O)C3=CCC3)CC2)ccc2oc(=O)oc2c1 44095,C1(C(N2C(CCNC(=O)COc3cccc(F)c3)CCC2)=O)CCCC(F)(F)C1 44096,c1(N2CCN(C)CC2)ncnc(NCCNC2(C)CCC(C(C)(C)C)CC2)c1C 44097,n1(C(C)C)cc2ncc(C(N3CCC4(CC3)CNC4C(=O)C3CC3)=O)cc2n1 44098,N1(C(c2n(CCC)nc(C)c2)=O)CCC2CCN(C(=O)C(F)CCC(C)C)CC12 44099,CC(C)CC(F)C(=O)N1CC(CNC(=O)Cc2ccc(O)cn2)C(C)(C)C1 44100,C=Cc1ccc(C(=O)NC(CCSC)C(=O)N2CCC(CC3CC3)C2)cc1 44101,c1(NC(C2C(C(=O)OC)C2)=O)sc2c(c1C(N1CCC(C)C(F)(F)C1)=O)CCC2 44102,N1(C(C2C(C(=O)OCC)CC2)=O)CCCC1CC(=O)NC(C(C)C)C1CC1 44103,C1(C(=O)NC(C=CC(=O)N(C)CCC2CC2)(C)C)CC2(CCO1)CC2 44104,CC1CCN(C(c2ccn(-c3ccccc3)n2)=O)CC1NC(C1CCC(=O)N1)=O 44105,N1(C(C(C(C)C)S)=O)CCn2ncc(CNC(=O)C(N3CCOCC3)O)c2C1 44106,c1(C(=O)NCCCCC(C)NC(c2cocc2C(N)=O)=O)nnc(O)cc1O 44107,C1(OCC)(CO)CCCCC1.C12CCCN(C1)C(=O)c1cscc1NC(=O)C2C 44108,N1(C(c2n(CC)cnn2)=O)CCCC2(C1)CN(C(C1CC1F)=O)C2 44109,CCC(C)(C)OCC(=O)N(CC(O)CN(C(=O)C=CCN(n1cncn1)C)C)C 44110,C(CC(C)C(=O)N(CC(C)O)CCNC(=O)Cc1cncnc1O)=CCC 44111,C12(NC(CCCC)=O)CCCC1N(C(=O)CSc1ccc(NC)cc1)CC2 44112,N1(C(c2c(CC)cccc2)=O)CCC2(CC2C(=O)NC2CCN(C(C)C)CC2)C1 44113,C(=O)(C(O)C(C)(C)C)N(CC(C)O)CCNC(C1CC(O)(CC#C)C1)=O 44114,N1(c2n(CC(=C)C)c(CN3CCCC(O)C3)nn2)CCC(O)CC(C)(C)C1 44115,c1(C(C(N2CCC(C)(CNC(C(CC)C)=O)C2)=O)C)c(C)nn(C)c1C 44116,c12ccc3c(c1)C(NCC2)CCO3.C1(C(=O)OC)CC(CC(=O)OC(C)(C)C)CO1 44117,c1(C(N2C(CN(C(CCSCCC)=O)C)COCC2)=O)ccc2c(n1)CCOC2 44118,C(=O)(CC(C(F)F)C(C)(C)C)NCC1CC(OC)CN1C(=O)CN1CCOCC1 44119,N1(C(Cc2scc(C)c2)=O)CCC(F)(C(N2CC(CN(C)C)C2)=O)C1 44120,C1(CNC(C2(OC)CCCC2)=O)CC(NC(c2cncn2C)=O)CC1O 44121,C1(C(=O)N(CCCCCNC(=O)Cc2ccsc2)C)(OC)CS(=O)(=O)C1 44122,N1(C(C(=O)NC)C(C)CC2CCOCC2)CCc2sc(C)nc2C1 44123,Cc1cc(CN2CCC(C(=O)Nc3ncc(Cl)cc3O)C(O)C2)cc(Cl)n1 44124,C(=O)(C(CC(C)C)C(N)=O)N(CC1CCN(C(CC(CC=C)(C)C)=O)CC1)CC 44125,c1(C(=O)OC)ccoc1C(=O)NC(C)CCNC(c1csc(C(F)F)c1)=O 44126,C(=O)(C(O)CCS(C)=O)N1CCC(N(CC#C)C(C2(CCO)CC2)=O)CC1 44127,N1(CC(=O)N(C2CN(C(C(C)OCC)=O)C2)CC)C(=O)C2CCCCC2C1=O 44128,C1(NC(=O)C(F)CC2CCOC2)CCCC12CN(C(C1CC3C(C1)C3(F)F)=O)C2 44129,O(N(C)C(=O)CNC(C(C)CCC)c1nnnn1CC1CC1)CC 44130,CCC(C)(O)C(=O)N(C)C.N1(CC2(C=O)CC2)CCN(C(=O)Cn2cccn2)CC1 44131,c1(SCC(N2CCC(CCCC(=O)OC)CC2)=O)nc2ccccc2n1C 44132,C1(O)(CNC(C(C)OCCC#C)=O)CCCN(C(=O)C(Cl)=CCl)CC1 44133,c1(C(=O)OC)cc(F)c(C(=O)NC(C(C)NC(=O)C(=O)N(C)C)C(C)C)cc1F 44134,C1(NC(c2cccnc2Br)=O)CC2CN(C(c3ccc(S)cc3)=O)CC2C1 44135,C1(C(=O)NCC(C(=O)NCCc2c(C)n(C)nc2)O)CCC(O)CN1C 44136,c1(CC(=O)NCC2N(C(CCC(C)SC)=O)CCCCC2)ccc2occc2c1 44137,C1(NC(CC(C)CF)=O)CCOC12CCN(C(c1cc3ccccc3[nH]1)=O)CC2 44138,C12(C(N3C(C(=O)NC(C)CCCO)CC(F)C3)=O)CCC(CC1)CC2 44139,c1(C(=O)NC(CC(C)NC(COC(C)=O)=O)C)cc(C)c(Br)o1 44140,N1(C(C(C=C)(C)CC)=O)CC(C)(C)C(NC(C2CC=C(C)CC2)=O)C(C)(C)C1 44141,CCC(CC(=O)N(C1CN(C(c2[nH]nnc2C(F)F)=O)C1)C)c1ccccc1 44142,N1(C(C(C)n2ccnc2)=O)CC=CC(NC(c2scc(Br)c2Cl)=O)C1 44143,C(=O)(CCCC(=O)NC1CCC(F)(CNC(=O)CCCCCOC)C1)NC 44144,c1(C(=O)NC2C(NC(CC3N(CC)CCC3)=O)C2)c(C)cn(C)c1CC(=O)OC 44145,C(=O)(C1=CCC(C)CC1)NCCC(C)NC(C1(CC(C)C)COC1)=O 44146,C(=O)(CCCCC(F)(F)F)NC1C(C)CCN(C(C(CC)C(C)O)=O)C1 44147,N1(C(C(CC)(C)C#N)=O)CC2CN(C(=O)C(C)c3ccsc3)CC2C1 44148,CC12CCC(C(=O)NC3COC4CN(C(c5ccon5)=O)CC34)(CC1)CO2 44149,N1(C(C2=C(C)OCCC2)=O)CC2(CCCCN2C(c2cc3c[nH]nc3s2)=O)C1 44150,Cc1nccnc1C(=O)N(CC(C)(C)C(=O)NCC(C)(C)CN(C)C)C 44151,C(C)(N=c1[nH]nco1)C1CCN(C(C23OC(C)C(C2)C3)=O)C1.C1CC1 44152,CN1CCOCC1C(=O)NCCC1CCCN1C(c1cnn(C)c1Br)=O 44153,C1(NC(C(CCC)c2ccccc2)=O)CN(C(c2ccc(F)cc2)C)CCC1C 44154,c1(C(=O)OC)cccn(CC(N2CCC2CNC(C2(C(C)C)CCC2)=O)=O)c1=O 44155,N1(C(C(CCSC)(C)C)=O)CCC2(CCCN2C(c2ncc(Cl)cc2Cl)=O)C1 44156,N1(C(c2cc(Cl)nn2C)C(=O)NC(CC)(C)C)CCOC2(CCSC2)C1 44157,C1(C(=O)NC(c2ncc(C)[nH]2)CC)CCN(C(C2CC23CCCC3)=O)CC1C 44158,C(=O)(C#CC(C)(C)O)N1C(CNC(C2CCCN(C(C)C)C2)=O)CC(COC)C1 44159,c1(C(=O)NCC2(C(=O)NC(C(C)(C)O)CCO)CC2)ccn2cncc2c1 44160,N1(C(C(CC)NC(N)=O)=O)CC2(CCN(C(=O)C=C3CCC(C)C3)CC2)C1 44161,c1(OCC)ncc(C(=O)NC2CCC(NC(C3(C)CCOC3)=O)CC2)cn1 44162,C(=O)(C(F)CC(C)(C)N(C)C)NCCCOCCN(C(=O)Cc1cnn(C)c1)C 44163,c1(C(=O)NCC(C)(C)NC(=O)CC2CCC(CC3CC3)O2)cc([N+](=O)[O-])n[nH]1 44164,c1(OC)cc(O)c(C(N2CCN(C(C3CCCC3(F)F)=O)C(C)C2)=O)cc1OC 44165,N1(CC)CCCC(C(=O)NCC2(C(=O)NCCSC3CCCO3)CC23CCC3)C1 44166,C1(C(N2CCOC(C)(CNC(=O)CSC)C2)=O)(COC)CCCNS1(=O)=O 44167,N1(C(c2cn(CC)nc2)=O)CCCC2(CC(NC(=O)CC3CCCC3C)C2)C1 44168,c1(SC)ccc(OCC(=O)NCCC2(C)CCN(C(=O)C(F)=CCCF)C2)cc1 44169,N1(C(C2C(OC)C2)=O)CCC(NC(C2CN(C(C)C)C2)=O)C1(C)C 44170,N1(C(c2c(C)c[nH]n2)=O)CC2CCCC2(NC(c2occ3c2CCC3)=O)C1 44171,C1(NC(CCC(=O)NCC)=O)CCN(C(=O)CCc2ccc(F)cc2Cl)CC1F 44172,CC(C)C(C)C(C)CC(=O)NC(C)(C)COCCCNC(c1cnc[nH]1)=O 44173,N1(C(C(CC)F)=O)CC2=C(C1)CN(C(c1cc(C)ncc1C)=O)C2 44174,C(=O)(C(CC)NC(C1(C)CN(c2ncccn2)C1)=O)NC 44175,N1(C(c2ccc(CCC=C)cc2)=O)CC2CC(NC(c3snc(C)c3N)=O)C1C2 44176,Cc1nc2ccc(C(=O)NC(C)CN(C)C(c3cc(C4CC4)ncn3)=O)cn2n1 44177,c1(N(CCCSc2cnc(-c3ncccn3)s2)C(=O)C2CC2)ccc(Cl)cc1F 44178,Cc1ccccc1C(=O)N(C1CCCC(N(C(=O)Cc2ccsn2)C)C1)C 44179,C(=O)(CC(C(=O)OC)NC(=O)CN1CCN(S(C)(=O)=O)C(C)C1)OC 44180,c1(OC)cc(N)c(Cl)cc1C(N1CC(N(C)C(C23COCC2C3)=O)C2(CC2)C1)=O 44181,c1(C(N(CC(C)NC(C2(CC)CCC2)=O)CC)=O)cc(C)c(Br)c(C)c1 44182,N1(C(C(CC)NC(C)=O)=O)CC(CNC(C2CCC(=O)N(C)C2)=O)CC(C)C1 44183,N1(C(c2cc(CNC(C(CCC)F)=O)on2)=O)CCC(O)C(F)C1 44184,c1(C(N2CCC(C(C)(C)NC(C(C=C)O)=O)C2)=O)cc2nc(C)[nH]c2cc1F 44185,C(C(O)C(=O)NC1CCOCC1)NC(C(C)=CC1CC1)=O 44186,c1(C(N2CC(CNC(COCCOC)=O)C(C)(C)C2)=O)cc2cc(Cl)ccn2n1 44187,N1(C(COCC=C)=O)CCC(O)(C2CCN(C(c3cnc(SC)[nH]3)=O)CC2)CC1 44188,c1(C(N(CCCNC(c2c(C)snn2)=O)C2CC2)=O)cncc(N)c1 44189,Cc1cccc(Br)c1-n1cc(CCN(C(=O)C(=O)OC(=N)O)CCS)nn1 44190,c1(CC(=O)NCCC2CCN(C(C(C)C3CC3)=O)CC2)cn(C)c2ccccc12 44191,c1(NC(C2C(NC(CN3CCC(C)C3)=O)COC2)=O)cncc(C2CC2)c1 44192,O(C=CC(=O)N(CCC(C)NC(=O)CC1CC(C)(C)C1)C)CC 44193,CC(C)C(C(=O)NC1CCCC1NC(C1CCCN(C)C1)=O)n1cncn1 44194,C(C)(CCC(=O)NCC(O)CNC(C1(c2nncs2)CC1)=O)OC 44195,c1(CC(=O)N(C2CCN(c3cc(Cl)c(O)nn3)C2)C)cn2cc(F)ccc2n1 44196,C1(C(=O)OC)CCCC2(CCN(CC3CC4(CN3)CC(F)(F)C4)CC2)O1 44197,c1(C(N(C2CCCN(C(c3cnsn3)=O)CC2)CC)=O)ccc2c(c1)CCNC2=O 44198,N1(C(C(C)NC(CC)=O)=O)CC(O)(CCNC(=O)CC2COCC2O)C1 44199,c1(NC(C2(C(N3CC(CC(=O)OC)(OC)C3)=O)COC2)=O)ccc(O)cc1 44200,c1(C(=O)NC(CC=C)CNC(c2ccn(CC#N)n2)=O)ccc(C(C)C)cn1 44201,N1(C(c2c(CNC(C3(C#N)CC3)=O)occ2)=O)CCC(O)(C(F)F)C1 44202,C1(CC)CCC(C)N(C(=O)CCOCCN(C)C(c2nnc(S)n2C)=O)C1 44203,N1(C(C(C(C)C)O)=O)CC2CN(C(C34CSCC3C4)=O)CC2C1 44204,C1(C(=O)NCCC#C)CCN(C(=O)c2cccc(Cl)c2)O1 44205,CC1COCCCN1C(=O)CC(C(F)F)NC(C1CCCCCCC1)=O 44206,C1(C)(C(=O)NC(CCC)CO)CN(C(=O)CC2(C)CCC2)CC1C 44207,c1(C(N2CCCC(NC(C3(COC)CC=CC3)=O)C2)=O)cc(C)c(C)nc1C 44208,Cc1nc2[nH]c(C(N3CCC4(NC(c5ccc(F)cn5)=O)CC4C3)=O)cc2s1 44209,C1(NC(CC(=O)OC)=O)CC2CCC1CC2NC(C1(C)CC=C(C)CC1)=O 44210,CC1(CNC(c2c[nH]nc2CCNC(=O)CC2CCOCC2)=O)CCOC1 44211,CC(C)(CO)CCCNC(C1CCCN1C(c1ccsn1)=O)=O 44212,C12(CNC(C3N(C(C4C=CC(N(C)C)C4)=O)CCOC3)=O)CCC(F)(CC1)C2 44213,C1(Cc2cn(CC=C)nn2)CN(C(C2CCCC2c2nc[nH]n2)=O)CCO1 44214,c1(NC(C(c2ccccc2F)NC(C(C)=O)=O)=O)cccc2cncc(C)c12 44215,CCCCCC(CC)C(=O)NCC1(CNC(=O)C(n2nccc2C)C)CCCC1 44216,Cc1cc(CC(=O)NC2CCCC2NC(=O)C(CCO)N(C)C)n(C)n1 44217,c1(C(=O)NC2(CC(=O)NCc3ccccc3F)CCCC2)ncncc1Cl 44218,C(c1cc[nH]n1)=CC(=O)NCC1CCC(NC(C2CCC(=O)N2)=O)C1 44219,Nc1cccc(F)c1C(=O)NCC1CCN1C(=O)C(c1ccncc1)n1cccn1 44220,C(=O)(CCCC(C)(C)C)N1CC(CCC)C(C(=O)NCC=CCOC)C1 44221,CC(C(C)n1cc(CCCC(=O)NOCc2ccc(Cl)cn2)nn1)S(C)(=O)=O 44222,c1(OC)cc(Cl)ccc1CNC1CC1C(N1CCC2(CC1)CC2)=O 44223,C1(C(N(CCNC(C2CSCCS2)=O)CC2CC2)=O)CCCC1c1nc[nH]n1 44224,N1(C(C(C(C)(C)C)N2CCCC2)=O)CCC2(CC1)CC2CNC(c1ccon1)=O 44225,C1(C(=O)NC2C(CNC(=O)CCC3CCCCO3)CCC2)CC2OC1C1CC21 44226,C(=O)(C1COc2ccc(Cl)cc21)NCCN(C(C1CCC1CF)=O)CC 44227,N1(C(CCC=C)=O)CCC2(CCCCN(C(=O)C(C)N(C)C)C2)C1 44228,C1(CC)CN(C(c2ncc(Br)cn2)=O)CCC1NC(=O)C=CC(C)(C)C 44229,c1(CCNC(C2(C)CN(C(=O)CC3CC4CCC3C4)C2)=O)cnc(CO)nc1 44230,n1(CC)cnc2c(NCc3cccc(C)c3F)[nH]c(=NCCC=CBr)nc12 44231,N1(C(c2c(C)nc(CCC)s2)=O)CCCC(C)(NC(c2cc(F)cc(Cl)c2)=O)C1 44232,c1(NC(C)C)cncc(NC(=O)C(C2CCCCC2F)(C)C)n1 44233,c1(C(=O)NCCCC(C)NC(C2(C)CC(C)C2)=O)cccc2c1COCCN2 44234,C(C(C)C)(C(O)C(=O)NCc1c(C)nsc1Br)OC 44235,N1(C(C2CCCN(CC)C2)=O)CCCC2CN(C(=O)C(F)CC3CCCC3)CC12 44236,c1(C(N2CC(CNC(C3(CCCC)CCC3)=O)C(C)C2)=O)cc2c([nH]1)CCCC2 44237,O(N(C)C(=O)CN=c1[nH]c(=NC(C)C(C)CC)[nH]c2c1COCC2)CC 44238,C=CCCCC(C(=O)NC1CCC(C(N)=O)C1)NC(=O)CC1(OC)CCC1 44239,[N-]=[N+]=NCCCCCCC(=O)NCC1CN(C(=O)CC23CCCC2C3)C1 44240,C1(C)(C(=O)NCCC2(C(=O)NCC=CC(C)C)CCC2)CCCCO1 44241,c1(OC)ccc2cc(C(N3CCC(NC(C4CCC(F)CC4)=O)C3C)=O)[nH]c2c1 44242,c1(NC(C2CCN(Cc3ccc(C)[nH]3)CC2O)=O)cccc2c1OCO2 44243,c1(OC)ccc(F)cc1CNCc1ncc(C2CCCO2)o1 44244,C(=O)(C1=C(Cl)CCCC1)NC1CN(C(Cc2c(C)scc2)=O)CC(F)C1 44245,C1(C(N2CCC(C(C)NC(=O)NCCNC(N)=O)C2)=O)CCN(C)C1=O 44246,Cc1sc(Br)cc1S(=O)(=O)NCc1c(F)cccc1F 44247,S(=O)(=O)(c1ccc(N2C3CCC(C3)C2CO)c(F)c1)NCc1cc(C)ncn1 44248,CC(CC(=O)NCC1C=CCN1C(=O)COCc1nccn1C)c1ccco1 44249,N1(C(CC(c2ccc(C)cc2)C)=O)CC2CC(NC(=O)CC3CC=CCC3)C2C1 44250,c1(CC(=O)NC2C(C(N(C(C)C)C)=O)C2)ccc(O)cc1 44251,CN1CCOCC1CC(=O)NCc1ocnc1Cn1cc(C2CC=CCC2)nn1 44252,C12(COC)COC(C(=O)NC3CCCCC3NC(c3c(C)coc3SC)=O)(C1)C2 44253,C1(CC(=O)NCC(CC)NC(C2CCC(C)(C)OC2)=O)CCS(=O)(=O)CC1 44254,C1(NC(c2ncn(C)n2)=O)COCCN(C(=O)Cc2cccc(Br)c2F)C1 44255,N1(C(CCOC)=O)CC(C(=O)N(C)Cc2cc(C)on2)CC(C)C1 44256,C#CCC(C)(C)CNC(=O)C(CCOC)NC(c1[nH]ccc1C)=O 44257,c1(OCC(=O)NCCC2CCCN2C(=O)CC2COCC2O)ccc(F)cc1 44258,N1(C(C(N2CCSCC2)C)=O)CC2CCN(C(c3cccc(N)c3)=O)C2C1 44259,C1(C(=O)NCCNC(C2CCCN(C(CSC)=O)C2)=O)CS(=O)(=O)CC12CC2 44260,C(=O)(CC(C)CF)N(CCCSC(C)C)CCOCCOCC#C.C1C(=O)N1 44261,C(=O)(N=c1c(Br)c[nH]cc1I)C1CCC(NC(c2ccc(F)c(F)c2O)=O)CO1 44262,C(N=c1[nH]c(=NCCC=CBr)[nH]c2c1CCCCCC2)C1(C)CCC(=O)N1 44263,c1(CC(=O)NCC2(O)CN(C(c3c[nH]nc3C3CCCO3)=O)C2)ccccc1 44264,N1(C(c2cc(C)no2)=O)CCC2CCC(C1)N2CC1CCC2CC2C1 44265,O=C1CCc2ccc(NC(=O)Cc3csc(=NCc4cc(Br)cnc4F)[nH]3)cc21 44266,c1(C(C)=O)ccnn1Cc1cn(CC(N2CCC(N3CCCC3=O)C2)=O)nn1 44267,C1(CNC(c2ccn(C(CC)CC)n2)=O)CCCCN1C(=O)CC1(C)CCCO1 44268,C1(CN(C(c2occc2Br)=O)CC)CCN(C(c2cccc(OC)c2)=O)CC1 44269,C1(NC(CCC)=O)CN(C(c2cc3cncn3c(O)n2)=O)CC2CCCC12 44270,C(=O)(C(CCC1CC1)NC(c1c[nH]c(=S)cn1)=O)N(CCCC)CC 44271,C1(NC(c2ccn3ncnc3c2)=O)CN(C(=O)Cc2cnns2)CC2(CC2)C1 44272,C(=O)(CC1(O)CCOc2ccccc21)N1CC(C)N(C(C2CC2F)=O)CC1 44273,c1(CCC)cc(C(N2CCC(C(C)CNC(C3(CO)COC3)=O)CC2)=O)n(C)n1 44274,c1(OC)cc(C)c(C(N2CC=CC(NC(c3c(Cl)noc3C)=O)C2)=O)cc1Cl 44275,N1(C(C(=O)N(C(C)C)C)=O)CCN(C)C(=O)C1.c1(C(C2(N)CC2)=O)ccc(F)cc1 44276,N1(C(C(C(C)OC)O)=O)CC2CCCC(C1)N2C(c1ccsc1Cl)=O 44277,c1(C(=O)NCC(CC)(CC)NC(=O)C(CC(C)C)OC)cc(OC)cc(C)c1N 44278,N1(C(CC2(NC(c3cc(CC4CC4)on3)=O)CC2)=O)CC(O)(CO)C1 44279,N1(C(c2c(CC)ocn2)=O)CCCC(NC(=O)Cc2ccsc2C)C(F)C1 44280,C(C(=O)NN1CCC(NCCC2CC2)CC1)(C(C)(C)C)NC(=O)OC(C)(C)C 44281,c1(C(=O)NCC2(F)CC(CNC(=O)C(Cl)=CCl)C2)cnn2ncccc12 44282,N#CC1CCCC(C(=O)NC2CC3(C2)CC(NC(=O)Cc2cccnc2Cl)C3)C1 44283,C12(NC(C34N(C(=O)CN5CCCC5=O)CCC3C4)=O)CCC(O)(CC1)CC2 44284,c1(-c2nc(OC(c3cccc(C)c3)CC)on2)c(F)cc(OC)c(F)c1F 44285,C1(C(=O)NC2(CC#C)CC2)CC(C)CN1C(=O)Cc1ccco1 44286,C1(C(N2CCCC(NC(c3c(CC)noc3)=O)C2)=O)CN(S(N)(=O)=O)C1 44287,c1(C(=O)NCC2C(NC(C3C(CC)C3)=O)C2)cc(N(C)C)cc(C#N)c1 44288,Cc1ccc(O)cc1NC(C1CCC2(CC2)N1C(c1ccoc1C)=O)=O 44289,CN1CCN(C(C2(O)CCCCC2)=O)CC1C(=O)NCc1ccc(C(N)=O)o1 44290,Nc1cc([N+](=O)[O-])ccc1C(N1CC(NC(=O)Cc2cncs2)C2(CCC2)C1)=O 44291,c1(C(=O)NC(C)(CNC(=O)C(F)C2CC2)C2CC2)cc(Cc2ccccc2)c[nH]1 44292,C(C(=O)NC(CCC1CC1)C(=O)NC1CC=CC1)(C(C)C)OCC 44293,c1(OC(c2nc(-c3nccs3)nn2C(=O)NC2CC2)C)ccc(F)c(Cl)c1 44294,C=CCN=c1[nH]c(C(N2CC3(C2)CN(C(=O)CO)C3)=O)cs1 44295,C=C1CCCN(C(=O)CCC(C)NC(=O)CC2(O)CCOCC2)C1 44296,c1(C(=O)OCC)cnc(SC)[nH]c1=NC(=O)NCc1noc2c1COCC2 44297,c1(NCC(N)=O)[nH]c(=NCC2CC=CCC2)nc2scnc12 44298,Cc1ccc(N2CCOC(CC3CC(NC(=O)OC(C)(C)C)C3)C2)nc1Br.C 44299,C#CCC(C)(CC)C(=O)N1CCC(c2nn[nH]n2)(COC)C1 44300,c1(C(CNC(c2sccc2F)=O)NC(C(c2ccccc2)OC)=O)cccnc1 44301,CCC(C)(COC)C(=O)NC(CNC(=O)C1=COCCC1)C1CC1 44302,C12(CC)CN(C(=O)Cn3cnnn3)C(CNC(C3CCS(=O)(=O)N3)=O)(C1)C2 44303,N1(C(CNC(C(C)N(CC)CC)=O)=O)CCC(O)C(C)(C)C1 44304,c1(-n2cc(C(C)(C)NC(CC(CNC)O)=O)nn2)cccc(C)c1Br 44305,O(NC(=O)C(Cc1cnn(C)c1O)NC(=O)CC=C(Cl)Cl)CC1CC(=C)C1 44306,N1(C(C2CCN(C(C(C)NC(C)=O)=O)C(C)(C)C2)=O)CCc2n[nH]cc2C1 44307,CC1CN(C(C2CCCO2)=O)CCCN1C(=O)CC(F)(F)F 44308,C1(CC)CN(C(CCC2CCC2)C(=O)NCc2ccco2)CC1O 44309,C(C(=O)NCC(O)CCNC(=O)CCCc1cccnc1)(C(C)O)NC(C)=O 44310,c1(C(=O)NC2(C(N(CCCF)CC)=O)CC2(C)C)cnn(C)c1C#N 44311,C(=O)(CC(C)(C)CN(C)C)NC(C(=O)N(C(CCC(C)C)C)C)C1CCOC1 44312,CC1(C)C(CC(=O)NCCCCCO)CCN1C(=O)C(O)CN1CCCC1 44313,Cc1nc(C(N2CC(NC(c3ncccc3Br)=O)C(O)C2)=O)n(C)n1 44314,CCC(C(=O)NC(C(=O)NCCC1CCCCO1)C1(C)CC1)N(C)CC 44315,C(=O)(C(F)(F)C(C)(C)O)N1CC(NC(C(CSC)C)=O)C(C(F)(F)F)CC1 44316,C1(C(=O)NC2CC(CC(=O)NC3C(NC)C3)C2)CC(=O)N(Cc2ccccc2)C1 44317,CCC(C)CCC(=O)N1CCCC1CCC1CCN(C(C2CC2(F)F)=O)CC1 44318,C1(C(N(C2CCN(C(c3ccn(C4CC4)n3)=O)C2)CCC)=O)CC12CC(C)(C)C2 44319,C1(NC(C(C=C)C)=O)CN(C(c2cnn3c2OCC3)=O)C2CCCC12 44320,C(=O)(CCCCC(N)=O)NCC1(F)CC(NC(C2CCC(=C)CC2)=O)C1 44321,C(=O)(C#CC1CCCOC1)NC1CC2CN(C(c3nc(CC)[nH]n3)=O)CC21 44322,C1(NC(C2C(CCOC)C2)=O)COCCC1NC(c1nc(OC)c(C)s1)=O 44323,C(C1c2ccsc2CCN1C(c1[nH]ncc1C#N)=O)NC(C(CC(C)C)OC)=O 44324,N1(C(C(C(=O)OCC)OC)=O)CCN(C(=O)CC(CC)C(C)C)CC2(CC2)C1 44325,CC(C)C(CN(C1CC1)C(C)C1CC1)C(=O)NC1CCC(F)(F)CC1 44326,C1(C(N2CC(C(N3CC(C(=O)NC)OCC3)=O)OCC2)=O)CCOC(=O)CC1 44327,c1(C(N2CCC(CSc3ccccc3)C2)C(=O)NCC)ccn2nccc2c1 44328,c1(C(CC)COC(N2CCCC(CC)C2)=O)ccc(Cl)c(F)c1 44329,C#CC1(C(=O)NC(C2(O)CCC2)C)CN(C(=O)CC2CCCC2C)C1 44330,O=C(C1=CCCN(C(=O)Nc2cc(Cl)ncc2F)C1)Nc1ccccc1 44331,CC1CC(NC(C2CCCS2)=O)CN(C(=O)C(C)(O)c2cscn2)C1 44332,c1(C(N(CC(C)CNC(=O)CCc2cnc[nH]2)C)=O)ns[nH]c1=O 44333,c1(OC)ccc(CC(C(=O)O)NC(=O)NCc2c[nH]cc(F)c2=O)c(C)c1 44334,N1(CCC)CC(N=c2[nH]c(=NCCN3CC4CCC3C4)[nH]c3c(F)cccc23)C1 44335,C(=O)(CN=c1cc[nH]cc1)N1C(CNC(C2(C)N(C)CC(OC)C2)=O)CC(F)C1 44336,C1(CNC(C(CC)F)=O)CC2(CCN(C(=O)CCc3cc(Cl)no3)CC2)C1 44337,c1(C(=O)NCC(c2ccsc2)O)cc2cccc(Br)c2o1 44338,N12CCN(CC1)CCSCCCC2=O.C1(CC(=O)N)CC2COCC12.CC(C)(C)O 44339,C1(NC(c2c(C)[nH][nH]c2=N)=O)CN(C(c2cc(C(N)=O)co2)=O)CCC1CO 44340,C(C1=Nc2cccc(F)c2S(=O)(=O)N1)N1C(C)CC(O)CC1 44341,c1(OC)c(CNC(=O)C(C)Oc2ccc(Br)cc2F)cccc1Cl 44342,c1(C(=O)NC2CC(N)C23CCOCC3)nc(O)nc2ccccc12 44343,c1(C(N2CCC(N(C(c3ccnc(C)n3)=O)C)C2)=O)ccc2c(C)noc2c1 44344,CC1=NNC(=O)C1CC(N1CCOC(CCNC(=O)C(C)(C)C2CC2)C1)=O 44345,C1(CC(=O)NCCOC(CC)(C)C)Cc2cccc(Cl)c2O1.C(C)(=O)O 44346,C1(CNC(CCSCCCC)=O)CN(C(=O)CC2(NC(C)=O)CC2)C2CCN1C2 44347,CCCC(O)C(CO)NC(=O)NC(Cc1ccccn1)CO 44348,c1(CC)ccc(OC)cc1C(N1CCCCC1CNC(C1CCC(=O)N1)=O)=O 44349,C1(NC(C(CCC)OC)=O)CC(F)CN(C(c2c(OC)ccnc2O)=O)C1 44350,C12(C(=O)NCCNC(C=C)=O)CCC(CC1)N(C(=O)C(C)(C)OC(C)=O)C2 44351,C(CC1c2ccccc2CCN1C(=O)C(C)SC)NC(CCOCCOC)=O 44352,C12(C(N3CC(O)(CN(C(Cc4ccc(OC)cc4)=O)C)C3)=O)CCC(C)(C1)OC2 44353,c1(NCCCc2c(C)noc2)[nH]c(=NCCn2ccnc2)nc2ncn(C)c12 44354,N1(C(C(=O)Nc2c(C)n(C)nc2)=O)CCOC2(CC1)CCS(=O)(=O)C2 44355,C=C(C)c1ccccc1NC(C1CC12CN(C(c1cc(C(C)C)n(C)n1)=O)C2)=O 44356,C1(CC(=O)NC23CC2CN(C(c2cc(O)nc(Cl)c2)=O)C3)CCn2cncc2C1 44357,C1(C(=O)Nc2ccco2)CCCN(C(C2COCC2OCc2ccccc2)=O)C1 44358,c1(C(=O)NCC2CC(COC)CN2C(C2CC(C)(F)C2)=O)cc2cccnc2s1 44359,CC1(C(N2CC(CNC(=O)C(c3ccc(F)c(F)c3)=O)C2)=O)CCCS1(=O)=O 44360,C1(CNC(C2C(CC)C2)=O)CN(C(c2ocnc2C)=O)CC12CC2 44361,c1(C(=O)OC)cc(S(=O)(=O)Nc2noc(-c3cnn[nH]3)n2)n(C)c1 44362,c1(NC(CNC(C(CC)C)=O)=O)ccc(Cl)nc1C(=O)OCC 44363,c1(OC)c(C(=O)Nc2cncc(-c3ccc(SC)cc3C)c2)ccc(Cl)c1Cl 44364,c1(C(=O)NC2C(C)N(C(=O)CCC3CCCCO3)CC2)cc(F)cc2ccoc12 44365,C=CCCC(C(=O)NC(CCO)C1CC1)NC(=O)COC(C)C 44366,C12(NC(c3c(C)cc(C)nc3O)=O)CC(C)(C1)OC21CN(C(C2CC2C#N)=O)C1 44367,c1(NC(C(C)C)CNC(C2CCCO2)=O)ncncc1I 44368,c1(-c2c(NC(N(CC(=O)OCC)CC)=O)csc2C)cccc2c1OC(F)(F)O2 44369,N1(C(C(C)(C)NC(c2ccccc2)=O)=O)CC(OC(C)(C)C)CC(C(=O)O)C1 44370,C1(CCNC(C2CC(=C)C2)=O)CN(C(C2OCCC2C(C)C)=O)CCS1(=O)=O 44371,C1(C)(CC(=O)NC2(CCCC)CC2)CCN1C(C1CC1C(=O)OC)=O 44372,Cc1ccc2c(c1)C(C(=O)NC1CC(NC(=O)Cc3nn(C)cc3Cl)C1)OCC2 44373,C(C(O)C(=O)N1CCC1c1cn(CC(n2cccn2)C2CC2(Cl)Cl)nn1)OC 44374,Cc1cc(C)c(C(=O)NC2CC(n3cc(-c4ccc(CO)cc4)nn3)C2)c(S)n1 44375,C1(NC(C(COC)(F)F)=O)CCC(C)N(C(c2ccc(-c3ccco3)[nH]2)=O)C1 44376,O(NC(=O)C(COC(C1COCC1OC)=O)OCC)CCCOCC 44377,N1(C(CC(CNC(C(CC)C#N)=O)OC)=O)CCCCC2(CCC2)C1 44378,c1(NC(C2C(C(=O)Nc3ccc4sncc4c3)C2)=O)c(O)cccc1[N+](=O)[O-] 44379,N1(C(CCCNC(C)=O)=O)CCN(C(=O)C(c2ccc(Br)cc2)C)C(C)C1 44380,n1(C(CC)C)nnnc1C(c1ccc(Br)s1)NCc1ccc(COC)o1 44381,CCC(C(=O)NCCCCCNC(=O)COCc1ccccc1)N1CCOCC1 44382,C=CCC(CNC(C1C2CCC(C2)C1C)=O)C(=O)NC1CCN(C(=O)CC)C1 44383,C1(c2cn(CC(C)NC(=O)CSC(F)(F)F)nn2)COC(C)(C)O1 44384,C1(NC(c2ccc(O)nn2)=O)(CO)CCCN(C(=O)Cc2ccc(O)cn2)C1 44385,Cn1cc([N+](=O)[O-])c(C(=O)NCC2(F)CCN(C(=O)CN3CSCC3=O)C2)n1 44386,c1(CC)oc(C(N2CC(CC(=O)N(CC(C)C(=O)OC)C)C(C)C2)=O)cc1C 44387,n1(CCC(=O)N(C2CN(C(c3c(C)oc(C4CC4)n3)=O)C2)C)ccc(O)nc1=O 44388,C1(CNC(C(C=C)O)=O)CCCCN(c2nc(Cl)ncc2C(N)=O)C1 44389,C1(N(C(c2ccccc2Cl)CC)C)CC2(C1)CC(C(=O)NC(c1ccc(Cl)o1)=O)C2 44390,C(=O)(C1=CCCC1C)NCC1CC(COC)CN1C(C1OCCC1C)=O 44391,C1(C(C)C)(C(=O)NCCC2CN(C(=O)C(F)C(C)C)C2)CNC(=O)C1 44392,c1(OC)ccc(NC(C2CC3CC3N2C(=O)Cc2ccccc2OC)=O)cc1C 44393,C(CCN(C)C)(C(=O)N1CCOCC1C(F)F)NC(c1scc(C)c1)=O 44394,c1(CCC(=O)N(C2CCN(C(=O)Cn3nccc3C)C2)CCC)nc(O)n[nH]1 44395,c1(C(=O)NC(C2CC2C(=O)NCCC2CC2C)C)cnnn1C 44396,N1(C(CC=C(C)C)=O)CCC2(CC1)CN(C(C1CC3CC1CC3(F)F)=O)C2 44397,C(C(=O)N1CCC(F)(C(=O)NCC2CC(N(C)C)C2)C1)(C(C)(C)C)OC 44398,C1(N2CCC(c3c(C)cccn3)C2)CC12CC=CCC2 44399,S(=O)(=O)(c1ccc(F)cc1)NC(CC(=O)N(CC(C)NC(=O)SC)CC)C 44400,C1(C(N2CC(CC=C)(NC(C3CC3COC)=O)C2)=O)CC2(COC(=O)N2)C1 44401,c1(C(=O)NCC(N(C(=O)CC2CCOC2=O)C)C2CC2)csc(S(N)(=O)=O)c1 44402,C(=O)(C(CNC(=O)CC(C)n1ccnc1)C(C)(C)C)NCc1cn(CC)nn1 44403,N1(C(c2c(C)cncc2)=O)CC2(C1)SCCC2NC(=O)CCCCN(C)C 44404,N1(C(COC(C)C)=O)CCC(C=CC(=O)NCC2CC(C)CO2)CC1 44405,N1(C(C2CC(C)OC2)=O)CCC2(CC1)CCN(C(c1cnc(N)c(Cl)c1)=O)C2 44406,c1(C(=O)NC(C2N(C(C(CC3CC3)OC)=O)CCC2)C)ncc(Cl)cc1F 44407,C(=O)(CC(C)P(C)(C)=O)NCC(CCCC)NC(c1cc(OC)n(C)n1)=O 44408,Cc1cc(Cl)c(C(=O)NCC2(F)CCN(C(c3cnncc3O)=O)CC2)cc1C 44409,n1(CCC(=O)NCC2C(NC(c3c(C(C)=O)[nH]cn3)=O)CC2)nc(C)cc1C 44410,C(=O)(C1=CCCCC1C)N1C(C(=O)NCCn2ncc(CC)c2)COCC1 44411,c1(C(=O)NC(CNC(C(N2C(CC)CCC2)=O)=O)C)ccc2c(c1)CCCCN2 44412,n1(CC(=O)NC2(CO)CN(C(=O)CCC3CC3(F)F)C2)nnc(C2CC2)n1 44413,CCCC(CC)C(=O)NC1(CC)CCCN(C(c2ccoc2)=O)C1 44414,c1(C(=O)NC(CN2CCN(C(C(CC)OC)=O)CC2)C)cc(C)ccc1F 44415,CCC(CCO)N=c1[nH]c(N2CC(Oc3ccccc3)C2)nc2c1CSC2 44416,CC1(NC(C2(CNC(=O)Cc3cncnc3)CCCCC2)=O)CC2(CC2)C1 44417,C12(CCNC(c3c(C)noc3)=O)CCC(CC1)N(C(c1ccc(F)c(F)c1)=O)C2 44418,c1(COC)ccccc1C(=O)NCCC(C)NC(c1cc(Br)cn1C)=O 44419,Cc1nc(Cl)c(NC(C2CC2C(=O)NCc2cc(F)cc(I)c2)=O)cc1Br 44420,Cc1c(C(=O)NCC2(CNC(C3CC(=O)OC3(C)C)=O)CCCC2)cncc1F 44421,c1(OC)cnc(C(=O)NCC(C)(C)OCC(=O)NCC(N)=O)cn1 44422,c1(C(N2C(CCNC(C(C)OCCCC)=O)CCCC2)=O)cc(F)c(C)cc1Cl 44423,CC1CCN(C(c2cccc3nsnc23)=O)C(C)C1NC(=O)CN1CC2CC2C1 44424,c1(CCC(=O)NCC2N(C(C(C)CC3CCC3)=O)CCOC2)nnc(S)nc1O 44425,C1(CC(=O)O)CC2(CCOCC2)CN1Cc1cc(N)c(O)c(F)c1 44426,c1(OC)cc(CC(=O)NCCC2CN(C(C3CC3c3cn[nH]c3)=O)C2)on1 44427,c1(N2CC3CN(S(CCCC)(=O)=O)CC(C2)O3)ncnc2ccc(OC)cc12 44428,C1(CC(=O)OC)(C(=O)NCC(=O)OC2CCN(C(=O)C)C2)CNC(=O)C1.C(C)(C)(C)O 44429,C1(NCC(=O)NC(=O)NCCc2ccc(OC)cc2)CCC2OCCC2C1 44430,N1(C(C(N2CCOCC2=O)C)=O)CCc2[nH]nc(-c3ccncc3)c2C1.[nH]1cccc1 44431,c1(C(=O)NC2CN(C(c3cc(SC)oc3)=O)C(C)CC2)ccc(P(C)(C)=O)cc1 44432,N1(C(C(c2cccc(OC)c2)C)=O)CC(NC(=O)Cc2csnn2)C(N=[N+]=[N-])C1 44433,c1(C(=O)NCC2C(NC(C(C)SC(C)C)=O)C2)cc(C(F)(F)F)ncc1Cl 44434,C12(CC(=O)O)CCC1CN(CC1=CCCCC1)C2.c1(-n2ccnn2)c[nH]ccc1=O 44435,N1(C(C(CNC(=O)OC(C)(C)C)F)=O)CC(C(=O)O)CC1CO 44436,c1(OC(C)C)ccccc1CC(=O)OCC1(C(F)(F)F)CCNCC1 44437,CC1CCCC(N(C)C(=O)NC2CC3(CC(NS(C)(=O)=O)C3)C2)C1C 44438,C(c1cc(C)c(C)cc1C)=CC(=O)NCC(c1cccc(C)c1)NC(=O)CO 44439,C1(OC)CN(C(=NCCc2sccc2C)NCc2ccco2)CC1O 44440,C1(C(=O)NCCCNC(C(C)C)=O)CC(C)N1C(=O)C=Cc1ccoc1 44441,O=S(=O)(c1cccc2cccnc12)NCc1ccnc2c(I)cnn12 44442,c1(C(=O)NC2C(n3cc(-c4ccc(C(=O)OC)o4)nn3)CCC2)ccc(F)cc1Cl 44443,N1(C(C(CC)N(C)C)=O)CC2C(NC(=O)CCc3cccnc3)CS(=O)(=O)C2C1 44444,C1(NC(C=CC(C)C)=O)CCC2(CC1)CN(C(C1CC1C1CC(F)(F)C1)=O)C2 44445,c1(C(=O)OC)ccc(O)nc1NC(C)CC(C)NC(C1CCS(=O)(=O)C1)=O 44446,c1(N2CCC(C(C)NC(c3ccc(COC)s3)=O)C2)ncc(Br)cc1C#N 44447,c1(C(CC)NCCNC(=O)CCCc2nc(-c3cccs3)no2)c(C)n[nH]c1C 44448,C1(C(=O)NC(C)C(CO)NC(=O)Cc2ccsc2)CCCC2(CCCCC2)C1 44449,c1(N2CCN(S(Cc3c(C)cc(Br)cc3)(=O)=O)CC2)c(C#N)oc2ccccc12 44450,N1(C(c2cc(C)n(C)c2C)=O)CCC(NC(=O)CCC2CCCO2)CC(C)(C)C1 44451,N1(C(CC2(CC(=O)OC)CC2)=O)CCC(NC(C2CCC(O)CC2)=O)C2(CC2)C1 44452,C1(C(=O)NCc2ncco2)(CC)CCCN1C(=O)CCN(C)C 44453,N1(C(CCC(=O)NCCC)=O)CC2CCCN(C(=O)C=CCOC)C2C1 44454,C1(CC(=O)NC2(CCO)CN(C(=O)CC3CCS(=O)(=O)C3)C2)CCCC1(F)F 44455,Cc1cnc2ccc(C(=O)NC3CCN(C(=O)CCS(C)(=O)=O)C3)cn12 44456,S(=O)(=O)(c1cnn(CCn2cccn2)c1)N1CC(C(=O)O)C1 44457,Cc1ncncc1C(N1CCC(N2CCN(C(C3CCCCN3C)=O)CC2)C1)=O 44458,c1(C(N2CC(CNC(c3scc(C)c3)=O)OCC2)=O)cccc2ncc(C)n12 44459,N1(C(CC2CCC(=O)N2)=O)CC2(CCCC2NC(c2cccc(C3CC3)c2)=O)C1 44460,c1(C(=O)NCCCC(C)NC(c2ncc(OCC)nc2)=O)c[nH]c2nccc-2c1 44461,C1(CNC(c2c(C)ccnc2)=O)CC2(CO1)CN(C(=O)CC(F)(F)C(C)C)C2 44462,c1(C(=O)NC2C(CNC(c3ccc(C#C)cc3)=O)COC2)cc2cn[nH]c2cn1 44463,C123CC(CC1C2)NC3=O.c1(COCCC(=O)OCC)ccc(CCC#N)cc1 44464,c1(C(N2CC(CC=C)(NC(=O)Cc3ccco3)C2)=O)ncnc(OC)c1F 44465,CC(C(=O)NCCNC(=O)C=Cc1cscn1)C(C)NC(N)=O 44466,N1(C(c2ccn(CCOC)n2)=O)C2CC1CN(C(c1ccc(F)cc1I)=O)C2 44467,C1(C)(CC)CCN(C(C2CC2C2CN(C(C3(C)CCCN3C)=O)C2)=O)CC1 44468,N1(c2nc(CC)nc(=N)[nH]2)C2CCCC1CN(C(=O)C=C1CCCC1)C2 44469,CC(C)C(C(=O)NCC1(O)CCN(C)C1)C(C)NC(C1CC(=O)NC(=O)N1)=O 44470,Cc1cnn(CC(N2CCC3C(NC(=O)C(CN(C)C)N(C)C)C23)=O)c(=O)c1 44471,c1(C(N2CCN(C(COCC=C)=O)C(C3CC3)C2)=O)cnn2cccc(Cl)c12 44472,c1(C(=O)NCc2c(C(N3CC(C)C3)=O)cccc2)ccc(O)cc1F 44473,C(C)(C(=O)NCCN(CCOC)C(C1CC(CC(N)=O)C1)=O)NC(CC)=O 44474,c1(CC(C)C)cc(C(N2CCC(CNC(=O)CC3(C)CC3F)CC2)=O)cc(O)n1 44475,C1(CNC(CCc2cc(C)sc2C)=O)CCC(C)(C)CN1c1ncnc(O)c1Br 44476,N1(C(COCP(C)(C)=O)=O)CCCCC(NC(c2ccc(N3CCC3)nc2)=O)C1 44477,Cc1ncn(C)c(=O)c1C(=O)NCC1C(C)CCCN1C(=O)C=CCF 44478,C1(CNC(c2csc(C(F)F)n2)=O)(CO)CCN(C(C2CC3(CC3)CO2)=O)C1 44479,c1(C(N2C(C)(CC(=O)N(C3CCOC3)C)CC2)=O)cnc(=N)[nH]c1 44480,CCC(C)C(C(=O)NOCc1nc[nH]n1)NC(c1ncc(F)cc1N)=O 44481,C1(CCNC(=O)C(COC)N(C)C)(NC(COCCC)=O)CCCC1 44482,C12(CNC(C3(C)CC(OC)C3)=O)CC(CNC(=O)CNC(=O)NCC)(CO1)C2 44483,C1(C(=O)NCC2CC(NC(=O)CC3CCCC34CC4)C2)CC2(C1)CC1(CC1)C2 44484,N1(C(C(=O)NC2CC2)=O)CCc2c(C(N3CCNCC3)=O)cccc21 44485,c1(OC)cc(CC(=O)NCC2(F)CC(NC(=O)C(C)OCC3CC3)C2)ccc1Cl 44486,Cc1cncc(C(=O)NCCOCCCN(C)C(C2CCC(N(C)C)CC2)=O)c1 44487,C(CN=c1cc(NCCc2ccc(Cl)nc2)nc(C(F)(F)F)[nH]1)(C1CC1)OC 44488,c1(CC)ccnc(C(N2CCC(O)(CSC)C2)=O)c1.C12(CC1)C(=O)NC2 44489,C1(C(N(CCN(C)C(c2cccnc2)=O)C)=O)CCCC2CCCN12 44490,c1(C(=O)NCCC2N(C(CC3CCN(C)C3)=O)CCC2)cn(C)ccc1=O 44491,N1(C(C(CC)F)=O)CCC(C2CCCN(C(=O)C=C3CCCC3)C2)C1 44492,CC1CN(C(C(C(C)O)C2CCC2)=O)CCN(C(=O)C(O)CC2CCCC2)C1 44493,c1(C(N2CCC(NC(c3n(C)cc(Cl)c3)=O)C(CO)C2)=O)ccc2nonc2c1 44494,C1(NC(c2cnn(CCC)c2C)=O)CC(C)CN(C(=O)CC2CCCC2(F)F)C1 44495,N1(C(C2C(=C)C2C(=O)OC)=O)CCC2(CC1)CC2NC(c1cc(C)cc(F)c1)=O 44496,c1(SCC)ccc(Cl)cc1C(=O)NCCN(C)C(C1(O)CC2CCC1C2)=O 44497,C(=O)(CCS(=O)(=O)CC(C)C)N1CCCC(O)(CNC(C(CCC)OCC)=O)C1 44498,Cc1cccc(C(N2CCC(CN(C)C(C3CCS(=O)(=O)C3)=O)C2)=O)c1Cl 44499,c1(C(=O)NC2(CCNC(CCCS(C)=O)=O)CC2)cccc2c1OCCO2 44500,C1(NC(C)(C)C)CC(O)C(F)C1.C1(=O)CC(=O)N(C2CCCC2)CCO1 44501,c1(C(=O)NCc2c(CC)noc2C)coc2c1CN(C(c1ccc(C)s1)=O)C2 44502,C1(n2c(C(C(C)(C)C3C(C)C3)NC(c3cnc(C)cn3)C3CC3)nnn2)CCC(F)(F)CC1.C 44503,N1(C(c2cccc(OC)n2)=O)CCc2ccc(C(=O)NCCCC(C)C)nc2C1 44504,CCCCCCC(F)C(=O)NCCN(C(=O)Cc1nc(F)c(F)cc1F)C 44505,c1(C2CN(C(C(CN(C)C)Sc3ccccc3F)=O)C2)cc(F)cc(F)c1 44506,C(=O)(C(CCOCCO)NC(=O)CC1CCOC1=O)NCCOCC 44507,c1(C(N(C2C3CN(C(CSCCCC)=O)CC32)C)=O)ncc([N+](=O)[O-])cc1C 44508,N1(C(c2c(C)cccn2)=O)CCC(NC(=O)CSC(F)(F)F)C2(CCC2)C1 44509,CC1C(=O)CCC(C(=O)NCC2CCCN2C(=O)CCN2CCC(F)C2)C1(C)C 44510,c1(C(=O)Nc2cncc(C(N3CCC(CC(=O)OC)C3)=O)c2)cc(Cl)ncc1I 44511,c1(OCC)cc(N2CCN(C(C3CC(C(C)(C)C)C3)=O)C(C)C2)nc(C)n1 44512,c1(SC)nc(C)c(CCC(=O)NCC2CCN(C(=O)C=C(Cl)Cl)C2)c(O)n1 44513,c1(C(N2CC(O)(C(C)NC(c3cc(CC)c(C)s3)=O)C2)=O)cc2ncccc2o1 44514,C(=O)(CCS(=O)(=O)NC)NCC1N(CCC)CCCC1.C12CCCC1C(=O)N2 44515,Cc1cc(Br)cc(C(=O)NC(C2CCCN(c3ccnc(Br)n3)C2)C)c1C 44516,C1(C(=O)NCC(CN(C(=O)CCc2nncn2C)C)O)CCN(C2CC2)CC1.C1(C)CC1 44517,N1(C(C2CC(C)(CC)C2)=O)CC2(CCCC2)C1C(=O)NOCCF 44518,C1(CNC(c2cc3occc3[nH]2)=O)CC2(CO1)CN(C(=O)CCc1ccc[nH]1)C2 44519,C(=O)(C(C)(C)C(F)F)NC(C)CC(=O)OC(C)(C)C.C12CC1OC2=O 44520,CCC(C)(CNC(=O)Cc1cccs1)C(=O)NCc1nc(C)ns1 44521,C1(OC(C)=O)C(CO)C2CCCC12.c12cc(sc1C)NC2=O 44522,C1(C(=O)NCCCC(CCC)Nc2ccc(COC)cn2)CC(C(C)(C)C)=NO1 44523,C1(CC(=O)NCC(CNC(C(C)c2ccco2)=O)O)COC(C)(C)C1 44524,N1(C(CNS(CC)(=O)=O)=O)CCN(C(=O)Cc2ccc(C)cn2)CC1C(C)(C)C 44525,C12(C(=O)NC3CC(N(C(C4C(C=C)C4)=O)C)C3)C3CC(CC13)C2(F)F 44526,Cc1nccc(Cl)c1C(=O)NC12CC1CN(C(=O)C(C)OCc1ccccc1)C2 44527,c1(C(N2CCCC(NC(C3C(C)CC(C)O3)=O)CC2)=O)ccc(F)c(Cl)c1F 44528,CC1CC(NC(=O)CN2CCCNC2=O)CCN1C(C1CC(=O)N(C)C1)=O 44529,CC1(C)OCC(CC(C)C(=O)Nc2cccc(C(N3CCCC3)=O)c2)O1 44530,N1(C(CCC(=O)NCC)=O)CCC(NC(=O)C(c2cn(C)nc2C)O)C(C)(C)C1 44531,N1(C(c2cnc(CC)o2)=O)CCC=CC1C(=O)NCC(C#N)CC 44532,C(=O)(C1=CCC2CCC1N2C(=O)C(C#N)C(C)(C)C)NCC(C)C(F)F 44533,N1(S(c2occ(C(C)=O)c2)(=O)=O)CC(C)OC2(CCCCC2)C1 44534,C(=O)(CCCN=[N+]=[N-])NCC(C)(O)CNC(C1CCCN1S(C)(=O)=O)=O 44535,Cc1cc(Br)c(F)cc1NC(c1cncc(C(F)(F)CF)c1)=O 44536,c1(NC2(c3ccccc3Br)C(NC(=O)C3CC3)C2)ccc(-c2nn[nH]n2)cc1 44537,C1(C(=O)OC)OC(C(=O)NC(CNC(=O)C=Cc2cnn(C)c2)C2CC2)CC1C 44538,C#CCCCCC(=O)NCc1nc(C(=O)NC(C)(C)C(O)CO)c(C)o1 44539,C(C#CC(=O)N(CCCCO)CC)NC(C1C(=C)C1)=O 44540,CC12CC(C(N3C4CCC3CN(C(C3C5CCCC35)=O)CC4)=O)(C1)C1(CCC1)O2 44541,C(=O)(C(O)C(C)CC)N(C(CNC(C=CC(=O)OCCCC)=O)C1CC1)C 44542,C(=O)(C1COc2ccc([N+](=O)[O-])cc21)NC(CC=C)CNC(=O)CC(F)F 44543,C1(C(N2CCC(C(C)(C)NC(CC(=O)NCC)=O)C2)=O)CN2CCC1(C)CC2 44544,C(=O)(C1=CCC(C)CC1)NCCC(C(=O)NC(c1onc(C)n1)CO)(C)C 44545,c1(C(=O)OC(C)(C)C)ccc(OC(C2CCC(C(=O)OC)C2)=O)cc1 44546,C1(NC(c2cnc(OC)s2)=O)CCC(C)N(C(C2CCS(=O)(=O)CC2)=O)C1 44547,C(=O)(C#CC(C)(C)C)N1CCC(C2N(C(C)=O)CCC2)CC1.c1cscc1Cl 44548,C(C)(CC)(CCNC(=O)CC1CCCCC1O)NC(C=CCCC)=O 44549,c1(CC(N2CCC(CCNC(COC(CC)C)=O)C2)=O)ccccc1F 44550,O(NC(=O)C(F)(F)C(C)(C)O)C(CC(C)C)C.N1CC2CC=CC1C2 44551,C(N=c1[nH]c2cc(Cl)ccc2s1)C1CC(NC(c2cc(CC)nn2C)=O)C1 44552,c1(C(N2CC(C)(OCC(=O)NCC(CC)C)C2)=O)cc(C#N)cn1C 44553,N1(C(c2c(COC)ncs2)=O)CCN(C(C2COCCO2)=O)C(C(C)(C)C)C1 44554,Cc1cc(Cl)ncc1NC(C1CCCCN1C(c1cn(C)cn1)=O)=O 44555,CCCCCC(=O)N1CCCC1(C)C(=O)N(C1CCOC1)CCN(C)C 44556,CCC(C)(C)CCCC(=O)N1CCC2(NC(c3coc(Br)c3)=O)CC2C1 44557,c1(C(N2C(CO)CC(NC(C3COC(=O)C3)=O)C2)=O)cc2nn[nH]c2cc1F 44558,Cc1ccc(SCC(N2CCC2CNC(=O)CCN2CCCCC2=O)=O)cc1 44559,N#Cc1cc(-c2ccc(CNC(c3ccc(OC(F)F)cc3F)=O)cn2)cc(F)c1 44560,C1(CC(=O)OC)CN(C(=O)CC=Cc2cccnc2)CCN1CCc1c(COC)cc[nH]1 44561,C1(C(N2C(CN(C(=O)C3=C(Cl)CCC3)C)COCC2)=O)CCC2(CCC2)CO1 44562,c1(OCC)ccc(C(=O)NCC(C)CN(C(=O)C(C)OCCC(C)C)C)cc1C 44563,C(C)(C(C(=O)NCc1cc(O)ns1)NC(c1nonc1C)=O)OC 44564,c1(C(N2CCN(C(C(C(C)C)OC)=O)CC2C2CC2)=O)cccc2nc(O)[nH]c12 44565,c1(C(N(CCNC(C=CCCC)=O)Cc2ccccc2)=O)nccnc1C(N)=O 44566,C(=O)C(=O)C(F)(F)F.CC1(C)CN(C(=O)C=CBr)C1C1CCNCC1 44567,N(C1CCCc2n[nH]cc21)C(C1N(C(CN2CCC(OC)C2)=O)CC(O)C1)=O 44568,c1(C(=O)OC)ccnc(C(=O)NC2CN(Cc3ccnc(Br)c3)C2)c1 44569,c1(C(N2CCN(C(C3CC(C)C3)=O)CC2CC(F)F)=O)cncc(S(N)(=O)=O)c1 44570,c1(OC)cc(C(N2CC(C(C)NC(=O)C#CC(C)C)C2)=O)ccc1C(N)=O 44571,C1(C(C)NC(c2csc(NC(=O)C(C)CC3CCC3)n2)=O)CCN(C(N)=O)CC1 44572,C(=O)(C1Cc2ccccc21)N1CCC(C)(NC(c2c(C)nc(CC)s2)=O)CC1 44573,c1(CC)ccc(C(=O)NC2CC2CNC(C2CC(C)(O)C2)=O)cc1 44574,C1(C(N2CC(C)(CCO)C2)=O)CCCN(C(=O)C(F)OC(F)(F)F)CC1 44575,c1(C(=O)NCC2N(C(CCOC(C)C)=O)CCC2)ccc(NC(C)(C)C)cc1 44576,CC1(C)OCC(C=CC(=O)NCC2CCN(C(=O)CCNC(=O)C=CCl)CC2)O1 44577,C1(C(N(CCCC)CCCO)=O)CCCCN1C(C1CCC2CC12)=O 44578,C1(C)(NC(CC(C)c2cccnc2)=O)CCCN(C(c2cnc(O)n2C)=O)C1 44579,C(=O)(C(C)(C)CC(C)C)NCC1(OC)CCN(C(C2(C)CCN(C)C2)=O)CC1 44580,n1(CC)ncc(Cl)c1C(=O)NC1CCC(C)(CC)C1 44581,c1(OC)c(C(=O)NCC2(F)CC(CNC(=O)C3=CCCC3C)C2)cc(Cl)cc1Cl 44582,Cc1nc(C)c(C(N2CCC(C)(CNC(c3scnc3C3CC3)=O)C2)=O)[nH]1 44583,N1(C(C(C(C)C)OCC)=O)CCN(C(C2CC(C)CCO2)=O)CC1CC(F)F 44584,Cc1cc(C(N2CC=CC(NC(=O)CN(C3CCCC3)C)C2)=O)c2c(c1)CCC2 44585,C12(C(N3CCC(CNC(Cc4c(C)ccs4)=O)C3)=O)CCC(CC1=O)C2(C)C 44586,c1(CC(=O)NC(CCCCNC(C=CC(CC)C)=O)C)cnc2cccnn12 44587,C(=O)(C1=CC(O)C(NC(=O)C2=CC3C=CC2C3)C1)N(C1CCCN(C)C1)C 44588,C1(C(N(CCCCNC(C2CC3(C2)CC3F)=O)C)=O)Cc2ccccc2C(=O)O1 44589,N1(C(CCCOC(C)=O)=O)CC(C2CN(C(C3(O)CC(C)(C)C3)=O)C2)C1 44590,C1(NC(Cc2cccc(OCC)n2)=O)CCCCN(c2cc(CC)ncn2)C1 44591,n1(CCOC)ccc2c(C(N3CCN(C(=O)CSC)CC(C)(F)C3)=O)cccc12 44592,S(=O)(=O)(CC(C)C)N1CC(N(C(C(=Cc2ccco2)C)=O)C)C1 44593,C12(NC(c3ccc(CC)nc3)=O)CC(CNC(=O)Cc3[nH]cnc3C)(C1)OC2C 44594,CN1CC(O)CC1(C)C(=O)NCCCN1CCC(NC(C2CC(F)C2)=O)C1 44595,N1(C(C2(C)CC3(CC3)C2)=O)CCN(C(=O)CNC(=O)C2CC2)C(CC(F)(F)F)C1 44596,c1(C(C(=O)NC(C)C)NC(c2c(C)n(C3CC3)nc2)=O)ccc2c(c1)C=CCC2 44597,N1(C(CCN(CCCCC)C(C)C)=O)CC2C(NC(C3(C)CCCS3)=O)C2C1 44598,C1(C(C(=O)NCCC(=C)C)F)CCN(C(=O)C=CCCC)C1 44599,CC(C)(C)C(CO)C(=O)NC1CCC(NC(c2ccc(F)o2)=O)CC1 44600,C(C(CNC(=O)CCc1ccccn1)S(C)(=O)=O)NC(C(C=C)C)=O 44601,C1(NC(CCC=CC)=O)CCN(C(c2ncccc2Br)=O)C12CCC2 44602,C#Cc1ccccc1NC(=O)C(CCC=C)NC(=O)CC(C)C(F)F 44603,C(CCCCC(=O)N(C)CCC1CCCN1C)NC(C1CC(C(C)C)C1)=O 44604,Cc1cc(C(N2CC(N(C)C(C3CCC3(F)F)=O)C(C)(C)C2)=O)ncc1C(N)=O 44605,N1(C(C2C(=C)C2)=O)CC(C(=O)Nc2cn(C)nc2C2CC2)CC12CCC2 44606,C1(O)(C(C(=O)NCC#CC)F)CN(C(=O)C=NOC)C1 44607,C1(CNC(CCC(C)SC)=O)CCN(C(c2cn3ccnc3s2)=O)CC1O 44608,N1(C(C=Cc2cn(C)nc2)=O)CCCC2(C1)CN(C(=O)Cc1ccsc1Cl)C2 44609,C(=O)(CC(C)(C)CNC(C1CC(F)(F)C1)=O)NCC(C)(C)C(F)F 44610,C(CC(=O)NCc1ccc(F)nc1C)(C(C)(C)C)NC(C(C)N(C(C)=O)C)=O 44611,Cc1cc(S(N)(=O)=O)oc1C(N1CCN(C(=O)COC2CCOC2)C(C)C1)=O 44612,CC1CC(C)(C)CCC1C(=O)Nc1cccc(COc2ccc(F)cc2)c1Cl 44613,C(=O)(C(C)(O)C1CCC1)NCC(C)CNC(C1(Br)CC1)=O 44614,N1(C(CC2(OC)CCC2)=O)CCCCC1C(=O)NC1CC(C)(O)C1 44615,C1(NC(C2CC(C)CN(C(=O)C(O)CC(F)(F)F)C2)=O)CCC2(CCCC2)C1 44616,CC1(C(=O)NCC#CC(=O)NCCC2CCOC2)CCC(=O)C1 44617,N1(C(COc2cc(C)c(F)cc2)=O)CC2CCN(C(c3csnn3)=O)CC2C1 44618,C1(N(C(c2cc(C)n(C3CC3)n2)=O)C)CN(C(=O)C(C)c2cccs2)CC12CC2 44619,c1(-n2cc(CN3CCN(C(C4CCCC4CF)=O)CC3)nn2)cnnc(O)c1Br 44620,C(=O)(C(C(C)(C)C)n1cc(C(C)N(C)C)nn1)NC1C(OCC)C2C1CCC2 44621,c1(CC(=O)NCC#CCNC(=O)CCc2nncs2)c(F)cccc1Cl 44622,C1(CN(C(C2COC(=O)O2)=O)CC)CCCCN1C(C1CC(O)CN1C(C)=O)=O 44623,c1(CN2CCC2)cc(S(N)(=O)=O)sc1Cl.C12(CC(O)C1)N(C)C2=O.C1(O)CCC1 44624,C1(C(N(CC(=O)NCC2CCCC(F)C2)CC)=O)CC2(CSC2)C1 44625,N1(C(C=CC(C)(C)SC)=O)CCCC12CCN(C(C1CCN(CC(C)C)C1)=O)C2 44626,N1(C(C2CC(OC)C2)=O)CCN(C(c2ccc(SC)s2)=O)C(C)CC1C 44627,C=C(C)CCCC(=O)NC1(CNC(c2cc(F)ncc2OC)=O)CCCCCC1 44628,Cc1cc([N+](=O)[O-])cc(C(=O)NC2CN(C(=O)C=CC3CCC3)CCC2F)c1Cl 44629,C(=O)(C1COc2ccc([N+](=O)[O-])cc21)N1CC(C)C(NC(c2cnc[nH]2)=O)CC1 44630,c1(C(=O)NCC2C(NC(c3c(C)n[nH]c3)=O)C2)coc(C#N)c1 44631,C(=O)(C#CC(C)(C)CNC(c1cnn(C(C)C)n1)=O)NC(C#C)CC1CC1 44632,c1(CCC)ccc(C(=O)NC2(C)CC(NC(=O)CC(C)C3CCCCC3)C2)cc1 44633,C(=O)(C(C)(C=C)CC)NC1CC(CCC(=O)NC(CCC=C)C2CC2)C1 44634,c1(C(N2C(C)CC(C(=O)NCC3(Oc4ccccc4)CC3)C2)=O)ncc(Cl)cc1F 44635,C=C1COc2c(C(=O)NCCC(C)NC(C3(Br)CC3)=O)cnn2C1 44636,C1(C(N(CC(CN(C(CN(C(C)=O)C)=O)C)O)C)=O)CCCCCN1C 44637,CC1COc2ccc(C(=O)NC3CC(NC(=O)CO)C3)cc21 44638,C1(CC(=O)NC2(CC)CCCCC2)CCCN(C(=O)C(O)C2CC2)CC1 44639,C1(CC=C)(C(=O)NCCc2cn[nH]c2)CCN(C(C2C=CC=CC=C2)=O)C1 44640,C1(CC(N2CC(CNC(c3ccc(C(F)(F)F)nc3)=O)C2)=O)(CC)CCCCO1 44641,Cc1cc(=NC(C)c2ccc(Cl)c(Br)c2)[nH]c(=NCCSCCO)[nH]1 44642,c1(CNC(C(COCC)n2cc(-c3ccns3)nn2)=O)csc2c(F)cccc12 44643,c1(OC)cccc(C(=O)NCC2(F)CCN(C(=O)CC3C=CCC3)C2)c1F 44644,N1(C(CC(=O)NCC#C)=O)CCCC12CCCN(C(=O)CN(C)C(C)C)CC2 44645,c1(OC)cc(CN2CCC(Cc3cc[nH]n3)CC2)ccc1OCC(=O)O 44646,C(=O)(C1CCCc2n[nH]cc21)NC1CN(C(CCCCC)=O)C(CC)(COC)C1 44647,Cc1c(CC(=O)NCCCCNC(=O)C=Cc2cn(C)cn2)ccc(Cl)c1Cl 44648,Cc1noc(C(N2CCCC2CNC(=O)C(C2CCCO2)C2CC2)=O)n1 44649,Cn1cc(C(C(=O)NC2CCC2(C)C)NC(=O)Cc2cc[nH]c2)nn1 44650,C(CSC)(CCOC)(n1c(C(c2cnn(CC)c2)NC2C(CC)C2)nnn1)C1CC1 44651,C1(CC(=O)NC(CN(C(=O)CNC(c2ccc(C)s2)=O)CC)C)CC2CC1C2 44652,N1(C(c2cc(F)c[nH]2)=O)CCC2(CC1)CCN(C(C13COC(CCO1)C3)=O)C2 44653,c1(OC)cc(CC(N2CC(N(C(=O)C(C)C(C)C)C)C(O)C2)=O)ccc1Cl 44654,Cc1cnc2nc(C(=O)NC3(C)CCN(C(c4cc(C)nnc4O)=O)C3)nn2c1 44655,Cc1cc(C)nc(SCC(=O)NCC(C)CN(C)C(C2(F)CCCC2)=O)n1 44656,C=CC1CN(C(C2CC3(CCC3)C2)=O)CC1NC(c1cn(CC)nc1C)=O 44657,C1(C(N(CC(C)C#N)C2CC2)=O)CCN(C(c2ccco2)=O)CC1 44658,n1(CC)cc([N+](=O)[O-])c(C(=O)N(CC(C)NC(=O)Cc2cc(C)cs2)C)n1 44659,C1(NC(COc2cc(C)on2)=O)CN(C(c2cnn(C(C)C)c2C)=O)CCC1F 44660,C#CCC(C)(C(=O)NC(c1nn(C)cc1O)C)NC(=O)C(C)=CC 44661,c1(C(=O)OCc2cccc(C(F)(F)F)c2F)nnn2c1COCC2 44662,Cc1ccc(C(F)CC2CCN(C(=O)C(=O)NCCC3CCC3)CC2)cc1C 44663,CN1C(=O)NCC1C(=O)NCCOCCNC(C1OC2CCC1C2)=O 44664,N1(C(C(CC)=CCCC)=O)CCN(C(C23CC(C)C2C3)=O)C(c2nccn2C)C1 44665,C1(C)(CCNC(c2nn(CC)c(C)c2)=O)CCN(C(=O)C(C)c2ccsc2)CC1 44666,c1(C(=O)NC(C2CCCCCC2)(c2nn[nH]n2)C)c(Br)ccc(F)c1I 44667,C(CCO)(CC(C)C)NC(c1cc(CNC(c2cc(COC)no2)=O)nn1C)=O 44668,C1(NC(Cc2nc(C)on2)=O)CCC(CNC(=O)CCc2ccc(O)cc2)CC1 44669,C(CCS(=O)(=O)c1ccccc1)N(CC(=O)NC1CCCC(C(N)=O)C1)CC 44670,c1(C(N2C(C)C(NC(C3CCC=CO3)=O)CCC2)=O)cc2ccccc2s1 44671,CCC1=C(C(=O)N2CCN(C(C3CC3C(N)=O)=O)C(C3CC3)C2)CCCO1 44672,C1(C(N2CC(F)(CNC(c3c(CC)ccs3)=O)C2)=O)CCCC2(CCC2)O1 44673,C#CCCCC(C)C(=O)N1CC(N(C)CCNC(=O)CC(=O)N(C)C)C(C)C1 44674,C(C(C)(F)C(C)(C)F)n1cc(C2C(C)CCN2C2(c3ncnc(O)c3F)CC2)nn1 44675,C(=O)(CC(Cc1cccc(F)c1)NCc1cnc(-c2cccs2)s1)OC 44676,c1(OC)cc(CCNC(=O)C(c2ccc(Cl)c(F)c2)O)cc(Br)c1 44677,c1(C(N2C(C)C(NC(c3csc4cncn34)=O)CCC2)=O)cccc2oncc12 44678,S(=O)(=O)(c1ccc(C#N)c(N2CC=C(C)C2)c1)N(C(CC)CSC)C 44679,Cc1cc(CCC(=O)NCCC(C)NC(=O)C(C(C)C)c2cccnc2)n(C)n1 44680,N1(C(C2CNC(=O)O2)=O)CC2CCCC1C2c1cn(Cc2c(F)cccc2Cl)nn1 44681,Cc1ccc(F)c(N)c1C(N1CCN(C(=O)CC2CC3(CCC3)CO2)C(C)C1)=O 44682,C(C(=O)N1CC(O)CC1CC(=O)NC1CC(CO)C2CC12)(C(C)C)SCC 44683,N1(C(c2cc(OC)c(C)cc2)=O)Cc2ccnn2CC(NC(=O)CCC(C)C)C1 44684,N1(C(C2(CC)CC2C(F)(F)F)=O)CCN(C(=O)CCC(C)C)CC1C1CC1 44685,N1(CC(=O)NC(C)(COc2ccccc2)CO)CC2(CCC2)CC1CO 44686,C(C(CO)C(F)(F)F)NC(c1sc(Cl)cc1Br)c1n(CCCOC)nnn1 44687,N1(C(=O)COCC2CCC2)CCOCC1CNC(C1(CO)CCCO1)=O 44688,N1(C(Cc2c(C)cco2)=O)CCCC(C)C1CCNC(c1cocn1)=O 44689,N1(C(C(C=C)c2ccccc2)=O)CCC(CC)C1CNC(c1cnc(S)n1C)=O 44690,c1(C(=O)NC2(CC=C)CN(C(=O)CCc3ccco3)C2)cccc2ccncc12 44691,C12(C(N3CC(NC(C=CC4N(C)CCC4)=O)C(C)C3)=O)CCCCC1CCC2 44692,c1(C(N2C(CC(=O)NCCCCOC)CCCC2)=O)cccn2ccnc12 44693,N1(C(c2c(CC(C)C)c[nH]n2)=O)CC2CCC(C1)N2C(=O)COC1CCC1 44694,C1(NC(C(=O)NCCOC)=O)C=CCN(C(=O)C(O)Cc2ccc(OC)cc2)C1 44695,N1(C(CC(=O)OCC)=O)CC(NC(c2ccc(C(C)C)o2)=O)CC2(CCC2)C1 44696,C1(NC(c2c(C)nn[nH]2)=O)CN(C(=O)CCSC(F)(F)F)CCC1F 44697,Cc1nnc2n1CCC(N=c1[nH]c(=N)[nH]c(=NCCOCCF)[nH]1)C2 44698,Cc1ccc(-n2cc(C(=O)NC(=O)CC(=O)OCC3CC(F)(CO)C3)nn2)cc1 44699,C1(CNC(c2c(CC)ocn2)=O)CC(C)(C)CN1C(c1cc(C#N)oc1C)=O 44700,C1(C(=O)NCC=CCNC(C2(CCc3ccccc3)CC2)=O)CCCCC1.COC 44701,C#CC1CN(C(c2sc(Br)cc2C)C(=O)NC(C)(C)CC)CC1O 44702,CC1CN(C(=O)CN(CC(C)(C)C)C)CC(C)N(C(c2ccoc2)=O)C1 44703,N1(C(c2c(CC)noc2)=O)CCC=C(C(=O)N(C2CCCC(C)C2)C)C1 44704,c1(C(N2CC3C(CNC(C4CC(=O)OC4)=O)C3C2)=O)ccc2nnn(O)c2c1 44705,CC1(CNC(c2ccc(C#N)o2)=O)CCCN1C(C1CCCOC1C(F)(F)F)=O 44706,c1(NC2C(NC(c3c(C)cc(C)s3)=O)CS(=O)(=O)C2)ncc(S(C)(=O)=O)cc1Cl 44707,C(C(=O)NCCC1CCN(C(=O)C(CC)N(C)C)C1)(C(C)C)NC(COC)=O 44708,C=CCC(F)(F)C(=O)N1CCCC1C(C)(C)CNC(=O)Cc1ncoc1C 44709,Cc1cc(C(C)NC(N2CCCC2C2CCCOC2)=O)cc(C)c1 44710,N1(Cc2c(C)nncc2)CC2CC1CN2C(=O)C(N1CCCCC1)=O 44711,C1(NC(C23CCC2CC3)=O)CCN(C(c2ccc(COC)cc2)=O)CC1CC1CC1 44712,c1(NC(CC2CCN(Cc3c(C)cc(F)cc3C)C2)=O)ccc(C#N)cc1C#N 44713,O=C(C1=CC2CC=CCC12)NCC(CNC(C1(O)CC(F)(F)C1)=O)CO 44714,C1(F)(CNC(=O)C=C(Cl)Cl)CCC(NC(c2cccc(C(F)(F)F)n2)=O)C1 44715,C1(NC(c2c(SC)cc(F)cc2)=O)COC2(CCN(C(c3ccsc3)=O)C2)C1 44716,c1(NC(CCc2onc(-c3c(Cl)cc(C#N)s3)n2)=O)cc2cc[nH]c2cn1 44717,CC1CCC(NC(=O)Cc2ccc(Cl)nc2)CN1C(c1cc(C2CC2)nn1C)=O 44718,N1(C(=O)CC2CCSC2)CCCCC2(CCN(C(c3ccncc3O)=O)C2)C1 44719,C1(C(=O)NCCCCCNC(C(C)OCCOCC)=O)CC2CC1CC2(F)F 44720,N1(c2nc(NC(CC)C)c3c(n2)scc3)C2CCC1c1ccccc12 44721,c1(C(=O)NCC(C)NC(C(C2CCCCC2)OC)=O)c(C)cc(Br)cc1C 44722,N1(C(C2CCC(C)O2)=O)C2CCC(C2)C1CC(=O)NCCCO 44723,CC1(C)OC(C(=O)NCC(O)CNC(=O)Cc2cccc3nsnc23)C(C)(C)O1 44724,C1(NC(COc2cc(C)on2)=O)CN(C(=O)C(C)C2CC2)CC1C(F)(F)F 44725,CC1(C(=O)NC(CNC(=O)C=C2CCC2)C2CC2)CCC(=O)N1 44726,CC(N=[N+]=[N-])C(=O)N1CCCC1C(C)NC(C1C2CCCOC12)=O 44727,CC(C)(C)CC(F)C(=O)NC1(C)CCCCC1C(=O)NCc1ncc(CO)[nH]1 44728,C1(NC(C(C)Cn2ccnc2)=O)CC2(CCN(C(=O)C3=CCCC3)CC2)C1 44729,C1(OC)CCC(NC(=O)C(c2ccoc2)NC(=O)CC2CCCO2)C1 44730,C1(OC)CCN(C(=O)CCC2(C)CN(C(c3ccns3)=O)C2)C1C 44731,C1(O)(CNC(c2cc(C(F)(F)F)cc(O)c2)=O)CCCN(C(=O)C=CBr)C1 44732,c1(OC)c(C(=O)NC2CN(C(=O)C(C)C#N)C2)csc1C 44733,C(=O)(CC1=NN(C)C(=O)C1)N1CCC2(C(C(=O)NC(CCOC)CO)C2)C1 44734,c1(C(c2n(CC)nnn2)NC(C2(C)COC2)C)ncc2ccccc2n1 44735,N1(Cc2occc2)CCC(NC(=NCC2CCCO2)NC2CCCCC2)CC1 44736,N#CC1(C(N2CCC(CC(C)NC(=O)C3=CCCOC3)CC2)=O)CC12CCCC2 44737,c1(OC2CN(CC)C2)ccc(S(=O)(=O)N(C(C)CCCl)C)cn1 44738,n1(CC)cc(Br)c(CC(=O)NC(CNC(=O)Cc2cncs2)C2CC2)n1 44739,CC(C)(C)CC(CO)NC(=O)CCCNC(=O)CC1CC(C2CC2)C1 44740,c1(C(N2CCC(c3ccccc3F)C2)=O)ccc(-n2ccnc2)cc1[N+](=O)[O-] 44741,C1(N(C(=O)Cc2cccnc2)CC)CCCN(C(c2ccc(Cl)cn2)=O)C1 44742,Cc1ccc(S(C)(=O)=O)cc1S(=O)(=O)N(C(CO)C(C)C)C1CC1 44743,c1(NC(C2CC(NCc3cc(C(=O)O)cc(Br)c3)C2)=O)nccc(Cl)c1Cl 44744,O=C(CCS(=O)(=O)Cc1ccccn1)NCC1CC(O)CN1C(=O)CC1CCC1 44745,N1(CCC)CCCC1C(=O)NCCC(=O)NCc1cc(C(=O)OC)co1 44746,c1(C(=O)NCC2CC(NC(CC3CCC(C)C3)=O)C2)csc(=NC2CC2)[nH]1 44747,c1(OC)cc(OC)cc(C(=O)NC(CNC(=O)C(C)OC2CCCC2)CC)c1 44748,C1(C(NOC(CC)C)=O)CN(C(C2CC3CCCC3C2)=O)CCN1C 44749,N1(C(c2ccc(OCC=C)cc2)=O)CCC(NC(c2cc(C)ns2)=O)C(F)C1 44750,S(=O)(=O)(c1ccc2[nH]c(=NCC(C)(C)C(N)=O)sc2c1)NCc1c(OC)cn(C)n1 44751,c1(C(N(CC(C)NC(c2c[nH]nc2Br)=O)C)=O)ccc(O)cc1F 44752,n1(CC)c(C(=O)NC(C)CNC(c2ccoc2Cl)=O)nc2ccccc12 44753,N1(C(C2C3COCC23)C)CC2CN(C(=O)COc3cccc(F)c3)CC2C1 44754,c1(Cc2cc(C(=O)NC(C)CCC3CCCO3)n[nH]2)ccccc1F 44755,C1(CC(=O)N(C)Cc2nnc(CC)o2)CCCC(NC(c2cscc2C)=O)C1 44756,c1(CNC(C(COC)(F)F)=O)cc(OC)ccc1OC1CCCC1 44757,C#CCC(CC(=O)NCCC(C)N(C)C(c1cnn(CC)c1)=O)c1ccccc1 44758,c1(C(=O)OC)cccc(CC(C)C)c1.CCC1CNC(=O)N1 44759,N1(C(C(C(COC)C)C)=O)CCCC2(C1)CN(C(=O)COc1cccc(F)n1)C2 44760,c1(CNC(CC2N(C(c3cn(CCOC)nn3)=O)CC2)=O)ccc(C)cc1C 44761,c1(C(N2CCCC(CNC(CC(C)SC)=O)C2)=O)cnn2c1S(=O)(=O)NCC2 44762,c1(C(=O)NC(CNC(c2cc(C)n(-c3ccccn3)n2)=O)C)cccc(N)c1C 44763,N1(Cc2ccc(N(C)C)s2)CCC(c2cc(N)ccn2)CC1 44764,C1(C(N2C(C(=O)NCCCC(C)O)CCCC2)=O)CC2CC1CC2O 44765,CCC(C)CC(=O)N1CC(CCNC(=O)COC(C)(C)C)C(C)C1 44766,N1(C(c2ncnc(C)c2C)=O)CCCC2(NC(C34CC(F)(C3)C4)=O)CC2C1 44767,N1(C(C)=O)CCc2cc(C(=O)NCC(CO)NC(=O)CN(C3CCC3)C)ccc21 44768,C1(CNC(C2CCC2)=O)CN(C(c2ccc(C(F)(F)F)nn2)=O)C2CCN1C2 44769,C(=O)(CCCC(CC)NC(=O)CCc1ccoc1)NC(C#C)(C)C1CC1 44770,C(=O)(CC(C)(C)CNC1CCC(=O)C1)NCc1c(COCC)occ1 44771,N1(C(C(C)N(C)C)=O)CCCC1(C)CNC(C1CCCC2CC12)=O 44772,c1(C(N(CCCC)C(C2CCC(C(C)C)CC2)=O)C)cccc(S(N)(=O)=O)c1 44773,c1(-c2nnn(CC(N3CCCC3C3CC3)=O)n2)ccc(Br)cc1 44774,N1(C(Cc2nn(C)c(Cl)c2)=O)CCC(C2CN(C(=O)CC(=O)NC3CC3)C2)CC1 44775,C1(CNC(c2ccc(C)o2)=O)N(C(c2ccc(F)c(Cl)c2)=O)CCC1(C)C 44776,Cc1nc2nccc(C(N3CC(C4CN(C(=O)CC(C)C(F)F)C4)C3)=O)n2n1 44777,N1(C(C2(SCC)CC2)=O)CCCCC(CNC(c2cc3sccc3[nH]2)=O)C1 44778,N1(C(Cc2ccn(C)n2)=O)CCC(CO)(CNC(C2CCCC23CC3)=O)CC1 44779,S(=O)(=O)(c1ccc(NCCC(C)CC(C)(C)C)c(C#N)c1)N1CCC(CSC)C1 44780,c1(C(=O)NCCN(C(C(C)=C2CC2)=O)C)cccc(SC(C)C)c1 44781,Cc1ccc(C(=O)NCc2nc(C(=O)N(C(C)(C)CO)C3CC3)c(C)o2)cn1 44782,c1(C(=O)NCC(C(C)C)NC(=O)C(F)C2CCCC2)cnn2cccnc12 44783,CCC(CC)C(C(=O)NCC(CCC)C(=O)N1CC(O)(C(F)(F)F)C1)OC 44784,CCC(C(=O)NC(C1(O)CN(C(c2cc(C)cs2)=O)C1)C)N(C)C 44785,N1(C(C2CC(=C)C2)=O)CCC2(NC(=O)COCC)CC2C1.c12ccccc1O2 44786,CCC(CNC(=O)CNC(c1ccccn1)=O)(CC)NC(=O)C(C)C#N 44787,C(CCC(O)C(=O)N1CCCC(O)C1)NC(c1c(CC)ocn1)=O 44788,O=C(O)CC(C(=O)O)NC(=O)NCC12COC(CF)(C1)C2 44789,c1(C(=O)NC2CCCN(C(C=CC(C)C)=O)C2)ccc(C(F)(F)F)c([N+](=O)[O-])c1 44790,Cn1nnc(C(=O)NCCCC(C)(C)NC(C2CC3(CC3)C2)=O)c1C(F)F 44791,C(=O)(C1=CCCSC1)NCc1cncc(C(=O)NC(CCCC)CC)c1 44792,O=C1C2CC3C(C2)C13C(=O)NC1CC(n2cc(CC(O)C3CC3)nn2)C1 44793,Cc1cn2c(n1)CC(C(=O)NCCCCCNC(C1COCCC1(F)F)=O)CC2 44794,n1(CC(=O)N(C2CCN(C(CC(C)(F)F)=O)CC2)CCO)ccc(O)nc1=O 44795,c1(-n2cc(C(=O)OCC)nn2)cnccc1C(c1nccn1C)NC(=O)C1CC1 44796,C(=O)(CCCS(N)(=O)=O)NC1(CCNC(C(c2ccc(CC)cc2)C)=O)CC1 44797,c1(C(=O)NCCC(C(C)C)NC(c2c(OC)cncc2)=O)n[nH]c2c1CCOC2 44798,Cn1nc(Br)cc1C(=O)NCCNC(C1CCC(NC23CC(CO2)C3)CC1)=O 44799,C1(C(C(=O)N(CCNC(c2ccc(C(C)O)cc2)=O)C2CC2)O)CCC(C)(C)CC1 44800,CC1CN(C(c2cncn(C)c2=O)=O)CCC1N(C)C(c1ccc([N+](=O)[O-])[nH]1)=O 44801,C(C)(CCC(=O)NCCOCC(C1(c2ncccc2Cl)CC1)=O)OC.C1CCS1 44802,C1(F)(CNC(c2n(C)ncc2)=O)CCCN(C(C2CC(=O)N(CC3CC3)C2)=O)C1 44803,N1(C(c2ncn(C)c2)=O)CCC2(CC1)CN(C(c1cc(F)nn1C)=O)C2 44804,N1(C(C(C)OCCCC)=O)CCCC(CCNC(C2(O)COC2)=O)C1 44805,C1(N(C(COCC(=O)NC)=O)C)CCC2CN(C(C34CCC(CC3F)C4)=O)CC12 44806,N1(C(Cc2cc(C)on2)=O)CCN(C(c2ccc(O)cc2C(F)F)=O)C2CC12 44807,N1(C(c2c(CNC(C(CCSC)O)=O)cnn2C)=O)CCN(C)C(=O)C1 44808,C(=O)(CCCC(F)(F)F)N1C(CNC(c2ccc(C(F)F)nc2)=O)CCCC1 44809,c1(CCC(=O)OCC)nc(O)c2c(C)c(C)sc2n1.C1(=O)C(C)N1C(CC)=O 44810,C1(NC(C(CC=C)NC(C)=O)=O)CC2CCC1CN2C(=O)C(C)OCC(C)C 44811,C12(CNC(CC(C(C)C)C)=O)CCC(NC(=O)COC(F)F)(CC1)CO2 44812,N1(C(C2(NC(CCCOC(C)=O)=O)CCSC2)=O)CC(CO)C(C2CC2)C1 44813,C1(CC)(NC(=O)CCCCc2cccc(O)c2)CCCN(C(C2CCC2)=O)C1 44814,C1(C(C)NC(C(C)c2cn[nH]c2)=O)CCCN1C(=O)Cc1cnc[nH]1 44815,C12(NC(c3cocn3)=O)CCCC1N(C(=O)CCc1ccccc1)CCC2 44816,C(=O)(CC(C(C)OC)NC(c1c[nH]c(=O)cn1)=O)N(C(C)C(C)C)CC 44817,N1(C(=O)Nc2nc(=N)[nH][nH]2)CCNCC1c1cccc(Cl)c1 44818,c1(CN)ccc(CCNC(=O)CCNc2ccc(-c3cccs3)cc2)cc1 44819,N1(C(C(COC)(F)F)=O)CCCCC(N(C(=O)Cc2cnn(C)c2C)C)C1 44820,N1(C(CN2CCN(C)CC2)=O)Cc2nccn2CC(NC(C2CCSCC2)=O)C1 44821,c1(C(C(=O)NCC2CC(NC(C3C(CC)OCC3)=O)C2)O)ccc(Cl)cc1 44822,C1(C(=O)Nc2cccc(CNC(C(C(=O)OC)OC)=O)c2)CCC2(CC1)CC2 44823,N1(C(Cc2cn(CC)nn2)=O)CCC(CNC(c2cnn(C)c2Cl)=O)C1(C)C 44824,N1(C(Cc2c(C)nc(C)s2)=O)CCCC(N(C)C(c2cnc(C3CC3)[nH]2)=O)CC1 44825,C(CCCCCC)(C(=O)NC(C)(C)CC)N1C(CCC)(CC)CCC1 44826,N1(C(c2ccc(CC)cc2)=O)CC(NC(=O)COCCOC)C2(CC2)C1 44827,C12(C(=O)NC(C)C(C)NC(c3ccc(O)nn3)=O)CCCN(CCC1)C2 44828,C(CC(C(=O)NCc1ccc(CO)o1)NC(=O)CC(O)c1ccccc1)OC 44829,CCC(C)(CNC(=O)CCC1CCCCO1)C(=O)N(C)CC1CCCS1 44830,O=C(C1=CCOC1)NCC1CN(C(=O)COc2ccc(F)cc2)C2CC12 44831,C(=O)(CCCC(=O)C1CC1)NCC1C(CNC(C(n2c(C)cc(C)n2)C)=O)C1 44832,c1(SC)cccnc1C(N1CCC(NC(c2cnc(O)o2)=O)CC1)=O 44833,N1(C(C(CC=CCC)C)=O)CCC2(CCC2NC(c2ccoc2C)=O)CC1 44834,N1(C(c2nncc(CCC)c2)=O)CCCCCCC1C(=O)NC(C)CC(N)=O 44835,C(CC1CC1)(C(=O)NCCOCCC(=O)N(C1CCOC1C)C)OC 44836,CCC(C)C(C(=O)NC(C(=O)NC1CC(C#N)C1)C1CC1)NC(=O)NC 44837,c1(C(=O)NCC23CC2CN(C(=O)Cc2nc[nH]n2)C3)cc2ccc(F)cc2[nH]1 44838,CC(CCN(C)C)C(=O)NC(C)CC(C)NC(=O)C(CCSC)N(C)C.N(C)C 44839,c1(OCC=C)ccccc1C(=O)NCCOCCCNC(c1c(C)nsc1N)=O 44840,C1(C(=O)NC(c2ncccn2)CC)CCN(C(=O)CS(=O)CC)CC1C 44841,c1(CC(=O)NCC2N(C(C(CC)F)=O)CC=C2)cc(C)cc(Br)c1 44842,CCC(O)C(C)(C)C(=O)NC1CC(C(=O)NCC2(CO)CCN(C)C2)CC1O 44843,C(=O)(CS(=O)(=O)NC)NC(CCC)CNC(C1CC2CC2C1)=O 44844,c1(C(=O)NC2C3CC2N(C(=O)C(F)OC(F)(F)F)C3)cc(F)ccc1F 44845,N1(C(C2N(C(CCN(CCC)C)=O)CC2)=O)CCCC1CC(N)=O 44846,CC1CC(NC(=O)CCc2nccs2)CN1C(c1ccccc1O)=O 44847,N1(C(C2N(C(CNC(C=C)=O)=O)CC(C)C2)=O)CCC(O)C(C)C1 44848,CC1(CNC(=O)C(C2(O)CCC2)NC(=O)CCc2ccccn2)CCCOC1 44849,C1(NC(=O)CCc2cncs2)CC1C1CCCN(C(c2cc(Cl)cs2)=O)C1 44850,C1(CN)C(CNCCC(O)C2CCCC2)C1(F)F 44851,C1(CN(C(C(c2ccccc2)SC)=O)C)CCCN1C(C1CN(C(N)=O)C1)=O 44852,N1(C(C2CC(CCNC(C#CC(C)C)=O)C2)=O)CC(C)(C)CC1CO 44853,N1(C(C2N(C(c3ccc(C#N)s3)=O)CC=C2)=O)CCCNC(=O)CC1 44854,O=C(Nn1ccccc1=O)C1CN(C(c2ncc[nH]2)=O)CC12CC2 44855,N1(C(CCn2ccc(C)n2)=O)CC2CCC2(CCNC(c2cc[nH]n2)=O)C1 44856,N1(C(CC)=O)CCN(C(=O)CNC(c2cccs2)=O)C2COCC12 44857,C(CS(=O)(=O)CC(=O)NC(C)(C)CC=CC(=O)NCCCN(C)C(C)=O)OC 44858,CC(CC(C)(F)F)C(=O)NCC=CCNC(=O)CCCc1nncn1C 44859,c1(C(=O)OC)ccc(NS(=O)(=O)NCC2CC(F)C2)cc1 44860,C(=O)(C(C)CC1CC1)NC(c1nc(C(=O)N(C)Cc2cn[nH]c2)co1)C 44861,C=CC(C)(C)CCN(Cc1ccnn1C)Cc1ccccc1C 44862,C1(NC(C(C(C)C)n2cnnc2)=O)COC2(CNC(=O)C=CC3CCC3)CC1C2 44863,C1(N(C(=O)C(C)C2CC2)CCC)CCN(C(c2cnn(CCF)c2)=O)C1 44864,Cc1ccc(C)c(C(=O)NC(C)CC(C)NC(=O)C=Cc2ccc(=N)[nH]c2)c1 44865,N1(C(c2c(C)cccn2)=O)CCCC(C2CC2NC(=O)CCC(F)F)C1 44866,N1(C(c2c(OCC)scc2)=O)CC(CNC(C2(CF)CC2)=O)CC1C 44867,c1(C(=O)OC)cc(F)cc(F)c1NCc1cnc(C(C)(C)C)s1 44868,C1(CC=C)(NC(c2ccc(OC)nn2)=O)CCCN(C(c2nsnc2O)=O)C1 44869,C=C1CC2(C1)CC(C(=O)NCC(C)NC(=O)CNc1cc(OC)ccc1OC)C2 44870,C#CCCC(O)C(=O)NC1CCC(NC(=O)CC2CCC(C)(O)CC2)CC1 44871,N1(C(c2cncc(C)n2)=O)CCC(NC(c2ccnc(Cl)c2)=O)C1(C)C 44872,C12(NC(=O)Cc3nc(F)c(F)cc3F)CCCN(C(c3cnsc3)=O)CC1C2 44873,C1(C(=O)NCC)CN(C(=O)C(=O)Nc2cnc(O)cc2OC)CCC1C 44874,N1(C(CCCC=C)=O)CCC(C(=O)N(CC(CC)OC)C)(CC)CC1 44875,C(N(C1CC1)N1CCCCC(F)(F)C1)c1ccc(OC(F)(F)F)cc1 44876,CCS(=O)(=O)c1ccc(S(=O)(=O)NC2c3ccccc3C3CC23)cc1 44877,C1(CC)CN(C(c2cc(C)ncn2)=O)CC1C(=O)NC(CC1CC1)C1CC1 44878,CC(CC(=O)N1CCC(=C(F)F)CC1)C(C)(C)C.N1CC2CCC(C1)O2 44879,c1(C(C(=O)N(CCCCNC(=O)C(O)CC2CC2)C)(C)N(C)C)ccc(F)cc1 44880,N1(C(CCCCOC)=O)CC2CCCC(CNC(=O)Cc3nnc(C)o3)C2C1 44881,c1(CC)cc(C(=O)NCC(O)CCNC(=O)COc2cccc(F)c2)ccc1C 44882,C(c1ccccc1F)=CCC(N1CCC(NC(c2cc(C#N)no2)=O)(CO)C1)=O 44883,C(=O)(C1OCCc2c(Br)cccc21)N1CC(C)(C)c2c1cncc2 44884,C(=O)(C#CC1CCCCC1)NCCCN(C(C1CCC(C)S1)=O)CC 44885,c1(CC)cc(C)nc(N2CCC(NC(=O)C(C)OCC3CCCCO3)C(C)C2)n1 44886,CCCCCCC(=O)N(CC(O)CN(C)C(c1[nH]nnc1COC)=O)C 44887,CC(=Cn1ccnn1)C(=O)N1CC2(CCN(C(c3cc4n(n3)CCO4)=O)C2)C1 44888,CCCCC(O)C(=O)NCC1COCC1NC(=O)Cn1ccnn1 44889,C1(CNC(CCC)(CC)c2nnnn2-c2ccccc2C)CCN(C)C(=O)C1 44890,c1(C(C)C)cc(S(=O)(=O)Nc2c[nH]nc2C(F)(F)F)c(Cl)cc1Cl 44891,c1(CC)cc(OCC(=O)NC2COCCC2NC(=O)CCCC(C)=O)ccc1Cl 44892,c1(OC)cc(C)ccc1OCC(=O)NC(C)CCCNC(=O)Cc1cc(C)on1 44893,c1(C(N(C)CC2CCCCN2C(C2CC23CCC3)=O)=O)c(F)cc(F)c(F)c1F 44894,O=S(=O)(c1c(Cl)cc(Br)cc1Cl)Sc1nc(C2CC(=O)OC2N2CCCC2)no1 44895,c1(OC)ncc(CO)cc1F.c1(-c2c(OC)ccnc2)cnc2cc1C(=O)N2 44896,C1(CNC(c2c(C)cns2)=O)CC2(CCN(C(C3COCCN3C)=O)CC2)CO1 44897,C1(C(N2CCCC(N(C(c3c(CC)scc3)=O)C)C2)=O)CCc2ncncc2C1 44898,c1(C(N(CC(C)N(C(C(C)n2cnnn2)=O)C)C)=O)c(O)nnc2c1COCC2 44899,C12(NC(Cc3c(C)nc(C4CCC4)s3)=O)CCN(C(=O)C(C)(C)C3CC3)CC1C2 44900,C1(N(C(CC2C(C)C2)=O)Cc2cc[nH]n2)CCCN(C(c2cncc(N)n2)=O)C1 44901,C=CC(F)(F)C(=O)N1CCC1CNC(c1ccc(C(C)(C)C)cc1)=O 44902,N#CC1CC12CCN(C(C1(F)CCN(C(C3CCNC3=O)=O)C1)=O)CC2 44903,C12(CNC(c3nc(COC)sc3)=O)CCC(CC1)N2C(c1cnn(CC)c1Cl)=O 44904,c1(CC(=O)NC)ccc(C(=O)NCCC(O)CNC(c2ccc(C)o2)=O)cc1 44905,c1(C(C)=O)cncc(C(=O)NC(CNC(=O)CCc2c(C)noc2Cl)CO)c1 44906,N1(C(c2c[nH]c(=N)o2)=O)C2CCC1C(NC(c1cc(Cl)c(Cl)s1)=O)C2 44907,CC(C)(C)CCCC(=O)N1CCN(C(c2ccc(C#N)[nH]2)=O)CC(CO)C1 44908,c1(C(C)NC(c2c(Br)cnn2C)c2n(CCOC)nnn2)ccc(F)cc1 44909,c1(OC)nccc(C(=O)NCC2CCCC2NC(C2C3CCCC23)=O)c1F 44910,CC(C)C(O)C(F)(F)C(=O)NC(C1CN(C(=O)C(C)O)C1)C 44911,C1(NC(c2cn3ccsc3n2)=O)CN(C(=O)C(Cl)=CCl)C2(CCCC2)C1 44912,C(CC)(C(=O)NCC(C)(F)F)NC(C(F)=CCC)=O 44913,Cc1cc(=NC(C)c2ccc(C)o2)[nH]c(=NCCC(=O)N(C)C)[nH]1 44914,C(C1=CCC2CC1C2(C)C)(c1nnnn1C)Nc1cccc(C(C)F)c1 44915,N1(C(Cc2c(C)noc2)=O)CCN(C(C23CC(CO)(C2)OC3C)=O)C(C2CC2)C1 44916,C1(CC)(NC(C2CCCCC2)=O)CCCN(C(C2CCS(=O)(=O)N2)=O)C1 44917,c1(C(=O)NC(CC=C)CNC(c2c(C)ncnc2O)=O)cnc2n1CCCC2C 44918,N12CC(C(F)(F)C1)C(=O)C2.c1(CC(C)C)ccccc1N(C)C 44919,c1(CNC(C(CC)NC(N)=O)=O)ccccc1CN(C)C(C1(F)CCC1)=O 44920,c1(C(C)=O)c(C)[nH]c(C(N2CCC(O)C(NC(=O)CC=C(Cl)Cl)C2)=O)c1C 44921,c1(COC)ccccc1C(=O)NCCCN(C(=O)CCC(=O)OC)C(C)C 44922,c1(NCC2C(NC(c3c(CC)ocn3)=O)CCCC2)ncc2cccnc2n1 44923,C1(NC(CC2(CNC(Cn3ncc(CC)c3)=O)CC2)=O)CCCC1N=[N+]=[N-] 44924,n1(CCC)nccc1C(=O)NCC1(C(C)NC(c2cc(C(C)=O)on2)=O)CC1 44925,c1(OCC)cccc(OC(=O)C(C2CCCCC2)NC(C2C3CCCC23)=O)c1 44926,N1(C(c2c(OC)cccc2C)=O)CC2CC3CC2C1C3NC(=O)C=C(Cl)Cl 44927,c1(OC(C(C)C)C(=O)NC2CCN(C(=O)CN(C)CCO)C2)ccc(F)cc1F 44928,N1(C(c2scc(COC)c2)=O)CC2(CCN(C(C34CCC(CC3)C4(C)C)=O)C2)C1 44929,c1(CNC2C(NC(C34CC(C(=O)OC)(C3)C4)=O)CCCC2)c(O)ccc(F)c1F 44930,c1(C(=O)NCCC(C)N(C(CCCN(C(C)C)C)=O)C)c(F)cc(O)cc1F 44931,CC(C)(C(=O)N1CC2CCC(NC(C3CCCSC3)=O)(C2)C1)S(C)(=O)=O 44932,c1(C(N2CCC(CNC(c3occc3Br)=O)C2)=O)ccc2c(c1)OCCC2 44933,C1(CCC)CCC(C(=O)NCC2(C(N)=O)CN(C(C3NC(=O)CC3C)=O)C2)CC1 44934,CCC(F)(CNC(=O)CC1CCCCN1C(=O)CCCOC(C)=O)CC 44935,N1(C(C2C(c3ccc(C)s3)C2)=O)CCC(C)C1CNC(=O)CC1OCCC1C 44936,Cn1cnc(C=CC(=O)NC2CCC2NC(=O)C(=O)NCc2ccccc2)c1 44937,C1(CNC(C2(C)CC2)=O)CCN(C(=O)C(c2ccc(Cl)cc2)(F)F)CC1O 44938,n1(CC)nccc1C=CC(N1CC(CNC(=O)Cn2ccccc2=O)C(C)C1)=O 44939,C(=O)(C1=COCCO1)NC1C(C2CCN(C(C(CC)=CC)=O)CC2)OCC1 44940,C1(CN(C(C(C)OC)=O)C)CN(C(C2C3CCC2(c2ccccc2)C3)=O)CCO1 44941,c1(CC)c(C(N2CC(NC(=O)C(C)(C)COCC(F)F)C(F)C2)=O)csc1C 44942,Cc1nc(Cl)ccc1C(=O)NCC(O)CNC(C1CCC(O)CC1)=O 44943,Cc1[nH]nc2ncc(C(=O)NC3CN(C(C4CCC(=O)C4)=O)CC3O)cc12 44944,C1(C)(C(=O)NCCN(C(c2nccc(N)c2Cl)=O)CC)CCC(F)(F)C1 44945,c1(C(=O)NCC(C)N(C)Cc2ccc(N(C)C)nc2)c(F)c(F)c(F)c(F)c1F 44946,c1(CCC(=O)NCC(CCOC)NC(c2cocc2C)=O)ccccc1F 44947,c1(C(N(C)CC2(O)CCN(C(=O)CSCC(N)=O)C2)=O)oc2ccccc2c1Cl 44948,C1(CNC(CC2CC(C)C2)=O)Cc2ccccc2CN1C(=O)C1=COCCC1 44949,c1(C(=O)NC(C(C)C)CNC(=O)C(C)CF)cccc(N)c1N 44950,N1(C(c2nc(COC)oc2)=O)CC(NC(=O)C(O)C2CCC2)CC12CCOCC2 44951,C(CC(C)(C)CC(=O)NCc1nnn(C)c1C(=O)NC1CCN2CCC1C2)OC 44952,N1(C(CSCCNC(C2CC(=O)NC2)=O)=O)CCN2C(=O)NCC2C1 44953,c1(C(=O)NCCNC(C(C(C)C)CN(C)C)=O)cccc2ncnn12 44954,C12(C(=O)NC3CCC(C)NC3=O)C3C4C1C1C2C3C41c1nn[nH]n1 44955,c1(C(=O)NCC2N(CC(=O)NCC)CCCC2)ccc(OCC)c(F)c1 44956,n1(CC)ncc2c1CC(Nc1nccc(N3CCCC(CSC)C3)n1)CC2 44957,C1(NC(c2ncn(CC)c2)=O)CC(C(=O)NCCc2csc(C)n2)C1(C)C 44958,N1(C(C(CC(C)C)OC)=O)CCC(C)(C)C(CNC(=O)C=CC2CC2)C1 44959,c1(C(=O)NCc2ccc3[nH]ccc3c2)cc2ccc(-c3cn[nH]c3)nc2[nH]1 44960,CC1OC2(CO)CC1(C(=O)NC(C)CN(C)C(C1CC3CCC(C1)C3)=O)C2 44961,C(CCC(C(=O)NCC=C(Cl)Cl)NC(=O)C(C)C(C)C)OC 44962,C1(CCNC(=O)C(CO)c2ccccc2)CC2CCC(C1)N2C(c1nncs1)=O 44963,C1(C2CCN(C(=O)CN3C(=O)CCC3=O)C2)(NC(=O)Cc2nccs2)CC1 44964,C(=O)(C(CO)NC(C1CC(=C2CCC2)C1)=O)N(CC(C)OC)C 44965,C(CC(F)(F)F)N(C(c1cn(CCNC(c2n[nH]cc2C(C)C)=O)cn1)=O)CC 44966,N1(C(c2ccc(C(=O)OC)[nH]2)=O)CCN(C(c2cc(C)ns2)=O)CC(C)(C)C1 44967,CC(CC1CCCO1)C(=O)NCC1CCCN1C(c1cc(C(F)F)cs1)=O 44968,C1(C(=O)OC)COC2(CCN(C(=O)C(F)(F)Cl)CC2)C1.c12cc-1cc(F)c2 44969,c1(C(=O)NCC2(CO)CCC2)coc2c1CN(C(c1[nH]ccc1CO)=O)C2 44970,C(C(CCOC)NC(=O)CCCc1nc(CCC)no1)NC(C1C(=C)C1)=O 44971,C1(CC)CC(O)CN1C(c1csc(C)c1)C(=O)NC1CCCCC1 44972,N=c1[nH]c2c(s1)CCCC2NC(c1cc(F)c(O)c(Cl)c1)=O 44973,Cc1occc1C(=O)NCCc1cc(C(=O)NCC(C)(C)C#N)no1 44974,C(=O)(C(CCSC)NC(c1cccnn1)=O)NCC(=O)NCC=C 44975,O=C1CCC(CCC(N2CCCC2CNC(=O)CC2CSC2)=O)N1 44976,C1(c2cn(CC3N(C)CCC3)nn2)CCOCCN1Cc1cc(F)ccc1N 44977,C1(C(=O)NOC(c2cccc(C)c2)C)(C)CCC(=O)CC1.C(=O)OCC 44978,N1(C(CCN(C(=O)Cc2cnn(CC(=O)OC)c2)CC)=O)CC(C)CC1CC 44979,c1(C(=O)NCCCN(C(=O)CN2CSCCSC2)C)ccc2ncc(=O)[nH]c2c1 44980,c1(C(C)=O)ccc(OCC(=O)NCCN(C(=O)CC2CC3CC3C2)C(C)C)cc1 44981,N1(C(C2C(C)C2)=O)CC2CCC1C(CNC(c1cc(-c3ccncc3)no1)=O)C2 44982,CCCCC(C(=O)NCCCC(C)(C)NC(c1cccc(CF)c1)=O)NC(N)=O 44983,C(CC(O)CNC(=O)CNC(=O)C(F)(F)F)NC(CCSCCC)=O 44984,c1(NC(c2c(C)cc(I)cc2)=O)ccc2c(c1)ncn2C 44985,C1(NC(C(C2CC(C)(C)C2)OC)=O)CCOCC1NC(=O)CCc1cnoc1 44986,N1(C(Cc2c(C)nc[nH]2)=O)CCC(NC(c2sc(F)cc2Cl)=O)C(CO)C1 44987,C(CC(C)(C)C)(C(=O)NCCCC(C)(C)C)NC(c1ccc(C)cc1)=O 44988,Cc1nc(C(N2CCC(OCCNC(c3ccnnc3)=O)C2)=O)n[nH]1 44989,C1(C(N2CC(COC)(NC(=O)CC(C)N(C)C(C)=O)C2)=O)CC2CCC1CC2 44990,C1(O)(C(=O)NC2C(n3cc(C(C)N(C)C)nn3)CCCC2)CCCC(C)(C)C1 44991,C1(C(NOCC2CC3CC2C3)=O)(COC)CCCO1 44992,C(C)(CCCC(=O)NC(CO)CCC1CC1)NC(c1n(CC)nnc1)=O 44993,Cc1ccc(CC(=O)Sc2cccc(N3CCC(C(=O)O)C3)n2)c(C)c1 44994,c1(C(=O)NCCC(C)N(C(C(C)OCCC=C)=O)C)ccc(C(C)C)s1 44995,C1(C2CCN(C(=O)CC3CCSCC3)C2)(NC(c2cc(C)sn2)=O)CC1 44996,C1(NC(C2N(C)CCOC2)=O)CCCC2CN(C(C3(F)CC4(CCC4)C3)=O)CC12 44997,CN1CCC(F)(F)C(CNC2C3(NC(=O)OC(C)(C)C)C4CC2CC34)C1 44998,C1(C=O)CCC(C)=C(C)C1.C1(CNCC)C2CN(C(=O)CS(=O)(=O)N(C)C)CC12 44999,CC(CCNC(=O)CCCCNC(=O)C(C)n1cncn1)CCO 45000,C=CCC(C(=O)NC(C)CCNC(c1cc2ncccc2s1)=O)C(C)C 45001,C1(NC(CC(C)CF)=O)CCCC12CCN(C(c1cnn[nH]1)=O)CC2 45002,N1(C(C2C(C(C)(C)O)C2)=O)CCC(O)(CCNC(C23CCC(C)(C2)OC3)=O)CC1 45003,c1(CNC(C(C)(C)CCl)c2n(C3C(C)C3)nnn2)nc2c(s1)COCC2 45004,CC1CN(C(=O)CCC2OCCO2)CCC1NC(C1CCC2(CCC2)C1)=O 45005,Cc1ccc(C2(NC(=O)NC(c3nnc(-c4ccc(Cl)cc4)s3)C)CC2)cn1 45006,C(=O)(C#CC1CCCCC1)N1CCC(NC(C(C)SC(F)(F)F)=O)C(O)C1 45007,Cc1cc(CC(=O)NCC23CC(CNC(=O)C(C(C)C)N(C)C)(C2)C3)cc(F)c1 45008,CC(C)CC(C)(CNC(C1(C#N)CC1(C)C)=O)NC(c1cnc(C(C)C)s1)=O 45009,N1(C(c2cccc(CO)c2)=O)CCN(C(C2CCN(C3CC3)C2)=O)CC(O)C1 45010,C(=O)(CCCCC(C)C)N1C2(C(=O)NCC3(COC)CCC3)CC2CC1 45011,N1(C(c2n(C)nnc2)=O)CCCC(C2CC2NC(C2CCCN2S(C)(=O)=O)=O)C1 45012,c1(C(=O)NC2CC(NC(C3(CC)CC3)=O)C2)cc(=N)[nH]cc1Br 45013,C1(CCC2N(C(CCOC)=O)CCC2)CCN(C(c2cncn2C(C)C)=O)CC1 45014,c1(C(=O)NC2(CNC(CCOCC)=O)CC2)cccc2nn[nH]c12 45015,c1(OC)ccc(C(C(=O)NC(C)C2CC2)N(C)C(C)C)c(Br)c1 45016,c1(C(=O)NC23CC(NC(C(c4cccc(C)c4)C)=O)(C2)C3)cc(F)c(N)cc1F 45017,c1(C(=O)OC)cc(NC(c2ccc3c(n2)OCCO3)=O)cc2[nH]ccc12 45018,C1(NC(c2nc(CC)sc2)=O)CC2CC1CN(C(=O)Cc1ccc(Cl)s1)C2 45019,c1(C(=O)NC2CC(CNC(C3CC=CC3)=O)C(O)C2)ccc2oc(O)nc2n1 45020,C=C(C)C1OCCCC1C(=O)NCC1(OC)CCN(C(=O)CN(C)C2CC2)C1 45021,CC1CN(C(c2cccc(=O)n2O)=O)CCC1NC(c1cncc(Cl)c1)=O 45022,c1(OC)ncnc(OC)c1CN1CC2CC1C2C(=O)Nc1ncc(Br)s1 45023,C1(NC(c2c(C)cccc2F)=O)CC1C1CCN(C(=O)Cc2csc(Cl)c2)CC1 45024,N1(C(C(C)OCCC#C)=O)CCOC(C)(CNC(c2ccc(OC)c(F)c2)=O)C1 45025,C1(C(C)C)N(C(=O)CCCn2cc(CNS(N)(=O)=O)nn2)CC12CCC2 45026,C(c1ccc(C)cc1)=CCC(=O)NC1CN(C(C(=CC2CCCC2)C)=O)CC1C 45027,C1(N(C(=O)Cc2cnoc2)CC)CCCN(C(=O)CC2CC(F)(F)C2)CC1 45028,N1(C(c2nc(Br)cs2)C(=O)NCCCSC)CCC(CCO)CC1 45029,C(=O)(CC(O)CC(C)(C)C)N1CCN(C(CCCCN(C(C)=O)C)=O)C(C)C1 45030,C1(S(C)(=O)=O)(C(=O)NCC(C)N(C(=O)Cc2nc[nH]n2)C)CC(O)C1 45031,O=C1CC2(CN1)CN(C(C1CC3(CCC3)CN1C(c1coc(CO)c1)=O)=O)C2 45032,n1(CCC(=O)N(CCF)CCc2ccccn2)cc(COc2ccccc2)nn1 45033,CCCCC(O)C(=O)N(C(CNC(C1CC1C(C)(F)F)=O)C1CC1)C 45034,C1(CNC(C(C2CN(C(C(C(=O)OCC)F)=O)C2)O)=O)OC(=O)NC1(C)C 45035,CC(C)CCC=CC(=O)N(C(C)C(=O)NCC(F)C1CCC1)C 45036,N1(C(C(C)OCCN(C)C)=O)CCC(NC(c2cncc(N)c2)=O)CC1 45037,N1(C(C(C)O)=O)C2CCC1CN(C(=O)CCCCC(N)=O)C2 45038,N1(C(c2ccc[nH]2)=O)CCC2(CCC(CNC(C34CCCC3C4(F)F)=O)OC2)CC1 45039,Cc1cccc(Cl)c1OCC(=O)NC1CN(C(C2CC(C)N(C)C2)=O)CC12CC2 45040,n12cc(nn1)CC2.c1(CN(c2ccn(C)n2)C)cc(Cl)cs1 45041,Cc1cc(F)ncc1C(N1CCN(C(=O)CCCCCF)CC1C)=O 45042,N1(C(c2ccc(N(CCC)C)nc2)=O)CC(C)(C)CC1CNC(=O)C(C)N(C)C 45043,NS(=O)(=O)c1cc(C(=O)NC2CCCC2NC(C2CC2F)=O)c(Cl)s1 45044,c1(CN2CC(F)(C(=O)Nc3cc(CC)cc(Br)c3)C2)cc(Cl)c(O)cc1F 45045,N1(C(C(C)=C(CC)C)=O)CCN(C(C2(S(C)(=O)=O)CCC2)=O)CC1CC(=O)NC 45046,CC1(C(=O)NC2CCCN(C(=O)C(C)(O)C(F)(F)F)CC2)CCC(F)(F)CC1 45047,CC1CCN(C(C2C=CCCC2)=O)C1C(=O)NCC(F)Br 45048,C1(NC(c2ccc(OC)cc2)=O)CCC(C)N(C(c2ccc(F)c(Br)c2)=O)C1 45049,N1(CC#N)CCCC1C1CCCCN1C(c1cccc2nc(O)[nH]c12)=O 45050,C(CC1CCC1)(C(=O)NC1(C(=O)NCCCNS(N)(=O)=O)CC(C)C1)NC(C)=O 45051,c1(N2CCC(CC=C)(NC(c3cc(C4(C)CC4)n[nH]3)=O)C2)ncnc(Cl)c1CC 45052,c1(CNC(C(C)(C)C2CCCOC2)=O)ccc(P(C)(C)=O)nc1 45053,N1(C(CC(C)N(C(N)=O)Cc2ccccc2)=O)CC(C(=O)O)C2(CCNCC2)C1 45054,c1(OCC2C(CC)C2)cc(OC)cc(OC)c1.c12ccccc1C(CC(C)C)O2 45055,C1(NC(C(COCC)C)=O)CC2CC(NC(=O)CCC(C)C)C1C2 45056,N1(C(c2c(OC)nccc2)=O)C2CCC1C(C(=O)Nc1ncccc1C(C)=O)C2 45057,c1(C(=O)NC2CN(C(C3C(=C)CC3)=O)C(C)C2)ccc2nnn(O)c2c1 45058,C(=O)(C1=CS(=O)CCC1)N1CCCC(NC(CCC(=O)NC)=O)(CO)C1 45059,Cc1nn(C)c(C(F)(F)F)c1C(=O)NC1CCCN(C(=O)CC2(O)CCC2)C1C 45060,N1(C(C2CC(N(C(CC3(N(C)C)CC3)=O)C)C2)=O)CC2(CCC2(C)C)C1 45061,C1(CN(C(=O)CCc2cccc(O)n2)C)CN(C(=O)CC2CCC2)CC12CC2 45062,c1(C(=O)NC2CC3CN(C(CCCCC)=O)CC2C3)ccc(S(C)(=O)=O)cc1 45063,N1(C(CC2(NC(C)=O)CC2)=O)CCC2(CCCN2C(=O)CC2CCCC2C)C1 45064,c1(NC2CN(C(CCS(=O)(=O)NC)=O)CC2C)cc(C)c([N+](=O)[O-])cn1 45065,c1(OCC)ncc(Cl)cc1C(=O)NC12CCC(CC1n1cc(CCCO)nn1)C2 45066,c1(C(=O)NCC2CC2CNC(C2CC23CCC3)=O)c(Cl)cccc1Br 45067,CCCC(C)CCCC(=O)NC1CCC(NC(C2(CF)CC2)=O)C1 45068,C(=O)(C#CC1CCCOC1)N1C(C2(NC(Cc3ncc(C)s3)=O)CC2)CCCC1 45069,C1(C(=O)NC2CN(c3nccc4c(Br)csc34)C2)CC2(CO1)CC1(C2)OCCO1 45070,N1(C(c2cncc(NC(C)=O)c2)=O)CC2(CCC(NC(c3ccoc3C)=O)C2)C1 45071,N1(C(CNC(=O)OCC)=O)CCCC2(NC(c3ncccc3F)=O)CC12 45072,S(=O)(=O)(c1cccc(N2CCOC(CCOC)C2)n1)NCC=CCCC 45073,C1(N(C(c2c(COC)cco2)=O)C)CCC(NC(C2CC3(CC3)CO2)=O)CC1 45074,N1(C(c2ccc(C#N)[nH]2)=O)CCC2(CCCN2C(=O)C(F)C(F)(F)F)C1 45075,CC1CN(C(=O)CC2OCCC2(C)C)CC1NC(=O)Cc1n[nH]c(=N)s1 45076,c1(CC(N2C(C)CC(NC(C3CCC(C)C3)=O)C2)=O)ccc2sccc2c1 45077,c1(C(C)C)nc(C(=O)N(C2CN(C(=O)C(C)CN3CCCCC3)C2)C)cs1 45078,C1(NC(CC2N(C(CCC(C)=O)=O)CCCC2)=O)CC2(COCCO2)C1 45079,S(=O)(=O)(CCC(F)(F)F)NC1CC(C)N(c2ncc(C#N)cc2Cl)CC1 45080,N1(C(c2ncc(C)cn2)=O)CCN(C(c2nccc(Cl)c2C)=O)CC1CC1CC1 45081,C1(CNC(=O)C2=CSCS2)C2CCCC1N(C(c1cncnc1)=O)C2 45082,N1(C(c2nc(CC)sc2)=O)CC2(CCC2)CC1CNC(=O)C(C)NC=O 45083,N1(C(c2c(C)nc(C3CCOC3)s2)=O)CC2(CCC2)CC1CNC(C1(C)CC1)=O 45084,N1(c2nccc(OC)n2)C2CCCC1CN(C(C1(O)CCOC1)=O)CC2 45085,C(C(=O)NCCCCN(C(=O)CC1C(=O)NN=C1C)C)(C(C)C)OCC(C)C 45086,C(C(CC)CCCC)NC(C1(CN(C(=O)C(C)CCC)CC)CC(=C)C1)=O 45087,c1(N2CCC(CC(C)NC(C3(C)CC(O)CN3C)=O)CC2)ccc([N+](=O)[O-])cn1 45088,N1(C(Cc2cnc(C)[nH]2)=O)CCCC2CN(C(=O)C(C)CS(C)(=O)=O)CCC12 45089,C(C(=O)N1CC(=O)NC(C)C1)(C(C)(C)C)n1cc(-c2ncc(OC)nc2)nn1 45090,C(=O)(CCC(C)(C)NC(C1CCC(=O)C(C)C1)=O)NCCC(CCC)C 45091,c1(CC(=O)N(C2CCN(C(C3CCCN3S(C)(=O)=O)=O)C2)C)ncc(F)cc1F 45092,C(CC(C)C(=O)NCCSCC(=O)NCCc1nnc(C)s1)=CCC 45093,C1(CC=C)(NC(=O)C(Cn2cccn2)NC(=O)Cc2cnn(CC)c2)CCCC1 45094,c1(NCC)ncc(C(N2CC3C(NC(C4CCCCNC4=O)=O)C3C2)=O)cc1Cl 45095,C#CCC(CC(=O)N1CCC1CC(=O)NC)NC(=O)C(C1CCC1)OC 45096,c1(C(N2C3CN(C(c4ccncc4)=O)C(CC3)C2)=O)nc(Br)n2ccccc12 45097,CC1(C)CC(c2cn(CC(C3CCN(C(=O)CS(C)(=O)=O)CC3)F)nn2)CO1 45098,CCCC(CCCNC(c1c(OC)noc1C1CC1)=O)NC(=O)C(CC)C(C)C 45099,CCP1(=O)CCN(C(c2ccc(OC(C)(C)C)nc2)C(=O)NC(C)C)CC1 45100,c1(C(C)CNC(=O)Cn2cnc(-c3cccs3)n2)cccc(Cl)c1 45101,N1(C(CC(=O)NCC)=O)CC2CN(C(=O)CC(C)C(C)C)CC2(C)C1 45102,C1(CNC(CCC=C=C)=O)CC(C)CN(C(=O)CCC)C1 45103,C1(C(N2CC(C=C)C(NC(=O)C3=C(C)CC3)C2)=O)CC12CCCCCC2 45104,C1(C(=O)OC)CCC(C(=O)NC(C)(C)C(C)NC(=O)CSCc2cscn2)O1 45105,c1(OC)ccnc(C(=O)N(CCCCNC(C2CCC(C(F)(F)F)O2)=O)C)c1F 45106,C(=O)(C(C1=CCC2CC2C1)NC(=O)OC(C)(C)C)N(C1(C2CC2)CC1)C 45107,N1(C(C2(CNC(=O)C=CC(F)(F)F)CC(C)(C)C2)=O)CCOC(C)(C)C1 45108,C1(CNC(c2nc(C)oc2)=O)CCCCN(C(=O)CC2(O)CCCC2)CC1 45109,Cc1cc(F)cnc1C(=O)NCC1CN(C(=O)CCn2ccnc2)CC1O 45110,N1(C(COC)=O)CCOC(CNC(=O)CNC(c2ccnc(N(C)C)c2)=O)C1 45111,C(C)(C(C)C(=O)Nc1ccsc1CC)NC(c1cn(CC=C)nc1)=O 45112,CCCCCC(C)(C)C(=O)NC1CN(C(=O)C(C)SC(F)(F)F)CCC1C 45113,C1(C(N2C(CNC(C3N(C)CC4(CC4)C3)=O)CCC2)=O)CCC(C2CC2)CC1 45114,N1(C(C(CC)=CCCC)=O)CC(=O)CC1C(=O)NCc1cc(O)ncn1 45115,c1(C(C)NC(=O)C(=O)NC2NCCCC2C(C)(C)C)ccc(F)c(Cl)c1 45116,CC1(CNC(=NCCCc2ccccn2)NCC2CCCO2)CCC(F)(F)CC1 45117,c1(C(N(CCCN)C)=O)ccn2cccc2c1.c1(OC)ccc(C(=O)NCCOC)s1 45118,C(=O)(C(C)(C)CN1CCCCC1)OC(C1C(C#C)C1)=O 45119,c1(C(=O)NCCC2N(C(C3CCCC(OC)C3)=O)CCC2)nn(C)c2c1CCC2 45120,c1(C(=O)NC2(CC=C)CN(C(=O)CC3CCC(C)O3)C2)cc(C)oc1COC 45121,N1(C(CC(CCC)(C)O)=O)CCC2C1CCCN2C(c1cn(C2COC2)nn1)=O 45122,c1(CC(=O)NCC(C2CCOC2)NC(C2(F)CC=CC2)=O)ccccc1Br 45123,CC(C(=O)N(C(C)CN(C)C(c1cncc(N)c1)=O)C)C(F)(F)C(F)F 45124,c1(C(=O)NCC2(F)COCCN(C(C=NOC)=O)C2)cnc2scc(C)n2c1=O 45125,C(CN=[N+]=[N-])(C(=O)NCCCc1ccccc1)NC(COCC=C)=O 45126,c1(C(=O)NC(C)CNC(=O)C(c2ccc(C#N)cc2)O)cnn2cccc(Cl)c12 45127,C(CC(=O)CCO)c1cn(CCCN(C(=O)C=CC2CCCC2)CC)nn1 45128,c1(NCCCC)ccc(C(=O)NC2(C)CC(NC(=O)CC3CC3)C2)cc1[N+](=O)[O-] 45129,c1(C(N2CCCC(C#C)C2)c2nnnn2CCC2CC2)ccc(Br)c(F)c1OC 45130,N1(C(COC(CC)(C)C)=O)CC2(NC(=O)CCOCC3CC3)CCCC2(F)C1 45131,CC1(C)CCCC1C1CCN(C(=O)C(=C2OCc3ccccc3C2=O)F)C1 45132,CC(C(=O)NC(CNC(c1c(F)cncc1Cl)=O)C1CC1)C(F)(F)C(F)F 45133,N1(C(C)=O)CCC(C(=O)OCc2[nH]nc3c2COC3)C(F)C1 45134,CCCCCCCCCC(C)CC(=O)N1CCC(CNC(=O)C=C(C)C)C1 45135,C(C1CCCc2cccnc21)NC(NC(CC)CC)=NCCNC(=O)COC 45136,C1(NC(c2cc(OC)ncc2Cl)=O)CN(C(C2CC=CCC2)=O)CC(F)(F)C1 45137,c1(C(=O)NC2(C)CCN(C(c3c(CC)c[nH]c3)=O)C2)ccc(N)c(C)c1Cl 45138,CCCCC(O)CNC(=O)COC(C1CCCC1)(C)C 45139,c1(CCS(CC(N2C3(CN(C(N)=O)C3)CC2)=O)=O)cncc2cnccc12 45140,C1(C(N2CC(C(C)C)OCC2)=O)C2CCN(C(C34CC3CNC4=O)=O)CC12 45141,N(C(=NCc1cnc(C)cn1)NCC(=O)NCc1ccccc1)C(C)C1CC1 45142,CC1CN(C(c2ccccc2CC#N)=O)CCN1C(c1ccc(C(N)=O)cn1)=O 45143,c1(C(=O)NCCCOC)cc(-c2cc(OC(C)=O)c(C)c(C)c2)c2cc[nH]c2c1 45144,c1(C(=O)NC2CCN(C(C(C)(C)N(S(C)(=O)=O)C)=O)CC2)ccc(CN)cc1O 45145,c1(CC(=O)NC(C2CN(C(=O)Cc3ccon3)C2)C)ccc(Br)cn1 45146,Cn1cc(C(N)=O)cc1C(=O)NCC1COC(CNC(=O)CC2CC(F)(F)C2)C1 45147,C(C(F)C(=O)N1CC(F)C1)C1CN(C(C2(CC#C)CC2)=O)C1 45148,C1(NC(=O)CC23CCCN2CCC3)CN(C(=O)Cn2cncn2)CC1C1CC1 45149,N1(C(CN(C(c2cccc(C#N)c2)=O)CC)=O)CC2(CC(F)C2)C1 45150,C(=O)(CCCN(C)C(c1ccn(C)n1)C)NC.c12cc(no1)C(=O)NC2 45151,N1(S(CC=C)(=O)=O)CCC(F)(F)C(C(=O)Nc2ccc3nccn3n2)C1 45152,c1(OC(C)C)cc(C(N2CC(CNC(=O)Cc3ccsn3)C(C)C2)=O)ccc1F 45153,C1(O)(CNC(=O)CCCC2CCCC2)CCCN(C(C2COC(=O)O2)=O)C1 45154,C#CCCC(O)C(=O)NC(C1CCCN1C(=O)Cc1c[nH]c(=N)nc1O)C 45155,N1(C(C2(COCC)CCC2)=O)CCC(C(N2CCOCC2)=O)CC1.C1(=O)CN1 45156,C(=O)(C(CC1CC1)NC(C1(CCNC(=O)CCc2nc(O)n[nH]2)CCC1)=O)NC 45157,CC1(C)CC(CNC(c2cccnc2)=O)N(C(=O)Cc2cncnc2)C1 45158,c1(C(=O)NCCCN(C(C2C(C#N)CC2)=O)CCO)ccc(CF)cc1.CCO 45159,c12ccc(nc1)N(CC)CCCCNC(=O)CC2.c1(C(=O)NC)nc(=O)n(C)[nH]1 45160,C(=O)(C(CN(C)C)C(C)C)NC(CC(=O)NCC(CC(C)C)OC)C 45161,Cc1c(NC(=O)CN2CCNC(=O)C2)cccc1-c1cncc(O)c1 45162,Cc1cc(N2CCC3(NC(C4CC5(CC5)C4)=O)CCCC23)n2nc(C)cc2n1 45163,C=CC1CN(C(C23CCOC(C)(C2)C3)=O)CC1NC(c1csc(F)c1)=O 45164,CCC(CC(=O)NC1COCC1C(=O)NC(C)Cc1ncn(C)n1)C(F)F 45165,c1(C(=O)NC(CC=C)CNC(C2CC(C)=NO2)=O)ccc(Br)c(Cl)c1 45166,C1(CNC(C2=CC(C)(C)C2)=O)CC2COCC2N1C(c1ccnn1CC1CC1)=O 45167,N1(C(C(=O)NCC2CC2)C2CC2(Br)Br)Cc2nccc(Cl)c2C1 45168,c1(C(C(=O)NCC(C(C)C)NC(CCCc2onc(C)n2)=O)C)c(C)n[nH]c1C 45169,c1(OCC(N2CCC(CN(C(C(n3ncc(C)c3)C)=O)C)C2)=O)ccc(Cl)cn1 45170,c1(CC)ccc(C(=O)NCC(C)(C(C)C)NC(=O)CCc2cnc(O)[nH]2)cn1 45171,C1(C(N(C2CCN(C(c3csc(=N)[nH]3)=O)C2)CC#C)=O)CC(C)(C)CCO1 45172,C1(N(C)C(c2cocn2)=O)CCN(C(C2CCCC(O)C2)=O)CC1 45173,Cc1cc(-c2nn(-c3ccc(Cl)cc3)cc2C(=O)NCCC(C)C)ccc1F 45174,c1(CC(=O)NCC2OCCN(C(CCCC#C)=O)C2)ccc(C)c(Cl)c1 45175,CC#CCC(C(=O)N1CCC1(C)CC)NC(c1cn[nH]c1)=O 45176,c1(C(=O)NC2CC(CNC(C(C)CC(C)(C)C)=O)C2)ccc2c(c1)CCCC2 45177,C1(C)(CNC(C(C(C)C)NC(N)=O)=O)COCCN(C(=O)C2=CCCCO2)C1 45178,C1(C(N(CCC(=O)NC2(CF)CCC2)CC=C)=O)CC12CCCCC2 45179,c1(CC)cc(Br)ccc1C(=O)Nc1nc(N2CCN(C(C)=O)C(C)C2)ncc1Br 45180,CC(O)C(C)C(=O)NCC(C)NC(C1CCCN1Cc1ccccc1)=O 45181,c1(C(=O)NCC(CC)NC(=O)C(N2CCCCCC2)C)nn2c(c1C)OCCC2 45182,Cc1cc(CC(N2CCC(c3nc(C(F)(F)F)cs3)CC2)=O)n(C)n1.C1CN1C 45183,C(C1CN(C(=O)CC)CC1N)=CC.N1(C=O)CCSCCC1C 45184,c1(COC)ncc(C(N2CC(=C(F)CNC(C3(C(C)C)CC3)=O)C2)=O)c(O)n1 45185,C=CC1CCCCN1C(=O)C(c1cnn(C)c1)NC(=O)CNC(N)=O 45186,C(=O)(C(F)C(C)(C)O)N1CCC1.c1(N(N2C(NC=O)CCC2)C)c[nH]c(C#N)c1 45187,c1(NC(c2n(CCCSC)nnn2)c2csc(Br)c2)cc(O)c(C)cc1C 45188,N1(CC(=O)NC(CNC(c2cc(C(=O)OC)c(C)[nH]2)=O)C)CCS(=O)(=O)CC1 45189,c12ccc(cc1)C(=O)NC2.C(C(C1CCC1)NC(=O)COCCCF)SC 45190,c1(CNC(C2CSCCN2c2ccncc2)=O)cc(C(F)(F)F)cc(C2CC2)c1 45191,N1(C(c2c(C)cc(C)s2)=O)CCCOC(CNC(c2cc(C)ncc2Cl)=O)C1 45192,c1(C(N2C(CCC(=O)NCC3CC34CCC4)CCC2)=O)cc(O)nc(O)c1 45193,C(=O)(C(C)CC(C)C(C)=O)N(CCNC(=O)CC1CC=CCN1C)CC 45194,c1(N(CC(O)CC(F)(F)F)CCN(CC)CC)cc(F)cc(F)c1 45195,c1(C(=O)NC(C2CN(C3CCOCC3)C2)C)nn[nH]c1Cl.C12CC(C1)NC2=O 45196,C#Cc1ccc(F)cc1C(N1CCOC(CNC(C2CC2CF)=O)C1)=O 45197,c1(OC)cccc(C2CC(=O)N2)c1.N1(C(=O)OC(C)(C)C)CC2CC2C1 45198,CC1CCC(C)C(C)C1NC(C1CCC(=O)N1CC1CCCCC1)=O 45199,C1(CC(=O)NC(C=CC(CC)C)=O)CCCCN1N1CCOCC1.C1C=CC1 45200,C(CC(C(=O)NCC1CCN(C(C)C)C1)NC(c1sccc1C)=O)OC 45201,c1(C(=O)NC(C)CCC(=O)N2CC(Oc3ccccc3)C2)ccc2sncc2c1 45202,C12(C(N3CCC(CCCC)C3)=O)CCCC1CCN2C(=O)Cc1cncn1C 45203,c1(CNC(c2ccc(OCC(=O)N(C)C)cc2)CC(C)C)ccc2c(c1)OCO2 45204,c1(CN2CC(C(=O)Nc3ccnc(F)c3)SCC2)c(F)c(F)cc(F)c1F 45205,Cc1cc(C#N)ccc1S(=O)(=O)N1CC(C2CCCOC2)C1 45206,CC(C)(C(F)(F)F)OCC(=O)NCCOCCCNC(C1(F)CCCC1)=O 45207,c1(C(N2CCC(C(=O)O)(C)CC2)=O)ccc(C)c(C)c1O.c1(CC)ccc(CN)o1 45208,N1(C(C2CC23CCOC3)C(=O)NCCCOC)CC(CO)OC2(CCC2)C1 45209,C1(CN(C(=O)CCc2cnco2)C)C2CN(C(=O)Cc3ccsn3)CC12 45210,c1(C(C(=O)NCCC(C)NC(C2(C(F)F)CC2)=O)=O)cc(F)cc(Cl)c1 45211,C1(C(N)=O)CCCC1CNC(=O)CNC(c1nc(CC(=O)N)cs1)=O.C1(S)CC1 45212,Cc1noc(C(F)(F)F)c1C(=O)NCC(F)CNC(C1(C2CC2)CC1)=O 45213,c1(CCC(N2C(CNC(c3ccc(COC)[nH]3)=O)CC2)=O)ccc(SC)cc1 45214,c1(N2CC(COC)C(SC)C2)cc(Br)ccc1S(=O)(=O)NCc1ccc(SC)o1 45215,C(=O)(C1COc2ccccc21)N1CCC(C2N(C(c3nccc(C)n3)=O)CCC2)C1 45216,Cc1cc(C(N2CCC(C(F)C(=O)N3CC(NC(N)=O)C3)C2)=O)c(C)cn1 45217,N1(C(c2c(C)nn[nH]2)=O)CCN(C2CCCN(C(=O)C(C(C)C)N(C)C)C2)CC1 45218,C1(C(N2CC(CC(C#C)C)C2)=O)CC(=O)CN1C(=O)CC1(N(C)C)CCC1 45219,N1(C(c2c(C3C(C)C3)noc2)=O)CCC(CNC(C2CC2(C)CN(C)C)=O)CC1 45220,n1(C(CC)C)ccc(=NC(=O)C2CN(C(c3ccccc3O)=O)CCC2(C)C)[nH]1 45221,N1(C(C2C(C(C)C)C2)=O)CCN(C(C2CC(=O)C2C(C)(C)C)=O)CC1CCO 45222,C1(CNC(C2C=CCN2C(=O)C(O)C2CCCC2)=O)CC2(CCC2)C1 45223,c1(C(c2n(CC=C)nnn2)NCc2ccns2)ccc(C)cn1 45224,N1(C(Cc2ccc(C)cc2)=O)CCCC(N(C)C(C2C(C)OC(C)C2C)=O)CC1 45225,C1(C(N(CC(C)C(=O)NC2C=CC(C)(C)CC2)C)=O)CCC(C)(O)CC1 45226,c1(C2C(C(=O)OC)C2)ccc(OCCCCOC(=O)C(c2ccccc2)F)cc1 45227,CC(CS(C)(=O)=O)C(=O)NCCC(C)CCNC(=O)CCSCC(N)=O 45228,C(C(C)(C(=O)NCC=CCC(=O)N(CC(F)Cl)C)OC)OC 45229,C(=O)(C1=CCS(=O)(=O)C1)N(C(c1cn(Cc2cc(Cl)ccc2Br)nn1)C)C 45230,C(=O)(CS(=O)(=O)c1cccc2nsnc12)N(CC(C)NC(=O)CCC1CC1)C 45231,c1(C(N(C2CCC(NC(=O)CCn3cccc3)C2)C)=O)cnc(Cl)o1 45232,c1(C(=O)OCC)cc(Cl)c(OC)cc1NCc1cc(C)ccc1Cl 45233,C#CC(CNC(=O)C(CO)NC(=O)C=Cc1ccco1)CC1CC1 45234,c1(SC2CCN(C(=O)Nc3cn(C)nc3)C2)ccc(F)c(NC(=O)OC(C)(C)C)c1 45235,c1(C(=O)NC2(CNC(c3cn(-c4ccn(C)n4)nn3)=O)CC2)c(Cl)cncc1Br 45236,n1(CC)nc(C(N2CCN(C(C3CCCC(C(F)(F)F)O3)=O)CC2)=O)cc1O 45237,N1(C(C)=O)CCCC1C(=O)NC(C)(C)CCNC(c1coc(Br)c1)=O 45238,C1(CNC(C(c2cnn(C)c2)C)=O)CCC(NC(=O)Cn2ncnn2)CC1 45239,C(=O)(C1=CCCC1C)NC(CCOCC)C(=O)NCc1cn(CCOC)nn1 45240,C1(C(=O)NC2CCC(NC(Cc3n(C)cnc3)=O)CC2)CCS(=O)(=O)CC1 45241,Cc1ncccc1C(N1CC=CC1CNC(C1C(F)(F)C12CC2)=O)=O 45242,c1(OC)ccnc(C(=O)NC2(CF)CCN(C(=O)CN3CCC(F)CC3)C2)c1 45243,c1(N(C(=O)CC(C)(C)C)C(=O)OCc2ccc(OC)cc2)cc(C)cc(C)n1 45244,c1(OC)cccc2c1OCCCC2NC(=O)C(=O)NC1CCN(C(C)C)C1=O 45245,N1(C(c2c(CC)cco2)=O)CCC(C2CC2)C1C(N1CC(CO)C2(CCC2)C1)=O 45246,N1(C(CCCN(C(=O)C(C)OC)C2COC2)=O)CCCOC(CCC2C(C)C2)C1 45247,CC1(C(=O)NC2CC(CNC(C3(C(F)F)CCCC3)=O)C2)CCCNC1=O 45248,c1(C(c2n(CCC)nnn2)NCC(=O)NC2CCCCCC2)c(C)nn(C)c1C 45249,C1(NC(=O)Cc2ccon2)CC2CCC(C1F)N2C(c1nc(Cl)c(Cl)s1)=O 45250,C1(C(N2CCN(C(=O)Cc3cccc(O)c3)CC2)=O)(OC)CC(C)CC(C)C1 45251,CC1CCC(NC(=O)CC2CN(C(=O)Cc3ccccc3)CCC2C)C(C)C1 45252,N#CC1CC(C(=O)NCC(O)CNC(C2(CC3CCC3)CC2)=O)C1 45253,C12(C(=O)NC(CC)CO)CC(CN(C(=O)CCn3ccnc3C)C1)C2 45254,CCCC(C)CC(=O)N1CCOC(CN(C(=O)CN(C)C2CC2)C)C1 45255,N(C(=NCCC)NC(c1cccc(Cc2ccccc2)c1)C)C(C#C)C 45256,N1(C(c2cc(C)[nH]n2)=O)CC(C(N2CCOCC(N(C)C)C2)=O)C(F)(F)C1 45257,N(C1CN(c2cc(Cl)ncn2)CCc2ccccc21)C(=O)CCc1cnc[nH]1 45258,C1(C(N2C(C)CC(CNC(c3cc(O)nn3C)=O)C2)=O)CCn2c(O)nnc2C1 45259,C(=O)(CC(O)C(C)C)NCC(c1ccc(C)cc1)NC(c1c(CO)noc1C)=O 45260,C12(CNC(c3c(CC)nc(=N)[nH]c3)=O)CCCC(CN1C(c1cnsc1)=O)C2 45261,c1(C(=O)NC2CCN(Cc3c(C#C)cccc3)CC2O)ccc(O)c(O)c1Cl 45262,c1(C(=O)NC23C(CCN(C(C4(SCC)CC4)=O)C2)C3)ccc2nccn2c1 45263,c1(CC(C)C)nc(C(=O)N(CC(=O)CC2CCC2)Cc2ccccc2)cs1 45264,c1(C(N(CCCNC(C2C(=C)C2)=O)CCO)=O)ccc(OC)c(S(N)(=O)=O)c1 45265,N1(C(C(C(C)C)NS(C)(=O)=O)=O)CCC(C)CC1CNC(=O)CN(C)C1CC1 45266,c1(OC)ccccc1C(N1CC(N(C(=O)CCC(C)N(C)C)C)C(O)C1)=O 45267,Cc1[nH]c2c(C(N3CCC(CNC(=O)CC4CC4(Cl)Cl)C3)=O)cccc2c1C 45268,N1(C(C(C(C)(C)O)F)=O)CCC(C2(NC(c3ccnc(C4CC4)c3)=O)CC2)C1 45269,c1(CN2C(C(=O)NC(CC=C)CO)CC(O)C2)cc(Br)ccc1F 45270,N1(c2c(OC)cnc(Cl)n2)CCCC(C2CC2NC(c2nccc(Cl)c2F)=O)C1 45271,c1(Cn2cc(CONC(c3cccc(C(C)=O)c3F)=O)nn2)cc(C)cc(C)c1Br 45272,C1(O)(CCNC(c2c(C)nc(CCC)s2)=O)CCN(C(=O)C(CC)OCC)CC1 45273,N1(C(=O)NCC(C(C)C)NC(=O)C(=O)Nc2ncc[nH]2)CSCC1NC(CC)=O 45274,Cc1cc(N2CC(O)(CSc3ccccc3)C2)nc(C)c1 45275,c1(C(=O)NC2(C3CC3)CCN(C(C(CC)(C)C#N)=O)C2)cnc2ccncc2c1 45276,C1(=O)C2=CCCN(C2)N1.c1(C(NOC(CC)CC)=O)[nH]cc(C)c1C 45277,c1(C(=O)NC(C(C)NC(C2CC(=C)C2)=O)(C)C)cc(Cl)cc(F)c1N 45278,c1(C(=O)NCCN(CCC)C(C2CCCSC2C)=O)occ2c1CCC2 45279,C1(NC(=O)Cc2cccc(-c3cn[nH]c3)n2)CC2CCC(C1)C2N 45280,c1(C(=O)NC2(COC)CN(C(c3n(CC)c(O)nc3)=O)C2)cncc([N+](=O)[O-])c1 45281,C#CC1(C(N2CCC(C3CCCN3C(=O)C(CC=C)CC)CC2)=O)CCCCC1 45282,N1(CC)CC(C)CC1(C)C.C1(=O)CCCn2nnnc2C(C)(CCSC)N1 45283,N1(C(CCCOCC)=O)CC(C)(CNC(=O)CC(C)c2ccccc2)CC1(C)C 45284,CC(C)CCC(C)N(C(=O)C(C)N(C(C1CCC2CC12)=O)C1CC1)C 45285,c1(C(=O)NC2CC3CN(C(C(CC)=CC)=O)C(C2)C3)ccc2cnnc(O)c2c1 45286,C(C1CCOCC1)=CC(=O)N(CC(C)N(C)C)C.C12(CCCO1)C(=O)NC2 45287,c1(C(=O)NC(CC)CNC(C2CN(C)C2)=O)cccc(F)c1C#N 45288,c1(C(=O)NC(C)(CNC(=O)C(O)CN2CCCC2)CO)csc2nnsc12 45289,N1(C(CCCC=C)=O)CC(C)(C)CC1C(=O)N(CCc1nccn1C)CC 45290,N1(C(c2nnn(C(C)(C)C)n2)=O)CC(NC(c2ncccc2O)=O)CC(F)C1 45291,c1(C(N(C(C)CNC(c2ccnn2C(F)F)=O)C)=O)oc2ccccc2c1Cl 45292,C1(F)(NC(C#CC(OCC)OCC)=O)CCCN(C(C2CCC=CCCC2)=O)C1 45293,C(CC(C(=O)NCCc1nncn1CC)NC(c1cnco1)=O)=CC 45294,N1(C(Cc2nc(C)oc2)=O)CCCC1(C)C(=O)NCC1(C)CCCC1O 45295,c1(OC)ccc(C(=O)NC2CCC2NC(C2CC2c2ccc(F)cc2)=O)c(F)n1 45296,Cc1ccc(F)c(OC(=O)C(c2ccc(F)cc2)OC(C)C)c1 45297,C1(NC(C(C)OCC#C)=O)CN(C(=O)CCc2cccs2)CC2(CCC2)C1 45298,c1(C(N(C)CCOCCNC(C2(C(C)(F)F)CC2)=O)=O)ccnn1C1CC1(F)F 45299,CC1CC(NC(=O)CCCNC(N)=O)CCN1C(=O)CNC=O 45300,C(N=c1nc(-c2ccccc2)[nH]s1)c1c(CNC(C2CC(=O)CN2)=O)cccc1 45301,c1(OC)c(C(=O)NC2CCN(C(=O)C=CSC)CC2SC)cccc1C(F)F 45302,N1(C(c2c(CC)nccn2)=O)CC(F)(F)CC1C(=O)NC(C)CC(C)(C)O 45303,CC1(C)CCC=C1C(=O)NC1CN(C(=O)CCC2CCCC(=O)N2)CC12CC2 45304,C(=O)(CC(CN(C)C)C(F)F)NC1CCN(C(c2cnc(SC)s2)=O)C12CC2 45305,N1(C(CCCC(C)C)=O)CC2(C1)SCCC2NC(c1ccc(Cl)cc1)=O 45306,C(=O)(C1=CC2(CCOC2)C1)OC(C(=O)N(CCC1CCCCC1)CC)C1CC1 45307,C(=O)(C(C)CC=CCC)N1CCC(CCNC(c2ccc(CCC)s2)=O)C1 45308,C1(NC(=O)CCc2cncs2)CC12CCN(C(C1CCCOC1)=O)C2 45309,Cc1nn(CC(=O)NCC(C)NC(c2ncc(Br)cc2F)=O)c(=O)n1C 45310,N1(C(CC(C)C2CC2)=O)C2CCC1CC(CNC(c1ccc(=N)[nH]c1Cl)=O)C2 45311,N1(C(C2N(C(C)=O)CC(O)C2)=O)CC(NC(c2ccnnc2)=O)C(C)(C)C1 45312,c1(CN(C(c2c(C(=O)OC)[nH]cc2)=O)Cc2cnc(C)s2)c(F)cccc1F 45313,N1(C(CC2CC(C)OC2C)=O)CCCC(C2CC2NC(=O)CC2(O)CCOC2)C1 45314,c1(CC(=O)NC(CNC(C2CN(C)C(=O)N2)=O)C(C)(C)C)cnn2c1OCCC2 45315,C1(C(N(C(C=C)C)C)=O)CCC(CNC(=O)Cc2ccn(CC)n2)C1 45316,C(=O)(C(C)(C)CCC#N)NCc1ccc(C(=O)NCC2(C#C)CCCC2)cc1 45317,C#CC(CC1CCC1)NC(=O)CC1(N(C(=O)CC=CCC)C)CC1 45318,C1(CS(=O)(=O)NCC2CC(C)(C)OC2)CCCC2(CCOC2)O1 45319,Cc1nc(CC(=O)NC2(CN(C(=O)C(C)C3CCOC3)C)CC2)n[nH]1 45320,C(=O)(C(C)(C)C(=O)N(C)C)NCC1(CNC(c2c(COC)noc2)=O)CCC1 45321,C1(C)(CCC(=O)N(CC(C)CNC(=O)CCOC2CCC2)C)CCC(=O)N1 45322,C1(C(=O)NC(C2(O)CN(C(C(C)(C)OC(C)=O)=O)C2)C)CC1C1CCCC1 45323,c1(C(=O)NC(CC)CNC(C2(Cl)CC2(F)F)=O)cccc(-c2cscn2)c1 45324,C1(CNC(CC2CCCN(C)C2)=O)CN(C(=O)CCc2cn(C)nn2)C(C)(C)C1 45325,CCC(C)C(O)C(=O)NC1CCC1C(N1CCCCN(C)CC1)=O 45326,C(=O)(C(CC(F)(F)F)c1ccc(F)cc1)NCc1nc(Cl)c(C)n1C 45327,c1(CC)[nH]nc(C(N2CC(OCCNC(c3cccnc3C(F)F)=O)C2)=O)c1Cl 45328,N1(C(c2cc(O)ccc2Br)=O)CC2CCN(C(=O)Cc3ccnc(Br)c3)C2C1 45329,C(=O)(C(O)CC(F)F)N(C)CC1CCN(C(c2c(OC)n[nH]c2)=O)C1 45330,CC1(C)CN(C(c2csc(S)n2)=O)CCC1NC(C1CCNC(=O)C1)=O 45331,CC1CC(NC(=O)Cc2ccn(-c3ccccc3)n2)CN1C(=O)C(=O)N(C)C 45332,c1(C(=O)OC)cc(C(=O)NCC(CNC(c2cc(Cl)c[nH]2)=O)CO)no1 45333,C(=O)(C(C)(O)CCc1ccccc1)NC1CC(NC(C(CC=CC)C)=O)C1 45334,C1(C(=O)NCCC(CNC(CN2CC(C)C2)=O)O)CCCN1C=O 45335,C1(NC(C(N(C)C)C2CC2)=O)CN(C(c2sccc2F)=O)CC(C)(C)C1 45336,CC1CCC(NC(=O)C(C#N)=CC2CC2)CN1C(=O)C=Cc1ccc(F)cc1 45337,c1(OC)ccc(F)c(C(=O)N(CC(O)CN(C(=O)CC2CCC(O)C2)C)C)c1F 45338,N12CCCCC(C1)CCC2=O.N1(C(Cc2n(C)ccn2)=O)CCOC(C(N)=O)C1 45339,N1(C(c2c(C)snc2)=O)CCCC2CN(C(c3ccc4cnccc4n3)=O)CC12 45340,C1(NC(CC2(C=C)CCOCC2)=O)C2CCN(C(=O)CC3(C#N)CC3)CCC12 45341,CC(C)(C)C(C(=O)NCCC1(NC(=O)Cc2ccccc2)CC1)C1CCCC1 45342,C1(C(=O)NCc2c(C)occ2)CCCN1NC(=O)CCCC1CCC1 45343,C1(N(C(c2c(COC)cco2)=O)C)CCCN(C(C2CCCOC2)=O)C1 45344,c1(C(C)(C)C)cc(C(=O)NC2CCCC(NC(C3(C)CC=CCC3)=O)C2)ccn1 45345,C1(CNC(c2ccnn2C2CC2)=O)CCN(C(c2ccsc2)=O)CC1(F)F 45346,C1(C(N(C)CC2N(C(C(C(=O)OCC)F)=O)CCCC2)=O)CC12CCCCC2 45347,N1(C(CN(C2CC2)CC)=O)CCCC1CC(=O)NCC1(C)CCCS1 45348,C1(NC(C(F)OC)=O)CCN(C(C2CNC(=O)N2C)=O)C12CCC2 45349,CCCCC(CNC(=O)CCCc1sccc1C)NC(C1(C)CCOC1)=O 45350,c1(C(N2CCC2CNC(=O)COc2ccsc2Cl)C)cccc2c1CCO2 45351,c1(C(=O)NC2CN(C(c3c(C)sc(Cl)n3)=O)CC2C)ccc2cnoc2c1 45352,c1(OC)cc(-c2cc(C(=O)NC(c3cc(F)cc(F)c3)CC(=O)O)no2)ccc1F 45353,C(=O)(C(C)(C)c1ccn(C)n1)NC(C)CN(C)C(c1ncn(C)n1)=O 45354,Cc1nc2cc(CC(N3CCCN(C(c4ccncn4)=O)C(C)C3)=O)ccc2o1 45355,C1(CC#C)CCCCN1C(=O)NC(c1cccnc1)C1CCNC1 45356,N(C1CCSc2ccccc21)C(C12C(NC(=O)OC(C)(C)C)C3CCC1C2C3)=O 45357,CC1CN(C(=O)CC2C3CCC(C3)N2C(=O)C(C)OC(C)(C)C)C(C)C(C)(C)O1 45358,c1(C(N2CC=C(CNC(C(C)OC)=O)CC2)=O)cnc2c(c1)COC2 45359,c1(C(=O)NC(CNC(CCCC)=O)C)ccc(OCC)cc1F 45360,N1(C(C(CC#CC)NC(c2nccnc2OC)=O)=O)CCN(C)C(=O)C1C 45361,C1(COC)(CNC(c2ccc(O)nc2)=O)CCN(C(C2CCC3(CC3)C2)=O)C1 45362,c1(SCC)ccc(C(N2CCOC(CCNC(C3(F)CCC3)=O)C2)=O)cn1 45363,Cn1cc(C(=O)NCCC2CCN(C(=O)CCCC#N)C2)c(=O)c(Br)c1 45364,NS(=O)(=O)c1ccc(F)c(C(N2CC3(C(=O)NCCC(F)(F)F)CC2CO3)=O)c1 45365,CCC(C)CN=c1[nH]c2c(c(=NCc3nc4c(s3)CCCC4)[nH]1)CCC2 45366,N1(C(C2CC3(CC3)CO2)=O)CCCN(C(=O)C(F)(F)CO)CCC1 45367,C(=O)(CC(CN(C)C)CC)N(C(C)CNC(c1ccc(NC(C)C)cc1)=O)CC 45368,C(C(C)(CCO)NC(=O)C(C)C(C)NC(c1nnsc1N)=O)OC 45369,c1(CC(=O)N(CCC(C(C)C)NC(C(CC)N(C)C)=O)C)ccc(F)c(F)c1 45370,N1(C(CC2CC(C(C)(C)C)C2)=O)CC2CCC2(CCNC(=O)C(Cl)=CCl)C1 45371,N1(C(C(C)Sc2ccccn2)=O)CCC(=CCNC(=O)CCC2CC2(F)F)CC1 45372,C1(C(N(C)N(C2CC2)CC)=O)CN(C(C2(CC#N)COC2)=O)C1.C1CC1 45373,N1(C(CC(C)(C)C)=O)Cc2cccc(CNC(=O)CC3CCCCC(=O)N3)c2C1 45374,c1(CCC(N2CC(N(C(c3c(OC)ccs3)=O)C)C2)=O)cccc2ccccc12 45375,S(=O)(=O)(c1cccc(C(=O)NC2CCC2CNC(=O)C(F)=C2CCC2)c1)NCC 45376,N1(C(c2ncns2)=O)CCOC2(CCN(C(C3CCn4nncc4C3)=O)C2)C1 45377,Cc1ccc2cc(C(=O)NC(C3CN(C(=O)C(C#N)C(C)C)C3)C)[nH]c2c1 45378,c12ncccc1NC2=O.C(=O)(CCCNC(NC1=NCCS1)=O)NC 45379,C1(SC)CCC(SC)CC1.c12cscc1C(=O)N1CCC(C1)n1cc-2nn1 45380,N1(C(CCNC(=O)NC)=O)CCC12CN(C(c1cnc3n1CCC3)=O)C2 45381,N1(C(C2(F)CCN(C(c3nc(CC)sc3)=O)C2)=O)CCC2C(O)C(C)(C)C12 45382,C(C)(N=c1ccnc(NC2CCCOC2)[nH]1)c1nc(CC)[nH]n1 45383,Cn1ncc(C(=O)NCC(O)CC(=O)NC2CC2C(C)(C)C)cc1=O 45384,N1(C(CCN(C(CC(C=C)C)=O)CC2CC2)=O)CC2(C1)OC(=O)NC2C 45385,C1(C)(CC)CCCN(C(C2C3CC2N(C(C2CC(=C4CCC4)C2)=O)C3)=O)C1 45386,N1(CC2CCC(=C)CC2)CC2OCCN(c3ccnc(-c4ccccc4)n3)C2C1 45387,CC1CCN(CCCC(N2CC(NC(=O)CSc3ccccc3)C3CC23)=O)CC1 45388,C1(C(N2CCCC(CCNC(CCC=C)=O)CC2)=O)C2CC3CC(C2)CC1C3 45389,C(=O)(C1=C(Cl)CCC1)N1CC(CN(C(C(CC)(C)C)=O)C)OCC1 45390,c1(OC)cc(C)sc1C(=O)NCC(C)(C)CNC(C1CCC(C(=O)OC)CC1)=O 45391,c1(CC)cc(C(c2nnnn2CC2CC2)NCc2occc2CO)n(C)n1 45392,C1(C)(CC)C=C(C(=O)NCCCC(C)NC(=O)C=CCCC=C(C)C)C1 45393,N1(CC(=O)NC(C2(O)CCN(C(=O)CS(C)(=O)=O)CC2)C)C(=O)C(=O)N(C)C1=O 45394,Cn1nc2ccc(Br)cc2c1C1CCCN1C(c1cnc(C2CCCCC2)s1)=O 45395,c1(OC(C(=O)N(CC(C)NC(Cc2c(C)con2)=O)C)C)ccc(F)c(F)c1 45396,CS(=O)(=O)c1ccsc1C(=O)NC1CCC(CNC(C2(n3cncn3)CC2)=O)C1 45397,N1(C(C#CC(C)C)=O)CC2(C1)CN(C(c1cccn3nnnc13)=O)CC2CO 45398,C(C(CC=C)C(=O)NC1CC(N2CCCC2)C1)NC(Cn1ncc(C#C)c1)=O 45399,Cc1ccc(C2CC2C(=O)NCC2CCCN(C(c3cnc(C)n3C)=O)C2)cc1 45400,CC1(C)CCOC1CC(=O)NC1CCN(C(=O)C=C2CCCCC2)CC1 45401,C1(CC=C)(NC(=O)C(Cc2cc[nH]n2)NC(C2C3(CC3)C23CC3)=O)CCCCC1 45402,c1(C(=O)NCC(C2CC2)NC(=O)C(O)CC2CCCCC2)cc(Cl)ccn1 45403,N1(C(CCN(CCCC)CCO)=O)CCC2C(O)CC12 45404,N1(CCc2ccc(OC)cc2)C(=O)C(CCCO)N(CCc2cccs2)C1=O 45405,c1(C(=O)NCC(C)(C)NC(=O)CCOC2CCCOC2)nncn1C1CC1 45406,C1(C(=O)OCC)CCN(C(=O)CC(C(F)F)NC(=O)CCCC(C)C)O1 45407,N1(C(C(CC)NC(C)=O)=O)CCC(F)(F)C(NCc2cc(Cl)ccc2Cl)C1 45408,C1(CNC(c2cc(C)sc2)=O)COC(C)(C)CN1C(=O)CCc1cncnc1 45409,C(=O)(N=c1ccn(Cc2ccccn2)[nH]1)c1ccc(COC)o1 45410,CCC(CC)CCCC(=O)N1CCCC(O)(CNC(=O)C(C)(C)N(C)C)CC1 45411,C(=O)(CS(=O)(=O)CCO)N(CCCNC(c1cn(CC(N)=O)nn1)=O)C(C)C 45412,C1(C(=O)NCC(CNC(=O)CNC(c2ccoc2CCCCl)=O)F)C2CCCC12 45413,N1(C(C=CC)=O)CCC(C2CC2)(CNC(=O)CC(C)P(C)(C)=O)C1 45414,C(CCCCC(=O)N1CCC(C(F)C(=O)Nc2ccccc2C)C1)OC 45415,c1(C(N2CC(OC)CC(NC(COCCC)=O)C2)=O)csc2c1CCC(C)C2 45416,C1(NC(c2ccc(CCC)s2)=O)CCCN(C(C2(NC(C)=O)CCC2)=O)C1 45417,Cc1cc(C2CC2)ccc1C(=O)NC(C)C(CO)NC(c1ccnn1C)=O 45418,c1(CC(N2CC(N3CCN(C(C4C(C)OCC4)=O)CC3)C2)=O)ccc(F)c(F)c1 45419,c1(N(C)Cc2cn(CC)nc2)nc(N2C3CCC2COC3)nc2ncn(C)c12 45420,C1(C(=O)NCC(CNC(C(C)C(F)F)=O)CO)CCC(O)CN1C 45421,c1(C(N2C(C(N(CCC(C)(C)O)C)=O)CCC(O)C2)=O)ccc2[nH]ccc2c1 45422,C(=O)(C1CCCc2nncn21)N1C(CCNC(C(C)OCCC(C)C)=O)CCC1 45423,CCCCS(=O)(=O)CC(=O)NCC(C)CNC(=O)COC(c1nccn1C)C 45424,c1(CC)nc2c(C(N3CCN(C(c4ccc(O)cc4)=O)C4CC34)=O)ccnc2[nH]1 45425,c1(C(=O)NC2CC(CNC(c3coc(O)n3)=O)C2)csc2ccc(F)cc12 45426,C1(NC(c2coc(-c3ccccc3)c2)=O)C2CC1N(C(=O)COC1CCOC1)C2 45427,C1(CC(=O)NCCN(C(Cc2n(C(C)C)cnn2)=O)C)CCCCN1C 45428,N1(C(CC2(NC(C)=O)CC2)=O)CC2CCC(C1)C(NC(=O)CC1CC=CCC1)C2 45429,N1(C(=O)OC(C)(C)C)CCC2(CC1)CC2(C)CNC(=O)Nc1cncc(Br)c1 45430,C1(F)(C(=O)NCC(CC=C)NC(=O)C(C)COC)CC2(CCC2)C1 45431,c1(COC(C)C)ccc(C(=O)NC2C3CCN(C(=O)C(C)(C)C#N)C23)cc1 45432,c1(C(N2CC(CCNC(C3(C#C)CC(=O)C3)=O)(OC)C2)=O)cccc(N=[N+]=[N-])c1 45433,c1(CC(=O)NCCN(CCC)Cc2ccccn2)c[nH]c2ccc(OCC)cc12 45434,C1(NC(c2cc(COC)on2)=O)CC(CNC(C2CCS(=O)CC2)=O)CC1O 45435,C(C)(CCC(=O)NC1CC(=O)N(C)C1)NC(C1CCN(CCOC)C1)=O 45436,N1(C(c2n(CC)nc(C)c2)=O)C2CCC1CN(c1ncc3ncn(C)c3n1)CC2 45437,c1(CNC(C(C=C)O)=O)ccc(CNC(=O)CN(C(=O)C(C)C)C)cc1 45438,N1(C(C(CC)(C)C)=O)CCC2(CC1)CCN(C(C1CCSC1)=O)CC2C 45439,C1(C)(CC)CC(F)(F)CN1C(=O)Nc1ccc(C(=O)OC)c(OC)n1 45440,Cc1[nH]c(=NC2CC(NC(c3cnc4n3CCC4)=O)C2)ccc1C#N 45441,N1(C(C2CN(Cc3ccccc3C(=O)O)CCS2)=O)CCC2(CC2)C1.CO 45442,c1(C(=O)NCC(c2ccccc2F)NC(C2CC(CC)C2)=O)cnc(C)cc1C 45443,N1(CC(=O)NCC(CNC(CCN(C(CC)CC)C)=O)O)OC(C)(C)CC1=O 45444,N1(C(C2C(C)C2C)=O)CCC2(CC1)CC2CNC(C1(C2(O)CCOC2)CC1)=O 45445,CCCCCCCC(=O)NC1(c2nnnn2C2COC2)CCCC(C(F)(F)F)C1 45446,c1(CC)ccc(F)c(C(N2CCCC(C)(CNC(c3nnccc3C)=O)C2)=O)c1 45447,C1(CNC(C(CC)C)=O)CCN(C(=O)C(C2COC(C)(C)O2)O)CCC1(F)F 45448,c1(C(=O)NC(CSC)(C)C(N2CCC3(CCO3)C2)=O)ccc(C)cc1F 45449,CC1C(NC(=O)COc2cc(F)cc(Cl)c2)CCCN1C(C1CC1C(C)(F)F)=O 45450,C1(CC)CC(C)(C)CN1C(c1n[nH]c(-c2ncc(F)cn2)n1)=O 45451,C1(CNC(C(c2cccc(C)c2)F)=O)N(C(C2CCNC2=O)=O)CCCC1(C)C 45452,N1(CCNC(C(COC(C)C)N(C)C)=O)CCC(NC(=O)C=CCF)CC1 45453,N1(C(Cc2cc(C)no2)=O)CCCC(C2CC2NC(c2cncc(C)n2)=O)C1 45454,C(=O)(C1=CCCCC1P(C)(C)=O)NCCCCN(C)C(C1Cc2nccn2C1)=O 45455,c1(C(=O)NCCC2CN(C(=O)CC3CCCNC3=O)CCO2)cccc(F)c1O 45456,C1(N(C(=O)CC(=O)NCCC(N)=O)C)CN(C(=O)CCCC2CC2)CC12CC2 45457,c1(C(=O)OC)ccc2[nH]nc(C(=O)NCC(C)CN(C(=O)C(O)COC)C)c2c1 45458,C1(N2CCC(NC(N3C(c4cccnc4)CC(C)C3)=O)C2)CC(C)N(C)CC1C 45459,C1(C(=O)NCCOCC)CCCN1C(C1(c2ccccc2)CCC1)=O 45460,Cc1cc(C(N2CCCC(CNC(c3cc[nH]c(=N)c3N)=O)C2)=O)c(C)cn1 45461,C1(C)(COC)CN(C(c2ccc(F)s2)C(=O)NCCC2(C)CC2)CCO1 45462,CC(CN(C)C)C(=O)NCCCC(C)NC(c1csc(-c2nc[nH]n2)n1)=O 45463,N(C1CN(C(C2CC2F)=O)Cc2ccccc21)C(=O)Cc1ccc2nc[nH]c2c1 45464,C1(CC)CN(C(C2CC=CCC2)=O)CCC1CNC(=O)Cn1ncc(O)nc1=O 45465,CC1C(NC(=O)C=Cc2cn(C)nn2)CCN1C(=O)CC1OCCO1 45466,Cc1ccc(NC(C2CN(C(=O)CNC=O)CC(C)(C)C2)=O)c(F)c1F 45467,c1(N2CCC(=C)C2)nc(N2CCC(CCN(C)C)CC2)nc2c1ncn2CC 45468,C1(NC(=O)CCC2NC(=O)NC2=O)CC12CCN(C(=O)C1=CCOCC1)C2 45469,C=Cc1cncc(C(=O)NCCC2CN(C(=O)C3=C(C)OCC3)CC(C)O2)c1 45470,C(=O)(C(C(=O)OC)OC)N1C(C(C(=O)N(c2ccccc2)CC)(C)C)CCC1 45471,C1(C(NOCC=CC)=O)CCCN(C(=O)C(C)(C2CC2)OC)CC1 45472,c1(C(CCN2CC2)=O)cc(-c2ccoc2)on1.C(=O)(COC1CC1)C1(N)CC1.CC 45473,C=C=C(C)CC(=O)N1CCCC1C1(NC(=O)CC2CCCCC2C)CC1 45474,c1(NC(C23CC(C(=O)NC(CC=C)CO)(C2)C3)=O)cc(Br)ncc1[N+](=O)[O-] 45475,N1(C(CC(C)CF)=O)CCN(C(c2cccn2Cc2cccs2)=O)C(C)C1 45476,CCC(O)(CC(=O)NC1CCC1CNC(=O)C=CCO)c1ccccc1 45477,C1(CC(=O)NCCOCCNC=O)CC(O)C12CCC2.c1(C(=O)CCN)ccc[nH]1 45478,c1(NC(C(C(C)OC)NC(c2csc(=N)[nH]2)=O)=O)cnn2c1CCCC2 45479,C#CCC(C)(C)C(=O)N1CC2CCC2(CCNC(c2cccc(F)c2OC)=O)C1 45480,C(CC(C)C)(C(=O)NCC1(OC)CN(C(=O)C(CO)NC(N)=O)C1)NC(C)=O 45481,c1(COC)cccc(C(N2CC(C(C)NC(c3ccc(C(C)(C)C)[nH]3)=O)C2)=O)n1 45482,N1(C(C(C)CNC(=O)CN(C)C)=O)CCCC(O)(CO)C1 45483,C1(C(=O)NCC(CNC(C2=CC(C)(CC)C2)=O)(C)C)CC2CCC(C1)C2O 45484,CC1CN(C(=O)CC(C)c2ccccc2)CC1NC(=O)CC(C)(F)F 45485,c1(NCC)ccccc1C(N1CC2CC2(CNC(c2csc(C(N)=O)n2)=O)C1)=O 45486,O=C(C1CCCn2cnnc21)NCC1(F)CN(C(C2C3CCCCCC23)=O)C1 45487,N1(C(c2c(C)onc2)=O)CCN(C(c2cnc(C3OCCO3)s2)=O)C(C)C1C 45488,C(=O)(C1=CCC(F)(F)CC1)N1CC(C(C)NC(=O)C=CC2CCC2)OCC1 45489,CP(C)(=O)CCC(=O)NCC1CCOC1C(=O)NCC#CC#CCO 45490,C1(CN(C(=O)C=C2CCOCC2)C)C2CN(C(=O)CCN3CCCS3(=O)=O)CC12 45491,C1(NC(C2CCC=CO2)=O)CN(C(=O)CCC2CCOC2)C2CCCCC12 45492,c1(C(N2CC(C)(NC(=O)Cc3cccnc3)C2)=O)cncc(N)c1 45493,N#CC1(C(=O)NCc2csc(C(=O)N(CCC(F)F)CCO)c2)CCCC1 45494,C1(F)(CNC(C2C(CC)CCC2)=O)CCN(C(=O)Cc2ccc(Cl)cc2F)CC1 45495,C#CCC(C)(CC)C(=O)NC(CNC(c1nccn1C(C)C)=O)C1CC1 45496,C1(CCNC(C(F)=CCC)=O)CN(C(=O)CCN2C(=O)CCC2=O)CC(C)O1 45497,c1(OC)ccc(Cl)c(COC(=O)Cn2c(C)cccc2=O)n1 45498,N1(Cc2nc(C)sc2)CCCC(NC(=O)NCCC2COCCO2)C1 45499,N1(C(CP(C)(C)=O)=O)CCN(C(=O)CCCn2cccn2)CC1c1cn[nH]c1 45500,C(C)(CCC(=O)N1CCC(C(C(C)C)NC(=O)COCCN(C)C)CC1)SC 45501,c1(CC(=O)NCCCC(C)NC(c2ccsc2)=O)cnccc1C(F)(F)F 45502,c1(C(N2C(CN(C(CSC(C)C)=O)C)COCC2)=O)n[nH]c2c1COC2 45503,N1(C(C(C2CCCCC2)NC(C2N(C)CC2)=O)=O)CCC2(CCOC2)C1 45504,c1(NC(=O)NC2(C(=O)OC)CC(OC)C2)ccc2c(c1)CC(N)CCC2 45505,Cc1ccc2oc(C(=O)N(C3CN(C(c4cn(C)c(C(F)F)n4)=O)C3)C)cc2n1 45506,C12(C(N(CCSC)CC)=O)CCC(CC1NC(c1cc(OC)n[nH]1)=O)C2 45507,CCC(C)C(O)CC(=O)NCC(N1CCN(C(=O)Cc2nnc(C)o2)CC1)=O 45508,CC(CCNC(C1(CNC(=O)CC2CCC(C)C2)CCCC1)=O)C(C)(C)C 45509,Cc1cccc(Cl)c1S(=O)(=O)NC1CN(Cc2cncc(O)c2)CC1C 45510,C1(N(CC(=O)N(CC(CC)NC(CC)=O)C(C)C)C)COC2COCC12 45511,C1(C(=O)NC2CCN(C(CC(C=C)(C)C)=O)C23CCC3)CCc2nnc(O)n2C1 45512,C1(C(=O)NC2CC(NC(C(CCC)NC(C)=O)=O)C2)CC2CCCC(C1)C2 45513,n1(CC)nc(C2CC2)cc1S(=O)(=O)NC1(CC2CC2(Cl)Cl)CCC1 45514,N1(C(c2cnc(NC(C)=O)o2)=O)CC(NC(=O)C(C)(C)N2CCCCC2)C2CC12 45515,C1(C(N2CCOC(CC3CC3)C2)=O)CCOCCN1C(=O)CC1CC=CCC1 45516,C1(Cc2nc(CCSC)nn2-c2cccc(C(C)C)c2)CCC(F)(F)CC1 45517,N1(C(CC(CC)C)=O)CC(NC(C2CC3CCC2CC3)=O)CC(C)(C)C1 45518,c1(-c2scc(C(=O)NCCCCC#C)n2)cnn2c1CCCC2 45519,c1(C(N2CC(CC)(CO)C2)=O)n[nH]c2c1CN(C(C1C3CCCCC13)=O)C2 45520,CCC(C(=O)NC1CCSC12CN(C(c1ccc(CC)nc1C)=O)C2)C(C)(F)F 45521,C12(C(N3CCC(N(CC#C)C(C4CCC(C)O4)=O)CC3)=O)CCC(N=[N+]=[N-])C1C2 45522,CCCC(F)C(=O)N1CC(F)CC1CC(=O)NCc1cncc(OC)c1 45523,CS(=O)(=O)c1ccsc1C(=O)NC1C2CC1N(C(C1(C#N)CC13CCC3)=O)C2 45524,C(=O)(C(O)C(C)(C)C)N(CC(O)CN(C)C(c1cc(F)n(C)n1)=O)C 45525,C1(CN(C)C(C2CCCS2(=O)=O)=O)CCCN(C(=O)CN2CCCC2=O)C1 45526,c1(C(=O)NCC(=O)NC23CCC(C2)N(C(=O)CC2CCC2)C3)cc(Cl)ccc1Cl 45527,C(=O)(C1=COCCO1)N1CCC(CCCCCNC(C2CCCS2)=O)CC1 45528,c1(C(=O)NCC2N(C(C(C)(Cl)Cl)=O)CC2)cc(C2CC2)oc1C1CC1 45529,Cc1cccnc1-c1cn(C2CCCN(C(c3cc(Cl)cn3C)=O)C2)nn1 45530,C1(C(=O)NCCCNC(C(C)Oc2ccc(F)cc2)=O)CCc2ncccc2C1 45531,C1(C(=O)OCc2nnnn2-c2ccccc2)CCc2cc(F)ccc2O1 45532,CCCC(C(=O)N1CCCC1(C)c1cn(Cc2cnco2)nn1)OC 45533,N1(C(C(c2cnn(C)c2)OC)=O)CC(NC(=O)COC(F)(F)F)C(C2CC2)C1 45534,CC(C)(C)C(C)(C)C(=O)NC1CCC(NC(c2[nH]ccc2C2CC2)=O)CC1 45535,C1(C(=O)NCC(C)CC(F)(F)F)CC2CN(C(=O)Cn3cnnc3O)CC2C1 45536,c1(C(N2CCC(CC(=O)OC)C2)=O)nccc(OC)c1OCc1ccccc1I 45537,c1(C(=O)NCCC2CN(C(CN(C)C(N)=O)=O)C2)cncc(N(C)C)n1 45538,C1(CNC(=O)C#CC2CCOC2)Cc2ccccc2CN1C(=O)CCC1CCC1 45539,Cc1ccc(C=CC(N2CC=CC(C(=O)NC(C3CCOC3C)(C)C)C2)=O)cc1 45540,C(c1cc(C)cc(C)c1)=CC(=O)NCCC(CCNC(C(C(C)C)OC)=O)C 45541,c1(CC)cnc(Cl)nc1N(C)CCOCCN(C)C(C1CCC2CC2C1)=O 45542,CCCC(CCC)=CC(=O)NC1CN(C(=O)Cc2ncccc2C)C2CC12 45543,Cc1ccccc1-c1nsc(N(CC(=O)NC2CC(O)C23CC3)C)n1 45544,c1(C(N2CCC(C(C)C)(CNC(C3CCN(C)C3=O)=O)C2)=O)c[nH]nc1[N+](=O)[O-] 45545,N1(C(c2cc(OC)ncn2)=O)CCC(NC(=O)Cc2c(F)cccc2F)C(C)C1 45546,c1(CC(N2CC(n3cc(C(C)OC)nn3)(C(=O)OC)C2)=O)ccc(O)c(F)c1 45547,Cc1ccc2nc(C(N3CCC3CNC(=O)C(C)OCC(F)(F)F)=O)c(N)n2c1 45548,c1(C(=O)NC(C2N(C(C(CC)n3ccnc3)=O)CCC2)C)ccccc1CO 45549,C(CC(C(=O)NCCCC1CC1C)NC(=O)CN1CCC(=O)CC1)OCC 45550,C(N=c1[nH]c(=NCCc2csc(=N)[nH]2)[nH]c2cc[nH]c12)c1nccc(NC)c1 45551,C12(NC(c3ccc(=N)[nH]n3)=O)CCCC1(F)CN(C(C1CCCSC1)=O)C2 45552,C(C(C(=O)NCC1(C2CCC2)CC1)NC(=O)CC1CCC1)SC(C)C 45553,c1(C(=O)NC2C3(CN(C(c4c(C)nsc4)=O)C3)SCC2)ccc2c(c1)CC(C)O2 45554,C1(C(=O)NC(CN(C)C(c2cc(Cl)c(Cl)n2C)=O)(C)C)CCC2CC2CC1 45555,c1(C(=O)NC(CC=C)CNC(=O)C(c2ccc(F)cc2)O)c[nH]c2nccc-2c1 45556,c1(OCC)cnc(C(=O)NC2CCC(CNC(c3cc(N)ccn3)=O)C2)cn1 45557,C(=O)(C1=CCN(C(=O)C(c2cnn(C)c2)=O)CC1)NC(CC(CC)C)C 45558,CCCC(CC(=O)NC1CCC(OC)CC1)NC(c1cc(C#N)oc1C)=O 45559,c1(OCC(=O)NCCCN(C(=O)CCc2ccncc2)CC)cnn(C)c1 45560,C(=O)(CS(F)(F)(F)(F)F)NCC1(C)CCN(C(C(C)OC)=O)C1 45561,CN1CCC(NC(=O)CC(C)(C)C)C12CCCN(C(=O)CCC#N)C2 45562,Cc1c(C(N2CCOCC2CCNC(c2cccc(Cl)c2)=O)=O)ccn1C 45563,c1(OCCOC)ccc(C(=O)N)cn1.c1(CNC(=O)C(O)CS)cccnc1SC 45564,Cc1ccnc2ccc(C(N3CCN(C(=O)CCC(C)(F)F)C(C)C3)=O)cc12 45565,c1(C(C)=O)ccc(S(=O)(=O)NC2COCCN(Cc3cc(C)ccc3Br)C2)cc1 45566,N1(C(C(C)(C)OC)=O)CCN(C(=O)C(=O)NC(c2nc(C3CC3)cs2)=O)CC1 45567,C1(CC)CC2(CCN2C(c2cn(C)nc2Cl)C(=O)NC2CCCC2)C1 45568,C1(NC(CCC(C)OC)=O)CCN(C(=O)CCc2cc(C)cc(C)c2)CC1(C)C 45569,N1(C(CC(C)O)=O)CC2CCC(N(C(=O)CCc3cnn(C)c3)C)C2C1 45570,CC(C)C(=O)NNC(=O)NC(C1CN(c2nnc(C3CC3)s2)CCO1)C 45571,CCC(C(=O)N(C(CNC(c1cccc2c1CCO2)=O)C1CC1)C)C(C)(F)F 45572,c1(CC(=O)NCC2C3CN(C(C4OCCN(C)C4)=O)C2C3)ccnc(Cl)c1F 45573,C1(C(=O)NC2(CNC(c3csc4nccn34)=O)CCCC2)CCCCC12CCC2 45574,CCCCCCC(C)OOC(c1cc(C2CC2)n(-c2ccccc2)n1)=O 45575,N1(C(COCC(=O)OC)=O)CCC(CNC(c2scnc2C)=O)C(C)C1 45576,Cc1c(C(=O)N(CCNC(C2(CO)COC2)=O)CC2CC2)sc2cccc(F)c12 45577,C=CCCCCC(=O)NC1CC1CNC(=O)CCCNC(c1scnc1C)=O 45578,CS(=O)c1ccc(CC(N2CCC(NC(C3CC(C)(F)C3)=O)C2)=O)cc1 45579,N1(C(C2CC(NC(=O)CSC(F)F)C23CCC3)=O)CCc2nc(O)[nH]c2C1 45580,N1(C2CCN(C(C(C)(C)SC)=O)C2)CCN(C(C2(CO)CCC2)=O)CC1 45581,c1(C(C)C(=O)NC(C2CCN(Cc3ccncc3)C2)C)cccc(Cl)c1 45582,C1(CC(=O)OCC)CCCCN1C(c1n[nH]c(CC)n1)C(=O)NCCN(C)C 45583,N1(C(C(CC)CC)=O)CC2CCC(C1)N2C(c1cc(Br)cc(F)c1F)=O 45584,c1(CC)ccc(C(=O)NCC2CCCN2C(c2cnc(C)nc2CC)=O)c(F)c1 45585,Cc1nccnc1C(=O)N(C)CCNC(=O)CC(C)Cc1cccc(F)c1 45586,N1(C(c2ccc(CC)o2)=O)C2CCC1(CNC(C1CC(CN(C)C)C1)=O)CC2 45587,C12(CC(=O)NCC3CCN(C(=O)CCc4ccncc4)C3)CCC(CC1)OC2 45588,Cc1c(C(N2CCCC(N(C(=O)C#CC3CC3)C)C2)=O)cc(N)cc1O 45589,C(CC1CCCO1)N=c1[nH]c2ccc(S(=O)(=O)N3CCCC(CCO)C3)cc2s1 45590,CC1(C)COC(CC(=O)NC2(C3CCCCN3C(c3coc(Cl)c3)=O)CC2)C1 45591,C(=O)(C(C)(O)C1CC1)NCC(C)CN(C)C(c1n[nH]cc1Br)=O 45592,N1(CCCc2ccc(C)cc2)C(=O)CN(CCc2ccc(F)cc2F)C1=O 45593,C1(F)(CNC(CCc2nc(C)c(C)[nH]2)=O)CCCN(C(=O)CCC(C)(F)F)CC1 45594,n1(CC)ncc(Cl)c1C(=O)NCC1CCC(F)(CNC(c2csc(C(N)=O)n2)=O)C1 45595,N1(C(C(C)(C)C2CCOC2)=O)CC2C(C(=O)NC3CC3F)C2C1 45596,C1(CC)CN(C(C2CC=CCO2)=O)CCN1C(C12CC(c3ccccc3)(C1)C2)=O 45597,c1(CC(=O)N(C(CNC(CSCC)=O)C)C)cc(Br)ccc1Cl 45598,c1(C(=O)NC2CCC(N(C(c3ccc(COC)o3)=O)C)C2)nc(C)ccc1F 45599,C(CC(=O)N=c1cc[nH]cc1O)c1c(-c2c(NC(C)C#N)nccc2)cccn1 45600,C1(NC(CNC(c2c(C(C)=O)cccc2)=O)=O)(CO)CC2(C1)OCCO2 45601,c1(NC(C2(CCNC(CS(CC)=O)=O)CC2)=O)cccc(F)c1O 45602,c1(C2CCCN(C(c3ncc(I)s3)C(=O)NC(C)(C)C)C2)ccc(F)c(F)c1 45603,n1(CC)cnc2c(NCCCC(C)NC(=O)COc3ccon3)nc(Cl)nc12 45604,CCCCS(=O)(=O)CC(=O)NC1CN(C(=O)COc2c(Cl)cccc2Cl)CC1C 45605,c1(CNC(N(C2(c3cc[nH]n3)CC2)C)=O)ncc(C(F)(F)F)n1C 45606,C1(CNC(C2(SC)CC2)=O)CCCCN(C(c2ccc(N)cc2Cl)=O)C1 45607,CN=c1[nH]cc(C(=O)NC(c2ccccc2SC)CNC(c2cc(C)sn2)=O)o1 45608,c1(C(=O)NCC2CC(C)(C)CN2C(c2cnsn2)=O)cc2ccccc2[nH]1 45609,c1(CC(=O)NCC2CCC2NC(C23C=CC(CC2)C3)=O)cc(F)ccc1F 45610,Cn1ccc(C(=O)NCC2CCN(C(C3CC4CCC3O4)=O)C23CC3)cc1=O 45611,C1(C(=O)NC(C)(C)CNC(=O)CC2SC(=N)NC2=O)CS(=O)(=O)CCO1 45612,c1(OC)cc(C(N2CC3CC(NC(C4CCOC4)=O)C3C2)=O)ccc1C 45613,Cc1ccc(C2(CNC(=O)Nc3cccc(CC#N)c3)CCC2)c(F)c1 45614,N1(C(c2ccc(C)nc2C)=O)CCCC(F)(CNC(=O)C(O)C(C)(C)C)CC1 45615,C1(C(=O)NCc2cc(C)nc(C)c2)N(C(=O)CC2CC(C)C2)CCCC1(C)C 45616,N1(C(C(C2CC(NC(C(CC=C)OC)=O)C2)F)=O)CCC12CN(C)C2 45617,c12ccnc(c1)NC2=O.C(CN(C)C1CC1)(CC(C)C)NC(CN(CCC)C)=O 45618,C1(CC(N)=O)(CNC(C2(C)CC(=C)C2)=O)CCN(C(=O)C(O)CC(=O)OC)CC1 45619,N1(C(CCC(=C)Br)=O)CC2CC(C1)CN(C(=O)CCC(CC)OC)C2 45620,CCCC(C)(C)C(=O)N1CCCCC(CNC(=O)C(O)CCSC)C1 45621,C1(CNC(C2CC(SC)C2)=O)CCCCCN1C(c1cc(N)ccc1C)=O 45622,c1(OC(C)C)ccc(C(=O)NC2CCCCC2CNC(c2ccnnc2O)=O)nn1 45623,C12(CCN=C(NCC3(COC)CCCC3)NC3CC3C)CC3CC(CC(C3)C1)C2 45624,c1(-c2nc(-c3c(C)cc(OC)nc3)nn2-c2cccnc2)ccc2cncn2c1 45625,C(C)(CC(=O)NC(c1nocc1C(=O)N(C)Cc1ccn(C)n1)C)SC 45626,Cn1ncc([N+](=O)[O-])c1C(=O)NCC(O)CCNC(c1cc(Cl)cc(Cl)c1O)=O 45627,CC12CC(CC1C(=O)NCC1(CNC(C3(O)CCOCC3)=O)CCCC1)C2 45628,n1(CC(=O)NCC(C)(C)NC(C2C(OCC)C2)=O)c(C)cc(O)cc1=O 45629,N1(Cc2cn(C)nn2)CCC2(CCN(C(c3ccn4ccnc4c3)=O)CC2)CC1 45630,C(=O)(CCCS(N)(=O)=O)N1CC(NC(C2(C#C)CCC2)=O)C(C)C1 45631,c1(C(=O)NCC2(C)C(NC(CP(C)(C)=O)=O)CCC2)ccc2nsnc2c1 45632,Cc1cnc(C(C2CC2)NC(C2CS(=O)(=O)C2)=O)s1 45633,n1(CC)ccc(C(=O)N(CCCNC(c2cc(C)cs2)=O)CC2CCCC2)n1 45634,C1(NC(=O)OC(C)(C)C)CCN(C(c2cncc(C3CC3)c2)=O)C(C)C1 45635,C(C(C)CC(=O)NC1(C)CC(NC(c2ccc(OC(F)F)nc2)=O)C1)OC 45636,Cc1ccc(F)cc1C(=O)NCC(O)CC(=O)N(C(C(N)=O)C1CC1)C 45637,C#CCC(CC)NC(=O)CCNC(C1(CO)CCOC1)=O 45638,C1(NC(CN2C(=O)NCC2)=O)CCN(C(C2CC3C=CC2C3)=O)C12CCC2 45639,C1(CN(C(C(n2c(C)ccn2)C)=O)C)CN(C(=O)CC2CC2(C)C)CC12CC2 45640,c1(C(=O)NC2CCCN(CC(CC)OC)C2)cnc2c(C)cccc2c1 45641,S(=O)(=O)(c1cccnc1N1CCS(=O)CC1)NCC(c1ccccc1Cl)C 45642,N1(C(C)=O)CCN(C(c2cc(N)c(Cl)cc2Br)=O)C2(CC2)C1 45643,N1(C(CC=C(C)C)=O)CC(F)(F)CC1CCNC(c1coc(Br)n1)=O 45644,C1(NC(c2cn(C)nn2)=O)CCN(C(=O)C(=Cc2cccc(F)c2)F)C12CC2 45645,C1(OCCC)CN(N2CC(N(C)CCOC)C2)C1 45646,CN1CC2(CC2)CC1C(=O)NC1CC(O)CN(C(C2(C3CC3)CC2)=O)C1 45647,CCCCCCCCNC(=O)N(C1CCC1)C(c1ccc(C#N)cc1)C 45648,c1(SC)cncc(C(=O)NCC=C2CCN(C(=O)CCn3cc(C)cn3)CC2)c1 45649,C#Cc1cc(C(=O)NNC(=O)Cc2ccccc2C)cc(I)c1 45650,C1(NC(CCCOC(C)C)=O)CCC(CNC(c2csc(S)n2)=O)CC1 45651,c1(C(C)C(=O)N(CCCCN(C)C(C23CC(F)C2C3)=O)C)ccccc1Cl 45652,C1(C)(NC(CNC(C(N2CCOC2=O)C)=O)=O)CN(C(=O)CC2CCCN2C)C1 45653,N1(C(CCc2c(C)noc2)=O)CCC(NC(c2cccnc2)=O)C1C(C)(C)C 45654,C1(NC(C2CC3CCC2CC3)=O)CN(C(=O)C(C2CCCCC2)O)CC2(CC2)C1 45655,C1(C(=O)NC2C(NC(CSc3cn(C)nc3)=O)COC2)CCCCNC1=O 45656,Cc1ccccc1C1(C(=O)NCC(CO)NC(=O)C(C)OCCN(C)C)CCC1 45657,C(=O)(C(CN(C)C)C(C)C)N1C(CNC(c2c(C)oc(C(C)C)c2)=O)CC(F)C1 45658,c1(Cc2cncc(C)c2)nn(C)c(Cl)c1-c1nc(CC2CC2)nn1CC 45659,N1(C(c2c(C)oc(CO)c2)=O)CC2(C1)CN(C(C1CC=CCC1)=O)CCO2 45660,C(C)(C)(C(F)(F)F)O.n1(C(C)(C)C)cc(CC(=O)NCCCNC(=O)CC2CC2)cn1 45661,N1(C(C=CC2C(C)C2(Cl)Cl)=O)CC2(CCN(C(c3cc(C(N)=O)no3)=O)C2)C1 45662,c1(OC)cc(NCC2CC(NC(C3CN(C)C(=O)N3)=O)C2)nc(OC)n1 45663,C=C1CCN(C(c2ccn(CCNC(=O)Cc3nocc3C)c2)=O)C1 45664,C123CN(C(CF)(C1)C2)C3=O.C1(C(=O)OC)CCCC(OC)C1.S1(=O)(=O)CCN1 45665,C1(NC(C=CC)=O)CCN(C(c2c(-c3ccccc3)cnn2C)=O)CC1F 45666,Cc1c(CNC(C2CCCN2C(=O)C(C)(O)C2CC2)=O)nnn1C 45667,Cc1nn(C)cc1CC(=O)N(CCCOCCNC(C1(C)CC=CCC1)=O)C 45668,N1(C(CC(=C)C)=O)CC(O)CC1CNC(C1CC(=O)N(c2ccc(F)cc2)C1)=O 45669,C(=O)(C1=CCCCCC1)N1C(C)CC(CC(=O)NCC2COCCOC2)C1 45670,C1(NC(C(C2CCC2)OCC)=O)CCN(C(=O)CN(C)C(C)C)CC12CCC2 45671,C(=O)(C1=C(C)OCCS1)N1CC(C(N2CCCC(O)(CC)C2)=O)OCC1 45672,N1(C(C(=O)NCC(C)NC(=O)C(N2CCC(C)C2)=O)C)CCOCC1 45673,C1(OC)CC(NC(=O)CCCCCn2cnnn2)CN(C(=O)C(C)(C)C2CC2)C1 45674,N1(C(C(CC)C(C)C)C(=O)NCC(F)F)CCC2(CC1)C(C)(C)C21CCC1 45675,CC#CCCC(=O)NCC(C)(O)CNC(C1COCCN1CC(F)(F)F)=O 45676,N1(Cc2c(OC)cccc2)CCc2sc(-c3cnccc3C)nc2C1 45677,c1(OC)cc(C(F)(F)F)[nH]c(=NCC(C)NC(=O)C(F)C(F)(F)F)n1 45678,C12(C(N(C)CC3CCN(C(=O)C(O)CF)C3)=O)CCC(C(F)(F)F)(CC1)CC2 45679,C(CCNC(C1CC1Cl)=O)N(C(=O)C=CCO)CC 45680,N#Cc1ccc(N)c(C(N2CCC(C(=O)NCC3CCC(F)(F)C3)C2)=O)c1 45681,C1(C(=O)OC)CC2CCC(C1)C2NC(C1OCCC1C)=O 45682,c1(C(N2CCCC2CNC(C23CCC(CC2)O3)=O)=O)cccc2ccnn12 45683,c1(C(=O)NCCC(C)N(C(c2[nH]cc(C)c2C)=O)C)onc2ccccc12 45684,c1(C(F)(F)F)cccc(CCNC2CC3CC3C2)c1Br 45685,CC(C(=O)N1CC(CN(C(=O)CCC2CC2)C)C(C)(C)C1)S(N)(=O)=O 45686,C12(NC(C(C)Cc3ccc(Cl)cc3)=O)CCC(C1)N(C(=O)CCc1cnc[nH]1)C2 45687,O=C(C#CC1CCC1)NCC1(CNC(c2ccc(C(F)F)o2)=O)CCC1 45688,Cc1cc(Cl)c(C(=O)NC(C2CCCN(Cc3ccncc3C#N)C2)C)c(Cl)c1 45689,Cc1cn2c(-c3cn(CCNc4cc(-c5ccc(F)cc5)ns4)nn3)csc2n1 45690,C(CC1=CCN(C(c2n[nH]c(C)c2N)=O)CC1)NC(C1(CC)CCOCC1)=O 45691,C1(NC(CC2CC(=C)C2)=O)CCN(C(C2CC3CC3CC2C)=O)CC1F 45692,C#Cc1cc(C(=O)NCC(C)NC(=O)C(C)C2CCC2)cc(F)c1 45693,N1(C(CCC=CC)=O)CC(NC(C2(C(C)(C)O)CC2)=O)CC12CCOC2 45694,C(=O)(CC(C)C(C)(C)NC(=O)CC1CCCSC1)N1CCC(C#C)(O)C1 45695,N1(C(c2cn(C)nc2-c2ccncc2)=O)CC2CCCC1(CN)C2 45696,C1(OC(CC)CNC(=O)NC(Cc2cccs2)CC)CCOCC1 45697,c1(CC(C(=O)NCC(CSC)(C)C)NC(C23CC(F)(C2)C3)=O)ccccc1Br 45698,c1(OC)ccnc(N(Cc2ccccc2-n2cncn2)CC2CC2)c1 45699,C1(CNC(C2CNC(=O)N2)=O)CCCN(C(C2CC3CC3C2)=O)C1 45700,Cc1nc(CNC(=O)C(C2CCN(C(c3cc(C4CC4)on3)=O)C2)F)c(C)[nH]1 45701,C(=O)(CCCC(C)(C)C)NC(CC#C)CC(=O)NC(CC1CC1)CC 45702,C1(CNC(C2(C(=O)NC)CCC2)=O)CC2CN(C(C3(F)CC3)=O)CC12 45703,CC(CNC(=O)C(=O)NCC(F)F)(C1CC1)NC(=O)CNC1CCOC1 45704,C1(C(N2CCCC2C(=O)NCCC2COCCO2)=O)(CC)CCCCC1 45705,O=C1CC2(CCN(C(C3CN(C(c4cccnc4O)=O)CCO3)=O)C2)CN1 45706,C12(CNC(c3c(OC)nccc3)=O)CCCC1N(C(=O)C(C)NC(N)=O)CCC2 45707,N1(C(C2C=CCC2)=O)CCN(C(C2(c3cccs3)CC(F)(F)C2)=O)CC1 45708,C1(CNC(CC2(OC)CC2)=O)CC(C)N(C(=O)CC2(c3ccccc3F)CC2)C1 45709,c1(C(=O)NCC2CCN2C(=O)COc2ccsc2)ccncc1F 45710,C12(C(=O)NCC3OCCN(C(C4(N5CCCC5=O)CC4)=O)C3)CC(C1)S(=O)(=O)C2 45711,c1(N(CC(C)(C)CNC(C)=O)C(=O)CC(=O)OC(C)(C)C)cn2cc(C)sc2n1 45712,Cc1ccc(C(N2CC3CCC(C2)N3Cc2c(F)cncc2F)=O)c([N+](=O)[O-])c1 45713,c1(C(=O)NC2(CO)CN(C(c3ccnc(C)n3)=O)C2)cccc2nccn12 45714,C1(CCNC(=O)NC(C)CN)CC(OCC(F)(F)F)C1 45715,N1(C(C2=CC(C)C2)=O)CCC2C(C1)CN2C(=O)Nc1nccn2nccc12 45716,c1(C(=O)NCC2C3CN(C(C(C)NC(CC)=O)=O)C2C3)ccc(C(C)=O)cc1O 45717,C1(C(=O)NCC2CN(C(c3cc(OC)n(C)n3)=O)C2)CCCC(C)(C)O1 45718,Cc1nn2ccccc2c1C(=O)NC(c1cn(CC(c2cccnc2)O)nn1)C 45719,CCC(CNC(C1CCN(C)C1C)=O)(CC)C(=O)NC1CC(C)(C)OC1(C)C 45720,Nc1nc(C(N2CC3CC(NC(c4cc(C(F)F)cs4)=O)C2C3)=O)ccc1O 45721,c1(CC(=O)NC2CC(CNC(c3nc(C(C)OC)sc3)=O)C2)ccc(Cl)nc1 45722,C1(C(N(C)CCC2CCOCC2)=O)(CO)CCN(C(=O)CC2CCOC2=O)C1 45723,Cc1c(C(N2CCCC2CN(C)C(C2(C#N)CC(C)C2)=O)=O)ncn1C 45724,C(C(=O)N1CCCC1C(=O)NCc1ccnc(C)c1)(C(C)C)NC(C)=O 45725,Cc1ccc(CNC2CC2Nc2ccc(C(=O)NC(C)C)nc2)c(Cl)c1Cl 45726,C=C(Br)CCC(=O)NC1CCC(CNC(=O)C=C(C)C)C1 45727,C1(C(N2CCC(CNC(c3ncc(C(F)F)s3)=O)CC2)=O)CCC2CC2CC1 45728,C(=O)(C(=O)C(C)CC)NCC(CC=C)NC(C(C=C)CC)=O 45729,c1(C(=O)NCCC(=O)NC(C2CC2c2cscn2)=O)ccoc1CCCO 45730,C1(O)(CN(C(=O)CCCc2cccc(Cl)c2)C)CCN(C(=O)C(O)CC2CC2)C1 45731,C(=O)(CCC(=O)NCC1CN(C(=O)CN2C(C)CCC2C)CC1C)NC 45732,N1(C(c2cc(C(C)=O)oc2C)=O)CC(NC(=O)Cc2sc(C)nc2C)CC(C)C1 45733,CC1CN(C(=O)COCC2CCCO2)CC1CNC(c1ccsc1C#N)=O 45734,CC1CC(C(N2CCC(NC(c3nsnc3O)=O)C(C)C2)=O)CC(C)O1 45735,S(=O)(=O)(CCC(=O)NC1CC(NC(=O)C(O)C(C)(C)C)C(O)C1)NC 45736,N1(C(CN(C(C)C)C)=O)CCC1CNC(=O)CC1(CO)CC1 45737,c1(NC(C2CN(C)C2)=O)ccc(O)c(CO)c1.c12nc(c(C)o1)C(=O)NC2 45738,N1(C(c2c(SC)cccc2)=O)CC2CCN(C(=O)C(F)n3cccn3)CC2C1 45739,Cc1ccc2c(N3CC(C)OC(C)C3)nc(=NCc3ccsc3Cl)[nH]c2c1 45740,c1(C(=O)NC2CCCC(NC(C3N(CC)CCC3)=O)C2)cc(C#N)oc1C 45741,CC1CCc2ncc(C(N3CC4CC(C3)N(C(c3occc3Cl)=O)C4)=O)n2C1 45742,N1(C(c2nc(F)ccc2F)C(=O)NC)CCCC1C1CCCO1 45743,C1(CNC(C(CC)C)=O)CCN(C(=O)Cc2cccc(NS(C)(=O)=O)c2)C1(C)C 45744,C12(C(N(CCCCCCNC(=O)C3=CCCSC3)C)=O)CC(C)(C1)OC2(C)C 45745,C1(CC(=O)N(C2C3CN(C(=O)COCC(=O)OC)CC23)CC)CC(C)(C)CCO1 45746,C1(CCC)CCCC1C(=O)NC12CC(C(N3CCC3(C)C(=O)NC)=O)(C1)C2 45747,Cc1ccc(CCC(N2CC3(C2)CN(C(c2cccc(=O)o2)=O)C3)=O)c(C)c1 45748,CC1CN(C(=O)CC2CN(C)C2)CCN1C(c1coc(C2CCC2)n1)=O 45749,Cc1ccc(C(=O)NCC2(O)CN(C(=O)C(C)N3CCC3)C2)o1 45750,c1(C(N(CCCCN(C(C(c2ccnn2C)C)=O)C)C)=O)cc(O)nn1C 45751,C1(NC(CSCC=C)=O)CCC2(CC1)CCN(C(=O)CC1CCCC(C)(C)O1)C2 45752,c1(C(N2CC(NC(=O)C=CCF)C2)=O)cc(F)cc2nc(S)[nH]c12 45753,c1(-c2cn(CC(=O)NCCCN3CCCCCC3)nn2)ncc(Cl)cc1F 45754,N1(C(C(CNC(c2cccc(CC)n2)=O)CC(C)C)=O)CC2(COCC(=O)N2)C1 45755,c1(C(C)NC(C(=O)NCc2c(Br)cn(CC)n2)=O)cccc2cnccc12 45756,c1(C(N2CCC(N3CCCC3=O)C2)=O)cc2cc(-c3ccccc3)sc2[nH]1 45757,n1(C(C)C)cc(Br)c(COC(=O)C(C)NC(c2ccccc2)=O)n1 45758,c1(CNC(N2CC(C)(CCc3ccccc3)C2)=O)ccc(Cl)cc1F 45759,c1(C(N(C2CCN(C(c3ccco3)=O)CC2)CC#C)=O)csc2c1CCCC2 45760,c1(SC)cc(C)ccc1C(=O)NCC(C(C)C)NC(=O)C(C)C(F)F 45761,N1(C(C2N(C(C)=O)CCOC2)=O)CCCN(Cc2ccc(Cl)o2)CC1C 45762,n1(CC)cc(-c2n[nH]cc2C(=O)NCC(C)N(C(=O)C(C)NS(C)(=O)=O)C)cn1 45763,C1(NC(c2cc(=O)cc[nH]2)=O)CN(C(c2ccnc(S)c2)=O)C2(CCCOC2)C1 45764,CN1N=C(C(=O)NC2CCN(C(c3cc(F)cs3)=O)CC2(C)C)CCC1=O 45765,C1(NC(c2c(C)nc(CC(C)C)s2)=O)CC12CCC(NC(c1csnn1)=O)CC2 45766,C1(F)(C(=O)NC2CCN(C(c3ncc(N(C)C)cn3)=O)CC2)CC2(CCC2)C1 45767,C=C=C(C)CC(=O)N(C1CN(C(c2cc(-c3ccn(C)c3)[nH]n2)=O)CC1O)C 45768,N1(C(=O)CCc2cc(Cl)sc2Cl)CCC2(CCCN2C(=O)C(F)F)C1 45769,N1(C(C(c2cn(C)nc2)=O)=O)CCc2ccccc2C1CCNC(C1(Cl)CC1)=O 45770,N1(C(CN(CCOC)C)=O)CCC2CCN(C(=O)COCCCOC)CC2C1 45771,CCCCC(O)C(=O)NC1(C2CCCN2C(c2cscc2SC)=O)CC1 45772,O=C(CN=c1cc[nH]cc1)NC1CC(CCNC(c2csc(C(F)(F)F)c2)=O)C1 45773,n1(CC(=O)NCC(CC)NC(=O)Cc2ccn(C)n2)c(-c2cccs2)nnc1S 45774,C(=O)(C(C)C(F)(F)C(F)F)NC1CC(CNC(COCCOCC#C)=O)C1 45775,Cc1ccc(C(N2CC(NC(c3coc(C(C)(C)C)n3)=O)CCC2C)=O)cc1F 45776,C1(N(C(C#CCNC(c2n(CC)ncc2C)=O)=O)C)CCCCC1(C)C 45777,CC1CCc2ccccc2N1Cc1ccc(Cl)cc1.C12CCCC(CC1)NC(=O)N2 45778,C1(OC)(CNC(C2CNC(=O)O2)=O)CCN(C(C2COCCC2C)=O)C1 45779,C(=O)(CS(=O)(=O)CC(=O)N1CC(NC(c2coc(SC)c2)=O)CC1C)OC 45780,Cc1ccnc(C(=O)NC2CC2CNC(c2ccc(Cn3cccc3)cc2)=O)c1 45781,c1(OC)cccc(NC(=O)CC(C)NC2(C)CC(C)=NO2)c1 45782,C1(NC(CCCCCC#C)=O)CCN(C(=O)CN2CCCS2(=O)=O)C12CCCC2 45783,c1(CCC)ccc(CC(N2CC=CC(NC(c3cnc[nH]3)=O)C2)=O)cc1 45784,C1(CNC(C=C(C)C)=O)(NC(C2CNC(=O)N2)=O)CCC(F)(F)CC1 45785,c1(CC(=O)NCC2(COC)CCCN2C(=O)C=C2CCC2)ccc(Cl)nc1C 45786,CCC(CC)C(F)C(=O)NCC1CN(C(C2CC3(CCC3=O)C2)=O)C1 45787,c1(OC)cc(C(N2CCN(C(C#N)C(C)C)CC2)=O)cc(C)n1 45788,N1(C(Cc2c(C(=O)NCOC)nccc2)=O)CCCC(NC(=O)C(O)CF)(CO)C1 45789,N1(C(C2CC(=C)C2)=O)CCSCC1C(N1CC(c2ncccn2)C1)=O 45790,N1(Cc2n(CC)ncn2)CCCC(O)(C(=O)OCC(=O)OC)C1 45791,S(=O)(=O)(c1ccc(Br)cc1NCc1ccccc1F)N(C)Cc1ccc(C)nc1 45792,CCC(CC(=O)NCC#CCNC(=O)C(C(C)C)c1cnc(C)s1)OC 45793,C1(NC(C(=O)N(C)Cc2ccc(OC)cc2)=O)CCc2cn(C(C)C)nc2C1 45794,c1(OC)cc(OC)cc(C(C)N(C)C(=O)Nc2ncc(F)cc2Br)c1 45795,C1(NC(c2cc(CC)n(C)n2)=O)CC2CC1N(C(=O)CCOC1CCOCC1)C2 45796,C(=O)(C(CCSC)NC(N)=O)NCC(CC=C)NC(=O)C=C(C1CC1)C1CC1 45797,C1(NC(c2c(C)nc(C(F)(F)F)s2)=O)CN(C(=O)C(O)C2CC2)C(C)(C)C1 45798,c1(C(N2CCCC(NC(c3ccc(C#C)cn3)=O)CC2)=O)cn2cc(C)sc2n1 45799,c1(CC)cccc(F)c1C(=O)NC1C2CC1N(C(=O)CC1(CO)CCCC1)C2 45800,c1(NC)cc(C(=O)NC2CCN(C(c3cccc(F)n3)=O)CC2CO)cc(Cl)n1 45801,c1(N2C(CCNC(c3ccc(NC)cc3F)=O)C(C)CC2)nc(Cl)nc2[nH]ccc12 45802,C1(NC(c2c(NC(c3cnc(OC)nc3)=O)cn(C)n2)=O)CCC(C2CC2)C1 45803,c1(C(=O)NC2(CNC(C=COCC)=O)CCOCC2)ccc2n[nH]cc2c1 45804,c1(CC(=O)NCCCNC(c2ccsc2Cl)=O)cc(Cl)ccc1O 45805,C(=O)(CCNC(=O)CC1CN(C(C2CC2(F)Cl)=O)C1)OC 45806,N1(C(C23CCC(OC)C2C3)=O)CCN(C)CC1CNC(=O)Cc1nocc1C(C)C 45807,N1(C(c2c(C)cc[nH]2)=O)CCCC2CCN(C(c3csc4c3CCCC4)=O)CC12 45808,C1(CCN(C)C(C2(C3CC3)CCCO2)=O)CCN(C(C2C(Cl)(Cl)C23CC3)=O)CC1 45809,C1(OC)CN(C(=O)NC2CCCN(C)C2)CCC1F 45810,Cc1ccc(C#N)cc1NC(C1CCN(C(C2CCCCC2F)=O)CC1(C)C)=O 45811,C(=O)(CC(C)CC(F)(F)F)NC1C(CNC(CC(CCC)C)=O)CCCC1 45812,Cc1ccc(NC(N2CCC(F)(c3ccc(Cl)cc3)CC2)=O)c(CN(C)C)c1 45813,c1(CC(=O)NC2CC(NCc3cccc(F)c3F)C2)ccc2c(c1)CCO2 45814,c1(C(N2C(CNC(c3cc(Br)ccn3)=O)COCC2)=O)c[nH]c2c(F)cccc12 45815,N1(C(CCCCC)=O)CCc2nc[nH]c2C12CCN(C(c1cccc(N)c1)=O)C2 45816,CC1(C)C2CCC(C(=O)NC34CCN(C(=O)Cc5ncc(Cl)s5)CC3C4)C1C2 45817,CC(C(=O)N(C)CCOCCCN(C)C(C1(C#N)CC1(C)C)=O)C(F)F 45818,Cc1ccc2[nH]cc(CN3CCC(O)C(C(N4CCC(OC5CC5)C4)=O)C3)c2c1 45819,C1(CNC(c2nsnc2O)=O)CN(C(C2(F)CCOC2)=O)CCC1(F)F 45820,c1(C(N2CCC(NC(=O)NC3(CCF)CCC3)C2)c2ccccc2)ccccc1 45821,c1(C=O)cc(F)cnc1O.N(CP(C)(C)=O)N(C)CCOCCC=O 45822,C1(N(C(CC(C)F)=O)C)CCCCC1N(C)C(c1cc(-c2ccccc2)cs1)=O 45823,c1(CC(=O)OC(CCC=C)C)cc(Cl)cc2ccccc12 45824,c1(OCC(=O)NCC(CNC(C2(NC(N)=O)CC2)=O)F)ccc(F)c(F)c1 45825,c1(OC)cc(C(F)CNCC2(C)CCCCCC2)ccc1Cl 45826,Cc1ncsc1C(=O)N(C)Cc1cocn1 45827,c1(C(=O)NCC2(NC(C3C(C)(C(F)F)C3)=O)CCC2)ccnc(-n2cccn2)c1 45828,C(C(=O)NNC(=O)C(C)(C)CCCCNC(=O)C(O)C1CC1)OCC 45829,C(=O)(CCCCN1CCCC1)NC(C1(O)CN(C(c2ccc(=O)oc2)=O)C1)C 45830,C(=O)(C#CC1CCCOC1)OCC(c1coc(-c2cccnc2)n1)=O 45831,C1(O)(CCNC(=O)CSC2CCS(=O)(=O)C2)CCCN(C(C2(O)COC2)=O)C1 45832,c1(C(=O)NC2C(SCC=O)C2)ccncc1.C1(CC(=O)NC)CCCCC1 45833,C1(CC(=O)NCCCN(C(c2cccc(COC)c2)=O)C)OCCCC1(C)C 45834,N1(C(CCOC)=O)C2CCC1(CNC(=O)Cn1cc(C3CCCC3)nn1)CC2 45835,C1(C(=O)NCCc2cc(C)nn2C)CCN(C(c2ccccn2)=O)CC1O 45836,N1(C(=O)CC2CCCCC2)CCCC(C2CN(C(c3cc(F)ccc3Cl)=O)C2)C1 45837,c1(CNC(C2(SC)CN(C(=O)CC3(C)OCCO3)C2)=O)cc(F)ccc1O 45838,N1(C(c2ccc(CC)s2)=O)CC(C2CN(C(C3CC(CC(F)(F)F)C3)=O)C2)C1 45839,C1(C2CC2)(CNC(C(C)OCCOC)=O)CCN(C(=O)CN=S(C)(C)=O)C1 45840,C1(NC(C2C(C(C)C)CN(C(=O)CC3COCCN3C)C2)=O)CC(=O)NC(=O)C1 45841,C12(C(=O)NC(CN(C(c3cscc3C)=O)CC)C)CCC(CC1)OC2 45842,C(=O)(C1CSc2ccccc21)NCc1c(OCC#C)nccc1 45843,N1(C(C2(C)CCN(Cc3ccc(F)cc3Cl)C2)=O)CC2OCCOC2C1 45844,N1(C(CNC(=O)OCC)=O)CCC(C(N2CCOC(COC)C2)=O)C(C)C1 45845,C(C(C)(C)CNC(=O)CC1CCC(C)O1)N(C(COCC(=O)NC)=O)CC 45846,C=C(C)CCCC(=O)N1CCC(C(C)(C)NC(=O)C2=CCC2)C1 45847,C12(C(=O)NCC(C)NC(=O)Cn3ncnn3)CC3CC(C(=O)N1)C2C3 45848,C=CCC(CNC(c1cc(C)on1)=O)C(=O)N(C)CC1CCCN1C 45849,Cc1nc([N+](=O)[O-])cn1CCC(=O)NC1CC(F)CN(C(c2ncn(C)n2)=O)C1 45850,C=CCC(CC)C(=O)N1CCN(C(=O)CNC(=O)OCC)CC1c1ccccn1 45851,N1(C(c2c(O)ccc(C)c2)=O)CCC(C(=O)NCC(c2cnc[nH]2)C)CC1(C)C 45852,C1(N(C(c2c(CC)ncs2)=O)C)CCN(C(C2(c3oncc3C)CC2)=O)CC1 45853,CCC(CSC)(CC)C(=O)N1CCC(C(=O)NCCn2cnc(CO)c2)O1 45854,C=C(Cl)CC(C(=O)NCc1cc(C)ccc1OC)NC(=O)CCCOC 45855,c1(CNN(C(c2ccc(C(=O)NCC)cc2)=O)CC)cccc(O)c1CC 45856,c1(C(=O)OC)nc(N2CC(OC)C(F)C2)cc(Cl)n1 45857,Cc1ccc(C)c(CCCC(N2CCC(CNC(=O)C=CC3CC3)C(C)C2)=O)c1 45858,C1(C(=O)NC2(C)CN(C(C3(c4ccccc4F)CC3)=O)C2)CCC2(CC1)CC(=O)C2 45859,c1(C(N(CCNC(c2c(CC)n(CC)nc2)=O)C(C)C)=O)cccc(C)c1F 45860,C(=O)(C(F)CC(C)(C)C)N(CCOC)CCNC(=O)C(CC1CC1)NC(C)C 45861,CC(CCNC(=O)Cc1cnc[nH]1)CCNC(C1CNC(=O)N1)=O 45862,CC1CC(CNC(=O)CC2(C)CC2(Cl)Cl)CN1C(c1n[nH]c(=N)s1)=O 45863,c1(CNC(CCC2CCN(C(C(CC)OC)=O)C2)=O)cnc(C)n1CC 45864,N1(C(C2(CCC)CCC2)=O)CC2CCCC2(NC(=O)C=C(Cl)Cl)C1 45865,N1(C(C(N2CCCC(CC(=O)OCC)C2)=O)=O)CCCNC(=O)C1CC(C)C 45866,C1(n2cc(C(N)=O)c(O)nc2=O)CCN(C(=NCCCCl)NCCC2CC2)C1 45867,c1(COC)ccc(C(=O)NCC(C2CCC2)NC(c2oncc2C)=O)cc1 45868,C1(NC(c2n(CC)ccc2)=O)CC2(C1)CC(NC(=O)CC13CC(C1)C3)C2 45869,N#Cc1c(Cl)nsc1NC1CCN(CCNC(=O)CNc2ccccc2)C1 45870,C=CC1(O)CCN(C(=O)C(CCOCC)NC(C2CCN(C)C2)=O)C1 45871,c1(C(N(C(c2n(CC)ccn2)C(=O)O)C)=O)cc(C)cc(O)c1 45872,N1(C(C(C)NC(CC)=O)=O)CCOC(CN(C(=O)CC2CN(C)C2)C)C1 45873,Cc1oc(C2CC2)nc1N(S(=O)(=O)CC1CC1F)C 45874,C(C(=O)N(C(C)CC)C)(C(C)CC)NC(c1cc(CC)on1)=O 45875,c1(C(N2CCC(CNC(C3CC34CCC4)=O)C23CC3)=O)cc2c([nH]1)CCCC2=O 45876,C#Cc1ccc(CNc2cccnc2C(=O)NC2(c3ccccc3F)CCC2)s1 45877,N1(C(c2cc(C)cc(O)c2)=O)CCC(C2(NC(c3cnnn3C)=O)CC2)CC1 45878,Cc1cncc(C(N2CCC(O)(C(C)NC(=O)Cn3cncn3)C2)=O)c1 45879,C1(N(C(CCN(CCCCC)C)=O)C)CCC(NC(=O)C(O)CC)CC1 45880,c1(CNC(C(N(C(CN(CCC)C)=O)C)C2CC2)=O)cnc(C)cn1 45881,c1(C(N(CC(C)NC(=O)CC(C)F)C)=O)ccccc1-c1cncnc1 45882,c1(C(N2CC(CC(C)NC(c3ccnc(F)c3)=O)C2)=O)cc2c(nn1)CCCC2 45883,c1(C(=O)NCC2CC=C(C)CC2)cc(C)ccc1F 45884,c1(NC(=O)C(F)CC2CNC2)cnccc1NC=O 45885,C1(CNC(CCSCCCC)=O)CCCN1C(c1c[nH]nc1-c1cnn(C)c1)=O 45886,N12CCC(CC1)C2.c1(C(=O)NC(c2nc(C)oc2)C)cnc(CN(C)C)nc1 45887,c1(NCC2OCCN(C(=O)C=Cc3ccccn3)C2)ncnc2c(Cl)cc(Cl)cc12 45888,N(C(=NCc1ccccc1)N1CCC(SC)C1)CC.c12ccccc1C(=O)NC2 45889,CC#CCCCCN=c1nc(N2CCCC(OC)CC2)c2[nH]ccc2[nH]1 45890,c1(C(N(C2CCCN(C(C3(Cl)CCCCC3)=O)CC2)CC)=O)ccc(C)c(O)n1 45891,C(=O)(C(C(C)(C)C)c1cc[nH]n1)N(CCNC(C(C(C)O)N(C)C)=O)C 45892,N1(C(c2n(C(CC)CC)nc(C)c2)=O)CCCC(NC(c2coc(C)n2)=O)CC1 45893,C1(CC(=O)N(C(C)C(N2CCCCC2C2CCC2)=O)CCC)CCN(C)CC1 45894,C#CCC(C)(C(=O)NC1(C)CCSC1)NC(=O)CC(C)(O)COC 45895,C1(NC(c2occ(C)c2)=O)(CO)CCN(C(c2ccc(CC(C)(C)C)cc2)=O)C1 45896,N1(C(C=C2CCN(C(C3(COC)CC3)=O)CC2)=O)C2CCC1CN(C)CC2 45897,c1(C(=O)NC(CC)CNC(c2sc(C)cc2C)=O)cn2c(n1)CCC(C)C2 45898,C(=O)(C#CC1CCOCC1)NC(C)CN(C)C(C1(C)CCNC(=O)C1)=O 45899,c1(C(=O)NCC2C(NC(=O)Cc3cscn3)CC2)cc2ncccc2s1 45900,N1(C(C(C)NC(N)=O)=O)CC2(CC(NC(=O)C(C)(C)NS(C)(=O)=O)C2)C1 45901,CCCCC(CC)CC(=O)NC(C(C)N=c1[nH]ncs1)c1ccccc1 45902,C1(F)(CNC(C(C)=C(C)C)=O)CCCN(C(C2(C)CC(C)C2)=O)C1 45903,c1(C(N2C(CNC(=O)C=CC3CCCCC3)CC3CC32)=O)cc(=O)cc(Cl)[nH]1 45904,C(c1ccccc1)=CCC(N1CCC(CN(C(C(COCC)C)=O)C)C1)=O 45905,N1(C(CCN2C(C)CCCC2)=O)Cc2c(ccc(F)c2Br)CC1C 45906,C(=O)(CCC(C(C)C)NC(=O)C(C)c1ccco1)N1CCCC(OC)C1CO 45907,N1(C(C)C)CC(C(=O)OCc2ccccc2C(F)(F)F)CC1=O.C1(C)C(=O)O1 45908,Cn1ncc(C(c2nnnn2CCONC)NC2CC3CCCC3C2)c1S(N)(=O)=O 45909,C(CCCCC(=O)NCC1CN(C)CCN1C(=O)C(C)C(=O)OC)=CC 45910,c1(C(N2CCC(c3ncc(C)cn3)CC2)C(=O)NCC2CC2)ccc(Cl)c(F)c1 45911,Cc1cccn2nc(C(=O)NC3CN(C(C4(C#N)CCCCC4)=O)CC3C)cc12 45912,CC1(C)CC(NC(=O)CC#N)CN1C(=O)COCc1cccc(Cl)c1 45913,C1(C(=O)NCCc2nc(C)[nH]n2)CCCC(NC(=O)C(F)CC2CCOC2)CC1 45914,N1(C(C2CC(C(C)(C)C)C2)=O)CCC(C(F)F)(CNC(=O)CN2CC=CC2)C1 45915,CC1CC(NC(=O)Cc2nc(C3CC3)cs2)CN1C(=O)C(c1ccc(F)cc1)C 45916,N1(C(c2c(=N)cc[nH]c2)=O)CCCC2CN(C(=O)C=CC3CCCC3)CCC12 45917,C1(C)(C(N(CCC(C)(C)C)C)=O)CCCN1C(=O)CCc1ncnn1C 45918,C1(C(=O)NC2C(CNC(C3(OC)CCCC3)=O)CCC2)CC(=O)N(C2CC2)C1 45919,c1(CCNC(CCc2cc(C)on2)=O)c(C)n[nH]c1C 45920,N1(C(c2cn(CC=C)nc2)=O)CCN(C(c2cn[nH]c2)=O)C(C2CC2)C1 45921,N1(CCCCCNC)CCN(CCOCCOCCC2CC2)CC1 45922,Cc1ccc2nc(C)c(C(=O)N(C3CCN(C(C4CC(Cl)(Cl)C4)=O)C3)C)cc2c1 45923,C1(C(=O)NC2CN(C(c3c(O)ccc(CC)c3)=O)CC2O)CCc2cnnn2C1 45924,c1(N2CCN(C(c3n(C)nc(CC)c3Br)=O)CC2)ccc(C(C)=O)cc1[N+](=O)[O-] 45925,CCCCC(C)CCC(=O)N1CCC=C(C(=O)NCc2cnccc2Cl)C1 45926,C1(CNC(COCC(=O)NC)=O)CC(C)CCN1C(=O)C(=Cc1ccncc1)C 45927,c1(C(CC(=O)OC)NC(c2c[nH]cc2C)=O)cccc2ccccc12 45928,C1(NC(c2c(=O)ccn(C)c2)=O)CCC2(CC1)CNC2 45929,N1(C(CCN(C2CCCCC2)C)=O)CC2C(NC(=O)CCc3ccn(C)c3)C2C1 45930,c1(CN2CC(O)(CNC(c3ccccc3F)=O)C2)ccnc(O)c1Br 45931,C1(NC(c2c(OC)nsc2)=O)CCC12CN(C(=O)CCc1csc(=N)[nH]1)C2 45932,C1(N(C(c2nc(OC)oc2)=O)C)CCC(NC(=O)CCc2ncc(C)[nH]2)CC1 45933,N1(C(c2cncc(C(C)(F)F)c2)C(=O)NCCOC)CCN(C=O)CC1 45934,c1(CC(=O)ON2CCC(CC(=O)NC3CC3O)CC2)ccc2c(c1)CC2 45935,N1(CC)CCN(CCC(N2CCC(C(F)CNC(=O)CCSC)CC2)=O)CC1 45936,N1(C(C2(CCCC)CCC2)=O)CCC2(CCCN(C(=O)CNC(=O)OC)C2)C1 45937,C(=O)(C(C(C)CC1CCC1)N1CC=C(CO)CC1)N(CCCCCC)CC 45938,Cc1cc(C(=O)NCCOc2ccccc2C(N)=O)c(F)cc1Cl 45939,C1(CN(C(=O)C(c2nc(C)cs2)C)CC)CCN(C(C2(C)CC=CCO2)=O)CC1 45940,C1(NC(C(N2CCCCC2)C)=O)(CO)CCCN(C(C2(O)CCSC2)=O)C1 45941,Cc1ccc(F)c(C(=O)NC2CC3(C2)CC3NC(C2CC(C#N)C2)=O)c1Br 45942,C1(C(=O)NCC(O)CNC(C2CCC(c3ccccc3)C2)=O)(CC)CCCC1 45943,N1(C(C)=O)CCC2(CCOCC2)C(NC(c2coc3c2C(=O)NCCC3)=O)C1 45944,c12ccccc1CNC(=O)C1CCCC1NC2.C(=O)(C(C)(C)OC(C)C)NC 45945,C1(C(N2CC(CC(C)NC(C3=C(C)OCC3)=O)C2)=O)CCc2nc(O)[nH]c2C1 45946,CCCC(C)CCCC(=O)N1CC2(NC(C3CC3CCOC)=O)CCC1CC2 45947,c1(C(=O)NC2(CN(C)C(c3ccc[nH]3)=O)CC2)ccnc(Cl)c1N 45948,CC1CCC(C(=O)NC2CCCC(CNC(C3(N4CCCC4)CCC3)=O)C2)CC1 45949,C1(NC(CCCSC)=O)COC2(C1)CN(C(c1ncnc(O)c1F)=O)C2 45950,c1(C(N2CCC3CN(C(C4C(C=C)OCC4)=O)CC32)=O)cnc2ccccc2n1 45951,c1(OC)cc([N+](=O)[O-])ccc1CN=C(NC1CC1C)NC1CCCCC1 45952,C(=O)(C1=CCC(NC(=O)C(n2cc(-c3sc(C)nc3C)nn2)C)C1)OC 45953,CCC(Cc1ccccc1)C(=O)NCCN(C(=O)Cc1nncn1C(C)C)CC 45954,N1(C(C2(C)CC2(F)Cl)=O)C(CNC(C2CCCO2)=O)CC2COCC12 45955,c1(-c2cn(CCOC)nc2)ccc2ccc(C(=O)NCCC(C)(C)C)nc2c1 45956,CC(C)CC(C)CC(=O)NCCC(C(C)C)NC(c1cnc(C2CC2)nc1O)=O 45957,CC(CN=c1[nH]c(=NC(C)c2nc(O)n[nH]2)[nH]c2cc[nH]c12)n1ccnn1 45958,N1(C(C2C(=O)NCC2)=O)CC(CO)C2(C1)CN(C(C1CCn3ncnc3C1)=O)C2 45959,C(=O)(C(C)CC(F)(F)F)NCC1CC(OC)CN1C(c1c[nH]cc1C)=O 45960,C(=O)(CS(=O)(=O)CC(=O)OC)N1C(CNC(C(CC)=CC)=O)C(C2CC2)CC1 45961,c1(C(=O)NC(CCCCNC(C)=O)C)cnc2c(C)cnn2c1 45962,C1(Nc2coc(C3CC3)c2)COCCC1CO.CC1(C)CNC(=O)CO1 45963,C1(n2cccn2)(C(=O)NCCC=C=C)CCN(C(=O)C(C)CC)CC1 45964,c1(OC(Cc2ccc(C(C)=O)s2)=O)cccc2[nH]ncc12 45965,c1(-c2cn(C3CN(C(c4c(C)coc4)=O)C3)nn2)cccc(CO)n1 45966,N1(C(C2CCCOC2)=O)CC2(CCCCN2C(c2ccnn2CC(F)(F)F)=O)C1 45967,c1(NCc2c(C)cn(C)n2)[nH]c(=NCC2CCCO2)nc2scnc12 45968,C1(C(=O)NCC(=C)CCNC(c2cc(Cl)ncc2O)=O)CCC2C(C1)C2(F)F 45969,c1(C(N2C(C)CN(C(=O)C(C)(O)C3CCC3)CCC2)=O)ccc(S(N)(=O)=O)nc1 45970,N(C(=NCCC(C)(C)S(C)(=O)=O)NCC(F)F)CC1CC(C(OC)OC)C1 45971,N1(C(C2(OC)CCSC2)=O)CC(CNC(=O)CCn2cncn2)C2(CCC2)C1 45972,c1(OC(C)C(=O)N(CC(C)NC(=O)CC2CCCCC2)C)cccc(Br)c1 45973,CC1(C)CC(CC(=O)NC(CO)C2CCC2)CN1C(=O)CC1CC(=O)C1 45974,c1(SCCNC(N(CCCC)C2CC2)=O)ccc(Cl)c(Cl)c1OC 45975,c1(C2CCN(C(C(=O)Nc3ccncc3F)=O)C2)ccc2ccccc2c1 45976,N1(C(CSCC)=O)CCSC(C(=O)NCCc2nc[nH]n2)C1 45977,C1(C2(CC(=O)NC(C)CC3CN(C(=O)C=Cc4nccs4)C3)CC2)CCN(C)C1=O 45978,C1(NC(c2ncn(C(C)(C)C)n2)=O)CCN(C(C2(C)CC2(Cl)Cl)=O)CC1(C)C 45979,c1(C(=O)Nc2ccc3c(c2)CCCS3)cc2n(n1)CCCC2=O 45980,C1(C(=O)NCC(C2CC2)NC(=O)Cc2ccc(Cl)nc2)CCOC(=O)CC1 45981,C1(CC(=O)NCCCNC(c2cncc(CSC)n2)=O)(OC)CCCCC1 45982,Cn1cnc2cc(C(=O)NCCC3CCCN(c4nnc(CO)s4)CC3)cnc12 45983,C1(CNC(C(C)(C)CC(F)F)=O)CN(C(=O)C(O)C2CCC2)C2(CCOCC2)C1 45984,c12ccc3c(c1)C(NC1=NCCN21)CCCO3.CO 45985,CN1CC(O)CC1NC(=O)C=CCN1CCCC1.C12(CC1)C(=O)N2 45986,C1(C(=O)Nc2c(C)n(CC(F)(F)F)nc2)CNC2(CCOC2)C1 45987,N1(C(=O)C(O)c2ccsc2)CCC(F)(C(=O)NCc2cn(C3CC3)cn2)CC1 45988,C1(CNC(c2ccc(O)nc2)=O)CC2(CCN(C(C3(CF)CC3)=O)CC2)CO1 45989,Cn1cnc2sc(C(=O)NC(C3CCN(C(C4(O)CCCCC4)=O)C3)(C)C)cc12 45990,c1(C(=O)NCC2N(C(Cc3c(O)nc(=N)[nH]c3)=O)CC2)cc2ccc(Cl)nc2s1 45991,N1(C(C(=O)NC2COC2)c2nccs2)CCOCC1c1cccc(F)c1 45992,C1(C2CN(C(c3cc(F)cs3)=O)C2)(NC(C(C)CCc2cccc(F)c2)=O)CC1 45993,C1(CC=C)(NC(c2ncoc2C2CCC2)=O)CN(C(=O)Cc2ccnn2C)C1 45994,C(=O)(C1CCCc2n[nH]cc21)NCC(C)NC(C1CC(C)(c2ccccc2)C1)=O 45995,CC1CCN(C(=O)CCCc2ccncc2)CC1CNC(c1ccc[n+]([O-])c1)=O 45996,C(=O)(C1=C(C)N(C)c2nnnn2C1)NCC(C)(CC)NC(CCCC=C)=O 45997,Cc1ccccc1N1CC(C(=O)N(CCCNC(=O)CC(C)F)CCO)CC1=O 45998,C=CC1(CC(N2CCC(NC(C3CCS(=O)(=O)CC3)=O)C(O)C2)=O)CCOCC1 45999,CC1(C)CCN(C(c2cc(C3CC3)on2)=O)C1CNC(=O)CCc1cnco1 46000,c1(C(C(=O)N(CCNC(C(COC)COC)=O)C)C)ccc(S(C)(=O)=O)cc1 46001,CCC(=O)CCC(=O)N1CC(C)(CCC(N2CCC(N(C)C)(CC)C2)=O)C1 46002,CC(C)CC(O)CC(=O)NCCC1(O)CC2CCC1CC2 46003,O=C1CCN(Cc2ncc(-c3cccc(-c4cncn4C(F)(F)F)c3)o2)CCN1 46004,C(=O)(CCC(=O)NCC1CC(O)CN1C(c1cc(Cl)cn1CC)=O)NCC 46005,c1(C(=O)NCC2(NC(C3CC3F)=O)CCOC2)cc(Cl)cc(C(F)(F)F)n1 46006,c1(C(=O)NC2CC(CNC(C(CC)(C)CO)=O)C2)cc(F)c(F)cc1Br 46007,CC1(c2ccc(NC(=O)CCc3cccc(NC(N)=O)c3)cc2)NC(=O)NC1=O 46008,c1(C(=O)OC)ccccc1CCC(=O)NCC1(F)CN(C(=O)Cc2ccon2)C1 46009,c1(C(=O)NCC2CCC(NC(C(CC(C)C)O)=O)C2)cc(C#N)ccc1F 46010,C(CC(C(C)(C)C)NC(=O)CC1(C)CCCCC1)N(C(=O)CC1(CO)CC1)C 46011,C(CCC(C)(C)C(=O)NCC(C)CCCO)NC(c1c(C)ncnc1)=O 46012,CCCS(=O)(=O)C(C)C(=O)NC1CN(C(=O)CCCCCN(C)C)C2(CCC2)C1 46013,C1(NC(c2c(C)occ2)=O)CN(C(=O)CCCCCNC(N)=O)C2(CCC2)C1 46014,N1(C(C2CN(Cc3cccc(C)c3)C2)=O)CCC2(CCC2)C(NC(=O)O)C1.ON 46015,c1(C(N(C2CCCC(NC(COCCCC#C)=O)C2)C)=O)ccc2nn[nH]c2c1 46016,c1(C(=O)NCC2(O)CN(C(c3ccc(C4CCCO4)s3)=O)C2)ccnc(Cl)c1Cl 46017,C1(CN(C(C2CCN(C(=O)Cc3cncc(C)c3)C2)=O)CC)CCCC2(CC2)C1 46018,N1(C(C(C(C)C)NC(C)=O)=O)CCC12CN(C(=O)C(C)NC(=O)C1CC1)C2 46019,C1(NC(c2cc3sccc3[nH]2)=O)CC2(NC(C3CC4(C3)CC4F)=O)COC1C2 46020,C12(C(=O)NCC(CC)O)CC(C)(CN1C(c1cc(COC)no1)=O)C2 46021,C(=O)(C1CCc2nccn21)N(CC(NOCC1(O)CCN(C)CC1)=O)C 46022,C#Cc1ccc(C(=O)NCCOC2CN(C(=O)COC3CCOC3)C2)cc1F 46023,C1(NC(CS(CC)=O)=O)CCC2(CCN(C(c3ccnn3C(C)(C)C)=O)CC2)C1 46024,c1(OC)ccc(CN(C(=O)C(C)NC2C3CCOCC23)C)c(OC)c1 46025,N1(C(C2CCC(F)(F)CC2)=O)CC2(CCN(C(C3(C)CC(F)C3)=O)CC2)C1.CC(C)(C)NC 46026,CC(C(=O)NO)NC(C1(NC(=O)CC#N)CC1(C)C)=O 46027,N1(C(C2OCCN(CC)C2)=O)C2CCC1CN(C(C1CCC3(CCC3)C1)=O)C2 46028,C1(CNC(CCCCSC)=O)CCC2(CN(C(c3cccc(C)c3C#N)=O)C2)O1 46029,C1(COC)C=CCCN1C(=O)CCC1(C)CN(C(=O)CCc2ccco2)C1 46030,C1(C(=O)NCC(C)(CO)NC(c2ccc(C)cc2)=O)CCCC2(CCC2)O1 46031,N1(C(C(CC=C)(C)C)=O)CCOC2(C1)CN(C(=O)C(O)CCSC)C2 46032,CC(=O)CCC(=O)OCC1CCCCC1F 46033,c1(CNC(CCC2N(C(CN(C)C(=O)C3CC3)=O)CCC2)=O)cccc(O)n1 46034,C1(C(N(CCCOCCNC(=O)C(CO)N(C)C)C)=O)CC2(C1)CC2(F)F 46035,c1(C(N2CCC(C)(NC(CC=C)=O)C2)=O)cccc2sc(C(F)(F)F)nc12 46036,C(CCCCC(=O)NC(C1(O)CCN(C(c2cc(CO)n(C)n2)=O)C1)C)OCC 46037,C(=O)(C(C)(C)C(O)C(C)C)N1CC2C(C(NOCCOC)=O)C2C1 46038,C1(NC(C2C(C)(C)C2)=O)CCC2(CCN(C(c3ccc4cc[nH]c4n3)=O)C2)C1 46039,C1(C(N2CCN(C(CC(=O)NCC#C)=O)C(CO)C2)=O)CC2OC(C)(C)OC2C1 46040,O=C1CC(C(=O)NC2CCC2C(N2CCn3nccc32)=O)=NN1 46041,C1(NC(C(C)c2ccsn2)=O)CCCN(C(=O)Cc2cccc(Br)c2)C1 46042,Cc1cc(CNCC2CCCCN2C(C2(O)CCCCC2)=O)n(C)n1 46043,N1(C(C2(C)C(C)C2)=O)CCC(C2CC2)(CNC(c2ccc3[nH]ccc3n2)=O)C1 46044,C(=O)(C(F)CC(CC)CC)NC12CCN(CC1)CC2.C12(CCC=C)CN(C1)C2=O 46045,N1(C(c2c(CC)[nH]cc2)=O)CCC2CC2(C(=O)NCc2n[nH]c3c2CCC3)CC1 46046,c1(OC)cc(Br)ccc1C(CO)NC(=O)NCc1oc(C)cc1C 46047,NC(=O)CCC(C(=O)NC1CC(C(F)F)C1)n1cc(Cn2cccn2)nn1 46048,c1(C(N2CC(CNC(C3C(OCC)C3)=O)(OC)C2)=O)c(O)nnc2c1COCC2 46049,c1(C2(C(=O)NC(C3CCCCO3)C#C)CCCC2)ccccc1Cl 46050,C1(NC(C2CCC(=C)CC2)=O)C(C)CCN(C(c2ccc(Cl)c(F)c2F)=O)C1C 46051,C(=O)(C1=CCC(C)(C)CC1)NC(CCNC(Cc1c(O)ccc(C)c1)=O)C 46052,c1(C(=O)NCC2C(C(=O)Nc3cnc(OC)nc3)C2)coc2c1COC2 46053,C(=O)(CCCC(F)(F)CO)NC1CC2CN(C(Cc3cncc(C#N)c3)=O)C1C2 46054,c1(OC(C)C)ccc(CC(=O)N(C2CCC(CNC(=O)CC(C)C)CC2)C)cc1 46055,c1(C(C(=O)NCC(=C)C)N(CCCN(C)C)CCC)ccc(-c2ccco2)cc1 46056,c1(CCOC)nc(=NC2CCCC(NC(C3(O)CCSCC3)=O)C2)s[nH]1 46057,Cc1cc([N+](=O)[O-])c(C)cc1C(N1CC2CN(C(c3ncccc3F)=O)C2C1)=O 46058,C(C(CNC(=O)C(C)Cn1ccnc1)S(C)(=O)=O)NC(C(COC)C)=O 46059,N1(C(c2c(C)[nH]cc2)=O)C(C(=O)N(C(C)C)Cc2ccco2)CCC1C 46060,O=C(C1CCCn2cnnc21)NC1CC(O)CN(C(C2C3(CC3)C23CC3)=O)C1 46061,c1(N2CC(C)=C(C)C2)nc(N(C)Cc2nc(C3CC3)n[nH]2)nc2cc[nH]c12 46062,C1(NC(CNC(C(CC)C)=O)=O)CN(C(c2ccn(C)c2)=O)C2(CCCCC2)C1 46063,c1(C(=O)NCC#CCNC(CC2CCCC(C)C2)=O)c(F)cc(Cl)c(F)c1F 46064,Cc1ncc(C(=O)N(CC(C)N(C(=O)CN2CC3CCC2C3)C)C)cc1N 46065,Cc1c(NC2CCN(CC(C)C)C2)ncnc1N(C)CCOC1CC1 46066,c1(N2CCC(N(C)C(c3ccc(O)nn3)=O)C2)nnccc1C#N 46067,C1(C(=O)NCCC(CNC(CN(C2CC2)CC)=O)O)CCCC(C)(C)O1 46068,c1(OC)ccc(-n2nc(C3CC3)nc2N(C)CC2(CS(C)(=O)=O)CC2)cc1Cl 46069,C(=O)(CC(C)(O)C(F)(F)F)N1C(C(C)NC(c2ccc(CC)cc2C)=O)CCC1 46070,c1(-n2c(CC(C3CCOCC3)F)nc(-c3cn(C)nc3)n2)c(C)cc(C)cc1C 46071,c1(C(=O)NC(c2c(NCc3nccc(C)c3)cccn2)=O)ccc2nc[nH]c2c1 46072,c1(C(=O)NCC2CC(O)(CNC(C(OC)OC)=O)C2)nc(C)ccc1F 46073,C(=O)(C1CCCn2nccc21)N(CC(C)(C)C)C(CNC(C=CCCC)=O)C 46074,c1(OC2CN(C(C3C(C)CCC3)=O)C2)cnccc1C(=O)Nc1cc(=O)cc[nH]1 46075,c1(C(=O)NC2CC(C)(CNC(=O)Cn3cnccc3=O)C2)ccc(F)cc1N 46076,n1(CC(=O)N(C(CNC(Cn2cc(C(C)=O)nn2)=O)C)C)ncccc1=O 46077,C#Cc1cnn(C)c1C(N1CCC(F)(CNC(c2cncn2C2CC2)=O)C1)=O 46078,CC1CC(NC(C2CC(=O)NC(=O)C2)=O)CCN1C(=O)CCCn1cccc1 46079,c1(C(=O)NCC(CC)(CC)Nc2cncc(C#N)n2)ccc2nc[nH]c2n1 46080,c1(CC(C)C(=O)NCCCNC(=O)C(C)(O)c2ccccn2)ccc(F)cc1F 46081,C1(=O)CCC(C)N1.N1(N(C(C(=O)N(C(CCOCC)C)C)=O)C)CCCC(C)C1 46082,C1(NC(c2ccc(OC)nc2)=O)CCCN(C(=O)CCn2cccc2)CC1F 46083,c1(C(CC)C(=O)N(C(C)CN(C(=O)COCC(=O)NC)C)C)c(C)noc1C 46084,C12(OC(C3C(C)CC(C)O3)=O)CC3CC(CC(NC(c4cccs4)=O)(C3)C1)C2 46085,C1(C(=O)NC2C(N(C)C)CC2)C=CCN(C(=O)C2=CCCC2)C1 46086,c1(C(=O)NCC2CCN(C(C3OCCN(C)C3)=O)C2)ccc2c(c1)CCCC2 46087,C1(CN(C(CC(C)O)=O)C)CCCCN(C(c2cccnn2)=O)C1 46088,N1(C(c2nc(C)oc2)=O)CCC(NC(=O)C(C2CCCN(C)C2)(C)C)C1C(C)C 46089,c1(C(=O)NC(CCC=C)C(=O)NCC2(CCO)CCC2)ccc2[nH]nc(Cl)c2c1 46090,c1(C(=O)NC2CCN(c3nnc(CC)c(CC)n3)C2)cc2c(=O)[nH]ccn2n1 46091,O=C1COc2ccccc2CN1N1CCCCCNS(=O)(=O)CC1(C)C 46092,C1(Cn2cc(CCC(C)O)nn2)(CNC(C2CCC(=O)NC2)=O)CC12CCC2 46093,CCCC(C(=O)N1CCN(C(C23CCCN(CC2)C3)=O)CC1C(C)C)C(C)C 46094,N1(C(CC2(C=C)CC2)=O)CC(C)CCC1CNC(=O)C(C)(CC)CC 46095,c1(C(=O)NC(c2cnn(C)c2)C(=O)OC)ccc(-c2ccc(F)cc2F)cc1C 46096,CC1(C)CN(C(=O)CC2CC2(C)C)C1C1CCN(C(=O)COCCCF)CC1 46097,C(=O)(CS(=O)(=O)CC1CCCN1)C(c1cn(CCS(CC)=O)nn1)(C)C 46098,N1(C(CCCOC)=O)CC2(C1)OC1(COC)CC2(NC(=O)C(C)CC(C)(F)F)C1 46099,CC(CCCNC(c1csc(F)c1)=O)NC(=O)C(c1ccccc1)F 46100,NC(Cc1ccccn1)C(=O)N1CCCC1CCc1ccncc1 46101,C1(CC)CCCN(C(C2CN(C(C)C)C2)=O)C1C(=O)NC1CN(C)CCC1O 46102,C1(SC)CCCCN(C(C2CCN(C(=O)c3cc([N+](=O)[O-])n[nH]3)O2)=O)C1 46103,Cc1cccc(C(C)N(C)Cc2cc[nH]c2)c1C 46104,C=CCCC(C(=O)N1CCC(C)(CCC)C1)NC(=O)CCC(C)OC 46105,c1(C(N2CCCC(O)(CNC(c3c[nH]c(=N)o3)=O)C2)=O)cc(=O)n2nccc2[nH]1 46106,C1(NC(CN(CCC)C(C2CN3CCN2CC3)=O)=O)CCCCC1C#N 46107,C1(CCNC(c2c(CC)c[nH]n2)=O)CCN(C(=O)C=C(C)C(C)(C)C)C(C)C1 46108,N1(C(c2ccc(CSC)o2)=O)CCC(C)C(N(C(=O)Cc2ncoc2C)C)C1 46109,CC1(C)OC2(C(=O)NCC(C3CCCO3)O)CC1C2 46110,C(CC(C(=O)NC1CCCN(C(c2csc(C(F)F)n2)=O)C1)OC)OC 46111,CC1(C)OC(=O)NC1C(=O)NCc1cccc(NC(=O)CCC(N)=O)c1 46112,c12c(cnn1C)CNC2=O.C1(C(C)C)CN(C(=O)CCc2nncs2)C1C(C)C 46113,C=C(C)CC1C(=O)NC(CCC)C(=O)N2CC3CC(C2)(C3)C(=O)N1.C(N)(=O)NC 46114,N1(C(CCC2CCC(=O)C2)=O)CCC2(CC2NC(=O)C2=C(Cl)CCC2)C1 46115,C1(C(=O)NC(C)CN(c2nc(C(C)(C)C)ns2)C)CCc2c[nH]nc2C1 46116,C1(=O)C(CCC2CCC2)N1.c1(C(C)NC(C(OC)OC)=O)nc(C)cs1 46117,C1(C)(C(=O)NCCc2cn(C)nc2)CCCN1C(=O)C(N)=O 46118,C=C(Cl)CC(C(=O)NC)NC(=O)C(N)Cc1cn(-c2ccccc2)nn1 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46153,Cc1ccc(OC(C)C(N2CC(CNC(C3(C#N)CCCC3)=O)C(C)C2)=O)cc1 46154,c1(N2CCC(C(=O)NCC(c3cc(C)sc3)(F)F)C2)ncnc2cnn(C)c12 46155,CC(C)CC(C)CC(=O)NCc1cc(C(=O)Nc2cncc(F)c2)ccn1 46156,c1(OC)ccccc1S(=O)(=O)NC1CN(c2cc(C)nc(C)n2)C1 46157,N1(C(C(N2CCS(=N)(=O)CC2)=O)=O)CCc2c(C(=O)NC3CC3)cccc2C1 46158,C1(C)(CNC(C(C=C=C)C)=O)CN(C(c2nc(O)nc(O)c2OC)=O)C(C)(C)C1 46159,CC(C)(C(=O)NCC1CC2CC2N1C(=O)CCP(C)(C)=O)S(C)(=O)=O 46160,CCCCCC(F)C(=O)NC(Cc1cc[nH]n1)C(=O)NC1CC(C)(C)OC1(C)C 46161,c1(N(C)Cc2c(OC)cccc2)cc[nH]c(=NCCCc2cccs2)n1 46162,Cc1ccc(C2CC2c2nc(-c3ccc(N)cc3)nn2-c2cnnn2C)cc1 46163,N1(C(CN2C(C)CC2)=O)CCC(O)(CNC(c2cnc(C3OCCO3)s2)=O)CC1 46164,C(=O)(CS(=O)C(F)(F)F)NCC1(C)CCCN1C(C12CCC(F)(CC1)C2)=O 46165,c1(CNC(c2nc(C)c(C)s2)=O)nc(CNC(=O)CC(C)C(C)C)cc(O)n1 46166,CCCC(C)C(=O)N1CC(CCNC(C2CC2Cc2conc2C(C)(C)C)=O)C1 46167,N(C1COCc2ccccc21)C(=O)C(c1cccnc1)Sc1ccc(Cl)cc1 46168,C1(C(=O)NCCC(C)(C)NC(C2C(C(=O)OC)CCO2)=O)CCCCC1(F)F 46169,c1(OC)cc(C(C(=O)Nc2nnn(C)n2)N(C)CCOC(F)F)cc2c1OCO2 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46188,C(=O)(C1OC(=O)c2ccccc21)NCCN(C(=O)C=Cc1cnn(C)c1)C(C)C 46189,N1(C(COC)=O)CC23CCCCC2(C1)CN(C(C1(C#N)CCOC1)=O)C3 46190,C1(C(=O)NC(C(C)C)CNC(C2COC3(C)CC2C3)=O)CC2COCC(C1)C2 46191,c1(C(=O)NC2CCN(S(CCCC)(=O)=O)C2)cc(Br)c(O)c(Br)c1 46192,c1(C(=O)NC2CN(C(c3c(C)noc3)=O)CC2C#N)cc(O)cc2ccccc12 46193,N1(C(c2c(N)cncc2)=O)CCCOC(CNC(=O)Cc2c(F)cccc2Cl)C1 46194,N1(C(C2N(CC)CC2)=O)CC=CC1(C)C(=O)NOCC1CC1 46195,C(CCN=C(NCc1ccc2c[nH]nc2c1)NCC1CC=CCC1C(C)C)SC 46196,c1(CC(=O)NC2(CC)CCN(C(c3cncn3C)=O)CC2)cnn2ccccc12 46197,C(=O)(C(C)(C)CS(C)(=O)=O)NC1C(C)CCN(C(c2ncnc3sccc23)=O)C1 46198,c1(C(N2CC(N(C(C3CN(C(C)=O)C3)=O)C)C2)=O)c[nH]c2cc(F)ccc12 46199,N1(C(c2ccc(C(=O)OCC)o2)C(=O)NC2CC2)CC2C(C1)C2(C)C 46200,C1(N(C(CC2CCN(C)CC2)=O)C)CN(C(c2c(F)cncc2Cl)=O)CC1(C)C 46201,n1(CC)nnc(C)c1CNC(c1ncc(CC2CCN(C)CC2)s1)=O 46202,Cc1ccc(C(=O)NC23CC2CN(C(C2(C)CC=CCO2)=O)C3)c(Cl)c1 46203,c1(CN(CCC)Cc2cnc(-c3ccccc3)nc2)ccc(C#N)cc1 46204,C1(NC(c2cc(OC(CC)CC)ncc2)=O)COC2(CCN(C(C)=O)C2)C1 46205,c1(NC(N2CCC(N3CCNCC3)C2)=O)ccnc2ccc(Cl)cc12 46206,c1(C(=O)NCC2N(C(CNC(=O)OC)=O)CC(O)C2)cc(N)ccc1F 46207,C1(C(=O)NCC2CCN(C(c3occc3CSC(F)F)=O)C2)CC12CCCCC2 46208,c1(NC(=O)NCC(CC(C)C)NC(=O)OCC)c(C)nn(CCO)c1C(F)F 46209,c1(C(=O)NC2CCN(C(C3(CCC)CC3)=O)CC2CO)n[nH]c2c1CCSC2 46210,C1(NC(C=Cc2cncc(C)c2)=O)(CNC(=O)CC(C)CF)CCC(F)(F)CC1 46211,C(=O)(CS(=O)C(F)(F)F)NCCCCC(=O)NCC(CCOC)(C)C 46212,c1(CC)ccc(C(=O)NC(C)(C)CNC(c2ccc(CN(C)C)[nH]2)=O)c(C)c1 46213,C1(NC(C(C)N(CCC)C(c2cc(CC)[nH]n2)=O)=O)CC2(CCOC2)C1 46214,Cc1noc2[nH]c(=N)c(C(=O)NCCCC3CCCOC3)cc12 46215,Cn1cc(CC(O)C(=O)NCCC2CC(NC(=O)CC3CCC=CCC3)C2)cn1 46216,N1(C(C(C)C2CCCC2)=O)CC(O)(CN(C(=O)CCCN(C)C)C)C1 46217,N1(C(CCSCC)=O)CC2CCN(C(c3ccc(OC)c(N)c3)=O)CC2C1 46218,N1(C(C(=O)NCCC)CC(C)CCC=C(C)C)CCC=C(c2ccco2)C1 46219,c1(C(N(CCNC(C2CC2C(F)F)=O)CC)=O)cc([N+](=O)[O-])c(Cl)cc1Cl 46220,CC1CCC(O)(C(=O)NCC(=O)NCC(=O)Nc2ccc(F)cc2F)CC1 46221,c1(OC)ccc2[nH]cc(CCN3C(=O)CCN(CC4=CCCOC4)C3=O)c2c1 46222,c1(C(N2CC(NC(C(C)CC(C)(C)C)=O)C2)=O)cccc2c1C(=O)NC2 46223,N1(C(C2(CCCC)CCC2)=O)CC(C(=O)NCC(C)(O)CO)OC(C)C1 46224,c1(C(=O)NCC2C(NC(CCC(C)(C)OC)=O)CCCC2)cccc2ccnn12 46225,C1(NC(C2(SC)CCC2)=O)CC2CN(C(=O)C(C)Cn3ccnc3)CC12 46226,CC1=C(C)CC(C)(C(=O)NCC2(CNC(C3CC(=O)N(C)C3)=O)CC2)CC1 46227,CC1CCc2cc(C(=O)NCCN(C(=O)CC3(O)CCCCCC3)C)ccc2N1 46228,O=C(C1=CCN(C(c2cc(C3CC3)on2)=O)C1)NCC1CC1C1CCCC1 46229,c1(OCCOC)cc(OC)ccc1C(=O)NCC(C)(C)c1ccsc1 46230,N1(C(c2ccc(COC)o2)=O)CCN(C(C2CC(S(C)(=O)=O)C2)=O)CC1CO 46231,c1(N(C)C)cnc(CN(C(=O)NOCc2ccco2)C2CC2)cn1 46232,c1(N2C(C)(C(N(C)C3CC3)=O)CC2)nc(C#N)nc2ccccc12 46233,c1(CCC#C)ccc(C(C)C(N2CCC(CN(C(=O)COC(F)F)C)C2)=O)cc1 46234,c1(C(=O)NCC2CCC(NC(C3(NC(C)=O)CCC3)=O)C2)cnc2c(C)cccn12 46235,CC1(C)CCC(F)(F)CC1C(=O)NC1CN(C(c2c[nH]nc2F)=O)CCC1CO 46236,C1(CNC(C(C)NC(C)=O)=O)C2CC1N(C(c1csc(-c3cnccn3)n1)=O)C2 46237,C(C(C)(C)CC(=O)Nc1cccc(CCF)c1)NC(c1cc(C)n(C)c1)=O 46238,N1(C(c2cc(CC)oc2C)=O)CCCC2(NC(c3cn[nH]c3)=O)CCCC12 46239,Cn1cc(CCNC(=O)NCCc2ccc(C(F)(F)F)nc2)c2ccccc12 46240,C(=O)(C(CC(C)(C)C)OC)NCC1OCCN(C(C2(COC)CCC2)=O)C1 46241,c1(CCN(C(C(N2CCC(OC)C2)C)=O)CC(C)C)cccc(OC)c1OC 46242,C1(NC(c2scc(COC)c2)=O)CCN(C(c2nc(C)c(C)s2)=O)CC1C(C)C 46243,Cc1cc(C(N2CCC(OCCNC(=O)Cn3cccc3)C2)=O)nn1C(C)C 46244,c1(C(=O)NC2C(C)CCN(C(C(COC)C)=O)C2)cc2cccc(Cl)c2nc1C 46245,C1(C(=O)NC(CCCNC(C(CSC)OC)=O)(C)C)Cc2cc(Br)cnc2C1 46246,C1(C(N(C2CCN(C(C3CC34CCOC4)=O)CC2)C)=O)CC(O)CN1C 46247,C1(CNC(C(C)O)=O)CCC(F)(CNC(c2ncccn2)=O)CC1 46248,N1(C(C2(C)CCNC2=O)=O)CCCC(NC(=O)CNC(c2ccccc2)=O)CC1 46249,C1(C(=O)NCC(CNC(C(c2c(C)cccc2)(C)C)=O)C)Cc2cscc2C1 46250,c1(C(N2CC(NC(c3cc(CCOC)on3)=O)C(F)C2)=O)nc(C)c(C)[nH]c1=O 46251,c1(C(=O)NCC(C)(C)NC(=O)CC(C)(C)C(F)(F)F)cnn2c1OCC(F)C2 46252,CCCCC(CN=c1[nH]nc(CC(F)(F)F)o1)NC(=O)CC(O)C(C)C 46253,c1(C(=O)NC2CCC(N(C(COC(CC)C)=O)C)CC2)cccc(Cl)c1O 46254,c1(C(C(=O)NCCOC)N(C)CCN2CCCC2)ncoc1C 46255,C(=O)(C1CCc2nccn21)N(CC(C)(C)CNC(c1coc(C)n1)=O)CC 46256,Cc1[nH]c2ccc(Br)cc2c1C(N1CC(NC(=O)CC(C)C(F)(F)F)C1)=O 46257,C=C(C)CC(C(=O)NC1CCC2CC1CO2)NC(=O)C(C)CN(C)C 46258,Cc1cccc(F)c1C(=O)NC1CCC(NC(C2(CF)CC2)=O)C1 46259,C(C(C(=O)NC(C)C(C)n1cccn1)N(C)C)NC(C(C1CCC1)OC)=O 46260,Cc1cnc(CNC(C2CN(C)CCN2C(=O)C(F)C(C)(F)F)=O)c(C)c1 46261,c1(C(=O)NC(c2nocc2C(=O)NOC2CCS(=O)(=O)C2)C)n[nH]c2ccccc12 46262,C1(OC)CN(C(=O)NC(c2c(C)nc3n2CCS3)=O)CCC1CC1CC1 46263,N1(C(CN(C)C(c2ncccn2)=O)=O)CCC(NC(=O)CN2CC3CC3C2)C1 46264,C12(CCOCC1)c1cn(nn1)CC(=O)N2.C1(C(=O)O)C2CC2C2CC12 46265,C1(CNC(c2ccn(CCC)n2)=O)CN(C(C23CCC(CC2O)C3)=O)CCN1C 46266,C(=O)(CC(CC(C)C)NC(=O)C(C)=C1CCC1)N(CCC(=O)OCC)C 46267,C(=O)(CCCS(C)(=O)=O)N1CCCC(C)(NC(=O)CCc2cncs2)C1 46268,n1(CC)nc(C(F)(F)F)cc1C(=O)NCCN(C(=O)CC(CC)=C(C)C)CC1CC1 46269,C1(CN(C)C)CCCCN1C(C1CNCC1c1cncn1C)=O 46270,c1(C(=O)NCC(CO)NC(c2ncn(C(C)C)c2)=O)cn(C)nc1Br 46271,C(=O)(C1=NOC(c2ccc(F)cc2)C1)NC1(C)CN(C(=O)Cn2cc(N)cn2)C1 46272,c1(C(N(C(CC)C(=O)OC)C)=O)coc2c1CN(C(=O)C(c1cncnc1)C)C2 46273,C(C(CC(C)C)NC(C1C(C)CCN1C(C)=O)=O)NC(c1nc(OCC)oc1)=O 46274,CC(C(CO)NC(C1CCC(=O)N1)=O)NC(c1cc(Cl)ns1)=O 46275,c1(OC)cc(CNC(=O)C(=O)Nc2ncc[nH]2)ccc1SC 46276,CCC(CC(=O)N(C(C(=O)NCC(C)(O)C(C)C)C1CC1)C)C1CCC1 46277,C1(C(=O)NCC2CCN(C(=O)CC34COCC(C3)C4)C2)C2CCCCCC12 46278,C1(C(C)NC(=O)C=CC(=O)NC2CC2)CCCCN1C(C1CC2CC1C2)=O 46279,c1(C(N(CC(C)NC(c2ccn(CC(F)F)c(=O)c2)=O)C)=O)cc(O)cc(O)n1 46280,C(C)(c1ccco1)=CC(=O)N(C(C)C(=O)NC1CCC(C(N)=O)CC1)CC 46281,CCCCC(CC(=O)NCC(N1CCC(C)C1)C)NC(=O)C=C1CCC(C)CC1 46282,C(=O)(CC1COCc2ccccc21)N(C)CC1CN(c2ncncc2Cl)CCO1 46283,C(=O)(CCCC(C)(C)C)NCc1nc(C(N2CCC(CC)CC2)=O)c(C)o1 46284,N1(C(CCC=CCC=C)=O)CCCCC1C(C)NC(=O)Cn1cccc1 46285,N1(C(C(C=C)O)=O)CCCOC(CCNC(=O)CCCn2ccccc2=O)C1 46286,C1(CNC(CC=CC)=O)CCCCN1C(c1cn(C)nc1COC)=O 46287,C(C(C(C)(C)C)NC(c1cc(Cl)c(Cl)[nH]1)=O)NC(C=C1CCC(C)C1)=O 46288,N1(C(c2cccc(OC(C)=O)c2)C(=O)NCCCSC2CC2)CCOCC(C)C1 46289,C(=O)(C(F)C(C)(C)O)NC1CCC(N(C(c2ccc(C)o2)=O)C)CC1 46290,C1(CNC(C2N(CC)CC2)=O)CN(C(c2c(Cl)c(C)nn2C)=O)CCC1(F)F 46291,S(=O)(=O)(c1ccccn1)NC1CC(C(N2CCN(C(C)C)CC2C)=O)C1 46292,N1(C(CC(C)(C)O)=O)CC(CNC(=O)Cn2cnnc2)CC12CCOCC2 46293,c1(CC)ncncc1C(=O)N(CCCNC(C1CCN1S(C)(=O)=O)=O)C(C)C 46294,C#Cc1ccccc1CN=C(NCCOCC)NC(c1ccccc1Cl)C 46295,N1(C(C2CC(N(C)C)C2)=O)CC=CC(NC(C23CCCC2C3)=O)C1 46296,C1(CNC(C2C(C)NCC2)=O)CC2(CC2)CO1 46297,CC(C)CCCC(=O)N(C1CCN(C(C2CC(C)CCC2C(C)C)=O)C1)CCO 46298,c1(C(=O)NC(C)CCNC(c2cccnc2F)=O)c(F)cccc1[N+](=O)[O-] 46299,C(=O)(CCCS(C)(=O)=O)N1CC(C)(C)C(NC(=O)CC2CC(=O)NC(=O)C2)C1 46300,N1(C(c2sc(C)c(C)c2C)C(=O)NC(C(=O)OC)C)CC2CCC(C1)C2O 46301,N1(C(CCc2cnc(C)o2)=O)CC(NC(=O)C(C)CC2CCC2)C2(CCCC2)C1 46302,NS(=O)(=O)c1ccc(C(=O)OC2CCN(CCCC=CC(=O)O)C2)cc1 46303,C1(C#N)(C(=O)NCCCN(C)C(c2cn(C)c(=O)n2C)=O)CC12CCCC2 46304,C1(NC(CNC(C(=O)NC2CC(=O)NC2)=O)=O)C2CC3COC1C3C2 46305,N1(C(C2(C)CCOC2)=O)CC2CCN(C(=O)CN3CCOCC3=O)C2C1 46306,CCC(CC)(C(=O)NCC1(C)CCCC1NC(=O)CSCCC(C)C)OC 46307,C(N=c1[nH]nc(C(F)F)s1)c1ccc(C(N(C2(CO)CCCCC2)C)=O)cc1 46308,c1(C(=O)NC(CN(C(C2(C(F)F)CC(=C)C2)=O)C)C)nc2ccccc2n1CC 46309,c1(C(=O)NCC2CCCN(C(C(C(=O)OCC)F)=O)C2)ccnc2nc(C)nn12 46310,CCCC(C)C(=O)N1CCC(N(C(=O)CCC#N)CC2CC2)C1 46311,CCCCCCC(=O)N1CCC(NC(c2c(C)c[nH]c2C(=O)OC)=O)CC1C 46312,C1(NC(c2ccc(N(C)C)nc2)=O)(CO)CCCN(C(=O)Cc2ccsc2Cl)C1 46313,c1(CC)ncc(C(=O)NCC(N2CCN(C(C3CNC(=O)N3)=O)CC2)C)c(O)n1 46314,C1(C(=O)NC2CCCN(C(COCCCOC)=O)CC2)Cc2ccccc2S1 46315,c1(C2(C(=O)NC3CCC(CCNC(CCC#C)=O)C3)CC2)cccc(F)c1C 46316,c1(CC)nc(=NCCOCCNC(c2ccn3nnnc3c2)=O)s[nH]1 46317,C(C)(C)(CN=c1[nH]c2cc(Br)ccc2o1)NC(Cc1c(C)noc1Cl)=O 46318,c1(CC(=O)NC2C(C)(C)C(CNC(=O)COc3ccsn3)C2)ccc(F)c(Cl)c1 46319,O=C(N=c1[nH]ccnc1Cl)C1CCCN(C(=O)C(F)Oc2ccc(Br)cc2)C1 46320,CC(COc1ccccc1)C(=O)NNC(=O)CN(C)C 46321,C#Cc1cnc(C(=O)NCC2C=CCN2C(c2cc3nc[nH]c3cn2)=O)c(C)c1 46322,S(=O)(=O)(c1ccc(Cl)cc1F)NCC1(F)CCN(C(C(CC)=O)=O)CC1 46323,N1(C(=O)C=Cc2ccco2)CCOC(C2CN(C(=O)C=CC(F)(F)F)C2)C1.c1nc[nH]n1 46324,C1(C(N2CCC(CC(C)(C)C)C2)=O)CSCCN1C(C1CCC(N(C)C)CC1)=O 46325,C(=O)(C1=CNC2=NCCC2=C1)N1CCN(C(C2C(OCC)C2)=O)CC1CC 46326,c1(N2CCCC(C)(CNC(c3n(CC)ccc3)=O)C2)ncnn2cccc12 46327,C1(CN(C(C2CC(=C)C2)=O)C)CCN(C(=O)CNS(=O)(=O)CCOCC)C1 46328,C(c1ccc(Cl)cc1F)=CC(=O)N(CC(CC)NC(C1(OC)CCCOC1)=O)CC 46329,Cc1nn(C)c(C(F)F)c1C(=O)NCCNC(C12CCCC1CCC2)=O 46330,CCCS(=O)(=O)NC(C)C(=O)NCC12CC(NC(=O)COCC(=O)OC)(C1)C2 46331,C1(CNC(CCSC)=O)CCN(C(C2(C3CCCCO3)CCC2)=O)CC1C 46332,c1(CO)ccc(F)c(NCCCN2CCC(F)(c3ccccc3)C2)c1Br 46333,N1(Cc2ccc(C(=O)OC)s2)CCCCC(NC(c2cccc(=O)n2C)=O)C1 46334,N1(C(CCCNC(=O)OC)=O)CC2(C1)CN(C(=O)CC1CC(C)(C)CO1)C2 46335,C1(NC(CCc2cnc(C)s2)=O)C=CCN(C(C2C(C)(C)C2(C)C)=O)C1 46336,c1(CNC(C2C(O)CCN(C(CCC=C)=O)C2)=O)ccc2nc[nH]c2c1 46337,N1(C(c2cnc(C)n2C)=O)CCC2(NC(=O)Cc3cncnc3)CCCC12 46338,N1(C(C(C)(Cl)Cl)=O)CCC(C)(CNC(c2cnn(CC3CCCC3)c2)=O)CC1 46339,N1(CC(=O)NCC2(C)CCCN2C(=O)C2=CSCS2)C(=O)C2CCCCC2C1=O 46340,C1(C(=O)NC(CC)(C)C2CC2)C2CC1N(C(=O)C=Cc1cn[nH]c1)C2 46341,C1(C(=O)N(C)CCOCCO)(CC)CCN(C(c2cc(O)nn2C)=O)C1 46342,c1(C(=O)NCC2CCCC(C#C)C2)coc2c1CN(C(=O)Cc1cncnc1)C2 46343,C1(CNC(c2c(CNC(c3ccoc3C3CC3)=O)occ2)=O)CC12CCOC2 46344,C(=O)(C(C(=O)NC1CC(C(=O)N(C)Cc2ccc(F)cc2)C1)OC)OCC 46345,C1(C(N(CCNC(=O)CC2COC3CC2C3)CC)=O)(OC)CCCCCCC1 46346,C12CN(CCO1)C2=O.C1(CC)CC2CC2N1C(=O)CCCN1CCCC1 46347,c1(C(=O)NCCCN(C)C(c2ccc(F)c(N(C)C)c2)=O)cc(S(N)(=O)=O)co1 46348,Cn1ccnc1C(N1CCC(n2cc(CCN(S(C)(=O)=O)CCO)nn2)C1)=O 46349,N1(C(c2n[nH]c(CC)c2C)=O)CC(CNC(c2cccc(C)n2)=O)N2CCC1C2 46350,C1(NC(C2C3(CC(OCC)C3)C2)=O)CCN(C(c2ccncc2C)=O)C(C)C1 46351,C1(C(=O)NCC2(C(C(C)C)O)CC2)CCC=CCC1 46352,c1(CC(C)N(C(=O)NCCN2CC=CCC2)CC)cccc(C#N)c1 46353,c1(C(N(C(C)CCNC(=O)Cc2cc[nH]c(=N)c2)C)=O)cc(F)c(F)c(Cl)c1F 46354,c1(C(N2CC(NC(C3C(F)(F)C34CC4)=O)C3(C2)CC3)=O)n[nH]c2ccc(F)cc12 46355,C(N=c1[nH]c2cccc(F)c2s1)C1C(C)CN(C(c2cc3n(n2)CCCC3)=O)C1 46356,CCC(C)(C)CCCC(=O)NC1CN(C(=O)CNC(=O)CC(F)(F)F)CC1C 46357,CC1(COC(c2ccc3ncc(Br)n3c2)=O)COCC2CCCN12 46358,C(c1ccc(OC(C)C)cc1)=CC(=O)NC(CNC(CC(=O)OC)=O)CC 46359,C1(c2cn(CCO)nn2)(NCCCn2ncc(CC(=O)N(C)C)c2)CCOC1 46360,C12(C(N3CCC(OCCNC(C(C)OCCOC)=O)C3)=O)CCC(CO)(CC1)C2 46361,N1(C(C(C)N(C(=O)C=CC(C)(C)SC)CC)=O)CC2CCN(C)C2C1 46362,c1(OC)ccc(N2CCCC2=O)cc1.N12CCC(CC1)CC(=O)NC(C)C2=O 46363,C(C)(C)(CC(C)NC(=O)CCN(C(c1ccc(C)s1)=O)CC1CC1)OC 46364,c1(CC(N2C(C)CN(C(c3csc(O)n3)=O)C(C)C2)=O)ccc2c(c1)CCN2C 46365,C1(N(C(c2cnc(C(C)C)s2)=O)CC)CCCN(C(C2(C#N)CCOC2)=O)CC1 46366,N1(C(C(CC=C)OC)=O)CCC(CNC(c2cnc(COC)nc2O)=O)C(C)C1 46367,c1(CC(=O)NC2C(C)(C)CN(C(=O)C(F)F)CC2)ccc(O)c([N+](=O)[O-])c1 46368,C1(O)(C(=O)NCC(C(C)C)Nc2ncc(C(=O)OC)cn2)CCCC(C)CC1 46369,N1(C(C2CSCC(=O)N2)=O)CC2(CCN2C(=O)C(O)c2ccsc2)C1 46370,c1(CCC(=O)NCCC(C)NC(C2CC2c2cnn(C)c2)=O)c(F)cccc1Cl 46371,CCC(CC)(CO)C(=O)NCC(C)(F)CNC(c1ccc(N)cc1F)=O 46372,Cc1cc(C(N2CCN(C(=O)Cc3cnsc3)C3CC23)=O)c(C)nc1C 46373,C#CCC(C)(C)C(=O)NC1CCCCC1NC(=O)Cc1ccsc1C 46374,c1(CC)nn(C)c(CC)c1CNC(c1ccc(F)cc1)c1nnnn1C1CCC1 46375,N(C1CCNc2c(C(F)(F)F)cccc21)C(c1ccc2sncc2c1)=O 46376,C1(C(CNC(=O)C=CC2CCC2)C2CC2)CCN(C(C2C3CNC(=O)C23)=O)CC1 46377,Cc1cc(=NCC2CCCC2C)[nH]cc1S(=O)(=O)NCC(O)C(C)(C)C 46378,c1(C(=O)NCc2ccccc2OCC2CCCCO2)ccc(CF)cc1 46379,c1(COC(C)=O)ncc(C)cn1.C1C(F)C(=O)N2CCCC2CN1CC 46380,C(CCCC(=O)N1CC(C(=O)NC(c2ccccn2)C)CCC1C)(OC)OC 46381,Cc1cc(C(=O)NCc2nc(C(N3CC(N4CCCC4)C3)=O)c(C)o2)c(O)nn1 46382,C1(C(N(CCCNC(=O)CC2CCCC2(F)F)C)=O)CCN(C)S1(=O)=O 46383,C(=O)(CCC1=CCCCC1)NCc1c(C(=O)NC2CN(C)CC2(F)F)[nH]cc1 46384,C1(N(S(c2c(C)onc2)(=O)=O)C)CCc2ccccc2C1 46385,C(=O)(C1OCCn2ccnc21)NCCCC(CCC)Nc1ncnc(CC)c1F 46386,CC(C)(CC(F)(F)F)C(=O)N1CC(NC(=O)COC2CCCCCC2)CC(F)C1 46387,N1(C(=O)NC2CC(COc3ccccc3)C2)CCCC2(CCCNC2=O)C1 46388,N(C(=NCCc1sccc1Br)N(C)Cc1cnn(C)c1)CC1CCCC(OC)C1 46389,N1(C(c2cc(C)no2)=O)CC(C)(C)CC1CNC(c1nnc(C)cc1O)=O 46390,C1(C(=O)NCC2N(N=O)CCC2)CCN(C(C2CN3CCN2CC3)=O)CC1O 46391,c1(C(=O)NCC2C(C)(C)N(C(=O)CC3CCCO3)CC2)cnn2cccnc12 46392,Cc1cccc2nc(N3CCC(O)(CNC(=O)Cc4ccccc4F)CC3)oc12 46393,CC#CCCC(=O)NCC(C)NC(=O)C(C)CC1CCCCC1 46394,c1(NC(C2CSCCN2c2ccncn2)=O)cc(Br)cc2cn[nH]c12 46395,C12(NC(CC(C)NC(=O)C#CC3CC3)=O)CCC(CC1)C2(C)C 46396,C1(C(N(CCNC(=O)CC2CC=CC2)C2CC2)=O)CCOC(=O)N1 46397,C1(C(=O)NC2CC(N(C(=O)C(=O)NCC3CC3)C)C2)CC(C#N)C1 46398,Cc1c[nH]nc1C(=O)NC(CO)C(=O)N1CCCC1 46399,C(=O)(CCC1CCc2ccccc21)NC1CC(C)(NC(CC(CCC)O)=O)C1 46400,N1(C(C)C)N=C(C(=O)N2CCCC2CNC(=O)C(O)CC2CCCC2)CCC1=O 46401,C(=O)(C(CC1CCOCC1)NC(=O)C=CC1CCC1)NC(C(C)F)C 46402,Cc1cc(C(=O)NCCC2CCCN2C(=O)C=CC2CCOC2)c(Cl)cc1Cl 46403,c1(C(=O)NC2C(NC(COCCOCC#C)=O)CCC2)cnn(C)c1C(F)(F)F 46404,CC(C)(C)S(=O)Cc1cccc(C(=O)OCC2CN(c3ccccc3)C(=O)O2)c1 46405,N#Cc1ccc(C(=O)NCC2CCC(NC(c3cnc(-c4ccco4)s3)=O)C2)[nH]1 46406,c1(C(=O)NCCCN(C(C(C)OCC=C)=O)CC)cccc2c1CNC2=O 46407,CCC1CNC(=NCCN2CCN(C)CC2)N1 46408,CCC(CN(C)C)C(=O)N(CCCNC(c1sc(C)nc1CC(C)C)=O)CCO 46409,N1(c2nccc(Br)c2Br)CCC2CCCCC2C1 46410,CCC(C)CC(C(=O)Nc1cnc(C(C)C)nc1)NC(c1ccsn1)=O 46411,c1(NC(CC)=O)ccc(NC(C)C(c2ccccc2)NC(=O)CCSC)cn1 46412,CC(CCNC(=O)CCC1CCN(C(=O)Cc2cc[nH]n2)CC1)C(C)(C)C 46413,C1(C(=O)NCC2(SC)CC2)CCCCCN1C(C1CCC(C(=O)N(C)C)CC1)=O 46414,c1(OCC)ccc(C(=O)NCCC2CN(C(C3(O)CC(C)(C)C3)=O)CC2C)cc1 46415,CC1CCOC(c2ccccc2)CN1c1nnnn1CCCCCS(C)(=O)=O 46416,Cc1cc(C#N)cc(C)c1C(=O)NC1CCN(C(C2CCCC2)=O)CC1O 46417,c1(C(N2CCC(CC(N3C4CCC3COC4)=O)C2)=O)ccc(F)cc1O 46418,c1(OC)ccc(C(=O)N(C)CC2CCCN2C(c2ccnn2C(C)C)=O)c(C)c1 46419,Cc1ccc(Br)c(NC(c2cc(-c3cccc(N4CCOCC4)c3)cs2)=O)c1 46420,N1(C(C2CC2NCc2c[nH]nc2-c2ccccc2)=O)CCN2CCCCC2C1 46421,N1(C(c2cc(SC)oc2C)=O)CCC2(CCCN(C(=O)C=C3CC3)C2)C1 46422,Cc1nn(C)c(C)c1C(N1CCC(N(CCO)C(C2CN(C)CC(C)O2)=O)C1)=O 46423,O=S(=O)(c1[nH]c(=NCC2C(F)(F)C23CCCC3)ccc1Br)NC1CC=CCC1 46424,Cc1cc(C(=O)N(CCN(C)C(c2scnc2C2CCCC2)=O)C(C)C)no1 46425,C1(CN(C(=O)C(C2CC2)NC(C2(C(N)=O)CC2)=O)C)CC1(C)C 46426,c1(C(N2CCC(CNC(C(CC3CC3)OC)=O)C2(C)C)=O)cccc2ccnn12 46427,c1(C(=O)NCC2C(C)CCN2C(C2CC2c2ccccc2)=O)ccc(F)cc1Cl 46428,N(C)(S(C)(=O)=NC(=O)c1[nH]c2ncccc2c1N)CC#C 46429,O=C(N=c1cc[nH]cc1O)C1CCCN1C(C1CCC2CCC(=O)N2C1)=O 46430,C1(NC(N(CCC)CCC)=O)(Cc2ccc(F)cc2)CCNCC1 46431,N1(C(C(C(C)O)(C)C)=O)C2CCC1CN(C(C13CCCN1CCC3)=O)CC2 46432,C1(C(=O)NC(C(=O)N2CC(N3CCOCC3)C2)C2(C)CC2)CCC2CC1CO2 46433,CC(C)(C(O)C(F)F)NC(C1CCCC1CNC(C1(n2cccc2)CC1)=O)=O 46434,Cc1cc(=O)oc(C)c1C(=O)NC1C=CC(CNC(C2COCCN2C)=O)C1 46435,CCCC(CCC)C(=O)NCc1cc(C)c(C(=O)NOCC2CC2)o1 46436,C#Cc1ccc(C(=O)NCCC2(C)CCN(C(c3cnccc3OC)=O)C2)cc1 46437,c1(C(=O)NC2C(c3ccc(Br)cc3)(CC)C2)ccc(S(C)=O)c(F)c1 46438,C1(C(N2CCC(O)(CC)CC2)=O)CN(C(=O)Cc2cccc(F)c2)CCC1(C)C 46439,N1(CC(=O)NC(C(=O)NCCN(CCC)CC)C2CCCO2)CCC(=O)CC1 46440,Cc1nc(C)n(Cc2cn(CCNC(C3CCC3C(F)(F)F)=O)nn2)n1 46441,N1(C(c2ccn(COC)n2)=O)CC(OC)CC1CNC(c1nocc1Cl)=O 46442,N1(C(c2nccc(C)n2)=O)CCCCC(NC(=O)C=CC(C)C)CC1 46443,C(=O)(CC1CCOc2ccccc21)NCC1C(NC(CCN(C)CCO)=O)CC1 46444,N1(C(C(c2ccc(F)cc2)CC)=O)CC2CC1C2NC(=O)CS(C)(=O)=O 46445,CCC(CC(=O)N1CCC(CN=c2nc(-c3ccccc3)[nH]s2)(C)C1)C(F)F 46446,C1(N(C(C)=O)C)CCN(C(=O)C(Cc2cn[nH]c2)C2CCC2)CC1 46447,Cc1c(C(C(C)C)NC(N2CCOC(c3ccccc3)C2)=O)oc2ccccc12 46448,c1(CN(C(C(=O)NC2CCCCC2)C2CCSC2)C)ccc(-c2ccccc2)o1 46449,N(C1CC2(CN(C(c3ccnn3C)=O)C2)n2ccnc21)C(CC(=O)NCC#C)=O 46450,C(=O)(CC(O)C(C)C)N(C1CCC(CNC(c2cc(C)ncn2)=O)CC1)C 46451,c1(SCC(N2CC(CNC(C3C(CC)OCC3)=O)C2)=O)ccc([N+](=O)[O-])cc1 46452,Nc1ccnc(C(N2CCC(F)(CNC(=O)CC3CSCCS3)C2)=O)c1Cl 46453,CCCCC(C(=O)NOCC(=O)Nc1cncc(Cl)c1C)N(C)C 46454,c1(NC(=O)CC2CCCN2C(=O)Nc2nnc(CC)o2)c(Cl)cccc1Cl 46455,N1(C(c2c(C)cccc2)=O)C(C(=O)O)CCC1(C)C 46456,C(=O)(C1CCCc2scnc21)N1C(C)CN(C(=O)COC2CCCCC2)CC1 46457,c1(C(=O)OC)nccc(NC(C2(C)CCN2C(=O)OCC(C)(C)C)=O)c1C 46458,c1(C(=O)NC2C(C=C)CN(C(=O)COCCC)C2)cc(S(N)(=O)=O)c(C)s1 46459,c1(NC(C2(F)CCN(C(CN(S(C)(=O)=O)C)=O)C2)=O)cc(O)nc(C(F)F)n1 46460,N1(C(CN(C(=O)C(O)c2ccsc2)C)=O)CC=C(CO)CC1 46461,CCC(C)CCCCC(=O)NCC(CC1CC1)C(=O)N1CC(C)C(F)C1 46462,C(CC(C)C(=O)NCCC1(O)CN(C(c2ccc(C3CC3)s2)=O)C1)OC 46463,c1(C(N2CC(NC(c3c(C)ccs3)=O)C(C3CC3)C2)=O)cc2nc(Cl)ccc2o1 46464,N1(C(CC=CCC)=O)CCn2c(CNC(C3C(Cl)(Cl)C34CC4)=O)nnc2C1 46465,C1(CNC(C(CC)N(C)C)=O)CCN(C(C2CCCCO2)=O)CC1C1CC1 46466,N1(C(C(C)N(C)C)=O)CCCN(C(c2cc(C(F)(F)F)ns2)=O)CC1C 46467,c1(CN2CC3(CCC(C(=O)Nc4ccnnc4Br)O3)C2)ccc2nc(O)[nH]c2c1 46468,CCP(=O)(CC)c1ccccc1C(N1CC(CCNC(=O)CCC(N)=O)C1)=O 46469,C1(NC(C(C)c2ccsc2)=O)C2CCN(C(C3CC3(Cl)Cl)=O)CC12 46470,Cc1ncnc(C(=O)NCC2(CN(C(=O)C(C)CC3CCCCC3)C)CC2)c1C 46471,Cc1oc2ncnc(O)c2c1C(=O)NC1CCN(C(c2cc(Cl)no2)=O)CC1O 46472,n1(CCNC(C2(CO)CCC2)=O)cc(C2CCCCO2)nn1 46473,c1(OC)cc(NC(=O)NCC2(O)CCOCC2)ccc1F 46474,C(C)(CC(C)N=c1c(C#N)c[nH]c2ccc(Cl)cc12)NC(Cc1cc(C)no1)=O 46475,n1(CCC2CN(C(c3csc(Br)c3)=O)C2)cc(CC2CCCCO2)nn1 46476,c1(C(C)C)nc(N2CCCC(NC(=O)Cc3cccc(F)c3)C2)cc(Cl)n1 46477,N1(C2CCN(C(=O)CC3COCCO3)CC2)CCN(C(c2cnns2)=O)CC1=O 46478,C1(NC(c2cc(C(=O)OC)oc2C)=O)CC2CC(C1)N(C(c1n[nH]c(O)n1)=O)C2 46479,C1(NC(c2c(C)noc2N)=O)CN(C(c2ccccc2)=O)C2(CCOC2)C1 46480,CC(C)CCCC(C)C(=O)NC1CCC(C)N(CC(=O)N(C)C)C1 46481,N1(C(=O)CCCn2cncn2)CC2CC2(C(=O)NC2CC23CCC3)C1 46482,C1(CC)(CC)CCCN1C(C1C(CNC(=O)CC2(C)CCC2)C1(C)C)=O 46483,CCC(C)C(C)C(=O)NCC(CC)(CC)NC(c1cccc(=S)n1O)=O 46484,c1(C(=O)NC2(C)CN(C(=O)C(c3ccc(Cl)cc3Cl)O)C2)cc(O)cc(Cl)c1 46485,c1(C(=O)NC2C(CNC(CN(C(C(C)C)=O)C)=O)COC2)cnn2cccc(Cl)c12 46486,c1(C(N2C(CNC(c3c(C)cccn3)=O)CC2)=O)cccc2c1C(=O)OC2(C)C 46487,N1(C(Cc2c(C)nc[nH]2)=O)CCC2CCN(C(=O)CNC(N)=O)CC12 46488,c1(C(=O)NC2C(CNC(C=COCC)=O)COC2)cccnc1Cc1ccco1 46489,N1(c2nccc(SC)n2)C2CCC1CN(C(=O)C(C)Cn1ccc(C)n1)CC2 46490,n1(C(C)C)c(=O)nc(O)c2c(C(=O)O)cc(NCc3conc3C(C)C)nc12 46491,C12(C(=O)NC(CCNC(C(C=C=C)C)=O)C)CC3CC1C2C3(F)F 46492,c1(C(N2C(C)C(NC(=O)C(CC#N)c3nn[nH]n3)CC2)=O)ccc([N+](=O)[O-])c(O)c1 46493,C1(CC(=O)NCCS(N)(=O)=O)C2CCCC2N1C(=O)COc1ccsn1 46494,c1(C(=O)OC)ccc(C(=O)NCCCC(C)(C)NC(C2CCS(=O)(=O)N2)=O)cc1 46495,C1(NC(C(C2CCC2)OC)=O)CC(O)(CNC(C2CCCN2C(N)=O)=O)C1 46496,C(=O)(C1=CC2CCCC12)NC1(CNC(CN2CC(C)C2)=O)CCCCCC1 46497,C(C(C(C)C)NC(=O)CC1(OC)CN(C(=O)CC(C)n2cccc2)C1)OCC 46498,C(=O)(CC(C)(C)C(=O)NC1CN(C(c2cn(C(F)F)cn2)=O)C1)OC 46499,c1(NS(c2ccc(C)cc2)(=O)=O)ccc(C2=CCC(O)CC2)s1 46500,C1(CC)(COC)CCN(C(C2(N(C)C(C3CCCO3)=O)CCCC2)=O)CC1 46501,CC(C)C(O)C(=O)N1CC(NC(C2(O)CC(CF)C2)=O)C(O)C1 46502,c1(C(N2C(C(C)NC(=O)Cc3ccno3)CCC2)=O)cc(Cl)ccc1Cl 46503,c1(C(=O)OCC)cc(CSCC(=O)NCc2c(C(C)OC)ccs2)oc1C 46504,c1(C(=O)OC)ccc(F)c2c1CN(C(=O)C(=O)N(C1CCC(C)C1)C)C2 46505,c1(CCCN2CCC(NCc3cn(CC(=O)NC)nn3)CC2)ccc(F)cc1F 46506,C1(CCC)(NC(=O)C(F)C(C)(F)F)CCCN(C(=O)C(C)Oc2cccnc2)C1 46507,CCCC(C)CCCC(=O)N1CCN(c2nccc(OC)n2)CC(O)C1 46508,c1(C(N2CCCC(CCNC(CCC=CC)=O)C2)=O)cc(N)c(C)cc1C 46509,c1(C(=O)NCCNC(C2CCCN(C(C)=O)C2)=O)ncc(Br)cc1F 46510,CCC(CC)C(F)C(=O)NCCC1COCCN1C(=O)CC(C)(C)O 46511,c1(OC)ncc(C(=O)NC2CCC(N(C)C(c3cnc(CC(C)(C)C)o3)=O)C2)s1 46512,c1(C2C(C(=O)NCCCCCNC(C(C)OCC#C)=O)C2)cc(F)c(F)c(F)c1 46513,N1(C(C(C)(C)CF)=O)CC2CC(F)(F)CCC2(NC(c2cc(Cl)cnc2O)=O)C1 46514,c1(NC(=O)C(=O)NC2CC(=C3CCC3)C2)ccccc1 46515,N1(C(C(C)C(=O)CN(C)S(N)(=O)=O)=O)CCN(C(=O)CC(=O)NC2CC2)C2CC12 46516,N1(C(C(C)(C)SC)=O)CC(NC(C2CN(C3COC3)C2)=O)C(n2ccnn2)C1 46517,c1(C(C)=O)cc2cc(C(=O)Nc3ccc(CS(C)(=O)=O)cc3F)sc2s1 46518,Cc1oc2c(F)c(F)c(F)c(F)c2c1C(=O)NC1CC1(C)C(F)F 46519,C1(C(N2CCC(CCNC(C(C)C3CCC3)=O)C2)=O)CCC2(CC1)CC2 46520,C1(CCCC)CN(C(=O)CCOC)CCN1C(=O)CCC1CC1 46521,c1(C(N(CCCC)CCCC)=O)ncccc1N(C)C 46522,C(=O)(C1CCCc2ncccc21)NCC1(F)CN(C(C2(C)CCCC2)=O)C1 46523,c1(-c2c(C)cc(OC(c3ccccc3)CCO)cc2)c(C)nc2ncnn2c1N 46524,CN1CC(C(N2CC(C(=O)NCC=CCNC(C34CC(C#N)(C3)C4)=O)C2)=O)CC1=O 46525,N1(C(Cc2n(C)ncc2)=O)CC2CC2(C(=O)NCC(F)CO)C1 46526,CC1CCN(C(=O)CC(C)n2cccn2)C(C)C1NC(c1ccccc1Br)=O 46527,c1(CS(N2C(C(=O)Nc3cccnc3F)CCC2)(=O)=O)cccc(Br)c1 46528,c1(N2CCC(C(=O)Nc3nccnc3F)C2)ncnn2cc(Br)cc12 46529,C1(C)(C(=O)NCC(CNC(c2nccc(C(C)(F)F)c2)=O)O)CCS(=O)(=O)CC1 46530,CCC(CC(=O)NC(C)CCC=C(C)C)N(C(=O)CCCN(C)C)C 46531,N1(C(C2(CC)CCCN2C(=O)C(C2CCCCC2)C)=O)CC2CCCC(C2)C1 46532,C1(C(=O)NC(C2(O)CCN(C(C3CCCC(C)C3)=O)C2)C)CCC2C(CC1)C2(F)F 46533,C1(NC(C(CN(C)C)NC(CSCC#C)=O)=O)CC=CC(O)C1 46534,c1(OC)nc[nH]c(=NCCC2CC(C)(C)CCO2)c1F 46535,C1(CC#C)(C(N2CC(O)(C(C)NC(=O)CSCc3ccccc3)C2)=O)CCOC1 46536,CC1C(C(=O)N2C3CCC2CC(C(=O)Nc2ccc(F)cc2)C3)=NOC1C 46537,c1(COC)cc(C(=O)NC2CC2CNC(c2cncnc2)=O)cs1 46538,c1(C(=O)NC2CC(NC(=O)Cn3ncnn3)C(O)C2)c(F)ccc2nc[nH]c12 46539,C1(CNC(c2cnn(CC)c2C2CC2)=O)CCN(C(=O)COC(C)C)CC1(F)F 46540,N1(C(C2CCC(CC)CC2)=O)CC(CC(=O)NCCc2cncn2C)CC1(C)C 46541,N1(C(C)=O)CCOC(C(N2CCC(CNC(c3ncsc3C3CC3)=O)CC2)=O)C1 46542,c1(C(=O)NC2C(N(C(=O)C=CC(c3ccccc3)=O)CC)COC2)ccnc(S)c1 46543,C1(C(C)C)CCN(C(=O)NCC23CC2CCN3C(=O)OC(C)(C)C)C1C 46544,Cc1cc(CC(N2CCC(C)(CNC(C3CCS(=O)(=O)N3)=O)C2)=O)n(C)n1 46545,N1(C(c2cc(CC)c(C)s2)=O)CCC2C(NC(=O)C3=CCC3)C2C1 46546,C1(C)(CC)CCN(C(=O)CC2CCCN(C(=O)C(C)C3CCC3)C2)CC1 46547,C(=O)(N1CCC(C(=O)NC(C)Cc2nc[nH]n2)O1)c1n(CC)nc(C)c1 46548,c1(NC(C2CN(C(=O)CCc3ccoc3)CC23CC3)=O)cc(CO)cc(CO)c1 46549,N1(C(CC=C=C)=O)CCCCCC1C(N1CCC1C1CCCCC1)=O.CC(=C)Cl 46550,S(=O)(=O)(c1c[nH]c2cc(F)ccc12)Nc1c(C)ccc(-n2cncn2)c1 46551,c1(CC)ccc(C(=O)N(C)CCOCCC(=O)NOC2CCOC2)cc1 46552,n1(CC(=O)NCC2N(C(CCCCC=C)=O)C3C(C2)C3)ncn2nccc2c1=O 46553,C(=O)(C(O)CCNC(C1(CN2CC3CC3C2)CC1)=O)NCC(C)N(C)C 46554,c1(C(N2CCC(C(CNC(C(C)(C)F)=O)O)CC2)=O)c[nH]cc(Cl)c1=O 46555,c1(C(C(=O)NCCC#N)N(C2C3CCCC23)CC)cc(C)nnc1C 46556,N1(C(c2cn(CC)nc2)=O)CC2C=CC1C(C(N1CCCSCC1C)=O)C2 46557,c1(C(N(CC(CNC(C2(COC)CC2)=O)(C)C)C)=O)cc2cc(Cl)cc(C)c2[nH]1 46558,c1(N(CCCNC(=O)NC2(CSC)CC2)C)ccccc1 46559,N#CC1(CNC(c2[nH]ccc2CNC(C2CC2(F)F)=O)=O)CCC1 46560,Cc1cccc(CC(N2CCC(CC(=O)Nc3c[nH]nc3C(N)=O)C2)=O)c1Cl 46561,N1(C(c2ccc(C)s2)=O)CC2CC(C1)CN(C(=O)C(C)C(C)O)C2 46562,C(=O)(C(C)(CC)CO)NCCC1N(C(c2cnc(CC)s2)=O)CCOC1 46563,C(CN=C(NCCc1cccc(F)c1)NCc1nc(C(F)(F)F)cs1)SC 46564,CC(O)(C(=O)NC1CC(CNC(c2coc(CC3CC3)n2)=O)C1)c1ccccc1 46565,C1(NC(c2n[nH]c(C)c2Cl)=O)CCC2(CC1)CCN(C(c1ccc(CO)s1)=O)C2 46566,c1(-c2c(F)ncc(C#N)c2)nc(C(=O)Nc2c(Cl)ccnc2Cl)n2ccccc12 46567,c1(C(N(C(C)CNC(c2ccc(-c3cccs3)[nH]2)=O)C)=O)ncc(F)cc1N 46568,C1(NC(C2(F)C(C)C2)=O)CCC(F)(CNC(c2ccc(Cl)cn2)=O)C1 46569,c1(C(N2CC(NC(c3cc(CC)no3)=O)C(C)C2)=O)c(C)nc2sc(C)nn12 46570,O=C(CS(=O)CCC(F)(F)F)NCC1CC(O)CN1C(c1cc(F)c[nH]1)=O 46571,C(CCCCCCCO)=CC(=O)NCC1(OC)CN(C(C2CCOC2)=O)C1 46572,N1(C(C(C)c2cccs2)=O)CCC(O)CC1C(N1CCC(c2ccco2)C1)=O 46573,C1(C(=O)NCC2(NC(C(CCC)F)=O)CCOCC2)CN2CCC1CC2 46574,N1(CC(C)(C)NC(=O)CCc2ccncn2)CCN(C(C2CC(O)C2)=O)CC1 46575,N1(C(COC2CC(NC(C(C)OC(C)(C)C)=O)C2)=O)CC2CN(C)CC2(C)C1 46576,CC(CNC(=O)CCc1cscn1)(CO)NC(=O)Cn1cccn1 46577,c1(C(=O)NCC(CNC(C(CC)N(C)C)=O)(C)O)cc(N)c(C)c([N+](=O)[O-])c1 46578,Cc1oc(C(N2CCOCC2CNC(=O)CC2=CCOCC2)=O)cc1S(N)(=O)=O 46579,c1(C(=O)Nc2c(C(=O)OC)nn(CC(F)(F)F)c2)c(C)cc(C)nc1C 46580,C=CCCCCC(=O)NC(C(=O)NC1CC12CCC2)c1ccco1 46581,Cc1cccc(COCC(C)C(=O)NC2CN(C(C3CCS3(=O)=O)=O)C2)c1 46582,N1(c2nccc(OCC)n2)CCC(NC(C2C=CC(=O)N=N2)=O)C(F)C1 46583,c1(N(C)CC2(OC)CCOCC2)nc(=NCC#CCCO)[nH]c2cccc(F)c12 46584,NC(=O)CCC(=O)NCC1CC(NC(=O)Cc2ccncc2Cl)CC1O 46585,c1(C(N2CC(C(N)=O)(CNC(C(COC)OC)=O)C2)=O)cc2c(cc1N)OCO2 46586,C1(CN(C(=O)C(C)(C)C)C)CCCN1C(c1ccsc1CCc1ccccc1)=O 46587,CCCCC(CNC(=O)CC1(CNC(=O)C(C)n2cccc2)CC1)CCC 46588,C(=O)(C1=Cc2ccccc2C1)NC1C2(CCN(C(COCCOC)=O)C2)CCC1 46589,CCCCCS(=O)(=O)CC(=O)N(C(C)CNC(=O)CC(F)(F)CS(C)(=O)=O)C 46590,N1(C(CSCC#C)=O)CCCC2(CCCCC2NC(c2cnn[nH]2)=O)C1 46591,C1(C(=O)OC)CC1C1CCN(C(=O)C(C)CC(C)C(=O)O)CC1 46592,C1(c2ncc(C)cn2)CCN(N(CC2CC2)C(C)C)CC1 46593,C(C(=O)NCCC(F)CN=[N+]=[N-])(C(C)(C)C)NC(C=C=C(C)C)=O 46594,C1(C(N(C2CCN(C(C(C)(C)O)=O)C2)CCO)=O)CCOC2(CCOCC2)C1 46595,CP(C)(=O)C1(O)CCN(CC(=O)NC(c2ccccc2Cl)C2CCCCC2)CC1 46596,C1(NC(c2c(C)cn(C)n2)=O)CC2CC1CN(C(=O)C(C)(C)C(F)(F)F)C2 46597,c1(C(CC)(C)NC(=O)CCn2cc(-c3cc[nH]n3)nn2)ccccc1Cl 46598,C(C(CNC(=O)Cc1ccno1)S(C)(=O)=O)NC(CCC)=O 46599,Cc1ccc(C)n1CC(N1CCCC1CN(C(=O)C(C)N1CCCC1)C)=O 46600,N1(C(=O)Cc2cccnc2)CC2(CCN(C(C3CCCN3C(=O)C3CC3)=O)C2)C1 46601,c1(CC(=O)N(C)CCOCCNC(c2cocn2)=O)ccc2ccccc2c1 46602,C1(NC(C2COCCN(C(C3(OC)CCCC3)=O)C2)=O)CC(C)N(C)CC1C 46603,c1(OC)cccc(CNC(=O)C(O)C2CN(C(=O)C(C)(C)C#N)C2)c1 46604,N1(C(Cn2c(C)cc(C)n2)=O)CCC2C(C1)NC(=O)CN2C(=O)CC1C=CCC1 46605,C1(NC(=O)Cn2cccn2)CC2(C1)CN(C(c1cc(O)ccc1I)=O)C2 46606,C1(CC=C)(NC(=O)CC#N)CN(C(=O)CC(C)c2ccco2)C1 46607,c1(N2C(C3CCN(C(C4(SC)CC4)=O)CC3)C(C)(C)C2)nc(C)nc(Cl)c1C 46608,C(=O)(C(C)(C)C(=O)N1CCCC(NC(=O)CC2(C#N)CCC2)C1)N(C)C 46609,C1(N(C(=O)Cn2cccn2)C(c2cc(Cl)cc(Cl)c2)CO)CCC12CCNCC2 46610,CC1CC(C#N)CN(C(c2cc3c(C)snc3s2)=O)C1 46611,N1(C(C2C(CC(C)C)C2)=O)CCCC(F)(C(N2CC3CC3C2)=O)C1 46612,N1(C(CN(C(=O)CCC(=O)C2CCCC2)C(C)C)=O)CC(O)CC1CO 46613,C(=O)(C(F)C(C)(C)O)N(CCNC(CCC#CC)=O)CCc1ccccc1 46614,c1(C(=O)NC(CNC(C=CCOCCOC)=O)CC)ncnc2sccc12 46615,Cc1cnc(Cl)[nH]c1=NC(=O)c1cnc2n[nH]c(-c3ccnc(F)c3C)c2c1 46616,c1(C(=O)NC2CC(CNC(C(C)(C)CF)=O)OCC2)cc(Cl)c2n[nH]cc2c1 46617,C(C(C)C)(C(O)C(=O)NCC1(O)CCCN(C(C2SC3C=CC2CC3)=O)C1)OC 46618,C(CC(C)C(=O)NCC(c1ccccc1F)NC(C1CCC1(F)F)=O)=CCC 46619,CCC(C)(O)CCNC(=O)C(C(C)OC)NC(=O)C(N1CCCCC1)C 46620,c1(C(=O)OCCOCCCC)cc(Cl)nc(-c2ccc(F)cc2)n1 46621,C1(NC(c2ccc(OC)s2)=O)CN(C(=O)CC(C2CC2)C2CC2)CC2(CCC2)C1 46622,CC(C(=O)Nc1ccsc1C(N)=O)C(C)O 46623,N1(C(c2csc(C)c2N)=O)CC(C)CN(C(c2sc([N+](=O)[O-])cc2Cl)=O)CC1C 46624,c1(SC(C)C(=O)NC2CCCCC2NC(=O)CCOCC2CC2)ccc(F)cc1 46625,C1(C(=O)NC2CCC(F)(F)C2)CC(F)(F)CN1S(=O)(=O)CCBr 46626,c1(C(=O)NC2(C)CN(C(c3sc(Cl)cc3Cl)=O)C2)cn2c(n1)CCC2 46627,Cc1nc2ccnn2c(C)c1C(=O)NCC1COCC1NC(=O)CCC(F)F 46628,N(C(=NCCc1cn(C)cn1)N1CCN(C(C)C(F)(F)F)CC1)CCCSC 46629,c1(CC(N2C(C)CC(NC(c3cnc(S)n3C)=O)C2)=O)cnc2c(=O)[nH]ccn12 46630,N1(C(C(CCC)NC(N)=O)=O)CCOC2(CCCN(C(=O)C(O)C(C)(C)C)C2)C1 46631,C(C(C)CC(=O)N1CC=CC1(C)C(=O)NCc1nnn(CC)n1)OC 46632,N1(C(c2n(C)nc(Br)c2)=O)CC(NC(=O)C2CC2)C2(CC2)C1 46633,CC(CCc1ccccc1F)C(=O)NCC1CCCN1C(c1c[nH]nc1Cl)=O 46634,N1(C(Cc2c(C)nsc2)=O)CCC2(C=C(C(=O)NC(C)CCC(C)(C)C)C2)C1 46635,C1(C(N(CCCCNC(c2cc(COC)on2)=O)C)=O)CN(C)CCO1 46636,Cc1nn2c(c1C(=O)NCC1(F)CCN(C(C3(CO)CC3)=O)C1)CCCC2C 46637,N1(C(c2cnc(C(C)C)nc2)=O)CC(NC(c2ocnc2C2CC2)=O)C2(CC2)C1 46638,C1(C(=O)NCCC(C)N(C)C(C2CCOC2)=O)CC(C)N(C)C1 46639,N1(C(c2cnc(CC)[nH]2)=O)CC(CNC(=O)CCn2ccnc2)C(O)C1 46640,c1(C(=O)NCC(C(=O)NC2(C)CCC2)OC)cccc(F)c1C 46641,c1(OC)ncc(C(N2CC(CNC(C3CCC(C)O3)=O)C2)=O)cc1C 46642,c12occc1C(=O)NC2.C(CO)(C(N)=O)NC(COCCSCC)=O 46643,C1(CNC(c2ccc3nn[nH]c3c2)=O)CN(C(c2cc(Cl)no2)=O)CCC1(F)F 46644,N1(C(c2cnc(C(C)OC)s2)=O)CC2C(NC(=O)Cc3cscn3)C2C1 46645,c1(CNC(C(c2cccc(Cl)c2)SC)C)cc(-c2nn[nH]n2)c(F)c(F)c1 46646,CC1(C)CN(C(=O)CCC2CC2(Cl)Cl)CC(CNC(=O)C(=Cc2cscn2)F)O1 46647,C1(N(CC#C)C(c2nocc2Cl)=O)CCN(C(C2(O)CCC2)=O)CC1 46648,N#Cc1ccc(C(c2ccccc2)=O)c(F)c1NC(C1C2CCC1(C(F)(F)F)C2)=O 46649,O=S(=O)(c1ccc(Br)cc1NC1CCCn2ccnc21)N1CC2CCC1C(CO)C2 46650,N1(C(=O)Nc2nnn(C)c2NC2(C)CCCCC2(C)C)CCCC(C2CC2)CC1 46651,c1(C(=O)NCCN(C(=O)COC2CCC2)C2CC2)snnc1CC1CCC1 46652,c1(C(N(CCNC(c2cccc(N(C)C)c2)=O)CC)=O)ccc2nc(S)[nH]c2c1 46653,c1(C(=O)NCCCN(C(C2CCC(C(N)=O)O2)=O)CC)cc(OC)cnn1 46654,N1(C(C(CO)N(C)C)=O)CCOC2CN(C(C3C4CC5C(C4=O)C35)=O)CC12 46655,CC1=C(CNC(=O)NC2(Cc3ccccc3F)COC2)S(=O)(=O)CCO1 46656,N1(C(c2nc(C)sc2C)=O)CCCC(NC(C23CC(C2)C(C(F)(F)F)O3)=O)CC1 46657,N1(C(C(=O)NCCC(=O)OCC)C2CC2(C)Br)CCC(C)(CC#N)C1 46658,C(=O)(C(C(C)C)OC)NCC(=O)OCCC.C1(=O)CC(C)=CCN1 46659,N#CC1(C(=O)NC2CCCCCN(C(c3cccnc3)=O)C2)CC12CCOCC2 46660,c1(-c2cccn(C)c2=O)c(C(=O)O)ccc2c1OC(F)(F)O2 46661,N1(C(CCc2c(C)ncs2)=O)CC=C(CCNC(=O)CCCOC(=O)N(C)C)CC1 46662,C(=O)(CC1COc2cc(O)ccc21)NC(CC(C)(C)C)CO 46663,C(=O)(C1=CCCN(C(=O)Cc2cccc(Cl)n2)C1)NCC(C)(C)CO 46664,c1(C(C(=O)NCc2cccc(Br)c2)N(CC)CC)ccc(Cl)cc1Cl 46665,C1(NC2(c3n(C(C)C4CC4)nnn3)CC3COCC3C2)CN2CCCC2CO1 46666,C=CCC(C)(CC)C(=O)NCC1CCC1C(=O)Nc1ccc(C)cc1CO 46667,C1(O)(CNC(C2(CC=C)CCC2)=O)CC(NC(=O)Cc2nc(C)cs2)C1 46668,C12(CNC(Cc3cc(C)[nH]n3)=O)CC1CN(C(C1(NC(C)C)CC1)=O)C2 46669,CCC(O)C(C)C(=O)N1CCCCC1CCNC(C1CCCCN1CC(F)F)=O 46670,N1(C(=O)NCc2nc(C(=O)OC)sc2)CCC(F)(C#N)C1 46671,CCCCC(CNC(N1CCOCC1)=O)NCC1CCC(NC(=O)CC2CC2)O1 46672,c1(C(=O)NCC(CNC(C(C)C2CC2)=O)O)cc([N+](=O)[O-])cc2c1OCCO2 46673,Cc1cc(C(=O)N(C(CNC(c2cccc(O)n2)=O)C2CC2)C)n2nccc2n1 46674,c1(C(N2C3CC(NC(C=CC)=O)CC2CC3)=O)ccc(=O)n2c1CCC2 46675,Cc1cc(C(=O)NCC(C2CC2)N(C(=O)COC2(C)CCC2)C)n2nccc2n1 46676,C(=O)(C(F)(F)C(C)O)NCC=CCNC(C1CC(C(=O)OC)C1)=O 46677,CC1CCCC(O)(C(=O)NC2CC(NC(c3cc(-c4ccns4)on3)=O)C2)CC1 46678,CC(C)C(O)CC(=O)N(CCC(N1CCCC(C)(N(C)C)C1)=O)C(C)C 46679,C1(N(C(=O)CCC2CCCCO2)CC)CCCN(C(=O)CSc2nncs2)CC1 46680,CC1CC(NC(=O)CCS(N)(=O)=O)CCN1C(C1CC2(C1)OCCO2)=O 46681,C(=O)(C(C)CCCc1cn(-c2ccncc2)nn1)NC(CCC=C(C)C)(C)C(=O)O 46682,c1(CC)cc(C(=O)NCC=CCNC(=O)C(F)(F)c2ccnn2C)oc1CC 46683,Clc1ccccc1OCCn1nnnc1N1CC2(CCO2)C1 46684,C(=O)(C(C)CC(C)(C)C)NCC(C)(C1CCC1)NC(CCc1ccnc(C)n1)=O 46685,N1(C(C=C(C)Cl)=O)CC2COCCC2(NC(c2nc(C)ncc2N)=O)C1 46686,C1(C(N(Cc2cn(CC(=O)NC3(C)CCCC3=O)nn2)O)=O)CCCCC12CC2 46687,c1(C(N2CC(NC(C=CCOCCOC)=O)C(O)C2)=O)cccc2cnsc12 46688,c1(C(N2CC(C(=O)NC3(CO)CCCC3(C)C)(SC)C2)=O)cc2ccccc2[nH]1 46689,c1(C(=O)NCCC(C)NC(CS(CC)(=O)=O)=O)cc2ccccc2nc1C(F)F 46690,C1(C(C)(C)NC(=O)CCCC2CCCO2)CCN(C(C2CCOC(=O)N2)=O)CC1 46691,C1(Cc2onc(CN3C(=O)COCC3)n2)CCC2(CCNC2)CC1 46692,c1(C(=O)NCC(c2cccnc2)NC(CSC(C)C)=O)cn(C)cn1 46693,CCC(CC(=O)NCC1CCN(C(=O)CC2CN(C(C)=O)C2)CC1)C1CC1 46694,CC1OCCC1CC(=O)NOCC(=O)NCC1(CCCO)CC1 46695,C1(CC(=O)N(C2CN(C(c3c(F)ccc(N)c3F)=O)C2)C)CCC2(CCC2)CO1 46696,C=CCCC(F)(F)C(=O)NC1CN(C(=O)Cn2cnnc2O)CC2(CC2)C1 46697,C1(NC(c2cc(SCC)ncc2)=O)CC2CN(C(=O)C=CCO)CC12 46698,C(CCCC(C)NC(c1ccnn1CCCC)=O)NC(C(C)=CC)=O 46699,O(P(=O)(OCC)C1(C)CCCN1C(=O)Nc1nc2cc(Cl)ccc2n1C)CC 46700,CCC(CN(C)C)CC(=O)N(C)CC1(O)CCN(C(c2cncn2C(C)C)=O)C1 46701,N1(C(c2ccccc2)C(=O)OC(C)(C)C)CCC2CC12C 46702,c1(NC2C3CN(C(=O)CCC4CCCC4)CC2C3)cc(=O)n2cc(Cl)ccc2n1 46703,c1(C(N2C(C)CC(CNC(C3COCCO3)=O)C2)=O)ccc2c(c1)CCN2 46704,C1(CN(C(=O)CC(O)c2ccccc2)C)COCCN1C(=O)C=CI 46705,c1(C(=O)NCC2CCC(NC(c3ccnnc3)=O)CC2)ccc2c(c1)COC2 46706,N1(C(c2nnn(CC)c2C)=O)CCCC(C)(NC(=O)CCc2cc(Cl)cs2)C1 46707,c1(OC)ccc(C(=O)NC2CCCC2NC(=O)C(O)CC(F)F)cc1OC(F)F 46708,N1(C(CCC2(C#N)CCC2)=O)CC2CCOC2(CNC(=O)CC2CCSC2)C1 46709,c1(N2CCC(CNC(C3CC4CC3C3CC43)=O)C2)ncnc(Cl)c1F 46710,c1(C(c2nnnn2C(C)C)NC(c2nccn2C)CC)cc(Br)ccc1Cl 46711,C1(NC(C2(C(C)C)COC2)=O)CC(CNC(=O)C(C)CC2CC2)CC1O 46712,N1(C(C(CC)=CC)=O)CC(OC)C(NC(=O)C(O)C2CC2)C1 46713,C1(n2cc(C(C(C)(C)C)O)nn2)CN2CCCN1CC2 46714,N1(C(COCCCOC)=O)CCOCC(C(=O)Nc2cc(Cl)ccc2C)C1 46715,C1(CNC(C2C(N)CCOC2)=O)CCC2(CCCCC2)O1 46716,CC1CCCC1C(=O)NCC(C)(C)CNC(=O)Cc1cnc(C2CC2)[nH]1 46717,c1(C(=O)NCC#CCNC(CN(CCC#C)C)=O)csc(O)n1 46718,Cc1ccc2cc(Cl)cc(C(=O)NCCn3cc(-c4csc(C)n4)nn3)c2n1 46719,c1(C(N2C(C)(C)C(NC(=O)C=CCN3CCCC3)CC2)=O)cc(P(C)(C)=O)cs1 46720,C12(C(=O)NC3CC(CCNC(C4(OC)CCCCC4)=O)C3)CCC(C)(CO1)C2 46721,C1(C(=O)NC(C(N2CCC(CN=[N+]=[N-])C2)=O)C2(C)CC2)CC=CC(O)C1 46722,c1(CCC(=O)NC(CC)CNC(C2CCC2(C)C)=O)ccc(OC(F)(F)F)cc1 46723,N1(C(C2C(C)C2)=O)CCC2(CCCN2C(C2CCC3(CCOCC3)O2)=O)CC1 46724,c1(C(=O)OC)ccc(SC(C2CC2CCCC(=O)N2CCC(CF)C2)=O)cc1 46725,C(=O)(CC(C)C(C)(C)NC(c1occc1C)=O)N1C(C(=O)NC)CCCC1 46726,c1(C(=O)NC2C(NC(C3N(C)CCCC3)=O)CCCC2)cccc(=S)n1O 46727,c1(C(=O)OC)cc(-c2cc(CO)cc(Cl)c2)cn(C)c1=O 46728,c1(C2C(C)C2)ncc(C(=O)N(C)CCOCCCNC(=O)C(C)(C)F)s1 46729,C1(NC(c2cccc(SC)c2)=O)CC2(NC(c3cnoc3C)=O)COC1C2 46730,C(C(=O)N1CCC(NC(C2CC3(CSC3)C2)=O)C(O)C1)(C(C)(C)C)NC(C)=O 46731,N(C1CCCc2c(Cl)ccc(Cl)c21)C(=O)NC1N(CC)CCOC1 46732,C(CC(C(=O)NC(CC1CC1)CC1CC1)NC(=O)CCC1CCC(=O)C1)OCC 46733,C12(C(=O)NCCN(C)C(C3(C)C=CCCC3)=O)CCCC1C2Br 46734,C(=O)(CCCCCn1cnnn1)N(CCCCCNC(=O)CC(C)(C)C)C 46735,C(C(=O)NC(C)C(CO)NC(=O)C1=CCC1)(C(C)(C)C)c1cccc(C)c1 46736,O=C(CC(F)(F)F)NCC1CCCCC1NC(c1ccc(OC(F)(F)F)cc1)=O 46737,N1(C(C(CC)(C)CO)=O)CCC2(CC1)COCC(CNC(C1(C)CCC1)=O)O2 46738,c1(C(N2CCCC(CNC(C3CCS3(=O)=O)=O)C2)=O)ccc(F)c2occc12 46739,C(=O)(C1Cc2ccc(Cl)cc21)N1CCC(CCCNC(C(C)SC(C)C)=O)CC1 46740,C(=O)(C(F)(F)C(C)O)NC1CC(CCNC(c2ccc(CCC)[nH]2)=O)C1 46741,c1(C(N2CCN(C(C3CCC(=O)C3)=O)CC2CC(F)F)=O)coc2c1CCCC2 46742,C1(CNC(C(C)Cc2ccco2)=O)CC2CC2N1C(=O)C#CC(=O)N(C)C 46743,C1(CNC(C(N2CCC(O)(Cc3ccc(OC)cc3)C2)C)=O)CCCCNC1=O 46744,c1(C(=O)NCCCNC(C(C(C)C)CN(C)C)=O)ccc2c(c1)C=CCC2 46745,C1(C)(C(=O)NC2(c3ccccc3)CN(C(C=CC=CCC)=O)C2)COCCO1 46746,c1(C(=O)NCC(C)N(C(C(CC)N2CCCC2=O)=O)C)[nH]c(C)nc1C 46747,N1(C(c2c(OC)n[nH]c2)=O)CCC2(CC2C(=O)NCC(C)(C)CN=[N+]=[N-])C1 46748,C(=O)(C(C)CCCOC(C)=O)NCc1cccc(C(N2CC(CC#C)OCC2)=O)n1 46749,C(CC(C)(C)C)N(CC(=O)NCC1CCCN1C(=O)CCC1CCOCC1)C 46750,c1(C(C(N2CCC(NCC3C(C(=O)O)CC3)C2)=O)O)cccc(F)c1 46751,CC1CC(N(C(=O)CC2CN(C(=O)CC3CCOCC3)CC2CO)C)CCO1 46752,c1(CN2CCC(N(C(C3C(C)CCC3)=O)C)C2)cc(F)c(O)c(F)c1 46753,c1(NC(C2C(CNC(c3c[nH]nc3Cl)=O)CC2)=O)ccc2n[nH]cc2c1 46754,C1(NC(C(N2CC3C(NC(c4n(C)cnn4)=O)(C3)C2)=O)=O)CCN2CCCCC12 46755,C#CCCCC(c1ccccn1)NC(c1cc(-c2ccc(F)cc2)n(C)n1)=O 46756,c1(C(=O)NC2CCN(C(c3cnc(-c4ccoc4)s3)=O)CC2)cnn2c1OCC2 46757,c1(C(N2C(CNC(c3cccc(F)c3Cl)=O)CCC2)=O)cc(F)c(Br)cc1F 46758,C1(CC)CCC(C)CN1C(C1CCN(C(c2cn(CCO)nn2)=O)C1C)=O 46759,CCC(CC(=O)N1CCCC1CNC(c1cc(C)nnc1O)=O)C(C)C 46760,c1(C(=O)NC(c2ccc(CNC(COC)=O)cc2)C)ccc(Br)nc1N 46761,c1(C(=O)NCCC2CC(NC(C(CC)(C)C)=O)C2)cc2c(C)c(Br)ccc2[nH]1 46762,C1(NC(c2cc(C)ns2)=O)CN(C(=O)CCSc2ccccc2)CC1C 46763,C1(NC(c2cnc(O)o2)=O)CCN(C(C2COC(=O)C2)=O)CC1 46764,c1(C(=O)NCCNC(C(C2CCOC2)OC)=O)cn2cccnc2n1 46765,N1(C(CCC#C)=O)CC2(CCOCC2)CC1CNC(c1cnc2sc(C)cn12)=O 46766,c1(CNCC)ccccc1SCCCCCC(F)(F)F.C1(C)C(=O)N1 46767,C1(C)(NC(CC2(C)N(C(c3ccc(CC)o3)=O)CC2)=O)CCCC1C 46768,C1(NC(C(CC)COC)=O)CN(C(c2cnc(OC)nc2)=O)CC1S(C)(=O)=O 46769,c1(CCC(=O)N(C2CCCN(C(C3CCOC3)=O)C2)C)cn2ccccc2n1 46770,C1(CC(=O)NC2(CC(=O)OC)CC2)CC(OC)CN1C(c1ccncc1SC)=O 46771,C1(NC(Cn2cc(CN(C)C)nn2)=O)COCCN(C(C2CCCCC2O)=O)C1 46772,N1(C(C(COC)OC)=O)CCC(C(=O)Nc2cc(OC)cc(O)c2)C(O)C1 46773,Cc1cc(C(=O)NC2CCCCC2NC(=O)C(c2ccc(Cl)cc2)O)nnc1C 46774,CCCCC(CC)C(=O)NCCOCCCN(C)C(C12CC(C(F)F)(CO1)C2)=O 46775,C1(NC(c2cc(C)c(Br)o2)=O)CN(C(=O)CN(C)S(N)(=O)=O)CC1C1CC1 46776,N1(C(c2n(CC=C)ccc2)=O)CCN(C(C2CCCS(=O)(=O)C2)=O)C(C(C)C)C1 46777,Cc1nc(CC(=O)NC2CCC2NC(=O)Cc2csc(Cl)c2)c(C)s1 46778,C#CC1(C)COCCN1C(c1cnn2c1CCC2)C(=O)NCC1CCOCC1 46779,N1(C(c2n(C)nc([N+](=O)[O-])c2)=O)CCCC2(CCCCC2NC(=O)C(Cl)=CCl)C1 46780,CN1CCCC(C(=O)NC(C2CCN(C(c3ccoc3)=O)CC2)(C)C)C1 46781,C1(CC(N2CC=CC(NC(c3c(C)cco3)=O)C2)=O)CCCC(F)(F)C1 46782,CC1=CC(C)C(c2cn(C3(C(=O)NC(CC(C)C)C(N)=O)CC3)nn2)CC1 46783,C1(C(N2C(C)CC(CNC(CCC(C)N(C)C)=O)C2)=O)CC2(CCO1)CC2 46784,C1(C(N(C)CCNC(=O)CSc2cc(Cl)ccc2Cl)=O)CCC2(CCC2)O1 46785,CC1CN(C(=O)C(CC2CC2)NC(=O)CC2C=CCC2)CCS1=O 46786,C1(O)(CNC(c2ccn(CCOC)n2)=O)CCCN(C(=O)C(C)NC(C)=O)C1 46787,C1(N(C)C)CCC(n2cc(CN(C(C3CC(O)C3(C)C)=O)C3CC3)nn2)CC1 46788,c1(C(N(CC(C)OC)C(C)C)=O)cc(CO)[nH]n1.C1(C=O)CN(C(N)=O)C1 46789,C1(N(C(C(C2CC2)OC)=O)C)CCC(NC(c2nnsc2C(F)F)=O)CC1 46790,C1(CNC(C(F)=CCC)=O)CC(C(=O)NCC(C)(C)CSC)=NO1 46791,c1(OC)cccc(C(=O)NC2CCN(C(C3(C#N)CCCO3)=O)C2)c1C 46792,CC1(CC(=O)NCC=CCNC(c2ccnc(O)c2)=O)Oc2ccccc2O1 46793,Cc1ccc(S(=O)(=O)NC(CN(C)C(c2ccoc2C)=O)OC)cc1 46794,C12(C(N3CCC(C(C)NC(=O)C(F)CC4CC4)C3)=O)CC3CC1C2C3 46795,N1(C(c2n(CC)ccc2)=O)CCOC2CN(C(=O)C(c3ccccc3F)C)CC12 46796,CCC(C)C(C(=O)N(C)Cc1nccn1CC)NC(C1CCCSC1C)=O 46797,C(CCC(C)(C)NC(=O)C=C(Cl)Cl)NC(C=CCCC(C)C)=O 46798,c1(C(=O)OCC)cnc(SC)[nH]c1=NCCCN(C(=O)CC(C)(F)F)C 46799,c1(C(=O)NC(CN(C(=O)C(C2CCOCC2)O)CC)C)cc(C(C)C)n(C)n1 46800,c1(C(N2C(C)(CC)CC(NC(=O)CCCCCF)C2)=O)nc2c(s1)COCC2 46801,CN1CCc2cc(C(N3CCC(N(C(=O)C=CS(C)=O)CCO)C3)=O)sc2C1 46802,CC(C)C#CC(=O)NCC1(C(N)=O)CN(C(C2CC(O)C(F)C2)=O)C1 46803,C1(C)(C(N(CCNC(C(C)c2ccsn2)=O)C)=O)CCCS1(=O)=O 46804,C12(CCNC(=O)Cc3ccccc3F)CCC(C1)N(C(c1ns[nH]c1=O)=O)C2 46805,C1(CC(C)NC(C2(CC=C)CCC2)=O)CCN(C(=O)CNC(C)=O)CC1 46806,C12(C(N3CC(SC)C(NC(=O)CC4CCCN(C)C4)C3)=O)CCC(CC1)CC2 46807,C1(CNC(CCSC)=O)CN(C(c2ccn(-c3ccccc3F)n2)=O)CC1C 46808,c1(C(=O)NC(C)CCF)ccc(CNC(C2CC2F)=O)nc1 46809,C1(NC(CCSCCC)=O)CC(C)N(C(=O)C(=O)NCC(F)F)C1 46810,C12(NC(CCCC#C)=O)CCN(C(c3cnoc3C(C)C)=O)CCC1C2 46811,CCCC(CNC(=O)C(CC)OC)C(=O)NC1CCN(CCF)C1 46812,c1(C(=O)NC(CNC)Cc2ccccc2)ccc(C2CC2)cc1OC 46813,C(CC(C(N)=O)NC(C(C)(C)C1CCCC1)c1nnnn1CCCF)OC 46814,C1(NC(C(=O)N(C)C)=O)CC2CCC1N(C(c1ccccc1Cl)=O)C2 46815,c1(C(N(C2CCN(C(=O)C(c3cscn3)N(C)CC)C2)CC#C)=O)ocnc1C 46816,N1(C(C(=C(C)C2CC2)F)=O)CCCC(NC(c2scc(Br)c2Cl)=O)C1 46817,C1(C)(NC(Cc2cc(CC)no2)=O)CCCCC1C(=O)NC1(C(C)(F)F)CC1 46818,S(=O)(=O)(c1sc(O)nc1C)N1C(NC(C2N(C(CC)=O)CCC2)=O)CC1 46819,C=C(Cl)CC(C(=O)N1CCC(F)CC1)C(C)C.C(=O)(C(C)C(F)(F)F)N 46820,c1(NNC(CC(C2CCOC2)CC)CC(C)C)cc(NCC(C)C)nc(C)n1 46821,NC(=O)C(N)CCC(=O)N1CCC2(CC1)CC2C(=O)NC(CC(N)=O)C(=O)O 46822,CC1CCN(C(C2(CC#N)COC2)=O)CC1CNC(=O)CCC(C)(C)F 46823,C1(C(=O)NC2(CNC(Cc3n(C)ncc3)=O)CCC2)CC2CCCCN2C1 46824,Cc1c(C(N2CCC(N(C(=O)Cn3ncnn3)C)C2)=O)ccn1C1CC1 46825,C(c1ccc(OC(F)(F)F)c(O)c1)=CCN1C2CN(C(CCC#C)=O)CC1CC2 46826,CCC(C(=O)OC)C(=O)N1CCCCC1CCNC(=O)CCc1c(C)n[nH]c1C 46827,c1(SCC(=O)NCCCN(C(CCCC#C)=O)CCO)ccc(Br)cc1C 46828,Cc1csc2ncc(C(=O)NC3CN(C(=O)C=Cc4ccoc4)CC34CC4)n12 46829,Cn1nc(I)cc1NC(=O)NCC1(C)CC(F)(F)C1 46830,c1(CCC)nc(C)c(C(N2CC(CNC(C3(C#N)CCC3)=O)CC2C)=O)o1 46831,C1(NC(c2onc(C)c2C)=O)CCCCC12CCN(C(=O)C1=COCC1)C2 46832,c1(C(=O)NC2CCN(C(C3(CC#C)CCOC3)=O)C2)cc(Cl)c(N)cc1OCC 46833,C#CCC(C)(C(=O)NC(COC)C(=O)OC)NC(=O)CN1C(=O)CNC1=O 46834,N1(C(c2n(C)c(S)nn2)=O)CCCN(C(=O)CCCc2ccc(O)cc2)CC1 46835,C1(C(=O)NCC(C)(CO)NC(=O)CN2CC3CC3C2)CCC(=O)NC1 46836,N1(C(COC(C)C)=O)CCCC2CN(C(=O)CN3CCN(C)CC3)CCC12 46837,N1(C(C(CCCC#C)C)=O)CCC2CN(C(c3c(C)[nH]c(C)c3C)=O)CCC12 46838,C(CC(C)C)(C(=O)OC)NC(N(C(CCC)C)C)=O.c12nc(n[nH]1)C2 46839,n1(CC)nc(C(N2CC(NC(=O)CCc3ncccn3)CC2C)=O)cc1O 46840,N12CC3CC1C3C2=O.CC1CCOC1c1cn(CCN(C)CCS(C)(=O)=O)nn1 46841,c1(CC)nn(C)c(C(=O)NCC2CCN2C(c2cc(C(F)(F)F)[nH]c2C)=O)c1Cl 46842,Cc1nc2ccnn2cc1C(N1CC(NC(=O)C=CCF)C(C)C1)=O 46843,c1(C(=O)NC23CC(NCc4cc(Br)cs4)(C2)C3)cc(Cl)cnc1O 46844,c1(C(=O)NCCC(CCNC(C2CC(C)C2)=O)C)cc(N)cc2c1OCCO2 46845,c1(N(CC(C)NC(CCc2c(C)cccn2)=O)C)ncc2c(n1)CCCCC2 46846,N1(C(c2ccn(C)c2)=O)CCC(NC(=O)CC2CCCCC2O)CC(C)(C)C1 46847,C1(NC(=O)CCCn2ccccc2=O)CN(C(=O)Cn2nccn2)CCC1CO 46848,c1(C(=O)NC2CN(C(C3C(c4ccc(OC)cc4)C3)=O)C2)nc2cccnc2s1 46849,C(=O)(C(O)CCCNC(=O)CC1CCOC1(C)C)NCC1CC(SC)C1 46850,S(=O)(=O)(c1cccc(Cl)c1Cl)N1CC2(CC(C(=O)Nc3cc(I)ncn3)C2)C1 46851,Cc1c(C(=O)N(CC(C)NC(=O)CCC=CBr)C)ccn1C 46852,N1(C(CN(C(C(c2ccn(C)n2)C)=O)C2CC2)=O)CCOC(C2(C)CC2)C1 46853,c1(CC)ncc(C(=O)NC2(CCNC(=O)CN3CC4CC4C3)CCCC2)c(O)n1 46854,c1(C(=O)NC2CCN(C(C(F)=CC)=O)CC2(C)C)cc2c(nc1O)CCCC2O 46855,Cc1nnc(N(c2ccnn2C)C(=O)CC2(C)CCCC2)nc1C 46856,c1(NC(c2n(CC)nnn2)c2ccccc2)cc(SC)ccc1OCC 46857,N1(C(C2(CC(C)=O)CCCC2)=O)C2CCC1C(CNC(c1cc(C)[nH]n1)=O)C2 46858,c1(CC(=O)NCC2(CCOC)CC2)cc(C(=O)NCCOCCOC)on1 46859,c1(C(N2CC(NC(C(C)(C)C3CCCCO3)=O)C(O)C2)=O)cccc(Cl)c1Cl 46860,CCCC(C(=O)NCC(CO)NC(c1c[nH]nc1C1CC1)=O)N(C)C 46861,CCCCC(O)C(C)C(=O)N(CC(=O)NCC1CC2C=CC1O2)C 46862,c1(C(=O)NCC2C(NC(=O)CCN3CCCC3)C2)cnc(C(F)(F)F)c(F)c1 46863,N1(C(C2CCC(=C)CC2)=O)CCCC(C)(NC(=O)CC2CCC2(F)F)C1 46864,c1(C(=O)NC2(C(NOCC(C)(C)O)=O)CC2(C)C)cnn2c1CCC2 46865,CN1CC2CCCC(C1)N2C(c1sccc1CNC(C1CC1C#N)=O)=O 46866,c1(OCC)ccc(C2CCN(C(=O)C(N3CCOC(CN(C)C)C3)=O)C2)cc1 46867,C(=O)(C(F)CCCCCCCC)NC1CCCN(C(CC2CC(=C)C2)=O)C1CC 46868,c1(CNC(c2nccc(OC)c2)=O)nc2c(s1)CCN(C(C1CC1Cl)=O)C2 46869,C1(C(N(CCCNC(CC(C=C)(C)C)=O)CC)=O)CCC2(CC1)CNC(=O)C2 46870,c1(C(N(C2CCN(CC(=O)NCCCC)C2)C)=O)c[nH]c2c(Cl)cccc12 46871,C1(C2CCC2)(CNC(C2C(=C)CC2)=O)CCN(C(c2cnc(O)c(C)c2)=O)CC1 46872,C1(CNC(c2ncn(C)c2)=O)C2CN(C(c3ccccc3C3CC3)=O)CC12 46873,C(CCC(C)CC(=O)NCC1CCN(C(C2COC(=O)N2C)=O)C1)=C(C)C 46874,c1(CN2C3C(C(=O)NCc4cccc(OC)n4)C(C3)C2)cc2ncccc2[nH]1 46875,CC(CCC(F)(F)F)(C(=O)O)NC(=O)Nc1ccc(CSc2ccccc2)cc1 46876,CCCC(CCCNC(=O)Cc1nonc1C)NC(c1c(C)nn(CC)c1C)=O 46877,N(C(=NCCC(O)C(F)(F)F)NCC(C)(C)C1=CCOCC1)CCOCC=C 46878,c1(N2CCN(CC)C(C)(C)C2)nc(=NC)[nH]c(=NCCCC(=O)N2CCCC2)[nH]1 46879,C(=O)(CCC(=O)c1cccs1)NCC(CNC(c1c(COC)ccs1)=O)(C)O 46880,C1(NC(c2sccc2F)=O)COC2(C1)CN(C(c1onc3ccccc13)=O)C2 46881,C12(C(=O)NC3CC(CNC(C(F)(F)C4(OC)CCC4)=O)C3)CCC(OC)(CO1)C2 46882,N1(C(CC(CC)C2CC2)=O)CCN(C(c2cc(SC(F)(F)F)c[nH]2)=O)C(CC)C1 46883,c1(SC)cc(C(N2CC(N(C)C(c3cc(C#N)cs3)=O)C2)=O)ccc1[N+](=O)[O-] 46884,C=CC(C)(CC)C(=O)N1CCCC1C(=O)NC1CCOC(C)(C)C1 46885,c1(N(C)C)cccc(CNC(c2ccn(C3CCNCC3)n2)=O)c1 46886,c1(C(=O)NC2C(NC(C3N(C)CCC3)=O)CC2)cc(C2CC2)nc2c1cnn2C 46887,N1(C(c2c(C)cnn2C)=O)CC(C)(C)CC1CC(=O)NC(c1nc[nH]n1)C 46888,CCCCCCCCC(=O)NC(C)(C)CC=CC(=O)NCCO 46889,C1(NC(CS(=O)(=O)NCC)=O)CCCC12CN(C(=O)C=Cc1ncc(C)[nH]1)C2 46890,C(=O)(C1=NNC(=O)CC1)NC1CCC(NC(c2cnc(C(C)O)s2)=O)CC1 46891,C(=O)(C1=CCC(C)(C)CC1)NCC1CCC(CNC(c2ncn(CC)n2)=O)CC1 46892,c1(NC(C2N(C(c3cc(CC)[nH]n3)=O)CC(O)C2)=O)ncc(Br)nc1C#N 46893,C=C(C)C(CC(=O)NCCCNC(=O)C(c1cc(F)cc(F)c1)O)OCC 46894,C(CCCO)N(C(=O)C(C1CC1)N(C(=O)C=CC1CC1)C)C(C)OC 46895,c1(CNC(COCC(=O)NC)=O)ccc(C(=O)NCC2(C)CC=CCC2)cn1 46896,C#Cc1ccc(Br)c(C(=O)NCC2CN(C(c3cc(C)oc3C)=O)C3CC23)c1 46897,c1(OCC(=O)NC(C)CNC(C2CC2Br)=O)cc(C(F)(F)F)ccc1O 46898,C1(C(=O)NCc2c(COC)cccc2)CCCCC1(C)NC(C1CCC=CO1)=O 46899,C(=O)(C(C(=O)NC(C(=O)N(CC(C)(C)O)C)C1(C)CC1)OC)OC 46900,C(C(O)(C(F)(F)F)c1nccn1C)NC(C1(CNC(CC(=O)OCC)=O)CC1)=O 46901,C(=O)(C(F)C(F)(F)C(F)(F)F)N1CC2(CC(NC(=O)CC3CC34CC4)C2)C1 46902,C(=O)(C1OC(=O)c2ccccc21)N(CCCNC(C1CCC=CCCC1)=O)CC 46903,N1(C(c2cn(CCOC)nn2)=O)CCC(C)(NC(=O)C(F)CC2CC2)CC1 46904,N1(C(C2(F)CC2)=O)CC2CCC(C1)N2C(C1C2CC2C2CC12)=O 46905,c1(C(C(=O)NCCCN(C(Cc2c(C)cc(C)s2)=O)C)O)ccc(Cl)c(Cl)c1 46906,C1(=CCNC(C(C)CO)=O)CCN(C(=O)C(c2ccccc2)N(C)C2CC2)CC1 46907,C1(NC(CC2CN(C(C(=O)NCC)=O)CC2C)=O)CCN(C)CC1C 46908,CCC(CC)(CC)C(=O)NCCN(CCc1ccccc1)C(c1cnsn1)=O 46909,N1(C(C(=O)OC2N(C)CCC2)=O)CCn2c(-c3ccc(F)cc3)nnc2C1 46910,CC1CN(C(C2(CF)CC2)=O)CCCN1C(=O)CC1CCCNC(=O)C1 46911,C(C1CC(C)(C)Oc2ccccc21)NC(C(CC)(C)C(F)F)=O 46912,c1(C(C)=O)cc(C(=O)NC2CCC(CNC(=O)Cn3cc(Cl)nn3)C2)ccc1C 46913,CCCC(C(O)C(=O)NC(C(C)C)C1CCC1)NC(=O)CCCn1ccnc1 46914,N1(C(c2cncc(C)c2C)=O)CCN(C(C2CCCN2C(C)C)=O)CC(CO)C1 46915,c1(C(N2C(CN(CCC#C)C)CCCC2)=O)cc(C)c(Cl)c(C)c1 46916,c1(CC)cccc(CS(=O)CC(=O)OC)c1.c12ccc(cc1)CN(C)CC2 46917,c1(CNC(C2(CC)CCCCC2)=O)ccc2c(c1)CN(C(=O)CCC(C)SC)C2 46918,c1(C(N2CC(CC=C)(C(=O)NCC(C)CCCO)C2)=O)nc(C)ccc1C 46919,CCC(C)C(C)C(=O)NC(C)(C)CN1CCN(C(c2ccnc(OC)c2)=O)CC1 46920,N1(C(Cc2cc(CC)no2)=O)CC2CC2(CN2CCCC(C(=O)NC)C2)C1 46921,c1(C(=O)NC2CN(C(c3c(OC)ccs3)=O)CC(O)C2)nccn2ccnc12 46922,C1(CNC(CCN(CC=C)C(C)=O)=O)CCCN(C(=O)CC2(C#N)CCC2)C1 46923,N1(CC)CCCC(C(=O)NCC(C)(C)CN(C)C(C2CCNC(=O)C2)=O)C1 46924,C(CN=[N+]=[N-])(C(=O)NCC(C)S(N)(=O)=O)NC(C(N1CC(C)C1)C)=O 46925,C(CCCSC)(C(=O)NCCS)N(CCN(C)C)CC.N1(CC)CCCCC1 46926,C1(NC(C(C)SCc2ccccc2)=O)CCCC(NC(c2ccnnc2O)=O)C1 46927,c1(C(N(C(c2cn(C(CC=C)CC)nn2)C)C)=O)cc2c(s1)CCC2 46928,c1(CC(=O)OC)ccnc(NC2CCN(C(C3CCCN3C3CC3)=O)C2)n1 46929,C1(C(N2CCSCC2)=O)Cc2nccnc2CN1C(=O)C1=NOCC1 46930,C(=O)(C(C)(C)CC(C)(C)C)N(c1ccccc1)CCNC(C1C(C)C1)=O 46931,N1(C(CCN(CCCCC)CC)=O)CCCCC1CCNC(C1CC2(CC2)C1)=O 46932,C(=O)(C(CC(C)C)ONC(=O)CCC1CCOC1)N(CC(=O)OC)CC=C 46933,C(=O)(CCCCCn1cnnn1)NC1CCCN(C(c2ccc(OC)cc2)=O)C1 46934,c1(C(N(CCN(C(=O)C(O)C(C)C)CC)CC)=O)cc(P(C)(C)=O)ccn1 46935,c1(C(=O)NCC(C)CN(C)C(C2(N(C)C)CCC2)=O)occc1C1CC1 46936,N1(C(CC2C(C)(C)C(O)C2)=O)CC(NC(c2ncccc2Cl)=O)CC2(CC2)C1 46937,CC1CCN(C(=O)CN(C2CCC2)C)C1C(=O)N(C)Cc1ccc(F)cc1 46938,c1(C(=O)NC2CC(C)(C)CN(C(=O)CCF)C2)cc(Br)c2nccn2c1 46939,C(=O)(CCCC(=O)N1CCOCC(CNC(=O)CNS(=O)(=O)C2CC2)C1)NCC 46940,c1(NC(C2OCCC2(C)C)=O)ccc(F)c(F)c1.CC1C(=O)N1.C1CNC(=O)O1 46941,c1(C(=O)NC2C(C)N(C(c3cccc(Cl)n3)=O)CC2)c(F)ccc(F)c1N 46942,C1(CNC(c2c(C)csc2)=O)C(C2CC2)CCN1C(=O)CC(C)C(F)(F)F 46943,C1(C(=O)OC)CCC12CC(C(=O)NC1(c3ccc(F)cc3F)CC1)C2 46944,c1(C(N2CCC(NC(CC(CC)C(C)C)=O)C(O)C2)=O)cccc2c1NCCC2 46945,C1(C2CCN(C(c3ns[nH]c3=O)=O)C2)CCCCN1C(c1cscn1)=O 46946,CN(C1CN(C(=O)CCCC2CCOCC2)CCc2ccccc21)C(=O)C1CC1 46947,C(=O)(C(C)(C)CC(C)(C)C)NCCC1(CNC(c2nccc(C)n2)=O)CC1 46948,CCC(N=c1[nH]c(Cl)nc2c1CCOC2)C=O.OC 46949,c1(C(=O)NC2CCC(C)CC2)nc[nH]c2nccc1-2.C1(CN)CCCO1 46950,C(=O)(C(F)n1ccnc1)N(C(C)C(=O)NCCOc1ccoc1)CCC 46951,C1(CNC(=O)C#CC2CC2)COCC2(CCN(C(C34CC(F)(C3)C4)=O)C2)O1 46952,N1(C(C2(CCN=[N+]=[N-])CC2)=O)CC(=O)NCC1C(N1CCNC(=O)C1)=O 46953,c1(C(=O)NC(CC(C)NC(c2c(NC)cccc2)=O)C)c(F)cc(C)cc1Cl 46954,C(C)(C(C)C(=O)NCC1(C2CCC2)CC1)NC(C(C=C)C)=O 46955,c1(C(=O)NC2CCC(CNC(C(N)=O)=O)C2)cccn2c(CC(C)C)nnc12 46956,N1(CC)CC(NC(c2nc(C)c(C)s2)=O)C(C)C1.n12cc(nn1)CN1CC2C1 46957,C1(C(N(C2CCN(C(=O)Cn3nccn3)CC2)C)=O)CCCCNC1=O 46958,c1(NC(C2CC2Cl)=O)cccc(Oc2cccc(F)c2)c1 46959,Cc1cn2c(n1)C(C)N(C(=O)CC1CCC3(CN(C(=O)OC(C)(C)C)C3)O1)CC2 46960,c1(C(=O)NC2(CO)CCN(C(c3cc(OCC)no3)=O)C2)cnn2ccsc12 46961,N1(C(C(n2cc(-c3nc(Br)nn3C)nn2)C)=O)CCCN(CCO)CCC1 46962,N1(C(CCCC=C)=O)CCC(C)N(C(C2CC(C)(C)CN2C)=O)CC1 46963,C1(CN(C(=O)C(C)(C)C(=O)NC)C(c2cccc(OC)n2)=O)CCCC(C)CC1 46964,c1(C(N2CCC(C)(CNC(CN3CC(CC)C3)=O)C2)=O)ncc(Br)cc1F 46965,n1(CC(=O)N(C)CC2CCN(C(=O)C=Cc3ncc[nH]3)C2)cc(C#N)cn1 46966,c1(OC)cc(F)cc(C(=O)NC(C)(C)CNC(C2(C)CC(F)C2)=O)c1N 46967,c1(C(=O)NC(CN(C(=O)CCc2cccnc2Cl)CC)C)ccc(Cl)c(C)c1O 46968,N1(C(c2[nH]nc(OC)c2Cl)=O)CC(NC(C2(C(C)C)COC2)=O)CC12CCOC2 46969,CC(C(=O)N1CC(C(C)NC(=O)CSCc2ccccn2)C1)C(C)(C)C 46970,c1(NCC2CCCN(C)C2)cccc(S(=O)(=O)NCCC2CC=CCC2)n1 46971,C(CCCC(CO)NC(=O)C(C(C)C)NC=O)NC(Cc1c(SC)cccc1)=O 46972,N1(CCNC(=O)NCC(c2cc(-c3ccccc3)no2)O)CCOCC1 46973,Cn1nc2c(cc1=O)CC(C(N1CCNC3(CC3)C1)=O)CC2 46974,c1(CNC(CCn2cc(C3CCN(C)C3)nn2)=O)ccc2c(n1)OCCO2 46975,C#Cc1ccnc(C(=O)NC2CCCC(C(=O)NC3CC4CC4C3)C2)c1 46976,c1(C(C(=O)NC(C)CCCNC(=O)C=CC2CCC2)O)c(F)cccc1Cl 46977,CC1CN(C(CCc2ccc(Cl)cc2)C(=O)NC)CCN1Cc1ccc(F)cc1 46978,C1(CNC(=O)NC(c2ccc([N+](=O)[O-])cc2)CC)CC(C)(C)CCC1O 46979,C1(CNC(Cc2c(C(=O)OC)scc2)=O)CCN(C(=O)C(c2cccnc2)O)C1 46980,CC1CCCC1CC(=O)NCCOC1CCN(C(=O)C(c2ccc(Cl)s2)=O)C1 46981,c1(C(=O)NCC2(CC)CN(C(=O)C(O)CC(N)=O)C2)cc(OC)c(C)c(OC)c1 46982,C1(OC)CCC(CNC(=O)C(=O)OC2CC(COC)(OC)C2)CC1 46983,C(=O)(C1Cc2c(Cl)cccc21)NCCCCNC1(S(N)(=O)=O)CC1 46984,c1(CC)c[nH]nc1C(=O)NC1CC(CCNC(c2cnn(CCN(C)C)c2)=O)C1 46985,C(C)(C)(CC(=O)N(CCC(=O)NCc1cc(C)ns1)CC1CC1)OC 46986,C1(NC(C2C(C#N)C2)=O)CCN(C(c2cnc3n2CCS3)=O)CC12CCC2 46987,c1(C(N2CC3CN(C(CN(C)CC)=O)CC3C2)=O)cc2c(F)ccc(F)c2[nH]1 46988,N#Cc1c(F)ccc(-c2cn3cnc(C(=O)NCC(O)CO)c3s2)c1F 46989,CC1(NC(c2cc(-c3ccoc3)on2)=O)CCN(C(=O)CCC2CCC(=O)C2)C1 46990,c1(-c2cnc(OC)c(CN3CCC4CCCC34)c2)cc2cc[nH]c2cn1 46991,N1(C(C(=O)NCCC2(C)CC2)CC2CC2(Cl)Cl)CC2CCCCC12C 46992,C1(NC(=O)COC2CCOCC2)CC(NC(=O)COCC(=O)O)C12CCC2 46993,N1(C(c2c(C)c(C3CC3)on2)=O)CCC2C(NC(=O)CCC(=O)N(C)C)C2CC1 46994,C1(Nc2nccc(C)n2)CC(NC(=O)CCc2ccon2)C12CCOCC2 46995,N1(C(CC=C(C)C)=O)CCC(C2(NC(=O)Cc3nnnn3CC3CC3)CC2)CC1 46996,c1(C(N2C(Cn3cc(CC=C)nn3)C(C)(C)C2)=O)cc(OC)cc(Br)c1C 46997,CC(C)CCC(C(=O)NCC1CCSC1)NC(C1CC2(CCCO2)C1)=O 46998,C1(CC(=O)NC(COCC)C(=O)NCCC(=O)N(C)CC)CC=CCN1C 46999,c1(C(=O)NCC2CC(C)N(C(c3cccc(CO)c3)=O)C2)ccc(Cl)c(C#N)c1 47000,c1(CC)cscc1C(=O)NCCC1(CNC(=O)CCCc2ccc(C)s2)CC1 47001,c1(C(N2C(Cn3cc(C(CC)=O)nn3)CCCC2)=O)nc(C)nc(C)c1F 47002,c1(CNC(=NCC=C)NC(CO)CCF)c(F)cc(F)c(F)c1F 47003,C1(C(=O)NCC2N(C(C(CC)C(C)C)=O)CCC2)(OC)CCCC(C)(C)C1 47004,CCC(Cc1cccc(F)c1)N=c1[nH]c(Cl)nc2c1CCC2 47005,Cn1c(C(=O)NCC2COCC2NC(=O)Cn2ccc(C(F)(F)F)n2)nnc1S 47006,N1(C(CCCNC(=O)OC)=O)CC(C)(C)CC1CNC(c1sc(C)c(C)c1C)=O 47007,C(=O)(CC1OB(O)c2ccccc21)N1CCC(C)C(NC(c2ncnn2C)=O)C1 47008,c1(OC)ccc(CN2CC3C(CNC(=O)C4=COCC4)C3C2)cc1C(F)(F)F 47009,c1(C(N2C(CNC(C3C(C#C)C3(C)C)=O)CC(C)(C)C2)=O)cc(F)c(F)cc1F 47010,C(=O)(CN=c1cc[nH]cc1)N1CC=C(C(=O)N2C(CC)CC(O)C2)C1 47011,c1(C(=O)NC2C(CNC(COC3(C)CCC3)=O)C2)cc2ccc(O)nc2s1 47012,C1(c2n(C)ccn2)CN(C(=O)CC2CCC2)CC1NC(=O)CCC1CCOC1 47013,c1(C(=O)NC2CC(NC(C(COCC)(C)C)=O)C2)ccnc(O)c1Br 47014,CCCCCCCC(O)CC(=O)N1CCNC(C(=O)NC2(CC)CCCCC2)C1 47015,CCC(CC)CC(=O)N1CCC(NC(=O)C(O)CC(N)=O)C1C(C)(C)C 47016,c1(C(=O)NCCCOCCNC(C(COC)C)=O)cccc2c1OCO2 47017,C12(CNC(c3c(CSC)cccn3)=O)CCC(CC1)N2C(C1C=CCC1)=O 47018,c1(OC)ccc(F)cc1C1CCCN1CCCCOCCCCCC(C)C 47019,C1(C)(CC)CC(NC(=O)CC2CCCCC2)CN1C(=O)CC1(OC)CCOCC1 47020,CC(CC(=O)NCCC(=O)NC1(C)CCC(=O)NC1=O)C(F)(F)F 47021,N1(C(C(CC(=C)Cl)NC(=O)COCC2CC2)=O)CCC2C(CCN2C)C1 47022,CCC(CC(C)C)C(=O)N1CC(CN=c2nc[nH]s2)C(C)(C)C1 47023,C1(NC(CCCC)=O)CC2CCC(C1F)N2C(c1ccc2c(c1)CCN2)=O 47024,C(=O)(C1=CC2(CCNC2)C1)N1CCC(NC(CCOCC)=O)CC1 47025,C12(CNC(c3c(C)ccnc3O)=O)CC(CCO1)N(C(=O)C(CO)C(F)(F)F)C2 47026,c1(CC)ccc(CNC(N2CC(N(C)C)C2)=O)cc1F 47027,N12CCC(O)(C1)C2=O.N1(CC(=O)Nc2cc(C)ns2)C(=O)CSC1=S 47028,c1(C(N2C(C)(CNC(C3CC(C)OCC3)=O)CCC2)=O)cn2ccccc2n1 47029,N1(C(CNC(c2n[nH]cc2Cl)=O)=O)CCN(C(=O)C(=Cc2c[nH]cn2)F)CC1 47030,c1(OC)cc(C(N2CCC(C)(NC(=O)CC3CCC3(C)C)C2)=O)ccc1F 47031,O(N=C(C(=O)N1CCCC(N(C)C(C)=O)C1)c1cc[nH]n1)CC(=O)OCC 47032,C=CC1(c2cn(CCCCO)nn2)COCCN1C(C1(CC(C)C)CCCC1)=O 47033,C1(NC(C(C)Cn2cccn2)=O)CN(C(c2ccc(F)c(I)c2)=O)CC12CC2 47034,c1(CC)sc(C(=O)NC(C)C(CO)NC(=O)CCC(C)N(C)C)cc1C 47035,C1(NC(c2ccc(Cl)nn2)=O)CCCN(c2ccccc2)C1 47036,C1(NC(c2cnoc2)=O)CCC2CN(C(C3CC3(F)F)=O)CCC2C1 47037,c1(OC)ccc(CC(N2CC(CNC(C3(C)CC3)=O)C(F)(F)C2)=O)cc1Cl 47038,C(CNC(C1CN(C)C(=O)N1)=O)(CC(=O)NC1(CO)CC(C)C1)OC 47039,N1(C(c2ccc(OC)s2)=O)CCC(NC(c2ccn3nccc3n2)=O)C2(CC2)C1 47040,[N-]=[N+]=NCCCCCC(=O)NCC1CCC(NC(c2ccc(C(N)=O)o2)=O)C1 47041,CC1(C)CCC(C(=O)NCC2CN(C(c3ccc(CO)nc3)=O)CCO2)CC1 47042,CCC(C(=O)NCCC(F)Cn1cc(-c2ccnc(C)c2)nn1)C(C)(C)CC 47043,C1(O)(CNC(C2(C#C)CC2)=O)CCCN(C(=O)C(C)NC(c2ccoc2)=O)CC1 47044,C(CC1c2ccccc2CCN1C(=O)C(O)C(C)C)NC(C(Br)=C(C)C)=O 47045,C(=O)(CCCC(=O)N(C)C)NCCN(C(CSc1nc(C)[nH]n1)=O)CC(C)O 47046,CCC(C)(CCC(C)C)C(=O)NC1COCC1NC(c1cncc2nc[nH]c12)=O 47047,CC(O)CCCC(=O)N1CCCC(C2CCCC2NC(c2cnc(F)c(Cl)c2)=O)C1 47048,C=C(C)CCCC(=O)N(C1CCN(C(c2ccncc2N)=O)CC1)CCCC 47049,CC(C)(C(=O)N1CCC(Oc2ccccc2C(F)(F)F)CC1)S(C)(=N)=O 47050,c1(CN(C2CC2)Cc2cccc(-c3c(O)cccc3F)c2)cnn2c1CCCC2 47051,CC1=C(C(=O)N2CCN(C(c3cscn3)=O)C(CCO)C2)CCS1(=O)=O 47052,S(=O)(=O)(c1cn(C)c(C)n1)NCC(N1CC2(C(NC(C=NOC)=O)CC2)C1)=O 47053,Cc1c(C(=O)N(C)CC2CCCCN2C(=O)CCc2cc[nH]n2)nn(C)c1N 47054,N1(C(C(C=C)(C)O)=O)CCC2(CC1)CC(NC(c1c(C)cc(C)nc1C)=O)C2 47055,C(CCCCC(=O)N1CCCC1C(C)(C)O)N(C(C(C)CC1CCC1)=O)C 47056,CC1COC2(C1)CN(C(=O)C(C1CC1)NC(c1nnc(O)nc1O)=O)C2 47057,N12CCCC1CCOCC2=O.CCCCCOC(=O)CCOC1CCC1 47058,c1(CCC(=O)N(C2CCN(C(c3cc(C)c[nH]3)=O)CC2)CC)cc(F)ccc1F 47059,CC1(C(=O)NC2CC(C)(NC(=O)C3=CCCOC3)C2)CCC2CC2C1 47060,C1(C(N2CC3C(CNC(c4cccnc4O)=O)(CC3)C2)=O)CN2CCCC2CO1 47061,c1(OC)cc(C)sc1C(=O)NC(C1CN(C(=O)CCCC2CCCC(=O)N2)C1)C 47062,C(=O)(CCCCCNC(=O)CC1CC(F)CN1C(c1cc(O)nc(Cl)c1)=O)OC 47063,c1(OC)c(C(=O)NCC(O)CN(C)C(c2cnc(Cl)s2)=O)csc1C 47064,c1(SC)c(C(=O)NC2COCC2CNC(C2Cc3cscc3C2)=O)cccc1F 47065,C(=O)(C(C#N)C(C)(C)C)N1CCC(CNC(CSCCC)=O)(OC)C1 47066,C1(C(=O)NCCNC(C(C)NC(=O)CCOC2CC2)=O)(CO)CC=CC1 47067,C(c1ccc(F)cc1F)=CC(=O)NCC1(OC)CCN(C(C2COC(=O)N2)=O)C1 47068,C(=O)(C(C1CC1)NC(C1(C)CC1)=O)NC.c1(CCNC(=O)CO)cccs1 47069,C1(NC(c2ccc(NC)nc2)=O)CCC(C)N(C(=O)CCSC)C1 47070,S(=O)(=O)(c1ccc2nc(C)oc2c1)NC1C(c2n(CC)ncc2)CCCCC1 47071,C(=O)(C(O)C(F)(F)F)N1CC(O)(CCNC(c2ccc(C#C)o2)=O)C1 47072,C(CN=c1[nH]c(=NCc2cnc(O)[nH]2)c2sccc2[nH]1)C1C(C)C1 47073,C(C(=O)N1CCCc2nccn21)C1N(C(CNC(C)=O)=O)CC(C)(C)C1 47074,c1(-n2cc(CCCNC(C3C(C(=O)OC)(C(C)C)C3)=O)nn2)cccc(C)c1Br 47075,C(C)(N=c1nc(Cl)[nH]c(C(C)C)c1C#N)C1N(C(C(c2ccc(C)o2)C)=O)CCC1 47076,C12CC=CCN1C2=O.C(=O)(C(C)N=[N+]=[N-])NCC(N1CC(OC)C1)=O 47077,C1(NC(c2c(C)nc[nH]2)=O)CC12CC(NC(=O)C(O)C(C)C)C2 47078,Cc1csc(=NCC(=O)N2CC3C(CNC(C4(C)CNC(=O)C4)=O)C3C2)[nH]1 47079,C1(NC(C2(CC#C)CCCC2)=O)CCN(C(c2cc(SC)oc2C)=O)CC1F 47080,c1(OC)ccc(CO)cc1.C1(C(N(CCC(=O)N2CC(O)C2)C)=O)CC1C1CCC1 47081,N1(C(CC(=O)OC)=O)CC2CC1C2NC(c1nscc1Br)=O 47082,C1(NC(CC(CC)OC)=O)CC(OC)CN(C(=O)CCCn2c(C)csc2=O)C1 47083,N1(C(Cc2ccn(CC)n2)=O)CC2(CCC(CNC(=O)CCn3cccn3)O2)C1 47084,CS(=O)CCCCNC(C1(CNC(C2CCOC2)=O)CC=CC1)=O 47085,C#Cc1cnc(NCC(CNC(=O)C(c2ccccc2C)C)CO)nc1 47086,c1(CC(=O)NCC2N(C(C(C(C)C)F)=O)CCCC2)ccc(C(F)(F)F)c(F)c1 47087,C(C1=CCN(C(c2ccnc(C(N)=O)c2)=O)CC1)NC(C(CC)NC(N)=O)=O 47088,C(C(C)C(F)C(=O)Nc1cccc(Cl)c1)NC(c1c(OC)nn(C)c1)=O 47089,Cc1ccnc(C(=O)NCCNC(=O)Cc2conc2C)c1Br 47090,C(CCC(O)C(=O)NC(C)C(O)C(F)F)NC(COCC)=O 47091,C1(CNC(CCN(C(=O)CCSCCC)CC#C)=O)CC2(CCCO2)C1 47092,N1(c2n(Cc3nn(C)c(Br)c3)nnn2)CCC2(CCCCOC2)CC1 47093,Cc1cc(C(N2CCSCC2C(=O)NC2CC(O)C2O)=O)cnc1C 47094,C(C(C)CC(=O)NCC1(F)CN(C)C1)NC(c1cn(CC)nn1)=O 47095,C1(CC#C)(NC(=O)C(CC2CC2)NC(C2CCC(=O)NC2)=O)CCOCC1 47096,c1(NC2CC3CN(C(CN4CCC(C)CC4)=O)C(C2)C3)ncnc2cccnc12 47097,C1(CC(=O)Oc2ccccc2)CCN(CCC2(C(F)F)CC2)C1 47098,CCCCCCCCC(C)CC(=O)CC#N.C1CCC1 47099,n1(C(C)CC(=O)NC2CCOCC2NC(=O)C2=CSCS2)cnc2ccccc12 47100,C(=O)(C(C)P(C)(C)=O)N1CCC(N(C(CC(C)OC)=O)Cc2ccccc2)CC1 47101,c1(C(=O)NCC2(O)CC(CNC(C=C(CC)C)=O)C2)cc(C)c(CO)cn1 47102,C1(CC(N2CCC(NC(c3cn(CCOC)nc3C)=O)C2)=O)CC2C=CC1CC2 47103,N(C)(S(=O)(=O)N(C)C)CC(N1C(CN(C(c2ncn(C(C)C)n2)=O)C)CCC1)=O 47104,Cc1cccc(N)c1C(=O)NC(C1CCCCN1C(=O)CCNC(N)=O)C 47105,c1(N(CCNC(CCC(C)(C)F)=O)CC2CC2)ncc(Br)cc1C#N 47106,CC(C)CCCC(=O)NCC(CC(=O)Nc1cscc1C1CC1)C1CCC1 47107,C(=O)(CC(O)CC1CCCCC1)N(CC(C)NC(c1cc(Br)co1)=O)C 47108,N1(CC)CCCN(C(=O)CONC(C2CCOC(NC(=O)NC)C2)=O)CC1 47109,CCC1=NOC(C(=O)NCC=CCNC(=O)CC2(C3CC3)CC2)C1.CC=O 47110,c1(C(N2CCCC3CNCCC3C2)=O)c[nH]c2ccc(F)cc2c1=O 47111,N1(C(c2c(OC)ncnc2C)=O)CCC(C)N(C(c2cc[nH]c2)=O)CC1 47112,Cc1ncc(C(N2CC(C(=O)NC(C)(C)CO)C3(CC3)C2)=O)cc1C#N 47113,C1(CNC(c2c(C)nc(O)[nH]2)=O)CC2CCCCC2N1C(C1CCSC1)=O 47114,C1(C(=O)NC2CCCCN(C(c3ccc(Cl)cc3)=O)C2)CC2CCCCCC12 47115,C(CC(C)C(=O)NC(C)(CC)CCNC(=O)CCc1nc(C2CC2)no1)=CC 47116,CC1CCN(C(=O)CN2CC3CC3C2)CC1CNC(=O)CNS(=O)(=O)C1CC1 47117,C(C1=NOC2CN(C(=O)C=C3CCC3)CC12)NC(c1cc(C)nnc1O)=O 47118,c1(C(N2C(C)CC(NC(C3CC(=C)C3)=O)C2)=O)cn2cccc(F)c2n1 47119,N1(C(c2n(C)cc(NC(c3csc([N+](=O)[O-])c3)=O)c2)=O)CCCC2(CC2)C1 47120,C1(C(=O)NC2(C(=O)OCC)CC2)CCCC(NC(C2CC2CC)=O)CC1 47121,C#CC1(C(=O)N(CC(C)(C)CNC(=O)C(CCSC)OC)CC)CCCC1 47122,C1(C(=O)NCC2C3CN(C(Cn4nnc(C)n4)=O)CC32)CCN2CCOCC12 47123,c1(CNNC(c2c(C)scn2)=O)cc(Cl)cnc1F 47124,CC1CC(C#N)(C(=O)NC2CC(NC(C3(Cl)CC3(F)F)=O)C2)C1 47125,N1(C(C(C)N(C(=O)C(C(C)O)N(C)C)CC)=O)CC(O)C(C2CC2)C1 47126,CCC(C(=O)N1CC2CC1(CNC(c1cccc(F)c1C)=O)C2)C(C)O 47127,c1(OC)ccc(COCCCN(C)C)cn1.c1(C(=O)NCCOC)ncccc1O 47128,N1(C(c2cn(CC=C)nc2)=O)CCC(NC(=O)C(F)C(C)(C)O)CC1C 47129,N1(C(c2nncc(OC)c2)=O)CCC(N(C)C(C2SCCS2)=O)C(C)C1 47130,C1(C(=O)NC2(CCNC(c3occ4c3CCOC4)=O)CC2)CCCC2(CCC2)O1 47131,N1(C(C(c2cccs2)NC(c2ccc(CC)nc2)=O)=O)CCC(N=[N+]=[N-])C(O)C1 47132,C1(CC(=O)NC2CC(CNC(CCCNC(C)=O)=O)C2)COCC(C)(C)O1 47133,N1(C(c2cc(F)c(C)c(F)c2)=O)CC2(C1)CN(C(=O)C(C)S)CC2C(=O)O 47134,C(CN=c1[nH]c(=NC)[nH]c(=NCC=CC2CC2)[nH]1)c1c(OC)c(C)c(C)cc1 47135,N1(C(CC2(NC(C)=O)CC2)=O)CCOC(C(C)NC(c2cc(Cl)cnn2)=O)C1 47136,c1(OC)cccc(=NC(=O)Cc2csc(C(=O)Nc3cc(Br)c(C)cc3F)n2)[nH]1 47137,c1(OC)ccc(OC)c(C2CC2C(=O)OCC(C)(O)COCc2ccccc2)c1 47138,C(N=c1[nH]c(N2CCc3nc(O)[nH]c3C2)nc2ccccc12)C1(C)C(C)(C)C1 47139,n1(C(CC)C)ncc2cc(C(=O)NCC3CCN3C(c3ccncc3)=O)cnc12 47140,CC1CCN(C(c2ccccc2O)=O)C1C(=O)NCC1(O)CC=CC1 47141,CCCCCCCC(=O)N1CCCC1C(C)NC(c1c(Br)nnn1C)=O 47142,C1(C(=O)NCC(CNC(C2CC23CCCCC3)=O)CO)CCC(=C(F)F)CC1 47143,C1(C(N2CCC3(CC2)CC3)=O)CC2CCCC2N1C(C1CCCC1F)=O 47144,C1(NC(COCCOC)=O)CCC2(CC1)CCN(C(c1csc3cncn13)=O)C2 47145,C(C(O)C(F)(F)F)CN(C(CNC(=O)OC)=O)C.C1CC(=O)N1 47146,c1(CCC(=O)NC2CC(C)N(C(=O)CC#N)C2)cc(F)ccc1Br 47147,N1(C(C2CCN(C)C2)=O)CC=CC(C(N2CCN(CC(N)=O)CC2)=O)C1 47148,C1(C(N(CCCF)CC)=O)CC2CC2N1C(C1CC=C(C)CC1)=O 47149,N1(C(CC2(CNC(C3CCN(C)CC3)=O)CC2)=O)CCCC(F)CC1 47150,C(=O)(C1=NOC(C)C1)NC(C(=O)NCC(CCC)O)CO 47151,N1(C(C(COC)C)=O)CCC(C2CC2)(NC(=O)C=C(C)c2cccs2)C1 47152,C=C(C)CCCC(=O)NC12CC(NC(c3cc(C4CCOCC4)[nH]n3)=O)(C1)C2 47153,c1(C(=O)NCC(C)NC(C2(CC)CC(C)(C)C2)=O)ccc(C(F)(F)F)c(F)c1 47154,N12CCCC(C1)NC(=O)C2=O.C1(C(N(C(C)C)CC)=O)(C(=O)NC(C)=O)CCC1 47155,c1(CC)cc(C(=O)NCC(C)CNC(=O)CC(CC)C2CCC2)ccn1 47156,Cn1ncc(C(=O)NC2CCCCC2NC(=O)Cc2nncn2C)c1Cl 47157,c1(N(CCOC)CCC2CC2)nnc(CC2CCCCC2)n1Cc1nnc(C)n1C 47158,C1(C(N(C(C)CCNC(=O)C=C2CC2)C)=O)CC(c2ccccc2[N+](=O)[O-])=NO1 47159,C1(OCCNC(C(=O)N(CCCCN(C)C)C)=O)CNC2CC2C1 47160,c1(C(=O)NCC2(O)CC(C(=O)NCC(C3CC3)OC)C2)cc(C)oc1C 47161,c1(CC(=O)NC23C(CN(C(C=CC(=O)OCC)=O)C2)C3)nsc2ccccc12 47162,N1(C(C2CCCCC2)=O)CC(C(N2CCC2CC2CC2)=O)C(F)C1 47163,c1(C(=O)OC)coc(C=CC(=O)NC2CCC(N(C)C(c3cc(C)sn3)=O)C2)c1 47164,C1(C(C)NC(C2(CCN(C)C)CC2)=O)CCCN1C(c1n[nH]c(O)n1)C1CC1 47165,C1(NC(CS(CCC)(=O)=O)=O)CCC2CCN(C(c3ccc(O)cc3Cl)=O)C1C2 47166,c1(NCC)ccc(C(=O)N(C2CN(C(=O)COC3CCOCC3)C2)C)c(F)c1Cl 47167,C1(n2cc(CC(C)(C)CO)nn2)CCC(NC(c2cc(F)n[nH]2)=O)CC1 47168,c1(C(N(CCCCN(C)C(c2csc(-c3cn[nH]c3)n2)=O)C)=O)cncc(F)c1 47169,C1(C(=O)NCC2N(C(Cn3nc(C)c(Cl)c3)=O)CCC2)CCCC1C1CC1 47170,CCN=c1[nH]cc(C(=O)N(CCCNC(C2CC2[N+](=O)[O-])=O)C)s1 47171,C1(NC(CCOc2cccc(C)c2)=O)CN(C(c2cscc2C#N)=O)CC12CC2 47172,CC(C)(C#N)CC(=O)NC1CC(NC(C2CCC=CCC2)=O)C(O)C1 47173,c1(CC)cccc(C#CC(=O)NCC2CCC3(CCCCCC3)O2)c1 47174,C1(C(C)O)CCOCCN1C(c1nc(Cl)cs1)=O 47175,c12ccc(c(F)c1F)CN1CCC(=CC(=O)N=CC(=O)N2)CC1.C(CC)=CC.OCC 47176,C1(CC)(CC)CC(NC(C2CCC3(CC2)CC3)=O)CN1C(c1csc(C)n1)=O 47177,N1(C(C(C)NC(C2CCC2)=O)=O)CCCC(O)(CNC(=O)Cn2nccn2)C1 47178,c1(OC)ccnc(O)c1C(N1CC(NC(=O)Cc2cnsc2)C(C)C1)=O 47179,Cc1cc(C(N2CCN(C(C3CCCO3)=O)CC2)C(=O)NC2COC2)cc(F)c1 47180,C1(S(C)(=O)=O)(CNC(=NCCSC)NCc2ccc(F)cc2)CCC1 47181,N(C1CC(C)(C)c2ccccc21)Cc1c(Br)cc(OC)c(OC)c1O 47182,c1(CC(=O)NC(C2CCN(C(C(CCC)O)=O)C2)C)cc(OC)ccc1F 47183,C(=O)(C(C(C)(C)O)NC(c1ncn(C)n1)=O)N1CC(C)SCC1 47184,CCC1=C(C(=O)NCC(C)(O)CNC(=O)CN=S(C)(C)=O)SCCO1 47185,C1(C(=O)NC2CC(NC(c3ccc(=O)oc3)=O)C2)CCN(C2CC2)C1=O 47186,n1(C2CN(C(CCN(C(CCC)C)C)=O)C2)cc(C2COCC2O)nn1 47187,c1(CNC(C(C2CN(C(Cn3nnc(C)n3)=O)C2)N(C)C)=O)cc(C)oc1C 47188,c1(CCCNC(=O)C(C2(O)CN(C(=O)CC3CCCCC3)C2)F)cncc(F)c1 47189,CCCC(C(=O)N1CC(=O)CC1C(=O)NCC1CC(C)C1)N(C)C 47190,c1(C(N2CCC(O)(CNC(c3cnn(C(F)F)c3)=O)C2)=O)noc2ncccc12 47191,c1(C(=O)OC(C(=O)OCCC)C)cn(CC2CCOC2)nn1 47192,c1(OC(C)C)ccc(C(=O)NC2CC2C(=O)NC(c2ccccc2)(C)C)cn1 47193,c1(CC)cc(C(=O)N(C(CNC(=O)C=CC2CC2)C2CC2)C)ccc1Br 47194,CN1CCC(O)(CC(N2CCC(NC(=O)CC3C=CCCC3)C(O)C2)=O)CC1 47195,Cc1ccc(CN2CCC(C(C)NC(c3ccnn3C)=O)CC2)c(F)c1F 47196,C12(CNC(c3n(C(C)C)ncc3)=O)CC1CN(C(C1CCCC1C(F)F)=O)C2 47197,C1(N(CCCC)C(c2n[nH]cc2Cl)=O)CCN(C(c2cc(OC)cs2)=O)CC1 47198,C#CC1(C(=O)NCC(CC(C)C)N(C)C)CCN(C(=O)CNC(=O)CN(C)C)C1 47199,Cc1ccc(C(F)F)cc1OCC(N1CCSCC1NC(=O)OCCO)=O 47200,N1(C(c2ncc3c(n2)CCC3)=O)CCC(F)(F)C(CO)C1.c1(N)ccc(O)cc1 47201,C=C(C)CC(C(=O)NC1CCCCC1N=[N+]=[N-])NC(=O)C(C1CCOCC1)F 47202,c1(OC)noc(C2CC2)c1C(=O)NCC1(NC(C2(C#N)CC2C)=O)CC1 47203,CN1N=C(C(=O)N2CC(CCNC(=O)C(c3cccc(F)c3)(C)O)C2)CCC1=O 47204,N1(C(C(C)c2ccco2)=O)CCC(NC(=O)C(C)(C)CC(F)F)CC(C)(C)C1 47205,C1(O)(CCNC(Cc2n(C)cnc2)=O)CCN(C(c2cnn(CCF)c2)=O)CC1 47206,C12(C(=O)NC(C3CCCCC3)CC)CC(CO1)N(C(c1ccc(Cl)cn1)=O)C2 47207,N1(C(CCOCCNC(c2ccnnc2O)=O)=O)CCc2ccccc21 47208,N1(c2ncnc(OC)c2OC)CCc2cc(C(N3CCS(=O)CC3)=O)ccc2C1 47209,C=C(C)c1cccc(NC(C2CC(=O)CN2C(=O)C(C(C)(C)C)OC)=O)c1 47210,c1(OC)ncc(C)c(C(=O)NC2CC(C)N(C(c3cccc[n+]3[O-])=O)C2)c1Cl 47211,c1(-c2ccc(CNC(C=C)C(=O)OC)cn2)ccc(OC)c(F)c1F 47212,Cc1c(C(=O)NC(C)CCNC(=O)C2=CCCC2C)c(O)nc2ccccc12 47213,CC1(NC(c2coc(Br)c2)=O)CCN(C(c2ccc(C3(C)CCO3)cc2)=O)C1 47214,N1(C(c2c(C)nco2)=O)CC(C)(CNC(=O)CC2CCCC(=O)N2)CC1(C)C 47215,c1(C(=O)NC(C)C(C)(C)NC(C23CC(C)C2C3)=O)cc(Br)cc2nc(O)[nH]c12 47216,C12(C(N3C(C)CC(NC(C(C4CCCCC4)C)=O)C3)=O)CCC(F)(CC1)CC2 47217,CC(C)CC(C)(CNC(=O)Cc1cccc(O)c1)NC(c1ccn(C2CC2)n1)=O 47218,N1(C(C(c2cccs2)NC(C2CCS(=O)CC2)=O)=O)C2CCCC1COC2 47219,CC(C)(C)CC(=O)N1CCC(C(C)(O)CC2CC2)CC1 47220,C=C=CCC(=O)NCC1COCC1NC(=O)CCc1cc(OC)no1 47221,c1(N(CCCN(C(c2nc(C)n(C)n2)=O)C)C)nc(Cl)ncc1Cl 47222,Cc1cc(-n2ccnc2)ccc1C(=O)NCCN(C(=O)C(F)C(F)(F)F)C(C)C 47223,C1(OC)CCCCCC1NC(=O)C(=O)N(c1ccc(Cl)c(F)c1)CC(C)C 47224,c1(C(=O)NCCCNC(=O)Cc2cnoc2)ccccc1SCCCO 47225,Cc1cc(=NCC2(CCO)CCCC2)[nH]c(NCC(c2ccccc2)F)n1 47226,CN1CCC(n2cc(C3(C)CN(C(=O)C(F)C4CCOC4)C3)nn2)C1=O 47227,CC(CN(c1ncc(C2CCCOC2)s1)C(=O)OCCCN=[N+]=[N-])(CO)CO 47228,C1(C(N(C2CCN(C(c3ncsc3C)=O)C2)CC)=O)CCCC2CC12 47229,N1(C(C(CC)OC)=O)CCC2(CCN(C(=O)C(O)C3CCC3)C2)C1 47230,c1(NC(N2CC3(CC2CO)OCCO3)=O)ccc(F)c2[nH]ncc12 47231,c1(C(=O)NC2(CNC(=O)CC3(C(F)(F)F)CC3)CC2)cn(C2CCCCC2)nn1 47232,c1(N2CCCC(C(C)C)CC2)cccc(S(=O)(=O)NCC(CO)N(C)C)n1 47233,C1(C)(CNC(c2c(CC)con2)=O)CN(C(=O)CC(C(F)(F)F)OC)C(C)(C)C1 47234,C1(NC(c2c(C)cc(SC)o2)=O)CCN(C(c2cn(C)ccc2=O)=O)C1(C)C 47235,C1(C)(C(N(CCN(C)C(c2ccnc(-c3ccco3)c2)=O)C)=O)CCC(=O)C1 47236,c1(CC)cc(C(=O)NC(C2CCN(C(=O)COC(C)C)C2)(C)C)c(C)o1 47237,C1(C)(C(C)NC(=O)COc2ccon2)CCN(C(=O)CC23CCCC2C3)CC1 47238,N1(C(=O)Cc2nc[nH]n2)CCOC2(CCN(C(C3CC4CCC3O4)=O)C2)C1 47239,CC(C)C(CN(C)C)N=c1nc(N2CC3CCC3C2)c2c(ncn2C)[nH]1 47240,Cc1nc(Cl)[nH]c(=NC2CC(CNC(=O)C3=NCC3C(F)(F)F)C2)c1Cl 47241,Cn1nc(C(N2CCC(NC(c3ccncc3)=O)C23CCC3)=O)c2c1CCC2 47242,CC(CC(C(=O)c1ccccc1)N1CC(n2cccn2)C1)C(C)(C)C 47243,C1(C(=O)NC2CN(C(C(C3CC3)OC)=O)C2)CC(=O)N(CCN(C)C)C1 47244,C1(OC)CN(C(=O)CC2CC(F)C2)CC1NC(C1(c2ccccc2Br)CC1)=O 47245,c1(C(N2C(CN(C(=O)CCF)C)CCC2)=O)csc2ccc(Br)cc12 47246,Cc1cnc(NC(C2CSCCN2Cc2c(C)cccc2Br)=O)c(Cl)c1 47247,c1(C(=O)NCC(CC)NC(c2cc3occc3[nH]2)=O)cc2n(n1)CC(C)(C)OC2 47248,C(C(CC1CCCC1)C(=O)N=c1ccn(C2CC2)[nH]1)NC(c1c(C)cnn1C)=O 47249,C(=O)(CC(C(F)F)NC(c1n[nH]c(O)n1)=O)NCCC(CC)(C)C 47250,N1(C(c2cnsn2)=O)CCCC(N(C(=O)C=Cc2ccco2)CCF)C1 47251,C1(C)(C(N(C)CC2(NC(=O)C=C3CCCCC3)CC2)=O)CCC(=O)N(C)C1.C(C)(C)(C)O 47252,CCC(C(C)O)NC(c1ccoc1CNC(=O)C(C)(C)OC(C)C)=O 47253,C1(NC(c2sc(CC)c(C)c2)=O)CN(C(=O)C(F)(F)C(C)O)CC1C1CC1 47254,Cc1c(CNC(=O)NCC2(F)CCCCC2)cccc1F 47255,CS(=O)c1cccc(NC(c2noc(-c3ccccc3)n2)c2nnnn2CC(F)F)c1 47256,C=CC1(C2(C(=O)NCCCCN(C(=O)CSc3cccs3)C)CCC2)CCC1 47257,C(c1ccc(F)cc1)=CC(=O)NCC12CCC1CCN2C(=O)CC1CS(=O)(=O)C1 47258,CC1CC(NC(c2cncc(O)c2)=O)CCN1C(c1cccnc1Cl)=O 47259,Cc1[nH]c(C#N)cc1C(N1CC(CC(N2CC3(CCC3)C2)=O)C(C)C1)=O 47260,N1(C(c2c(C)ncnc2)=O)CCC(F)(C(=O)NCCC(O)C(C)C)CC1 47261,c1(OC(C(N2CCC(C)CC2)C)=O)ccc2ccccc2c1 47262,c1(Nc2sc(C(C)=O)c(C)n2)ccc(NC(=O)CN2C(=O)CCCC2=O)cc1C 47263,C#CCCCCCCC(=O)N1CCN(C(=O)CCCNS(C)(=O)=O)C2CC12 47264,N1(C(c2c(C)cn(C)n2)=O)CCC2(CC(NC(c3c(C)ncn(C)c3=O)=O)C2)C1 47265,C(CC(O)C(=O)NCCCCC(C)NC(c1ccc(NC=O)cc1)=O)SC 47266,N1(C(c2c(C)nc(C(F)(F)F)cc2)=O)CCC2(NC(=O)COC(C)C)CCCC12 47267,Cc1nn(C)c(C)c1S(=O)(=O)NC1CCN(C(C2CNC(=O)C2)=O)CC1 47268,c1(OC)ccc(CCC(=O)NC2CCC(CNC(C3CN(C(N)=O)C3)=O)C2)cc1 47269,c1(C(N2C(CNC(C3CCCC(=O)N3)=O)CC2)=O)nc2cnccc2s1 47270,c1(C(N(C(c2ccccc2)CNC(C2CNC(=O)C2)=O)C)=O)cc2cccnn2n1 47271,C1(N(CCOC2CC(c3ccccc3F)(C(=O)OC)C2)C)CC2CCC1C2 47272,CC(C(=O)NCC1CN2CCC1(C)CC2)N1C(=O)COc2ccccc21 47273,Cn1cnc2c1CCN(C(=O)CC(C)(C)C)C21CCN(c2nnc(C#N)s2)C1 47274,C1(C)(CC(=O)N(CCC(C)O)C)CCN(C(C2CCCCN2C)=O)C1 47275,Cc1cc(C(F)F)nn1CC(N1CC(NC(C2(C)CCOC2)=O)C(F)C1)=O 47276,C=Cc1ccc(C(=O)N(C2CCCCN(C(C3(C(C)C)COC3)=O)C2)C)cc1 47277,c1(C(=O)NCC2CCCN(C(C(C3CCC3)OC)=O)CC2)nc2ccccn2n1 47278,C1(NC(CC2CC(C(=O)OC)C2)=O)CCCN(C(C2CC(=O)N(C3CC3)C2)=O)CC1 47279,N1(C(C(CCSC)(C)C)=O)CC2CC(C1)CN(C(C1CC3CC(=O)C1C3)=O)C2 47280,C1(OC)CC2(C1)CC2NC(=O)C(C1CCOC1)NC(=O)C=Cc1cc[nH]n1 47281,C(CC(O)CC(=O)NC1CCC(N(C(=O)C(C)n2cncn2)C)CC1)SC 47282,N1(C(Cc2c(C)nccc2)=O)CCC(O)(CNC(c2ccc([N+](=O)[O-])o2)=O)CC1 47283,c1(CC)cccc(OCC(=O)NCC2CN(C(c3ccc(CCF)cc3)=O)C2)c1 47284,N1(CCn2c(C)cc(C)n2)CCCC(NC(=O)CN2CCCCC2=O)CC1 47285,C1(CC(=O)N(C2(C#C)CC2)C)CC(O)CN1C(=O)CN1CCCC1 47286,c1(C(C)=O)cc(C(=O)NCC23CC(NC(=O)Cn4ccnn4)(CO2)C3)n(C)c1 47287,N1(C(c2n(C)c(S)nc2)=O)CC2CN(C(c3coc(C(F)(F)F)n3)=O)CC2(C)C1 47288,C1(C(N(CCCNC(=O)CSCc2ccncc2)C)=O)CCC(=O)N2CCCC12 47289,C1(C(N2CC(C(C)C)OCCC2)=O)C2CCCC2CN1C(=O)CC(C)(C)O 47290,C1(NC(=O)C=CCNC(=O)CC2CC=CCC2)CCC(C2CC2)O1 47291,CCC(N)CCC(=O)N1CCC12CN(Cc1ccccc1)C2 47292,C1(NC(CNC(=O)CC(F)(F)F)=O)CCN(C(=O)CCc2cnccn2)CC1O 47293,c1(CC(=O)NCC(CCOC)NC(=O)Cc2c(Cl)cnn2C)ccc(F)cn1 47294,C(=O)(C(F)C(F)(F)C(F)(F)F)N1CCC2CCC(NC(C3CC(C)(C)C3)=O)C1C2 47295,C1(C(N(CCCC(C)C)C)=O)CN(C(C2C3CCC(C3)C2C)=O)CC1(C)C 47296,c1(OCC)ncc(C(=O)NCCC2(NC(=O)C(C)(C)O)CCCC2)s1 47297,N1(CCNC(C(=O)NC(c2ccc(I)cc2)COC)=O)CCC(C)CC1 47298,C1(CC(N2CC(NC(c3c(C)cn(C4CC4)c3)=O)C2)=O)CCCC(C#N)C1 47299,CC12CC(C(=O)NC3(C4CCCCN4C(c4ccco4)=O)CC3)(C1)C(C)(C)O2 47300,N1(CCNC(C(C)(C)C2CCC2)=O)CCN(C(=O)C(C)(C)C2(C)CC2(F)F)CC1 47301,C1(CNC(c2c(C)onc2Cc2cscn2)=O)CN(CCOC2CC2)CCN1C 47302,c1(CNC2(c3nnnn3CCCF)C(CN(C)C)COC2)ccccc1[N+](=O)[O-] 47303,CCCCC(O)C(C)C(=O)NC1CCCC1CNC(=O)CCc1nc[nH]n1 47304,O=C(N1CC(O)CO1)C1CC12CCN(C(c1cnn3c1CCC3)=O)C2 47305,c1(CCC(=O)OCC(CNC(=O)OC(C)(C)C)O)cncnc1O 47306,c1(C(c2nnnn2C2CCOC2)NC2C(OCC)C2)cc(C)ccc1Cl 47307,C=CCCC(C(=O)NOCCC)NC(C1CC=CCO1)=O 47308,C(=O)(CC(C)(C)C(F)(F)F)NCC1N(C(C(C(=O)OC)OC)=O)CC2(CC2)C1 47309,S(=O)(=O)(C(Cl)(Cl)Cl)NC1(C(N(CCC#C)C2CC2)=O)CC1 47310,N1(C(Cc2c(C)nn(C)c2)=O)CCC(C)C(CC(N2CCC(SCO)CC2)=O)C1 47311,N1(C(COCC=C)=O)CC2CC(C(=O)NCCOCCC3CC3)C(C2)C1 47312,CCCCC(C)CCC(=O)NC1CN(C(C23CCC(CC2)CC3)=O)CC1C(F)F 47313,C12(NC(Cc3n(C(C)C)ncc3)=O)CC(CNC(=O)Cn3cnccc3=O)(C1)C2 47314,N1(C(CCOC(C)=O)=O)CC(NC(=O)CN2CCC(C)(O)C2)CC(C)(C)C1 47315,C1(C(N(CC)OC)=O)N(C(=O)CC(=O)OCC)CC12CCCC2 47316,C(CNC(=O)CCCc1ncco1)(CC(=O)N1CCC(C(N)=O)C1)OC 47317,C1(NC(c2c(CC)cccc2)=O)CC2CN(C(=O)CCc3cn(C)nn3)CC12 47318,Cc1sc(C)c(S(=O)(=O)NC2CN(C)CC2c2cncn2C)c1Br 47319,N1(C(=O)CCCc2ncco2)CCC(C(F)F)(CNC(=O)C(F)OC(F)(F)F)C1 47320,Cc1cc(C(N2C3CCC2CN(C(=O)CC(F)(F)Cl)CC3)=O)nc2ccccc12 47321,N1(CC)C(=O)CCC1CC(=O)NC1(C)CCN(C(=O)CCc2nccn2C)C1 47322,C(=O)(C1CCc2c[nH]nc21)N1C(C)C(NC(C2(F)CCOCC2)=O)CCC1 47323,C(=O)(C(C(C)(C)C)N(C)C)NC(CC#C)C(=O)N(CC(C)C#C)CC 47324,c1(-c2scc(C(=O)NC(c3ccc(Cl)cc3)CF)n2)ccc2c(c1)OCO2 47325,C(C)(C(O)C(=O)NCC1CCC(NC(c2n[nH]cc2Br)=O)CC1)OC 47326,N1(C(C(C)SCC)=O)CC(C2(NC(=O)C(CC)CC)CC2)C1 47327,CCCCC(O)C(=O)NC(C)CC(C)NC(c1cc(C(F)(F)F)ncc1N)=O 47328,C1(C(=O)OC)(N(CC(=O)Nc2ccc3c(c2)OCO3)C)CC(O)C12CCC2 47329,c1(C(=O)NC2CC(C)(CNC(c3sc(C)c(O)n3)=O)C2)c(O)cccc1Cl 47330,c1(NCC(N(C)C(c2ccncc2F)=O)C2CC2)ncc2scc(Br)c2n1 47331,N1(C(c2ccc(OC)nc2)C(=O)NCCCF)CC2C3C=CC(CC3)C2C1 47332,N1(C(CC=CCC)=O)CCCOC(CCNC(C2(C)CN(C(C)C)C2)=O)C1 47333,C1(C(=O)NCC2(F)CC(NC(C(C)OCCC=C)=O)C2)CCCC(=O)N1C 47334,N1(CCCC)CC2CCC1C1CN(C(=O)C3Cc4ccccc43)CC21 47335,O(C1CCCC(=O)c2ccccc21)CC(N)(CC(=O)O)C(F)(F)F 47336,c1(C(C)=O)ccnc(NCC2CCCCN2C(=O)CSc2ccncc2)n1 47337,S(=O)(=O)(c1ccc([N+](=O)[O-])cc1Cl)NCC(=O)N(CCNC(COCCC)=O)CC 47338,C(CCCCCC(=O)N(CCCCCO)C)n1cc(SC)nn1 47339,C1(CC=C)(NC(=O)C(O)C2CC2)CCCN(C(=O)CCCN(C)C)C1 47340,C1(C(N(C2CN(C(C3CCC(C)CC3)=O)CC2(C)C)C)=O)COC(C)(C)CO1 47341,C1(NC(C2CC2(F)F)=O)CCCN(C(c2cnn(-c3ccccc3)c2)=O)C1 47342,Cc1cc(C2CC2)cnc1C(=O)NCCNC(=O)CCc1ccccc1O 47343,N1(C(C(CSC)(C)C)=O)CCC2(NC(=O)Cn3ccc(=O)cc3C)CC2C1 47344,N1(C(Cn2ncc(CC)c2)=O)CC(O)CCC1C(=O)NCc1ccc(F)c(F)c1 47345,c1(C(N(CCCNC(CC(CCC)C)=O)C(C)C)=O)ccc2c(c1)CNC2=O 47346,CC(C)(O)C#CC(=O)NCCCNC(c1ccc(CC(=O)NC2CCC2)cc1)=O 47347,CC(C)C(O)CONC(c1cc(CNC(C2COCOC2)=O)[nH]n1)=O 47348,CC1(C)COC(CC(=O)NCC2CCCN2C(=O)CCC=CBr)CO1 47349,N1(C(c2nc(OC)c(C)s2)=O)C2CCC1CN(C(c1cnc(C)[nH]1)=O)CC2 47350,C1(NC(C=C(COC)C)=O)COC2(CNC(=O)C3=CCCC3)CC1C2 47351,N1(C(N)=O)CCCC1C(N1CC(CCNC(=O)CCc2cnn[nH]2)C1)=O 47352,N1(C(C2C(=C)C2)=O)CC(C)(C)CCC1CNC(c1ccc(C(N)=O)cc1)=O 47353,C1(C(N2CCC(NC(c3cc(C(=O)OC)sn3)=O)C2)=O)CCS(=O)(=O)C1 47354,C1(NC(C2C(c3cn(C)nc3)C2)=O)CN(C(=O)CSc2nncn2C)CC1O 47355,C1(C(N)=O)CCN(C(=O)CC2CCCC2NC(c2ocnc2C(F)F)=O)O1 47356,c1(CC(C(=O)OCC(N2CCC(C(F)(F)F)C2)=O)O)cccc(Br)c1 47357,N1(C(C(C)(C)F)=O)CCC2(C(=O)NCC3CCCC3)CC2C1 47358,C(=O)(C(CC(F)F)N(C)C(c1ccc(C#N)cn1)=O)NCC(C1CCCC1)C 47359,N1(C(c2cc(OCC)n[nH]2)=O)CCC2(NC(=O)Cn3ccc(C)cc3=O)CC2C1 47360,C#CC1(O)CC(C(N2CCC(N(C(=O)CC(C)(O)C3CC3)CC)CC2)=O)C1 47361,C1(CC(N)=O)(NC(C2(COC)CCOC2)=O)CCN(C(=O)C(C)CN(C)C)CC1 47362,C(=O)(CCC(C)C#N)N1CCN(c2nnc(-c3c(C)nc(Cl)s3)n2CCC#N)CC1 47363,Cc1conc1C1CN(C(C2(CNC(C3C4COCC34)=O)CCOC2)=O)C1 47364,C#CCCCC(C)C(=O)N1CCC1CC(=O)NCCCCSC 47365,C1(C)(CC(=O)NCC2CC(C(=O)OC)C2)CCN(C(C2CC2(F)F)=O)C1 47366,C(CCCCC(=O)NC1(C)CC(N(C)C)C1)N(C)C(C1CCC2CC12)=O 47367,C1(N2CCN(C(C(c3cccc(C#N)c3)C)=O)CC2)CC(C)(C)OC1=O 47368,C12(CNC(c3c(C)nc(Br)s3)=O)CCC1CCN2C(=O)CC1=CCCC1 47369,c1(NCC(N2CCC(NC(C3CCCSC3)=O)C(O)C2)=O)ccccc1[N+](=O)[O-] 47370,c1(CC)ncoc1C(=O)N(CCCC(=O)NCC(c1ccccc1)F)C 47371,c1(C(=O)Nc2sc(C(C)=O)c(C)n2)cc(O)ccc1Br 47372,C1(NC(CNC(C(CC)CC)=O)=O)(CO)CCN(C(=O)CCCC(N)=O)CC1 47373,C(=O)(CS(=O)(=O)C(C)(C)C)NCC1N(C(C2(CCOCC)CCC2)=O)CC1 47374,C1(CCNC(C(c2cncnc2)C)=O)CCN(C(c2nn[nH]c2C(F)(F)F)=O)C1 47375,C1(NC(C(C)C2CCCO2)=O)CN(C(C2CCCS2)=O)CC(C)(C)C1 47376,N1(C(C2(OCC)CCC2)=O)CCN(C(CNC(C2(C)COC2)=O)C(F)(F)F)CC1 47377,C(=O)(CCCC(F)(F)F)N1CC(C(C2CC2)NC(=O)C=Cc2ccco2)CC(C)C1 47378,C(CCC(C)C)(C(=O)NCC1CC(C)C1)NC(C1CC=C(C)CC1)=O 47379,C1(C(N2CC(CCC)C(C(=O)O)C2)=O)CC2CN(C(=O)OC(C)(C)C)CC2C1 47380,C1(NC(CCC(=O)N(CC)CC)=O)CCN(C(c2nn(C)cc2Cl)=O)C12CCC2 47381,c1(CNC(N2CCC(=CCc3nn[nH]n3)CC2)=O)n[nH]c2c1CCOC2 47382,c1(OC)cc(C=CC(=O)NCC2CC2NC(C2(n3cnnn3)CCCCC2)=O)sn1 47383,C1(CNC(CN(C(C2CC3CCC(C2)O3)=O)CC)=O)CC12CCCCC2 47384,N(C1CCc2cccnc21)C(C1C(CC)N(C(C2COCC2(C)C)=O)CCC1)=O 47385,C1(NC(CC2CN(S(CC)(=O)=O)C2)=O)CCC(NC(c2scnc2C2CC2)=O)C1 47386,c1(C(N2C(C)CN(C(=O)CC#N)CC2)=O)cccc2c1CC(=O)N2C 47387,C1(C(=O)NC2C(NC(c3n(C)cc(C#N)c3)=O)CCCC2)CCc2nccn2C1 47388,C(=O)(C(C)CC(C)C)N(CCCC(=O)N(CCC)CC)C(C)C 47389,c1(NC(C2CCN(C(C3(C)CCCCO3)=O)CC2)=O)ccc2c(c1)CCC2 47390,c1(C(=O)NCC(CNC(CC2CCN(C)C2)=O)C(F)(F)F)cnn2c1OCCC2 47391,C=CC(C)(O)C(=O)NCC(CNC(c1sccc1Cl)=O)OC 47392,C(=O)(C(F)(F)C(F)(F)C(F)(F)C(F)F)NCC(CO)NC(c1c(C)nns1)=O 47393,N1(C(C2(C)CC2(F)Cl)=O)CCC2(CCCC2NC(c2cnc(O)nc2O)=O)CC1 47394,C=C(C)C1OCCC1C(=O)NC1CCC1CNC(=O)C(C)NC(=O)CC 47395,C(CCC(C)CC(=O)NC1CCC(N(C(=O)CCc2cnn[nH]2)C)C1)=C(C)C 47396,c1(CC(C)C(=O)N2CCC(N(C(=O)Cn3ncnn3)C)C2)cccc(Cl)c1 47397,CC1CN(C(C2CCC(NC(=O)CC3CCOC3(C)C)CC2)=O)C(C)CO1 47398,N1(C(C2(NC(CNC(CC)=O)=O)CC(O)C2)=O)CC2(CCC(=O)O2)C1 47399,C#CCCCC(C)C(=O)N1CCC(C)(CNC(c2c(F)ccc(OC)c2F)=O)C1 47400,c1(C(C)C)ccc(C(=O)NCC(C)NC(=O)CCC2CCC(O)CC2)cn1 47401,c1(SC(C)C)ccc(C(=O)NCCC2CCCCN2C(C2CC3CC2C3)=O)cc1 47402,c1(OC)ccc(C(N2CC(OCCNC(=O)C(N)=O)C2)=O)c2ccoc12 47403,N1(C(CSCCCC)=O)CC(CNC(=O)CN2CCN(C3CC3)C2=O)CCC1C 47404,C12(CNC(c3ncc(Cl)cn3)=O)CC1CN(c1ncc(I)cn1)C2 47405,Cc1c(C(=O)NC23CC(CNC(c4cccs4)=O)(C2)C3)nn2ccccc12 47406,C(=O)(Nn1cccn1)C1(F)CNC1.c1(-c2[nH]c(=N)sc2)ccccc1F 47407,C(=O)(C(C#N)C(C)(C)C)NCC1(F)CCC(NC(COCCSC)=O)C1 47408,c1(NC(C2N(C(c3ccc(Cl)cc3)=O)CCC(=C)C2)=O)cnc2c(c1)CCC2 47409,Cc1ccc2c(C(N3CCCC(NC(=O)CC(O)C(C)(C)C)CC3)=O)c[nH]c2c1 47410,c1c(Br)cncc1Br.Cc1cccc(C2CCN(CCNC(C3CCC3)=O)C2)c1 47411,N1(C(C2(C#C)CCN(C(c3ccc(F)c(O)c3)=O)C2)=O)CCCCC(C)(F)C1 47412,N1(C(CC2(OC)CCC2)=O)CCC(CF)(NC(c2ccc(C(F)F)o2)=O)C1 47413,C1(C(N)=O)CC(C(=O)NCCCNC(=O)CSCC2CC2)=NO1 47414,N1(c2n(C)c(C3CCN(S(C)(=O)=O)CC3)nn2)CCC2(CCCCO2)C1 47415,N1(C(CCC=C=C)=O)CC(NC(=O)CC(C)COC)C(N=[N+]=[N-])C1 47416,C1(C(=O)NC2(C)CC(NC(C3CCC(C)CC3)=O)C2)CCn2c(O)nnc2C1 47417,Cn1nccc1CCC(=O)NC1CCCC1NC(c1coc(Cl)n1)=O 47418,Cc1cc(=O)n(C)cc1C(=O)NC(C)CNC(=O)C(C1CCC(O)CC1)(C)C 47419,C1(NC(C(CC)C#N)=O)CC(O)(C2CCN(C(c3csc(C)n3)=O)CC2)C1 47420,N1(C(c2cc(COC)on2)C(=O)NCC(F)F)CC2CC2(CO)C1 47421,n1(C(C)(C)C)ccc(=NC(=O)C2N(C(=O)CC3CCCCC3)CC23CCCC3)[nH]1 47422,c1(C(N2CCC(NC(c3cc(C=O)ccc3O)=O)CC2)=O)cn2c(n1)CCC2.CO 47423,C1(C(N2CC3(NC(C(=O)NC)=O)CC2(COC)C3)=O)CCCC2CCCCC12 47424,N1(C(C(=O)N(C)C)=O)C2CCC1CC(N(C)C(c1nocc1Cl)=O)C2 47425,c1(C(C(=O)NC23CN(C(C(C)O)=O)C(C2)C3)=O)cc(F)ccc1F 47426,c1(SC)nc(Br)c(N(C2CC(N)C2)C(c2ccc(-c3cccs3)o2)=O)n2ccnc12 47427,N(C(=NCc1ccccc1C(N1CCCC1)=O)NC(C)CC)C(C=C)C 47428,C1(NC(C=CC=CCC)=O)CCC12CN(C(=O)C1=NNC(C(F)(F)F)C1)C2 47429,N1(C(C(CC(=O)OCC)C)=O)CC2(CCCC2)C1C(=O)NCCCCC(C)(F)F 47430,C1(C(C)NC(c2cn(CCC)nc2)=O)CCCCN1C(=O)Cn1nnc(C)n1 47431,S(=O)(=O)(c1cc(C)cnc1NC(CCO)c1ccco1)NC(CCCC(=C)C)C 47432,C(=O)(CN=c1cc[nH]cc1)NC(CN(C(C(CCC)C)=O)CC)C 47433,C1(NC(C2C(=C)CC2)=O)CN(C(c2cc(Br)cn2C(C)C)=O)CC1F 47434,C(C)(C)(CC(=O)NC(Cc1cn[nH]c1)C(N1CCC(F)(C(N)=O)C1)=O)OC 47435,C1(C(=O)NC(C)CN2CCN(C(c3ccon3)=O)CC2)CC12CCCCC2 47436,c1(CC)cc(NC(=O)CCc2ccncc2)cnc1C.C12CCCCC1NC2=O 47437,c1(C(N2CCC(C)(NC(Cc3nc(C)sc3)=O)C2)=O)cnn(C)c1C#N 47438,c1(C(=O)NC(CNC(c2cnc(CC)s2)=O)C(C)C)cnn2ccnc(N)c12 47439,N1(C(c2ccc(OCC=C)cc2)=O)CC2=C(C1)CN(C(=O)CC1(C#N)CCC1)C2 47440,C1(CNCc2cnc(C#N)c(F)c2)CC2(CCC(F)(F)CC2)CO1 47441,C1(=O)C#CC2(COC2)CC2CN1C2.C1(C(=O)NC23CC(CC)(C2)C3)CCC2CC2C1 47442,c1(C(=O)NC2CN(C(C3=CC(C)(C)C3)=O)CC23CC3)c[nH]c2ccc(F)cc12 47443,C#CCCCC(=O)NC(COC)CC(=O)N(CCCC(C)O)C 47444,C1(NC(C=C(COC)C)=O)CC2(C1)CC(NC(=O)CCC1CC1(F)F)C2 47445,CC1(F)CN(C(=O)CCOC2CC2)CCN(C(=O)CC(O)CCSC)C1 47446,C(=O)(C1CCCn2cnnc21)NCCC1N(C(c2ncn(CC)n2)=O)CCSC1 47447,c1(-n2cc(CN(C(C(C)CNS(=O)(=O)C3CC3)=O)C)nn2)ccc(O)nn1 47448,Cc1ccc(N)c(C(N2CC(C)(C)CC2CNC(c2cn(C(F)F)cn2)=O)=O)c1 47449,C(=O)(C(C)(C)C1=CCSCC1)NCC1CC(C)(C)CN1C(C1CCC(=O)C1)=O 47450,c1(CNC(CCc2onc(SC)n2)=O)cccc(Br)c1O 47451,C1(CNC(C=CC=CC)=O)CN(C)CCN1C(C1CCCN1CC(C)C)=O 47452,N1(C(C2(c3ccccc3F)CC2)=O)CCc2c(C(=O)O)cccc2C1 47453,c1(C(N(C2CN(C(=O)C(O)c3ccco3)C2)C)=O)ccc(S(N)(=O)=O)s1 47454,c1(CNC(C(C2CCN(C(C(OC)OC)=O)C2)C)=O)cnn(C)c1O 47455,CCC(F)(C(=O)OC)C(=O)N1CCOC(CN(C(=O)Cc2cnoc2)C)C1 47456,CC(N=[N+]=[N-])C(=O)NC(C1(O)CCCCC1)C(N1CCCCC1C)=O 47457,S(=O)(=O)(CCCCCl)N1CC(NC(c2occc2Br)=O)C(F)C1 47458,c1(C(=O)OC)cn(C)nc1C(=O)NCC1CC1CNC(C1CCCCC1C)=O 47459,N1(C(C(CC)CC)=O)CCCCC(CNC(=O)CCn2nc(C)c(C)c2C)C1 47460,C1(NC(CCC(N)=O)=O)CCN(C(C23CC(CN2C2CC2)C3)=O)C(C2CC2)C1 47461,c1(C(=O)NC(CNC(CC(CC)C(C)C)=O)C)c(O)cnc2cc(F)ccc12 47462,CC(C)(O)C(F)(F)C(=O)NCC1(NC(c2cc(C3CC3)ccn2)=O)CCOC1 47463,N1(C(C(C)Cc2ccnn2C)=O)CCC(CF)(NC(=O)C(C)NS(C)(=O)=O)C1 47464,c1(COC)ccc(CO)o1.C(C(=O)NCC1CCC1C(=O)N(C)C)(C1CCCO1)OC 47465,N1(C(CC2(OC)CCC2)=O)C(C(=O)N(CCCSC)C)CCC1C1CCCC1 47466,N1(CCCC(=O)NCc2c(C)cc(Cl)nc2)CC23CCCC2(C1)C3 47467,C(=O)(C(C(F)(F)F)C(F)(F)F)NCCC1N(C(c2ncn(CC)n2)=O)CCOC1 47468,Cc1cc([N+](=O)[O-])ccc1C(=O)NC1CCC1NC(=O)C(=O)NC(C)C 47469,Cc1ccc(C(=O)NCC2CCCCN(C(c3ncccn3)=O)C2)cc1Cl 47470,C1(C)(C(N(C(c2ccccc2)CNC(c2cnsc2)=O)C)=O)CC(=O)N(C)C1 47471,C1(C(N(CC(O)CNC(C2(c3ccsc3)CC2)=O)C)=O)CCCN1C1CC1 47472,N1(C(CCCn2cc(-c3cc(C(N)=O)ncc3)nn2)=O)CCCCS(=O)(=O)CC1 47473,C1(c2ccc(C)o2)CCCCCN1C(=O)COc1ccccc1Br 47474,C1(NC(C2(OC)CCOCC2)=O)CN(C(C2COCCOC2)=O)C(C)(C)C1 47475,CC1CCCC=C1C(=O)N1CCC(C(=O)N(C2CCOC2)C)CC1 47476,C(C)(C(C)(C)NC(c1cccn1C1CCCC1)=O)NC(C(C)n1cncn1)=O 47477,c1(CCCC(=O)NC2C(NC(C(CCC)NC(N)=O)=O)C2)cc(O)ccc1C 47478,CCC(C(=O)N1CCC(NC(=O)CCOCc2ccccc2)C1C1CC1)C(C)C 47479,N1(C(c2c(C)nc(C)s2)=O)CCC2(NC(c3nc(Cl)ccc3N)=O)CC2C1 47480,C(C(C)(C(=O)NCC1CCSC1)NC(c1ccc(F)cn1)=O)SC 47481,C1(N(C(CN(C)C(=O)C2CC2)=O)C)CN(C(=O)CCCCCF)CCC1O 47482,CC(C)(O)CCC(=O)NC1CCN(C(=O)C(N2CCNC(=O)C2)c2ccccc2)C1 47483,c1(C(=O)NCCC2CN(C(C3C(C)C3C)=O)C2)n[nH]c(C2CC2)c1Cl 47484,C(CCN(C)C(C12CCCC1C2(F)F)=O)(C(C)(C)C)NC(C=CC=CCC)=O 47485,c1(C(=O)NCC(C)CNC(C2CCOC(C)C2)=O)ccc2c(c1)C(=O)CCCC2 47486,c1(NC(CN(C(C2CC2(Cl)CC)=O)C)=O)cn(CCF)nc1C 47487,C1(C(=O)NC(C#C)CCC)CCCCCC1NC(C1(C)CNC(=O)N1)=O 47488,C(=O)(CCCCCCCC(=O)NCCNCc1ccc2cn(C)nc2c1)OC 47489,C(CN=c1[nH]cc(-c2cc(CO)cc(ON)c2)o1)OC 47490,C1(NC(CCc2ccc(C)cc2)=O)CC12CCN(C(C1CC1C(N)=O)=O)C2 47491,C(C1=NOC2CN(C(c3ocnc3C(F)(F)F)=O)CC12)NC(CCCC(=C)C)=O 47492,C(=O)(CC(C)(O)C1CC1)N(C1CN(C(c2cscn2)=O)C1)C 47493,Cc1[nH]c(C(=O)Nc2cncnc2Cl)c(C)c1C(=O)NCc1ncccc1Cl 47494,N1(C(c2cc(C)[nH]c2C)=O)CCCC(C)(NC(c2cnoc2C)=O)C1 47495,c1(NC(=O)NC2CN(S(=O)(=O)Cc3ccc(Cl)cc3)C2)c(Br)ccc2c1OCO2 47496,N12CCCCC(C1)NC(=O)C2=O.c1(OCC)ccc(C(C)=O)cc1 47497,c1(CC)cccc(C(N2CC(C)C(O)C2)C(=O)NC2CCOCC2)n1 47498,n1(CC(=O)NC2CCCN2C(C2(C(F)F)CC2)=O)cc(C2(C3CC3)CC2)nn1 47499,C1(C(=O)NC2(CNC(=O)CC3CCCC3)CC2)CC12CCCCCC2 47500,c1(C(=O)Nc2nc(C(=O)OC)sc2C)cncc(Br)c1C 47501,N1(NC(C(N2C(c3nc(C)[nH]n3)C3CCC2C3)=O)=O)CCn2ncc(Cl)c2C1 47502,Cc1ncnc(C)c1C(=O)NCC(F)CNC(=O)C(c1cccc(F)c1)(C)O 47503,C(=O)(CC1=CCOCC1)NCC1CCC(C(N2C(CC)CCC2)=O)CC1 47504,CCC(C)C(O)CC(=O)NCc1ccc(C(=O)NCC2CCC3(CC3)C2)cn1 47505,Cc1nc(O)sc1C(N1C(C(=O)NCC(C)N(C)C)CC1C)=O 47506,n1(CC(=O)NCC(C)N(C(=O)CCC2CCCN2C)C)cc(Cl)c(O)nc1=O 47507,c1(C(=O)NCC2(NC(=O)CC3CCC(O)C3)CCOCC2)cnc2[nH]nnc2c1 47508,c1(C(=O)NCC(CNC(C(CC)C#N)=O)F)nc2ccc(Br)cn2c1F 47509,C1(C(C)C)(C(=O)Nc2cnsc2)CCN(C(c2ccncc2O)=O)C1 47510,C12(NC(C(n3cc(CCc4ccccc4)nn3)C)=O)CCCCC(F)(C1)C2 47511,c1(C(N2C(C(=O)Nc3cnccc3I)CC(C)C2)=O)ccc(Cl)c(C(F)(F)F)c1 47512,CCCC(C(=O)N1CC2CC1C2CNC(=O)CCc1cc(C)cs1)N(C)C 47513,C1(C(N2CCN(C(c3occ(C)c3)=O)CC(O)C2)=O)Oc2ccccc2OC1C 47514,N1(c2cc(C)nc(N3CCC(C4CCCO4)C3)n2)CCC2(CCOC2)CC1 47515,C1(CC2(C(=O)NCC3CC3)CN(C(c3c(C)ncs3)=O)C2)CCCN(C)C1=O 47516,c1(C(=O)NCC2C(NC)CN(C(=O)C(O)Cn3cncn3)C2)cccc(Cl)c1F 47517,c1(C(N(C2CCCCC2)C)=O)ccc(CC2CCC(F)(F)C2)cc1 47518,C1(N(C(CC=CC=C)=O)CCOC)CCN(C(C2CCCCN2C(C)=O)=O)CC1 47519,c1(C(=O)NCCC2(O)CN(C(C3CN(CC)C(=O)N3)=O)C2)ccc(=N)[nH]c1Cl 47520,C1(NC(C=CC(N)=O)=O)CCCC2CN(C(=O)Cc3nc4c([nH]3)CCCC4)CC12 47521,N1(C(CCCC#C)=O)CCC2(NC(=O)CSc3cnn(C)c3)CCCCCC12 47522,c1(C(=O)NCC(CC)N(C)C(c2cccn2CC)=O)cc(C)sn1 47523,N1(C(Cc2nc(C(=O)OC)sc2)=O)CCC(NC(=O)C(C)(Cl)Cl)C(C)C1 47524,c1(CC)ncc(C(=O)NCC2CCN(CC3CCOCC3)CC2)c(C)n1 47525,CC1CCC2CN1OC2=O.C(CO)(C1CC1)OC(C(C)(C)C)=O 47526,c1(C(N2CC(F)(CNC(=O)CCn3cccn3)C2)=O)cc(Cl)ncc1C(F)(F)F 47527,C1(CC)CN(C(c2c(F)cccc2Cl)=O)CCC1NC(=O)CC1=CCCC1 47528,Cc1cnc(CCNC(C2C3CN(C(=O)CCCc4cnn[nH]4)CC23)=O)cn1 47529,c1(C(=O)NCC(C)CNC(C2(CCF)CCC2)=O)c[nH]cc1-c1cnn(C)c1 47530,N1(C(C2C(C)=CCS2)=O)CCC(NC(C2CS(=O)C2)=O)C(C)(C)C1 47531,CC1(C)CC(NC(C2(C3CCC3)CCC2)=O)CN1C(=O)CC1CN2CCC1CC2 47532,C1(C2CC2)(NC(c2ccc(CCC)s2)=O)CCN(C(=O)C(C)C(C)C)C1 47533,N1(C(C(C(C)C)n2cnnn2)=O)CC(NC(=O)CC2CC3(CC3)CO2)C2(CC2)C1 47534,C(C)(c1cccc(Cl)c1)=CC(=O)NC(CC)CN(C)C(c1cccc(C)c1F)=O 47535,C12(CN(C(=O)Nc3cn(CCC)nc3)C3CC3)CCC(CC1)CC2 47536,CON1CCC(C(=O)NC2CCC(CC(=O)NCCC3CCOCC3)C2)CC1 47537,C(=O)(C(C)(C)C(=O)NC(C)C(C)NC(=O)CSc1ccccn1)OCC 47538,c1(COCC(N2CC(C)S(=O)CC2)=O)nc2ccccc2s1 47539,N1(C(CC=C=C)=O)CCc2sccc2C1CNC(C12CC(C(=O)OC)(C1)C2)=O 47540,C1(C(N(C(C2CCOCC2)C)C)=O)CCCC(NC(=O)Cc2cccnc2O)C1 47541,C1(CC(=O)N(C(C)CN(C(=O)CN2CCCC2=O)C)C)CC=CCN1C 47542,N1(C(C(C)Oc2cccc(Cl)c2)=O)CC2CCN(C(C3CC=CC3)=O)CCC2C1 47543,c1(SCC#N)cccc(C(=O)NCCNC(=O)CC2CC3(CC3)C2)c1 47544,c1(C(=O)OCC(=O)N(C2CCS(=O)(=O)C2)CCC)ccc(Br)cc1Cl 47545,N1(C(C(=O)N(CCc2cccc(OC)c2)C)=O)CC2CC(C)C2C1 47546,c1(C(=O)NCC2CCCN(C(CCC=C)=O)CC2)nnc2n1CCCCC2 47547,C1(OC)(CNC(C2CCC(=O)N2)=O)CCN(C(=O)C(c2ccc(F)cc2)O)CC1 47548,CC(CN(C)C)CCC(=O)NCC(CNC(=O)CCc1ccc(F)c(F)c1)CO 47549,C(=O)(CC(C(C)(C)C)NC(c1c[nH]c(=S)cn1)=O)NC(CCC)C(F)(F)F 47550,N1(C(C(CC)(C)C#N)=O)CCC=C(C(=O)NOC(C2CC(OCC)C2)(C)C2CC2)C1 47551,CC#CCC(C(=O)NC1CCN(C(C)C)C1=O)NC(=O)CCC(C)(C)OC 47552,n1(CC)ccc(C(N2CC(NC(=O)Cn3ccnn3)CC2C)=O)cc1=O 47553,N1(C(C2OCCN(C)C2)=O)CCN(C(c2cnn(C)c2Cl)=O)CC(CO)C1 47554,N1(C(COCC(C)C)=O)CC2CC1CCC2NC(=O)CSCc1cscn1 47555,CN1CC=C(CCNC(=O)C(C2CCCO2)NC(=O)CNC=O)CC1 47556,c1(SCCCC(CCC)N)ccc2c(c1)OCCO2.C1(=O)CCCN1 47557,C1(C)(C(N(C)CC2CN(C(CNC(C)=O)=O)C2)=O)CCCO1 47558,C1(O)(C(=O)NC2COCCN(C(c3cnc(C)s3)=O)C2)CCCC(C)CC1 47559,N1(C(CN(CCC)C(c2cc(COC)on2)=O)=O)CCCC2(CC2)C1 47560,CC1=NN(C)C(=O)C1CC(=O)NC1CC(NC(C2CC(F)(F)C2(C)C)=O)C1 47561,C1(CN(C(c2c(C)coc2)=O)C)CCCN(C(C2CCC(C(N)=O)CC2)=O)C1 47562,c1(CCC(=O)NC(C)CN(C(=O)CC2CCC2(C)C)C)ccc(N)cn1 47563,c1(C2(C(N(C3CCN(C(C4CC4Cl)=O)CC3)C)=O)CC2)ccc(Cl)cc1 47564,C12(CC=CC1)C(=O)N2.c1(C(C(=O)NCC2CCN2C(C)=O)OC)ccccc1 47565,C1(C(=O)NCC(CCNC(C(N2CCOCC2)C)=O)O)CCCC(F)(F)C1 47566,C1(C)(C(N2CC(NC(CCCNC(C)=O)=O)C(C)C2)=O)CCC2(CC1)OCCO2 47567,c1(CNC(N2CCCCC2c2cccs2)=O)ccc2cc(Br)ccc2n1 47568,CC1(CNC(c2cccc(O)n2)=O)CCCN1C(=O)CCc1cnc[nH]1 47569,S(=O)(=O)(c1cccnc1)N(C)CCCSCCC(C)(C)C.C(CC(N)CO)N1CCCC1 47570,C1(C(N(C)CC2CCCN2C(c2cocn2)=O)=O)CC2C=CCC(C1)C2 47571,c1(C(C)NC(c2n(CC)nnn2)c2snnc2C)cccc(NC(C)=O)c1 47572,c1(CC)ccc(C(=O)NC2CCC(CCNC(=O)Cn3cnc(=N)[nH]3)C2)nc1 47573,C(=O)(C1CC(=O)Nc2ncccc21)NCCN(C)C(c1cnc(CC(C)(C)C)o1)=O 47574,C(=O)(C(C)(C)CCCNC(=O)CC1CC=CCN1C)NC1C(O)CCC(C)C1 47575,C(=O)(C1CCc2c[nH]nc21)NC1CC2CC(NC(CCNC(=O)NC)=O)C2C1 47576,C1(CNC(Cn2c(N)cc(C)n2)=O)CN(C(c2ccc(F)o2)=O)CC(C)(C)C1 47577,c1(NC(CC)=O)cncc(C(N2CC(NC(c3cccnn3)=O)C(C)C2)=O)c1 47578,N1(C(CCC)=O)CCCC1C(=O)N(CCCNC(=O)C(C)(C)N(C)CC)C(C)C 47579,C1(C(=O)NC2CC(C)N(C)C2)CN(Cc2cnn(CC(F)(F)F)c2)CCC1O 47580,C1(NC(c2cc[nH]c2)=O)CC12CC(NC(c1cncc(C(F)(F)F)c1)=O)C2 47581,c1(NC(=O)CC#N)ncnc2c1ncn2CC.N1(C(CC)=O)CC2CCC1(C)C2 47582,c1(C(=O)NCC(C)(C2CCC2)NC(CN(CCOC)C)=O)cccc(C(F)F)c1 47583,N1(C(c2c(O)ccc(C)c2)=O)CC2(NC(C3CCCCS3(=O)=O)=O)CCC1CC2 47584,C(=O)(CC(O)CNC(=O)CCCC1CCCC1)NC(Cc1cc(C)[nH]n1)C 47585,N1(C(C(=O)NC)c2nc[nH]n2)CCC2(CC1)C(=O)N2.CCCC(C)C(=O)NCC 47586,C1(CC(=O)N(CC#C)CC)CCCN(C(c2ccc(SC)o2)=O)C1 47587,C(=O)(CS(=O)(=O)C1CC1)NCC(C1CCN(C(COCC=C)=O)CC1)O 47588,O=C1OC2CC(C(N3CC(OCCNC(=O)C=CCO)C3)=O)CC2O1 47589,CC1(C(=O)NC2(CN)COC2)CCCN1C(C1CCOCC1)=O 47590,N1(C(C(CCC)F)=O)CCN(C(=O)CC2COC(=O)C2)CC1CCC 47591,C1(CNC(C(CC2CCC2)OC)=O)CN(C)CCN1C(=O)CC1CC1 47592,C(c1cccc(Cl)c1Cl)=CC(=O)NCCCCCCNC(=O)CC1CCOC1 47593,CONC(=O)C(=O)NCC(C1CC1)NC(c1nnc(S)n1C)=O 47594,C1(C(=O)NC2(C(=O)NC3CSCC3C)CC2)(CC)CCOCC1 47595,N(C(=NCCCCN1CCN(C)CC1)NC1CC1)CCN(CCOC)C 47596,c1(NC(CCC(CC)NC(=O)CC(=O)NC(C)C)=O)ccc2c[nH]nc2c1 47597,C(C(=O)NCC(C1CC1)NC(=O)C=CC(=O)N)=CCN(C1CC1)CC.SC 47598,CCC(CC(=O)NCC(C)(O)C1CCCC1)NC(=O)C(C)OCCOC 47599,C(=O)(C(O)CC(F)F)NC(CC=C)CNC(=O)Cc1csc(Br)c1 47600,c1(OC)cc(C(N2CCC(NC(=O)Cn3ccc(C)n3)C(F)C2)=O)c(F)cn1 47601,C(CC(CC)C(=O)NCC1CCC12CN(C(c1csc(SC)n1)=O)C2)=CC 47602,c1(C(=O)NC(C)CCNC(=O)CSC(F)(F)F)cnn(CC(F)(F)F)c1 47603,c1(SC)c(C)nn2c1CN(C(=O)OC(C)(C)C)CC2.N12CC(CC1=O)NC2=O 47604,c1(CNC(C2CN(C[Si](CC)(C)C)C2)=O)cnc(O)cc1O 47605,n1(CC)nc(C(=O)NC2(CNC(=O)Cc3ccns3)CCCCC2)cc1O 47606,c1(OC)ccc(CC(N)C(=O)NC(C)C(=O)N2CCC2)c(C)c1 47607,C1(C(=O)NCC2CCC(C#C)CC2)CC2(CCC2)CN1C(=O)CSC(C)(C)C 47608,N1(C(c2c(C)snn2)=O)CCCC(C(=O)NC2CN(C(=O)OC(C)(C)C)C2)C1 47609,C1(n2cc(CC3(O)CN(C(C4(CSC)CC4)=O)C3)nn2)CC2CCC1(C(=O)O)C2 47610,C1(F)(C(=O)NC2CCC(C(=O)NC(C)Cc3ccccn3)C2)CCOCC1 47611,Cc1cc(C(=O)NC(C2CCN(C(=O)C(c3cncnc3)C)CC2)C)ncc1Cl 47612,c1(C(N2CCC(NC(C3C(CC)C3)=O)C2)=O)cccc(OC)c1Cl 47613,c1(C(N(CCCNC(c2csc(Cl)n2)=O)CC)=O)ccc(CO)cc1 47614,C12(NC(c3nc(Br)n4ccsc34)=O)CCCC(CN(C(=O)CO)C1)C2 47615,N1(C(c2cncc(OC)c2)=O)CCC(F)(F)C(CNC(=O)C(F)=CCCF)C1 47616,S(=O)(=O)(c1ccc(F)cc1)N1C(CCNC(N2CCOCC(F)C2)=O)CCCC1 47617,c12cc(F)c(cc1F)CN2.c1(NC(C2C(C(=O)OC)C2)=O)c(OC)cccc1Cl 47618,C#Cc1cccc(C(=O)NC2(CCNC(C3CCC(C)CC3)=O)CCC2)c1Cl 47619,N1(C(CCc2cccc(OC)c2)=O)CCC2CN(C(C3CCCS3)=O)CC12 47620,C1(C(C2CCCCC2)NC(COC)Cc2nnnn2C2(CF)CCC2)CC(F)(F)C1 47621,c1(NCC(=O)NCC=CCNC(c2c(C)ccnc2)=O)ccc2ccccc2c1 47622,CC1(C)CC(CC(N2CC(O)(CNC(=O)CCCNC(N)=O)C2)=O)CC(C)(C)O1 47623,c1(CC)ccsc1C(=O)N(CC(C)C(=O)N(CC(CC)OC)C)C 47624,C1(CC(=O)NCC(C#C)CC2CC2)CN(C(=O)Cn2c(C)ccc2C)C(C)(C)C1 47625,CC1(C)CC(CNC(C2CC=CCO2)=O)N(C(c2ccnc(C#N)c2)=O)C1 47626,C1(NC(c2n(CC)ccc2)=O)CC2CN(C(C34CC3C4)=O)CC2C1 47627,N1(C(COC(C)=O)=O)CC2CN(C(c3nccc(N4CCCC4)n3)=O)CC2C1 47628,N1(C(c2c(C)nns2)=O)CC2(CCN2C(c2ncn(C)n2)=O)C1 47629,c1(CC)ccccc1C(CNC(=O)CC(C)CC)NC(=O)Cc1cnns1 47630,C1(NC(Cc2c(C)nc[nH]2)=O)CC(CC(=O)NC(C)CC(N)=O)C1(C)C 47631,Cc1cc(CC(=O)NC2CCN(C(c3csc(Br)n3)=O)CC2)nn1C 47632,N1(C(c2nc(C)sc2)=O)CCCCC(CNC(C23CC(CO2)C3(C)C)=O)C1 47633,N1(c2cc(C)nc(NC(c3ncccc3F)C)n2)CCc2nc(Br)sc2C1 47634,N1(C(CCC(=O)N(C)C)=O)CCC2CN(C(C3CCn4nnnc4C3)=O)CC2C1 47635,c1(C(=O)NC(C)CC2CN(C(=O)CC3(C(F)(F)F)CC3)C2)ccc(N)cc1 47636,c1(CN=C(NC(CC)CO)NC2CSC2(C)C)ccc(F)c(Cl)c1 47637,C1(C2CCCCO2)(C(=O)NC2CC(NC(c3ccn(CC)c3C)=O)C2)CCCO1 47638,CCC(C)C(C(=O)NCC=CCNC(c1ccc(C2CCC2)nc1)=O)OC 47639,C=CC(O)(C(=O)NCC1CCN(C(=O)C(=O)NCC(F)(F)F)CC1O)C(F)(F)F 47640,C(=O)(C(O)CC[S+](C)C)NC1C(NC(c2ncc(C)c(C)c2)=O)CCCC1 47641,CC1CC(S(C)(=O)=O)CN1C(=O)NC1CC2CC1C(O)C2O 47642,C1(C2CCC2)(C(=O)NCC(C)(C)OCCNC(C2CCC(F)(F)C2)=O)CCC1 47643,C=CCCCCCCC(=O)N1CC(CN(C(=O)CC2CCOCC2)C)C2(CC2)C1 47644,c1(C(=O)NCC=CCNC(=O)CC23CCCC2C3)cc2cccnc2o1 47645,C1(NC(C2(CC=C)CCOC2)=O)CC=C(C(=O)NC2CC3(C2)CC(O)C3)C1 47646,CC1CCc2[nH]nc(C(=O)NC3CN(Cc4ccc(F)cc4F)CCC3C)c2C1 47647,C1(NC(c2ccnc(C)n2)=O)COC2(CCN(C(c3cnsn3)=O)C2)C1 47648,Cn1cccc(C(=O)NCC23CC(CN2C(=O)C(F)C(F)(F)F)C3)c1=O 47649,N1(C(C2C(C(C)(F)F)C2)=O)CCC2CN(C(c3ccc(Br)cc3)=O)CC12 47650,CCC(CC)(CN=c1nc(C#N)[nH]cc1C)NC(C1CC2CC2C1)=O 47651,N1(C(C(N2CCCC(C)C2)=O)=O)CCCC2(NC(C3CC4CC4C3)=O)CC2C1 47652,c1(NC)ncccc1C(=O)NCCC(O)CNC(=O)CCC1CC(C)C1 47653,c1(C(=O)NCC2CC(NC(c3cccs3)=O)C2)cc2c(nc1O)CCCC2O 47654,C1(NC(C(CSC)C)=O)CCC2(CCN(C(c3ccoc3Cl)=O)C2)C1 47655,CN1CCC(N(C(c2csc(-c3ccco3)n2)=O)C2CC2)C1 47656,c1(C(=O)NC2CC(C)CN(C(c3ccncc3Cl)=O)C2)c(N)c(F)cc(F)c1F 47657,c1(OC)ccc(C(=O)NCC2CCCN(C(C3CC(=C4CCC4)C3)=O)C2)c(Cl)n1 47658,CCCCCC(O)C(=O)N1CC2=C(C1)CN(C(c1ncc(Br)cc1N)=O)C2 47659,c1(C(N(CC(C)Nc2ncc(C)c(O)n2)C)=O)ccc2nnc(O)n2c1 47660,C#Cc1nccnc1NC(=O)Cc1ccccc1NCc1cnc(SC)nc1Cl 47661,C(=O)(C(O)C(F)(F)F)N1C(C(N2CCC(C(C)C)C2)=O)C(C)C1 47662,CC(C)CC(CNC(=O)C(C)(C1CC1)NC(=O)CN1CCOCC1=O)N(C)C 47663,CC1CN2CCN1C(C(=O)NCCCCNC(=O)CCCN1CCCC1)C2 47664,c1(OC(C)(C)C)ccc2c(c1)CCN(C(=O)NCC1CC(O)C13CCC3)C2 47665,CCC(C)(O)C(=O)N1CCN(C(CNC(=O)C=CC2CCCCC2)C(F)F)CC1 47666,CC1(C)CC(NC(=O)CC2CCCC2)CN(C(c2ccc(S(=O)(=O)F)[nH]2)=O)C1 47667,C(=O)(C#CC1CC1)NC1CCN(C(CCN(C)CCO)=O)C1 47668,N1(C(CC2N(C)CCCC2)=O)CCN(C(=O)CSc2ccncc2)C(CCO)C1 47669,C(C(C)N=c1[nH]c(=NC2CSC2)c2c(ncn2C)[nH]1)(c1ccc(Cl)cc1)OC 47670,c1(C(N2CC(C)C(CNC(C3CC34CCCC4)=O)C2)=O)ccc(F)c2c1OCC2 47671,CC1(C(=O)NCC(C2CCCC2)NC(c2cc(Br)no2)=O)CC(F)C1 47672,N1(C(C(COC)C)=O)CCC2(CCCN2C(c2cncc(OC(F)F)c2)=O)CC1 47673,C1(NC(c2c(CC)scc2)=O)CC(CNC(c2cn(C)nc2OC)=O)C1(C)C 47674,C1(C(=O)NCC=CCNC(c2cc(C)on2)=O)CCn2nccc2C1 47675,Cn1ccc2cc(C(=O)NCC3CC(CNC(=O)Cc4cnc[nH]4)CO3)cnc12 47676,C1(NC(c2nc(CC)sc2)=O)CN(C(=O)Cc2cc[nH]c(=N)c2)CC2(CC2)C1 47677,N1(C(C(C)(C)F)=O)CC2(CC(C(=O)NCc3cccnc3)CO2)C1 47678,c1(C(=O)NCC(C)(C)NC(C23CCCN2CCC3)=O)ccc2c(c1)NC(=O)CC2 47679,c1(OC)ccc(C(N2CCCC2CN(C(=O)CC2CCCC2C)C)=O)cc1 47680,C1(NC(C(CCC)CNC(=O)C(C)(C)N(C)C)=O)CC(C2CCCC2)C1 47681,C1(C)(C(N2CC(C(C)(C)O)(CNC(CCSCC)=O)C2)=O)CC2CC2C1 47682,C12(C(=O)NC3CC(CC(=O)NCC4CCCCC4O)C3)CCCC1C2(F)F 47683,CC1(C(=O)NC2C=CC(CC(=O)NCCn3cncn3)C2)CCCOC1 47684,c1(OC)cc(C(=O)NCC(C)NC(c2cc(SC)oc2C)=O)c2ccccc2n1 47685,C1(c2nc(C(C)OC)nn2C)CCN(c2ccccc2Cl)S1(=O)=O 47686,C1(c2n(CCC)nnn2)(NC(c2cccc(Br)c2)C)CNC(=O)C(C)(C)C1 47687,c1(C(N2C(C)CC(NC(c3nn[nH]c3Cl)=O)C2)=O)nccc2ncccc12 47688,c1(C(=O)NC2CC(NC(CN(C3CCC3)C)=O)C2)c(F)cccc1F 47689,c1(-c2c(C(=O)OCC)cccc2)cnc(C(=O)Nc2cnc(C)[nH]2)cc1OC 47690,C1(CNC(C2(N(C)C)CCC2)=O)CCCN(C(=O)CCc2cncnc2)CC1 47691,c1(C(=O)NC(CC)CNC(=O)CC2CCCOC2)cccc(N)c1C 47692,C1(F)(CNC(C2(C(C)C)CCC2)=O)CCN(C(C2CC(F)(CO)C2)=O)C1 47693,N1(CCC(CC(=O)OCC)(C)C)CC23CCCC2(C1)CN(C)C3 47694,C1(C#N)(C(N2CCC(NC(C(C)n3cncn3)=O)(CF)C2)=O)CC2CCC1CC2 47695,C12(C(N3CC(CC(C)NC(C=CC(CC)C)=O)C3)=O)CC3CC1C2C3O 47696,C(=O)(C(C#N)C(C)C)N1CCC(C(=O)NCc2c(C)scn2)C1 47697,C1(C#N)(C(=O)NC2CC(CNC(C(C)C(F)F)=O)C2)CC2CC2C1 47698,N1(C(c2cnc(OCC)s2)=O)CCC(CCNC(=O)COc2cnn(C)c2)CC1 47699,CC1CC(C)C(C(=O)NC2CCC(CNC(c3n[nH]c(O)n3)=O)C2)O1 47700,N1(C(C(CCC)NC(c2c(C#C)c[nH]n2)=O)=O)CC(=O)NCC1CC 47701,S(=O)(=O)(c1c[nH]c(C(N2C3CCC2CN(C(c2ccon2)=O)C3)=O)c1)N(C)C 47702,N1(C(CNC(C(N2C(C)CC3(CC3)C2)=O)=O)=O)CC2(CCN(C)CC2)C1 47703,CN1CCC2CCC(C1)N2C(=O)Nc1ccnc(Oc2ccccc2)c1 47704,C(c1cc2ccccc2o1)=CC(=O)Nc1cc(-n2cccc2)ccc1F 47705,C(=O)(C(C)(C)S(C)(=O)=O)N(C1CCCN(C(=O)C(C)(C)COC)C1)CC 47706,C1(NC(C2(C)CC2(F)Cl)=O)CCC(NC(=O)Cn2nnc(=O)[nH]2)CC1 47707,Cn1ccc2cccc(C(=O)NCC(O)CCNC(C3(C)CCCO3)=O)c12 47708,CCC(CC(=O)N1CC(F)CC1CO)NC(=O)C=Cc1cn(C)cn1 47709,CC1CCCN(C(=O)CC2CCCC2)C1CCNC(c1csc(C(C)(F)F)n1)=O 47710,c1(OC)ccc(-c2onc(C(=O)NC3CC(CNC(=O)CSC)C3)c2C)cc1 47711,c1(CSC(C(=O)N(CC(CC)NC(=O)C(F)=C(C)C)C)C)ccc(F)cc1 47712,C(CC(C)CN=C(NC(C)C)N1CCC(NCC(F)(F)F)C1)OCC 47713,Nc1cnc(C(=O)NCCCNC(C2(Cc3cccs3)CCCCC2)=O)cn1 47714,C(=O)(CC(C(F)(F)F)NC(c1sccc1F)=O)NCC1C(C(C)C)C1 47715,c1(C(C)C)oncc1C(=O)NCC1CCN(c2ccccc2)C1 47716,c1(C(=O)NC2(C(N(CC=C)C)=O)CC2C)cc(CC)[nH]n1 47717,CN1C(C)(C)C(NC(=O)Nc2ccc3[nH]ncc3c2)CS1(=O)=O 47718,N1(C(C(CCCC)F)=O)CC2CCC1C(NC(=O)C(C(=O)OCC)OC)C2 47719,C1(NC(=O)CCc2cnn[nH]2)CC1C1CCCN(C(C2C3CC4C(C3)C24)=O)C1 47720,C1(C(N2CCC(CC(=O)N(CC(C)C)C(C)C)C2)=O)CC(=O)NC1=O 47721,C(=O)(CC(C)CNC(=O)OC(C)(C)C)N(CC(C)N(C(=O)Cc1cc[nH]c1)C)C 47722,c1(OC)ccc(CCNC(=O)C(=O)N(C2CC2)CC2(C)CCCC2)cc1C 47723,c1(C(c2nnnn2C2CC2)NC(c2cc(Cl)nc(Cl)c2)C)cnc2ccnn2c1 47724,C1(C(N2C(C)CCC(NC(C(c3ccn(C)n3)C)=O)C2)=O)CC2(C1)CC(C)(C)C2 47725,N1(C(c2cn(C)nc2-c2ccnn2C)=O)CCCc2cc(OC(F)F)ccc21 47726,N1(C(c2c(C)n(C3CC3)cc2)=O)CC(NC(c2ccncc2)=O)C(C)(C)C1 47727,C(=O)(CCCCCF)N(C(C)C(=O)NC(C)(C)CCCO)CC 47728,C12(C(N3CCCC(NC(C(c4cccc(OC)c4)O)=O)C3)=O)CC(N=[N+]=[N-])C1C2 47729,C=CC(C)(C)CC(=O)NCC(=O)NC1CCC(CCNC(=O)OCC)C1 47730,C(=O)(CS(=O)(=O)C1CC1)NCC1C(NC(C(C)Cc2ccncc2)=O)C1 47731,C(CN=c1ccc(C(=O)NCC2(CNC(c3ccon3)=O)CCCC2)c[nH]1)OC 47732,N1(C(C2C(C=C)CC2)=O)CC(CO)C2(C1)CN(C(c1cnc(O)c(F)c1)=O)C2 47733,C1(NC(=O)C=C(Cl)Cl)CCCCCC1NC(C1CC2CCC(C1)C2)=O 47734,CCCCCC(=O)NCCCC(C)NC(c1ccnc(N2CCCCC2)n1)=O 47735,c1(NC(C2N(C(C(C)O)=O)CC2)=O)nc(Cl)ccc1F 47736,CC(C)C(CCN(C)C(c1csc(CO)n1)=O)NC(C1(O)CC1(C)C)=O 47737,CC(C)(C)CC(O)CC(=O)NC(CCF)C(=O)Nc1conc1C 47738,C1(ON2CCOCC2)C2CNC2(C(=O)O)C1 47739,C(=O)(C(C)CCCOC)NCCN(C(=O)CCC(C)CC)CCCCCC 47740,C1(c2n(CC)nnn2)(NC2CC3CC2CC3c2ccccc2)CC2CCOC12 47741,N1(C(CC2CC(CC)C2)=O)CCOC2CN(C(C3CC3CC)=O)CC12 47742,CC1COCC(CCNC(=O)OC(C)(C)C)O1.O1NC(=O)NCC1 47743,C(=O)(C1=CC2(CCOC2)C1)N(C1CCN(C(c2ccc(O)c(F)c2)=O)CC1)C 47744,c1(C(=O)NCC(CC=C)NC(=O)Cc2ccc(F)c(F)c2)onc2c1CCCC2 47745,CCC(C)CC(C)C(=O)NC1(CNC(=O)C(C)(C)Oc2cccc(Cl)c2)CC1 47746,C(CC(=O)NCC1=CCN(C(c2sc(C#N)cc2Cl)=O)CC1)(C(N)=O)NC(C)=O 47747,c1(C(N2CCCN(C(C(C(CC)C)O)=O)CC2C)=O)cc2c(C)ccc(C)c2[nH]1 47748,N1(C(CNC(CC)=O)=O)CCC(O)(CCNC(c2c[nH]nc2C)=O)CC1 47749,Cc1cc(NC(C2CCC3COC2O3)=O)ccc1NC(=O)CSC1CCCC1 47750,c1(C(=O)NCC(CNC(C=CCCC)=O)F)cccn2cc(C(F)(F)F)nc12 47751,CC1CN(c2nnnn2CC2CCCSC2)CCCO1 47752,Cc1cccc(C2CC2C(N2CCC2CNC(=O)CSc2cn[nH]c2)=O)c1 47753,C(=O)(CCCCC(=O)NCC1CCCN(C(=O)C(C)(C)C2CCOC2)C1)NC.CO 47754,N1(C(c2cnc(C)nc2C)=O)CC(NC(C2(Cl)CC2)=O)C(N=[N+]=[N-])C1 47755,c1(C(=O)NCC2(C)C(C)CN(C(c3cc(C#N)c[nH]3)=O)C2)cc2ncccn2n1 47756,c1(CN2C(C(N3CCN(CCO)CC3)=O)CC(C)C2)c[nH]c2ccc(Br)cc12 47757,N1(C(C(N2C(C3C(C)(O)CCCC3)CCC2)=O)=O)CCCc2ncc(F)cc21 47758,C=CCC(C)(C)CCNC(c1ccc(OC)cc1)c1ccn(C)n1 47759,C12(NC(C=CCN(C)C(C3CCC(=C)CC3)=O)=O)CC1COC2(C)C 47760,C1(NC(C2C(=C)CC2)=O)CC2CC(NC(=O)CCC3CCOCC3)C1C2 47761,C12(NC(CNC(C)=O)=O)CCCN(C(=O)C(Cc3cccnc3)C3CCCC3)C1C2 47762,C1(CNC(=NC)NC2CCC(C(N)=O)C2)CNCC(C)(C)O1 47763,C1(CCCC)(C(N2CCC(C(C)(C)NC(C)C(=O)NCC)C2)=O)CCCC1 47764,CC(c1cccnc1)=CC(=O)NCC1(C(C)(C)C)CCCO1 47765,C(=O)(C1=Cc2ccccc2C1)N1CC(C)(C)C(C(=O)NCCCCCF)CC1 47766,C(=O)(CC1=CCCCC1)N1C(C)CCC(C(N2CCC2c2cnccn2)=O)C1 47767,C1(C(=O)NC(C(C)NC(=O)Cc2nncn2C(C)(C)C)CO)CC12CCCCC2 47768,CC1(C(=O)NCc2ncccc2O)CCCN(C(C2CCOC2C2CC2)=O)C1 47769,C(=O)(C1=NOC(C)(C)C1)NC(CC#C)CC(=O)NCc1ccc(O)nc1 47770,C(CC1=CCN(C(c2cc(C(C)(C)C)on2)=O)CC1)NC(c1n(C)c(Cl)cn1)=O 47771,C1(CC(n2cc(C3CCN3)nn2)C)CCCCN1C(=O)Cn1nccn1 47772,c1(Cc2nc(C(CCCCC(=O)NCC=C)=O)on2)ccc(S(C)=O)cc1 47773,c1(NC(C2C(C(=O)Nc3cc(OC)c(Cl)cc3Cl)C2)=O)ccc2c(Br)nn(C)c2c1 47774,C1(OC)CC2(CCN(C(=O)CCC3CC(NC(=O)Cn4nc(C)nc4C)C3)C2)C1 47775,c1(C(N2C(CN(C(C3CC(F)(F)C3)=O)CC)CCCC2)=O)ccn2cncc2c1 47776,c1(C(=O)NCc2ccc(C(=O)NC(C)Cc3cccs3)o2)cccc(F)c1O 47777,CCCCC(CC)C(=O)N1CCCN(C(=O)Cc2ccc(Cl)nc2)CCC1 47778,N1(C(CCC#CC)=O)CCC(NC(c2nn(C)c(Cl)c2C(F)(F)F)=O)C(C)C1 47779,O=C1CC(C2CC2)(C(=O)NC23CCC(NC(=O)C(O)C(F)(F)F)(CC2)C3)C1 47780,C1(C(=O)NCCOCCCNC(=O)Cn2cccc2)(CO)CCCO1 47781,c1(C(N2CCn3ncc(I)c3C2)=O)cc(C(F)(F)F)nc2ccccc12 47782,C(=O)(C(F)(F)C(C)(C)O)NC1(CN(C(C(C)SC)=O)C)CC1 47783,C(=O)(CC(O)CC(C)(C)C)N1CCC(C(C)C(=O)NC2CCOC2(C)C)CC1 47784,n1(CCC)cc(C(C(=O)NCCCF)N(c2cnn(C)c2)CC)c(C)n1 47785,c1(C(C)C)cccc(F)c1C(=O)NC(C)CNC(=O)C(C)Cc1cccc(Cl)c1 47786,N1(c2snc(C(C(=O)NC)OC)n2)CC(F)(F)CC1CN(C)CC1CCCOC1 47787,c1(N2CCC(CCC)C2)nccc(=NCCC2CC(n3cc(Br)cn3)C2)[nH]1 47788,N1(C(C(C)C2CCCC2)=O)CC2CCN(C(=O)Cc3ccc(F)cc3Br)CC2C1 47789,C1(N(C(CCN(C(=O)CC2CCOC2(C)C)CC=C)=O)C)CCCC(C)(C)C1 47790,C1(C(=O)OC)C(C)OCCN1C(CC(C)C)C(=O)NCc1cccc(Cl)c1 47791,c1(CC)ccc(CNC(N2C3CN(Cc4cccc(OC)c4Cl)CC23)=O)cc1Cl 47792,Cc1nc(N2CC3CC3(C(=O)Nc3cnccc3C#N)C2)c2c(n1)CCC2 47793,N#Cc1cc(C(=O)NCC2(NC(c3cn(C4CC4)nn3)=O)CCOC2)on1 47794,n1(CC(=O)NC(C)CNC(=O)Cc2cnccn2)cccc(C(F)(F)F)c1=O 47795,Cc1nn(C)cc1CNC(=O)C(=O)N(CCCCC(=O)O)C 47796,C1(CNC(C2N(CC)CC2)=O)CC(C(C)(C)C)CN(C(C2(O)CC(C)(C)C2)=O)C1 47797,C(=O)(CCC1=CCc2ccccc21)NC1C(CNC(c2nnc(C)s2)=O)C1 47798,c1(C(C)(F)F)cccc(C(=O)NCC(CO)NC(c2cccn2C2CC2)=O)c1 47799,N1(C(c2ccc(C)[nH]2)=O)CCCCC(CCC(N2C3CCC2COC3)=O)C1 47800,C1(N(C(CN(S(CC)(=O)=O)C)=O)CCF)CCCN(C(C2CC(C)N(C)C2)=O)C1 47801,Cc1cc(C(C)Nc2cc(CN3CCCCC3)ncn2)cc(C)c1 47802,c1(NC(=O)NC2CC(=O)SCC2)ccc(F)c(-c2cn(CCCO)nn2)c1 47803,C1(COC)CN(C(c2ccc(-c3ccncc3)cc2Cl)=O)CC(C)O1 47804,C1(CC)(NC(c2ccccc2C(C)=O)=O)CCN(C(=O)COC2CCCC2)C1 47805,Cc1ccc(C(=O)NC2CC(N(C(=O)CCc3cscn3)C)C2)c(F)c1C 47806,C(CCNC(C12CC(F)(C1)C2)=O)(C(C)C)NC(C(C1CCOC1)OC)=O 47807,N1(C(c2cn(C)nn2)=O)CCC2(CC1)CN(C(C1CC3CC3C1)=O)C1COCC21 47808,N1(C(C(CC(C)C)C)=O)CCC(C2CCCN(C(=O)CC3SC(=N)NC3=O)C2)C1 47809,C1(CSC)CCc2nc(C)nn2C1.N12CCN(C(C#N)C1)C(=O)C2=O 47810,CC(CN=c1[nH]c(=NCC2CC(F)(F)C2)[nH]c2c1CCC2)n1ccnn1 47811,C1(NC(COCCCC)=O)CN(C(=O)C(n2nc(C)cc2C)C)CC1SC 47812,C(=O)(CCC(=O)C(C)(C)C)NC1CCC(CCC(=O)NCC(N(C)C)C2CC2)C1 47813,Cc1ccccc1OCC(=O)NC1COCC1C(=O)NC(CO)C(C)C 47814,C(=O)(C(CC(C)C)C(N)=O)NC(CC(C)NC(c1n(CC)cnn1)=O)C 47815,c1(C(=O)NCC2C(CNC(c3cc(OC)n[nH]3)=O)C2)cc2c(cc1O)OCO2 47816,C(C(CC(C)C)C(=O)NC1(Cc2ccccc2C)CN(C(=O)CC2CC2)C1)OC 47817,CCCC(CCCO)C(=O)N1CCN(C(C2CCCN(C(C)=O)C2)=O)C(C)C1 47818,CN(S(N)(=O)=O)CC(=O)NCc1cn(C2CN(C(=O)CSc3cn[nH]c3)C2)nn1 47819,CCCCCCC(C(=O)NC1(C)CCN(C(=O)C(C)(C)C2CC2)C1)NC(C)=O 47820,c1(C(N2CC3C(CNC(C=C(C)C(=O)O)=O)(C3)C2)=O)ccnc(Cl)c1C 47821,Cc1nc(F)ccc1C(=O)Nc1cccc(OCF)c1 47822,C1(CNC(C2(OCC)CCCC2)=O)CCCC(NC(=O)COCC(C)C)C1 47823,N1(C(C(C)(C)c2nccs2)=O)CC2CCCC(NC(C3(C)CC(=O)C3)=O)C2C1 47824,c1(C(=O)NCC23C(CN(C(c4cn(CC=C)nn4)=O)C2)C3)cccn2cnnc12 47825,CCC(C)C(C)C(=O)N1CC(C)(NC(c2csc3nnsc23)=O)C1 47826,C(CC(C(=O)NOC(CO)C(C)C)NC(C1CC(C(C)C)C1)=O)=CC 47827,CCC(C(=O)NCC(CNC(=O)CC1CCC1)OC)Sc1nc(=N)[nH][nH]1 47828,N1(CCNC(C2CCCCC2)(C)C)CC(=O)N(Cc2ccc(SC)o2)C1=O 47829,c1(CC)cc(NCC2(C)OCCCO2)n2ncc(Br)c2n1 47830,C1(NC(c2nc(OC)c(F)cn2)=O)CCN(C(C2CSCN2C(C)=O)=O)CC1C 47831,C1(C(=O)NCCCc2c(C)noc2)C2CCN(C(=O)CCC(C)CN(C)C)CC12 47832,C1(NC(N)=O)CC2CCC1C(NC(C(CC)N(C)CC)=O)C2.C12CC(C1)NC2=O 47833,C(C)(C(C)(C)NC(c1ccn(CCC(F)(F)F)n1)=O)NC(C1N(CC)CC1)=O 47834,CC1CCN(CCC(=O)NCC2C(C)CCN2C(c2cc(C#N)on2)=O)CC1 47835,c1(OC)cc(OC(C)C)ccc1SCCCC(C)C1CN(C(=O)OC(C)(C)C)C1 47836,CC(C)C(C)CC(=O)NCC1(C(C)(C)O)CN(C(C2(CO)COC2)=O)C1 47837,C(c1ccc([N+](=O)[O-])s1)=CC(N1C(C(C)NC(=O)C2=COCCC2)CCC1)=O 47838,Cc1oc(C(C)(C)C)cc1C(=O)NCC1CC1NC(c1cnoc1C(C)C)=O 47839,c1(C(N(CC(CN(C)Cc2cc(C)sc2)O)C)=O)coc2ccccc12 47840,N1(C(C)(C)C)CCN(C(c2nccn2C(F)(F)F)C(=O)NCCC2CC2)C1 47841,CCC(CCCO)N=c1[nH]c(=NC(C)c2c(F)cccc2F)[nH]c2cccnc12 47842,N1(C(c2ccc(F)s2)C(=O)NC2CC2)CCCCC2(CCC2)C1 47843,C1(C(C)(C)C)CN(C(=O)C=CC2CCCO2)CCN1C(=O)C(Cl)=CCl 47844,CC(CN(C(=O)C(CCN(C)C)NC(C1CC(O)C(F)C1)=O)C)C(C)(C)C 47845,c1(C(N(C(C(C)SC)C)C)=O)cc(CNC(=O)CN(c2ccccc2)C)on1 47846,N1(C(C(C)(C)N2CCC2)=O)CCC(C2CCCN(C(C3CC3C(F)F)=O)C2)CC1 47847,c1(OC)cc(-c2cnc3cc(C(N4CCC(O)C4)=O)ccn23)cc([N+](=O)[O-])c1 47848,C1(N(C(c2cc(CCC)[nH]n2)=O)C)CCCCC1N(C(=O)C=CC(C)C)C 47849,N1(C(C(CC(C)C)F)=O)CCC2CCC(C1)N2C(c1cccc(SCC#N)c1)=O 47850,N1(Cc2cc(Cl)ncc2Br)CCc2ccc(F)cc21 47851,C(CC1c2ccccc2CCN1C(c1ccon1)=O)NC(=O)C(C1CC1)C1CC1 47852,CC1CN(C(c2cscc2C(F)F)=O)CC(CCNC(=O)C2=CCSC2)O1 47853,c1(C(N(CC(C)(C)CNC(=O)C(O)Cc2cnc[nH]2)C)=O)cc(C(F)F)ncn1 47854,C1(CC)CN(C(=O)Cc2ccc(Cl)cc2)CCC1CNC(=O)COCCCF 47855,CCCC(CC(=O)NC1CC12CCCCC2)NC(=O)C(=O)NCC1CC1 47856,c1(C(N)=O)ccccc1C(=O)NC1CCC1CNC(=O)C(C1C=CCC1)=O 47857,C1(NC(Cc2ccc(C)s2)=O)CCN(C(c2ccsc2C(F)F)=O)CC1F 47858,Cc1ncc(C=CC(=O)NCC2CCCN2C(=O)C=CC(c2cnn(C)c2)=O)s1 47859,c1(CC)ccc(C(=O)NCCC(C)N(C(=O)C=CC(=O)N(C)C)C)s1 47860,C1(CNC(C=CC(C)(C)SC)=O)CCCN(C(C2(C)C=CCCC2)=O)C1 47861,CC(C)C(O)C(C)(C)C(=O)NCC1CCC(NC(=O)CSc2nnnn2C)CC1 47862,CC1CN(CC2(c3nnnn3C(C)(C)C)CC(C)(C)C2)CC1(C)CO.C(C)(C)(C)OC 47863,c1(NCCc2cnc(C)[nH]2)ncnc(N(C)Cc2nc(=N)[nH][nH]2)c1C 47864,C1(NC(C2CC2(F)F)=O)CC2(C1)CN(C(c1ccc(OCC(F)F)cc1)=O)C2 47865,N1(C(CC(C(C)C)O)=O)CCC(CNC(=O)CN2CCCS2(=O)=O)C12CCC2 47866,C1(CNC(C2C3CNCC23)=O)CCN(C(=O)CCC2CCCC2)CC1 47867,c1(C(=O)OC(C)(C)C)cc(Cl)cc(Cl)c1Cl.C1(C(C)(C)C)C(=O)N1 47868,O=C1CNC(=O)N1CCC(=O)NC12CC1CN(C(c1ccoc1C1CC1)=O)C2 47869,c1(OC)ncc(-c2c[nH]c(=NCc3ccccc3I)s2)cc1O 47870,C1(NC(c2c(COC)cco2)=O)(CO)CCN(C(c2ccsc2SC)=O)C1 47871,c1(C(=O)NC(CCOC)CNC(c2cnco2)=O)c(C)noc1C(F)F 47872,c1(C(=O)NC2(CN=c3[nH]nc(C)s3)CCCC2)cnc2nncn2c1C 47873,N1(C(=O)NC(C)CCNS(=O)(=O)C(F)(F)F)CCCC(C)C1C1CCCO1 47874,CN1CCN(C(c2ncncc2F)=O)C(CNC(C2(F)CCOCC2)=O)C1 47875,Cc1nccn1CCCC(=O)NCC1CCN(Cc2ncnn2C)C1 47876,c1(C(=O)OCC)cnc(SC)nc1N1CC2CC1CN2Cc1ccc(SC)o1 47877,Cc1ncc(N(C(=O)CCC2CC(c3c(C)ccnc3C)C2)C(=O)C(Cl)(Cl)Cl)c(C)c1C 47878,N1(C(CCCCCSC)=O)CCC(CNC(c2cc(F)c[nH]2)=O)C(F)(F)C1 47879,Cc1nc(NC2CN(C(c3c[nH]c4c(Cl)cccc34)=O)CC2C)c2sccc2n1 47880,C1(C2CCOCC2)(NC(C2CC(CNC(=O)C=CC3CCCC3)C2)=O)CC1 47881,C1(NC(CN(C(C)C)C)=O)CCN(C(=O)C(C)(C)C2(C)CC2(F)F)C1 47882,N1(C(CCCCCC)=O)CC(NC(C2CCCNC2=O)=O)CC2(CC2)C1 47883,c1(NC(=O)Nc2ccc(-c3ccncc3)cc2)nc(C(F)(F)F)ccc1F 47884,c1(CCC(N2C(C(C)NC(C(C)=C3CCCC3)=O)CCC2)=O)ccc(N)c(F)c1 47885,CC(C)CC(CNC(C1CC1C1CCCC1)=O)C(=O)Nc1cc(O)cc(F)c1 47886,c1(OC)ccc(S(=O)(=O)Nc2cncc3ncnn23)cc1Cl 47887,c1(C(N2CCCC(CC=C)C2)C(=O)NC2(C)CC2)cc(F)cc(F)c1 47888,c1(NCCC(=O)N(CC(C)Cn2cccn2)C2CC2)cnc(C#N)cn1 47889,N1(CCC(=O)N(C)CC2(CNC(C3CC34CC(O)C4)=O)CC2)CCCC(N(C)C)C1 47890,C1(NC(COCC(C)C)=O)CCN(C(C2CN(C3COC3)C2)=O)C(C)C1 47891,C(=O)(C(CNC(=O)CCC1CCCCC1)OC)N(C1(C#C)CC1)C 47892,C(=O)(CCCC(=O)NCC(C)(Cn1cccn1)NC(c1n[nH]c(C)n1)=O)OCC 47893,C(CCc1cn(CCC[N+]([O-])=O)nn1)(C(=O)O)NC(C(C)(C)c1sccc1Cl)=O 47894,C(C(C)CC(=O)N1CC(C)(C)C1)NC(c1cn(CC=C)nn1)=O 47895,c1(CC)onc(C(N2CCC(NC(=O)CCc3cnn[nH]3)C2C(C)(C)C)=O)c1C 47896,c1(C(=O)NC2CC(CNC(C3C(C)C3C)=O)C2)cnc2ccc(F)cc2c1 47897,CC(C)CS(=O)(=O)CCC(=O)N1CC(CC(C)NC(=O)CCc2ccco2)C1 47898,C(=O)(C#CC1(C)CCCO1)N1CC(N2CCN(C(C3(F)C(C)OCC3)=O)CC2)C1 47899,N1(C(C2C(C)(C(=O)OCC)C2)=O)CCN(C(=O)C(C2CCC2)OCC)C(CC)C1 47900,C1(NC(NCC(c2ccc(OC(F)F)cc2)OCC)=NC)CCCCC1(C)C 47901,C1(NC(CN(C(=O)Cn2c(C)ccc2C)CC#C)=O)CCn2ncnc2C1 47902,c12ccccc1C(C)N2.N1(C(C)C)CCN(c2cccc(Br)n2)CC1 47903,N1(C(c2ccc(CC)[nH]2)=O)CC(C)(C)CC1C(=O)NCCC1CCCN(C)C1 47904,c1(C(=O)NCC2CN(C(c3n[nH]c(CC)c3C)=O)C2)nnc(O)nc1O 47905,C(C(C)(C)CC(=O)N1CCCCC1C1(NC(C2CCN(C)C2=O)=O)CC1)OC 47906,c1(C(=O)NCCNC(c2cn(C)c(Br)c2)=O)ccnc(Cl)c1O 47907,CCC(C)C(O)CNC(=O)COC(=O)CC1CCCS1(=O)=O 47908,N1(C(CCc2ccc(C)nc2)=O)CCN(C(=O)CC2CCCC2)C2CC12 47909,c1(C(=O)NC2C(CNC(c3n[nH]c(CC)c3Br)=O)C2)cc(F)cc(Cl)c1O 47910,CON(CCCO)C(=O)C1CC(C)(C)CN1C(c1ccc(C)cc1O)=O 47911,C1(C(=O)NCCC(CNC(C(C)CN(C)C)=O)O)COCCOC1 47912,c1(CC)c(C(=O)N(C)CC2(NC(=O)CCC#N)CC2)cnc2ncnn12 47913,c1(CC)nn(C)c(C(=O)NCC2C(C)CCCN2C(=O)C(C(C)(C)C)OC)c1Cl 47914,C1(CNC(c2noc(CC)c2C)=O)C(C2CC2)CCN1C(c1ncccc1Cl)=O 47915,C=CCCC(F)(F)C(=O)N1CC(N(C(=O)CC(C)(C)C(F)F)C)C2(CC2)C1 47916,N1(C(C(CC)N(C)C)=O)CCC(OCCCNC(=O)C(C)(C)F)CC1 47917,C1(CCC)CN(C(=O)Cc2occc2C)CC1NC(=O)C(C)CNC(C)=O 47918,C(C(=O)NC1CC(F)(F)C1)(C1=NOC2CC12)N1C(CC#N)CC(F)(F)C1 47919,N1(C(=O)OC(C)(C)C)CCC(N(CC(=O)NC2(F)CCOC2)C(c2ccco2)=O)C1 47920,c1(NC(C2CCCN(C(C(C=C)O)=O)C2)C)ncc(C)c(C)n1 47921,C1(CNC(CCCCC)=O)CCC(C)CN1C(c1ccc(Cn2cccn2)o1)=O 47922,C1(NC(CCC#CC)=O)CCCCN(C(=O)CCCNC(C)=O)C1 47923,C1(CNC(c2cn(-c3ncccn3)cn2)=O)CN(C(C2CC2C(F)F)=O)CC1O 47924,C(=O)(CC(C)(C)N(C)C)NCC(CC=C)NC(=O)Cn1cc(Br)c(C)n1 47925,Cc1cc(C(C)C)ccc1C(=O)NC(C1CCN(C(=O)CC2CCOC2)CC1)C 47926,C1(CC)C(NC(C2CC2COC)=O)CCCN1C(c1ccc(SC)o1)=O 47927,c1(C(=O)NC(CN(C(c2cc3cnccc3[nH]2)=O)CC)C)cnn2cccnc12 47928,N1(CC)CCOC(C(N2CCCC(CNC(c3ncoc3C(C)(C)C)=O)C2)=O)C1 47929,Cc1cc2ncc(C(=O)NCCC3CC(NC(C4(C)CC4(Cl)Cl)=O)C3)c(C)n2n1 47930,CC1(CNc2nccnc2F)CCN(C(=O)C(=O)Cc2cccc(F)c2)CC1 47931,C(=O)(C1=CCC(C)(C)CC1)NC(CCC)C(=O)Nc1ccsc1C 47932,C=C(Cl)CC(C(=O)NCc1cccnn1)NC(c1cc(Cl)no1)=O 47933,N1(C(c2ncn(C)n2)=O)CC2CCCC(C1)N2C(=O)CC=C(Cl)Cl 47934,CCC(C)C(C(=O)NC(c1cncn1C)CO)N(C(=O)C#CC(C)(C)C)C 47935,Cc1ccc2c(CN3CC4(CC4C(=O)Nc4c(C)cccc4Br)C3)c[nH]c2c1 47936,C1(NC(C2N(CC)C(=O)CC2)=O)CCC12CN(C(C1(O)CCOCC1)=O)C2 47937,N1(c2sc(C#N)c(Cl)n2)CCc2sc(-c3ccc(OC(F)F)cc3CO)cc2C1 47938,CCCCC(CCC)NC(=O)C(C1CCN(C(C2(CO)COC2)=O)CC1)C 47939,N1(C(c2c(C)ncn(C)c2=O)=O)CC(NC(=O)C(Cl)=CCl)CC2(CCC2)C1 47940,c1(C(=O)NCc2cccc(NC(C(CC)C(C)O)=O)c2)cc2oc(C)cc2[nH]1 47941,C1(C(=O)NC(C=C)C2CC2)CCC(C)(C)N(C(=O)CCC(C)CN(C)C)C1 47942,CCC(C(=O)NC)N(C(=O)COC1CC(N(C(C)Cc2nc[nH]n2)C)C1)C 47943,N12CCC3(CC3C1)C2=O.c1(OCCOC)cccc(Cl)c1.c12cn(nn1)CC2=O 47944,c1(N(CCCC(C)C)CC(CC)C)nnc(-c2cccc(Br)c2)n1CCC#N 47945,C=C1CCN(C(=O)C(C)CN(C)C(C2(C)CC=CCC2)=O)CC1 47946,c1(C(C)O)ccc(C(=O)NC(C2CN(C(=O)COCP(C)(C)=O)CCO2)C)cc1 47947,N1(C(C=Cc2ccc(C)o2)=O)CC(C)CCC1CNC(=O)CC1(C)CCCC1 47948,C1(C(N(CCNC(CN2CC(CC)C2)=O)CC2CC2)=O)CCc2ccnn2C1 47949,C(C(N=c1ccnc(CC)[nH]1)c1n(CC=C)nnn1)NCC1CCN(C)C1 47950,C1(NC(C(C2CC2)SC)=O)CC(C)(NC(=O)CCC=CC(C)C)C1 47951,CCC(CN=c1ccc(Br)c(S(=O)(=O)Nc2cc(C)cc(C)n2)[nH]1)OC 47952,C(=O)(C(O)C1=CCCCC1)NCC1N(C(c2c(C)nc(COC)s2)=O)CCCC1 47953,c1(CC)ncc(NC(C2CCN2Cc2ccc(Br)o2)=O)cn1 47954,CCCC(CCCNC(=O)COc1ccsc1)NC(=O)C=Cc1c(C)coc1C 47955,N1(C(c2cc(C)[nH]c2)=O)CCC(NC(C2CC(F)C2)=O)C12CCC2 47956,CC(C)CC(O)CC(=O)NC(c1nocc1C(N1CCC(N2CCC2)C1)=O)C 47957,CC1CCC(c2nnnn2C2COC2)(NCCc2cscn2)C1 47958,c1(C(=O)NC2CCN(C(C=C(C)C(C)C)=O)C2C)cc2cccc(C)c2s1 47959,c1(CC(N2C3(CNC(c4c(C)snn4)=O)CCC3CC2)=O)cc(F)c(F)cc1F 47960,n1(CC(=O)NC2C(CNC(c3c(C)nc[nH]3)=O)C2)sc2ccccc2c1=O 47961,c1(CC)cc(C(=O)NCCCN(C)C(C2CCCCN2N=O)=O)ccc1Cl 47962,N1(C(CC2(OC)CN(C(C3CSC3)=O)C2)=O)CC(CO)OC(C)C1 47963,C1(CC(C)C)CCN(C(C2CCN(C(=O)CCc3cn(C)cn3)C2)=O)C1 47964,C1(NC(C2(CCC=C)CN(C(c3cc[nH]c3)=O)C2)=O)CCn2cncc2C1 47965,c1(CC(=O)NC(C(=O)N(CC)Cc2ccncc2)C2CCOC2)cncnc1O 47966,C1(NC(C(=O)NCC)=O)COC2(C1)CN(C(c1cnc(OCC(F)F)cn1)=O)C2 47967,c1(C(=O)NC2C(C)CCN(C(c3c(C)nc(C)o3)=O)C2)c(C)nc2sc(C)nn12 47968,N1(C(C=CCC(C)(C)NC(CN2C(C)CCCC2)=O)=O)CCCC2C(=O)NCC12 47969,c1(C(N2C(C(=O)NC(C)CO)C(O)CC2)=O)cc2c(s1)CSC2 47970,C12(CCNCC1)C(=O)O2.N1(CC)CCC1(C)CCO 47971,C(=O)(C(F)C(C)CNC(c1ccc(O)cc1)=O)NCC(C1CC1)OC 47972,C12(CNC(=O)C=CC(F)(F)F)CCC1CCN2C(=O)CCN1CCCC1 47973,C(=O)(CC(O)C(Cl)(Cl)Cl)NC(C1CN(C(c2cc(CN(C)C)on2)=O)C1)C 47974,N1(C(C2N(CC)CCC2)=O)CCC(C)(CNC(c2sncc2C)=O)C1 47975,C1(CCOC)(NC(=O)CCC2CC2)CCN(CC=C(Cl)Cl)CC1 47976,c1(OCC=C)c(OC)cc(CC(C2(OC)CCCCC2)C(N)=O)cc1Br 47977,c1(OC)c(C(=O)NC2CCN(C(=O)COc3cc(C)cc(C)c3)C2)ccnc1F 47978,C1(C(=O)NCC2(NC(=O)COc3cccc(Cl)c3)CC2)CCN(CCO)C(=O)C1 47979,C(CC(O)CC(=O)NCC(C(C)(C)C)NC(=O)CSC(F)F)SC 47980,[N-]=[N+]=Nc1ccnc(NC(=O)CC2CC(O)CN2C(=O)OCC(C)(C)C)c1 47981,c1(C(=O)NC(CCC)CCCNC(=O)C(F)=C(C)C)cnc2ncccn12 47982,Cc1nc2ccc(C(=O)NC(C3CCN(C(c4nccn4C)=O)C3)(C)C)cc2s1 47983,C(C)(CNC(c1ccncn1)=O)(CC(C)C)NC(Cc1nc(C(C)OC)sc1)=O 47984,N1(C(C2CC(=C)CN2C(=O)Cc2cc(Br)ccc2Br)=O)CCC(O)C(C)(CO)C1 47985,c1(CC)nc(C)oc1C(N1CC2C(N(C(=O)C(CC)SC)C)C2C1)=O 47986,Cc1cc2c(C(N3CCC(CNC(=O)CSC(F)F)CC3)=O)cccc2[nH]1 47987,C1(C)(N(CC(=O)N(c2ccccc2)CC)C)CCCN(c2ccnc(C)n2)C1 47988,c1(N2CC(CNC(C(c3cccnc3)OC)=O)OCC2)cc(C)c([N+](=O)[O-])cn1 47989,n1(CC=C)c(N(CCc2ccccc2OC)CC)nnc1CC(F)F 47990,Cc1nc(C(=O)NCC(C)(C)CN(C)C(C2CCSC(C)C2)=O)cn1C 47991,CC1(F)CN(C(c2cccc(S(C)(=O)=O)c2)=O)CCN(C(c2cccs2)=O)C1 47992,C1(CC=O)C(=O)N(C)C(C)(C(=O)NCCOC(F)F)C1CC 47993,Cc1ncc(N)cc1C(=O)NC1COCC1NC(=O)Cc1cc(C2CC2)nn1C 47994,Cc1cccc(Br)c1S(=O)(=O)NCCCc1ccc([N+](=O)[O-])cc1 47995,CN1C(C(=O)NCC2CC3(CC3)CN2C(=O)CC2(O)CCCC2)CCS1(=O)=O 47996,c1(C(=O)NC(C=C)C)ccc(-c2ncc[nH]2)cc1 47997,Cc1nsc(C)c1C(=O)NCC1CCCC1C(N1CCC(N2CC=CC2)C1)=O 47998,C(CC(=O)NC(CO)C(C)(C)C)(C(F)F)NC(c1cc(C)n(C)n1)=O 47999,C1(O)(CCNC(C2(CC=C)CCOC2)=O)CCN(C(=O)Cn2ncc(Cl)c2C)C1 48000,c1(C(C2CCCC2)OC)nc(-c2cccs2)nn1-c1ccnc(F)c1 48001,C(=O)(C(F)(F)CC(C)C)NC1(COC)CCN(C(=O)Cn2cc(Cl)cn2)C1 48002,C1(CN(C)C(C2CCN(c3ncccn3)C2)=O)CCCOC1 48003,C(CS(=O)(=O)CC(=O)NCC1COCCN1C(c1cc[n+]([O-])cc1)=O)OC 48004,N1(C(C2C(CC)C2)=O)CC(CNC(c2cccc(CC)c2N)=O)CC12CCC2 48005,c1(C(=O)NCC(CNC(c2n(C=C)nnc2)=O)(C)O)cnc(O)c(C(F)(F)F)c1 48006,C(C(C)(C(=O)NCC(C)O)OC)OC.C1(CCOCC(=O)NCCO)CCCO1 48007,N1(C(C2(C)C(C)OCC2)=O)CC(C2(NC(c3cnnn3C)=O)CC2)C1 48008,C1(C(N(CCC(=O)NCC2CC2CC)CC)=O)CC=CCC1 48009,CCC1=NOC(C(=O)NCC(CO)NC(c2cccc(C(=O)OC)n2)=O)C1 48010,N1(C(C(C2CCOCC2)C)=O)CCC(C)(C(=O)Nc2cccc(C(F)F)c2)C1 48011,Cc1nc(C(=O)NCC2CC(NC(c3cn(C)nn3)=O)CCO2)c(C)n1C 48012,C1(CNC(c2cncc(OC)n2)C)CN(OC)CC1c1cnn(C)c1 48013,c1(CC(C)C)c[nH]c(C(=O)N(C)CCNC(=O)CC2C=CCC2)c1 48014,c1(C(=O)N(c2ncc3cn[nH]c3n2)C2(CO)CCNCC2)cc(C(=O)O)ccc1F 48015,c1(C(=O)NCCCN(C)C(C2(F)CC=CC2)=O)cc(C2CC2)nc(O)c1 48016,O=C(C(O)C1=CCCCC1)NCC1CCN1C(=O)Cc1ccc(C(F)(F)F)cc1 48017,CCCC(O)CC(=O)NCC(C1CCCC1)NC(=O)C(c1cccc(F)c1)C 48018,Cc1ncncc1C(N1CC(NC(C2OCCC2C)=O)C(C)C1)=O 48019,C(N=c1[nH]c(N2CC(C(F)F)C3(CCC3)C2)nc2c1COC2)c1c(C)cncc1 48020,c1(C(=O)NC(CC=C)CNC(=O)CCC=C=C)c(C)[nH]c2ccc(OC)cc12 48021,N1(C(c2c(C)sc(Cl)n2)=O)CCC2CC1CN2C(c1ccc(Cl)cc1F)=O 48022,c12ccc(cc1)C(=O)NC1CC21.CC(C(=O)N(C)C)c1ccco1 48023,CC1CCCN(C(=O)C=CC(C)(C)NC(C23CC2CNC3=O)=O)C1CO 48024,N1(C(C)C)C(=O)COCC1C(N1CCC(CNC(=O)CC2C=CCC2)C(C)C1)=O 48025,C(CCCCC(=O)N(C(CC(C)C)C(N)=O)C)NC(C)=O.N12C(CC1C)C2=O 48026,N1(C(CCN(C)CC)=O)CC(C)C(NC(c2nccc3cc[nH]c23)=O)C(C)C1 48027,N1(C(C(CC)C2CCC(=O)N2)=O)CCN(C(=O)CCCCCSC)CC2(CC2)C1 48028,N1(C(c2cn(C)nc2)=O)CCc2c(C(=O)Nc3cc(Br)cc(Cl)c3O)n[nH]c2C1 48029,Cc1cc(F)sc1C(=O)NCc1cccc(CN(C)C(c2nncn2C)=O)c1 48030,C1(C(C(N2CC(CNC(=O)CCn3cccn3)OCC2)=O)O)CCCCCCC1 48031,N#Cc1cncc(C(N2CCCCC(C(N3CC(CO)C(O)C3)=O)C2)=O)c1 48032,c1(C(=O)NC(CN(C(=O)C(C)NC(C)=O)CC)C)ccccc1C(F)F 48033,C1(CC)(Nc2nn(C)c(C)c2Cl)CCN(C(c2ncc(I)cn2)=O)CC1 48034,C1(NC(CC(c2ccc(F)cc2)C)=O)CCCN(C(=O)CC2COC(=O)C2)CC1 48035,c1(C(N2C(CNC(c3c(C)ncnc3)=O)CCCC2)=O)cccn2cncc12 48036,C(=O)(CCCCCOC)NC1CC(F)(CNC(c2ccnc(C(CC)C)n2)=O)C1 48037,Fc1cccc2nc(N3CCC4CC4C3)[nH]c(=NCC3(CC(F)F)CCC3)c12 48038,c1(C(N(CCC(C)NC(C(C(C)C)O)=O)C)=O)ccc(F)c(C#N)c1 48039,c1(C(N(C(C)CNC(=O)CC2CCC3CC23)C)=O)ncc(C2CC2)cc1F 48040,Cc1ccc(C(=O)NC2CC(NC(=O)CO[Si](C)(C)C)C23CCC3)nc1O 48041,c1(C(=O)NCC(C2CC2)NC(CC=C=C)=O)cccc2c1OCCN2 48042,C1(CNC(C2CC(CC)OCC2)=O)CC2CCC1N2C(C1CNC(=O)N1)=O 48043,Cn1cnc2c(NC3(C4CN(C(C5CCC(C)(O)CC5)=O)C4)CC3)ncnc12 48044,c1(COC)c(C(=O)NC2(C)CC(NC(c3ccnn3C)=O)C2)sc2ccccc12 48045,C1(NC(c2c(OC)nsc2)=O)CCN(C(c2[nH]cc(C)c2C)=O)C(C2CC2)C1 48046,CC1CC(C(=O)NC2CC(NC(c3cn(C)cn3)=O)CC2O)CN1C 48047,C(=O)(C(O)C(F)(F)F)NCCC(CNC(c1n(CC)ncc1)=O)O 48048,N1(C(=O)Nc2c(C)c(F)ccc2)CCCC12CCCN(C(c1csc(Br)c1)=O)C2 48049,c1(CCC(=O)NC(CN(CC)CC)C)ccc(C(=O)NC2(C)CC2(F)F)cc1 48050,c1(CCC)ccc(C(c2nnnn2C2CC2)NCC2CCCOCC2)cc1 48051,C1(C(=O)NCCCC(C)NC(C(C2CCCCC2)OC)=O)CN2CCCN1CC2 48052,C1(CC)(CNC(C2CN(C(=O)CC3CSC3)CC2CC)=O)CCC(=O)N1 48053,c1(C(=O)NC(C(CO)NC(C(CSC)C)=O)C)ccc(Br)c(SC)c1 48054,C1(C(=O)NCCCCN(C(C(C)C#N)=O)C)CCn2cncc2C1 48055,N(C(=NCCNS(C)(=O)=O)NCC(c1cccc([N+](=O)[O-])c1)=O)C(C#C)C(C)(C)C 48056,c1(CC(CC)NCC2(C(C)(F)F)CCOCC2)ccc(F)cc1 48057,Cc1ncc2n1CC(C(=O)N(CCCN(C(=O)CCCC1OCCO1)C)C)CC2 48058,C1(C2CC2)(NC(c2ccc(OC(C)C)cc2)=O)CCN(C(C2CC3(CC3)C2)=O)C1 48059,C1(CNC(C2C(CC)CCC2)=O)CN(C(=O)C=Cc2cnc(C)s2)CCCO1 48060,c1(C(OC)NC2(CS(C)(=O)=O)CC2)ccc(OC)cc1C#N 48061,N1(C(C2CCC(=O)NC2)=O)CCOC2CN(C(c3cnc4ccccn34)=O)CC12 48062,c1(C(N2CC(NC(Cc3cc(C)[nH]n3)=O)C2)=O)cc2cccc(Br)c2cn1 48063,N1(C(C2(NC(=O)CCP(C)(C)=O)C(C)CCC2)=O)CC2C3CCC(C3)C2C1 48064,c1(NC(c2n[nH]cc2I)=O)ccc2c(c1)CN(C(c1cncnc1)=O)C2 48065,C1(C)(CNC(C(CC)NC(C)=O)=O)CN(C(C2(c3cccnc3)CC2)=O)CCO1 48066,Cc1cccc(CC(=O)N(C2CCC(NC(=O)Cc3nccn3C)C2)C)c1 48067,C(=O)(C(F)CCC(C)C)N1CCN(C(C2N(CC)CCOC2)=O)CC1C 48068,C(=O)(C(CC(C)C)C(C)C)NC1CC2(C(C(=O)NCCOCC)C2)C1 48069,C1(CC(=O)NC(CNC(C(c2cnn(C)c2)C)=O)(C)C2CC2)CNC(=O)C1 48070,c1(C(=O)OC)c(F)ccc(COC2CCC(CONC=O)CC2)c1F 48071,CC(N=[N+]=[N-])C(=O)NCC1CC(F)CN1C(=O)CC1NC(=O)NC1=O 48072,c1(C2C3CN(C(C4C(C(=O)OC)C=C4)=O)CC32)cccc(NC(C2CCC2)=O)c1.C 48073,C1(CCC#C)CCCN1C(=O)C(CNC(c1[nH]nnc1C)=O)N(C)C 48074,Cc1nc(S)nc(C)c1CCC(=O)NCCN(C(C1CCN(C)C1=O)=O)CC1CC1 48075,C1(C(CC)C)CCN(C(=O)COC2(C)CN(C(=O)C(O)CC)C2)CC1 48076,c1(OC)ccc2c(c1)CN(C(c1nc(C(=O)Nc3cnc(C)c(C)c3)cs1)=O)C2 48077,N1(C(=O)OC(C)(C)C)CC2CC(NCc3ccn(C4CCCCC4)n3)C(C2)C1 48078,N1(C(C)=O)CS(=O)(=O)CC1C(N1CC(NC(c2cn3cccnc3n2)=O)C1)=O 48079,c1(CN2CCC(NC(C(COC)OC)=O)C2)ccncc1[N+](=O)[O-] 48080,N1(C(C(F)OC)=O)CCC2CCN(C(C3CN4CCN3CC4)=O)CC12 48081,c1(CC)nn(C)c(C(=O)NCC2CN(C(c3ccc(SC)o3)=O)CCC2C)c1Cl 48082,C1(C(=O)NCC(CN(C(C(C=C)(C)C)=O)C)C)CC(C2CCOCC2)=NO1 48083,c1(C(=O)OC)cc(=NCC2CCC(NC(c3cc(C(C)(C)C)on3)=O)C2)[nH]cn1 48084,C1(CNC(c2cnnc(O)c2)=O)CC2CCCCC2N1C(c1ncc(F)cn1)=O 48085,c1(COc2csc(CNC(C(=O)OCC)=O)c2OC(F)F)ccc(F)c(OC)c1 48086,C(CCCCCCC(=O)N(CCNC(c1cnccc1Cl)=O)C(C)C)SC 48087,CCC(CC)C(C)C(=O)NCC1(C)CCCN(C(C2(C3CCC3)CCC2)=O)C1 48088,C#CC1(C(=O)NCC2CCN(CCC)C2)CCN(C(c2cccc(=O)n2C)=O)C1 48089,N1(C(C2(CC#C)CCCCO2)=O)CC(NC(=O)CCCC2CCCC2)CC(F)C1 48090,N1(C(COCCC)=O)CC=C(CC(=O)N2CCC3CC23C)CC1 48091,c1(C(CC)(C)C)nnc(N2CCN(c3cccs3)CC2)n1CCC1CCCCC1 48092,c1(C(=O)NCC2N(CC(=O)NC(N)=O)CCC2)ccn2ccnc2c1 48093,C1(C(C(=O)N(CCCC)CC)C)CCCN(C(=O)C(OC)OC)C1 48094,c1(OC)ccc2c(=NCc3csc(Br)c3)[nH]c(NC3CCOC(C)C3)nc2c1 48095,c1(OC)cc(N)ccc1C(=O)NC1C2CN(C(C3CC3C3CC3)=O)CC12 48096,C1(c2nnnn2C)(CSc2n(C)nnn2)CCC(Cc2ccccc2)CC1 48097,c1(C(N2CC(NC(C3C(C)C3C)=O)C3(C2)CC3)=O)cc2cc(F)ccc2[nH]c1=O 48098,c1(CC)cc(F)c(NC(=O)Nc2ccnn2Cc2cccnc2)c(F)c1 48099,CCS(=O)(=O)CC(=O)N1CCCC(C)(NC(=O)CN(C)C(c2ccoc2)=O)C1 48100,Cc1cc(CC(=O)NC(C)C(C)(C)NC(=O)Cc2csc(Cl)c2)n[nH]1 48101,N1(C(CC2CC(C)C2)=O)CCC2C(CCCN2C(c2cccc(N(C)C)n2)=O)C1 48102,N1(C(c2ncn(CCNC(=O)CCOCC(F)F)c2)=O)CCC12CCC(O)CC2 48103,C1(F)(CNC(c2n(CC)ncc2Cl)=O)CCN(C(C2CC3CC3CC2C)=O)CC1 48104,c1(CC)nc(=N)[nH]c(=NCCCCNC(C2CC(N(C)C)C2)=O)[nH]1 48105,N1(C(C(C)n2ccnn2)=O)CC2(CCC(CNC(=O)CCF)O2)C1 48106,C(=O)(C1CCCc2ncnn21)NCC(=O)NCCCN(C)C(C1CCCC1)=O 48107,C1(CNC(c2on(C)c(=O)c2)=O)(CO)CCN(C(=O)Cc2cnns2)CC1 48108,C(=O)(C1=NOC(C)C1C)NC1C(OC)CN(C(=O)CCCC2CCCCC2)C1 48109,c1(NC)cc(C(=O)NCC2CCCN2C(=O)CCC2CCOC2)cc(Cl)n1 48110,C1(C(N2CCOCC(F)(CNC(C(C#C)(C)C)=O)C2)=O)CC2(C1)CC21CCC1 48111,CC(CSC(F)(F)F)C(=O)N1CC(O)(C(C)NC(c2coc(C(F)(F)F)c2)=O)C1 48112,C1(C(=O)NC(C)C(CO)NC(c2cnncc2O)=O)CN(C)CCN(C)C1 48113,CC1=C(C(=O)NC2(CC(=O)NCC3OC(=O)NC3(C)C)CC2)CCCO1 48114,Cc1nc(Cl)nc(N2CCCC(C(C)NC(=O)C=Cc3ccncc3)C2)c1F 48115,CCS(=O)(=O)CC(CO)NC(=O)CNC(c1scnc1C)=O 48116,C1(C(=O)NCC2CCN(C(=O)CN3CCCCC3)C2)CCC2(CC1)OCCO2 48117,Cn1cncc1C=CC(=O)NCc1cc(C(=O)NCCCc2ccccc2)no1 48118,C(=O)(C1CCc2cccc(F)c21)NC(CNC(Cc1ncc(C)o1)=O)(C)C 48119,Cc1ncccc1C(=O)NCc1cc(C(N2CCC(C(C)(C)O)CC2)=O)ccn1 48120,N1(C(C2CN(CC(C)C)C(=O)O2)=O)C(=O)CCC(N(C)CCC2CCOC2)C1=O 48121,c1(C(=O)NC2C(NC(C(C)(C)n3cccn3)=O)C2)cc(F)c(Cl)cc1Cl 48122,N1(C(CC(C)c2cccnc2)=O)CC2CC2(CNC(=O)CN(C)C(N)=O)C1 48123,CCCCC(CC)CC(=O)NCC1CCC2CN(C(c3ncc[nH]3)=O)CCC2C1 48124,C1(O)(CNC(=O)COC2CCCC2)CN(C(=O)CCc2cncs2)C1 48125,CC(C)C(O)C(=O)N(C(C)CCNC(=O)CCc1cnco1)C 48126,C(C)(CCC(=O)N(CCCNC(=O)Cn1nc(C)cc1C)C1CC1)SC 48127,C1(CNC(c2ccc(C)cc2C)=O)CC2COCC2N1C(=O)Cc1cccnc1 48128,c1(C(N(C2CN(C(C3C(C(C)C)(CC)C3)=O)C2)C)=O)ccc(C(C)(C)C)c(Cl)c1 48129,C12(NC(=O)CSCc3ccncc3)CCCN(c3ccn4nccc4n3)CC1C2 48130,Cc1cccc(Cc2cc(NC(=O)NC3CCNCCC3C)c(F)cc2)c1C 48131,n1(CC(=O)NC2C(SC)CN(C(C3(CO)CCCC3)=O)C2)nc(C)c(Cl)c1C 48132,CC1CC(C(N2CCCCC2C2CCC2)C(=O)NCC2CCOCC2)CC(C)C1 48133,Cc1nc(O)c(C(=O)NC23CC(C2)N(C(c2ocnc2C)=O)C3)c(C)c1[N+](=O)[O-] 48134,N1(C(CNS(NC)(=O)=O)=O)CCCC2CCN(C(=O)Cc3nonc3C)CC12 48135,c1(C(=O)NC2CCN(C(c3cscc3C3CC3)=O)C2)ccc(SC(F)(F)F)nc1 48136,c1(C(N2C(CN(C(C(F)=CC)=O)C3CC3)CCC2)=O)cc(Br)c(CC)o1 48137,C1(NC(=NCCC=C)NCC2(C3CCC3)CC2)CCOC2(CCOCC2)C1 48138,N1(C(CCC(=C)C)=O)CC(CNC(=O)CCCC)CC12CCOCC2 48139,Oc1cnc(Br)cc1Cn1nnnc1N1CCC(CCCF)C1 48140,N1(C(c2cccc(Cl)n2)C(=O)NCC=C)CCn2c(cnc2C2CCC2)C1 48141,N1(CCC)C(=O)CCC1C(=O)N(C(CNC(=O)C=C1CCSCC1)C1CCC1)C 48142,CCC1(C(=O)NCC(O)CN(C(=O)Cc2cscn2)C)CCCc2ccccc21 48143,Cc1nn(CC(=O)NCC2CCCN2CC2CCC3CC3C2)c2ncccc12 48144,C1(NC(CCC=CCC=C)=O)CC2(C1)CC2C(=O)NC(CO)C(=O)N(C)C 48145,c1(C(=O)NCC(CNC(C(C(C)(C)C)SC)=O)C)cc(Cl)c2n[nH]cc2c1 48146,Cc1cc(Cl)cc(C(N2CCOC(CN(C)C(c3ccc(F)s3)=O)C2)=O)c1N 48147,C(=O)(C1=CCOCC1)NCC(CCNC(CCC1CC(OC)C1)=O)O 48148,c1(C(N2CCC(CCOC)CC2)C(=O)NC(C)C)ccc(Br)c(C)c1 48149,CCCCCC(C)(C)C(=O)NC1CCOC(CNC(C2CCC2COC)=O)C1 48150,c1(OC)ccc(F)cc1CNC(=O)NCC1CC2(CCC2)CN1 48151,Cc1ccc(CC(=O)NC(C2CN(C(C3CC3(C)C)=O)C2)C)cc1Cl 48152,C1(C(=O)OC)CCCC1NC(=O)NCCOCc1scnc1C 48153,Cc1cccnc1C(=O)N(CC(O)CN(C)C(c1cc(CC(C)C)nn1C)=O)C 48154,CC1(C(=O)Nc2cc(O)ncn2)CCN(Cc2cccc(F)n2)CC1 48155,c1(NC2CCCN(CC)C2)ccc(S(=O)(=O)NC2CCCn3ccnc32)cc1Br 48156,c12cc(oc1C)S(=O)(=O)NC2.c1(CCNC(C)=O)ccns1 48157,C1(C(=O)OCCC2(O)CCC2)CC(F)(C(=O)OC(C)(C)C)C1.CCOC 48158,N1(C(C(C)(C)C)=O)CCCC(F)(CNC(c2cccc(C3CC3)c2Cl)=O)C1 48159,c1(CCC(=O)NCCCCNC(C2CCC2C2CC2)=O)c(Cl)cccc1Cl 48160,c1(C(=O)NC2CC(NC(C(C)C3(O)CCC3)=O)C23CCC3)cc2c([nH]1)CCCC2 48161,N1(S(c2cn(C)nc2)(=O)=O)CCC2C(CCN2S(=O)(=O)CCCCCCCl)C1 48162,C(=O)(CS(=O)(=O)CCOC)N1CC(NC(CCCCCC)=O)C2(C1)CC2 48163,C1(C=C)(C(N(CC#CC)Cc2ccsc2)=O)CCN(C(=O)CN2CCCC2)CC1 48164,c1(CCC(=O)NCC(C2CC(=O)C2)N2CCCC2)c(F)cccc1F 48165,N1(C(=O)CN2CC3CC3C2)CC2CCCN(C(C3CCC(F)C3)=O)C2C1 48166,CN1CC(C(=O)NCC(C2CC2)NC(=O)Cn2ccnn2)NC1=O 48167,C(C(=O)NNc1ccc(S(=O)(=O)N(CC)CC2CCOC2)cc1)(C(C)(C)C)SC 48168,C12(Cn3c(N4CC(CC)OC(CO)C4)nnn3)CCCN(CCC1)C2 48169,N1(C(C2C(C)CCC2)=O)CC2CCC1CC2NC(c1cnn(C)n1)=O 48170,c1(C(N2CC(OC)C3C2COC3)=O)cc2ccnc(Cl)c2s1 48171,Cc1nc2cc(C(=O)NCCN(CC(C)O)C(C3CC(=C4CCC4)C3)=O)[nH]c2s1 48172,c1(C(=O)NCCCCN(C(c2cc(C(C)=O)on2)=O)C)cc(C)c(Cl)cn1 48173,c1(N(CCN(C(C)C)C(C2(F)CCS(=O)(=O)C2)=O)C)ncc(C#N)cc1F 48174,N1(C(C(c2cnccn2)C)=O)CCCCC1CNC(=O)C1=CCOC1 48175,c1(C(C(=O)N(CCN(C(=O)Cc2cc(C)no2)CC)CC)=O)ccccc1 48176,CCC(CNC(C1(C)CCCOC1)=O)(CC)c1ccccn1 48177,N1(C(C2N(CC#C)CCC2)=O)CCC(NC(C2C(C)OC(C)C2C)=O)C(F)C1 48178,CP(C)(=O)c1ccc(C(N2CCC(CNC(=O)C3=CCCCC3)C2)=O)cc1 48179,c1(C(=O)NCC2(NC(C3CSC3)=O)CC2)cnc(C2CC2)s1 48180,c1(C(N2CC(CNC(c3c(OC)cnc(Cl)c3)=O)C2)=O)ccc(F)c(C#N)c1 48181,C1(C(N(CCCNC(=O)NC)CCNC(C(C)SCC)=O)=O)CCCCC(F)(F)C1 48182,c1(OC(C)C)ccccc1C(=O)NCC1CCCC1NC(c1ccc(C#N)o1)=O 48183,N1(C(C2(CF)CC2)=O)CCCC2(NC(C)C)CC2C1.c1(CCC=O)cccc(F)c1 48184,c1(C(=O)NC2C=CC(CC(N3CC=CC3)=O)C2)ccc2cccnn12 48185,N1(C(C)=O)CCOCC1C(N1CCC(C(C)NC(C2CCCCC2C)=O)C1)=O 48186,CC(CCNC(=O)CNS(N)(=O)=O)CCNC(=O)C(C)(C)C1CCOCC1 48187,C1(C(=O)NC2CC2(F)F)CC12CCN(C(c1cccc(Br)c1)=O)CC2 48188,CC(CC(F)(F)F)C(=O)N1CC(CCNC(c2cc(=O)cc(Cl)[nH]2)=O)C1 48189,C1(CCCC)CN(C(C23CCC(C2)C3(C)C)=O)CCN1C(=O)Cc1conc1C 48190,C1(C(N2CCOCC2CNCc2ccc(Br)[nH]2)=O)CCCCC1(F)F 48191,c1(C(=O)NCCC2(NC(c3c(C)n(C)cn3)=O)CC2)cccn2c(C)cnc12 48192,CC1(NC(=O)Cc2csc(C(F)(F)F)n2)CN(C(=O)CC2CC3(CC3)C2)C1 48193,N1(C(C2C(CC(C)C)C2)=O)CC2CN(C(=O)Cn3ccccc3=O)CCC12 48194,C1(CNC(C(CC)(CC)CO)=O)CCN(C(C2(C(=O)OC)CC2)=O)CCC1(F)F 48195,CCCCCCC(C)C(=O)N1CC2CN(C(c3cc(Cl)cc(OC)c3N)=O)C2C1 48196,Cc1nc[nH]c(=NCC(C2CC2)NC(=O)C(c2c(C)nn(C)c2C)=O)c1C#N 48197,c1(C(N2CC(NC(CCCC)=O)C(C)CC2)=O)ccc2cccnc2c1 48198,C12(CNC(CN(C3CCSC3)C)=O)CCCC1N(C(C1OCCCO1)=O)CCC2 48199,N1(C(C(COC)COC)=O)CCN(C)C(C(=O)NCCCN(C)C(C)=O)C1 48200,CCCC(C)(C)C(=O)NC(C)C=CC(=O)NCC1(C)CC2(CC2)C1 48201,N1(C(C(C#C)(C)C)=O)CC(NC(c2ccccc2C2CCOC2)=O)C(N=[N+]=[N-])C1 48202,CCCC(C)CCNC(=O)C(C1CCN(C(c2ccccc2O)=O)CC1)C 48203,C1(N(C(=O)CCOC(N)=O)C)CCCC(N(C(=O)CN2CCC(C)(C)C2)C)C1 48204,N1(C(C(CNC(C(C=C=C)C)=O)C)=O)CCN(C)C(C)C1 48205,c1(C(=O)NC2CC(C)N(C(=O)CC3CC=CCC3)C2)cnc2cccnc2c1 48206,Cc1cc(NC(C2CCCCCC2)C)ncc1C(F)(F)F 48207,C1(=O)CC(C2CC2)C(C(=O)N(CC)CC2CCCCO2)N1.C1(C2CC2)CCOC1 48208,C1(C(=O)NC(C=C)(C)C)CCC(C2CC2)N1C(c1cc(Cl)cs1)=O 48209,N1(C(c2cn(CC)nn2)C(=O)NCCCC2CC2)CC2(CO)CC2(C(F)(F)F)C1 48210,C1(C(=O)NCC(C2CCCCC2)NC(C2(C)CCNC2=O)=O)CC12CCSCC2 48211,N1(C(C(CC)(C)C)=O)CCC(C2CC2)C1CNC(=O)CSc1ccccc1 48212,N1(C(c2scc(OC)c2)=O)CC(C2CN(C(c3nc(C)[nH]c4nccc3-4)=O)C2)C1 48213,c1(-c2nc(C(N3CCOC4CC34)=O)sc2)cccnc1C(F)(F)F 48214,C(=O)(C(C)CC(C)(C)C)N1CCCC(NC(c2ccc(OC)nc2C)=O)C1 48215,C#CCC(CC(=O)NC(CC)C(C)(C)C)NC(C1CS(=O)C1)=O 48216,c1(CNC(C=C2CCC(C)CC2)=O)nc2c(s1)CCN(C(=O)Cc1nccs1)C2 48217,C(CC1CC1)(C(=O)NCCCC1CC1)N(CCCF)C 48218,N1(S(C(=O)C#N)(=O)=O)CC2CCN(C(C3CC=CCC3)=O)CCC2C1 48219,C12(C(=O)NCC(CNC(c3ccn4ncnc4c3)=O)O)CCC(O)(CC1)CC2 48220,C1(CCC(=O)NC(C#C)C2CC2)CCCN(C(=O)CC(O)c2ccccc2)C1 48221,C1(CCNC(C(C)(C)OC)=O)C(C)CCCN1C(=O)C(=Cc1ccc(C)cc1)C 48222,C1(NC(c2c(C)ncs2)=O)CC2CC(NC(=O)C(O)CC(C)C)CC2C1 48223,C1(NC(c2nn(C)c(C(F)F)c2)=O)CC2CCC(C1)N2C(=O)C(O)C1CCC1 48224,C1(NC(N2CC(CCNC(c3ccccc3)=O)C2)=O)CCC2C(CC1)C2(F)F 48225,N1(C(c2cc(C)ncn2)=O)CCC(C2CCN(C(c3ccccc3C)=O)C2)C1 48226,C(=O)(CCCC(C)(C)C#N)NCC1C(C(=O)NCCc2cnc(C)[nH]2)C1 48227,C1(C(=O)NOC(CSCC(=O)OC)=O)N(CC2CCCO2)CC12CCCC2 48228,Cc1n[nH]c(C)c1SCC(N1CCC(C)(NC(=O)C(C)NCCN(C)C)C1)=O 48229,C1(CNC(Cn2nc(C)oc2=O)=O)CC(C(=O)NCC(C)F)=NO1 48230,CCC(C)(COC)C(=O)NCC(C1CC1)N(C(=O)Cn1cccc(C)c1=O)C 48231,c1(C(=O)NC2CCC(NC(c3c(Cl)cn(C)n3)=O)C2)cc(F)ccc1Cl 48232,S(=O)(=O)(c1cc(Br)cc2c1OCC2)NS(CC1(Cc2ccc(C)cc2)CC1)(=O)=O 48233,Cc1c(C(=O)NC(CNC(c2cc(C3CC3)[nH]n2)=O)C(C)C(C)C)cc(O)cc1N 48234,CCS(=O)(=O)CCCNC(=O)NCC1CCC(C2CC2)C1 48235,C(=O)(C1CCCc2c[nH]nc21)N1CC(CNC(CC(C=C)C)=O)C1 48236,C12(CNC(C3C(OC)CCC3)=O)CCC1CN(C(=O)Cc1cccc(F)c1F)C2 48237,c1(N2CCCN(CC=C)CC2)nc(=NC)nc(N2CCn3nncc3C2)[nH]1 48238,C12(C(=O)NCCCOC(=N)O)CC(CN1C(=O)CC1CCOC1)C2 48239,O=C(C#CC1CCOCC1)NCC1CN(C(c2ccc(C(F)F)o2)=O)CC1(F)F 48240,c1(C(=O)NCC(C2CC2)NC(C(C(=O)OCC)OC)=O)cc(S(C)(=O)=O)oc1C 48241,C1(CC)CN(C(=O)Cc2cc(C)n(C)n2)CCC1CNC(=O)C(CC)(CO)OC 48242,c1(NCCCc2n(C)ncc2)ccc(S(=O)(=O)N2CCC(CCN(C)C)C2)c(Br)c1 48243,CC(CS(C)(=O)=O)C(=O)NCCN(C(=O)C=Cc1cnccn1)C 48244,S(=O)(=O)(c1cc(-c2ccccc2)no1)C1(N(C)C)CCC1 48245,C#Cc1cccc(C(N2CC(CC(=O)NC3(CC)CCCOC3)(OC)C2)=O)c1C 48246,c1(C(=O)NCC(C)N(C(c2c(C)nns2)=O)C)cc(C2(Cl)CC2)n(C)n1 48247,C(=O)(C(C)(C)C(C)NC(c1ncccc1C)=O)NC(CCC)CC 48248,S(=O)(=O)(c1ccc2c(c1)CCO2)N1CCN(C(c2c(C)nc(C)s2)=O)C(C)C1 48249,CC(C)CC(O)C(=O)NCC(CNC(c1cncc(N(C)C)c1)=O)CO 48250,CC(C)CC(C)(O)CNC(c1cc(CNC(C2(C)CC2C)=O)ccn1)=O 48251,c1(C(N2C(C(=O)NCc3scc(C)n3)C(C)CC2)=O)ncn2c1CCC2 48252,CCCC(CNC(c1coc(C(C)C)n1)=O)C(=O)Nc1cn(C)nc1O 48253,C1(CNC(CCN(CCC)C)=O)C(C2CC2)CCN1C(c1cnc(CO)s1)=O 48254,C1(C(N(CCNC(CCOCC)=O)C(C)C)=O)CCC(N2CCOCC2)CC1 48255,C=CCCCCCCCC(=O)N1CC2(CCCC(CNC(C3(O)CCC3)=O)O2)C1 48256,Cc1cc(Br)c(Cl)cc1NCC1CCN(C(=O)OC(C)(C)C)CC1C 48257,C(=O)(C1CCc2c(Cl)cccc21)NC1CN(C(CC)=O)CC1C 48258,c1(NC(C)=O)nc(C(=O)NCC(C)NC(C2CC23CC3)=O)cs1 48259,c1(C(=O)NC2C(CNC(c3cc(SC)oc3)=O)CC2)c(F)ccc(C)c1F 48260,N1(C(C2(CCCC)CCC2)=O)CC(NC(=O)Cc2coc(C(F)F)n2)C(C)C1 48261,C1(C)(NC(CN(CC)CC)=O)CCCCC1C(=O)NCCc1ncon1 48262,N1(C(Cc2nc(CNC=O)sc2)=O)CCC(NC(c2cc[nH]n2)=O)CC1 48263,c1(C(N(C2CCN(C(c3ccc(CC)s3)=O)C2)CC)=O)c(OC)nsc1OC 48264,C1(OC(CCCOCC(C)C)=O)CCCC(C(C)(C)C)CC1 48265,C(C(=O)NCCC1CN(C(c2cnccc2Br)=O)C1)(C(C)(C)C)NC(C)=O 48266,N1(C(C(C)(CO)NC(C)=O)=O)CC(NC(c2ccn(CC(C)C)n2)=O)C2(CCC2)C1 48267,C(CO)(C(C)NC(=O)Cn1nnnc1C(C)C)N(c1ccccc1)CC(=O)OC 48268,C(C(C)C(C)C(=O)NCCOCCN(C)C(c1cc(C)nn1C)=O)OC 48269,C1(CC#C)CN(C(C2CCN2C(=O)COCC2CCCO2)=O)CCO1 48270,C1(Cl)(C(=O)NC(CNC(C2CC(SC)C2)=O)C)CC12CCOCC2 48271,N1(C(CC(C)c2ccco2)=O)CC2(CCCC(CNC(c3cc(Cl)no3)=O)O2)C1 48272,c1(C(N2CC3(CN(C(c4cccc(C)c4)=O)C3)C2)=O)c(N)cc(Cl)nc1Cl 48273,C=CCC(CC=C)C(=O)NCC1CN(C(=O)CC2CCC(=O)NC2=O)CCN1C 48274,c1(C(=O)NCCC(CCC)C)ccc(CS(C)(=O)=O)c(F)c1 48275,c1(C(=O)NC2CCCN(C(c3c(NC)scn3)=O)C2C)cccc(C=C(F)F)c1 48276,c1(NC(CC)CC(C)O)ncccc1S(=O)(=O)NCCCc1nncs1 48277,Cc1nccc2cc(CNCC3CCCOC3(C)C)[nH]c12 48278,c1(C(=O)NCC(C)N(C(=O)CCCN(C)C)C)cccc2cncn12 48279,c1(CNC(C2(C#C)CC2)=O)nc(C)c(C(=O)N(CCCCC(=O)OC)C)o1 48280,C(N=c1[nH]c(=NC(C)CC(C)(C)N(C)C)c2ncccc2[nH]1)c1sc(C)c(Br)n1 48281,C1(C2CN(C(C=CC)=O)C2)CN(C(=O)CN2CCC(=O)CC2)CCO1 48282,Cc1cn2c(n1)CCC(C(=O)NC1CCC1NC(c1ccccc1[N+](=O)[O-])=O)C2 48283,C(=O)(C(C)(C)CC(=O)OCC)N1CCC(N(C(C(CC(=C)C)C)=O)CCC)C1 48284,C(CCCCC(=O)NC1CCOCC1C(=O)NC(C)(C)CCCF)(OC)OC 48285,c1(C(N(CCCCCNC(CCC(=O)OC)=O)C)=O)c(F)ccc2cnn(C)c12 48286,C(C(=O)NC1CC(NC(c2nc(C)[nH]c2C(F)(F)F)=O)C1)(C(C)(C)C)NC(C)=O 48287,Cc1csc2c(C(N3CC4CC(NC(=O)Cn5cnnn5)CC3C4)=O)ncnc12 48288,C(=O)(C(O)CCC(F)(F)F)N1C(C(C)C)C(NC(C2CCSC2)=O)CC1 48289,C1(C(=O)NC2CCC(NC(C3C(C(=O)OC)CC3)=O)CC2)CCc2nncn2C1 48290,c1(C(N2CCC(N(C(=O)CC(C)F)CC)CC2)=O)ccc(-n2cnnn2)c(C)c1 48291,C1(CNC(C2CCC(C)(C)CO2)=O)N(C(c2cnoc2)=O)CCCC1(C)C 48292,c1(C(=O)NC2C(NC(C(C)n3ccnn3)=O)CCC2)cccc(Cl)c1Cl 48293,C1(C(=O)NC(C(=O)NCCCN=[N+]=[N-])C2(C)CC2)CCCC(=O)C1 48294,N1(CC(COCC(C)C)O)CCC(N(C)C(c2cnon2)=O)CC1 48295,C(=O)(C1=CC2C=CC(C1)C2)N1CC(N(C(=O)CSC(F)F)C)OCC1 48296,C(C1CCCC1)=CC(=O)N(C(C)C(=O)N(CC(O)CCC)C)CCC 48297,N1(C(C(C)NC(CC)(C)C)=O)CC(C)C(NC(C2C3CC4C(C3)C24)=O)C(C)C1 48298,Cc1ccc(=O)n(CC(=O)NCC2(O)CN(C(C3CCN(C)S3(=O)=O)=O)C2)n1 48299,c1(CNC(c2nccn2C)CC)c(C)cc(C)cc1C 48300,c1(C(=O)OCC)ncccc1S(=O)(=O)NC(c1ccccc1F)CN(C)C 48301,CC1(CNC(C2CCCC3(CC3)C2)=O)CN(C(c2cn3ccnc3s2)=O)CCO1 48302,C1(NC(COC2(C)CCC2)=O)C2CCCN(C(=O)CN3CCNC3=O)C2C1(C)C 48303,c1(C2(C)C(C(=O)NCC(=O)NCCc3ccccc3)C2)ccc(Br)cc1 48304,C12(CO)COC(CCN1Cc1n[nH]c3cccnc13)C2 48305,c1(CC(N2CC(COC)N(C(C3CCCO3)=O)CC2)=O)ccc2c(c1)CCN2C 48306,N1(C(CC(CCC)O)=O)CC2CCC(C1)C2NC(c1cc(C)cc(F)c1)=O 48307,c1(NC(c2c(C)nns2)=O)cnc(F)cc1C(=O)Nc1cccc(CCO)c1 48308,C1(NC(c2ccsc2C(F)F)=O)CN(C(C2CCCC(O)C2)=O)CCC1CO 48309,Cc1ccc(F)cc1C(N1CCCC1CC(=O)NCC1CCC(F)(F)C1)=O 48310,N1(C(Cc2cn(CC)nc2)=O)CCCC(CCCCNC(c2cn(C)nn2)=O)C1 48311,C(=O)(CS(=O)(=O)Cc1cccs1)NC(CNC(C(C)=C1CCC1)=O)(C)C(C)C 48312,C1(CC)CN(C(=O)C(C)(C)C2CCC2)CCC1NC(c1cc(O)cc(F)c1)=O 48313,CCC(C)(CNC(=O)C1=NOC(CNC(c2cc(C(N)=O)co2)=O)C1)C(N)=O 48314,S(=O)(=O)(c1cccs1)NCC(=O)NCC(C)CNC(=O)Cn1cccnc1=O 48315,C1(N(C(=O)C=CC(F)(F)F)C)CCN(C(C2CC(=O)OC2(C)C)=O)C12CCC2 48316,c1(C(=O)NCCC2N(C(C3(OC(C)=O)CC3)=O)CCC2)cnc2onc(C)c2c1 48317,c1(OC)nccc(Br)c1C(=O)NC(N1CC(O)(Cc2cc3occc3[nH]2)C1)=O 48318,C(=O)(C(C)CS(C)(=O)=O)N1C(COC)CN(C(=O)CCc2cnoc2)CC1 48319,c1(CN(C)C(=O)Nc2c(SC)ccs2)ccc(F)c(C)c1 48320,N(C1CCCn2cnnc21)C(=O)NCC(c1cc(OC)cc(F)c1)N(C)C 48321,C1(CNC(C2CCCC(C)C2)=O)CC2(CC2)CN1C(=O)CCCN1CCCC1 48322,c1(N(C)Cc2nccs2)ccc(Br)c(S(=O)(=O)NC2CCCC(C(F)F)CC2)n1 48323,N1(C(C2CC(OC)C2)=O)CCCC(C)(NC(=O)COCc2ccncc2)C1 48324,CS(=O)c1ccc(C(N2CCOC(C3CN(C(C4CCC4)=O)C3)C2)=O)cc1 48325,CC(C)(C)C(CO)C(=O)NCC(F)CNC(=O)CCc1cccc(C(F)(F)F)c1 48326,C(=O)(C(F)C(F)(F)F)N(CCCN(C(C(N1C(C)CCC1C)C)=O)C)C 48327,c1(C(N(C(C)CN(C)C(c2ccc(CO)c(F)c2)=O)C)=O)sccc1S(C)(=O)=O 48328,C1(NC(c2cnco2)=O)CC(O)(C2CCN(C(c3ccccc3)=O)CC2)C1 48329,CCCC(CC)CC(=O)N1CCN(C(C2SC3C=CC2CC3)=O)C2(CC2)C1 48330,c1(C(=O)NCC23CC2CN(C(=O)C2=C(Cl)CC2)C3)ccn2c1CCCC2 48331,N1(c2ncnc(=N)[nH]2)CCC2(CC1)CN(C(=O)CC1=CCCCC1)CCC2CO 48332,C1(C(N2CCCC(C)C2)=O)CCN(C(=O)CCCC2CCC2)C12CCC2 48333,N1(C(CC(CC)O)=O)CCCC(C2CC2NC(c2cc(C)cs2)=O)C1 48334,N1(C(C2CCCCC(=O)N2)=O)CCCC12CCN(C(C1(F)CC=CCC1)=O)CC2 48335,C1(C(=O)NC2CCN(CC(=O)Nc3ccccn3)CC2)CCc2ncccc2C1 48336,C(CC(O)C(=O)N(C)CC1CCN(C(=O)CCOC2CCN(C)CC2)C1)SC 48337,C(=O)(C(O)C(C)(C)C)N1CCN(C(CNC(C(C2CCC2)OCC)=O)C)CC1 48338,c1(NC(c2scc(-c3ccc(OC)c(OC)c3)n2)=O)c(Cl)nc(C)nc1Cl 48339,C1(C(=O)NCC(C)(F)CNC(C2CC(F)C2)=O)CCOC1(C)C 48340,CC(C)(C)CC(O)CC(=O)NC1CC(C(=O)Nc2ccc3occc3c2)C1(C)C 48341,C1(C(=O)Nc2cc(C)sc2)CN(C)CCN1C(C1CC(C2CC2)=NO1)=O 48342,c1(NC(C(CC)(F)F)=O)cc(NC(=O)CC2CCC2OC)cc(C)c1 48343,C(=O)(CCC(C)NC(C1CN(C(=O)C(C)c2cc[nH]n2)CC1C)=O)OC 48344,C(=O)(C(CC1CC1)CC1CC1)N(CC(c1ccccc1)NC(C(CC)O)=O)C 48345,c1(OC)cc([N+](=O)[O-])ccc1NC(=O)NC1(C(C)Sc2ccc(OC)cc2)CC1 48346,N1(C(CSCCN)=O)CCOC(Cc2cn(-c3ccccc3)nn2)C1 48347,C1(NC(C(F)=CC)=O)CCN(C(c2cccc(N)c2OC(C)C)=O)CC1O 48348,CN1CC=C(CC(=O)N2CCC3CCN(C(=O)CN4CCCNC4=O)C3C2)CC1 48349,c1(OC)nc(N2CCN(C(=O)Cc3cc(Cl)cc(Cl)c3)CC2CO)ncc1Br 48350,C1(CNC(c2ncc(C)cc2C)=O)CC2CCCC2N1C(c1cc(Cl)ns1)=O 48351,N1(C(C(CSC)OC)=O)CCC(C2CCN(C(c3cnc(C(C)C)s3)=O)CC2)C1 48352,C(=O)(CC(O)CN(C)C)NC(C(c1ccccc1)NC(Cc1c(C)scc1)=O)C 48353,C(CC(N)=O)(c1cn(CCCC(=O)O)nn1)NC1CC(CCSC)C1 48354,N1(C(CCCC#C)=O)CCC(C(N2CCC(C)(NC(C)=O)C2)=O)C12CCC2 48355,C1(NC(=O)COCC2CC2)CCC2(CC1)CCN(C(=O)C(F)C(F)(F)F)C2 48356,NC1(C2CCN(C3(C(=O)NC4CCCCC4)CCC3)CC2)CC1 48357,C(=O)(CCS(=O)(=O)NC)N1CC(C)(NC(C2N(CC)CC2)=O)C1 48358,C1(C(=O)Nc2ncccc2-c2ccccc2)CCCCC1NCc1ncco1 48359,c1(C(N2CC(O)(C(C)NC(Cn3c(C)ccn3)=O)C2)=O)ccnc(CN(C)C)c1 48360,C1(C(N2CCC(C)(NC(c3cc(C)nn3C)=O)C2)=O)Cc2nnsc2S1 48361,C(CC(C)C)(CS(C)(=O)=O)NC(c1cn(CCC)nc1C)c1nnnn1C1CC1 48362,C1(NC(c2c[nH]nc2-c2ccccc2)=O)CCCCN(C(=O)C(F)(F)CF)C1 48363,Cc1ccc2c(C(N3CCNCC34CCCC4)=O)ncnc2c1 48364,CC#CCC(C(=O)Nc1ccc(Cl)nc1C)NC(=O)C(O)CN1CCCC1 48365,c1(C(N2C(C(=O)Nc3c(COC)scc3)CCC2)=O)cc(=O)n(C)cn1 48366,c1(C(=O)OC)c(NC2(CC(=O)N(CCCN(C(=O)C)C)C)COC2)n[nH]c1C 48367,C1(OC)CC(CCNC(=O)CCN2CCCCC2=O)N(C(=O)CCS(C)=O)C1 48368,N1(C(c2ccn(COC)n2)=O)CCCC12CCCN(C(=O)C(C)CC(C)(F)F)C2 48369,C12(C(=O)NC(c3cnc(C)s3)C)C(NC(=O)Cn3cnnn3)C3CC1C2C3 48370,c1(C(=O)NCC2(O)CCCN(C(COC(CC)(C)C)=O)C2)ccc(C#N)c(O)c1 48371,C=CC(C)(C)C(=O)N(CCCNC(=O)C(=O)NCCCN1CCCC(C)C1)C1CC1 48372,Cc1nc2ccccc2cc1C(=O)N(C)CC1CC(F)CN1C(=O)C(C)O 48373,CN1CCCC(CNC(=O)C(O)CNC(c2ccccc2F)=O)C1 48374,c1(C(C)C)ccc(NC(C2(N(C)C(C3(CO)COC3)=O)CC2)=O)cc1O 48375,C1(F)(CNC(CSC)=O)CCCN(C(c2ccc(F)cc2F)=O)CC1 48376,Cc1cc(CC(=O)NC(C)(C(=O)N2CC(OC(=N)O)C2)C2CCC2)nn1C 48377,n1(CC(=O)NC(CN(C(c2cnn(COC)c2C)=O)C)C)nc(C)c(Cl)c1C 48378,C1(C(N(CCOC)C)=O)CCCCC1(C)NC(c1cnc[nH]c1=N)=O 48379,N1(C(C(c2cccs2)SC)=O)CC2(C1)CN(C(c1ccc(Cl)cc1F)=O)C2 48380,C12(CC#N)CC(CN1CC1C(O)CCN1C(=O)OCc1ccccc1)C2 48381,C=C(CNC(C1CC(C)CO1)=O)CCNC(=O)CNC(N1CCCC1)=O 48382,N1(C(C2C(C)CCCC2)=O)CCC=C(C(=O)NCCCOC2CC2)C1 48383,Cc1ccc(F)c(O)c1C(N1CC(CNC(=O)CCc2ccon2)C(C)C1)=O 48384,C1(CC(=O)O)CCCCCN1C(=O)CCc1nc(C23CCCCC2C3)no1 48385,C1(CC(=O)N(CC(C(=O)NCC(C(=O)NC)O)C)C)NC(=O)NC1=O 48386,CC1=C(C(=O)NC2CCOCC2NC(C2CC(CN(C)C)C2)=O)CCS1(=O)=O 48387,C12(C(=O)NC(C(CO)SC(C)C)C)CCCN1CC(O)C2 48388,CCC(C)C(=O)C(=O)N1CCC(C)(C(=O)NCC2CCCC2)C1 48389,c1(C(=O)NC2C(C)(C)CN(C(C3(F)CCOCC3)=O)C2)c(F)ccc2occc12 48390,C(C(C)(CC(C)C)NC(=O)CCc1cc(C)n(C)n1)NC(C=C(C)Cl)=O 48391,Cc1c(C(=O)NC2CC2NC(c2ccc(C(C)C)o2)=O)cnn1C1CC1 48392,N12CCC(O)C(C(=O)O)(C1)C2=O.Cc1nn2c(C)c1-2.CC(F)(F)F.N(C)C 48393,c1(CN(C)CC2CCN(C(=O)CCCCc3cccs3)C2)ccc(C#N)cc1 48394,C=C(Cn1cc(CNC(=O)COC)nn1)C1CCOCC1 48395,C12(NC(=O)COCC3CC3)CCC(C(=O)NCC(F)Cl)(CC1)C2 48396,N1(C(c2nc(C(F)(F)F)cs2)=O)CCC12CN(C(C13CCCCC1C3)=O)C2 48397,N1(C(c2ccc(C(N)=O)nc2)=O)CCCCC(NC(C2C=CCS2)=O)C1 48398,N1(C(C2CC(C)(c3ccccc3)C2)=O)CCCCC12CC2 48399,C1(C(=O)NC2C3(CC(OC)C3)C2)CCC2(CC2)N1C(=O)C(C)N=[N+]=[N-] 48400,N1(C(CCn2ncc(C)c2)=O)CCC2(CC1)CC2NC(C12CCCC1C2)=O 48401,c12nccc(n1)N(C)CC1CCN2C1.N1(C(CN(CCC)C)C)CCCC1 48402,c1(OCCC)cccc(C(N2CC(O)(C(C)NC(=O)CC3(C)CCC3)C2)=O)c1 48403,c1(C(=O)NCCN(C(=O)C(C)(C)CF)CC(C)O)c[nH]c2cc(F)ccc12 48404,CN=c1nc(C(N2CC(NC(=O)C(C)(C)C(F)(F)F)CC(O)C2)=O)cc(C)[nH]1 48405,N1(C(C2CC(=C)C2)=O)CCC2OCCN(C(c3ccc(C(F)F)cc3)=O)C2C1 48406,N1(C(CC=CC)=O)CCCC2(CCC2NC(C2CCCCO2)=O)C1 48407,n1(CC(=O)N(CC(C)O)CCNC(C2CC(O)(CC#C)C2)=O)c(C)csc1=O 48408,c1(C(N2CC(C)C(CCNC(c3cccc(F)c3)=O)C2)=O)cncc([N+](=O)[O-])c1 48409,C1(NC(c2cc(SC)oc2)=O)CC(NC(=O)C2=CCCOC2)C12CCOCC2 48410,N1(C(=O)OC)CC2CCC1C(C(=O)NCCCCNC(C1(CSC)CCC1)=O)C2 48411,C1(NC(CC(C)OC)=O)CCN(C(=O)C(C)Sc2ccccc2)C12CC2 48412,C1(NC(c2n(CC)nnn2)c2cscc2C)(CSC)CCOCC1 48413,C(=O)(C(Cc1ccoc1)NC(=O)C(F)=CC1CC1)N(CC(C)OC)C 48414,c1(CC)nnc(N2CC(O)(C(C)NC(C3(C)CC3)=O)C2)c(C#N)c1CC 48415,C1(CNC(CC=C)=O)CC2CCC(C1)N2C(=O)CS(=O)(=O)NC1CCC(C)CC1 48416,CC1(CNC(=O)Cn2ccc([N+](=O)[O-])n2)CN(C(c2cccnn2)=O)CCO1 48417,C1(CNC(CCc2cccc(OC)c2)=O)CN(C(=O)Cc2ccsc2)CCCO1 48418,c1(C(=O)NCC(CC2CN(C(CCCCC)=O)C2)(C)C)ccc2oncc2c1 48419,c1(C(=O)NC2C(NC(C3(COC)CCCCO3)=O)CC2)cc(C)ccc1C 48420,N1(C(c2nnn(CC)c2C)=O)CCC(NC(C2(Cl)CC2(C)C)=O)CC(O)C1 48421,C1(NC(c2n(CC(C)C)ncc2)=O)CN(C(c2cc(C(=O)OC)cs2)=O)CC1C 48422,N1(C(CCC2CC(NC(CC3(C)CCC3)=O)C2)=O)CC2CCC2(C)C1 48423,C1(C(=O)NC2C(C)N(C(C3COC(C)(C)CO3)=O)CCC2)CCC(C2CC2)CC1 48424,S(=O)(=O)(c1ccc(NCC2CCOC2)c(C#N)c1)N1C(C)CN(C)CCC1 48425,CC1CCC(C(N2CCC(N(CC(C)C)C(=O)C=Cc3cn[nH]c3)CC2)=O)CC1 48426,C1(NC(Cn2cc(CNC(C3CC(C)OC3)=O)nn2)=O)CC(C)(C)C12CCC2 48427,C1(C(N2CC(CNC(Cc3cn(C)nc3)=O)OCC2)=O)CC2C=CC1C21CC1 48428,c1(OC)cc(C(=O)NC2C3CN(C(=O)C=CSC)CC23)cc2nc(O)[nH]c12 48429,c1(C(C(=O)NCCC2CC(NC(C(C)=C(CC)C)=O)C2)C)ccncc1C 48430,c1(C(N(CC(CC)NC(=O)CC#N)C)=O)cc(C)c(F)cc1Br 48431,Nc1ccc(C(=O)NC2CCCN(C(=O)Cc3cnccc3Cl)CC2)nc1Cl 48432,C=Cc1ccc(C(=O)NC(Cn2cncn2)C(=O)N(CC(C)(CC)OC)C)cc1 48433,N1(C(Cc2cccc(COC)c2)=O)CCN(C(=O)CCCCSC)C2COCC12 48434,N1(C(=O)OC(C)(C)C)CCC(NC(N2CC(C(F)(F)F)CC(CO)C2)=O)C(O)C1 48435,CC1CN(C(c2ncn3c2CCC3)=O)CCCN1C(c1cccc(N)c1O)=O 48436,N1(C(C2OCCN(CC)C2)=O)CCN(C(c2scc(C)c2C)=O)CCC1C 48437,C(=O)(C1=C(Cl)CCCC1)NCC1N(C(CCC2(OC)CCCCC2)=O)CCC1 48438,CCCC(C)CC(=O)N1CCCCC(NC(c2ccnc(-c3ncc[nH]3)c2)=O)C1 48439,N1(C(c2ccc(CCCC#N)cc2)C(=O)NCC(=C)C)CCC=C(C(=O)OC)C1 48440,c1(N2CCCC(C(C)NC(C(Br)=C(C)C)=O)C2)nc(N(C)C)cc(C(F)(F)F)n1 48441,c1(CC(=O)NC(c2ccccc2)C(=O)NCc2nc(=N)[nH][nH]2)cccnc1F 48442,N1(C(c2cc(C)ccc2F)C(=O)NC(CC)C)CCC2(CCCCO2)C1 48443,Cn1nnc2c(C(N3CCC(NC(C4CCC(F)CC4)=O)C3)=O)ccnc12 48444,c1(C(C(N2CC=CC(OCC)C2)=O)NC(CCN(C)CC)=O)c(C)cccc1Br 48445,N1(C(C(OCC)OCC)=O)CCC(F)(CC(=O)NCC(C)(C)CC2CC2)CC1 48446,Cn1nc(Br)cc1NC(C1CCCN1C(=O)COc1ccccc1)=O 48447,C(N=c1[nH]c(=NC(C)C(C)CC)c2c(ncn2C)[nH]1)c1n(CCC)cnc1 48448,c1(C(=O)NCCC(C)NC(C2C3CCCCCC23)=O)c(F)ccc(F)c1Cl 48449,Cc1ccc(CCCC(=O)NC(C)(CNC(C2CCCCC2O)=O)C2CC2)cc1 48450,C1(C)(C(N2CCC(NC(CC(C)(C)OC)=O)(CO)C2)=O)CCC(F)(F)CC1 48451,c1(C(=O)NC2CC(CNC(CCSCCC)=O)C2)cc(C)nc2c1nc(C)n2C 48452,c1(C(=O)NCCCC2(NC(CCn3ccc(C)n3)=O)CC2)nccc(F)c1Cl 48453,C1(CSC)(CNC(N(CCNC(=O)OC(C)(C)C)C)=O)CCCCC1 48454,C1(C(N2C(CCCNC(CCC=C)=O)CCC2)=O)CCOC(C)(C)C1 48455,Cc1cc(C(=O)NC2CCC2C(=O)OC(C)(C)C)ccc1OC(F)(F)F 48456,C1(COC)(NC(=O)C(C2(O)CCCC2)F)CCN(C(c2cc[nH]c(=N)c2)=O)CC1 48457,C1(NC(CCCNS(C)(=O)=O)=O)CCC2CCN(C(c3c[nH]cc(F)c3=O)=O)C12 48458,c1(CNC(C2CCSCC2)(c2nnnn2-c2ccccc2)C)cccc(CO)c1 48459,N1(C(C2(C)CCC2)=O)CC2CCN(C(=O)CCCn3cccn3)CCC2C1 48460,CC1(NC(c2nccnc2Cl)=O)CCCN(C(c2ccc(=O)oc2)=O)C1 48461,C12(C(N3C(CCNC(c4cnc(COC)s4)=O)COCC3)=O)CCCC1OCC2 48462,C1(C(C)(C)C)CCCN(C(=O)C(CO)NC(C2CC(F)(CF)C2)=O)C1 48463,N1(C(C=CCC)=O)CC(CNC(c2cccs2)=O)CC12CCOCC2 48464,c1(CC(=O)NC(C)C(CO)NC(=O)Cn2nnc(=O)[nH]2)coc2ccc(F)cc12 48465,c1(C(=O)NCC2(O)CCCN(C(c3ncc[nH]3)=O)C2)ccc2c(c1)CCCO2 48466,N1CC(OC(c2c(C(C3CCCCC3)=O)cccn2)c2ccccc2)C(F)C1 48467,CCCCCC(C)(C)C(=O)N1CC(C)(NC(c2c[nH]c3cccc(F)c23)=O)C1 48468,CC1CN(C(=O)CC2CCC(NC(C3CCCCC3)=O)C2)CCS1(=O)=O 48469,c1(OC)ccccc1OCC(=O)N(C1CN(C(C2(C)COC(=O)N2)=O)C1)C 48470,C(=O)(CCCCCCS(N)(=O)=O)NC1C(NC(=O)C2=COCCC2)C1.CN1C(=O)C1 48471,N1(C(C2(NC(=O)COC3CC=CC3)C(C)(C)C2)=O)CCc2nc[nH]c2C1 48472,C(c1ccc(C)c(C)c1)=CC(=O)NC1C2(CC(NC(C(CC3CC3)OC)=O)C2)C1 48473,Cc1cc(CNC(=O)CNC(c2cn[nH]c2)=O)sn1 48474,Cc1cccn2c(C(N3CCC4C(NC(=O)C(C#N)C(C)(C)C)C34)=O)cnc12 48475,Cn1ncc2c1CCCC2N=c1[nH]c(=NCc2ccccc2Br)[nH]c2cc[nH]c12 48476,C1(CCO)CCN(C(=O)NC2(CNC(=O)OC(C)(C)C)CCCCC2)CC1(C)C 48477,c1(N2CCN(CC)CC2)nc2cccnc2c(=NCC2CCCC(F)(F)CC2)[nH]1 48478,c1(C(=O)Nc2cccc(NC(CC3C(CC)C3)=O)c2)c(Br)c(C)nn1C 48479,C1(N(C)C(C2CC2(F)Cl)=O)CCC2CN(C(=O)OC(C)(C)C)CCN12 48480,C1(F)(C(=O)NC(C)CN(C(=O)C2=NNC(=O)CC2)C)CS(=O)(=O)CC12COC2 48481,C(=O)(C#CC1CCOC1)N1CC(C)N(C(c2ncnc3[nH]cnc23)=O)CC1 48482,Cc1cc(F)sc1C(=O)NC(C1CCCCC1)CNC(=O)CC1CN(C)C1 48483,C1(NC(=O)COC(F)F)CN(C(=O)C(O)CC2CCOCC2)Cc2ccnn2C1 48484,c1(OC)ccc2c(c1)N(C(c1ccc(Br)cc1Cl)C(=O)NCC(F)F)CCC2C 48485,c1(CN(C(=O)C(=O)NC(C)C(C)(C)C)CCC)ccc(-n2cccn2)cc1 48486,N1(CC(N2CC(CNC(C(=O)N(C)C)=O)OCCC2)=O)CCCC2(CC2)S1(=O)=O 48487,CCCCCCC(=O)N(CCCN(C)C(c1sccc1COC)=O)C 48488,C1(C(N2CCCC2C(C)C)C(=O)NC)C2CN(Cc3cnn(C)c3C)CC12 48489,Cc1cc(C(=O)NCCN(C(=O)CCCc2ccc(F)cc2)C)c(O)c(C)n1 48490,c1(OC)cccc(C)c1NC(=O)C(N1CC2CC1(CNC(=O)CSC(F)F)C2)=O 48491,N1(C(CC(CC)NC(c2cscc2C)=O)=O)CCCC2(CC2)C1 48492,C1(NC(C(CC)SC)=O)CCN(C(=O)Cn2cnnc2)C12CCC2 48493,[nH]1ccccc1=O.C1(N)CC(c2ccccc2)(C(=O)NOC(c2nn[nH]n2)C)C1 48494,C(=O)(C1CCCc2cccnc21)N(C(CNC(c1cn(CC=C)nn1)=O)C)C 48495,CCC(COCC)(CC)C(=O)N1CC(C2CC2C(=O)NOCCN(C)C)C1 48496,c1(C(=O)NC(C2CCCO2)C)ccnc(CNC(C2(C(N)=O)CC2)=O)c1 48497,c1(OC)cc(C(N2CCCCC(CNC(=O)CCC(C)(F)F)C2)=O)cc(C)n1 48498,c1(C(=O)NC2CC(CNC(CCn3ncc(C)c3)=O)C2)ccc2cccnc2c1 48499,CC1CN(C(c2nnn(C)c2C(F)F)=O)CCC1NC(=O)CC1CSCCS1 48500,C#CC1(O)CCN(C(=O)C(CN=[N+]=[N-])NC(c2cccc(O)c2F)=O)C1 48501,C1(CCC=C)CCCN(C(C23CC2CCN3C(=O)C(=O)NOC)=O)C1 48502,CC1CN(C(c2cncn(C)c2=O)=O)CCC1N(C)C(c1ccc(CO)cn1)=O 48503,CC(C(C(=O)O)C1CCCCC1)NC(=O)CCNC(=O)OC(C)(C)C 48504,C=CCC(CC)C(=O)N1CC2(CC(CC(N3CCC(c4ccon4)C3)=O)C2)C1 48505,c1(NC(C2CC(C)CN2C(=O)Cc2ccc(Cl)s2)=O)ncnc2c1c(Br)cn2C 48506,C12(C(N(CC(=O)NC(c3cnccn3)C)CC3CC3)=O)CCCC1C2(F)F 48507,c1(C2C(C(=O)NCCCOCCNC(C(CC#C)O)=O)C2)cccc([N+](=O)[O-])c1 48508,CC1CCCC(OCC(=O)NCCC(C)(C)NC(=O)Cc2cnc(C3CC3)[nH]2)C1 48509,c1(C(N(CCCC(=O)NC2CC2)C)=O)ccc(OCCNC23CCC(C2)C3)cc1 48510,c1(C(=O)OCC)cn(C)[nH]c1=NC(=O)C(c1ccccc1)Nc1ccccc1 48511,c1(C(N2CC(NC(C=CCN(CC)CC)=O)C(C)C2)=O)c(C(F)F)nn(C)c1C 48512,N1(C(C(C2CC(F)(F)C2)OC)=O)CC(NC(=O)CCN2CCCC2)C(C)C1 48513,c1(C(N(CCNC(C2C(CCOC)C2)=O)C)=O)cnc(C(F)(F)F)c(F)c1 48514,C(=O)(C1=CCN(C(C2CCN(C)C2=O)=O)CC1)N(C(C)C1CC1)C1CC1 48515,C(CCCCC(=O)NCC1C(C)CCN1C(=O)CC1(C)CC1(Cl)Cl)OCC 48516,C(=O)(CC(CC)SC)NCCOCC(=O)N(CCC)CCN(C)C 48517,C1(CNC(C(CC)OC)=O)(NC(C23CC(C(=O)NC)(C2)C3)=O)CC(F)(F)C1 48518,CCC(CCOC)C(=O)N1CC(CNC(=O)C(C)(C)N(C)C)C2(CC2)C1 48519,N1(c2cc(C(=O)OC)nc(Cl)n2)CC2(C1)SCCC2NC(=O)Cc1n[nH]c(C)n1 48520,c1(C(=O)OC)ccc(C(C)=O)c(NC(C2(COC3(C)CCC3)CC2)=O)c1 48521,C1(C)(CC)COCCC1NCCCS(Cc1cccc(OC(C)=O)c1)(=O)=O 48522,N1(C(C2C(C)=CCS2)=O)CC2CCC(CNC(=O)CC(C)(C)C)C2C1 48523,c1(-c2ccc(OC)c(F)c2)cccc2c1CCN(c1cccc(Cl)c1[N+](=O)[O-])C2 48524,c1(C(=O)NCC2(C)CC(NC(=O)CNC(=O)NC3CC3)C2)ccc2nccn2c1 48525,Cc1cc(=NC(=O)CCNC(c2cc3ccccc3o2)=O)[nH]n1CCO 48526,C1(C(=O)NCC(C(C)C)CO)C2CC3C(C2NC(c2cncn2C)=O)C13 48527,c1(C(=O)NC2CN(C(c3cc(C)ns3)=O)CC(C)(C)C2)cnc2ncnn2c1C 48528,c1(CC(=O)NC2C(C)CN(C(=O)CCCCN(C)C)C2)ncn2c1CCC2 48529,CCC(CC(=O)NCC1(N(C)C)CCCC1)N(C)C(C1CC(OC)C1)=O 48530,C1(SC)CC(n2ccnc2-c2ccc(F)cc2C)CN(CC2CC2)C1 48531,O=C(CCCC(F)F)NCC1CCN1C(c1ccc(CO)nc1)=O 48532,C1(=CCNC(c2ccc(SC(F)(F)F)cc2)=O)CCN(C(=O)C(O)CF)CC1 48533,C1(C(N2C(C)CCN(C(C3CCC(=O)N3)=O)CC2)=O)CC(F)(F)CCC1(C)C 48534,N1(CCc2nn[nH]n2)CCN(C(c2ccccc2)C2CC2c2ccco2)CC1.SC 48535,C1(C(=O)NC(c2ccccn2)(C)C)CCCCC1NC(C1CNC(=O)C1)=O 48536,c1(CC)ccnc2nc(=NC(=O)NCC(=O)OC(C)C(=O)OCC3CC3)[nH]n12 48537,N12CCC3(CC1)CC(C)N2C3.c1(CCC)ccccc1S(C)(=O)=O.C 48538,C(=O)(C(C)CC(C)CC(C)C)NC1CN(C(C(C(CC)(C)C)O)=O)CC(C)C1 48539,CCC(CC(=O)NC1CC(C(=O)NCc2cc[nH]n2)C(O)C1)C(C)C 48540,CC(C(=O)OC(C)(C)C)C(=O)N1CC=CC1CNC(=O)C=Cc1nccs1 48541,C1(C(=O)NC2(CC)CN(C(=O)C(C)C)C2)C2CC2C2CC12 48542,Cc1noc(C)c1CC(C)C(=O)NCC1CCN(C(=O)CCc2cccnc2)C1 48543,C(C1CSc2ccccc21)NC(=O)Nc1cn(CCOC2CCCCC2)nn1 48544,c1(CNC23CCC(NC(C=CC)=O)(CC2)C3)cc(F)cc([N+](=O)[O-])c1 48545,C(C)(CN=c1ccnc(NCCCS(C)=O)[nH]1)c1ccc(OC)cc1 48546,C=CCC(CNC(c1cc(Cl)no1)=O)C(=O)NCc1cc(C)cc(O)c1 48547,c1(CN2CCCC(NC(CCC(C)C)=O)CC2)cc(Cl)c(O)cc1F 48548,Cc1cc(F)ccc1CC(=O)NCCC(C)N(C(=O)Cc1cccc(F)c1O)C 48549,c1(C(=O)NC2CC(N(C(C3(OC)CCOCC3)=O)C)C2)cc(F)c(Cl)cc1F 48550,Cc1cc(C(=O)O)sc1C(=O)NC(C1(CC(=O)O)CCOC1)c1ccccc1 48551,Cc1ccnc2c(C(N3CCC(CNC(=O)C(C)N4CCC4)C(C)C3)=O)cnn12 48552,C1(CC(=O)NCC(C)(C)CC2CN(C(c3ccncn3)=O)C2)CCC=CCC1 48553,Cc1ccc(-c2ccc(C(N3CCCCC3c3nncs3)=O)cc2)cc1Br 48554,C1(NC(c2ccc(C#C)cc2)=O)CN(C(c2ccc[nH]2)=O)CC12CCC2 48555,N1(C(=O)Nc2ccc(OCCCN(C)C)cc2)CCC(O)C2(CCC2)C1 48556,Cc1ccc(C)c(CNC(=O)N(c2ncc[nH]2)Cc2ccccc2)n1 48557,N(C(=NCC1CNCc2ccccc21)N1CCC(Nc2ccccn2)C1)C(C)C 48558,c12cn(nn1)C1(CC1)C(=O)NC2C.c1(C(=O)NCCCC(F)F)ccccc1 48559,N1(C(c2sncc2Br)C(=O)NCCCCCC)CCCC(NC(=O)OC)C1 48560,CC1CCC(C)N1CC(=O)NC1CCC(CC(=O)NC2(C)CCOCC2)C1 48561,N1(C(CC=CC)=O)CCC(C2CCCN(C(=O)CS(=O)(=O)CC)C2)C1 48562,CC(C)CCCCCC(=O)NC1CCN(C(c2cnn(C3CC3)c2)=O)C1 48563,c1(CCC(N2C(C)CC(NC(c3c(OC)c[nH]n3)=O)C2)=O)csc2nc(C)cn12 48564,CCC(CNC(=O)C(C)(F)F)(CC)NC(C1COCC1C(=O)OC)=O 48565,N1(C(c2cn(CC)nc2C)=O)CCN(C(c2ccc(N)c(C)c2F)=O)C(C)C1C 48566,CC#CC1CCN(C(C2(CCNC(=O)C(F)C(CC)CC)CC2)=O)CC1 48567,C(C(O)C(=O)NC(C(=O)N(C)Cc1ncc(C)o1)C1CCCO1)N(C)C 48568,c1(OC)cnc(Cl)cc1C(N1CCC(NC(=O)C(C)(Cl)Cl)C(C)C1)=O 48569,C1(C(C)(C)C)(CNC(C(C)OCC)=O)CCN(C(C2CCC(N(C)C)CC2)=O)C1 48570,C(=O)(C1=NOC2(CCC2)C1)N1CC(C)N(C(=O)CC(O)CCNC(N)=O)CCC1 48571,c1(C(=O)NCC(C)CN(C)C(C2CC(O)CN2C)=O)n[nH]c2c1COCC2 48572,C1(CNC(CC2CCN(C)C2=O)=O)CN(C(c2cnc(S)[nH]2)=O)CC12CC2 48573,C(=O)(C1(C)CCn2ccnc21)NC(CCCCNC(C(C(C)C)F)=O)C 48574,c1(C(C(C#N)C(=O)NCCC2CCCCC2)=O)ccnc2c1CC(=O)N2 48575,N1(C(CCCCCCC)C(=O)NC(C)(C)CC)Cc2ccccc2CC1(C)C 48576,CC1(C)CC(CNCCc2c(F)cccc2F)CCO1 48577,Cc1ccc(C(N2CCCC(NC(=O)C(C3CC3)N(C)C)C2CO)=O)c(Cl)c1 48578,C(CCCN=c1[nH]nc(C2CCCC2)s1)NC(c1cnn(C2CC2CO)c1)=O 48579,N1(Cc2c(C)sc(C(=O)O)c2)CC(F)(C(=O)O)C2(COC2)C1 48580,C1(NC(CCC2(C)N(C(c3c(C)csn3)=O)CCC2)=O)CNC(=O)C12CC2 48581,CCC(CC(=O)NCCCCNC(c1cccc(O)c1F)=O)C(F)F 48582,c1(C(CN2CCCN(C(C(N)=O)=O)CC2)=O)cccc2c3c([nH]c12)CCCCC3 48583,S(=O)(=O)(c1ccc(Cl)nc1)N(C(C)CNC(C1COC2(CCNCC2)C1)=O)C 48584,Cc1n[nH]cc1CC(N1CC(CN(C(=O)COC2CCCOC2)C2CC2)C1)=O 48585,n1(CC)ncc(C(N2CC(NC(=O)C(C)c3ccsc3)C2)=O)c1C(F)(F)F 48586,CC1=C(C)CC(C)(C(=O)NC2C=CCN(C(c3ncsc3S(N)(=O)=O)=O)C2)CC1 48587,C=CCCCCC(=O)NCC1CCC(Cn2cc(C3CC3COC)nn2)CC1 48588,CC(CCNC(=O)CCc1n[nH]c(=N)s1)CCNC(=O)CNS(C)(=O)=O 48589,N1(C(COCc2cc(C)no2)=O)CCC(C)C(CNC(=O)CCCF)C1 48590,C1(C(N2CC(C3CN(C(CNC(C)=O)=O)C3)C2)=O)Cc2cccc(Cl)c2C(=O)O1 48591,C(=O)(CCCCC(N)=O)N1CCC(NC(C(C)(C2CC2)NC(C)=O)=O)C1 48592,Cc1ccc(C)n1CC(N1CCOC(C(C)NC(=O)C(C)(C)c2cnc[nH]2)C1)=O 48593,Cc1cccc(C)c1OCCC(=O)NC1CCN(C(C2CNC(=O)C2)=O)C1C 48594,C1(CC(=O)N(CCNC(c2sccc2C(F)F)=O)CC)SC2=NCCN2C1=O 48595,c1(CC(N2C3(CN(C(c4c(C)nns4)=O)C3)CC2)=O)n[nH]c2ccccc12 48596,c1(C(C)N(C)C(C2CCN(c3ccccc3Br)C2=O)=O)ccc(Cl)cc1 48597,C(CCCC(=O)N1CCC1C1CCCC1)NC(Cn1c(C)ccn1)=O 48598,c1(C(=O)NC2C(CNC(C=C(COC)C)=O)CCC2)ccc2cnoc2c1 48599,C1(NC(=O)CC2CCC(O)C2)CC2(CCN(c3nnc(C4CC4)s3)CC2)C1 48600,CC1COCCC1N(C(=O)C(C1CCC1)NC(=O)CCC1CCC(=O)C1)C 48601,N1(C(CO)=O)CCCCC(C2CN(C(COCC(C)(C)OCC)=O)C2)C1.C(C1CC1)=CC 48602,C(c1ccc2occc2c1)=CC(=O)NC1(CCCSCc2ccccc2)CC1 48603,N1(C(C2(C(C)=O)CC2)=O)CCC(C2CCN(C(c3ccc(Cl)s3)=O)CC2)C1 48604,c1(NC(C(COC(C)C)NC(C(CC)OC)=O)=O)ccc(OC(C)C)c(C)c1 48605,c1(C(=O)NC(C2CN(C(C3CCS(=O)(=O)C3)=O)C2)C)cnc(-c2ccoc2)[nH]c1=N 48606,N1(C(CC(C)(F)F)=O)CC2COCCC2(NC(c2ccnc3[nH]cnc23)=O)C1 48607,c1(CCC(=O)NC2CC(NC(=O)CCC3CCC3)C(O)C2)ccc(Cl)cc1 48608,C1(NC(CC(CN(C)C)(C)C)=O)C2CC(O)C1N(C(C1CSCCS1)=O)C2 48609,n1(CC(=O)N(C(C2CCCCC2)C2CCCC2)C)ncn(C)c1=O 48610,N1(C(C=C(C)C(C)(C)C)=O)CCC(C2CC2)(CNC(=O)C#CC(C)(C)C)C1 48611,C(=O)(C(C(F)(F)F)=Cc1ccccc1)N1C(CNC(c2c(C)csc2)=O)CCC1 48612,n1(CC(=C)C)nnnc1C(c1nc(C2CC2)cs1)NC(C1CCC1)C1CC1 48613,C1(C2CCC2)(C(=O)NCCCC2(NC(=O)CC3CCCC(=O)N3)CC2)CC1(F)F 48614,n1(CCCC)nc(C)c(C=CC(=O)N(CC(C)C(=O)OC)CC(C)C#N)c1Cl 48615,C1(CNC(COCCOCC)=O)C(C)CCCN1C(c1cccc2c1OCC2)=O 48616,Cc1cnoc1C(=O)NCC1(NC(C2CC(CC3CC3)C2)=O)CCC1 48617,N1(C(C2CCN(CC(C)C)CC2)=O)CCC(NC(=O)CCC(C)(C)C)C(C)(C)C1 48618,C1(NC(CN2C(C)CCC2)=O)CC(O)CCN1Cc1cc(O)cc(F)c1 48619,N1(CC(=O)NCC2CCCC2C(=O)NC2CC3CCC2O3)C(=O)CCCC1=O 48620,C(CC(C(=O)NOCCC(C)O)NC(=O)C1=C(Cl)CCC1)OCC 48621,N1(C(CCC=CC)=O)CCC(NC(=O)CSCC(F)F)CC(O)C1 48622,Cc1cc(C(N2CC(CC(C)NC(c3cccc(=S)n3O)=O)C2)=O)c(F)cc1F 48623,c1(OC)cccc2c(C(=O)N(CC(C)NC(=O)Cc3cncc(O)c3)C)csc12 48624,S(=O)(=O)(c1ccc2c(c1)CC(C(N1CCOCC1C(=O)OC)=O)C2)NC 48625,c1(C(=O)NC(C(N2CC3(CCC(=O)N3)C2)=O)C2(C)CC2)cccc2cncn12 48626,c1(NC)cc(Cl)ccc1C(=O)NCC1COCC1NC(=O)C(C)(C(C)C)OC 48627,C1(NS(CCC)(=O)=O)CC2CN(C(c3c(I)ccnc3F)=O)CC2C1 48628,CN1CC(NC(C2C3CC3CN2C(=O)CCc2nncn2C)=O)CC1=O 48629,C1(CNC(CCCCC=C)=O)CCN(C(C2(OC)CCOC2)=O)CCC1(F)F 48630,C(=O)(CCCC(=O)N1CC(CNC(c2cnc(F)cc2C)=O)CC1C)NC 48631,C1(N(C)CC2CCCN2C(C2CCCC2)=O)CCCC(c2cncn2C)C1 48632,N1(C(C(c2cc(C)oc2C)C)=O)CC2CCCC2(CNC(c2ccsc2)=O)C1 48633,c1(C(N2CC(CCNC(=O)C(O)CCSC)(OC)C2)=O)c(C)c(C)nn(C)c1=O 48634,c1(OC)cc(CNC(C23CC(CCO2)C3)C(=O)O)cc(OC)c1Br 48635,C(CC(C(=O)N1CC(OCCO)C1)NC(C1CCOCC1)=O)SC 48636,c1(C(=O)NCCCN(C(C(CC)N(C)C)=O)C2CC2)cc2nc(=O)ccn2[nH]1 48637,C1(N(C(COC)=O)C)CCCC(N(C)C(c2cn(C3CC3)cn2)=O)C1 48638,C1(C)(CNC(C(F)=CCC)=O)CCN(C(C23CCCCC2CCC3)=O)CC1 48639,CC1CC(NC(C2COC(=O)N2)=O)CN1C(C1CCN(C2CC2)CC1)=O 48640,N1(C(CN(C(C)(C)C)C2CC2)=O)CCC(C(C)(C)NC(=O)CC2C=CCCC2)C1 48641,c1(NCC)ncc(C(N2CC(NC(=O)CC3=CCCC3)CC(C)C2)=O)cc1Cl 48642,N1(C(C(C=C)O)=O)CCCN(C(c2nc(OC)c(C)s2)=O)CC1C(C)C 48643,C1(C#N)(C(=O)NC2CCC(NC(c3cccc(SC)c3)=O)CC2)C(C#N)C1(C)C 48644,C1(C(N2C(CC)C(C(=O)NCCc3cnccc3C)CC2)=O)CCOC(C)(C)C1 48645,CCC(C)CCC(=O)NC(C)C(C)(C)C(=O)NCCN(CC(F)F)C 48646,C1(N(C(C(C)=C2CCC2)=O)C)CCN(C(=O)Cn2ncccc2=O)CC1C 48647,C(CCC)(C(=O)NC1COCC1CNC(C1CSCCS1)=O)=CCC 48648,N1(C(=O)CNS(=O)(=O)C2CC2)CCCC12CCN(C(C1CC3CCC1O3)=O)C2 48649,C1(C)(C(=O)NCC(C2CCC2)NC(CCc2cn(C)nc2)=O)CCCCO1 48650,c1(C(N2CCNC(=O)C2c2cccs2)=O)cc2c(s1)CCC(c1ccccc1)C2 48651,CC(CN(C)C)CC(=O)N1CCC(CC(=O)NC2CC(CN(C)C)C2)CC1 48652,Cc1cc(Br)ccc1CC(=O)NCC#CCNC(c1cc(C2CC2)nn1C)=O 48653,C1(C(=O)NCC2CCCN(C(CN3CCC(OC)C3)=O)C2)CCC2(CCCC2)C1 48654,CCC(CCCC(=O)N(C)CC1CCCC1)NC(=O)C(C)N(C)C 48655,c1(CC)cc(C)c(C(=O)NCC(=O)NCCCN(C(=O)C2=CCCC2)C)o1 48656,N1(C(c2ccc(C#N)o2)=O)CCC2(NC(c3cc(C4CC4)cc(F)c3)=O)CC2C1 48657,C(=O)(C(O)CC(C)(C)C)NC1CCN(C(Cc2c(C)sc(Br)n2)=O)C1C 48658,C1(O)(CNC(CC2(CS(C)(=O)=O)CC2)=O)CCCN(C(c2nnc(O)nc2O)=O)C1 48659,C1(CC(C)NC(=O)CC(C)(F)F)CCN(C(C2CCCCN2C)=O)CC1 48660,c1(C(C)C(=O)Nc2cc(Cl)c(Br)cc2O)cc2ccccc2nc1O 48661,n1(C(C)C)cccc(C(=O)NCc2cn(CCNC(C3CC(F)C3)=O)nn2)c1=O 48662,c1(C(=O)NC2CCN(C(C(C=C)O)=O)CC2)ccc(Cl)c(OC)c1 48663,CCC(C)C(O)C(C)C(=O)N1CCCC(CC(=O)NCC2(O)CCCCC2)CC1 48664,c1(C(=O)NC2CCN(C(C3C(OC)C3)=O)C2C2CC2)ccc(C)c(C)n1 48665,N1(C(CSC)=O)CCC(CNC(=O)COc2c(Cl)cccc2Cl)(COC)CC1 48666,C1(C(N(C(c2ccccc2)CNC(=O)CC(C)(F)F)C)=O)CCCCC1(C)C 48667,C1(NC(CCCSC)=O)CN(C(=O)C(C)(C)C2CCCC2)CC1C 48668,N1(C(c2c(OC)nc(C)cc2)=O)CCCCCC(NC(=O)Cc2cnc[nH]2)C1 48669,N1(C(c2c(OC)ccnc2)=O)CC(NC(=O)Cc2cc(C)[nH]n2)CC(F)(F)C1 48670,C(=O)(C1CCc2cccc(F)c21)N1C(CCNC(=O)Cc2cc[nH]n2)CCCC1 48671,N1(C(c2c(C)ccs2)=O)C2CCCC1CC(NC(c1c(C)nc3ncccn13)=O)C2 48672,c1(C(=O)NCCOCCN(C(C(COC)(C)OC)=O)C)c(C)cccc1[N+](=O)[O-] 48673,CCCC(C(=O)OC)C(=O)N(C(C)CNC(c1cccn2cnnc12)=O)C 48674,N1(C(C2CC(=C)C2)=O)CCC2(C1)CN(C(=O)C(C1CCC1)OC)CCO2 48675,c1(C(=O)NC2C(NC(Cc3cn(C)nc3)=O)CCC2)ccc2cnnc(O)c2c1 48676,C(=O)(CCC(C)(C)C(=O)NC1CC1NC(C1CCCc2ccccc2C1)=O)OC 48677,N1(C(C2(c3cc(C)n(C)n3)CC2)=O)CC2(C1)CN(C(=O)COCCF)CCO2 48678,C1(CNC(c2ccnc(-n3ccnc3)c2)=O)CN(C(C2CCOC2=O)=O)CCO1 48679,c1(CC(N2CCC(n3cc(C4CCCC4O)nn3)C2)=O)cc(C(=O)O)co1 48680,c1(C(=O)NC2C(CNC(CCNS(CC)(=O)=O)=O)C2)csc(-c2ccco2)n1 48681,N1(C(CCC(C)C)=O)CC2CCC(NC(c3cccc(CN=[N+]=[N-])c3)=O)C2C1 48682,CCC(C)(C)CCN=c1[nH]c(N2CC(CCOC)OC(C)C2)nc2cccnc12 48683,CC(C)C(=O)C(=O)NC(c1ccnn1C)C(N1CCC(OCCO)C1)=O 48684,N(C(=NCc1ccccc1)N1CCOC(C2CC2)C1)CC(CC)(C)C 48685,C1(NC(Cc2cc(C)ns2)=O)CN(C(=O)C(O)CC(=O)OC(C)(C)C)CCC1F 48686,c1(NC(N(c2cc(OC)ncn2)C2(CO)CNC2)=O)cc(C)cc(C)c1 48687,Cc1cc(C=CC(=O)NC2CC(NC(c3csnn3)=O)C23CCC3)c[nH]c1=N 48688,c1(SCc2nc(C(C)(C)C)sc2)nnc(N2CCC3CC23)o1 48689,c1(C(=O)NC(CC)CN(C)C(c2cnn(C)c2C)=O)ccc(C)c(Cl)c1F 48690,Cc1scc(C(=O)NCC2OCCC2C(=O)NCCc2ccccc2F)c1C 48691,C1(C(N2CC(OC)C2)=O)CC(C)CN1C(=O)CCc1nncs1 48692,CCC(CC(=O)NCC(C1CCN(C(c2cc(C)c(C)o2)=O)CC1)(C)C)C(C)C 48693,CC(CCC=O)NC(=O)OC(C)(C)C.C1(C(=O)OC(C)(C)C)(CN)CC12CCC2 48694,CC1CCCC1(C)C(N1CC(O)(CNC(=O)CC(=O)Nc2ccccc2O)C1)=O 48695,C1(C(=O)NCC(CC)NC(C2(N(C)C)CC2)=O)CCc2cc(OC)ccc2C1 48696,C1(NC(CCC(=C)Cl)=O)CC2CC1N(C(c1sc(C(=O)OCC)nc1C)=O)C2 48697,N1(C(c2ncn(C)n2)=O)CCCC1C1CCCN1C(c1n[nH]c2c1CCC2)=O 48698,CC(C)C(C)C(CNC(c1csc(-c2ccsc2)n1)=O)NC(C1OCCO1)=O 48699,N1(C(C(CC(=C)C)C)=O)Cc2ccnn2CC(NC(c2ncc(Cl)cc2F)=O)C1 48700,O=C1CCC(=O)N1CCCCC(=O)NC1CC(C(F)(F)F)C1 48701,c1(CC(=O)NC2(CC=C)CN(C(C3CCCS3(=O)=O)=O)C2)c(C)nc(C)nc1O 48702,C1(C2CC2)(CNC(CC=C)=O)CCN(C(=O)CCCC2CCC2)C1 48703,c1(C(=O)NCCN(C(C(CC)n2cccn2)=O)C(C)C)c[nH]cc(F)c1=O 48704,c1(C(=O)NCCC2N(C(C(N)=O)=O)CC(F)(F)C2)cc(Cl)cc([N+](=O)[O-])c1 48705,N1(CC)CC(C(=O)N2CCC(C)(NC(=O)CS(=O)(=O)CC)C2)c2ccccc21 48706,Cc1nc2c([nH]1)CC(CNC(N1CCC1CC1CC3(CC3)CO1)=O)CC2 48707,C1(=CC(=O)NC2CC(O)CN(C(=O)CCCc3ncco3)C2)CN2CCC1CC2 48708,CC1CN(C(=O)C(C2CCCCCC2)O)CC(C)N(C(c2cc(C#N)c[nH]2)=O)C1 48709,Cc1nc(C(N2CC3CC(C2)N3C(=O)Cc2cnn(C)c2)=O)cc(O)n1 48710,c1(OCC(=O)NC(C2CCOC2)CNC(c2c(C)nc[nH]2)=O)cc(F)cc(Cl)c1 48711,c1(C(=O)NCC2(O)CN(C(CC(CCC)CC)=O)C2)cccc2c1CC(C)(C)C2 48712,C1(OC)CC(CN(C)C(=O)NCC2CC3(C2)CC3F)CC1OC 48713,N1(C(c2n[nH]cc2Br)C(=O)NC(CC)(C)C)CCCCC12CCN(C)C2 48714,C1(NCC)OCCC1C(=O)NCCOCCN(C)C(c1cc(C(C)(C)C)on1)=O 48715,c1(C(=O)NCCCN(C(C2CCCO2)=O)C2CC2)ccc(Cn2cccn2)o1 48716,Cc1oc2cc(C(=O)NCCN(C)C(C3(O)CC3(C)C)=O)[nH]c2c1C 48717,N1(C(CNC(C)=O)=O)CCc2[nH]nc(C(=O)Nc3cc(Cl)c(F)c(Cl)c3)c2C1 48718,C=CC1(C(=O)NCC(N2CCCC2C)C)CCN(C(=O)COCCCF)C1 48719,C(=O)(C1CCCc2nc[nH]c21)N(C1CCCN(C(C(COC)(C)C)=O)C1)CCO 48720,CC(C)CC(CCO)NC(=O)CC1CCC(NC(c2csnc2Cl)=O)C1 48721,c1(C(=O)NCCC(C)N(C(C(CC)n2cccn2)=O)C)cc(C)nc(N(C)C)n1 48722,N1(C(Cc2ccc(OC)cn2)=O)CCN(Cc2ccnn2C)CC1CO 48723,N1(C(C(c2ccc(Cl)s2)C)=O)CCC(N(C)C(C2(C)CC(F)(F)C2)=O)CC1 48724,c1(C2C(C(=O)NCCNC(C3CC(C)(F)C3)=O)C2)c(F)cc(Br)cc1F 48725,N1(C(CC)=O)Cc2ccccc2C1C(=O)Nc1nc2ccccc2nc1OC 48726,C1(NC(C(CC=C)OC)=O)CC2(C1)CC(C(=O)NC1(C)CCCOC1)C2 48727,C1(CN(C)C)CC(O)CN1C(c1ncoc1CNC(c1ncncc1N)=O)=O 48728,CC(F)(F)CC(=O)N1CCC(C)(NC(c2[nH]nnc2C2CC2)=O)C1 48729,C1(NC(C2C(CCOC)C2)=O)CCCCN(C(=O)Cn2nccc2C)C1 48730,C(CN=C(NCc1ccco1)NC(c1ccccc1Cl)C)N(CC)CC 48731,C(CCC(C)(C)C(=O)N1CCC(OC=O)C1)NC(c1c(C)sc(O)n1)=O 48732,C(=O)(CCCC(=O)NC1CC(CNC(c2cccc(NC3CC3)c2)=O)C1)NCC 48733,N1(C(Cc2cn(C)nn2)=O)CCCC2(CCC(NC(=O)C(=O)N=S(C)(C)=O)C2)C1 48734,CC1CC2(CCN(C(=O)CCCCCNC(=O)C(C)(C)C(C)(C)O)C2)CO1 48735,CC(CC(=O)NCc1cc(C(N2CCC(C3(C)N=N3)C2)=O)no1)N1CCCC1=O 48736,Cc1n[nH]c(C)c1SCC(=O)NC1(CNC(=O)C(C)(C)N2CCCC2)CCCCC1 48737,CC1(NCCSc2ccccn2)CC(F)(F)C1 48738,C#CCC(CC(F)F)C(=O)N1C2CCC(C2)C1CC(N1CC=CC1CF)=O 48739,N1(C(c2n(CCC)ncc2)=O)CC2CC1CN2C(c1c(Cl)sc(C)c1C)=O 48740,N1(C(CCOCC#C)=O)CCC=CC1C(N1CC(C(C)C)C1C(C)C)=O 48741,Cc1cc(C)cc(C(N2CC(NC(C3(C)CCCCO3)=O)C(O)C2)=O)c1O 48742,C1(C(=O)NCCC(C)(C)NC(C2CCCC2C(F)F)=O)(OCC)CCOCC1 48743,N1(C(C2(C)COC2)=O)CCCC(CCCCNC(C23CCCC2(C(N)=O)C3)=O)C1 48744,N1(C(C(C)=C(C)C)=O)CC2CCC(CNC(=O)C=Cc3cccc(C#N)c3)C2C1 48745,Nc1cc(C(=O)NC2CC(CNC(c3ccc(F)cn3)=O)C23CCC3)cnc1N 48746,C(=O)(CS(=O)(=O)C1CCCC1)NCC1(C)CCCN1C(C1CCCC12CC2)=O 48747,C=CCCCCC(=O)NCC1CC(O)CN(C(=O)CCCc2ccccc2N)C1 48748,Cc1nc(C)c2c(C)c(C(=O)NCC(C)(C)NC(=O)C(C)C(C)O)sc2n1 48749,C(c1cccc(Cl)c1)=CC(=O)N(C1CCN(C(C2C(C)(COC)C2)=O)C1)C 48750,c1(CC(N2CC(CCCCNC(C(C)NC(C)=O)=O)C2)=O)c[nH]c2ncccc12 48751,c1(CN2CC3(CC(C(N4CC(C(N)=O)OCC4)=O)C3)C2)c(Br)cc(F)c(F)c1F 48752,N1(C(C(C)=C(C)C)=O)CCC2(CCN(C(=O)C(=O)Cc3ccccc3)C2)C1 48753,C#CCCCCC(=O)NCc1cc(C(=O)NCC2(C3CC3)CCCO2)n(C)n1 48754,c1(C(=O)NC2C(C(C)C)CN(C(=O)C3=CCCS3)CC2)n[nH]c2ccccc12 48755,C1(CCC(=O)NC(c2c[nH]nc2OC)C)CCCCN(C(=O)C2=C(Cl)CC2)C1 48756,C=C(Cl)CC(C(=O)N1CC2CC1C2)NC(c1ccncc1NC)=O 48757,c1(CNC(C2CCCN2C2CC2)=O)nc2c(s1)CCN(C(C1CCCS1)=O)C2 48758,c1(CN2CC(C(=O)NC(C(C)C)CO)SCC2)nccc2occc12 48759,C1(C(=O)NCCCC(=O)NC)CCN(C(C2C3(CC3)C23CC3)=O)C(C)C1 48760,CC(C)S(=O)(=O)C(C)C(=O)N1CCC(NC2CN(C(c3cncc(N)n3)=O)C2)CC1 48761,CCC(C)C(O)C(C)C(=O)N1CC(N(C(=O)Cc2cnc(C)s2)C)C1 48762,c1(NC(c2c(OC)ncc(-c3cscn3)c2)=O)cccc2ncsc12 48763,C1(C(=O)NC(C)CCNC(c2conc2C(C)(C)C)=O)CCN(S(N)(=O)=O)CC1 48764,C1(NC(C)=O)CCCCC1N(C(=O)Cc1c(Br)cnn1C)C 48765,C12(NC(C=CS(C)=O)=O)CCCC1N(C(c1cnn3c1CCCC3)=O)CC2 48766,c1(C(N(CC(C)NC(COC(C)C)=O)C)=O)ncccc1N(C)C 48767,CCCCC(F)C(=O)N(C1CCCN(C(=O)C(C)(C)OCC)C1)C 48768,N1(C(C(CCC)(C)C)=O)CC2(NC(=O)CSc3nc(C)cc(C)n3)CCC1CC2 48769,c1(C(N(C(CCC)Cc2ccccc2)C)=O)nccc(C)c1[N+](=O)[O-] 48770,C1(C(=O)NC(CC#C)CO)(CSC)CCCN1C(C1CCC1NC)=O.C 48771,CC1CCC(CNC(c2csc(=N)[nH]2)=O)CN1C(=O)CC1(O)CCCCCC1 48772,C(CCCCC(=O)NCCC1(NC(c2csc(C)c2N)=O)CCC1)OCC 48773,CCC(CNC(=O)C(C1CCOCC1)O)(CC)NC(c1cnn(C)c1C1CC1)=O 48774,C(=O)(CC(C)CC(=O)NCC1CCN(C(c2cncc(OC(C)C)c2)=O)C1)OC 48775,c12cc(no1)C(N(C1CCC(C)C1)C)C(=O)NC2.C(COC)OCC 48776,C1(C(=O)NC(C)CN(C(=O)COCP(C)(C)=O)C)CCCCN1CC(F)F 48777,C(C)(CCC(=O)N1CC2C(NC(C3CC(=O)N(C4CN(C)C4)C3)=O)C2C1)SC 48778,CCC(CC(=O)NC(CN(C)C(c1cccc(C(C)C)n1)=O)CC)OC 48779,C(=O)(C1CCCn2nccc21)NC(c1ccc(F)cc1F)COC.C1(=O)CN1 48780,N(C1CCc2cccc(C)c21)C(N1C(C(=O)OC)CNc2n[nH]cc2C1)=O.C(C)S 48781,c1(OC)c(C)cc(-c2ccc(CC(=O)NCc3c(C)noc3C)cc2F)cc1C 48782,C1(O)(C(C)NC(c2n(CC)ccc2)=O)CCN(c2ncncc2C#N)CC1 48783,c1(C(N(C2CCN(C(c3cc[n+]([O-])cc3)=O)CC2)C)=O)ncc(N)cc1Cl 48784,CCCC(C#N)C(=O)N1CCN(C(=O)Cc2ccncc2Cl)C(COC)C1 48785,c1(NCC(=O)NC(C2CN(C(=O)C(c3ccccc3)=O)C2)C)cnn(C2CC2)c1 48786,N1(C(c2ccc(CC)[nH]2)=O)CCOCC1CNC(=O)C(c1ccc(OC)cc1)O 48787,N1(C(CC(=O)OC)=O)CCC2(CCC(CNC(c3cccnn3)=O)O2)CC1 48788,C1(NC(C(C)CO)=O)CN(C(=O)C(C)(C)c2ccnn2C)CC2CCCC12 48789,c1(C(=O)OCC(c2cnc(C)s2)=O)cncc2nc(O)[nH]c12 48790,c1(CCC)cc(C(N2CCC(NC(C3(NC(C)=O)CCCC3)=O)C2)=O)nn1C 48791,C1(NC(c2ccc(N(CCC)C)cc2)=O)CCN(C(=O)C(=O)NC2CC2)CC1C 48792,CCCC(C)(O)C(=O)NCC1CCC(C(=O)NC2(C)CCCCC2)CC1 48793,N1(C(C(c2ccco2)NC(C2OCC(C)(C)C2)=O)=O)CCC(C2(C)CC2)CC1 48794,C1(C(C)NC(=O)COC(F)F)CN(C(=O)CCCC2CCCO2)CCO1 48795,c1(CC)ccc(OOC(F)(F)F)cc1.C12(NC(=O)C(C)CC3CC3)CN(C1)C2 48796,c1(CC(n2cc(CNC(c3scc(OC)c3)=O)nn2)C)ccc(F)cc1F 48797,C1(O)(CCNC(C2COCCC2(F)F)=O)CCCN(C(=O)CCc2cnoc2)C1 48798,C1(NC(Cc2ccc(C)nc2)=O)CCN(C(=O)CC2OCCCO2)CC1(C)C 48799,c1(CNC)cccc(NC(=O)C(N2CC(CN)C(C)C2)=O)c1 48800,N1(C(c2c[nH]cc(C)c2=O)=O)CC(NC(=O)Cc2nc[nH]n2)C2(CCCC2)C1 48801,C(=O)(C(F)(F)C(C)(C)O)NCC1C(C(=O)NC2CCN(CC)C2)C1 48802,CC(C)C(C(=O)NOCCCF)C(C)NC(C1(O)CCCC1(C)C)=O 48803,C(=O)(C(F)(F)CO)N1CC2(C1)C(=O)N2.N1(CC)CCC1COC 48804,C=CC(C)(CCOC)C(=O)NC1CCC1C(=O)OC.c1(C(=O)N)ncoc1COC 48805,C1(NC(Cc2cccc(OC)c2)=O)CC2CN(C(c3cc(Cl)ccc3Cl)=O)CC12 48806,N1(C(CNC(CC)=O)=O)CC(N(C(=O)C(C)Cc2c(C)n[nH]c2C)C)C(C)(C)C1 48807,c1(CCC)cc(C(N2CC(C(C)(C)O)(CNC(C3(F)CC3C)=O)C2)=O)no1 48808,c1(C(N(CCOCCNC(C(CCC)C#N)=O)C)=O)c(F)ccc(F)c1Cl 48809,C#CCCC(O)C(=O)N1CCCN(C(C2CCC(F)(F)C2)=O)CC1 48810,Cc1cc(C(N2CCC(C)(C)C2CC(=O)NOCC(C)(C)C)=O)nc(O)c1 48811,C1(CNC(=O)CCN2CCCCC2)COCCN1C(=O)COC(F)(F)F 48812,C#CCCCCCCC(=O)NC(C1CC(NC(c2nccc(OC)c2N)=O)C1)C 48813,C1(C(=O)NCCCC(C)NC(=O)CN(C)Cc2ccccc2)(COC)CCOC1 48814,CC(C)CCC(=O)N1C(CNC(c2ccc(N3CCCC3=O)cc2)=O)CC2CC12 48815,N1(C(C2CCSCC2)C(=O)Nc2ccc(F)cc2)CCC(CC2CC2)CC1 48816,C1(C(N2CC3CC3(CO)C2)=O)(NC(=O)OC)CC(OC)C1(C)C 48817,c1(C(N2C(C(N3CC(OCC(=O)NC)C3)=O)CC2)=O)cc(C#N)[nH]c1C 48818,C#Cc1ccc(C(=O)NC2CC(C)(NC(c3cccc(C(C)C)n3)=O)C2)cc1F 48819,N(C(=NCCCCCOc1ccc(Cl)cc1Cl)NCC(F)C(F)(F)F)CC(F)F 48820,C=C=CCCC(=O)NC(C1CCN(C(c2nnn(C(C)C)c2C)=O)C1)C 48821,c1(C(=O)NC(C2CCCN(C(c3csc(C4CC4)n3)=O)C2)C)c(O)cccc1Cl 48822,N1(C(CCC(=C)Cl)=O)CCC(C(=O)NC(C(C)C)C2CCC2)C(C)(C)C1 48823,CCCCCC(O)CC(=O)NC1CCC(NC(c2nc[nH]c3ncnc2-3)=O)C1 48824,C1(CNC(CN(C2CCC2)C)=O)CCC2(CCC2)CN1C(=O)C(O)C(C)(C)C 48825,Cc1cccc2c1C(NC(C1(N(C)C)CCSC1)=O)CC2 48826,c1(-c2nc(C)oc2)ccc(C(N2CC(NC(c3cncn3C)=O)C(O)C2)=O)cc1 48827,c1(C(N2CCC(C(C)CNC(c3ccoc3)=O)CC2)=O)nc(Cl)c(=O)[nH]c1N 48828,C1(CN(C(=O)CSc2cccc(F)c2)C)CCCCN1C(=O)CC1CC12CC2 48829,c1(OC)cc(C(=O)NCC(CC(C)C)NC(=O)C=CC2CCOC2)n(C)n1 48830,N12CCCC(CC1)NC(C)CC2=O.C1(CC)CCC(CC(=O)OC(C)(C)C)CC1 48831,N1(C(CC2(C#N)CC2)=O)CCc2c(CNC(=O)CC3=CCOCC3)cccc2C1 48832,c1(C(=O)O)cn2c(n1)CCCN2c1nc(-c2ccccc2)ns1 48833,CC(C)CCCCC(=O)N1CCCC1C(C)NC(=O)C(C)n1cccc1 48834,C1(COC)(NC(=O)CCn2cncn2)CCN(C(=O)COC2CC=CC2)C1 48835,C#CCC(C)(CC)C(=O)NCC1(O)CCN(C(=O)COCCCC)C1 48836,Cc1cc(NC(=O)CC2COCCO2)ccc1NC(=O)CNS(=O)(=O)C1CC1 48837,C(CC(=O)N1CCCC(CNC(c2cc(F)cc(C)c2N)=O)C1)(C(F)(F)F)OC 48838,c1(OC(C)C(=O)NCCC(C)N(C(=O)CSc2cccnc2)C)ccccc1Cl 48839,C(=O)(C1CCc2nccn21)NCC1CC(OC)CN1C(c1cc2occc2[nH]1)=O 48840,N1(C(=O)CCc2ccon2)CCC(NC(C2CC(n3ccnn3)C2)=O)CC(O)C1 48841,C(CCCC(=O)NON(C)C(c1ccc(F)c(O)c1)=O)N(C)C 48842,C(=O)(CCC(F)(F)F)N1CCN(CC2(NC(=O)COC3CCOC3)CC2)CC1 48843,C1(NC(c2c(OC)cnc(Cl)c2)=O)CC2CCC(C1)N2C(C1(C)CCCS1)=O 48844,N1(C(C(C(C)C)NC(C)=O)=O)CC2(CCN(C(c3cnc(S)nc3)=O)CC2)C1 48845,O=S(=O)(c1cnccc1N1CC2C3CCC(C3)C2C1)NCC(C1CCOCC1)O 48846,C1(NC(CC2(C)CCOCC2)=O)CC(C(=O)NCc2nnc(O)o2)=CC1O 48847,c1(N(C(CCC#N)c2ccccc2)C)ccc(S(=O)(=O)NC2CCOCC2)cc1Cl 48848,Cc1ccc2occ(C(=O)NCC3CN(C(C4CC(O)C4)=O)CC(C)(C)O3)c2c1 48849,N1(C(C=NOC)=O)CCC2CN(C(=O)Cc3cc(C)ccc3C)CC12 48850,c1(C(N2CCC(CCNC(C(C)c3ccco3)=O)C2)=O)ccc2nc(O)sc2c1 48851,C1(C(=O)NCCN(C(=O)CC2CCCOC2)CC)CCC(Oc2ccncc2)C1 48852,C(C)(CC(=O)N(C1CCN(C(=O)Cc2csc(NS(C)(=O)=O)n2)C1)C)OC 48853,Cc1snnc1C(=O)NC(CN(C)C)C(=O)NCCC1(O)CCOC1 48854,c1(OC)cccc(NC(=O)CN(CC(C)C)C(c2ccnn2C(C)C)=O)c1 48855,CC1CN(C(=O)C(c2c(Br)cnn2C)C)CC1n1cc(-c2cccc(F)c2)nn1 48856,N1(C(CCCOCC=C)=O)CCC(C)(CNC(=O)COc2ccon2)C1 48857,C#Cc1ccc(C(=O)NC(c2ccccn2)C(C)C)c(CC)c1 48858,CCCCCCCCCC(CC)C(=O)N1CC(C2(NC(C3CC=CC3)=O)CC2)C1 48859,c1(OC)ccc(Cl)cc1C(N1CCC(NC(c2c(C)[nH]c(C)c2C)=O)CC1C)=O 48860,CCCC(CCCNC(=O)CCNC(C1CCCO1)=O)NC(=O)CNC=O 48861,C1(NC(c2ncc(OCC)nc2)=O)CCC(C)N(C(=O)CCC#N)C1 48862,c1(CC)cccc(NC(C2(C)CCCN2C(=O)C(c2ccc(C)o2)C)=O)c1F 48863,N1(Cc2n(CC)ncn2)CCCCC(NC(=O)CC2COC(=O)C2)C1 48864,C12(NC(c3cnco3)=O)CCN(C(c3ncoc3-c3ccco3)=O)CC1C2 48865,C1(C)(C(N(CCCC#C)C)=O)CC12CCN(c1ncc([N+](=O)[O-])c(C)n1)CC2 48866,N1(C(c2ccc(OC)cc2O)=O)CC2CCN(C(=O)CCCCC(C)=O)CC2C1 48867,N1(C(CSCCNC(C(COCC)N=[N+]=[N-])=O)=O)CCCC(C)(CC)CC1 48868,Cc1ncccc1CCC(=O)N(CC(O)CN(C)C(C1C=CCS1)=O)C 48869,N1(C(CNCc2n(C)c(O)nn2)=O)CCC2(CC1)CC2(C)C(=O)NC1CC1 48870,C12(C(=O)NC(C(C)(C)NC(Cc3c(C)n(C)nc3)=O)C)CC(CO)(C1)OC2C 48871,C(=O)(CCCCCC(C)O)NCCC1(NC(c2c(CCC)cccc2)=O)CC1 48872,C(=O)(C(C)(C)CCC#N)N(CC(C)(C(C)C)NC(C=NOC)=O)c1ccccc1 48873,c1(CC)cccc(NC(=O)C(Cn2cncn2)NC(c2nonc2N)=O)c1C 48874,C(c1cc2ccccc2o1)=CC(=O)NC1C=CCN(c2cc(CC)nc(Cl)n2)C1 48875,O=C(C(=O)C(F)(F)F)NCc1cn(C2CCN(C(=O)C3=CCC3)C2)nn1 48876,N1(C(C=NOC)=O)CC2(CC(NC(c3cc(Cl)ns3)=O)c3nccn32)C1 48877,CC(C)(C)C(=O)NCCCC(=O)NCC1(NC(=O)Cn2ccc(=N)[nH]2)CC1 48878,C1(C(N2CC(CC(=O)NC(CC)COCC3CC3)C2)=O)CCCOCC1 48879,N1(C(C2(C3(C)CC3)CC2)=O)CC(C(=O)NC2(C)CC2)C2(CCC2)C1 48880,N1(C(C(COC)(C)C)=O)CC2(C)CC1(C(=O)NC(C)CCC1CCCO1)C2 48881,C(=O)(C1(C)CCOc2ccccc21)N(CCNC(C(CCCC)CC)=O)C 48882,C1(C(N2CC(CCNC(=O)CSc3ccccc3Cl)C2)=O)CCCC2CCCN12 48883,C(=O)(C(CCCC)NC(C1CCCSC1C)=O)N1C(C=C)CCC1 48884,Cc1nc(C(N2CCCC(NC(=O)C(C)Cc3ccnn3C)C2)=O)c(C)s1 48885,C#Cc1cccc(C(N2CCC(N(C)CC)C2)C(=O)NC2CCOCC2)c1 48886,C#CCCCCCC(=O)N(CCCN(C)C)CCNC(C1(F)CC=CC1)=O 48887,N1(C(CC2CCN(CC)C2)=O)CCC(CCCCNC(C2C3COCC23)=O)CC1 48888,C12(C(=O)NC3CCC3C(=O)N(C3CC(N(C)CC)C3)C)CCC(OC)(CC1)C2 48889,NC(=O)N=Nc1ccc(C(=O)NC2CC(CNC(C3CCCN3C=O)=O)C2)cc1 48890,n1(CC)ncc(CNC(=NCc2ccnn2C)NC2CC(=O)N(C3CC3)C2)c1C 48891,Cn1nc(-c2nc(-c3ccccn3)no2)c2c1CCN(Cc1ccccn1)C2 48892,N1(C(CCSCC)=O)CCC2(CC1)CC2CNC(=O)C(C)(C)F 48893,N1(C(Cc2ccc(C)o2)=O)CC(NC(c2cncn(C)c2=O)=O)CC1(C)C 48894,c1(OC)ccc(F)cc1CNC(=O)NC(c1cccc(Br)c1)C1CC1 48895,CC1CN(C(C2(C)CCCN2C)=O)CCC1C(N1CCCC(CO)(CO)C1)=O 48896,n1(CC=C)cccc1C(=O)NCC(C)NC(=O)Cc1ccoc1C 48897,Cc1noc2nc(C(C)C)cc(C(N3CCCC(S(N)(=O)=O)CC3)=O)c12 48898,C1(NC(C2CN(C)C(=O)C2)=O)CC2CCCC(C1)N2C(c1cccn1C)=O 48899,C1(C(=O)NC(CNC(c2c(C)cnnc2)=O)C)CCCCCS1(=O)=O 48900,c1(OC)cc(F)c(CSc2ccnc(Cl)c2Br)cc1F.c12sc(cc1C)[nH]c2=O 48901,c1(C(=O)NC(C)CNC(=O)C(F)Cc2ccccc2)cccn2ccnc12 48902,CN1CC(C)(C(=O)NCCCNC(c2ccccc2SC(C)(C)C)=O)CC1=O 48903,n1(CC)ncc(CNC(C2(C)CCN(C(=O)CN=[N+]=[N-])C2)=O)c1C 48904,CC(C)(CCCF)NC(C12CC(NC(=O)CC=C(Cl)Cl)(C1)C2)=O 48905,C1(C(N2CC(OCCCCC)C2)=O)CCN(C(c2cc(C)c(C)cn2)=O)CCO1 48906,c1(C(N2CCC(O)(CCNC(C3C(C)(C)CO3)=O)C2)=O)cc2scnc2[nH]1 48907,Cc1ccc(C(c2nnnn2CC2CCOCC2)NCCc2scnc2C)s1 48908,N(C(=NCCOC1CCCCC1)NCC(C)(C)OC)C1(OCC)CCC1 48909,C1(CC#C)(C(=O)NCc2ccnc(OC)c2)CCN(C(=O)C(O)c2ccsc2)C1 48910,N1(C(c2ccc(OCCO)cc2)=O)CCCN(CC(=O)NCC(F)F)CC1 48911,C(=O)(CCCCC(C(F)(F)F)NC(=O)NCC1COC2(CCCC2)O1)OC 48912,N1(C(C(C=C=C)C)=O)CCCN(C(c2cnc(C)s2)=O)CC1C(C)C 48913,C#Cc1ccccc1CC(N1CCC(C)(C(=O)NC(C)C(C)(C)CC)CC1)=O 48914,c1(CN(CCCNC(c2ncccc2C2CC2)=O)CC)ccc2n[nH]cc2c1 48915,NC(CCc1ccncc1)C(=O)N(c1nccn1C1CC1)Cc1ccccc1F 48916,Cn1nc(O)cc1C(=O)NCc1csc(CNC(=O)Cn2cc(C(F)F)cn2)n1 48917,C1(C(=O)NCC(N2CCCCC2)=O)CC2CNCC1O2 48918,C(C(C)(C)CC(=O)N(CCCNC(C1CCCN1CC(C)C)=O)CCO)OC 48919,c1(C(N2C(CNC(CC=CCC)=O)CCCCC2)=O)ncc(Cl)c(N)c1Cl 48920,c1(C(=O)NCC2C(C(=O)NC(CC)C3CC3)CCO2)ccc(F)cc1C 48921,n1(CC)c(C(=O)NCCN(C2CCCCC2)C(=O)CCOC2COC2)cnc1O 48922,C1(CNC(C2NC(=O)OC2)=O)N(C(C2Cc3ccccc3O2)=O)CCCC1(C)C 48923,C(=O)(C(C(C)C)C(C)C)NC1CC(N(C(c2c(C)cc[nH]2)=O)C)C1 48924,N1(CC(=O)NCC2ON=C(C)C2)CCN(C(=O)C=C(Cl)Cl)CC1 48925,C(C#CCN=c1[nH]c2c(c(=NC(=O)CC3SCCS3)[nH]1)COC2)OC 48926,Cc1cc(Br)cc2cc(CNC(=O)C(=O)N(C(C)CN(C)C)C)oc12 48927,CC1ON=C(C(=O)NCCC2CN(C(=O)C#CC(C)(C)C)CCCO2)C1C 48928,c1(N(S(C)(=O)=O)C)cc(Cl)c(Cl)cn1.n12cc(nn1)C1(C)CN(C1)CC2 48929,N1(C(c2n(C)ncc2Cl)=O)CC2CCC(C1)C2CNC(=O)C(O)CC(F)(F)F 48930,C1(C(=O)NCC2=NOC(C)C2)CCCCCC1NC(c1nccs1)=O 48931,C12(NC(c3cc(C(N)=O)oc3)=O)CCCC1N(C(c1cscn1)=O)CC2 48932,C12(NC(CCS(C)=O)=O)CCOCC1CN(C(C1(c3cc[nH]n3)CC1)=O)C2 48933,C=CCC(C(=O)NC(C1(O)CN(C(c2cccc3ncsc23)=O)C1)C)C(C)C 48934,N1(CC(=O)NC2C3CN(C(c4[nH]n(C)c(=O)n4)=O)C2C3)CCC(=O)NC1=O 48935,c1(C(C)C)cc(C(=O)NCC(C2CC2)NC(=O)C(C)(C)c2cnco2)cc(O)n1 48936,C1(C(N2C(CNC(=O)Cc3cccnc3)COCC2)=O)CCc2ccccc2O1 48937,CC1CN(C(=O)C=CS(C)=O)CCCN1C(=O)CCCn1ccc(C(=O)O)n1 48938,C(CN=c1cc(N2CC(N3CCCCC3)C2)nc[nH]1)c1ccc(OC(F)F)nc1 48939,c1(C(=O)NC2(c3ccccc3)CCN(C(C=CSC)=O)C2)cc(C)nnc1O 48940,C1(C(=O)NCC(CC)NC(=O)CCc2cn(C)nn2)CCCC1c1ccccc1 48941,C1(C(=O)NOC2CCOCC2)CCCCN(C(=O)Cc2ncccc2F)C1.CN 48942,C(=O)(C(C)(C)C#N)NC(C1(C(=O)NC(C(C)C)CO)CC1)C 48943,c1(C(=O)NC2CCCC(N(C(=O)CC(C)(C)C)C)C2)cc(C(F)F)cc(Cl)c1 48944,C(c1c(Cl)cccc1Cl)=C(C(=O)NCC1(F)CN(C(C(=O)NCC)=O)C1)C 48945,Cc1nn(CC(N2CCCCCC(NC(c3ccsc3C)=O)C2)=O)cc1[N+](=O)[O-] 48946,C(CCCCC(=O)N(C(C)CNC(C1CC(OC)C1)=O)C)=CC 48947,C(C(C)(CO)NC(=O)CNC=O)NC(C1(OC(C)C)CCC1)=O.c1cccnc1 48948,CC(N=[N+]=[N-])C(=O)N(CCCC(N1CCC(C)(N(C)C)C1)=O)C 48949,CC1CCCC=C1C(=O)NC1CCN(C(=O)CC(F)(F)C(F)F)CC1(C)C 48950,c1(OC)cc(C(=O)NC23COC(C2)C(NC(c2cocn2)=O)C3)cc(OC)n1 48951,c1(C(N2CCC(N(C(=O)CCC3CC(OC)C3)CC)C2)=O)ccnc(Cl)c1OC 48952,N1(C(C2N(C(c3c(C)c[nH]c3)=O)CC2)=O)CCC2(CCCO2)C1 48953,C=CC1CCN(C(C2CCN2C(=O)C(C)OCC)=O)CC1 48954,C(CCC(C)C)(C(=O)N(C)CCc1ncccn1)NC(C1C(CCC)CCC1)=O 48955,CCS(=O)(=O)C=CC(=O)N1CCC(C)(C)C(CNC(c2cccn2C2CC2)=O)C1 48956,C1(OCC)CC(CNC(=O)CNC(=O)Cc2cc[nH]n2)C1 48957,C(c1cn(C)cn1)=CC(=O)NC(C(=O)NC(c1onc(C)n1)CO)CO 48958,C(=O)(CC1=NN(C)C(=O)C1)NC1CC=C(C(=O)N(CCCN2CCCC2)C)C1 48959,N1(C(c2c(CC)cns2)=O)CC(O)CCC1C(=O)NCCn1ncnn1 48960,C(=O)(NNC(=O)C1CCOC1)NCc1cc(C)[nH]n1 48961,C1(S(N)(=O)=O)(Cc2cc(-c3ncc(C(=O)OCC=CC(=O)OC)s3)on2)CCCC1 48962,N1(C(C(CC)(C)O)=O)CCCCC2(C1)CN(C(c1nn(C)cc1C)=O)C2 48963,c1(C(N2CC(O)(C(C)NC(C(CCCC)O)=O)C2)=O)cc(=O)c2ccccc2o1 48964,C1(C2CCCN(C(=O)C=Cc3cn[nH]c3)C2)(NC(=O)C(O)CN2CCCC2)CC1 48965,Cc1cc(=NCc2nc[nH]n2)[nH]c(=NCCS(=O)(=O)C2=NOC(C)(C)C2)[nH]1 48966,N1(C(C2(CCN(CC(=O)O)C)CC2)=O)CCOCC(C(N2CCC(C)(C)C2)=O)C1 48967,C1(C(N(C2CCN(C(c3cc(I)on3)=O)C2)C)=O)C2CCCC12 48968,CCCCCC(O)C(=O)N1C(C)C2CC1C2NC(C1(C(F)(F)F)CCCCC1)=O 48969,c1(C(N(C2CCCN(C(c3cc[nH]n3)=O)C2)C)=O)ccc(N)c(Br)n1 48970,CCC(C)(C)CC(=O)N1CCOC(C)(CNC(=O)COCP(C)(C)=O)C1 48971,c1(C(=O)NCC2(NC(c3ccc4c(c3)NCC4)=O)CC2)cnc2[nH]ccc2n1 48972,N1(C(C2N(C)CCC2)=O)CCOCC(NC(c2cccc(O)c2O)=O)C1 48973,c1(OC)ncc(Br)cc1CN(C1CCN(C(C2CCN(C)C2)=O)C1)C 48974,C=CCC(CC(C)C)C(=O)N1CC(NC(C2(C#N)CC(C)C2)=O)CC(F)C1 48975,C1(C2CCOCC2)(C(=O)NCC2N(C(CCCN(C(C)C)C)=O)CC(O)C2)CC1 48976,N1(C(C=C(C)C2CC2)=O)CC(O)CC1(C)C(=O)N(C)CC1(C)CC1 48977,Cc1sc(O)nc1C(=O)NC(C)CC1CCCN(C(C2(N3CCCC3)CC2)=O)C1 48978,CC(C)CC(C)CC(C)C(=O)NC1CN(C(=O)C(F)(F)CO)CC1C(F)F 48979,c1(C(=O)NCC(CNC(C(CN(C)C)N(C)C)=O)(C)C)cnc2ncccc2c1 48980,C1(CC)CNC(=O)CN1C(c1sccc1Br)C(=O)NCCCOCC1CC1 48981,c1(C(=O)NCCCN(C(C)C)C(C2CCCCC2(F)F)=O)cccc2occc12 48982,C(C(CO)NC(=O)Cn1cccn1)NC(C1C(CC)C1)=O 48983,N1(C(Cc2ncc(C)s2)=O)CCOC(CNC(C2CN(C3CCCCC3)C2)=O)C1 48984,CC#CCCCC(=O)NC1CCC1CNC(c1ncn(CC)n1)=O 48985,CCC(CC(=O)NC(C)CC(C)NC(c1c(C)cncc1C)=O)C(C)(C)C 48986,C(=O)(CC(C)C)NC(C(=O)N(CCOC)CCOC)c1cccs1 48987,C1(NC(C(C2CC(F)(F)C2)OC)=O)C=CCN(C(=O)CC2CC(=O)NC2=O)C1 48988,N1(C(N)=O)CCCC1C(=O)NC1CC(NC(c2cn(C3CCOC3)cn2)=O)C1 48989,c1(CN2CC(CNC(C3(CC)CCNC3=O)=O)OCC2)c(F)cccc1Cl 48990,Cc1ccc(C)c(C(=O)NC2CC3CC2N(C(C2(O)CC2(C)C)=O)C3)n1 48991,C(=O)(C#CC1(C)COC1)N1C(C)CCC(NC(C(C)(CO)OC)=O)C1 48992,C1(CNC(=O)CCCC2CCC2)CC2(CCC2)CN1C(=O)Cc1ccncc1Cl 48993,N1(C(CNC(CCC)=O)=O)CC(F)CC1CNC(c1c(C)ncn1C)=O 48994,c1(C(N2CCC(C)(CNC(c3cnc(C)o3)=O)C2)=O)cnc2ccncc2c1 48995,n1(CC(N2CCC(N(C(C3CCC(C)O3)=O)CCO)C2)=O)cc(S(N)(=O)=O)cn1 48996,C(=O)(NNc1cc(F)c(F)cc1Br)NCc1c(CC)onc1C 48997,c1(CC=C)cccc(NC(c2cc(CNC(=O)C(F)=C(C)C)nn2C)=O)c1 48998,N1(C(C2N(C(CNC(=O)NC)=O)C(C(C)C)CC2)=O)CCOCC1CO 48999,CS(=O)(=O)c1cscc1C(=O)NCC(CO)NC(C1(F)CC=CCC1)=O 49000,c1(NC(C2(OC)CCN(C(=O)CC3CC(F)(F)C3)C2)=O)cnn2c1CCCC2 49001,c1(C(C)=O)cc(S(=O)(=O)N2Cc3cccc(C)c3C(C)C2)cc2c1CCC2 49002,CC(C)CC(C)(O)C(=O)N1CCCC(CNC(=O)C#CC2CCC2)C1 49003,Cn1ncc(CC(=O)NC2CCC(NC(c3ccon3)=O)C2)n1 49004,c1(OC)ccc2c(c1)C(NC(=O)NCC1(C(F)F)CCCCC1)CCC2 49005,CCC(C#N)C(=O)NCCCCCNC(c1ncccc1OC)=O 49006,C(=O)(C(CC1CN(C(=O)OC(C)(C)C)C1)NC(C1CC1F)=O)NCC(=C)C 49007,CC1(C(N2CCCC(O)C2)=O)CCCN(C(c2ccccc2-c2cccs2)=O)C1 49008,c1(C(=O)NC(CNC(c2c(CC)non2)=O)CCOC)coc2ccccc12 49009,c1(C(COC)NC(=O)C(=O)NCc2ncc(Cl)s2)ccc(C#N)cc1 49010,c1(C(N2CC3(C(NC(C(CCC)C)=O)CC3)C2)=O)ccc2cc(C)cn2c1 49011,n1(CCC(=O)NC2CCN(C(c3c(C)ncnc3)=O)C2)cc([N+](=O)[O-])nc1C 49012,c1(N)ncc2ccccn12.N12CCCC(C1=O)N1CC2C1.C1(CC)CCC(F)(F)CC1 49013,C1(C2CN(C(=O)CC3CCC4CC34)C2)(NC(c2cc(OCC)ncc2)=O)CC1 49014,N1(C(C(CC)SC)=O)CC(CNC(=O)CSC(F)F)C(F)(F)C1 49015,C(C(=O)NCC1(NC(c2cnn(CC(C)C)c2C)=O)CC1)(C(C)C)SC 49016,c1(NC2CCC(SCC)C2)ccc(S(=O)(=O)NCc2nnc(C)o2)cc1C#N 49017,C#CCC(CC(=O)OC)NC(=O)CC1(NC(=O)CC(O)C(C)C)CC1 49018,C1(C(=O)NCCN(C(C(CC)(C)O)=O)CC2CC2)CCc2ncnc(C)c2C1 49019,C(=O)(C(CC1COCCO1)C(F)(F)F)NCCNC(CN(c1cnccn1)C)=O 49020,C(=O)(C(C)(C)C(C)O)NC.C12CCC1C(=O)N(CC)CCCNC2=O 49021,c1(OC)ccc2cc(C=CC(=O)NC3CCN(C(=O)C(C)C)C(C)C3)ccc2c1 49022,C#Cc1ccc(CNC(=O)CC2(NC(=O)CC3CCSC3)CC2)cc1 49023,C#Cc1ccc(C(=O)NCC2CC2C(N2CC3CC3(CC)C2)=O)c(C)c1 49024,CCCCCS(=O)(=O)CC(=O)N1CCCC2(NC(c3ccc(C)o3)=O)CC2C1 49025,O=C(CCC(CF)CF)NC1COCC1CNC(c1cncc([N+](=O)[O-])c1)=O 49026,CCCCC(C(=O)NCC1CCCN(C(c2cccc[n+]2[O-])=O)C1)C(C)C 49027,C(=O)(CS(=O)(=O)C(C)C)N(C)CC1CCN(C(c2c(CCC)nco2)=O)CC1 49028,C(=O)(C1=NOC2(CCC2)C1)NCC1(C2(O)CN(C(c3ccnc(C)n3)=O)C2)CC1 49029,c1(NC2CC(C)N(C(=O)CCc3ccccc3)C2)ncc2ncnc-2[nH]1 49030,c1(C(=O)NCCCCC(CO)NC(C2CC(OC)C2)=O)cccc2c1OCC2C 49031,C1(NC(=O)C(F)OC(F)(F)F)(CO)CCCN(C(C2(Cl)CC2)=O)C1 49032,c1(C(=O)NC(C(=O)OCC2CC(=C)C2)CC2CCCO2)c[nH]nc1[N+](=O)[O-] 49033,c1(OC)nc(N2CC3(CCN(C(c4cncc(C)n4)=O)C3)C2)ncc1C#N 49034,N(C(=NCCF)NC(C)CC(F)(F)F)CC1CC(CC)C1 49035,CC1C(NC(c2cn(C3CC3)nn2)=O)CCCN1C(c1cncc(F)c1)=O 49036,Cc1nc(C(=O)NCC(CO)NC(C2CCC(=O)N2)=O)co1 49037,N1(C(=O)C=CCc2ccon2)CCC2(NC(=O)C=C3CCC3)CCCC12 49038,c1(OC)ccc(C(N2CCC(NC(=O)Cc3ccnc(Br)c3)C(O)C2)=O)cc1O 49039,C(=O)(CC(O)CNC(C1CCN(C)C1)=O)N1C(C(=O)NC)CC1 49040,C1(C(=O)Sc2cccc(NC(C)C)c2)CC(C)(C)CO1.C1(OC)CC2(C1)CN2 49041,c1(C(=O)NC(CC)CNC(=O)CC2COC(=O)C2)nnc2n1CCCCC2 49042,C(c1ccc(S(C)(=O)=O)o1)=CC(N1CCC(NC(C#CC2(C)CC2)=O)C(O)C1)=O 49043,C(C(=O)NNC(=O)c1ccc(I)c(I)c1)NC(c1c(C)cccn1)C1CC1 49044,CC1CCCCC1(CNC(c1ccc(=N)[nH]c1)=O)NC(C1(CN(C)C)CC1)=O 49045,N1(C(C=CSC)=O)CC(NC(=O)Cc2cc(COC)on2)C(C(F)(F)F)C1 49046,c1(NC=O)ccccc1C(=O)NCC1(F)CC(NC(c2conc2C2CC2)=O)C1 49047,C1(NC(CCOC(CC(C)C)C)=O)CN(C(=O)CNS(C)(=O)=O)CC1C(F)(F)F 49048,N1(C(c2c(C)ncn2C)=O)C2CCC1CN(C(=O)Cc1ccncc1Cl)C2 49049,CC1CC(CNC(C2(C)CCSCC2)=O)CN(C(c2cn(C)[nH]c2=N)=O)C1 49050,C1(CNC(C=CC=CCC)=O)CCCC2CN(C(c3ccc(CC)cc3)=O)CC12 49051,N1(C(c2ccc([N+](=O)[O-])[nH]2)=O)CC2CC(C1)N(C(c1coc3ccccc13)=O)C2 49052,N1(C(C=CCCC)=O)CCN(C(=O)CC2CN3CCN2CC3)CC1CO 49053,c1(C(=O)NC2CC(NC(C3C(C)(C)CCCC3)=O)CC2O)cc2ccccn2c1 49054,c1(CNC(CCCCOC)C)cc(O)ccc1[N+](=O)[O-].c1(N)ccccc1 49055,C1(NC(c2c(OC)cccc2)=O)CCCN(C(=O)C(=O)CC(C)C)C1C 49056,C1(CNC(CC2ON=C(C)C2)=O)CCC(N(C)C(c2cncs2)=O)CC1 49057,c1(C(N2C(COC)(CNC(c3occc3C)=O)CCC2)=O)csc(=NC2CC2)[nH]1 49058,C(=O)(C1CCSc2ccccc21)NC(CC=C)CNC(=O)CCCC(=O)OCC 49059,C(=O)(CCC(C)(C)C)C(CC1C(C)CN(C(=O)CC2(C)CCOC2=O)C1)=O 49060,C(=O)(C#CC1CCOC1)NC(C)C(C)NC(c1ncsc1Br)=O 49061,c1(C(=O)NCc2ncc(CC)o2)ncc[nH]c1=NCC1(SC)CCC1 49062,c1(C(=O)NC2CN(C(C(CCC)(C)C)=O)CC3C2C3)nc2ccccc2cc1Cl 49063,c1(C(N(CCC)CCNC(C2CC(C)(C)CO2)=O)=O)cc(F)ncc1OCC 49064,c1(C(=O)NCC2CCC(C(N3CC(C)(O)C3)=O)O2)occ2c1CCC2 49065,c1(NC(C(c2ccco2)NC(COC(CC)CC)=O)=O)ccc(F)cc1O 49066,N1(C(c2cc(CC)[nH]n2)=O)CCCC(CCC(=O)NCC(C)C(C)C)C1 49067,C1(C)(c2cn(C(C(=O)OC)C)nn2)CCCN1C(=O)CO 49068,Cc1[nH]c(C#N)cc1C(=O)NC1CC2CC(NC(c3cnsn3)=O)CC12 49069,c1(NC)cnc(C(=O)NC2CCCC2NC(=O)CC#N)cn1 49070,CC(C)(C)C(O)C(=O)N1CCCCCC1CNC(c1cnc2sccn12)=O 49071,CCCC(O)C(=O)N1CCC(C)(NC(=O)Cc2nc(C)sc2C)C1 49072,C1(SCC)CCN(C(=O)CC2CCCC2NC(C2CCOCC2)=O)CC1 49073,Cn1nnc2cc(N3CC(C(=O)Oc4ccc5c(c4)OCO5)CC3=O)cnc12 49074,CCC(CC)(CC)C(=O)N1Cc2occ(C(=O)NCC3CCCCC(O)C3)c2C1 49075,CC1(C)C(CC(=O)NC2CCCC2)CC1c1cn(C2CCOC2)nn1 49076,C1(NC(CCn2c(C)ncc2)=O)CC2CC(C1)N(C(=O)C(=O)NC(C)C)C2 49077,N1(C(c2cc(C)on2)C(=O)NCCCN(C)C)C(CN=[N+]=[N-])CC2CC12 49078,C(=O)(C1=CCCN(C(c2cc(F)ncc2Br)=O)C1)NC(C)CN1CCCC1 49079,C1(CNC(C(C2CC2)OCC)=O)N(C(=O)C=C2CCCC2)CCCC1(C)C 49080,C12(CNC(c3ccc(OC)nc3)=O)CCCN(C(=O)CCc3nccs3)C1C2 49081,C(=O)(C(O)CC(C)(C)C)NC(C(C)NC(=O)CSc1nccn1C)C 49082,C12(CC(=O)NCCSCC)CCC1CN(C(C1(OC(C)=O)CC(C)(C)C1)=O)C2 49083,CCC(C)C(O)C(C)C(=O)N1CCC(O)(CNC(=O)C(C)S(N)(=O)=O)C1 49084,C#Cc1cnn(CC(N2CCC(NC(c3n[nH]cc3CC)=O)C2CC)=O)c1 49085,C(CC(C)N(C)CC)OCCO.C(CCCC)SCC 49086,C=C(C)C(CC(=O)N1CCCCC1C1(CNC(c2csnc2C)=O)CC1)OCC 49087,C(=O)(C(CN=[N+]=[N-])NC(C12CCCC1C2(F)F)=O)N(C1CC2(CCC2)C1)C 49088,Cc1cncc(C(=O)NC2CC2CNC(=O)C=CCOC(C)(C)C)c1Cl 49089,O=C(CC1CN(S(=O)(=O)Cc2ccc([N+](=O)[O-])cc2)C1)N=c1cc(C2CC2)[nH][nH]1 49090,C(=O)(C(C)C(C)(F)F)N1CCCC(CN2CCN(C(C(C)NC(N)=O)=O)CC2)C1 49091,C(=O)(C1CCc2ccccc21)NCCN(C1CCCCC1)C(c1c(C)con1)=O 49092,C1(N(C(=O)CC2(C)CCC2)CC)CCCN(C(C2(C)CCCOC2)=O)C1 49093,C1(C(=O)NCc2c(C(=O)NC3(CCC)CCC3)c[nH]n2)CCNC(=O)C1 49094,c1(NC(c2cccc(OCCC)c2)C)cc(C)c(C(=O)O)cn1 49095,N1(C(=O)CCOC2CCC2)CC2(CC2)CC1CNC(C1(CF)CCC1)=O 49096,Cc1cccnc1C=CC(=O)NCC(C)CN(C(=O)CN1CCC(F)CC1)C 49097,CS(=O)c1ccc(C(N2CCC(C)(C)C2CNC(=O)Cc2nc[nH]n2)=O)cc1 49098,C1(C(=O)NC2CC(NC(c3ccc(-n4ccnc4)cc3)=O)C2)CC2(CC2)CO1 49099,C(=O)(C1COc2ccc(Cl)cc21)NCC1CN(C(c2ccn(C)c2)=O)C(C)(C)C1 49100,CC(C)(CC(=O)N1CCCC1N1CCN(C(=O)CCN2CCC(F)C2)C1)C(F)F 49101,c1(OC)ccc(C2(C(=O)NC3CN(C(C4CC(OC)C4)=O)C3)CCC2)cc1 49102,C(C1CN(C(=O)CNC(C)=O)Cc2ccccc21)NC(C1C(OCC)C1)=O 49103,c1(CCC(=O)NC(C2CCCN2C(c2cnc[nH]c2=N)=O)(C)C)ccc(Cl)nc1 49104,C1(C(=O)NC(C(=O)NC)C)CC(N=[N+]=[N-])CN1C(c1sccc1Cl)=O 49105,NS(=O)(=O)CCCC(=O)NCC1CCCCO1.C12CCCCN(C1)C2 49106,N1(C(C(CC)F)=O)CCOC(CN(C)C(c2csc(-c3ccsc3)n2)=O)C1 49107,C(=O)(CCCC(=O)NCCNC(C)=O)N1CCN(C(C(CN(CC)CC)F)=O)CC1 49108,C(=O)(C(C)(C)C(=O)N1CC2(NC(=O)CCc3ncccc3C)CC1C2)OC 49109,C(F)(F)(C(=O)NOCC(=O)NC1COCCC1(F)F)c1cc(OCC)no1 49110,CN1CC(C)(C(=O)NCC2CN(C(=O)CCc3cnc(O)[nH]3)CCO2)CCC1=O 49111,C(N=c1[nH]cnc2c(Br)cccc12)C1CN(C(c2c(OC)nsc2)=O)C(C)C1 49112,C1(NC(c2cncs2)=O)CCCOC12CCN(C(c1cc(Cl)cs1)=O)CC2 49113,n1(CC(=O)NC2CCC(CNC(CC3CC(CC)C3)=O)CC2)ccc(O)nc1=O 49114,C(C)(C)(CCC(=O)NCC(O)C(N1CCCC(C(C)OC)C1)=O)OC 49115,N1(C(=O)COCC(F)(F)F)CCN(C(C2(CCc3cccs3)CC2)=O)CC1CO 49116,C1(CNC(C(CC)CO)=O)CN(C(C2CNC(=O)O2)=O)CC(C)(C)C1 49117,c1(NC(=O)C(=O)NC2CCN(c3ncco3)C2)ccc2c(c1)C(=O)NCCO2 49118,Cc1c(-c2cccc(NS(=O)(=O)c3cccc(Cl)c3)n2)cccc1[N+](=O)[O-] 49119,C1(NC(C=NOC)=O)CC(C2CCN(C(c3cc(N)c(O)c(F)c3)=O)C2)C1 49120,O=S(=O)(c1[nH]c(=NCC2OCCOC2F)ccc1Br)N1Cc2cccc(Cl)c2C1 49121,c1(C(N2C(C)C(NC(=O)CC(C)(C)C)CC2)=O)cc(S(=O)(=O)NCCO)c[nH]1 49122,CC(C)C(C(=O)NCc1cnn(C(C)C(=O)O)c1)c1ccnc(C(=O)O)c1 49123,Cc1nccnc1N1CCN(c2nnc(-c3ccnn3C)n2CCC#N)CC1 49124,C(C(=O)NCCCF)(C(CC)CC)N(CC(CCCC)CC)c1cccc(Cl)c1 49125,C1(NC(CC(=C)C)=O)CC(O)CN(C(c2ccc(-c3nccs3)cc2)=O)C1 49126,CC(C)(C)C(CCn1cc(-c2ccc(Br)c3[nH]ccc23)nn1)C(F)F 49127,C(=O)(C(C)(C)CSC)NCCN(C(C(C)NC(CC)=O)=O)C1CCCC1 49128,C1(NC(C2(C)CC2(Cl)Cl)=O)CCCN(Cc2cn(Cc3csc(Br)n3)nn2)C1 49129,N1(C(C(C=C)(C)CC)=O)CCC(NC(=O)C2=C(C)OCCS2)C(F)(F)CC1 49130,c1(-c2cn(CCN(C(=O)C(c3cccnc3F)(C)C)C)nn2)cnccc1Cl 49131,c1(C(N(C(CCNC(C2N(C(C)=O)CSC2)=O)C)C)=O)cc2ncccc2o1 49132,c1(C(=O)NC2CN(C(c3cc(CC)c(CC)o3)=O)CC2C)c(N)ccc(F)c1C 49133,N1(C(C=CCC)=O)CC2CC(NC(c3cn(C)nc3-c3ccco3)=O)C1C2 49134,C(C)(c1cccnc1)=CC(=O)NC(CCOC)CNC(C1(C)CC=CCO1)=O 49135,C(c1ccccc1Cl)=C(C(N1CC(CNC(CN(C2CC2)CC)=O)OCC1)=O)C 49136,CCN=c1cc(C(N2CC(NC(=O)CC(C)c3ccncc3)C(O)C2)=O)cc[nH]1 49137,C1(C(=O)NC(c2ncnn2C)C)CCN(C(=O)CN2CCSCC2)C(C)(C)C1 49138,Cn1ncc(Cl)c1C(=O)NCCCCCCNC(C1CCCCS1)=O 49139,C1(CC(N2CC(N(C(=O)COc3ccn(C)n3)C)C2)=O)CCCC(C)O1 49140,N1(C(CCCCN(C)C)=O)CCC2(CCC2)C(CNC(C2CS(=O)(=O)C2)=O)C1 49141,N1(C(C(C(C)(C)C)(C)C)=O)CCC(NC(c2ccc(N)c(Cl)n2)=O)C(F)(F)CC1 49142,c1(C(=O)NCCC(C)(C)NC(c2cc(OC)no2)=O)ncccc1SC 49143,N1(C(CCSCC)=O)CCN(C(=O)CN2CC(C)C2)CC1c1nccn1C 49144,C1(C(=O)NC(C(=O)N(C(C2CCCC2)C)C)C2CC2)CN(C)CCN1C 49145,c1(CCC(N2CCC(c3cn(C(C=C)C)nn3)C2)=O)cc(OC)c(Cl)cc1OC 49146,C(CN=c1nc(N2CCN(C(C)C)C(=O)C2)c2c(ncn2C)[nH]1)N(CCO)CC 49147,N1(C(C2(C)COCCO2)=O)CC2=C(C1)CN(C(=O)CN1C(=O)CCC1=O)C2 49148,N1(C(c2cn(CCNC(CCC#C)=O)nn2)=O)CC(F)CC1CO 49149,c1(C(=O)N(C2CCN(C(=O)C=C(Cl)Cl)C2)CCO)ncc(C2CC2)cc1F 49150,c1(CC(N2CC(=C(CNC(CCC(C)C)=O)F)C2)=O)cc(F)cc(Cl)c1 49151,N1(C(C2N(N=O)CCC2)=O)CC2CCCC(C1)N2C(c1ccn2ccsc12)=O 49152,c1(OC)ccc(CCCCNC(C(C)C)C(C)(C)O)c2c1C(=O)CO2 49153,c1(C(N2CC3CC(C)C3C2)C(=O)NCCCSC)cccc2cc[nH]c12 49154,N1(S(Cc2ccc(C)cc2)(=O)=O)CCC2(CC1)CCN2C(=O)Cc1cc(Br)cs1 49155,n1(CC(=O)NCC(CNC(CC(C)c2ccco2)=O)O)cnc([N+](=O)[O-])c1 49156,c1(CC)ccc(NC(C2(CNC(=O)C(C)CC3CCCC3)CCOC2)=O)cc1 49157,c12ccc(cc1Cl)NC(=O)N2.C(=O)(C(C(C)(C)C)c1cc[nH]n1)NC 49158,Cc1nc2cccc(C(=O)NCC34CCCC3CCN4C(c3cnsn3)=O)c2[nH]1 49159,N1(C(C2CC(CC)C2)=O)CCCC(O)(CN(C(=O)CCC(C)C)C)C1 49160,C1(NC(CC(=O)OCC)=O)CN(C(C2CC(=O)NC2(C)C)=O)CC2(CCC2)C1 49161,c1(NCCc2cn(CC)nn2)cc(F)ccc1CN 49162,[N-]=[N+]=NC1COCC1NC(=O)CC(CNC(=O)CN1CC2CCC1C2)C1CCC1 49163,N1(Cc2cc(OC)cc(Cl)c2)C(=O)C2C(C)CCCN2C1=O 49164,C1(C(=O)NCCc2cnc(C)s2)CN(C(=O)CC2CCOC2)CC1(F)F 49165,c1(CCC(=O)NCC2(O)CCN(c3snc(C(=O)OC)n3)C2)c(C)ncnc1O 49166,c1(C(=O)NCC2CCCN(C(c3c(OC)ccs3)=O)C2)ccc([N+](=O)[O-])c(F)c1 49167,c1(OC)c(Cl)ccnc1NC(C1CCC(Nc2ncc(F)c(C)n2)CC1)=O 49168,N1(C(=O)Cc2c(F)cccc2Cl)CC2CCC(C1)N(C(c1ccns1)=O)C2 49169,C1(NC(c2cccc(C)n2)=O)CC2CCC1CN2C(c1ccn(C(C)(C)C)n1)=O 49170,Cc1cc(Cl)c(C(=O)NCc2ccc(CN(C)C(C3CCCCC3C)=O)cc2)s1 49171,CCCC(C#N)C(=O)NC(C1(C(=O)NCC(C)CCC)CC1)C 49172,N1(C(CN(C(C)C)C)=O)CC2(CCCCN2C(C2CCCC3CCCCC23)=O)C1 49173,C1(F)(CNC(c2c(C)cc(F)s2)=O)COCCN(C(=O)C2=CCSC2)C1 49174,CC1CCC(C)(C(=O)NCc2cc(C(N3CC(C(C)(C)C#N)C3)=O)n[nH]2)C1 49175,Cc1cc(F)cnc1C(=O)NC1(CO)CCN(C(c2sccc2OC(F)F)=O)C1 49176,C(=O)(C(C(C)OC)N(C(c1ccnn1C)Cc1ccccc1)C)NCC=C 49177,C(=O)(CCCC(F)(F)F)N1C(CCC)CN(C(=O)COC2CCCC2)CC1 49178,CCCC(CC(=O)N(C)CC1(N(C)C)CCC1)NC(c1cc(Cl)c[nH]1)=O 49179,N1(C(C2CN(C)C2)=O)CCC2(CCC(C(=O)NCC3CCN3C(C)(C)C)O2)CC1 49180,c1(CCC(=O)NCCC(=O)NCCOC)ccnc(C)n1 49181,N1(C(C(C)(C)CF)=O)CC2(CCN(C(=O)CCCC3CCCCC3)C2)C1 49182,N1(C(CCCCOC)=O)CCOC(C)(CNC(=O)C(F)(F)C(O)C2CC2)C1 49183,C1(NC(C2CC3CCC2O3)=O)CN(C(=O)CCc2ncc[nH]2)C2(CCCC2)C1 49184,c1(C(=O)NCC2(C(=O)Nc3c(C(=O)OC)sc(I)c3)CC2)ccc(C#N)cc1F 49185,c1(C(=O)NC(CC)CNC(c2occc2F)=O)cc(N)c(F)cc1C 49186,C12(C(=O)NC(c3cccs3)C)CCC(CN(C(=O)CCCCCC#N)C1)C2 49187,C1(C(=O)Nc2ccc(COC)nc2)CCN(C(=O)C(C)C2CC2)O1 49188,C(=O)(C(C(C)(C)C)OC)N1CC(NC(CN(C)CC)=O)C(c2ccnn2C)C1 49189,N1(C(C=CC(C)NC(=O)C(F)CC2CCOC2)=O)CCCCCC1 49190,CCC(C)(C)CCNC(=O)CC(CNC(C1CCCS1)=O)C1CCC1 49191,C(=O)(C1CCc2nccn21)N1CCN(C(CC2C(C)(C)COC2)=O)CC1CCO 49192,c1(C(N2CCC3(C(=O)NC4CCC(OC)CC4)C(C2)C3)=O)c(Cl)ccc(F)c1Cl 49193,CC(C)CCCC(=O)NCCC1CC(NC(=O)C(C)CC(N)=O)C1 49194,C=CCC(C(=O)N(CCC(C)(C)NC(=O)C(C)CC1CCCC1)C)NC(C)=O 49195,c1(C(=O)NCCOCCNC(c2ccn(CC)n2)=O)ccc2ccsc2c1 49196,C1(CC(=O)NCC2N(C(c3c(C)nn(C)c3Cl)=O)CCC2)CCC2(CCC2)CO1 49197,C(C(CNC(=O)Cc1ccn(CC(C)C)n1)CO)NC(C1C(C(=O)OC)C1)=O 49198,c1(CN(C2CCNCCC2C)C(c2c(C)cccn2)=O)ccc(F)c(Cl)c1 49199,C(=O)(C1CCCn2nccc21)NC(C)CCNC(c1cnc(C(F)(F)F)s1)=O 49200,c1(C(=O)NCC2N(C(CC(CCSC)O)=O)CCCC2)[nH]nc2ncnc(O)c12 49201,C1(C(N(c2ccc(OC)c(Cl)c2)C(CC)C)=O)CCC2CC1C2(C)C 49202,CN1C(=O)CCC1C(=O)NCC1CCCC(CNC(=O)Cc2csc(=N)[nH]2)C1 49203,C1(NC(C(C)(F)F)=O)CC2CC(NC(C3(c4cncc(F)c4)CCC3)=O)C1C2 49204,N1(Cc2ccc(NC(CC(=O)OCC)=O)cn2)CCC(C(C)(C)C)C(O)C1 49205,C(=O)(CCCCCNC(C1(C#N)CC1C)=O)NCC1CC=C(C)CC1 49206,c1(C(N(CC(=O)OC)CCN2CCNCC2)=O)nnc(O)cc1O 49207,C(C(=O)N1CC(CO)(NC(=O)CCCCN2CCCC2)C1)(C(C)C)SC 49208,C1(NC(C2C(CC)C2)=O)CCC(NC(=O)CCOc2ccc(Cl)cc2)CC1 49209,N1(C(C2C(=C)CC2)=O)CCCC(C2CN(C(c3nc[nH]c3C(C)(C)C)=O)C2)C1 49210,C1(N(C(C2C(OC(C)=O)C2)=O)C)CCCCC1N(C)C(C1(C)CCSCC1)=O 49211,c1(CCC)ccc(C(N2CCC(CCOC)(NC(=O)OC(C)(C)C)C2)=O)cc1 49212,C(=O)(C1=CC(O)CCC1)NC1CCN(C(C2CC(C)(C(=O)OC)C2)=O)CC1 49213,Cc1csc2c(C(N3CCN(C(c4cc(Cl)cc(Cl)c4O)=O)CC3)=O)ncnc12 49214,c1(CN2CCN(C(=O)CCc3cccc(F)c3)C3C2C3)cccc([N+](=O)[O-])c1Cl 49215,C1(NC(c2cn(CC)nc2C2CC2)=O)CCN(Cc2ccccc2F)CC1C 49216,N1(Cc2cn(C)nn2)Cc2ccccc2C1C(=O)NC.NC1CCc2ccc(Br)cc21.N 49217,c1(CN2C3C(C(N4CCC(C(N)=O)CC4)=O)C(C3)C2)c(F)cc(Br)cc1F 49218,c1(CNC(c2cncs2)=O)cccc(-c2cccnc2)c1 49219,N1(C(c2c(N)ccc(C(C)C)c2)=O)CCC2CN(C(c3nccn3C)=O)CCC12 49220,N1(C(CC(CC)O)=O)CCCCC2(CCN(C(=O)CC=C(Cl)Cl)C2)C1 49221,c1(-c2ccc(OC)cc2SC)cc2c[nH]nc2cc1C(=O)Nc1ccc(I)nc1 49222,Cc1c(C(N2CCC(C(=O)NCc3noc(C(N)=O)n3)(CO)C2)=O)nnn1C 49223,Cc1cc(C(=O)NC(C)CCNC(=O)C2=CCCC2)cc(Cl)c1 49224,c1(C(=O)OC)ccc(CNC2CC2C(=O)Nc2cccc(F)c2)cc1 49225,C(=O)(C(C)(C)C(C)(C)O)NC(CCCNC(C1N(CC)CCCC1)=O)C 49226,C(=O)(C(C)(O)CC(C)C)N1CCN(C2CCN(C(CS(=O)(=O)NC)=O)C2)CC1 49227,c1(C(=O)NCc2cccc(F)c2)ccc(F)c(S(=O)(=O)N2CCC2)c1 49228,N1(C(C=C(CC)CC)=O)CC2CC(NC(c3ccnnc3S)=O)CC2C1 49229,C1(C(=O)NC2(CC=C)CN(C(C3(CF)CC3)=O)C2)CCCCC1C1CC1 49230,c1(C(N2CCN(C(C3C(C(=O)OC)CCC3)=O)CC2C)=O)ccc2n[nH]cc2n1 49231,CC1CC(CNC(=O)COC2CCC2)CCN1C(c1ncoc1-c1ccco1)=O 49232,C(=O)(C(F)CCC(C)C)NC(CC)CC(=O)NCCCC(C)O 49233,C1(CC)CN(C(=O)C(O)C(C)C)CCC1NC(=O)Cc1cc[nH]n1 49234,N1(C(C(C)=C(CC)C)=O)CCC2(CCN(C(=O)C(C)(C)C(F)F)C2)C1 49235,C1(NC(c2c(C)scn2)=O)CCCC(N(C)C(C2CCC(C)CC2)=O)C1 49236,C1(C(N(C2CC3C=CC2C3)C)=O)CCCN(C(=O)CN2CC(=O)NC2=O)CC1 49237,c1(CNC(c2cnc(C)n2C)=O)ccc(CNC(c2ccncc2C)=O)c(F)c1 49238,c1(C(=O)NC2(C)CCN(C(C3CC(C4CC4)=NO3)=O)C2)csc(=NC2CC2)[nH]1 49239,Cc1cc(CN2CC3CC3(C(N3CCCC(C)(O)CC3)=O)C2)c(F)cc1Br 49240,CC(C)(C)CCC(N)CNCc1cnccc1Cl 49241,C(=O)(CCCS(C)(=O)=O)NCC1C(NC(Cc2c(C)cccc2)=O)CCC1 49242,c1(CNC(c2c(C)scc2)=O)ccc(C(=O)NCCC2CCCC23CC3)nc1 49243,N1(C(C)=O)CCc2cc(C(N3CCCC(C(C)(C)C)CC3)=O)ccc21 49244,CC1=C(C(=O)N2CCC(NC(=O)CC3CCCC3)C(CO)CC2)CCS1(=O)=O 49245,C1(C#N)(C(=O)OCc2cc(C)c(Cl)cc2)CCCCCCC1 49246,c1(CC(=O)NCCOC2CCN(C(C(C)=CC)=O)C2)nn(C)cc1Br 49247,Cc1cn(C)cc1C(=O)NCC(C(=O)NCCC(=O)NC1CC1)N(C)C 49248,N1(C(Cn2c(C)nc(C)n2)=O)CCC2CCN(C(C3CC3C#N)=O)CC12 49249,C1(NC(C2CCN(C3COC3)C2)=O)CCN(C(c2ccncc2Cl)=O)C12CCC2 49250,C(=O)(C1=NN(CCO)C(=O)CC1)N1C(C)C(CC2CC2)CCC1 49251,CC(CC(F)(F)F)C(=O)NC(C)CC(C)NC(c1c(O)cc(O)cc1O)=O 49252,N1(C(c2cnc(COC)nc2O)=O)CCC2(C1)CN(C(C1CC1Br)=O)C2 49253,c1(OC)ccc(CC(=O)NC2CCCC2NC(C2CN(C)CCO2)=O)cc1Cl 49254,CCC(C(=O)N1CCN(C2CN(C(c3nncs3)=O)C2)CC1)C(C)C 49255,C(C(=O)NOC(CO)C(C)C)(C1CN(C(c2csc(F)c2)=O)C1)OC 49256,c1(CC)onc(C)c1CN(C(=O)NC(c1ccc(C(C)C)cc1)C)CC 49257,C(=O)(CC(C)(C)C(F)F)NC1C(NC(C(C)S(N)(=O)=O)=O)CCC1 49258,CN1CCN(C(c2cc3occc3s2)=O)C(CNC(c2ccc(O)c(O)c2)=O)C1 49259,Cc1nc(Cl)[nH]c(=NCC2CCCC(NC(=O)C(F)=C3CCCC3)C2)c1Cl 49260,N1(CC(=O)N(C)CC2(NC(C3CCC(CC)O3)=O)CC2)CCC(=O)NC1=O 49261,C#CCCCCCC(=O)N1CC(C)(C)CCC1CNC(c1cnn(C)c1)=O 49262,N1(C(C(C)NC(COC)=O)=O)CC2CCC(C1)C2NC(=O)CC1CC=CCC1 49263,c1(C(=O)NCC2(C)CCN(C(C3C(C(=O)OC)CC3)=O)C2)c(C)nn(C)c1OC 49264,c1(CNC23CC(NC(c4cc(Br)cc(Cl)c4Cl)=O)(C2)C3)c(F)cc(O)cc1F 49265,Cc1cc(C)c(CC(=O)NCCOCCCN(C(=O)C=CCOCCO)C)s1 49266,c1(NC(C(C)(N(C)C(c2ccnnc2)=O)C2CC2)=O)ccc(O)c(=O)cc1 49267,c1(C(=O)NC2CN(C(C(C=CC)O)=O)CC2O)cnc2c(c1)COCC2 49268,C(CC(=O)N(C1CC2CCC1O2)C)(C(F)F)NC(CC1C=NN(C)C1=O)=O 49269,C1(O)(CC(=O)NCc2cc(C(=O)NCc3ccc[nH]3)no2)CCCCC1 49270,c1(CC)cc(C(=O)N(CC(C)(C)C(=O)NC(CO)C(=O)OC)C)nn1C 49271,C(C)(CCC(=O)NC1CC(NC(c2cscn2)=O)C1)OCC 49272,C(=O)(CC(C)P(C)(C)=O)NC1C(CNC(C=C(C)c2cnn(C)c2)=O)COC1 49273,C1(CCC)CN(C(CC(C)C)C(=O)NC)CCN1CC(C)O 49274,C(=O)(C(C)C(F)(F)F)NCC(CCOC)NC(=O)C(O)C(C)(C)C 49275,c1(N)ccc2nn[nH]c2c1O.C1(C(C)(C)C)CCC(NC(=O)COC(=O)C2CC2)CC1 49276,C1(CCCC)CN(C(=O)C(C)c2cccs2)CCN1C(c1cnc(O)c(F)c1)=O 49277,N1(CC(=O)NCC2C(N(C(=O)CCCc3cccs3)C)CCC2)CCCOC1=O 49278,C(=O)(CC(CC(C)C)NC(=O)CC1CCC(C)(C)O1)NC(CCOC)CO 49279,C1(C(=O)NC23C(CN(C(c4cc(C)[nH]n4)=O)C2)C3)CCc2ccc(F)cc2C1 49280,c1(C(=O)NC(CC)CNC(c2csnn2)=O)cc(N)c(N)cc1F 49281,N1(C(CCN(CCCCC)C)=O)CCN(C(C2CC2C(F)F)=O)CC1COC 49282,c1(C(N2CC(O)(C(C)NC(C3CCCN3N=O)=O)C2)=O)ccc(C#N)nc1O 49283,c1(C(N2C(COC)CN(C(=O)C=C3CCC(C)C3)CC2)=O)cc(S(C)(=O)=O)co1 49284,C1(COC)CN(C(=O)Cc2cnoc2)CCN1C(C1CC(=O)N(C)C1)=O 49285,C12(NC(c3ncn(CC)c3)=O)CCCC(NC(c3ccsc3C)=O)(C1)C2 49286,c1(C(=O)NCC2(NC(COCC)=O)CC3CCC2C3)ccc2snnc2c1 49287,C12(NC(=O)COC(F)(F)F)CCC(CC1)N(C(=O)C=CC1CCOC1)C2 49288,C(=O)(CCC(=O)N1CC(N2CC(NC(C3CCC(CO)CC3)=O)CC2=O)C1)NCC 49289,S(=O)(=O)(CC(=O)NC1CCCC1CNC(C1CCN(C2CC2)CC1)=O)NCC 49290,C1(C(=O)OC)CC(n2cc(C3CC=CCC3)nn2)CN1C(C1CCCCC1O)=O 49291,c1(OC)cccc(C=CC(=O)NC(C)CC(C)NC(c2ccc(C)nc2C)=O)c1 49292,c1(C(=O)NC(c2cn(C3CC3)cn2)C(=O)NC(C=C)(C)CC)cn(C)nc1CC 49293,c1(C(=O)NCCCCNC(C2C(C(=O)NCC#C)C2)=O)cccc(C(N)=O)c1F 49294,c1(C(C)C)nc(C(N2CC(CO)(NC(C3CCC3CF)=O)C2)=O)co1 49295,C(C)(C)(CCC(=O)N1CCN(C)CC1C1CC1)NC(C(CSC)OC)=O 49296,c1(OCC(=O)NCC2(NC(CC3CCC(C#N)C3)=O)CC2)cccc([N+](=O)[O-])c1 49297,c1(C(=O)NCC2(OC)CN(C(=O)C(C)(CO)OC)C2)nc2ccccc2cc1Cl 49298,C1(C2(O)CN(C(C3(CC4CC4)CC3)=O)C2)(CN(C(=O)CC2(O)CCC2)C)CC1 49299,C1(C(N)=O)CCCN1C(=O)CC1(CNC(c2ccn(C3CC3)n2)=O)CC1 49300,c1(C(=O)NCC(CC)NC(C2CC2c2sccc2C)=O)nnn(CC2CC2)c1C 49301,N1(C(C(CC)O)=O)CCN(C(=O)C(F)(F)c2csc(Cl)n2)C2(CCC2)C1 49302,C1(C(=O)OC)C=CCCN1C(=O)CC1CC1OC.c12ccc(cc1)Cn1cc-2nn1 49303,N1(C(=O)NCCCCNC(=O)OC(C)(C)C)CC2C(CC1CO)C2 49304,c1(C(=O)NC(C(C)(C)NC(Cc2c(C)nsc2)=O)C)cc(C(F)(F)F)cc(Cl)c1 49305,C(N=c1[nH]ccn2cnnc12)c1cc(OC)c(Br)cc1 49306,C1(C(=O)OC(C)(C)C)CCN(C(=O)NC2(Cc3nc[nH]n3)CCC2)CC1 49307,C=Cc1cnn(C)c1C(N1CC2CC1CC2NC(=O)C(=O)C(C)(C)C)=O 49308,CC1(C)CCC(NC(=O)Cc2cc(O)nc(O)n2)C(CN)C1 49309,Cc1ccc2c(c1C)OCCC2NC(c1cc(F)ccc1C(F)F)=O 49310,C(CCC(O)C(=O)Nc1ccc(C)nc1)NC(C(C)=C1CC1)=O 49311,n1(CCCC)ncnc1C(=O)Nc1cc(C)sn1 49312,c12ccc3cc([nH]c3c1)c(=O)[nH]c1c2ccc(C)c1.C1(NC2CC2)CC(O)C1 49313,C1(C(=O)OC)CC(F)(F)CCN1C(c1ccccc1Br)C(=O)NCCSC 49314,C#CC1CN(C(=O)C(CC(C)C)ONC(=O)CO)CC1O 49315,N1(C(c2cc(C)oc2)=O)CCC2(NC(c3cc(CC(C)C)c[nH]3)=O)CCCC12 49316,c1(CC(C)(C)C)nocc1C(N1CCCC1CNC(=O)CSCc1cccs1)=O 49317,c1(C(N(C2CCN(C(C3C(=C)C3)=O)CC2)CCO)=O)[nH]c2ccc(Cl)cc2c1Cl 49318,C1(C(N(C)Cc2ccoc2)=O)CC(NC(c2nc[nH]n2)=O)CCO1 49319,N1(C(C2(F)C(C)C2)=O)CCC2(CCC2CNC(c2cccs2)=O)CC1 49320,CC(C)CC(=O)NCC1CCN(C(C2CNC(=O)N2)=O)C1 49321,CC(C)CCCOCC(=O)NCC1CC1C(=O)NCCCN(C)C 49322,C1(OC)CCC12CC(C(N1CCN(C(C3CCC(=O)N3C)=O)C(C)C1)=O)C2 49323,c1(C(=O)NCC2CC3(CC(NC(COC(C)(C)C)=O)C3)C2)cnc2n1CCCC2 49324,CC(C)(C(=O)NCC(C1CCN(C(C2(CC3CC3)CCC2)=O)CC1)(C)O)C(N)=O 49325,c1(CC(=O)NC(C2CN(C(c3ccc(F)cn3)=O)CCO2)C)ccc(Cl)cc1F 49326,Cn1nc(CC(=O)NC(C)(CNC(C2CC23CCC3)=O)CO)cc1C(F)(F)F 49327,c1(OC(C)C(=O)NCC(=O)NCc2nc(-c3ccccn3)no2)ccccc1Br 49328,N1(C(COCCC=C)=O)CC2CCC2(NC(c2ccc(Cl)cc2NC)=O)C1 49329,c1(C(=O)NC(CNC(c2c(C)cno2)=O)C(C)(C)C)c(Cl)ccc2ccoc12 49330,C1(C)(C(NOCc2cn(CC=C)nn2)=O)CCOC1C.c1(C(=O)NC)ccc(CO)s1 49331,c1(CC(=O)NCCCCCNC(=O)CC2(O)CC2)ccc2n[nH]cc2c1 49332,c1(C(=O)NC(CC)CNC(=O)CCCOCCOC)cnc(Cl)n1C 49333,n1(CC)nncc1C(=O)NC1C=CC(CC(=O)NCCOC(F)(F)F)C1 49334,N1(C(Cn2c(C)ncc2)=O)CC(C)(C)OCC1CNC(c1nnn(C)c1C)=O 49335,C1(CNC(C#CC2(CC)CC2)=O)CCC(C)(C)CN1C(C1CC12CCC2)=O 49336,C=CCC(C(=O)NC1CCSC12CN(C(c1ccc(Cl)o1)=O)C2)C(C)C 49337,N1(C(C(CCC)NC(N)=O)=O)CC(NC(=O)CCCCc2cnc[nH]2)C(C)(C)C1 49338,C1(c2c(C(=O)OC)cccc2)CCCN(C(=O)C(C)C(=O)OC)CC1 49339,n1(CC=C)nnnc1C(c1conc1CC)NCc1ccc(SC)o1 49340,C(=O)(C(C)(C)CCC(=O)OC)NCC(CCCC)NC(=O)C(F)(F)C(F)F 49341,CC12CCC(C(=O)NCC(O)CNC(=O)C(C)(C)n3cc(Br)cn3)(CC1)CO2 49342,C1(NC(=O)NC(CC(C)C)C)C2CN(CCn3cnnc3C)CC12 49343,N1(C(COCC(=O)NC)=O)CCC2CN(C(C3C4CCCC34)=O)C2C1 49344,C1(C(N2C(C(C)C)CNC(=O)C2)=O)CCN(C(=O)C(C)c2ccco2)CC1(C)C 49345,c1(NC(=O)NC(CCS(C)(=O)=O)C(=O)N2CCC2)ccc(Br)c2nccn12 49346,c1(SC)ccccc1C(N1CCOC(CCCNC(C2CCCN2C=O)=O)C1)=O 49347,N1(C(=O)C=Cc2nccs2)CCCC1C1CCCN1C(=O)C=Cc1ccccc1 49348,C1(CC(=O)NC(CCNC(C(C)O)=O)C)CC(F)(F)C1 49349,C1(CNC(C)=O)CC2(CCN(C(c3ccc(N)c(Cl)c3)=O)C2)CO1 49350,N1(C(CC(=O)OC(C)(C)C)=O)CCC(NC(C2CC2(F)F)=O)C12CCCC2 49351,CCCC(C)CC(=O)NC1CCC12CN(C(c1cc(C)cc(F)c1)=O)C2 49352,C(=O)(C(O)C(C)(C)C)NC1(CC(=O)N(C)CC2CCCC2)CCC1 49353,CC1CN(C(C2(C)CCC(=O)C2)=O)CC1NC(=O)CSc1cccc[n+]1[O-] 49354,C(=O)(C1=CS(=O)CCC1)NCCCN(C(C)C)C(C1CCCN1N=O)=O 49355,CCC(C)(CO)C(=O)NC(CNC(c1cncc(F)c1)=O)C(C)(C)C 49356,c1(C(N2CC(NC(c3n(CCC)ccc3)=O)C(F)C2)=O)ccc2c(c1)COC2 49357,c1(NC(=O)CC2CCN(C(=O)Cc3ccc(F)cc3Br)C2)ccc2c(n1)CCC2 49358,N1(C(c2cc(O)cc(Cl)c2)=O)CCC12CN(Cc1csc(Br)c1)C2 49359,c1(OC)ccccc1SCNC(=O)C(c1sc(Br)cc1C)N(CC(C)(C)C)C 49360,c1(C(N2CCN(CC)C(C)C2)=O)c(C)ccc2cnccc12 49361,C1(N(C(=O)Cn2ncnn2)C)CCC(NC(c2ccnn2CC(F)F)=O)C1 49362,CCCS(=O)(=O)CC(=O)NCC1CCN1C(c1ccc(Cl)nc1)=O 49363,C1(CNC(C2(C(=O)OCC)CC=CC2)=O)CN(C(C2SCCS2)=O)CC12CCC2 49364,C=C(C)c1ccccc1NC(c1cc(CNC(C2C3CC(=O)CC23)=O)no1)=O 49365,N1(C(c2c(CC)cns2)=O)CCOCC(C(N2CC(C)(N(C)CC)C2)=O)C1 49366,CN1CCCC(CCC(=O)NCC2CCN(C(C3CCC3)=O)CC2)C1 49367,c1(OC)cccc(C)c1C(N1C2CC1CN(C(=O)OC(C)(C)C)C2)=O 49368,C#Cc1ccc(C(=O)NCCC2CC(NC(c3ccc(C#N)o3)=O)C2)cc1C 49369,C(C(C)CC(=O)N(C1CC1)C1CC1)NC(CC=CCC)=O 49370,c1(C(=O)NC(CN(C)C)C(=O)NC2CCC(C)(C)C2)ccc([N+](=O)[O-])o1 49371,N1(C(c2cc(CC)nn2C)=O)CC(C(=O)NC(CO)C(N)=O)C(C2CC2)C1 49372,C1(C)(C(=O)NC(CN(C(C(CC)F)=O)CC)C)C(C)(C)C1(C)C 49373,Cc1cc(CC(N2CC(F)(CNC(=O)Cn3ncc(Cl)c3C)C2)=O)n(C)n1 49374,CCC(C(F)(F)F)OC(C1CCCCN1C(=O)NCC(F)(F)F)=O 49375,CC(C)C(C(=O)N1CCC(NC(C2CC3(CC3)C2)=O)C1)n1cncn1 49376,c1(-n2c(-c3ccc(C(CC)C)cc3)nc(CC3(C)CC3)n2)ccc(F)c(Cl)c1F 49377,c1(C(=O)NC2(C3CN(C(CC4CCCC(C)C4)=O)C3)CC2)ccc2scnc2c1 49378,c1(OC)ccc(C(=O)N(C)CC2CCCN2C(c2coc(O)n2)=O)c(O)c1F 49379,CCC(C)(C)C(C)CC(=O)NCCC(C)NC(c1ccc(OCCOC)nc1)=O 49380,C1(CNC(COCCOCC)=O)C2CN(C(=O)C(O)Cc3cccc(Cl)c3)CC12 49381,C1(C(=O)NCCc2nc(-c3ccc(C)cc3)oc2)CN(C)CC(C)O1 49382,N#Cc1ccc(C(N2CC(CO)(NC(=O)C=Cc3cscn3)C2)=O)s1 49383,C1(NC(=O)CC2CCCC(=O)N2)CC(C(=O)NCC2CCCC3(CC3)C2)=CC1O 49384,c1(C(=O)NCCCC(C)NC(=O)CC(=O)N(C)C)ccccc1NC(=O)C(C)C 49385,C1(C(=O)NC(CNC(=O)CCCC2CCCC2)C2CC2)CCCC(CC2CC2)C1 49386,c1(C(=O)NC2(n3cccn3)CC2)cc(O)nc2c1CN(C(C1(F)CC1)=O)CC2 49387,C1(NC(C=NOC)=O)CCC(O)CN(C(=O)CC(C(F)F)n2cccn2)C1 49388,C(=O)(CC(C)CCC)N(C1CC(C)(NC(C2N(C(CCC)=O)CSC2)=O)C1)CC 49389,CCC(CC(=O)NC(CNC(c1cc(-c2cccnc2)[nH]n1)=O)C(C)C)OC 49390,C1(C(=O)NC(C)CC2CN(C(c3ccsc3C)=O)C2)(OC)CCC(C)CC1 49391,CCCCC(C(=O)NO)NC(=O)NC1CCOCC1F 49392,C1(C(N(C(C)C(F)F)C)=O)CCC2CCCCN2C1 49393,c1(OC)cccc2c1N(C1CC1)C2=O.c1(CNC(=O)C(F)(F)Cl)ccc(F)cc1 49394,c1(COC)nc(NCC2CC(=O)N(C)C2=O)cc(=NCc2cccs2)[nH]1 49395,c1(OCC)ccnc(C(N2CCC(OCCCNC(=O)CCOC)CC2)=O)c1 49396,c1(C(=O)NC(Cc2ncn(C)n2)C(=O)O)ccc(CO)cc1 49397,c1(C(=O)NC23CC(NC(C(CCC)C)=O)C(OC2)C3)scc2c1OCCO2 49398,N1(C(c2cc(-c3ccco3)on2)=O)CC2(CCN(C(C3(C(F)(F)F)CC3)=O)C2)C1 49399,C1(C(=O)NCC2N(S(CCOCC)(=O)=O)CC(OC)C2)Cc2ccccc2C1 49400,C1(CC(NOC(C(C)C)CO)=O)CC(O)CN1C(=O)CC1CCOC1C 49401,N1(C(c2n(C)cc(Br)c2)=O)CC2(CCC2)CC1CNC(=O)CCC(N)=O 49402,c1(C(=O)NC2CN(CC)C2)cc(C2CC2)[nH]n1 49403,C1(C2CCCN(C(c3csc(=N)[nH]3)=O)C2)(NC(CCC(=O)NCCC)=O)CC1 49404,C(=O)(CCCCCC)N(CC(=O)NCC12COC(COC)(C1)C2)CC#C 49405,c1(C(=O)NC(CC)CN(C(=O)C(C)c2cncs2)C)ccc(F)cc1OC(F)F 49406,C(=O)(CCC(=O)c1cc(C)sc1C)NCCN(C(=O)C(=Cc1c[nH]cn1)F)CC 49407,CC(C)CC(F)(F)C(=O)N(C)CCNC(=O)C(c1ccc(Cl)c(F)c1)O 49408,O=C(CC(C(F)F)NC(=O)C=CC1CC1)NCC1(F)CCOCC1 49409,CN1CCC2C(CCN2C(C2CC2C(N2CCC2c2ccccc2)=O)=O)C1 49410,C1(C(=O)NC2(C(=O)NCC(=O)N(C)C3CC3)CCN(C)C2)CCCC1C1CC1 49411,C(=O)(N1CCC(C(=O)NCC(F)CO)O1)c1nc(=N)[nH]cc1 49412,C1(NC(c2c(CC)ncs2)=O)CN(Cc2ccn(C(C)C)n2)CCC1C 49413,C1(C)(C(=O)NC(C2CC(NC(c3cc(=O)cc[nH]3)=O)C2)C)CC(=O)N(C)C1 49414,C(=O)(N=c1[nH][nH]c2cccnc12)C1C=CC(NC(c2ccccc2O)=O)C1 49415,C(=O)(CCC(F)(F)F)NCC(CCNC(c1cc(C(C)C)on1)=O)O 49416,C(=O)(C1CCc2c(Br)cccc21)NCCN(C)C(c1ccnc2ncnn12)=O 49417,c1(C(=O)NC(C(=O)N2CCC(CCC)C2)C(C)C)cnn(C)c1C#N 49418,c1(C(N(C2CCN(C(=O)CC(C)(F)F)C2)C)=O)cn(C)ccc1=O 49419,N1(C(c2c(CCC)[nH]cc2)=O)CCC(C)(CNC(c2cn(CCC)nn2)=O)C1 49420,Cc1cc(F)c(C(c2nnnn2C2CCCCC2)NC2CC(C)C2)c(Br)c1 49421,c1(OC)ccc(CC(=O)NCC2CCCN(C(C3(CF)CC3)=O)C2)cn1 49422,C(=O)(CCS(N)(=O)=O)NCC(C)(C)OCC(=O)N(C)Cc1nccn1C 49423,C(=O)(CCCCC(C)(C)C)NCC(C)(CC)NC(CCC(=C)Br)=O 49424,CCCCC(CNC(=O)Cc1cc(Cl)cnc1Br)CCC 49425,C1(C(N2CC(C)C(CCNC(=O)CCCCCF)C2)=O)CCc2c[nH]nc2C1 49426,c1(CC)nnc(C)cc1C(=O)NC(C)(CNC(c1cc(C(F)F)[nH]n1)=O)CO 49427,Cc1cc(O)cc(O)c1C(N1C(C(=O)Nc2cc(Cl)cc(Cl)c2Cl)CC2CC12)=O 49428,Cc1nc2sccn2c1C(=O)NC1CN(C(c2cc[nH]c2)=O)CC1C 49429,C1(C(=O)NC(C)C(=O)NO)CCC(C)(C)N(C(=O)CC2CCCCCC2)C1 49430,C(=O)(CCC(=O)Nc1nccs1)NCC(C)N(C)C(c1cccc(O)c1)=O 49431,N1(C(CC(C)CF)=O)CCN(C(=O)CCC2OCCO2)C(CS(C)(=O)=O)C1 49432,c1(C(=O)NC2(C)CC(C(=O)Nc3cnc(OC)nc3)C2)nccc(C)c1F 49433,c1(Cn2c(C(=O)NCC3N(C(C=CC)=O)CCC3C)ccc2)cc(Cl)cc(Cl)c1 49434,Cn1cc(C(F)=CC(=O)NC2CC(NC(c3conc3C3CCCC3)=O)C2)cn1 49435,C(=O)(C(CC(C)C)C(C)C)NC1CCC1.N1(C(CC2(CSC)CC2)=O)CCOCC1 49436,c1(NC(CCOCC#C)=O)ccc(-c2ccc(O)nn2)cc1 49437,c1(C(=O)NCCC2N(C(Cn3ncc(C)c3)=O)CCC2)cncc2cnccc12 49438,C12(CNC(=O)C(=O)Nc3ccc(N4CCCC4)nc3)CCC(O)(CC1)C2 49439,CCCCCC(F)C(=O)N1CCC(C(=O)NCC23CCC(CO2)C3)(CC)C1 49440,C1(CC)CC(NC(=O)CC(C)(C)NC(C2CC(CF)C2)=O)CCO1 49441,C1(CNC(c2nncc(OC)c2)=O)CN(C(=O)CCC(C)C)CC(C)(C)C1 49442,C#CC1CCCN(C(=NCCOc2ccccc2)NCC(CC=C)CCSC)C1 49443,C1(C(C)C)CN(C(=O)CC2CCC(C#N)C2)CC1C(=O)NCc1ccc(F)cn1 49444,C=CC(C(=O)NCCOCCNC(=O)C(C)(C)c1cccnc1)c1ccccc1 49445,N1(C(C(C(=O)OCC)F)=O)CCN(C)C(C(=O)NCC2=CCCC2)C1 49446,c1(OC)ccc(CC(=O)N(C)CC2CN(C(=O)Cc3ccsc3)CCO2)c(F)c1 49447,c1(C(C)OCC)nc(C(N(C(C)CN(C(=O)C=C(C)I)C)C)=O)cs1 49448,C(=O)(NNc1ccc(P(C)(C)=O)cc1)c1ccc(OC)c(N)n1 49449,N1(C(C2CCCC(N(C)C)C2)=O)CC2=C(C1)CN(C(=O)CCF)C2 49450,C1(C)(C(N2CCC(N(CC#C)C(c3cnc[nH]3)=O)CC2)=O)CCCNC1=O 49451,N1(CCc2ccc(NC(=O)N(C(C)C)C)cn2)CCC2CCN(C(C)C)CC12 49452,c1(C2(C(N3CC4CCN(C(=O)C=CCO)C4C3)=O)CC2)nccc2ccccc12 49453,C(C)(CCCCNC(=O)C(C)c1cccs1)NC(C1N=C(C)SC1)=O 49454,C1(CNC(C(C)OCC)=O)CC2(CCN(C(=O)Cc3ccnc(Cl)c3)CC2)CO1 49455,c1(C(=O)NCCN(C(C(F)OC)=O)CC(C)O)ccc2cnn(C)c2c1 49456,CC1(C(=O)NCC=CCC(N2CC(CO)C3(CC3)C2)=O)CC2C=CC1C2 49457,CON(CCC(=O)N(C1CCC(=O)N(C(C)C)C1)C)C(=O)c1cccc(C)c1F 49458,c1(C(=O)NCC23OCC(NC(CNC(=O)NC)=O)(C2)C3)cc(C(F)F)ccc1Cl 49459,Cn1ccc2c(C(N3CC4CCC(NC(c5cnc(O)s5)=O)(C4)C3)=O)ncnc12 49460,N1(C(c2cnc(C(C)(C)CF)o2)=O)CCN(C(C2C=CCC2)=O)CC1 49461,C1(NC(C2CC(C)SCC2)=O)CCCC2CN(C(=O)Cc3ccn(C)n3)CC12 49462,n1(CCCC)nc(-c2ccnc(SC(C)(C)C)c2)nc1C(CC)C(C)O 49463,C(=O)(CCCCC(C)CC)NC1CC(C)N(C(=O)CC#N)C1 49464,C12CCN(CC1O)c1ncncc1NC2.c12cccc(c1)OC(=O)C2.CO.OC 49465,c1(C(C)C)nc(=NC(=O)N2CCC(C)(COC(C)(C)C)CC2)[nH][nH]1 49466,Cc1ccnc(C(=O)NCC(O)CCNC(C2CCCCCN2C)=O)c1F 49467,Nc1ncccc1C(N1CC2C(CNC(c3cc(=O)cc[nH]3)=O)C2C1)=O 49468,C(=O)(C(O)CC(C)(C)C)N1CCCC(N(C(COCc2ncc(C)o2)=O)C)C1 49469,c1(C(N(C)CC)=O)cccc(NC(c2coc(Cl)n2)c2nnnn2CCCF)c1 49470,C1(NC(C2CN(C)C(=O)C2)=O)COC2(C1)CN(C(c1cc(C3CC3)sn1)=O)C2 49471,N1(C(C(CC=C)C)=O)C2CCC1CC(C(=O)NC1CC13CCCC3)C2 49472,c1(C(=O)NCCC2(CNC(=O)C=CBr)CC2)ccnc2c1CCC2 49473,C1(C(N2CCN(C)C(C3CC3)C2)=O)CN(C(c2cc(C#N)cs2)=O)CCC1(C)C 49474,C1(C#N)(C(N2CC(O)(C(C(=O)NC(c3c(C)nns3)C)F)C2)=O)CC(F)(F)C1 49475,CN=c1nc(N2CC(=O)NC(C)C2)[nH]c(=NC(C)c2cccc3cccnc23)[nH]1 49476,N1(C(c2c(CCCC)ocn2)=O)CCCC(NC(=O)C(C)c2ccco2)CCC1 49477,CCC(CC(=O)NC(C1CN(C(=O)C=Cc2ccc(C(F)F)o2)C1)C)OC 49478,C1(CNC(c2ccco2)=O)COCC2(CCN(C(=O)CC3CC4CC4C3)CC2)O1 49479,c1(OC)cc(C(N2CC(C(=O)N(C3CC3)CC3(F)CCCC3)C2)=O)ccc1Cl 49480,Cc1cnc(Cl)c(CC(=O)NCc2cccc(CN(C)C(C3CC3F)=O)c2)c1 49481,N1(C(C2N(C)CCOC2)=O)CC2CCN(C(c3ccc(Cl)c(Cl)c3)=O)C(C2)C1 49482,C(=O)(CS(=O)(=O)C1CC1)NC1CCCC(NC(=O)COc2cccnc2)CC1 49483,N1(C(CN(S(C)(=O)=O)C)=O)CCC2C(NC(c3sc(F)cc3Cl)=O)CC12 49484,C(=O)(C(C)(F)C(=O)N(C)C)NC(C)(C)C(=O)NCCC[Si](C)(C)C 49485,c1(SC)cn(C)nc1C(N1CCCC(C(C)NC(C2(O)CCOCC2)=O)C1)=O 49486,N1(C(c2cccc(C(=O)NC)n2)=O)CCC(NC(C2(CN(C)C)CC2)=O)CC1C 49487,c1(CN2CC(C(N3CCC(c4ccccc4)C3)=O)C2)cc(F)ccc1[N+](=O)[O-] 49488,C(=O)(CCCCCN=[N+]=[N-])N1CC(N(C(C2CC(C(F)(F)F)C2)=O)CC)C1 49489,Cc1ccc2cc(C(=O)NC3CCCC34CCN(C(C3(CO)CC3)=O)C4)[nH]c2c1 49490,C1(C(=O)NCC(C2CCOC2)OC)CC(C)(NC(=O)CSC2CC2)C1 49491,CC(C)(C(=O)NCCC12CC(CO1)C2)NC(=O)CCc1nnc(C2CC2)o1 49492,N1(C(CN(CC)CC)=O)CC=CC1CN(C(=O)CN1CCC(C)C1)C 49493,Cc1ccn2ncc(C(=O)NC3CN(C(=O)CC4CC=CCC4)CC3(C)C)c2n1 49494,c1(C(N(CCCCNC(=O)CC2C=CCCC2)C2CC2)=O)n[nH]c2nccc(Cl)c12 49495,CC1CN(C(c2nnn(C)n2)=O)CC1NC(C1(F)CCOCC1)=O 49496,N1(C(C2N(C(COC)=O)CCC2O)=O)CCN(C)C(=O)C1C 49497,c1(C(=O)NCCC(CCC)N2CCOCC2)c(C(F)(F)F)ccc(Cl)c1Cl 49498,C(C(N=[N+]=[N-])C(=O)NCCC1(NC(=O)C(C)Sc2ccccc2)CC1)OCC 49499,CC1CN(C(=O)CC(C(F)(F)F)NC(=O)CC(C(Cl)Cl)N(C)C)C12CCOCC2 49500,C12(C(=O)OC)CC(C(=O)NCC3CCC(NC(=O)CCc4ccncn4)C3)(C1)C2 49501,c1(C(N(C)CC2COCCN2C(=O)Cn2ncnn2)=O)cnc2c[nH]nc2c1 49502,C1(C(=O)OCC#Cc2cccc(Cl)c2)CCOC2(CCOCC2)C1 49503,c1(CCC)cccc(C(N2CCCCC2c2cc[nH]n2)=O)c1 49504,N1(C(c2c(CC)ccs2)=O)CCN(C(C2CCN(C)CC2)=O)C(CF)C1 49505,c1(CC(N2CC(C)N(S(C)(=O)=O)CC2)=O)c[nH]c2ccc(-c3cn[nH]c3)cc12 49506,c1(C(=O)NC2C3(CC(NC(Cc4cnc(C)[nH]4)=O)C3)C2)ccc(N)c([N+](=O)[O-])c1 49507,c1(C(C)(N)C(=O)NC(C(F)(F)F)C2CCCCO2)cccc([N+](=O)[O-])c1 49508,C#Cc1ccc(F)c(C(N2CCOC(CN(C(=O)C(F)=CC3CC3)C)C2)=O)c1 49509,C1(CC)CCCCN1C(N1CCC(CN(c2ccn(CCF)n2)C)C1)=O 49510,O=C(C#CC1CCCO1)NCC(c1ccc(F)cc1)NC(c1cc(Cl)no1)=O 49511,C1(N(C(C(CC)C)=O)C)CCCCN(C(C2CC=CC2)=O)C1 49512,C12(OC)CC(C(=O)NCC(C)(C)NC(c3cccc(F)c3)=O)C(C1)C2 49513,c1(C(N2CCN(CC3(C(N)=O)CC3)CC2)=O)n[nH]c2c1CCC(F)(F)C2 49514,c1(C(=O)OCC2CCOC2)c(O)cccc1Cl.c12nc(co1)OC2C 49515,c1(C(=O)NC2C3CN(c4ncnc5c4CCC5)CC23)cc(=O)c2ccccc2o1 49516,c1(OC)ccc(C(C)NC(C2(C)CCCN(C(C3(Br)CCC3)=O)C2)=O)cc1OC 49517,C1(NC(C(CCC)OCC)=O)CCN(C(c2cc(C)n(C(C)C)c2)=O)CC1F 49518,N(C1CCOc2ccccc21)(CCC1CCOC1=O)CC.C(=O)CCc1nccs1 49519,CC1Cn2nc(C(=O)NC3CCN(C(c4occ5c4CCC5)=O)C3)cc2C(=O)N1 49520,c1(CC(C)C(=O)NCC#CCNC(C2CC3(CCCO3)C2)=O)ccc(C#N)cc1 49521,C1(C(N2CC(CNC(C=C(C)C)=O)OCC2)=O)CCN(C)S1(=O)=O 49522,c1(NC(C(C)C)C(C)NC(=O)Cc2cnccc2Cl)ncnc2c1cnn2C 49523,Cc1cc(Cl)c(Br)cc1C(=O)N(c1nc(C(C)C)c(C)s1)C1CC2CNC1C2 49524,C=CC1(C(N2CCC(CC(F)F)C2)=O)CCN(C(C2CCCSC2)=O)C1 49525,N1(C(COCCCC)=O)CC2CCC1C(CNC(=O)CCCc1cnn[nH]1)C2 49526,N1(C(c2ncn(CC)n2)=O)CC(CNC(=O)C=Cc2ccsc2)C2(CCC2)C1 49527,C1(C(=O)N(C2CC(SC)C2)C)(CC)CCCN1C(c1ccccc1O)=O 49528,n1(C(C(=O)N(C(CCNC(CSCC#C)=O)C)C)C)ccnc1C 49529,c1(OC)ccc(CCC(=O)NCC2CCC2NC(C2CC3C=CC2O3)=O)c(F)c1 49530,N1(C(C(C)=C2CCCC2)=O)CCC2C(C1)CN2C(c1cnc(OC(C)C)cn1)=O 49531,c1(CC)nc(C)c(C(=O)N(C)CC2CCCN2C(C2CCCOC2C)=O)s1 49532,N1(C(C2(C)CCCCC2)=O)CC(CO)C2(CCN(C(C3COCCO3)=O)CC2)C1 49533,C1(C(N2CC(NC(CCOCCCOC)=O)(CO)C2)=O)CN(CP(C)(C)=O)C1 49534,c1(CC)ccc(O)c(C(=O)N(C(C)CCNC(C2CCC2(C)C)=O)C)c1 49535,C1(CC)C(NC(=O)COc2cccc(C)c2)CCN1C(c1ccsn1)=O 49536,N1(C(c2ccc(C(C)=O)cc2)=O)CCN(C(=O)C(C)C(C)O)CC1CC(F)F 49537,C1(N(C(C2C(CNC(c3c(CC)non3)=O)OCC2)=O)C)CCC(O)CC1 49538,Cn1cc(C=CC(=O)NCCC(=O)NCCC2CCSC2)nn1 49539,N1(C(c2cc(C)c(O)nc2)=O)CCC=C(C(=O)N2CCCCC2C#N)C1 49540,C12(C(=O)NC3CC(N(C)C(c4ccc(NC(N)=O)cn4)=O)C3)CC=CC(C1)OC2 49541,c1(C(C)=O)ccc(C(N2CC3C(CNC(C4CC(C)(C)CO4)=O)C3C2)=O)cn1 49542,CC12CCOC(C(N3CCC(CO)C(NC(C45CCN(CC4)CC5)=O)C3)=O)(C1)C2 49543,CCCC(C(N)=O)NC(=O)CN(C(=O)C=CC(F)(F)F)C 49544,C(c1cccc(Cl)c1)=CC(=O)NC(C1CCN(C(c2cc(C)c(C)[nH]2)=O)C1)C 49545,N1(C(C=C(C)Cl)=O)C2CCC1CC(N(C)C(c1ccncc1Br)=O)C2 49546,S(=O)(=O)(c1ccc(C(N2CCC(C(C)NC(c3cc[nH]c3)=O)C2)=O)o1)NC 49547,c1(CNC(=NCCCCC)NCCc2ccccc2)ccc2nc(O)oc2c1 49548,C1(C)(CNC(C2C(CC)C2)=O)CCN(C(=O)CC2CCC(=O)NC2=O)CC1 49549,C1(CCOC)(NC(=O)CC2CC2CF)CCN(C(C2CC2C(F)(F)F)=O)CC1.C(C)C 49550,N1(C(C(C(C)C)N(C)C)=O)CC(CN(C)C(c2csc(C(F)F)c2)=O)C2(CC2)C1 49551,c1(CNC(=O)C(C2CCN(C(c3ccnn3CCF)=O)C2)F)cccc(CO)n1 49552,CC(C)C(O)CCNC(C1CC=CCN1C(C1CC2C=CC1O2)=O)=O 49553,C(C(CNC(=O)CC1CCC(=O)N1C)C(F)(F)F)NC(c1c(SC)nn(C)c1)=O 49554,Fc1cccc2nc(N3CCC(C4CC4)C3)[nH]c(=NCCc3nccs3)c12 49555,n1(CCOCC)cc(C(=O)N(C)CCNC(C2CCC(C(N)=O)C2)=O)cn1 49556,c1(OCC(N2CCC(N(C)Cc3cccnc3O)C2)=O)cc(F)cc(Cl)c1 49557,CCC(C)C(=O)NC(C1(O)CN(C(C2COCCO2)=O)C1)C 49558,c1(C(N2CC(NC(C(CCC)O)=O)C(OC)C2)=O)cnc2c(c1)CNC2=O 49559,Cc1ccc(C(=O)O)c2c1N(CCOC1CCC1)CCC2.CCCN 49560,c1(N(CC=C)C)[nH]c(=NC2CC3(CCCC3)C2)nc2c1ncn2C 49561,CC(C)CCCC(C)NC(=O)CN1CCN(C(C2C=CC=CC=C2)=O)CC1 49562,N1(C(c2c(C)ocn2)=O)CCN(C(c2ccc(F)cc2O)=O)C2CCCC2(C)C1 49563,N1(C(Cc2ccc(OC)nc2)=O)CCCC(NC(=O)C(C)COC(C)=O)CC1 49564,CC1=C(C(=O)NC(CNC(c2cc(C(F)(F)F)n[nH]2)=O)CC(C)C)CCCO1 49565,N1(C(Cn2c(C)ncc2)=O)C2CCC(C2)C1CNC(C1COC2(CCC2)C1)=O 49566,N1(C(c2c(C(=O)OC)cncc2)=O)CC(C2CCCN(C(=O)C(C)(C)C(C)O)C2)C1 49567,N1(C(c2n(CC#C)cnn2)=O)CCC2C(C(=O)N(CC(=O)NCC)C)C2C1 49568,Cn1ccc(C(N2CC(C)(NC(=O)CC3(O)CCOC3)C2)=O)c1C1CCC1 49569,C1(NC(C2CC2(F)Cl)=O)CCN(C(=O)C(C2CCCC2)C2CCCC2)CC1 49570,N1(C(C2CC(CC)C2)=O)CC2CC2(NC(=O)COCCc2cccc(OC)c2)C1 49571,C1(CC(N2CC(C)C(NC(c3ccn(CC(F)F)n3)=O)C2)=O)CCC(C)(C)CO1 49572,c1(C(N2CC(NC(C3(OC)CCOC3)=O)C2)=O)cc2c(C)c(Cl)ccc2[nH]1 49573,N1(C(CCC2CC(OC)C2)=O)CCCN(C(c2cc(C#N)ccc2C)=O)CC1C 49574,Cc1cc(N2CCCCC2)cc(-n2cc(-c3ncc(F)cc3N)nn2)c1 49575,C1(CNC(c2ncn(CC)n2)=O)(CO)CCCN(C(C2CCCC(F)C2)=O)C1 49576,c1(C(N2CC(C(=O)NC3(C4CCCO4)CC3)C2)=O)ccc(F)c(F)c1F 49577,c1(C(=O)NC(C)OC(c2c(C)nsc2N)=O)coc2c1CCCC2 49578,C1(C(=O)NC(C)CNC(=O)Cc2nc[nH]n2)CCCCN1S(N)(=O)=O 49579,CC1CCN(C(=O)C(N2CCC(C)(c3ccccc3)C2)=O)CC1C 49580,CC1=NOC(C)(C(=O)NCCC(=O)NCCS(C)(=N)=O)C1 49581,C1(CC(N2C(CNC(CSC)=O)COCC2)=O)CN2CCN1CC2 49582,Cc1ccc(NC(C2CCN(C(C(=O)NCC3(NCCN)CC3)=O)CC2)=O)cc1 49583,c1(NC(COC)(C)C)nc(N2CCCC(OC(C)(C)C)C2)nc2scnc12 49584,CC1CC(=O)NC1C(=O)NCC1CC(NC(c2cnn(C(C)(C)C)c2)=O)C1 49585,CC1CC(NC(c2cc(C(C)(C)C)on2)=O)CN(C(c2cnco2)=O)C1 49586,C12(NC(C(n3c(C)cc(C)n3)C)=O)CCOC(CNC(C3(C)CCCO3)=O)(C1)C2 49587,CCCC(C)(O)CC(=O)NC1CC(F)CN(C(=O)CCC(C)CN(C)C)C1 49588,Cc1oc(C(=O)NCCC2(O)CN(C(c3ccc(C(C)C)cn3)=O)C2)cc1CO 49589,C#Cc1ccc(CC(N2CCOC(C)(CNC(c3cnnc(O)c3)=O)C2)=O)cc1 49590,c1(C(N2CCC(NC(c3n(C)nc(C4CCC4)c3)=O)C2)=O)c(F)cc(Cl)cc1F 49591,c1(C(N2CCCC(O)(CNC(CCCOC)=O)C2)=O)cc(OC)cc([N+](=O)[O-])c1 49592,CC1CC(C)(C)CN1C(C1(c2cn(C(C)(C)C(=O)O)nn2)CC1)=O 49593,Cc1c(Br)sc(CNCC(C)(C)CN)c1Br 49594,c1(C(N2CCC(COC)(NC(c3cocn3)=O)C2)=O)ccc(F)c(CSC)c1 49595,N1(C(C2(NC(c3n(C=C)ncc3)=O)CCN(C)C2)=O)CCC2(CCC2)C(O)C1 49596,N1(C(=O)Cn2cncn2)CCC2C(C1)CN2C(C1CC(c2ccc(F)cc2)C1)=O 49597,c1(N2CCCC(NC(C)=O)C2)ncnc(N(C)CC2CCCC2(C)C)c1C 49598,C1(C(=O)NC(C2CCCN2C(C2CC2(C)C)=O)C)CCN(C(=O)OC(C)(C)C)CC1 49599,C1(N(C)C(C2CC23CCCC3)=O)CC2CC1N(C(c1ccc(N)cc1F)=O)C2 49600,C1(CNc2c(Br)cnc(C(=O)OC)n2)(OC)CC(C2CCC2)C1 49601,N1(C(c2c(SC)ccs2)=O)CCOC2(CCN(C(C3CC(C)(C)C3)=O)CC2)C1 49602,C1(NC(c2cnsn2)=O)CC12CCC(NC(c1cccc(F)c1Cl)=O)CC2 49603,Cc1cnc(C(N2C3CC2CN(C(=O)C=CC(=O)N(C)C)C3)=O)c(F)c1 49604,Cc1oc(C(C)C)cc1C(N1CCCC1C1CCN(C(=O)C=CC(F)(F)F)C1)=O 49605,CN(CCCC(=O)NCC1CN(C(c2cnc(S)nc2)=O)C(C)(C)C1)N=O 49606,c1(C(N2CCC3(C2)CC3(F)F)C(=O)NC2(C)CC2)cnc2ccc(Cl)cn12 49607,C1(COC)(CNC(C2CCCCC2O)=O)CCCN1C(=O)CC1(C)OCCO1 49608,c1(CCNC(C2(CNC(=O)COC3CCOC3)CC(=C)C2)=O)ncc(C)cn1 49609,C#CCC(C)(C)C(=O)NCCC1CCC(NC(=O)CNC(c2n[nH]c(C)n2)=O)C1 49610,N1(Cc2ccc(OCC#C)cc2)CC2CC(C1)N2C(c1cc(F)c[nH]1)=O 49611,c1(C(N2CC(O)(C(C)NC(C(CCC)CC)=O)C2)=O)ccc2c(c1)NC(=O)CN2 49612,O=C(CCCCCCCO)NCCCO.C12CC(c3ccccc3)CN1C2 49613,c1(C(=O)NC(C(C)NC(C2(F)CCCC2)=O)C)cc(Cl)cc(Br)c1N 49614,N1(C(c2cccc3nonc23)C(=O)NCCSC)CC2CCC(O)CC2C1 49615,C1(NC(C2CCC(C)C2)=O)CN(C(C2C3CCCC23)=O)CCC12CCC2 49616,n1(CC(N2CC(CC(C)NC(C(C=C=C)C)=O)C2)=O)ccc2ccccc2c1=O 49617,C(=O)(CC(C)(C)Cn1cc(CN2CC(=O)CCC2=O)nn1)N(C(C)C)CCO 49618,c1(CC)onc(C)c1C(=O)NC1CN(C(=O)CCc2ccc(OC)cc2)C1 49619,C1(NC(=O)COCc2ccccn2)COCCN(C(C2CC3(CCC3)CO2)=O)C1 49620,C=C=CC(C)C(=O)NC(c1cccnc1)C(=O)N(CCCC)C(C)C 49621,C12(C(N(C3CCN(C(c4ccc(Br)cn4)=O)CC3)CC)=O)CC(C)(C1)OC2C 49622,c1(CC)cccc(C(=O)N(C(C)CN(C)C(C2(Br)CC2)=O)C)n1 49623,C(CCCC(C)(C)C(=O)NNC(=O)C(C)CC=C)OCC#C.N1CCCC1 49624,N1(C(Cc2cnc(C)[nH]2)=O)CC2CCC(C1)C(NC(C1CCC3CC13)=O)C2 49625,CC1CC2(CC2)CN1C(=O)CCn1cc(-c2c(F)cncc2F)nn1 49626,C(=O)(C(O)CC(F)F)NC(CC)CNC(c1cc(-c2ccccc2Cl)on1)=O 49627,c1(C(=O)NCC(C(C)(C)C)NC(C=C=C(C)C)=O)cc2ccccc2cc1N 49628,c1(C(=O)NCC(COC)NC(=O)CC2CCNC2=O)cccc(OC(C)C)n1 49629,N1(C(=O)Cc2ccc3c[nH]nc3c2)CC2(C1)CN(C(C1CCNC1=O)=O)CCO2 49630,c1(-c2nc(CNC(C3C(OCC)CCC3)=O)nn2C)cn2ccnc2s1.C(=O)(NC)NCC 49631,C1(NC(C2CCC(C)O2)=O)CCCC(C(N2CCOC(C3CCC3)C2)=O)C1 49632,c1(OC)cnc(F)cc1C(=O)NC1(CNC(C2CC2Cl)=O)CC(F)(F)C1 49633,Cc1ccc2c(C(N3CC(CC(C)NC(C4(S(N)(=O)=O)CC4)=O)C3)=O)csc2c1 49634,C1(C(N(C2(CC(=O)N(CC(COC)(F)F)C)CC2)C)=O)CCCC(C)C1 49635,c1(C(=O)OCC=CC)ccc(OCCOC(=O)C(C)=CCO)nc1 49636,C1(C(N(CC)Cc2ccsc2)=O)(CC)CCCN(C(c2ncc(C)cc2F)=O)C1 49637,c1(C(=O)NCc2c(CNC(CC3(COC)CC3)=O)ocn2)ccc(F)c(SC)c1 49638,n1(CC(N2CC3C(NC(c4c(C)cns4)=O)(C3)C2)=O)nc2n(c1=O)CCCCC2 49639,C(CC(C)C(=O)N(C1CCC(CNC(c2cc(Cl)cs2)=O)CC1)C)=CC 49640,C1(C(=O)NC2C=CCN(C(C3N(CCC)CCCC3)=O)C2)CCc2nncn2C1 49641,C1(C(=O)NCc2ccc(CC)o2)CCCN(C(=O)C(C2CC2)OC)C1CC 49642,CCC(C)(CNC(=O)C(F)OC(F)(F)F)C(=O)NCC1(CN=[N+]=[N-])CC1 49643,c1(SCCNC(c2cn(C3CC(N)C3)nn2)=O)cccc(Sc2ccccn2)n1 49644,CC12CCC(C(=O)NCCC3CN(C(=O)C(C4CCCCCC4)O)C3)(CC1)CO2 49645,c1(CC)ccc(F)cc1C(N1CCCC1C1(O)CN(C(C2CC2(Cl)Cl)=O)C1)=O 49646,c1(CS(N2CCC(NS(CCC)(=O)=O)C2)(=O)=O)cc(F)ccc1Br 49647,C1(CC(=O)NCCCOCCC(=O)N2CC(c3ncc[nH]3)C2)CCCSC1 49648,N1(C(c2cc(C)nn2C)=O)CCn2nc(C(=O)NC3CCC3)cc2C1 49649,C1(C(N2CC(NC(c3csnc3Br)=O)C2)=O)CC2C=CCC(C1)C2 49650,c1(CC)c(C(=O)NC2CCCC2CNC(=O)Cc2csc(Cl)c2)csc1C 49651,N1(C(CCN(CCC)C)=O)C2CCC1C(C)C(NC(c1nc(C)oc1C)=O)C2 49652,c1(OC(C(=O)N(CC(C)NC(=O)C(C)n2ccnn2)CC)C)ccc(C)cc1 49653,c1(C(N2CC(F)(CNC(c3cc(C(F)F)no3)=O)C2)=O)nccc(F)c1Cl 49654,N1(C(=O)NCc2c(OCCOC)cccc2)CCCC(CN)CC1 49655,C(=O)(C(CN(C)C)NC(=O)Cn1ccnn1)N(C(C(C)SC)C)C 49656,N1(C(C(C)N(C(c2cnc[nH]c2=N)=O)C2CC2)=O)CCSC(C)C1C 49657,c1(CC(=O)NC(C)CC2CN(C(C3CC(C)(O)C3)=O)C2)cc(F)ccc1Br 49658,Cn1cccc1C=CC(=O)NCC1CCCC1NC(C1CCOC1(C)C)=O 49659,OC1(C2CCCC2)CCN(CC2CCn3ccnc32)CC1 49660,C1(C(=O)NCCOCCNC(c2nn(CC)nc2C)=O)C2CS(=O)(=O)CC12 49661,N1(C(C(c2ccc(F)cc2)=O)=O)CC(NC(C2CC3C=CC2CC3)=O)CC(O)C1 49662,C1(C(N(C)CC2(NC(C(C)Oc3cccc(C)c3)=O)CC2)=O)CC2(CCCC2)C1 49663,C(CCCCCNC(=O)CCc1cccnc1Br)N(C(C1C(=C)CC1)=O)C 49664,C(=O)(CCCN(C)N=O)N1CC(CNC(CCC2CC(OC)C2)=O)OCC1 49665,c1(CC)cnccc1C(=O)NC1CC(C(=O)NCC(c2ccccc2)F)C1(C)C 49666,N1(C(C23CC(NC(Cc4c(C)con4)=O)(C2)C3)=O)CCC2(CC(F)C2)C1 49667,C=CC(CCC)CC(=O)NC(C(=O)NC1CCCCCC1F)C(C)(C)C 49668,N1(C(c2cn(CC)nc2)=O)CCCC(C2(NC(c3cn(CCO)nn3)=O)CC2)C1 49669,c1(OC)cc(CN2CC(OC(C)(C)C)C2)c(OC)cc1I.C12CCCN(C1)C2=O 49670,c1(C(N2CCN(C=O)CC2)c2ccc(OC(F)F)c(F)c2)cc(Cl)c(Cl)c(Cl)c1 49671,N1(C(=O)Nc2cccc(Cn3c(C)cc(C)n3)c2)CC2CNCC2(C)C1 49672,N1(C(c2nc(C(N)=O)sc2)=O)CC2(COC(CNC(c3coc(Cl)n3)=O)C2)C1 49673,NCCCC(O)C(=O)NCC(=O)NC(C1CCC1)=O 49674,C(=O)(CC(F)(F)C(C)(F)F)N1CC(NC(C2C(C)(C)S(=O)(=O)CC2)=O)C(O)C1 49675,N1(C(c2c(CC)noc2)=O)Cc2n[nH]cc2C1C(=O)N1CC(OC(F)F)C1 49676,c1(N(C)CC2CCCC2O)nc2c(c(=NCc3ccsc3Cl)[nH]1)CSC2 49677,C(=O)(C1=NOC2COCC12)N1C(C(=O)NC(CC#C)CO)(CC=C)CCC1 49678,Cc1nc(C2CCCC2)sc1CC(=O)N(CCCNC(C1CC1CF)=O)C1CC1 49679,N1(C(CCC(CC)=O)=O)CC2(CCCC2NC(=O)C=CC2CCCN2C)C1 49680,c1(C(=O)OC)cc(C(=O)NCC2CC(SC)C2)co1 49681,CC(CCCNC(=O)C(CN(C)C)c1ccccc1)NC(=O)Cn1nccc1N 49682,C1(NC(C2(C)C=CCC2)=O)COCCN(C(=O)Cc2ccsc2Br)C1 49683,N1(C(C=CC)=O)CC(F)(n2cc(COCC(C)C)nn2)C1 49684,n1(CC=C)cc(C(=O)N(CCCN(C(=O)C(C2CCC(=O)N2)C)C)C)nn1 49685,N12CCC(CC13CCC3)NC(=O)C2=O.N1(C(c2ccccc2)C)CCC(C)C1 49686,C1(C(=O)NCC2CN(C(Cc3cc(C)on3)=O)C(C)C2)CCC2(CCOCC2)O1 49687,c1(C(N(C2CCN(C(C3CC4CCCC4C3)=O)C2)CC)=O)c(OC)cccc1F 49688,c1(CO)ccc(C2CCN(CCn3cccn3)C2)c2ccccc12 49689,C=Cc1ccc(C(N2CCN(C(C3C(F)(F)C34CC4)=O)C(CCC)C2)=O)cc1 49690,CC1(C)CC(C(=O)N2CC(NC(=O)CCC3CCC(=O)C3)C(C)(C)C2)=NO1 49691,C1(C2CC2)(OC)CN(C(C2CCN(C(=O)C(C)=C3CCCC3)C2C)=O)C1 49692,c1(C(=O)NC2(CC=C)CN(OC(C3CC=C(C)CC3)=O)C2)ccnc(OC)c1F 49693,n1(CC)ncc(C(=O)NC(C2CCN(C(=O)CNC(=O)COC)C2)C)c1C1CC1 49694,C1(NC(C(C)Oc2ccccn2)=O)(CNC(C2(C(N)=O)CC2)=O)CCOCC1 49695,C12=CC(=NCCCOCCc3nc(cs3)CN1)NC=N2.CCC(C)C1CCC1 49696,Cc1nn2cccnc2c1C(=O)NCC1COCC1NC(c1nc(O)sc1C)=O 49697,n1(CC=C)nnnc1C(c1csc(-c2ccccc2)c1)Nc1cc(C(C)C)no1 49698,c1(CNC(C2CCCN2C(=O)Cc2ccc(F)cc2Br)=O)c(F)ccc(Cl)c1Cl 49699,CC1CN(C(=O)CN2CC(=O)N(C)C2=O)CCCN1C(c1cocc1F)=O 49700,c1(OCCC(=O)NCC(C)N(C(=O)CCC2CCCCO2)C)ccc(Cl)cc1 49701,C1(C(=O)NCC2(C=C)CCOCC2)CCN(C(=O)CC2OCCO2)CC1(C)C 49702,Cc1cccc2c(C(=O)NCC3CC3NC(=O)CSc3cccc(Cl)c3)n[nH]c12 49703,N1(C(C(N2C(C)CCC2C)C)=O)CCC2(CCCN(C(=O)CCCCF)C2)C1 49704,c1(C(N2CC(NC(CSCC)=O)C(C)CC2)=O)ccc2nncn2c1 49705,N#Cc1cc(C(=O)Nc2ccc(Cl)cc2)ccn1.C12(CC=CC1)C(=O)NC2 49706,C12(C(N3C4C(NC(c5cc6c(s5)CCC6)=O)C(C4)C3)=O)CCC(O)(CC1)CC2 49707,C1(C(=O)NC(CC=C)C(=O)N(CCOC2CCC2)C2CC2)CC2CCCC2C1 49708,N1(C(c2c(C)nccn2)=O)CCC(NC(=O)COC2(C)CCC2)C12CC2 49709,CC1(C)COC1CC(N1CCC(c2ccccc2)C1)=O 49710,CN1CC2(CCN(C3CC4(C3)CN(C(C3CCS(=O)(=O)C3(C)C)=O)C4)CC2)C1 49711,C1(N(C)C(=O)OC(C)(C)C)COC2(C1)CC1(CN(C(=O)CC3(C)COC3)C1)C2 49712,N1(C(C2C(NC(C(C)c3cc[nH]n3)=O)C3CCC2C3)=O)CCc2nc[nH]c2C1 49713,Cc1cccc(CC(C(=O)NC(C2CC2(F)F)C2CC2)NC(=O)OC(C)(C)C)c1 49714,c1(C(=O)NCc2cn(CCCC)nc2C)ccc2ncc(I)n2c1 49715,c1(C(=O)OC)csc(CN2CC(CC(C)(C)CN)C2)c1Cl 49716,N(C(=NCC1CCCCC1)NCc1cc(C(F)(F)F)nn1C)C(C#C)C(C)C 49717,c1(C(=O)NCC2N(C(C3C(C)C3(F)F)=O)CCC2)cc2c(cc1Br)CCN2 49718,c1(CC)ccc(NC(=O)C(C)=CCNC(=O)CC2C=NN(C)C2=O)c(F)c1 49719,N1(C(c2cc(C3CC3)nc(O)c2)=O)CC2CC1CN2C(C1C=CC=CC=C1)=O 49720,CC1CC=C(C(=O)NC23CCC(CC2)N(C(C2CC4(CCCC4)CO2)=O)C3)CC1 49721,C(=O)(C1=C(SC)CCCC1)NCC(CNC(CCC(=C)Br)=O)OC 49722,CC1CCC(CCNC(=O)C(Cc2ccoc2)NC(C2CCC(O)C2)=O)CC1 49723,C(C)(CCC(=O)NCCCNC(c1cnc(C)[nH]1)=O)SC 49724,c1(CNCC(C)(C)OCCNC(CCCCSC)=O)ccc(C(C)(C)C)cc1C 49725,C(C(C(C)C)NC(c1ccccn1)=O)(C1CCCCC1)NC(CCCC)=O 49726,CN1CC(F)CC1C(N1CCC(C(F)C(=O)NCC2CNC(=O)C2)C1)=O 49727,Cc1cnc(CC(N2CCC2c2cn(C3CCCCC3F)nn2)=O)c(C)c1 49728,N1(C(C(C2CCN(C(c3cc(C(C)=O)on3)=O)C2)C)=O)CCc2nnnn2CC1 49729,CCC(CNC(C1(F)C(C)(C)C1(C)C)=O)N=c1[nH]nc(C(F)(F)F)s1 49730,N1(C(C2CCC(C)O2)=O)CCCC2C1CCN2C(c1cccc2c1CC(=O)N2)=O 49731,c1(CC)sc(C(=O)NCC2(C)CCN(C(=O)C(c3cccnc3)C)C2)cc1C 49732,CC1CC2(CC(C(=O)NCC3(C(=O)NC(CCF)C(N)=O)CC34CCC4)C2)C1 49733,c1(CN2CC(C(=O)Nc3ccc(CN(C)C)cc3)OCC2)cc(F)cc(F)c1 49734,C1(C(N(CC)Cc2ncc[nH]2)=O)C2CC3C(C2NC(=O)C(C)(C)CSC)C13 49735,C1(C)(CC)CC(C(=O)NCC(C2CCC2)NC(=O)CC#N)CCO1 49736,c1(C(=O)NC(CCNC(CCc2ncc(C)[nH]2)=O)c2cccs2)ncccc1CO 49737,Cc1nnn(C)c1C(N1CCC(C)(CNC(c2ccccn2)=O)C1)=O 49738,c1(C(=O)NC2CCN(C(C(C)=CC)=O)C2CC)cnn2cccc(Cl)c12 49739,C1(C(N2CC3(CN(C(CCNC(=O)CO)=O)C3)C2)=O)CCC2(CCOC2)O1 49740,C#CC1CN(C(=O)OC(C)(C)C)CCN1C(=O)NC1CCC(F)(F)CC1 49741,N1(c2c(C#N)nccn2)CCCC(C2(NC(C3CCCC(O)C3)=O)CC2)C1 49742,CC1(C(=O)N(CC(O)CO)C2CC2)CCN(C(=O)C(=O)NC2CC2)CC1 49743,CC(O)C(C(=O)N1CCN(C2CCC2)CC1)NC(=O)CC1CC2C=CC1C2 49744,CC(C)(C)C(CNC(C1CC1Cl)=O)C(=O)NCC1(c2ccon2)CC1 49745,C1(NC(c2cc(C)[nH]n2)=O)CC2C1CCN2C(c1cnn(C(C)C(C)C)c1C)=O 49746,c1(C(N2C(C)(CNC(CC(CC)OC)=O)CCC2)=O)ccc2c(c1)CNC2=O 49747,Cc1cc(C)c(C(=O)NCCC2CCC(C)(NC3(C4CCC4)CC3)C2)c(O)n1 49748,N1(C(CC=CC=C)=O)CCN(C(c2cc(C(F)(F)F)ccc2Br)=O)C(C2CC2)C1 49749,C1(CCOC)(NC(=O)CSc2nncs2)CCN(C(c2ccc(CO)cn2)=O)C1 49750,CC1CC(CO)(NC(=O)CCN(C(=O)C(c2cccn2C)=O)C2CC2)C1 49751,N1(C(c2c(C)nn(C)c2C)=O)CC(C)OC2(CCN(C(=O)CC3(C)CC3)CC2)C1 49752,Cc1ccc(C(=O)NCC2(O)CC(CNC(C3CCN(C)C3=O)=O)C2)cn1 49753,C1(NC(=O)COC2CC2)CC2CN(C(c3cc(Br)c(F)cc3F)=O)CC2C1 49754,C1(n2cc(CCCCC)nn2)CC2CCC(C1)N2C(c1ccc2c[nH]nc2c1)=O 49755,S(=O)(=O)(c1ccc(=NCCOCCCOC)[nH]c1)NC(COC)CN(C)C 49756,C1(CCC)CCCCN1C(=O)CC1(NC(=O)C=Cc2cc[nH]n2)CCCC1 49757,N1(C(c2cc(C(C)=O)oc2)=O)CCCC(CNC(=O)CP(C)(C)=O)CC1 49758,C1(n2cc(-c3c(C)nccn3)nn2)CC2CCC1(NC(=O)Cn1cc(Cl)cn1)C2 49759,N1(C(c2c(NC)ccc(Cl)c2)=O)CCC=C(C(=O)N(C)Cc2ccncc2)C1 49760,N1(C(c2cn(C3CC4(C(C)=O)CC34)nn2)=O)CCN(CC(=O)NC(C)(C)C)CC1 49761,C1(CNC(C(C)=C2CCC2)=O)CN(C)CCN1C(c1cnc(Br)c(N)n1)=O 49762,C#CCC(C(=O)NC)NC(C1(NC(=O)Cc2nccn2C)CCC1)=O 49763,C1(O)(CC(=O)N(C)CCOCCC(=O)NCCCc2ncc[nH]2)CCOC1 49764,c1(Cn2cc(C(C)N(C(=O)C(O)C(F)(F)F)C)nn2)cccc(S(C)(=O)=O)c1 49765,C1(C2CC2)(NC(c2c(C)nc[nH]2)=O)CCN(C(=O)CC2OCCOC2(C)C)C1 49766,c1(OC)cccc(CN2CCC(CNC(c3c(C4CC4)noc3C)=O)CC2)c1 49767,CC1(C)CC(F)(F)CCC1C(N1CCOC(CCNC(=O)C2=CCC2)C1)=O 49768,n1(CC)cc(C(=O)NCCCC2CN(C(=O)C(C)c3cc[nH]n3)CCO2)c(C)n1 49769,c1(OC)ccc(F)c(C(=O)NC2CCCCC2NC(c2cccnc2)=O)c1F 49770,C12CCC(CC1)NC2=O.n1(CC(=O)NC)cc(OCCOC)cn1 49771,Cc1cc(C(=O)N(C)CC2CCCN2C(C2CCCCO2)=O)ccc1N 49772,C1(CNC(c2c(C)cn(C)c2)=O)C2CCC(C2)N1C(c1ccccc1CC#N)=O 49773,C1(NC(C2(COC)C=CCN2C(=O)CCc2ccc[nH]2)=O)CCCCCC1(C)C 49774,c1(C(N(CC(C)NC(C2CCC3(CCC3)O2)=O)C)=O)csc(S(C)(=O)=O)c1 49775,CC1(C(=O)NCCNC(=O)CCc2nc(O)n[nH]2)CCc2ccccc21 49776,C1(C(N(CCC(=O)N(C)CC2(C)CCC2)CC#C)=O)CCC(C)(C)OC1 49777,c1(C(=O)NC(C2N(C(C=CSC)=O)CCC2)(C)C)c(C)nn(C)c1Cl 49778,N1(C(c2cccc(OC(C)(C)C)n2)C(=O)NCCCF)CCOC(C)(CCO)C1 49779,C1(C(C)NC(=O)C(=O)NC2CC2)CCN(C(c2cnccc2Br)=O)CC1 49780,c1(C(=O)OC)nc(=NC2CCCN(CC(c3ccccc3)=O)C2)c(F)c(Cl)[nH]1 49781,C1(CNC(CCC(C2CCC(C)CC2)=O)=O)C(C)CCCN1C(=O)CSC(F)F 49782,c1(C(N(CC(CC)NC(CC2(OCC)CC2)=O)C)=O)cnn(CC)c1 49783,N1(CCCCCCC)C2CCCC1COC2 49784,C=CC1(CC)COCCN1C(c1ncc(Br)cc1Cl)C(=O)NCC(C)C 49785,c1(CN2CC3CN(C(C4C(OC)CC4)=O)CC3C2)cc2ccccc2nc1C 49786,Cc1ccc(CC(N2CC3(NC(=O)COc4cccnc4)CCC2C3)=O)cc1F 49787,Cc1cc(C=CC(=O)NC(C(=O)NC2COCC2CO)C2CCCO2)on1 49788,N1(C(C(COC(C)C)(C)C)=O)CCCC(NC(c2cnc(O)c(F)c2)=O)C(F)C1 49789,c1(C(=O)NC(C)CCCCNC(=O)C2CC2)coc2c1COC2 49790,N1(C(CC=CCC)=O)CC2CC1CC2N(Cc1ccccc1)NC(=O)CCC 49791,N1(Cc2c(F)cc(OC)c(I)c2)CCC(C)(C)CC(C)(C)C1 49792,N1(CCOC)CCC2CN(c3ncc(-c4ccccc4)cn3)CC2C1 49793,C1(NC(C2(CSC)CCC2)=O)CCN(C(=O)CCCc2ccccc2)CC1O 49794,N1CCN(C(=O)CC2CCN(c3ncc(I)cn3)C2)C2(CCC2)C1.CNC 49795,c1(CC)cccc(F)c1C(=O)NC1CCN(C(=O)CCC(C)(C)C)C1(C)C 49796,c1(C(=O)NCC2(O)CN(C(c3c(C)cccn3)=O)C2)c(C)nc(C2CC2)nc1C 49797,C1(NC(C2CC3CC2C2CC32)=O)(CO)CCCN(C(=O)CCn2cc(Cl)cn2)C1 49798,c1(C(CCOCCC)NC(=O)C(C)O)cc(C(F)(F)F)ccc1C(F)(F)F 49799,c1(OC)cc(C=CC(=O)NC23CCCC2CN(C(c2cscn2)=O)C3)ccc1F 49800,c1(C(=O)NC(C)CCN(C)C(c2ccco2)=O)nccc(Cl)c1Cl 49801,c1(NC(C2CSCCN2Cc2cc(F)c(O)c(Br)c2)=O)ncc(Br)cc1[N+](=O)[O-] 49802,C(=O)(C(C)CC(N)=O)NCc1cc(N2CCN(C(CN(C)CC)=O)CC2)ncc1 49803,C1(C(=O)NC(C#C)CC(C)C)CN(C)CCN1C(=O)CCC(C)SC 49804,c1(C(=O)NCCCCNC(c2cncn(C)c2=O)=O)scc2c1CCCC2 49805,c1(C(N(C(CNC(c2cc(CSCC)on2)=O)C2CC2)C)=O)cc(Cl)ccc1F 49806,c1(C(=O)NCC2C(NC(C(C3CC3)N)=O)CCCC2)cnc(O)c(C)c1.CCOC 49807,C1(CNC(C(CC)(C)OC)=O)C2CCC(C2)N1C(=O)CCc1ccc(Cl)cc1 49808,c1(CCC)ccc(C(=O)NCCC(C)N(C(=O)C(N2CCNC2=O)C)C)[nH]1 49809,N1(C(C(CCCC)C)=O)CC2=C(C1)CN(C(C1CCCCC1CC)=O)C2 49810,Cc1cc(Cl)c(C(=O)NCC2CN(C(c3cncnc3)=O)CCO2)cc1N 49811,N1(C(c2ccc(CC)o2)=O)CCC(NC(=O)Cc2sc(C)nc2C)CC1C1CC1 49812,N1(C(CCC=CC(C)C)=O)CCN(CCNC(C2(C)CC=CCC2)=O)CC1 49813,C1(NC(c2c(C)ncc(C)c2)=O)CCCC12CCN(C(c1cn[nH]c1)=O)C2 49814,c1(C(=O)NC2(CCCNC(c3n(CC)nc(C)c3)=O)CC2)cccc2c1CCN2 49815,c1(C(C)NC(=O)CN(C(=O)CCC2CC2(F)F)C)nncn1C 49816,C(=O)(C(F)(F)CC)N(C(CC(=O)NC1CCN(C(CC)=O)C1)C)C 49817,C1(C(=O)NCC(C(C)C)NC(=O)CCn2cccn2)CCC2(CC2)C1 49818,c1(C(N(C)CC2(CNC(c3cccs3)=O)CC2)=O)nc(O)nc(O)c1N 49819,c1(-c2ccc(CCNC(c3cn(-c4scc(CC)n4)nc3)=O)s2)ccc(O)cc1 49820,c1(C(=O)NC2(CCOC)CCN(C(C3(O)CC3(C)C)=O)C2)ccc(=O)n(C)n1 49821,N1(C(C(C)OCC)=O)CCCC1CNC(C1CC(Oc2ccccc2)C1)=O 49822,C(CC(F)F)(C(=O)NCC(=O)NC1CCCC1)N(C(c1cncc(CC)c1)=O)C 49823,C(C(=O)N(CCCCCCNC(=O)C=C1CCC(C)C1)C)(C(C)C)OCC 49824,C1(C)(C(N(CCC)CCNC(c2ccc(Cl)o2)=O)=O)SCCCS1 49825,C1(NC(CCc2cc(C)n(C)n2)=O)CCCCC12CCCN(C(C1(O)CC1)=O)C2 49826,Cc1nn(C)c(Cl)c1CC(=O)NCC1CCN1C(C1(C)CC(F)(F)C1)=O 49827,c1(N2CC(C)C(O)C(C)C2)nc(N2C3CCC2CC(F)C3)nc2c1COC2 49828,c1(N2CCC(NC(c3c(C)cc(OC)cc3C)=O)C2)ncnc2cc(C)[nH]c12 49829,C12CN(CCN1C(c1scnc1C)=O)C(=O)C2.c1(CC)nocc1Br 49830,C#Cc1cnc(C(=O)NC(CC2CCC2)C(=O)NCC=CCl)c(C)c1 49831,C1(CCC)CN(C(c2cnc(Br)c(OC)c2)=O)CCN1C(=O)CCSC 49832,C(=O)(CC(CC1CC1)NC(C1(CC)CCOC1)=O)NCC(CC)O 49833,N1(C(c2ccn(CC(C)C)n2)=O)CC2(C1)CN(C(c1ncc(Cl)n1C)=O)CCO2 49834,c1(C(=O)NCCC(=O)N(C)Cc2ncc(CC)o2)cc(C#N)cn1C 49835,C1(OC)CN(C(c2c(Cl)cccc2Br)=O)CCC1NC(C1CNC(=O)C1)=O 49836,C1(C(N(CC(=O)OC)C2CC2)=O)CCC(n2cc(CCCNC(C)=O)nn2)C1 49837,N1(C(Cc2c(F)ccc(C)c2)=O)CC2CCN(C(c3cncc(C)n3)=O)CC12 49838,N1(CC(N2CC(O)(CNC(C3(c4cccnc4)CCCC3)=O)C2)=O)CSCC1=O 49839,N1(C(COCC)=O)CC2(CC(NC(=O)CCc3ccc(F)nc3)C2)C1 49840,N1(CC2N(CC)CCC2)CCCC(C(=O)N(C)Cc2nncn2C)CC1 49841,C(C(C(=O)NCc1ccc(CN(C)C)s1)NC(=O)C(C)O)OC(C)C 49842,C1(C(=O)NCC2C3CN(C(=O)CCN4CCOC4=O)CC23)CCc2cnnn2C1 49843,c1(NC(C2CC(NC(c3cc4ccccc4o3)=O)C2)=O)cnc2ccnn2c1 49844,CCC(CCCC(=O)NC1CCN2CCCC2C1)NC(=O)C=C(CC)CC 49845,Cc1ccnc2ccc(C(=O)NC3CCC(C)N(C(c4cnn(C)c4)=O)C3)cc12 49846,c1(C(N(C(CNC(C(C)OC)=O)C)C)=O)ccc(F)c2c1OCC2 49847,CC(C)C(O)C(C)(C)C(=O)NC1CCN(C(=O)Cc2cncnc2)CCC1CO 49848,Cc1ccc(F)c(NCC(c2nnnn2CCN2CCOCC2)NC(N)=O)c1Br 49849,c1(OC)ccc(C(=O)NCC(C2CCOC2)NC(c2cnc(N)cn2)=O)c(C)c1 49850,C(N=c1ccnc(CNC(=O)C(C)(C)C)[nH]1)c1c(N(CCN(C)C)C)cccc1 49851,C1(CNC(c2c(C)scc2)=O)CCCCN1C(=O)CC1C=NN(C)C1=O 49852,C(=O)(CCCCCC(C)(C)C)N(CCCNC(CCc1ccc(C)s1)=O)C1CC1 49853,c1(OC)ncc(F)cc1C(N1CC2CC(NC(c3ccc(C)s3)=O)C1C2)=O 49854,N1(C(c2c(C#N)cncc2)=O)CCCC(C2CCCN(C(=O)C3=CCCC3)C2)C1 49855,C(CC(C(C)C)NC(C1CCC(=O)C1)=O)NC(C(=O)NCC)=O 49856,c1(C(N(C(CC)C(=O)NCCOC(=N)O)C)=O)cccc2cc[nH]c12 49857,C(=O)(C1=CCCCCC1)NCC1(OC)CCN(C(CSCCCC)=O)C1 49858,C(=O)(CC(CC=C)NC(c1ccnc(O)c1F)=O)NC(C#C)CC1CCC1 49859,C(=O)(C(CC(C)C)C(N)=O)NC(C(C)NC(c1cc(C)nc(C)n1)=O)CO 49860,c1(NC(C)=O)cccc(NC(c2csc(C(=O)Nc3cc(CO)n[nH]3)n2)=O)c1C 49861,c1(CC(=O)NC(CC)CN(C(C2CC2F)=O)CC)ccc2scc(C)c2c1 49862,c1(C(=O)NC(CN(C(C(N2CC(C)C2)C)=O)C)C)cc2ccccn2n1 49863,c1(C(=O)NC(COC)CO)cccnc1CNC(=O)COC1CCOC1 49864,C1(NC(C(C)(C)C(F)(F)F)=O)CC(C2CCN(C(=O)COc3ccccc3)C2)C1 49865,c1(C(=O)OC)[nH]c(=NCC23CCC(CO)(CC2)CO3)sc1Cl 49866,C(C(F)(F)C(F)(F)F)NC(CCC#C)=O.C12(CCOC1)CNC(=O)CCO2 49867,c1(C(=O)NCC(CCNC(=O)CC2CC(=O)NC2=O)O)cnc2[nH]cncc1-2 49868,c1(NCC(CCCC)NC(C2CC2(C)C(C)C)=O)cnc(C#N)c(C#N)n1 49869,CCCC(CC)C(=O)NCCNC(c1cc(F)ccc1NS(C)(=O)=O)=O 49870,C1(CNC(CC(C=C)C)=O)CCN(C(c2cc(C)ccn2)=O)CC1(F)F 49871,c1(OC)ccc(C(=O)NC(C)(CNC(=O)CC(C)(C)O)C(C)C)cc1C 49872,N1(CC)CCCC1CC(=O)NCC#CCNC(=O)CCOCC(F)F 49873,c1(OC)ccccc1C(=O)NC(C)C(CO)NC(C1CCCOCC1)=O 49874,C1(OC)(OC)C(C(=O)NCC2(C)CCCN2C(C)=O)CC1(F)F 49875,c1(SC)ccccc1OC(=O)Cc1ccc(OCC2CCCC2)cn1 49876,Cc1cncc(C(=O)N(C2CCCN(CC=Cc3ccccc3)C2)C)c1Cl 49877,S(=O)(=O)(c1ccccc1C(=O)OC)N(C(COC)C)C 49878,c1(SC)ccc(N)cc1C(N1CCC(NC(=O)C=CC2CCOCC2)C(O)C1)=O 49879,Cc1nc2c(C#N)cnn2c(C)c1CCC(=O)NO 49880,C1(NC(C2CCN(CC)C2)=O)CCC12CN(C(=O)Cn1cc(C(F)(F)F)nn1)C2 49881,C1(C(N(CC(C)NC(=O)C(c2cnn(C)c2)C)CC)=O)CC(=O)N(CC)C1 49882,C(CC(C)C)(C(=O)NCC(=O)NCC1CC1NC(c1cscn1)=O)NC(C)=O 49883,CCCC(CCC)CC(=O)NC1CC2(C1)CC2Nc1ncc(C)cn1 49884,c1(C(=O)NC(CC=C)CNC(=O)Cc2ccsc2C)cc2c(O)ncnc2cn1 49885,c1(N(C2CC2c2ccc(-c3nn[nH]n3)cc2)C(C)=O)nc(C=NO)c(C)o1 49886,C1(Nc2c(C(=O)OC)c(Cl)ncn2)CC1C1CCCN(C(=O)C2=NOCC2)C1 49887,c1(N2CC(C)SC(C)C2)nc(=N)[nH]c(=NCc2cn3ccccc3n2)[nH]1 49888,CC1(C)CCN(C(c2cc(C3CC3)no2)=O)C1CC(=O)NC1CC1C1CCC1 49889,CCCCC(O)C(=O)NC(CNC(=O)CC1OCCCO1)C(C)C 49890,Cc1cc(C(=O)N(C(C)CCNC(c2cc(Cl)c(Cl)n2C)=O)C)c2nccn2c1 49891,C1(NC(C(C(C)O)N(C)C)=O)CCN(C(=O)CC2CC(C(C)(C)C)C2)CC1O 49892,c1(OC)cc(Cl)ccc1C(=O)NC1CCCC1CNC(C1CC2CCC1CC2)=O 49893,CC1(CNC(=O)C(F)=CC2CC2)CC(NC(c2cn(C3COC3)nn2)=O)C1 49894,c1(OC)c(F)ccc(-c2nccn2CCc2ccc(F)c(-c3cn[nH]c3)c2)c1F 49895,c1(C(N2CCCC(C)C2)C(=O)Nc2c(OC)cccc2)cc(Cl)cc(Br)c1F 49896,C(=O)(C1=CCc2ccccc21)N1C(CNC(C2CCCCC2O)=O)CC2(CC2)C1 49897,CCC(C)(C(=O)NC(C)C(CO)NC(C1CC(F)(F)CS1)=O)C(N)=O 49898,c1(C(=O)NCCn2cc(C(=O)NCC(=O)NCC(C)C)nn2)ncccc1F 49899,C(=O)(C(O)CC(C)C)N1C(C=CC(N2CCC(CCC)C2)=O)CCC1 49900,C1(C(N2CCC(NC(=O)N(C)C)C2)C(=O)Nc2nc(C)sc2)CC12CCOC2 49901,c1(OCC)ccc2c(C(=O)N(CC(C)C)CC(C)O)c[nH]c2c1.C(C)(COC)S 49902,C(CC(=O)NOCC1CC2C=CC1C2)C1CCN(C(c2c(C(=O)OC)c[nH]n2)=O)C1 49903,N1(C(c2cc(C)no2)=O)CC2(CCCC2)C1C(=O)NCC1=NOC(C)C1 49904,C1(C(=O)NC2CC(=C)C2)CC(C(F)(F)F)CN1C(C1CCC(O)CC1)=O 49905,N1(C(c2n[nH]c(CC)c2Cl)=O)CCC2(CCC2CNC(=O)C(C)C(C)C)CC1 49906,c1(CCC)sc(C(=O)NCC2CC2CNC(=O)C(C)(C)O)cc1CC 49907,c1(C2(C(N3CCC(C(=O)O)C3)=O)CCC2)ccc(C2=COCC2)cc1 49908,c1(OCC)cccc(C(=O)NC2C3CC2N(C(=O)CC(C)C2CCCO2)C3)c1 49909,c1(C(=O)NC(C2(O)CCN(C(c3[nH]cc(C)c3)=O)C2)C)ccc2ncn(C)c2n1 49910,N(C(=NCC1CCCSCC1)NC1CCN(CC(F)(F)F)CC1)C(C)C 49911,CON(CCC(=O)N1CCCC(CC2CC2)C1)C(=O)C=C1CCOC1 49912,C(=O)(CCS(C)=O)NCCCOC.C1(=O)CC(c2ccccc2)O1 49913,CCCC(CCCNC(C1(C)CCN(C)C1=O)=O)NC(c1c[nH]nc1OC)=O 49914,N1(C(c2cc(C)oc2C)=O)CC(NC(c2c(Br)noc2C)=O)CC(C)C1 49915,N1(C(C(CCC)CC)=O)CC2(CCCN(C(C3COC(=O)C3)=O)C2)C1 49916,Cc1oc(C(N2CCCC(C3(NC(C4CC4(F)F)=O)CC3)C2)=O)cc1S(C)(=O)=O 49917,c1(C(=O)NCCCCC(C)NC(c2cnc(C3CC3)o2)=O)cccc2c1CCN2 49918,C(=O)(C(C)C(C)(F)F)N(CC(=O)NCCOC)C 49919,CC(C)C(C(=O)N1CCC(C)(C)CC1C(N1CCCC1CF)=O)C(C)C 49920,c1(CC)ccc(C(=O)N(C)CC2CC(F)CN2C(=O)COC2CCOC2)cn1 49921,c1(C(=O)NC2(CC=C)CN(C(=O)CC(C)C(F)F)C2)c[nH]c2cc(OC)ccc12 49922,C1(NC(C(CC)n2cccn2)=O)CCCN(C(=O)C=CCOCC(F)(F)F)C1 49923,CC1(C(=O)NCC2CC3CCC2N3C(C2(CO)CCC2)=O)CCCNS1(=O)=O 49924,C1(NC(c2cc(Cl)cnn2)=O)CCN(C(c2ccc(Cl)cn2)=O)CC1O 49925,N1(Cc2cnc(-c3cccs3)o2)CCC2CC2C1 49926,C1(C)(CNC(c2c(CC)c[nH]n2)=O)COCCN(C(C2CC2CC)=O)C1 49927,C1(OC)CC(C(N2CCC2CF)=O)N(C(=O)Cc2ccoc2C)C1 49928,Cc1cccnc1CC(=O)NC1CC(C)N(C(=O)CN2CCOCC2)C1 49929,N1(C(CN(C(COCC(N)=O)=O)C2CC2)=O)CCOC2CC12 49930,C1(CC)C(NC(=O)COc2cccc(F)c2)CCN1C(=O)C(C)SC 49931,c1(C(N2CC(CN(C(C3N(C(C)C)CCC3)=O)C)C2)=O)nccn2ccnc12 49932,C(=O)(C1=NOC(CNC(=O)CC2NC(=O)NC2=O)C1)NCC(C)NC(=O)OC 49933,c1(C(N2CC(CCn3cc(CC4CCOC4=O)nn3)C2)=O)ccnc2cc[nH]c12 49934,c1(C(N(CC(C)NC(C2CCCN2Cc2nnn(C)n2)=O)C)=O)ccc(Cl)cc1 49935,Cc1cc(C(=O)NC2CC(F)(F)CC2NC(=O)C2=CCOCC2)cc(Cl)c1 49936,N1(C(=O)C=Cc2ccco2)CCN(C2CCOC2)C(=O)C1 49937,c1(C(N2CCN(C(=O)OCC)CC2)=O)cc(OC)nc2cc(Br)ccc12 49938,N1(C(C(CC)=CCCC)=O)CCC2CN(C(c3sc(C)cc3Cl)=O)CCC12 49939,CCC(CCCC(=O)NCCCN1CCCCC1)NC(c1cc(C)c(F)cn1)=O 49940,N1(CCC2N(C)CCC2)CC(=O)N(CC2(n3cc(Br)cn3)CC2)C1=O 49941,c1(C(N2CC(O)(CNC(CN(C3CCSC3)C)=O)C2)=O)ccc(Br)cc1O 49942,Fc1cccc(CN=C(NCC2CCN2C2CCOCC2)NC2CC2)c1F 49943,c1(C(N2CCC3CCN(C(CC(C)(C)O)=O)CC32)=O)c[nH]c2ccccc2c1=O 49944,Cc1ccc(CCC(=O)NC(C)CCNC(C2CCCC(C)C2)=O)cc1 49945,c1(CC)nc(=NCC(C2CC2)N(C(=O)COC2CCOC2)C)s[nH]1 49946,C1(C(=O)NC2(C)CN(C(c3cnn(CC(F)(F)F)c3)=O)C2)CC2(CCCC2)CO1 49947,c1(OCC=C)ccc(Cl)nc1C(=O)NC1CCC1NC(=O)C(C)c1ccco1 49948,c1(CS(N2CCC(N3CCCC(c4onc(C)n4)C3)C2=O)(=O)=O)cc(F)ncc1Br 49949,N1(C(C2C3(NC(=O)OC(C)(C)C)CCC2C3)=O)CCSC(C)(C)C1CC1CC1 49950,C1(NC(C2CN(C(C3CC(CF)C3)=O)CC23CC3)=O)CCOC12CCC2 49951,C(C1CN(C(=O)CC(C)C(=O)OCC)CC1C(N1CCC2CCC12)=O)=CC 49952,N1(C(C2N(C(C(C)C)=O)CCCC2)=O)CCC(NC(c2cnc(S)[nH]2)=O)C(F)C1 49953,C(CCNC(C1CCCCC1CNC(C1(C2(C)CC2)CC1)=O)=O)(C(C)C)OC 49954,N1(C(C2CC(C#N)(O)C2)=O)CCC2(CCN(C(C34CCC(C3)C4)=O)CC2)C1 49955,CCCS(=O)(=O)C(C)C(=O)NC1CN(C(=O)CCn2cc(C)cn2)C(C)(C)C1 49956,CC1CN(C2CCCCC2NCCC2CC2(Cl)Cl)CCO1 49957,C1(C(=O)NCC2(C)N(C(c3ncc(N(C)C)nc3)=O)CCC2)C2CCCCCC12 49958,C12(NC(C(C3CCCOC3)OC)=O)CC(NC(c3ccn(C)c3C)=O)(C1)OC2C 49959,Cc1ccc(C(=O)NCC(C)(C2CC2)NC(=O)COCP(C)(C)=O)c(C)c1 49960,c1(C(C(=O)NCCCC(=O)OC)N(CC(C)SC)C)cc(OC)cc(O)c1 49961,c1(NCCCC(=O)N(C)C)cc(Br)ccc1S(=O)(=O)NCC1CCOC(CO)C1 49962,C1(C(N(CC#CCC)C(C)(C)C)=O)CCN(C(C2C(C)CC2C)=O)C1 49963,C(CCCC(=O)N1CC(O)(CCNC(c2cccc(O)n2)=O)C1)OCCC=C 49964,c1(C(=O)NC(C2CCCN(C(c3n[nH]c(C)c3O)=O)C2)C)cc(Cl)nnc1O 49965,N1(C(CSCCCC)=O)CCC12CN(C(=O)CCC(C)(C)F)C2 49966,C1(NC(c2c(F)cc(CC)c(F)c2)=O)COC2(C1)CN(C(=O)C(C)(C)O)C2 49967,C(CCCCC(=O)NC1CCC1O)N(C(=O)Cc1cncnc1)C 49968,N1(C(CN(c2ccncc2)C)=O)CCCCCC1CNC(c1ccccc1F)=O 49969,CC1=C(C(=O)NC2COC3(C2)CN(C(=O)CCc2scnc2C)C3)CCS1(=O)=O 49970,c1(C(=O)NCC(CC)NC(C2CCC(C)(C)O2)=O)cc(C)cc2c1NCCC2 49971,CC1CC(NC(c2c[nH]c(C(N)=O)c2)=O)CCN1C(=O)CC1(C)CC1 49972,C(=O)(CCCCCc1cn(C(C)CO)nn1)OCCC 49973,CC(C(=O)N=c1ccn(CF)[nH]1)C1CCCN(C(c2ccc3occc3c2)=O)C1 49974,c1(N(C)CC2CN(C(C(n3cc(Cl)cn3)C)=O)C2)nccc(CC#N)n1 49975,CCCCCC(O)C(=O)N1CCCC(CCNC(C2(OC)CCSCC2)=O)C1 49976,C(C(CCOC)NC(C1CCCC1)=O)NC(COCCC)=O 49977,N1(C(CC2CC(C(=O)O)C2)=O)CCCC1C(N1CCC(N2CCCCC2)C1)=O 49978,C#Cc1ccc(C(N2CCC(NC(C3(F)CCOC3)=O)C(O)C2)=O)c(F)c1 49979,C#CC1CCC(C(N2CCC(CCNC(C3CCC(C4CC4)C3)=O)CC2)=O)CC1 49980,CCCCC(C)CCC(=O)N1CCC(CNC(c2coc(Br)n2)=O)C12CC2 49981,c1(C(N2CC(c3ncc(C(=O)OCC)o3)C2)=O)cccc(CC(F)(F)F)c1 49982,n1(CC)nnc(C(=O)NCCC2(C)CCN(C(C3CCS(=O)(=O)N3)=O)C2)c1C 49983,C1(NC(CSc2n(C)ccn2)=O)CC2CCC1N2C(=O)C(O)C1CC1 49984,n1(CC(=O)NC2(CC(=O)NCC(C3CCC3)OC)CCCC2)ncccc1=O 49985,CON1CCC(C(=O)N(C2CCC(NC(c3cccs3)=O)CC2)C)CC1 49986,C(=O)(C1=C(F)CN(C(c2ccc(C#N)cc2)=O)CC1)NC1C2C3CCC(C3)C12 49987,Cn1cnc2ncnc(N(C3CCCCNC3)C(c3ccc([N+](=O)[O-])c(Cl)c3)=O)c12 49988,C(=O)(CCCS(C)(=O)=O)N(C1CCC12CN(C(=O)CC(C)(C)C(F)F)C2)C 49989,c1(C(=O)NC2CC2NC(C23CCCC2(C(=O)NC2CC2)C3)=O)ccn2nnnc2c1 49990,c1(C(C(=O)NC2(CC=C)CC2)NC(=O)CC2(OC)CC2)ccccc1 49991,CC1CCC(CNC(=O)CCC(F)(F)F)CN1C(=O)CC1CCCNC1=O 49992,C1(C(=O)NCC(C)NC(C2CC2C(F)(F)F)=O)CCn2nnnc2C1 49993,c1(CC(=O)NC(C2CN(C(c3ccccn3)=O)C2)C)ccc2c(c1)COCC2 49994,Cc1ccc(C(=O)NC2CC(C)N(C(=O)CCc3ccon3)C2)c(=O)n1C 49995,C1(C(c2n(CCC)nnn2)NCCc2ccncc2)CC2CCC1O2 49996,N1(CC)CCC1C(=O)NC(CNC(C1(COC2CC2)CC1)=O)C1CC1 49997,N1(C(CC(c2ccc(C)cc2)C)=O)CC(CNC(=O)C2=CCOCC2)C(C)(C)C1 49998,CC1(C)CC(NC(c2occc2C2CC2)=O)CN1C(=O)CCc1ccc(N)cn1 49999,Brc1cc(-n2cccn2)ccc1-c1noc(-c2cccc(Oc3cccs3)n2)n1 50000,c1(OC)ccc(CC(N2CCNC(C(=O)Nc3c(C)ccnc3Br)C2)=O)cc1Cl 50001,N1(C(c2c(CC)non2)=O)CCCC(C2CCN(c3ncnc4n[nH]cc34)C2)C1 50002,C1(C(=O)NC(C2CC3(CCC3)C2)C)CN(C(C2(C)CCOC2)=O)CCO1 50003,C1(C(CNC(C2(C)CC2)=O)F)CCN(C(=O)CCc2ccncn2)CC1 50004,c1(C(N(C)CCOCCNC(c2cc3n(n2)CCO3)=O)=O)cn2c(n1)CCCC2 50005,N(C(=NCCC1CC1)NCC1CCC(C)CO1)C(C)C 50006,N1(C(c2c(CC)occ2)=O)CCCC(C2CN(C(=O)C(C)OCCC(C)C)C2)C1 50007,CCCC(O)CC(=O)N(CCCN(C)C(c1occc1-c1ccc(F)cc1)=O)C 50008,N1(C(c2c(C)n(CCO)cc2)=O)CCN(C(=O)CCc2cncs2)CC(CO)C1 50009,N1(C(CCc2cncc(C)c2)=O)CCN(C(=O)Cc2ccc(C)nc2)CC(O)C1 50010,C1(CNC(C=Cc2ccc(C)o2)=O)CN(C(c2c(Cl)cnn2C(C)C)=O)CCN1C 50011,N1(Cc2cccc(OC(F)F)n2)CC2CC3CCCN3C2C1 50012,C12(NC(=O)Cc3cc[nH]n3)CCCC1CN(C(c1c(F)cncc1Cl)=O)C2 50013,Cc1cn2ccnc(C(=O)NC(C3CCN(C(=O)Cc4cc[nH]n4)CC3)C)c2n1 50014,c1(CCC(=O)OC)ccc(CC2CCC2(OC)OCC)cc1.N12CC(C1)OC2=O 50015,C1(CC(N)=O)CC(O)CN1C(=O)NCC1(c2ccn(C(F)(F)F)n2)CC1 50016,C1(CNC(CC2C(C)(C)C2)=O)CCC(F)(F)C1O 50017,C1(n2c(C3c4cc3nn4C)nnn2)CCC(F)(F)CC1.CCCCC(C)CNC 50018,c1(NC(C2(F)CN(C(C3CC(O)C3)=O)C2)=O)c(Br)cccc1[N+](=O)[O-] 50019,c1(OCC=C)ccc(CC(N)=O)cc1.C(CNC(=O)COC)(C(C)C)NC(CS)=O.CCl.N 50020,Cc1nsc(C(=O)N(CCCN(C(=O)C(C)Cn2ccnc2)C)C)c1N 50021,CC(C)(C#N)CCCC(=O)NOCC(=O)N(CCF)C1CC1 50022,c1(CC)cnccc1C(=O)NCC1CCN(C(C2CS(=O)(=O)C2)=O)C1 50023,CC(C(=O)NCCCCNC(=O)C=Cc1c(Cl)cccc1Cl)C(F)(F)C(F)F 50024,C(C(C)(C)SC)(c1nnnn1CCCC(=O)OC)NCC.C12CC(C1)OC2 50025,C1(NC(c2cccc(OC)c2)=O)CCN(C(=O)C(C)S(N)(=O)=O)CCC1(F)F 50026,c1(C2CN(C(CCN(CC(C(C)C)C)C3CC3)=O)C2)ccc(Br)cn1 50027,C(C(O)C(=O)NCC1(NC(=O)C(=O)NCC2CC2)CCOC1)OC 50028,Cc1nn(CC(=O)N(CC(C)NC(c2n[nH]cc2C(F)(F)F)=O)C)cc1Cl 50029,C12(C(N(C3CCN(C(C(C(C)C)F)=O)C3)C)=O)C3CC(CC13)C2(F)F 50030,c1(CN=C(NC(c2ccc(OC)cc2)C)NC(C)C2CC2)cn(C)c(=O)nc1O 50031,CC1(C)OCC(CCN=C(NCC2CCCO2)NC2CC2)CO1 50032,C(C(C(=O)N(C)CCF)C(C)(C)C)NC(C(C)SCCN(C)CC)=O 50033,C(=O)(CCCS(N)(=O)=O)N1CC(N(C(=O)C(c2ccccc2)O)C)C(O)C1 50034,C1(c2nnc(N(CC)CC)n2CC(n2cc(F)ccc2=O)C)CC2C(C1)C2(F)F 50035,N1(C(c2c(OC)cccn2)=O)CC2(NC(=O)Cc3ccc(F)cn3)CCC1CC2 50036,CCCC(C)(CCC)C(=O)NC(C)C(C)NC(=O)C=Cc1ccccc1 50037,N1(C(C=C(C)Cl)=O)CC2CCC1(CNC(=O)C(c1ccc(F)c(F)c1)O)CC2 50038,c1(CCC(=O)O)ccccc1Cl.C#CCOCCOCCOCCC1CC1 50039,C1(CC(N2CCC(OC)(CNC(c3ncn(C)n3)=O)C2)=O)CCCC2(CCC2)O1 50040,c1(OC)noc(C)c1C(=O)NC1COCCC1NC(C1CC12CCC2)=O 50041,CCC(C(=O)NC1COCC1CNC(=O)CNC(c1ccoc1)=O)OC 50042,C1(C(N(CCCNC(C2(C)CCN(C)C2=O)=O)CC)=O)COCCN1C=O 50043,C(C(CC(C)C)C(=O)NCCC(=O)N1CCCC1)NC(CC1(C(=O)OC)CC1)=O 50044,S(=O)(=O)(c1ccnc(C(F)(F)F)c1)N1CCCC(NS(CCC)(=O)=O)C1 50045,C1(C(N(CCCC)CCOC)=O)N(C(=O)C(C)C(=O)OC)CCCC1(C)C 50046,CC(CC(=O)NCc1cc(C(=O)NCCOC2(C)CCC2)cs1)CC(C)(C)C 50047,CC(C)CCC(C(=O)NCC(CO)C(C)C)NC(=O)CCN(C)CCO 50048,c1(C(=O)NC(CNC(c2c(C)ccnn2)=O)C)cn2cccc(F)c2n1 50049,CCCC(CC(C)C)C(=O)NCC(C)(C(C)C)NC(C1CCC=CCC1)=O 50050,C(=O)(C(C)(C)Cc1ccccc1)N(CCN(c1nnc(C)s1)C)C 50051,c1(C2(NC(N(CC(C)(C)OC)C)=O)CCCC2)ccc(Br)cc1 50052,C(=O)(C(C)CC(F)F)N1C(C(CC)NC(c2cc(OC)ccn2)=O)CCC1 50053,C(c1ccc(Br)cc1)=CC(=O)COCC(=O)NCCOCCOCCOC 50054,C#CCCC(C(=O)NCC(F)(F)C(N)=O)NC(c1cnc(O)cc1C)=O 50055,c1(OC)cccnc1C(=O)N(C1CCN(C(C2CCOC2C2CC2)=O)CC1)C 50056,c1(CNC(c2cccc(CO)c2)c2nnnn2CC(F)F)c(Cl)cnc(F)c1F 50057,C1(C(=O)NCCOCC(C)(C)O)CC2(CC2)CN1C(=O)C(F)OC(F)(F)F 50058,N1(C(CN(C(=O)CC(O)CN(C)C)CCC)=O)CCC(C)(C)C1C 50059,N1(C(C2C(C)C2)=O)CC2(C1)CN(C(C1CCC(=O)N(C)C1)=O)CC2CO 50060,Cc1cnncc1C(=O)NCC(C1CCC1)NC(=O)C(C)Cc1cccc(Cl)c1 50061,C1(OC)CN(C(=O)C(C)(F)F)CC1NC(=O)C(C(C)C)c1cc(C)no1 50062,C(=O)(C(C)C(C)NC(=O)CCN1CCCC1=O)N(C)CC1C(C)OCC1 50063,n1(CC)nnnc1C(CCC)(C1CC1)NCc1cnc(C(C)C)s1 50064,c1(C(=O)NCCN2CCN(C(CC(C(=C)C)OCC)=O)CC2)ccc2n[nH]cc2n1 50065,CCC(C)C(O)C(C)C(=O)NC1(CC(N2CCC2C2CCC2)=O)CCCC1 50066,C1(CCNC(C2CN(C(N)=O)C2)=O)CN(C(c2nnsc2C(F)F)=O)CCO1 50067,N1(C(=O)C(c2cccc(Cl)c2)(F)F)CCCC(NC(C2CC(O)C2)=O)CC1 50068,c1(CC(=O)NCCCN(C)C(C2(c3nc[nH]n3)CC2)=O)cnsc1 50069,CC1CC(NC(=O)C(C)(C)CC2CC2)CN(C(=O)Cc2cncn2C2CC2)C1 50070,C1(NC(C(c2cnn(C)c2)OC)=O)CC12CC(NC(=O)CCCC1CCCC1)C2 50071,CC1(CNC(=O)Cc2ccc(Cl)s2)COCCN(C(=O)CN(C)C2CC2)C1 50072,C=CCC(C)(C)C(=O)NCC1(C)CCN(C(C2CCC(C(=O)N(C)C)CC2)=O)C1 50073,Cc1ccc2c(c1)C(C(=O)N1CCCC(CCNC(=O)CC(C)C)CC1)OCC2 50074,C1(NC(CCOCC)=O)COC2(CCN(C(c3ncsc3NCC)=O)C2)C1 50075,C1(N(C(C(CCCC)N(C)C)=O)C)CC2CCC(C1)N2C(c1ocnc1C)=O 50076,c1(C(=O)NCC2CC2NC(C2CCC2(F)F)=O)cncc(N2CCCC2=O)c1 50077,Cc1c(C(=O)NC(CNC(C2CCS(=O)CC2)=O)C2CCC2)c[nH]c2nccc1-2 50078,N1(C(C2CN(C)C(=O)N2)=O)CCN(C(=O)CCCC2CCOCC2)CC(O)C1 50079,N1(Cc2cn(CC(C)NC(c3c(Cl)nsc3Cl)=O)nn2)CCN(C)C(=O)C1 50080,[N-]=[N+]=NCCCCC(=O)NC1COCC1C(N1CC(NC(N)=O)C1)=O 50081,C1(OC)CCC2(C(=O)NC3CN(C(c4sncc4C)=O)CC3C)CC12 50082,C1(NC(Cc2n(CC)cnc2)=O)CCCC(N)CC1 50083,N1(C(C(C)O)=O)CC(NC(c2c[nH]cc2C2CC2)=O)Cc2ccccc21 50084,c1(OCCOC)cc(C)cc(C(=O)N(C2CCCCCC2C)CC2CC2)c1O 50085,C(CCC(C)(F)F)N(C)C(c1sccc1CNC(=O)CC1CCCOCC1)=O 50086,N1(C(C(CC)n2cccn2)=O)CC(NC(=O)CN(C)S(N)(=O)=O)C2CCCC12 50087,N1(C(CC(C)(C)O)=O)CCC2(CCN(c3nccc(N4CCCCC4)n3)C2)C1 50088,c1(OC)ccc2[nH]c(C(=O)NCCN(C(=O)C(C)CCCC(C)C)CC)cc2n1 50089,c1(C(N2C(C)C(NC(=O)CCCC(F)F)CCC2)=O)cnc([N+](=O)[O-])n1C 50090,CC1CN(C(=O)CO)CC(C)N(C(c2cc(Cl)cc(Br)c2F)=O)C1 50091,C=CCC(C)C(=O)NC1(C)CC(C(N2CCC(C)(F)C2)=O)C1 50092,C1(C(N2CC(NC(c3occc3F)=O)C(C(F)F)C2)=O)CC2(CCCO2)C1 50093,Cc1cc2ccccc2n1CC(=O)NC1(C)CCN(C(C2(C)CCN(C)C2)=O)C1 50094,Nc1cc(C(=O)NCC2CCCN2C(c2cncc(N=[N+]=[N-])c2)=O)cc(F)c1O 50095,S(=O)(=O)(c1cccc(=NCc2cnc(NC)nc2)[nH]1)NC(C(CC)(C)C)C.C=O 50096,N1(C(CSC)=O)CCc2nc(CNC(C3(C)CC3(F)Cl)=O)sc2C1 50097,CC1CCN(C(c2ccc(SC(C)(C)C)nc2)=O)CCN1C(=O)C#CC1CC1 50098,c1(OC)c(C(N2CC(OC)C(NC(c3c(C)cccc3Br)=O)C2)=O)cccc1F 50099,S(=O)(=O)(c1ccccc1Cl)NCC(=O)N(C1CC(NC(c2occ(C)c2)=O)C1)C 50100,c1(NCCC(C)F)[nH]c(=NC2CSCCC2O)nc2c1ncn2C 50101,N1(C(Cc2cncc(C(C)=O)c2)=O)CCC2C(NC(=O)C=C3CCC(C)CC3)CC12 50102,C1(C(N(C(CC(=O)NCC(C(C)O)O)C)C)=O)C(C#N)C1(C)C 50103,c1cnn(C)c1Cl.C12(C)CC(C1)OC2=O.CC(C)(C)NC(C1CC1C(=O)NCC)=O 50104,C1(C(N(CCCN(C(C(CC)NC(C)=O)=O)C)C)=O)CC(F)CN1C 50105,C1(C(=O)NC(C2CCCC2O)C)CCCC1CNC(c1cc[nH]n1)=O 50106,c1(C(N2C(CNC(=O)Cc3ccc(F)cc3F)CCC2)=O)ncnc2[nH]cnc12 50107,c1(CC)ccsc1C(=O)N(C)CC1CCN(C(C2CC3CC3C2)=O)C1 50108,Cc1nc2ccnn2cc1C(N1CC(O)(CNC(C2CC2(C)Br)=O)C1)=O 50109,N1(C(COC(CC)CC)=O)CCC(F)(C(=O)Nc2cc(CC)cc(O)c2)CC1 50110,C1(CN(CCNC(c2ccoc2)=O)Cc2cnn(CCF)c2)CC12CC2(F)F 50111,CCCC(C)C(=O)N1CCC(CC(=O)NOCC(O)CO)CC1 50112,N1(C(C2C(C(C)(F)F)C2)=O)CCC2(CC(C(N3CC(CO)C4(CCC4)C3)=O)C2)C1 50113,C1(C#N)(CNC(CC2(C)N(C(Cc3nc(C)[nH]n3)=O)CC2)=O)CCCC1 50114,CC1CCCCN1C(C1CC(NC(C2C=CCS2)=O)C1)=O 50115,C1(NC(CCC(CC)NC(=O)CCCn2ccnc2)=O)CCC(=O)N(C)C1=O 50116,c1(C(N2C(CNC(CC(CC)C)=O)C=CC2)=O)cc2occ(C(=O)OC)c2[nH]1 50117,C(C(CC)CCO)NC(CCN(CC#C)C(c1cnc(Cl)n1C)=O)=O 50118,N1(C(CCCC#CC)=O)CC2(C1)CN(C(c1cc(C)c(Cl)s1)=O)CC2CO 50119,Cc1cc(C(=O)NC(c2cn(-c3ccccc3CO)nn2)C)cc(C)c1 50120,C1(c2nnnn2CCN2CCOCC2)(NCc2ncc(C)s2)CC(C)SC(C)C1 50121,C1(NC(c2ccc(N)cn2)=O)CC(C(=O)NCC(O)CF)C12CCC2 50122,CCCCC(C(=O)NCC(C)N(C)C(c1nc(C(F)(F)F)cs1)=O)C(C)C 50123,N1(C(c2cc(Cl)c3c(c2)OCCO3)=O)CCC2(CCN(C(C3CC3F)=O)CC2)C1 50124,C(=O)(CC1=NNC(=O)C1)NC1CN(C(C(CC)(C)C)=O)CC(C(F)(F)F)C1 50125,CC#CCC(C(=O)NC1CCC12CCCC2)NC(C1CCC1COC)=O 50126,C(=O)(C(C)CC(=O)NCCOCCCNC(C1CNC(=O)C1)=O)OC 50127,C1(N(C(C23CCC(OC)C2C3)=O)C)CN(C(C2CC3(CCOC3)C2)=O)CCC1O 50128,S(=O)(=O)(c1ccc(C(=O)NCC2CC2NC(c2cnn(C3COC3)c2)=O)o1)NC 50129,N1(C(C23CC(COC)(OC2)C3)=O)CCCC(NC(C2ON=C(C)C2C)=O)CC1 50130,C1(CC=C)(NC(=O)C2=CCC2)CCN(C(c2ccc(CCC)cc2)=O)CC1 50131,c1(C(=O)OCC)nc(C(=O)NCCN(C(C2COCCO2)=O)CC2CC2)cs1 50132,CC1(C)C(CC(=O)NCC23CCCN(CC2)C3)CCN1C(c1ccsn1)=O 50133,N1(C(C(COCC)C)=O)CC2CCC(C1)N2C(c1cccc(F)c1O)=O 50134,Cc1nc(C(C)C)sc1C(N1CC(NC(=O)C2=CCC2)CC1CO)=O 50135,c1(C(=O)NCC(C)NC(CNC(COC)=O)=O)sc(Cl)c(Cl)c1C 50136,c1(C(C)NC(CC2(N(C(c3cn(CC)nn3)=O)C)CC2)=O)ccc(F)cc1 50137,C1(C(C)NC(=O)CCN(CC(F)(F)F)C)CCCN1C(=O)CC1(C)CCCO1 50138,N1(C(C2(C(C)(F)F)CCC2)=O)CC(NC(C2OCCC2C(F)(F)F)=O)CC(F)C1 50139,C1(C(=O)N(C)Cc2cncnc2)(CC)CCN(C(=O)C(C)NC(=O)NC)C1 50140,CC1=C(C(=O)NCCN(C)C(c2c[nH]nc2C(F)F)=O)CCCO1 50141,C(=O)(C(C)CCCOC)NCC1CN(C(C(c2cccc(Cl)c2)CC)=O)C1 50142,Cc1c(Cl)c(C(C)(C)N)nc2ccccc12.n1(C(C)C2CC2)cc(C(N)C(C)(C)C)nn1 50143,CCCC(C)CCCC(=O)N1CCCC1C1(O)CN(C(c2ccc(C)nc2)=O)C1 50144,c1(NC)c(C(N2CCC(N(C)C(c3csc(CO)n3)=O)C2)=O)cccc1F 50145,c1(OC)ccccc1C(O)C(=O)NC(C)C(C)NC(=O)Cn1cccn1 50146,c1(C(=O)NCC2CC(C)N(C(c3cscc3C(F)(F)F)=O)C2)ccnc(C#N)c1 50147,C1(C(C)NC(=O)C(F)n2cccn2)CCCCN1C(c1ccc(CO)cc1)=O 50148,N1(C(CC2CCC(C)(C)O2)=O)CCC2CN(C(=O)CCCC#N)CC2CC1 50149,N1(C(C2=NC=C2C(=O)OC)=O)CCN(C(c2ccon2)=O)C(CC(F)(F)F)C1 50150,C(=O)(C1(OC)CCc2c(NC(c3c(Br)cccc3Br)=O)cccc21)OC 50151,C(CCC(C)C(C(=O)NCC1CC1)N(c1ccc(Cl)cc1F)C)=C(C)C 50152,CC(CNCc1cc(C2CC2)n[nH]1)CC(F)F 50153,c1(OC)ccnc(C(N2CC(CN(C)C(c3cnc(Cl)s3)=O)C3(CC3)C2)=O)c1O 50154,c1(C(=O)OCC)ccc(CC(N2CCC2C(=O)Nc2cc[nH]c(=N)c2)=O)cc1 50155,N(C(=NCCN1CC2CC2C1)NCc1ccco1)Cc1scc(C#N)n1 50156,O=C(C1=CCC(NC(c2cc(C3CC3)ns2)=O)C1)NC(CO)C1CCC1 50157,CCCC(F)(F)C(=O)NCC1CC1CNC(=O)CCn1cncn1 50158,C(=O)(C(C)(C)C(C)(C)C)NCC1CN(C(C(C)N=[N+]=[N-])=O)CC1(C)C 50159,N1(Cc2n(CC)nc(C)c2)CC(=O)N(Cc2nc(C(F)(F)F)n[nH]2)C1=O 50160,C12(NC(=O)CCF)CN(C(=O)C3=CC4C=CC(C3)C4)CC1CS(=O)(=O)C2 50161,c1(C(N(C2CCCN(C(=O)CCc3cocn3)C2)CC)=O)cc(F)cnc1O 50162,C1(C(N2CCC(CNC(CCC(C)OC)=O)C2)=O)(OC)Cc2ccccc2C1 50163,c1(CC(=O)N(CCOCCN(C(C2N(CC)CC2)=O)C)C)n[nH]c(C)n1 50164,C12(NC(c3cc(CCC)[nH]n3)=O)CCC(CC1NC(=O)C(C)n1cncn1)C2 50165,c1(SCC(=O)NCC(CNC(CCOCCCC)=O)C)nnnn1C1CC1 50166,Cn1cc(-c2ocnc2C(N2CCC(NC(=O)CC3CCC3(F)F)C2)=O)cn1 50167,C1(NC(C2(C(O)C(F)(F)F)CC2)=O)CCC2CCN(C(c3coc4c3COC4)=O)C12 50168,CC(CN(C)C)CN=c1[nH]c(=NCC2CC23CCC3)[nH]c2c1CCCCC2 50169,c1(CC(=O)NC(C)(CNC(C2(C(N)=O)CC2)=O)CO)c(F)c(F)c(F)c(F)c1F 50170,C(CCCCC(=O)NCC1CC(C)N(C(=O)Cn2cnc([N+](=O)[O-])c2)C1)OC 50171,CC1CN(C(=O)Cn2ncnn2)CC(CCNC(c2cnc(O)s2)=O)O1 50172,CCCCC(CN(C(=O)NC(c1ccc(Br)s1)C)CC1(C)CCC1)CC 50173,CC(C(=O)Nc1ccccc1C(N)=O)S(N)(=O)=O.C1CN1CC1CC1 50174,CC#CCCCC(=O)NNC(=O)Nc1ccc(CCC(=O)OC)cc1OC 50175,N1(C(C(=Cc2cn[nH]c2)C)=O)CCN(C(c2csc(CC(C)C)n2)=O)CCC1C 50176,N1(C(C(=CC2CCCC2)C)=O)CC2OCCN(C(=O)CCS(C)=O)C2C1 50177,CCCCC(F)C(=O)N(C1CCCN(C(c2cc(CC3CC3)on2)=O)CC1)C 50178,C(=O)(CCC(C)S(C)(=O)=O)NCC1CC(NC(CC(C)C(F)(F)F)=O)C1 50179,Cc1cc(CC(=O)NC2CC(C)(CNC(c3c(C)cccc3F)=O)C2)cc(F)c1 50180,Cc1ncc(C(N2CCCC2(C(=O)Nc2ccc(O)nc2)C(C)C)=O)c(=N)[nH]1 50181,c1(C=O)ccccc1NC1COC1.c1(N(C(C)CNC(C2(CSC)CC2)=O)C)nnnn1C 50182,C(=O)(CCCCCC#N)N(C)CC1(O)CN(C(=O)Cc2csc(C(F)(F)F)n2)C1 50183,Cc1ccc2[nH]c(C(N3CC4CCC4(NC(C4(F)CCOC4)=O)C3)=O)cc2c1C 50184,N1(C(CC2N(CC)CCC2)=O)CC2(NC(C3CC(n4cccn4)C3)=O)CCC1C2 50185,C(CC(O)CNC(c1cnn(C2CC2)c1)=O)NC(C(N1CCCC1=O)C)=O 50186,C1(CN(C(Cc2cc(C)no2)=O)C)CCCN(C(c2occc2Cl)=O)C1 50187,C=Cn1nncc1C(=O)Nc1cccc(NC(=O)CC(O)c2ccccc2)c1 50188,C(C(N=[N+]=[N-])C(=O)N1CC(=O)CC1C(=O)NC1CCOC1C)OCC 50189,N1(C)CCC(=O)N(CCOc2cccnc2Cl)C1=O.C1OCCC1COC 50190,N12CCN(CC1)CC2=O.C1(CSCC)CCC(CNC(C2CC(OC)C2)=O)C1 50191,C1(CC)(NC(=O)CC2CCC(=O)O2)CCN(C(=O)CCCn2ccnn2)CC1 50192,C1(S(C)(=O)=O)(C(=O)NCC2C(CNC(CSC)=O)C2)CCCCC1 50193,c1(CN(C(=O)CN(C(=O)CCC(C)SC)C)CC)ccc(C)cc1 50194,C(CC1=CCN(C(=O)CC2CC23CC3)CC1)NC(c1n[nH]c2c1CCCC2)=O 50195,Cc1cccc2c(C(N3CCCN(C(=O)COC(C)C)C(CO)C3)=O)csc12 50196,N1(CC)Cc2ccc(NC(C3(OC(COC)C(C)(C)C)CCCC3)=O)cc2C1=O 50197,N1(C(C2CN(C)C2)=O)CCC2(CCCCN(C(C3CCC4(CCC4)CC3)=O)C2)C1 50198,Cn1nc(C(N2CC3CC3(CNC(=O)CN3CCC(C(N)=O)CC3)C2)=O)cc1O 50199,C(=O)(C1c2c[nH]nc2CCC1C)N(C(CCNC(c1c(O)ccc(C)c1)=O)C)C 50200,C1(=O)CCC(C)(C)N1CC(=O)N(C1CN(C)C1)C.C1(C)(N(C)C)CCCC1 50201,c1(C(N2CC3C(NC(C(CCC)OC)=O)(C3)C2)=O)ccc(Br)cc1F 50202,C1(NC(CCC#C)=O)CN(C(=O)C(CC(=C)C)NC(C)=O)CC1(C)C 50203,S(=O)(=O)(c1cc(C(=O)OC(C)(C)C)c(C)c(Cl)c1)N1CCN(CCCOC)CC1 50204,C(=O)(CS(=O)(=O)N1CCN(C)CC1)N(CCCNC(C(C)SCCCC)=O)C 50205,N1(C(c2c(C)cc(CO)o2)=O)CCC(C)CC1CNC(c1sccc1F)=O 50206,C1(C)(C(=O)NCC2C(COC)C2)CCN(C(=O)CC2CC23CC3)CC1 50207,CN1CC(C(N2CC(CC(F)C(=O)NCC3CC(O)C(O)C3)C2)=O)CCC1=O 50208,c1(C(=O)NCC(CC)NC(C(CCC)O)=O)cccc(S(=O)(=O)NCC(N)=O)c1 50209,c1(NC(C(N2C(c3c(C)noc3C)CCC2)C)=O)c(C)nn(C)c1C 50210,C(=O)(CC(O)CC(C)(C)C)N(C(CC(C)C)C(=O)NCC1(F)CCN(C)C1)C 50211,c1(SCC(=O)NC2CC(C)N(C(=O)CCNC3CC3)C2)ccc(F)c(F)c1 50212,c1(CC(N2CC(NC(C3C(CCC)C3)=O)C(C)C2)=O)cc(SC2CC2)cc(F)c1 50213,N1(C(C(C)O)=O)CCN(C(c2cc(C3CCCN3C)[nH]n2)=O)CC1 50214,c1(OC)cccc(C(=O)NCC2CN(C(C3CC(=O)CCO3)=O)CCO2)c1OC 50215,CS(=O)(=O)c1ccccc1CN1CCC(CC(N2CC3C(C2)C3(F)F)=O)C1 50216,C(=O)(C1CCc2cc(Cl)ccc21)N1CC(NC(c2nc(C)n(C)c2)=O)C(F)C1 50217,c1(C(=O)NCC2CN(C(C(CC=C)NC(C)=O)=O)C2)cc2nc(OC)ccc2[nH]1 50218,C1(C(N(CCCNC(C2CCC2C(C)(C)C)=O)C)=O)CCS(=O)(=O)CC1 50219,C1(CNC(c2ccc(Cl)o2)c2nnnn2CC2CCCO2)CCCCCC1 50220,c1(C(N2CCC(NC(c3cnco3)=O)C2)=O)ccc2c(n1)CCCC2 50221,C(CCCCNC(C1CC1(F)Cl)=O)N(C(C)C)C(c1ccc[nH]1)=O 50222,c1(CNC(c2c(C)onc2)=O)cccc(NC(C2CCCCC2C)=O)c1 50223,c1(C(=O)NC2CCN(C(COCC)=O)C2(C)C)cc2c(Br)c(C)ccc2[nH]1 50224,c1(C(C)C)cccnc1NC(=O)NOCCCS(N)(=O)=O 50225,N1(C(COCC(C)C)=O)CCC(C)CC1C(=O)Nc1ccc(CCF)cc1 50226,C1(C(=O)OCc2c(C)occ2)CN(C(=O)OC(C)(C)C)C(C)CO1 50227,C1(C(N2CC3CC3(C(N3CCC(c4ncco4)C3)=O)C2)=O)CC2CC1CC2O 50228,c1(CC)ccc(Br)cc1C(=O)NC1CC(N(C(=O)CC2CCOCC2)C)C1 50229,c1(CC(C)C(N2CC3CC2CN3C(C2(O)CCCCCC2)=O)=O)ccc(Cl)cc1Cl 50230,C1(NC(CCOCC(C)C)=O)CCCN(C(c2ccc3nn[nH]c3c2)=O)CC1F 50231,CCCCC(C)(F)C(=O)NCC1CC(NC(=O)CC2(N(C)C)CCCC2)CCO1 50232,Cc1oncc1C(=O)NC(C)C(=O)NCC(C)N(C(=O)C=CC(C)(C)C)C 50233,N1(C(C)C)CC(NC(=O)CN2CCN(C(=O)Cn3ncccc3=O)CC2)CC1=O 50234,C1(NC(C=C(C)C(C)C)=O)C2CC1N(C(=O)Cn1cc(C)cn1)C2 50235,C1(CNC(CCCN(C)C(C2(C3CC3)CC(=O)C2)=O)=O)CC2CCCC2C1 50236,c1(C(N2CCCC(CCNC(C(COCC)(C)C)=O)C2)=O)cnc2scc(C)n12 50237,N(S(=O)(=O)N1CCCC(C2CCOCC2)C1)CC(C)(C)OC(F)F 50238,C1(C2CC2)(C(=O)NCCCOC=C)CN(C(c2ccc(Cl)cn2)=O)C1 50239,N1(C(C2CCN(CC(CC)C)C2)=O)CCC(O)(C(=O)O)CC1 50240,N1(C(C(CSC)(C)C)=O)CC2(CC(NC(c3cn4cc(C)ccc4n3)=O)CO2)C1 50241,C1(C(=O)NCC2N(C(c3n[nH]c(CC)c3Cl)=O)CC(O)C2)CCOC(C)(C)C1 50242,c1(SC)nc(C)c(C(C)(C)NC(N2C(C(C)(C)NCCC(C)C)CCC2)=O)s1 50243,N1(C(C2N(C)CC(O)C2)=O)CC2CCC(Nc3ncc4c(n3)CCCC4)CC2C1 50244,C1(CC(=O)OC)(N(C(C=[SH]c2ccccc2)=O)C=S)CCOC1 50245,C1(CNC(C(C)c2ccon2)=O)(NC(c2cc(Cl)no2)=O)CCCCC1 50246,C1(C(=O)NCC(C(C)(C)C)NC(c2c(CC)c[nH]c2)=O)CCCCC(=O)N1 50247,c1(OC)cc(OC)c(OC)cc1CNCC1(c2ccc(C)nc2)CCC1 50248,CC(CC(=O)N1CCCC(CCO)CC1)C(C)(C)NC(=O)CC1(O)CCCC1 50249,N1(c2c(Cl)cnc(OC)n2)CCC(C2(NC(=O)CC(C)SC)CC2)CC1 50250,c1(OC)ccc2c(c1)C(C(=O)Nc1ccc(C(=O)NCCC(C)(C)O)cc1)CC2 50251,n1(CC)cc(C(=O)NC(C)CC(C)NC(=O)CN2CCNC(=O)C2)c(C(C)C)n1 50252,C(=O)(C(CC(C)c1ccccc1)N(C)Cc1cccnc1)NCC(C)C 50253,C1(OC)CCCC(C(=O)N(C2CCCC2)CCCNC(c2cn(C)c(C)n2)=O)C1 50254,C(N=c1[nH]cnc(Cl)c1C)C1C(NC(CCCn2c(C)ncc2)=O)CCCC1 50255,CCC(CC)CCC(=O)NCC1(C)CCN(C(=O)C(C)CNC(=O)OC(C)(C)C)C1 50256,C(=O)(C(F)C(=O)NC(C)(CSC)C(=O)NCC=C(C)C)OCC 50257,C(=O)(C(C)(CCC(N)=O)N=[N+]=[N-])NC1C(C)(C)CN(C)C1 50258,N1(C(C(CC)=O)=O)CCC2(CC2C(=O)Nc2cc(CO)nc(C(F)(F)F)c2)C1 50259,c1(C(N(C(CNC(C=COCC)=O)C)CC)=O)ccnc2ncnn12 50260,c1(OC)ncc(C(=O)N(C2CC3CC2N(C(=O)CSC(C)(C)C)C3)C)cc1Cl 50261,Cn1nc(Br)c2c(NCCNC(c3ccc(Cl)cc3F)=O)ncnc12 50262,c1(C(=O)NC(C(C)NC(c2cccc(O)n2)=O)(C)C)ccc(Cl)c(F)c1 50263,N1(C(CCCC#C)=O)CC2CCCC1C2CNC(=O)CC=C 50264,c1(CC)ncc(CNC(=O)C(C(C)C)NC(=O)OC(N)=O)c(=N)[nH]1 50265,c1(SC)ccncc1OCCNC(c1nncn1C)=O 50266,N1(C(c2cc(C#C)c(Cl)cc2)=O)CCC2(C1)CN(C(=O)CCN(C)CC)CCO2 50267,N1(C(C(C)=CC2CC2)=O)CC(C(N2CCC(CC(F)F)C2)=O)(N(C)C)C1 50268,Cc1cnc(NCc2cscc2C)c(S(=O)(=O)NC2CC3CC(CO)CC23)c1 50269,c1(C(c2nnnn2CC)NCCC(COCC)(C)C)cc([N+](=O)[O-])c(C)cc1C 50270,c1(C(=O)NCC2(NC(C(C)c3ccsc3)=O)CCC2)ccnc(F)c1O 50271,C1(C)(C(=O)OCC)CCCN(C(=O)CC(CC#N)C(=O)OC(C)(C)C)C1 50272,CC(C)C(O)C(C)(C)C(=O)NC1COCC1C(N1CC(C)(CF)C1)=O 50273,c1(Cn2c(C(C3(CSC)CC3)NC(CC)CC)nnn2)cccc(C(C)(F)F)c1 50274,C1(NC(CCC)=O)CC(CNC(=O)CCCOC(C)C)C1(C)C 50275,N1(C(C(CC(C)C)NC(C23CCC(OC)(CC2)C3)=O)=O)C2CCC1CC(CO)C2 50276,N1(C(c2c(C)cnnc2)=O)CC(NC(=O)CC(O)CN(C)C)CCC1C 50277,C1(C(=O)NCCC(C(C)C)NC(C2(C)CCC(=O)N2)=O)CC1C1CCCC1 50278,C1(NC(=O)NC2C(C)C2C)CC2CC3C(C2)C13 50279,Cc1ccc(C(O)C(N2CCCC(NC(c3ccc(Cl)nc3)=O)C2)=O)cc1 50280,CC(CN(C)C)CC(=O)NCC1C2CC1N(C(=O)Cc1nc[nH]n1)C2 50281,N1(C(C(CC)(C)CO)=O)CCCCC(CNC(c2ccon2)=O)CC1 50282,c1(NC(C2N(C(CC)=O)CCSC2)=O)cc(CO)ccc1C 50283,C1(CC#C)(C(=O)NCC(O)C(F)F)CCN(C(=O)CCCC#N)C1 50284,c1(C(C(=O)NCCCOC)N(CCC(N)=O)CC2CC2)nc(C#N)cs1 50285,Cc1cc(C(=O)NC2(CC(=O)Nc3nnc(C)o3)CCC2)nc(C)c1 50286,Cc1cnc2c(NCC3(Oc4ccccc4Cl)CCCSCC3)nccc2n1 50287,C(C)(C)(CC(=O)NC1C2CC1N(C(=O)CCc1ccccc1OC)C2)OC 50288,c1(C(N2C(CN(C(c3nccc(C)c3)=O)C)COCC2)=O)cc2c(ncn2C)[nH]1 50289,C1(NC(c2sc(C)c(O)n2)=O)CC2CC(C1)N(C(C1(C)CCCCC1)=O)C2 50290,c1(C(C)C)nc(C(=O)NCC2C(NC(=O)Cc3cnns3)CC2O)co1 50291,c1(-n2cc(CN3CCCC(NC(c4ccno4)=O)C3)nn2)ccc2c(c1)CCO2 50292,C(=O)(C(C)(F)F)NCC(C)CN(C)C(c1ccc(CSC(F)F)o1)=O 50293,CC1CN(C(c2nc(=N)cc[nH]2)=O)CCCN1C(=O)Cc1cc(F)ccc1Cl 50294,CC(CCCNC(c1nc(Cl)cs1)=O)NC(=O)C(C)(C)c1cscn1 50295,C1(COC)(NC(=O)C(C)n2cccc2)CN(C(=O)C(C2CCCCC2)O)C1 50296,C(C)(CNC(=O)C(c1ccnn1C)C)(C(C)C)NC(CNC=O)=O.CC#N 50297,c1(OC)ccc(N)c(C(=O)NCC2C(C)CCCN2C(=O)Cc2cc(Cl)cs2)c1 50298,C1(C(=O)NCCCCN2CCOCC2)CC12CCN(CCSC1CCCO1)CC2 50299,CC1N(C(C2N(C(c3ccc[n+]([O-])c3)=O)CCC2(C)C)=O)CCOC1(C)C 50300,c1(C(=O)NCCN(C(=O)CCC2CC2)CC)nn2cccnc2c1Cl 50301,Cc1cnc(CC(=O)NCCCC2CCCN2C(=O)C(C)(F)F)o1 50302,c1(C(N2CCCCC3CCC23)C(=O)NCCOC)ccc(F)c2ncccc12 50303,C1(CC)CNC(=O)CN1C(=O)CC1CN(C(=O)Cc2cccc(C)c2)CC1C 50304,CC1(C)CN(C(=O)Nc2ccc(C#N)cc2)CC1NC(C12CCC(C)(C1)OC2)=O 50305,Cc1ccc(Cl)cc1OCC(=O)NC1COCCN(C(c2ccc(=N)[nH]n2)=O)C1 50306,C(=O)(C1SCCc2sccc21)N1C(Cn2cc(-c3c(C)nn(C)c3Cl)nn2)CCC1 50307,CN1CCC(N(C)C(C2CCN(C(=O)COC3CC3)CC2)=O)C1=O 50308,C1(C)(CNC(CN2CCC(C)CC2)=O)COCCN(C(c2cnsn2)=O)C1 50309,C(=O)(CCC(=O)NCC(CC)NC(C1CCCN1c1ncccn1)=O)NCC 50310,C(=O)(C1=COc2ccccc2O1)N(C)CCN(C)C(=O)NC12CCCCC1C2 50311,c1(C2(CNC(C(C3CCCO3)NC(=O)Cc3cn[nH]c3)=O)CC2)ncccc1F 50312,CC1CN(CC2CCCC2)CCN1C(=O)CCCCN1CCOCC1 50313,N1(Cc2n(CC)cnc2)CC(N(C)C)C2(CC2)C1.N12CCC(C1)C2=O 50314,C#CC1(C(=O)NC2CC3CCCCN3C2)CCN(C(c2c[nH]c(C#N)c2C)=O)CC1 50315,c1(C(C(=O)N(CCNC(C(CC)(C)F)=O)Cc2ccccc2)=O)c(C)nn(C)c1C 50316,C1(CC(=O)NCC(CNC(=O)Cn2cc(C3CC3)cn2)OC)CCC(=O)NC1=O 50317,Cc1cc(I)c(Cl)cc1N(C(=O)CC1CCCC1)Cc1ccncc1 50318,C(=O)(C(C)(C)C(=O)N1CCOCC(C(N2CCN(C)C(CO)C2)=O)C1)OC 50319,N1(C(COC(C)C)=O)CCN(C(=O)Cc2cncnc2)C(CS(C)(=O)=O)C1 50320,CCCC(CNC(c1cc(CC)[nH]n1)=O)C(=O)NCc1cnn(CCO)c1 50321,C(CCCC(=O)NC1CCC(NC(C2(C)CSC2)=O)C1)SC 50322,C(=O)(CC(C(F)(F)F)OC)N(CC(=O)NCC1(CC)CCC(=O)N1)CCOC 50323,N1(C(C2(N(C)C)CCC2)=O)CCC(C(=O)NC(c2nc[nH]n2)C2CC2)=C(F)C1 50324,C1(NC(C(C)C(=O)OC(C)(C)C)=O)CN(C(c2ccoc2Cl)=O)CC1(C)C 50325,CC1Cc2cc(NC(=O)Cc3ccc(C(C)C(F)(F)F)cc3)ccc2O1 50326,CN1C(=O)CSC1=CC(=O)NC1CCC1NC(C1CC2(C1)CC21CC1)=O 50327,Cc1ncc(C=CC(N2CCC3CN(C(c4cc(C)n(C)c4)=O)CC23)=O)c(O)n1 50328,N1(C(CCc2cc(OC)no2)=O)C2CCC1CC(NC(C1CC(=O)N(C)C1)=O)C2 50329,Cc1ccc(C)c(C(=O)NC2CN(C(c3ccco3)=O)CCC2(F)F)c1O 50330,c1(C(C)NC(C2C(C(C)NC(=O)Cc3nccn3C)C2)=O)ncc(F)cn1 50331,C1(C(N2CC(C(Cn3cc(CCOC)nn3)F)C2)=O)CCn2cncc2C1 50332,C1(CC(=O)OCC)CCN(C(c2cccc(Br)c2Cl)C(=O)NCCSC)C1(C)C 50333,c1(C(=O)NC(CC)(C)CNC(C2C(C)(C)C2(F)F)=O)ccc2c(c1)OCC2 50334,N1(C(C(C=CC)O)=O)CCN(C(=O)CCNC(=O)Cc2ccccc2)C2CC12 50335,CC1CC(C(=O)NCC2CCC2)CN1C(C1(C(=O)OC(C)(C)C)CC1)=O.C(=O)(C(F)F)N 50336,N1(C(c2c(OC(C)C)nccc2)=O)CCC2(CC(NC(=O)CC(F)(F)F)CO2)C1 50337,c1(OC)ccc2c(C(=O)NC(C)CNC(C3CC4(CSC4)C3)=O)coc2c1 50338,c1(OC)ccc2c(c1)OCC2C(=O)N1CCC(C)C2(CCCCC2)C1 50339,C(=O)(CCC(C)(F)F)NCC1(OC)CN(C(=O)CC2CCCOCC2)C1 50340,c1(C(=O)NCC2C(OCC)CN(C(CS(CC)=O)=O)C2)cccc(F)c1Cl 50341,CC1(C)OCCC1NC(C1(NC(C2C=CCS2)=O)CCCC1)=O 50342,CS(=O)(=O)C1CCC(CNC(=O)C(=O)NC2CCC(F)(F)CC2)CC1 50343,C(CC(C)C)(C(=O)NC1CC(NCc2ccoc2)C12CCC2)OC 50344,CC(C)CC(C)(O)C(=O)N1CCN(CC(C)(C)NC(=O)CC(=O)NC2CC2)CC1 50345,c1(C(N2CCC(N(C(C(CCOC)C)=O)CCO)CC2)=O)c[nH]c2nccc-2c1 50346,CCC(CC(=O)NC1(CNC(c2cnc(C(C)C)[nH]2)=O)CCCC1)C(F)F 50347,c1(C(=O)NC(CNC(C2(COC)CCCC2)=O)CO)c(OC)cc(OC)cc1N 50348,c1(OC)cc(C(=O)NC2CCCC2NC(=O)CC2CC2(Cl)Cl)cc2c1OCC2 50349,C(=O)(CC1OCCc2ccsc21)NCC1C(C)CCCN1C(=O)Cc1ccco1 50350,CC1CCN(CC(=O)Nc2ccnc(CNC(=O)Cc3cccnc3O)c2)CC1 50351,N1(C(C=C(C)C(C)(C)C)=O)CCOC(CCNC(=O)CN2CC(C)C2)C1 50352,Cc1cc(CCC(=O)NCC2CC(NC(c3cnsn3)=O)C(O)C2)nn1C 50353,c1(C(=O)NC(CNC(C2(CC)CCOC2)=O)(C)C2CCC2)cncc([N+](=O)[O-])c1 50354,C12(NC(C=C(C)C3CCCCC3)=O)CCCCCC1N(C(C1CCC1)=O)CC2 50355,c1(CNC2C(C(N3CC(CC)OCC3)=O)C2)cc2ccc(Br)cc2[nH]1 50356,Cc1nc(O)sc1C(=O)NC1CCOCC1C(=O)NCCC1CC(C)(C)C1 50357,Cn1c(COC(C2OCC2(C)C)=O)ccc1Cl 50358,c1(C(=O)NC2CN(C(C3(C=C)CCC3)=O)CC2C)ccc(OCC2CC2)cc1Cl 50359,c1(CC)ncc(C(N2CC(NC(=O)C(C)CN(C)C)C(C(F)F)C2)=O)c(O)n1 50360,C1(CNC(C(CC#C)C2CC2)=O)CN(C(c2cccn2CCC)=O)CC12CCC2 50361,CCC(C(=O)NC(C)(C)C=CC(=O)NC(C)CC1CCC1)n1cncn1 50362,c1(-n2c(C3N(CC)CC3)nc(CS(C)(=O)=O)n2)ccc(C)cc1C(=O)O 50363,CCC(C)CC(=O)C(=O)N(C(C)C(=O)NCCc1cc(C)on1)C1CC1 50364,C1(CC(N2CC(C)(C(=O)NCC3(F)CCOCC3)C2)=O)(OC)CCOCC1 50365,C1(NC(c2cnc(CC)o2)=O)CC(CNC(=O)COCc2ccncc2)C1(C)C 50366,c1(NC(=O)NC(COCC)COC)cn2c(c1C#N)CCC(C)C2 50367,S(=O)(=O)(c1nc(N2CCC(C(C)CO)CC2)ccc1Br)NC(CC)CO 50368,c1(C(=O)NCC2(C)CCN(C(C3CCCCO3)=O)C2)ccc2cnsc2c1 50369,N1(C(C2C(=C)C2)=O)CCCCCC1CNC(c1cc(C(C)C)nn1C)=O 50370,C1(CC(=O)NCCCNC(c2cc(Cc3cccs3)on2)=O)CCCCO1 50371,c1(CNC(C(N2C(=O)CCC2=O)CC)=O)ccccc1CNC(C1SCCS1)=O 50372,c1(C(=O)NCc2c(C(=O)Nc3ccc(CCC)cc3)c[nH]n2)cc2occc2[nH]1 50373,c1(N(C)C)ccccc1N(C(=O)C(=O)NCC(=O)Cc1ccccc1)C 50374,C(=O)(C(C)C(O)CCCC)N(CC(N1CCCC(C)C1CCO)=O)CC#C 50375,Cc1ccc2nnnn2c1N(CC(C)C(F)(F)F)C 50376,CCCCCCC(CC)C(=O)N(CC(CC)NC(c1nnn2c1CCC2)=O)CC 50377,C1(C(=O)NC(CCCC)CCO)CC2(CCOCC2)CCO1 50378,N1(C(=O)Cc2ccccc2F)CCC(C(O)CNC(C23CCC2C3)=O)CC1 50379,N1(C(CC(C)F)=O)CCN(C(c2csc(CO)n2)=O)CC1c1ccc(F)cc1 50380,N1(C(C(CCCC=C)NC(C2CSCC(=O)N2)=O)=O)CC(C)OC2(CCC2)C1 50381,C1(C(=O)NCCC2N(C)CCC2)CCCC(NC(C2(CO)CCCC2)=O)CC1 50382,N1(C(C=NOC)=O)CC(C(N2CC(c3nc(C(F)F)no3)C2)=O)CC(C)C1 50383,C1(C(N2C(C(N(CCn3c(C)ncc3)C)=O)C(C)C2)=O)CCCC(C)(C)C1 50384,C12(C(=O)NC(CNC(c3cc(C)nc(O)n3)=O)C(C)(C)C)OCCCC1C2(F)F 50385,C1(C(N(CCCC(=O)NCC(CC#C)O)C)=O)CCCC(C#N)C1 50386,c1(C(N2CCC(NC(c3c(C(C)C)[nH]cc3)=O)C(C)C2)=O)cccc2cnnn12 50387,c1(C(N2CCC(CC=C)(NC(C3CC3F)=O)C2)=O)cc2c(Br)cccn2n1 50388,N1(C(=O)C2=CS(=O)CCC2)CCOCC2(COCCN2C(c2coc(O)n2)=O)C1 50389,CCS(=O)(=O)CC(=O)N1CCCCC1C1CCN(C(C2CC2F)=O)C1 50390,c1(NC(c2ccn3nncc3c2)=O)cc2c(cc1Br)CCC(=O)N2 50391,N1(C(C2C(C(C)C)C2)=O)CCC(O)(CN(C)C(c2ccc(CC3CC3)cc2)=O)C1 50392,CC1CN(C(=O)CC2C(C)(C)C2(C)C)CC1NC(c1ccc(C2CC2)o1)=O 50393,c1(CC)cnccc1C(N1CCOC(C(=O)NCC2(C)CCCO2)C1)=O 50394,N1(CC(CC(C)C)c2ccccc2)CCNCC(O)C1 50395,c1(C(N(C)CC2CCCN2C(=O)CCOc2cccnc2)=O)cn2c(n1)SCC2 50396,CC1(C)CCCCC1(C)NC(c1ccc(CNC(C2(C#N)CCC2)=O)nc1)=O 50397,N1(C(c2ccccc2)C(=O)NC2C(C)OCC2)CC2CN(C)CC(C1)O2 50398,c1(C(=O)NCCCN(C(CC2CC(OC)C2)=O)C(C)C)cnn2ccc(C)nc12 50399,CCN(Cc1ccc(C)cc1)N1CCN(C)CC(P(C)(C)=O)C1 50400,c1(C(=O)NCC=C2CCN(C(CC(C)C3CC3)=O)CC2)cc(Cl)cc([N+](=O)[O-])c1 50401,C1(NC(=O)CCCC2CCCC2)CC2(C1)CC2C(=O)NOC1CCOC1 50402,c1(C(=O)NCCCCCCO)cc2cc(-c3cnc4n[nH]cc4c3)ccn2n1 50403,N1(C(CCCCC#C)=O)CCC2(CC1)CC2CNC(c1c[nH]ccc1=O)=O 50404,C1(C(N(c2cnccn2)C)=O)CCCN(CC(F)(F)F)C1=O.C12CCCN1C2 50405,N12C(=O)CN(C1=O)N(C)c1cccc(c1)C2.C1(C)CC(F)C(=O)N1.CO 50406,CC1CN(C(=O)CCP(C)(C)=O)CC1(C)C(N1CCCC(CN=[N+]=[N-])C1)=O 50407,c1(C(C)NCc2noc(C(C)(C)C)n2)ccoc1CNC(C1(CCC)CCC1)=O 50408,C(C)(CN=c1[nH]c2ccccc2cc1C#N)NC(C1CCC(C)CC1)=O 50409,c1(OC)cncc(CC(=O)N(C2CCN(C(=O)C(C)(F)F)CC2)CC(C)C)c1 50410,C(=O)(C1=NOC2(CCC2)C1)NCC(CN(C)C(c1ncc(C(F)F)s1)=O)(C)C 50411,c1(CC)cccnc1C(N1CCC(C(C)NC(=O)CNC(C2CCC2)=O)CC1)=O 50412,C1(NC(C(Cc2ccsc2)NC=O)=O)CC2CCC1N2C(=O)Cc1ccn(C)n1 50413,N1(C(CCCCOC)=O)CCC(C2CCN(C(=O)Cc3c[nH]ccc3=O)C2)CC1 50414,c1(C(N2CC3(NC(CCC)=O)C(C2)CS(=O)(=O)C3)=O)cc2c(OC)cccc2s1 50415,Cc1ccncc1C(=O)N(C)CCOCCN(C(=O)Cc1cscc1F)C 50416,CCC(CC)C(F)C(=O)N1CCCC(O)(CCNC(=O)C(C)(C)C(C)(F)F)C1 50417,Cc1ccc(Cl)c(F)c1C(=O)NCC1CCC2(CN(C(C3CC34CCC4)=O)C2)O1 50418,C1(C2CCCN(C(c3cc(C)cs3)=O)C2)(NC(C(F)OC)=O)CC1 50419,c1(NC(Cn2c(C(C)C)cc(-c3nc(C4CC4)no3)n2)=O)nn(C)cc1S(C)(=N)=O 50420,N#CC1(CC(=O)NC2CCOC(CNC(=O)C=CC3CC3)C2)CCCCC1 50421,c1(CC)nc(O)c(C(=O)NCC(CC(C)C)NC(=O)CC2CCCOC2)cc1C 50422,c1(C(N2CCC(O)(CNC(C(COC)(C)C)=O)C2)=O)ccc2c(C)[nH]nc2c1 50423,C1(C(=O)NCc2c(OC)ccc(C)c2)CC12CCN(Cc1ccc(Cl)nc1)CC2 50424,c1(C(N2CC3C(NC(c4ccn(C(C)(C)C)n4)=O)C3C2)=O)ccc(O)nc1Cl 50425,C1(N(C(=O)CNC(=O)COC)CC#C)CCN(C(=O)CCc2nncn2C)CC1 50426,c1(CNC(N2C(CC)C(=O)NCC2)=O)ccc2c(c1)cc(C)n2C 50427,C(C1CN(C(=O)CC2CCN(C)C2=O)CC1C(=O)NCC(F)C1CCC1)=CC 50428,c1(NC(C2N(C(CCNC(C)=O)=O)CCC2)=O)nnc2ccc(Cl)nn12 50429,O=C(NN1CC(CO)C1)C1CC=CCC1C(N1CCC(O)CC1)=O 50430,CCC(C)C(CC(=O)N1CC(O)C1)NC(C1CCCS1)=O 50431,c1(C(=O)NCC(C)(C)NC(C2CC3(CCC3O)C2)=O)cc(F)cc(F)c1O 50432,C(=O)(CCCC(=O)N1CC2(CNC(=O)CC3(C)CC(F)(F)C3)CC1CO2)N(C)C 50433,c1(NC(C2(C)CCCN2Cc2ccc(O)cc2O)=O)ncnc2sc(Br)cc12 50434,c1(C(N(CC(CNC(CSCC(C)C)=O)C)C)=O)cc([N+](=O)[O-])c[nH]1 50435,c1(C(=O)NC(CNC(C2=C(CC)OCCS2)=O)CO)cccc2nc(O)n(C)c12 50436,c1(NC(C2CCCN(C(=O)CSc3cnn(C)c3)C2)C)ncc(C#N)cc1Cl 50437,N1(C(C(C2CC2)OCC)=O)CC2CC2(C(N2CC(OCC(=O)NC)C2)=O)C1 50438,Cc1cnc(C(=O)NCC(C)CNC(C23CC(F)(CO2)C3)=O)cc1Br 50439,C1(NC(C2C(C)(C)C2CNC(=O)CC2CC3CCC2C3)=O)CCC(C2CC2)C1 50440,C1(O)(C(C(=O)NCCSCC(=O)Nc2cc[nH]n2)F)CCCC1 50441,C1(NC(Cc2ncc(C(C)(C)C)[nH]2)=O)CCCC2CN(C(=O)C(N)=O)CC12 50442,C1(C(=O)NC2(C3CCC3)CN(C(C(C)(C)C3CC3)=O)C2)CCCCC1F 50443,N1(C(C(CC)OC)=O)CCC(CCN(C)C(c2cnn(C(C)C)c2N)=O)CC1 50444,C1(CC#C)(C(=O)NCC2CCN(C(=O)C(c3ccccc3)C)C2)CCCC1 50445,n1(CC(=O)NC2(C3N(C(CC(C)F)=O)CCC3)CC2)cc2ncccc2n1 50446,N1(C(Cc2cccc(C)c2)=O)CCCC2(NC(c3cnc(Cl)[nH]3)=O)CC2C1 50447,C#CC(CC(C)C)NC(=O)CCN(C(=O)C(C)(C)CC)C 50448,CN1CCCC12CN(C(=O)CC1(CNC(C3CCOC(=O)CC3)=O)CC1)C2 50449,c1(OC)ccc(C(N2CCN(C(C3CC(O)C3)=O)C3CC23)=O)c(OC)c1Cl 50450,C(CC(C(C)C)NC(c1cccc(-n2cncn2)n1)=O)N(C(C(C=CC)O)=O)C 50451,C(CN=c1nc(C(=O)OC)nc[nH]1)C1CC(NC(=O)NC2CC(CC)C2)C1 50452,C(=O)(C1CCCc2nccn21)N1CCN(C(c2cc(C)oc2)=O)CC(O)C1 50453,c1(CCCC)cccc(C(N2CCC(C(N)=O)(N(C)C)C2)C(=O)NC2CC2)c1F 50454,c1(OC)c(F)ccc(F)c1C(N1CC2CC2(NC(=O)COCC(F)F)C1)=O 50455,N1(C(Cn2ccc(C)n2)=O)CC2(CC2)CC1C(=O)NCC1CCCO1 50456,c1(C(=O)NCCCCC2CN(C(C3CC(CCC)C3)=O)C2)cc(C)nn1C 50457,C12(NC(C3(S(C)(=O)=O)CC3)=O)CCOC(CNC(C3CC3C3CC3)=O)(C1)C2 50458,c1(C(=O)NCC2(O)CN(C(C(C)NC(=O)NC)=O)C2)ccc2cc[nH]c2c1 50459,Cc1cccc(C(=O)NC2CCCCC2CC(=O)NC(C(C)C)C(C)C)c1N 50460,C1(C(=O)NCCc2ncccc2F)COCCN(C(c2n[nH]c3c2COC3)=O)C1 50461,c1(CNC(=O)NC2(C)C(C)OCC2)ccc(S(N)(=O)=O)cc1 50462,c1(C(N2CC(C(=O)Nc3ncc(SC)s3)NCC2)=O)cc(O)c(O)c(Cl)c1 50463,c1(C(=O)NC(C2CN(C(=O)C=CCN(C)C)C2)C)ccnn1C1CC1 50464,C1(C(=O)NC2CC(OC)C2)CCCCC1NC(C1CC(F)(F)CS1)=O 50465,C(C)(CCC(=O)NCc1ccsc1C(=O)N(C1CCN(C(C)C)C1)C)OCC 50466,N1(C(CS(=O)(=O)NC)=O)CC(NC(c2cc(-c3ccc(C)o3)[nH]n2)=O)CC(O)C1 50467,N1(C(C(C)(F)F)=O)CCCCC(NC(c2cnnc(C3CC3)c2)=O)C1 50468,N1(C(c2c(C)cn(C)n2)=O)C2CCCC1CC(NC(c1cn(C)[nH]c1=N)=O)C2 50469,N1(C(c2cc(C)nnc2)=O)CC(=O)NCC1C(=O)N(CC(=O)N(C)C)C 50470,C1(C(=O)NC(CC2CN(C(C3CCC(C(=O)OC)C3)=O)C2)C)CC12CCOC2 50471,N(C(=NCCc1ccccn1)N1CCCC(O)CC1)CC(C(=O)OC)C 50472,C(C(C)C(C)C(=O)N1CC(CNC(c2cccc(C)c2Cl)=O)(OC)C1)OC 50473,CCC(C)CCC(=O)NCC12CC1CN(C(=O)C=CSCc1ccco1)C2 50474,N1(C(c2c(C(C)(C)C)ncnc2)=O)CC2(C1)CN(C(=O)CC1CCC(C#N)C1)C2 50475,N1(C(C2C(NC(c3c(C)n[nH]c3)=O)CCC2)=O)CCN2CCOCC2C1 50476,C1(CC(N2CCC(COC)(NC(=O)CC3(C)CCOC3)C2)=O)CN2CCN1CC2 50477,N1(C(c2c(OC)ccs2)=O)CCN(C(c2cnccc2Cl)=O)CC1C 50478,C1(CNC(CC2ON=C(C)C2)=O)(CNC(c2cnnc(O)c2)=O)CC12CCC2 50479,c1(C(=O)NCC(CNC(CN(CC)CC)=O)CO)ccc2c(n1)CCC2 50480,C1(NC(C(C)Cn2cccn2)=O)CC(F)CN(C(c2csc(-c3cnc[nH]3)n2)=O)C1 50481,Cc1c[nH]cc1C(N1CCC(NC(c2ccsc2-n2cnnn2)=O)C1)=O 50482,Cc1cnn2ccc(C(=O)NC(C)C(CO)NC(=O)C(n3nccc3C)C)nc12 50483,N1(C(C(c2ccncc2)C)=O)CC2CCCC(NC(C3CC34CCOC4)=O)C2C1 50484,C(N=C(NC1CCCC1)N1CCCC(O)(CO)C1)c1c(COC)cco1 50485,C=C(C)CCC(=O)NC1CCC(CCNC(c2nccnc2C)=O)C1 50486,C1(CC)(CO)CCN(C(C2(COC)CC2c2ccncc2)=O)C1 50487,n1(CC(N2C(C(CNC(C)=O)Cc3ccccc3)CCC2)=O)cc(F)ccc1=O 50488,c1(C(N2CC3CN(C(C4=C(C)CCC4)=O)CC3C2)=O)c([N+](=O)[O-])c(C)nn1C 50489,C=C(Cl)C(C)(C)C(=O)N1CC(CNC(=O)CCn2cc[nH]c(=O)c2=O)C(C)C1 50490,c1(C(N(CCCN(C(C(C)NC(=O)C(C)(C)C)=O)C)C)=O)nc2ncccn2n1 50491,O=C1CC2(C1)CC(C(=O)NCc1ccc(C(N3CC(F)C3)=O)cc1)C2 50492,N1(C(C=C(C)Cl)=O)CC2CCCC1C2CNC(=O)CN(C)C(=O)C1CC1 50493,Cc1occc1C(=O)NCC(=O)NC(C)CNC(=O)CCC1CCC(=O)N1 50494,C1(CC)CCCN(C(c2cc(CNC(=O)CCc3ccn(C)n3)nn2C)=O)CC1 50495,c1(C(N2CC(CC(N3CC(O)C(F)C3)=O)C2)=O)ccn2nccc2c1 50496,C(=O)(C(C)(CO)NC(C1CCC(F)(F)C1)=O)N(CC(C(=O)NC)C)C 50497,N1(C(c2ccc(SCC)nc2)=O)CC2CC(C1)C2NC(=O)Cc1ccccc1F 50498,N1(C(C2(COC)CCCCO2)=O)CCC2(CCC(NC(C3CCCO3)=O)C2)CC1 50499,N12CCC(F)(CC1)C2=O.c1(CNC(C2(CC)CC2)=O)ccc(N(C)C)cc1 50500,c1(C(c2n(C(C(=O)OC)C)nnn2)NCC(C)(C)CO)ccc(Br)c(F)c1F 50501,n1(C(C)C)cc(NC(c2nnnn2CCC2(C)CC2)(C)CC2CCC2)cn1 50502,N1(C(c2c(OC)cccc2O)=O)CCOCC(NC(c2n[nH]cc2[N+](=O)[O-])=O)C1 50503,c1(C(=O)NCC2(NC(C3CN(C)C3)=O)CCCCC2)cc2c(cc1N)CCC2 50504,C1(C(=O)NC(COC)CO)N(C(=O)CCOC2CC2)CCCC1(C)C 50505,c1(C(N2CC(CNC(CCC=C(C)C)=O)C(C)C2)=O)cc(Cl)c2ccccc2n1 50506,Cc1ccc(OC(C)C(C)NC(=O)C(N2CCC(N(C)C)CC2)=O)c(C)c1 50507,N1(C(C(C(C)O)(F)F)=O)CCC2(CC1)CCN(C(C1(CCN(C)C)CC1)=O)CC2 50508,C1(CCNC(C2(C)CC3CC3C2)=O)CCN(C(=O)CC2CC2)CC1(F)F 50509,c1(N(C)C)ccc([N+](=O)[O-])c(C(=O)NC2CN(C(C3CCC3(F)F)=O)CC2O)c1 50510,C1(C(N(CC(C#C)OCCO)C)=O)(CO)C=CCN1C(=O)CCOCCOC 50511,CC1(C)CC(CCNC(=O)Nc2cc(C(C)(F)F)on2)CO1 50512,c1(C(N2CCCC(C(=O)NCc3ccc4c(c3)CC4)CC2)=O)ccc(Br)cc1Cl 50513,C1(CNC(c2c(CC)noc2C)=O)CCN(C(c2c[nH]c(C)c2)=O)CCC1(F)F 50514,N1(C(CC(C)F)=O)CCCC(CNC(C2(F)CCCCC2)=O)CC1 50515,CC(CF)CC(=O)NC(CNC(=O)C(c1ccc(Cl)cc1)(F)F)CO 50516,c1(C(=O)NCC(C)NC(c2c(F)ncc(OC)c2)=O)ccc(F)c(C)c1N 50517,C1(C(=O)NCC2(C(=O)OC)CC2)CCCN(CC(C)C)C1.C12CCCN1C2=O 50518,CCC1(C)CN1.c1(CNC(=O)COC)cn(CC2CCCCC2)nn1 50519,c1(C(=O)NC2(CC(=O)OC)CCCOC2)sc2ccsc2c1C 50520,c1(CC(=O)OCC(c2c(C)ocn2)=O)ccnc(Cl)c1F 50521,C(=O)(C(CC(C)C)NC(C)=O)N(C1C2CN(C(C3(CC)CCCO3)=O)CC12)CC 50522,c1(C(=O)NC(CN(C(c2c(COC)nn(C)c2)=O)C)C)cc2cc(Cl)ccc2s1 50523,c1(CN(C=O)Cc2cccc(CNCc3nn(C)nc3Br)c2)ccc(Cl)c(F)c1 50524,c1(CC)ccc(C=CC(=O)N(C(C)CNC(C2CCCC2(F)F)=O)C)o1 50525,CC(CS(C)(=O)=O)C(=O)NC(C1CCN(C(c2cc3c(ccn3C)[nH]2)=O)C1)C 50526,C1(OC)CC(NC(=O)NCC(C)Oc2ccc(C)cc2)C12CCOCC2 50527,c1(CCC(N2CC(NC(CSCCCC)=O)C2)=O)cc2ccccc2o1 50528,C1(C(=O)NCC(CCC)C)(C(C)C)CCN(C(=O)C(CO)NC(N)=O)C1 50529,Cc1cc(C)n(CC(N2CC(N(C(=O)Cc3c(C)noc3Cl)C)C2)=O)c(=O)n1 50530,c1(C(N2CC(NC(c3c(SC)csc3)=O)C3C2C3)=O)cc2cccnn2n1 50531,C1(CC(=O)NCC(=O)OCCCC)CCCN(C(=O)C2=NOC(C)C2)CC1 50532,c1(OC)ccc2c(CC(C(=O)O)NC(c3cnn(C(C)(C)C)c3C)=O)c[nH]c2c1 50533,c1(C(=O)NC2CC2C(N2CCC(N3CCOCC3)CC2)=O)cccc(F)c1Br 50534,C1(C(N(C)CC2(C)CC2)=O)CC(C)(NC(=O)Cn2cc(CO)nn2)C1 50535,c1(CC(=O)NC(CNC(=O)Cc2ccsc2Br)CO)ocnc1C(F)F 50536,c1(CC(=O)NCCN(C(c2nc(CC)sc2)=O)C)ccc(CO)c(C)c1 50537,C1(NC(c2csc(Cl)c2Cl)=O)CC2CC1N(C(c1cnco1)=O)C2 50538,c1(C(N2CC=CC(O)C2)=O)cnc2[nH]ccc2n1.CCC(F)(F)F 50539,N1(C(C2C(=C)C2C(=O)OC)=O)CCC(C)N(C(C2CC2F)=O)CC1 50540,N1(C(c2n(C)c(=O)ccc2)=O)C2CCCC1CN(C(C1CCC13CCC3)=O)CC2 50541,Cc1cccc(C)c1CS(=O)(=O)NC(C1CCC(F)(F)C1)=O 50542,C1(C(=O)NC(C2CC=CCC2)C(=O)NCCC2(O)CCCC2)(SC)CC(=O)C1 50543,C1(NC(Cc2c(C)occ2)=O)CN(C(=O)CC#N)CC12CC2.C12CC(C1)C(=O)N2 50544,Cc1nc(-c2c[nH]c(C(=O)NCC(C3CCCC3)NC(=O)C=CCF)c2)cs1 50545,N1(C(c2ccc(CC)nc2)=O)CCC2(CCN(C(c3ccc(F)cc3Cl)=O)C2)C1 50546,C1(NC(C2=C(C)OCC2)=O)CCCC2CN(C(=O)CC3COC(C)(C)C3)CC12 50547,n1(CC(C)C)cc(NC(C(c2ccn(C)c2)N(C)Cc2cccs2)=O)cn1 50548,CC1CCC(C2CCCC2)CN1Cc1cn(Cc2cccnc2)nn1 50549,c1(OC)ccc(Cl)cc1C(N1CCC(CNC(=O)CC2CC2)C(O)C1)=O 50550,N1(C(CC2(C=C)CCC2)=O)CC2CC2(CNC(C2CCC(=O)N2C)=O)C1 50551,c1(C(N(C2CCN(C(=O)C=CC3CCC3)CC2)C)=O)cc(O)cc(C#N)c1 50552,COn1cnc(C)c1C(=O)NCC(c1ccccc1F)NC(=O)Cc1ccns1 50553,C(=O)(CC(C)CC(C)C)N(CCCCNC(c1cccc(NC(=O)NC)c1)=O)C 50554,C(=O)(C1CCc2c[nH]nc21)N1C(C(N(CC#C)CCO)=O)C2(C1)CCCC2 50555,N1(C(C(CC)(C)C)=O)CC2CCC2(NC(=O)CCOc2cccc(F)c2)C1 50556,C(=O)(C1CCCc2scnc21)NCC1CN(C(c2c(C)cns2)=O)CC(C)(C)O1 50557,Cn1nc(C(=O)NC2CCN(C(C3CCC34CCC4)=O)CC2O)c2c1CCCC2 50558,C1(CNC(C(C)NC(CC)=O)=O)C(C)CCCN1C(C1CCCC(=O)N1C)=O 50559,C1(CNC(C=C2CCN(C)C2)=O)CCN(C(=O)C=CC(C)(C)C)CC1O 50560,CC1(NC(=O)C(O)C(C)(C)C)CCN(C(=O)Cn2cnnc2)CC1 50561,C(=O)(C(C(C)O)NC(=O)CC1CCCN(C)C1)N1CC(C)C1C(N)=O 50562,C1(C(N(CCCNC(=O)COC2CCOC2)CCO)=O)CC=CCC1 50563,Cc1noc2nc(C(=O)NC3CCCN(C(=O)CC4CNC(=O)C4)C3)ccc12 50564,CC(c1ccccc1)=CC(=O)NCC(C)N(C(=O)C(C)C1(O)CCC1)C 50565,C1(C(=O)NC(C#C)CCC)CC2CN(C(C3C4CCCC(=O)C34)=O)CC2C1 50566,C1(CC)CN(C(C2CCCOCC2)=O)CCN1C(=O)COCC1(F)CC1 50567,N1(C(CC2OCC(C)(C)C2)=O)CC(C(N2CC(N3CCCCC3)C2)=O)C(F)(F)C1 50568,c1(C(=O)NCC2(F)CC(CNC(=O)C=Cc3ccc[nH]3)C2)cc(Cl)cc(Cl)c1 50569,c1(CNC(C2(C)CCN(Cc3ncn(C)c3)CC2)=O)ccc(C#N)c(F)c1 50570,c1(N(CCC)C)nnc(C(c2ccsc2)O)n1CCCOCC1CC1 50571,c1(N2CCN(C)C(CNC(c3cn4c(n3)CCC4)=O)C2)ncnc2[nH]ccc12 50572,c1(C(C(=O)N(CC(C)(F)F)C)NC(C(C2CCC2)OCC)=O)ccccc1 50573,C1(C)(C(=O)OC)CNCCN1Cc1ccncc1 50574,c1(C(C(=O)NC)N(C)Cc2ccc(Cl)o2)ccc(Oc2ccccc2)cc1 50575,CN(CCN1CCNCC1)N1CCC2CC1CO2 50576,n1(CCOC)nc(COc2ccccc2C)nc1-c1ccc(C(C)C)cn1 50577,C1(NC(C=C(C)Cl)=O)CCCCC12CCN(C(=O)C=Cc1ccoc1)CC2 50578,N1(C(Cc2ccc(OCC#N)cc2)=O)CC(O)C2(CCOCC2)C1 50579,c1(CC)cc(C(N2CCCC2CCC(C)C)C(=O)NCCCF)ccc1Cl 50580,Cc1nc2ccc(C(=O)NC3CCC(NC(=O)CCOC4CCC4)C3)cc2n1C 50581,C12(CNC(c3ccn(CC(F)F)n3)=O)CC1CN(C(C1CC=CC1)=O)C2 50582,CCC(O)C(C)(C)C(=O)NCC(O)CCNC(=O)CCc1nncn1C 50583,c1(OC(C(=O)NCCC(C)N(C(c2n(CC)ncc2)=O)C)C)cccc(CO)c1 50584,c1(C(=O)NCC2CC(C)N(C(c3ccoc3Cl)=O)CC2)ccc2c(n1)CCC2 50585,CCN(NC(=O)C(O)CCn1ccnc1)C(=O)OC(C)(C)C 50586,C1(C(N(CC(=O)NC(C)C)C)=O)(NC(c2ccc(F)cc2)=O)CCCC1C 50587,N1(CCCC(=O)N(C)C)CC2C(Cc3ccccc3)CS(=O)(=O)C2C1 50588,CCCC(C)(C)C(=O)NCC1CN(C(c2nncs2)=O)CC(C(F)(F)F)O1 50589,C(=O)(CC(P(C)(C)=O)c1ccccc1)NCC1N(C(CCOC)=O)CCCCC1 50590,C1(CCOC)CN(C(C2(CC(F)(F)F)CC2)=O)CCN1C(=O)CCS(C)=O 50591,N1(C(=O)NCc2c(C)cccn2)CCN(S(=O)(=O)N2CCN(C)CC2)CC1 50592,CC(C)(C)S(=O)(=O)CC(=O)NCC1CCN1C(C1(C)CCC(=O)N1)=O 50593,C1(C(=O)NC2(c3onc(C)n3)CC2)CCCCCCN1C(=O)C(C)CC(F)F 50594,CCCC(CCNC(=O)CCC1(C)CN(C(C2CCC(O)CN2C)=O)C1)CCC 50595,C(C(C)NC(c1cccn1CC)=O)(C(C)C)NC(CCC)=O 50596,c1(OCC(N2CC(NC(=O)C=Cc3ccccc3)C(O)C2)=O)ccc(F)c(Cl)c1 50597,C(c1ccccc1)=CCN(C(C1N(C(C)=O)CCC1)=O)C.C12CN(C1)C2=O 50598,C1(C(=O)NCCCOCCCNC(C=CC(CC)C)=O)CCC2(CCC2)O1 50599,CCC(CC(=O)NC1CN(C(c2ccc(F)c(-c3ccccc3)n2)=O)C1)C(F)F 50600,N1(C(C=CC(C)(C)C)=O)CC(O)(C(C)(C)CNC(=O)CC2COCC2O)C1 50601,Nc1cnc(C(=O)NC2CC2NC(=O)C=Cc2ccccc2Br)c(Cl)c1 50602,C=CC(C)(O)C(=O)NCCCC(C)NC(=O)CC(O)Cc1ccccc1 50603,CC#CCC(C(=O)NCCC(O)CCC)NC(=O)C(C)OCC1CC1 50604,c1(C(C)(CO)NC(C(C)Sc2nn[nH]n2)=O)ccccc1Br 50605,N1(C(CCCOCCC)=O)CCN(CC(=O)N(C(C)CC2CC2)C)CC1 50606,C(=O)(CC(CC)C(C)(C)C)NCCC(C(=O)Nc1cnc(CCC)nc1)OC 50607,c1(C(N2CC(C)(NC(CC(CCC)C)=O)C2)=O)cc2c(nc1O)CCC(CC)C2 50608,c1(C(=O)NCC(CC(C)C)NC(C=CSC)=O)cc(Cl)cc2c1NCCC2 50609,Cc1c(CCNC(=O)Cc2ccc(O)nc2)cccc1Cl 50610,N1(C2(C(=O)NC(C(C)NC(=O)Cn3ccnn3)C)CC2)CCOCC1 50611,C(=O)(C(F)C(C)(C)O)NCC1(CNC(c2ccc(OCC#C)cc2)=O)CCCC1 50612,C=CCCCCCC(=O)N1CC2CC(NC(c3cc(C)oc3CC)=O)CC2C1 50613,C=CCCCCC(=O)NC(C1CCN(C(=O)C=C(Cl)Cl)C1)C 50614,c1(C(N2CC(O)(CN(C(=O)CS(N)(=O)=O)C)C2)=O)cnc(F)c(F)c1 50615,C1(C(CNC(C2(C)CCCC2)=O)O)CCN(C(c2ccc(O)nc2)=O)CC1 50616,C(CNC(c1ccc(O)nn1)=O)(CC(F)(F)F)NC(c1cncc(OC)c1)=O 50617,S(=O)(=O)(c1ccc(-c2ccc(NCCC)cc2)s1)N(CC=C)CC=C 50618,c1(C(N(C2CCCN(C(c3c(CC)c(C)sc3)=O)C2)C)=O)c(C)cc(O)cc1C 50619,C1(NC(C=C(COC)C)=O)CC(CNC(=O)CCc2cccnc2)C1(C)C 50620,c1(CC(N2CCC(C(C(=O)N(C(C#C)C)CCCC)C)C2)=O)ccnc(Cl)c1 50621,C=C(C)CCCC(=O)N1CCC(C)C(CC(N2CC(CO)CC2CO)=O)C1 50622,c1(C(N2CC(C)C(NC(=O)CCCCC3CC3)C2)=O)ncc(C(F)F)cc1Cl 50623,c1(N(N2CCCC2)C)nc2c(c(=NC3CCCn4ccnc4C3)[nH]1)CSC2 50624,C(=O)(CCCCCNC(N)=O)NC1(F)CN(C(CN2CC(C)(OC)C2)=O)C1 50625,C12CCN(C(=NCC(C3CC=CCO3)C3CC3)NC1)C2.N(C(C)C)(CC)CC 50626,N1(C(c2c(-n3c(C)ccc3C)scc2)=O)CC(=O)N2CCOCC2(CO)C1 50627,c1(CC)cccc(C(=O)NC(C(=O)NC2CN(C)NC2=O)C2CCCC2)c1 50628,C1(COC)(NC(=O)CCSC(F)(F)F)CCN(C(c2c[nH]nc2C(C)(C)C)=O)C1 50629,c1(CC(=O)NCC2CN(C(c3[nH]ncc3C#N)=O)CC2O)csc2ccccc12 50630,C1(C)(CN2C(C(C)C=O)CCCC2)CC12CCN(CCc1ncccc1Cl)CC2 50631,c1(C(=O)NCCC(CNC(C2(CSC)CC2)=O)O)ccc(-c2cnc[nH]2)cc1 50632,N1(C(C(C)C#N)=O)CCN(C(=O)CNC(c2ccccc2)=O)C(CC2CC2)C1 50633,CCCC(O)CC(=O)N1CCC(C(C)NC(c2cc(C)c(C)[nH]2)=O)CC1 50634,Oc1nccc(=NC2CC(c3ccc(Cl)cc3)C23CCC3)[nH]1 50635,c1(OC)cc2c(cc1OC)C(N(C)C(=O)NC(c1cccnc1)C(C)C)CC2 50636,c1(OC)c(Cl)cc(C(N2CCC(NC(=O)CCC3CCC(=O)N3)C2)=O)cc1Cl 50637,N1(C(C(CC)NC(C)=O)=O)CC2(CCCC2)C1C(=O)NC(C(C)C)C1CC1 50638,c1(N2CCC(CC)C2)nc(=NCc2nc(C(C)C)n[nH]2)[nH]c2c1CCCCCC2 50639,c1(C(C(=O)NCCCCN(C(C(COCC)F)=O)C)N(C)C)c(F)cccc1F 50640,CC(=NOCC#N)C(=O)NCC(O)CCNC(C1CC(O)CN1C(N)=O)=O 50641,c1(C(N2CC3(C(NC(c4c(C)onc4)=O)CC3)C2)=O)cnc2cc(O)ccc2c1 50642,C(=O)(C#CC1CCCCO1)N(C(CNC(C1C(C=C(C)C)C1(C)C)=O)C1CC1)C 50643,c1(CCC)cc(C(=O)N(CCC(C)NC(=O)C(=C2CCCCC2)F)C)ccn1 50644,Cc1cccc(CCNC(=O)CCC2(C)CN(C(C3CC(C(C)C)C3)=O)C2)n1 50645,C(C(CO)C(C)(C)C)c1onc(-c2ncc(C)o2)n1 50646,C1(C(N2CC(NC(Cc3cc(C)c(Cl)cc3)=O)C2)=O)CCCC(F)(F)CC1 50647,C1(C#N)(C(=O)NCC2OCCN(C(Cc3nc(NC=O)sc3)=O)C2)CCOCC1 50648,S(=O)(=O)(c1nc(N2CCCC(F)C2)ccc1Br)N(C)CCOC(C)(C)C 50649,C1(C(N(CCCNC(c2cscn2)=O)C2CC2)=O)CC2CC(=O)C1O2 50650,N1(C(C(CC)O)=O)CCC(F)(C(=O)NCC2CC23CC3)CC1 50651,C12(NC(c3ccc(Cn4c(C)cc(C)n4)o3)=O)CCCC(CC1CO)C2 50652,C(=O)(C(F)CC(CC)CC)NC(CC#C)(C)C(=O)NC1CC(C#N)C1 50653,O=C1CCC(C(=O)NC(Cn2cccn2)C(=O)NCCCCN2CCCC2)O1 50654,c1(OC)c(F)ccc(F)c1C(=O)NC1CCN(C(c2cc(C)ccn2)=O)CC1F 50655,C1(C(N2CCN(CC(C)NC(C3(C)CC3(C)C)=O)CC2)=O)Cc2cscc2C1 50656,N#CC1CN(Cc2ccc(O)c(O)c2)CC1NC(=O)Cc1cccc(C(N)=O)c1 50657,N1(C(c2ncn(C)n2)C(=O)N2CC(NC(N)=O)C2)CCC(O)C(F)C1 50658,Cc1ccccc1C(C)CC(=O)N(C1CCN(C(=O)C(C)(C)O)C1)C 50659,N1(C(C2(C)CSC2)=O)CC(O)(CNC(=O)CNC(c2cccnc2)=O)C1 50660,C1(NC(C=Cc2scc(C)n2)=O)CC2CC(C1)N(C(=O)CC(C)C(F)(F)F)C2 50661,c1(CC(=O)OC)c(N2CCOC(c3nc[nH]n3)C2)nnc(Cl)c1C 50662,CCC(C)(C(=O)N(CC(C)C(=O)N(C)Cc1n[nH]c(C)n1)C)OC 50663,CC#CCCC(=O)NCCCCN(C(=O)COc1ccc(O)cc1)C 50664,Cc1cn(C)cc1C(=O)NCCNC(c1ccnnc1S)=O 50665,c1(CN2CC3(N(C(=O)NCCCl)CC3)C2)cc(O)c(F)c(F)c1 50666,CCC(O)(CNC(=S)N)CC.C1(c2cccc(C)c2)CCN(C)C1 50667,C1(NC(c2c(CC)scc2)=O)CC(NC(=O)C(C)C)C12CCOCC2 50668,N1(C(CCCOC)=O)CC(N=[N+]=[N-])CC1C(N1CCC(CF)C1)=O 50669,c1(OCC)nc(Cl)ccc1C(c1nnnn1-c1ccc(Cl)cc1F)NCCOC 50670,c1(C2(C(=O)NCCc3ncc(Br)s3)CNC2)cccc(F)c1 50671,N1(C(COc2ccc(OC)cc2)=O)CC(NC(=O)C(F)C2CCC2)CC(O)C1 50672,CC(C)CC(F)C(=O)NCC1(C)CCCN(C(c2c(Br)cnn2C)=O)C1 50673,N1(C(C2N(Cc3c(OC)ncc(F)c3)CC(O)C2)=O)CCCC2(CCO2)C1 50674,CC(CC(=O)NCC(C)NC(c1cnc(C(F)(F)F)s1)=O)C1CC1 50675,CCC(C)(COC)C(=O)NCC(C)N(C(=O)CC1CCC=CCC1)C 50676,N1(c2n(CCC#C)c(-c3ccccc3Cl)nn2)CCc2cc(Cl)c(Cl)cc2C1C 50677,N1(C(c2cncc(N=[N+]=[N-])c2)=O)C2CCCC1CN(C(c1coc(Br)c1)=O)C2 50678,CCCCC(CNC(c1cccc(OC)c1)=O)NC(=O)CC1(OCCF)CCC1 50679,CC1CCN(C(=O)Cc2cnc(C(C)(C)C)[nH]2)C1C(=O)NCC1COCC1(C)C 50680,CC1CN(C(c2sc(C(F)F)cc2Br)C(=O)NC2CCC(F)(F)CC2)CC(=O)N1 50681,N1(C(c2cccc(C)c2)=O)CC2CC(NC(C3CC4CCC3CC4)=O)CC1C2 50682,N1(C(C(C=C)(C)O)=O)CC2CCCC(NC(=O)Cc3ccn(C)n3)C2C1 50683,N1(C(Cc2cc(C)[nH]n2)=O)CCN(C(=O)CCN2CCSC(C)(C)C2)CC1CO 50684,N1(CC(=O)OCCOC2(C)CC2)CCN(C(=O)Cc2cnoc2)CC1 50685,C(C)(CNC(C1(F)CCC1)=O)(CC(C)C)NC(CCOc1c(C)cccc1)=O 50686,C1(NC(CCCC#CC)=O)CCC(C)(C)CC1CNC(c1cnc(N)c(N)c1)=O 50687,C(C(=O)NCc1ccccc1Cl)(C(C)CCc1ccccc1)N(CCC)CC 50688,C1(O)(c2cn(CC(CC)O)nn2)CCN(C(=O)Cn2cccnc2=O)CC1 50689,C1(NC(c2cc(C)[nH]c2)=O)CC2CCC1N2C(=O)Cc1cccnc1 50690,N1(C(C(C)NC(C)=O)=O)CCC(NC(C2CC(O)CN2C(N)=O)=O)C(C)C1 50691,S(=O)(=O)(c1ccc(N)c(NC(C2CCCC(COC)O2)=O)c1)NCC 50692,C1(CC(C)NC(C(COC)O)=O)CCN(C(c2cncc(F)c2)=O)CC1 50693,C=Cc1ccc(C(N2CCC(C)C(NC(=O)CCC(C)(C)F)C2)=O)cc1 50694,c1(C(=O)NCC(C)N(C)C(c2ccoc2Br)=O)c[nH]cc(Cl)c1=O 50695,N1(C(c2c(C)cn(C)c2)=O)CC2(C1)CN(C(=O)Cc1cnccn1)C2 50696,C1(C(=O)NCCC2(C)CCN(C(C3CC(O)C(F)C3)=O)C2)CN2CCCN1CC2 50697,C1(C(=O)NCCNC(CC(C)F)=O)CC(c2cccc(Br)c2)=NO1 50698,c1(C(N(C(CCNC(C2N(C(C)=O)CCOC2)=O)C)C)=O)nccc2n[nH]cc12 50699,c1(C(=O)NC2CC(C)(COC)N(C(=O)CCSC)C2)cnc(O)c2ccsc12 50700,n1(C2CC(C(=O)O)C2)nnnc1C1(c2cc(C(=O)NCC3CCCC3O)cs2)CC1 50701,Cc1c(NC(=O)C(N2CC=CC2(CO)Cc2ccccc2)=O)cnn1C(F)F 50702,c1(CC(=O)NCC(C2CCCC2)N)cc(C)oc1C.C(C(=O)N)CCSC 50703,C1(C(C)C)N(C(=O)CN2CCOCC2)CC12CC(N)C(O)C2 50704,CCS(=O)(=O)CC(=O)N(C1CCCCC1NC(=O)C(O)CCc1ccccc1)C 50705,N1(C(C2(C)COC2)=O)CCC2C1CCCN2C(=O)C(F)(F)c1ccccc1 50706,C1(F)(C(=O)NC2CC(C#N)C2)CCN(C(=O)C(O)Cn2cncn2)C1 50707,CC1COC2(C1)CN(C(c1cnc(CNC(C3(C)CCC(O)CC3)=O)nc1)=O)C2 50708,C1(C)(NC(C(C)Cc2cnn(C)c2)=O)CCN(C(=O)CCC2CCCOC2)CC1 50709,Cc1sc(Cl)nc1C(N1CCN(C(C2CCCSC2)=O)CC1)=O 50710,N1(C(CN(C(C)C)C)=O)CCC2(NC(c3cc(F)ccc3Cl)=O)CC2C1 50711,C1(NC(c2cccc(C(=O)NC)c2)=O)CN(C(=O)CC2CN(C)C2)CCC1C 50712,C(C(C)C(F)C(=O)NCCc1cccnc1O)NC(C1(CC#C)CC1)=O 50713,c1(NC(=O)Cc2cccc(-c3cn[nH]c3)n2)cc(Br)cnc1O 50714,c1(C(N2C(C)CN(C(C3CC34CCC4)=O)CCC2)=O)noc2cc(F)ccc12 50715,CCCCC(F)C(=O)N1CC(O)(CNC(=O)C=Cc2ccc(C)s2)C1 50716,N1(Cc2c(C)noc2)CCC2(NC(c3ccnn3CC3CCC3)=O)CCCC12 50717,C1(C)(OC)CCN(C(C2C=CC(NC(c3cccc(Br)c3F)=O)C2)=O)CC1 50718,N1(C(C=C(C)C(C)C)=O)CCCC12CCCN(C(=O)CC1(O)COC(C)(C)C1)C2 50719,c1(OC)ccc(C(=O)N(CCCCN(C(=O)C(F)OC(F)(F)F)C)C)nc1N 50720,c1(C(=O)NC2CN(C(c3cn(CC=C)nc3)=O)CC(C)C2)cc(C)c(=O)n(C)c1 50721,N1(CCC=CCC)CCC(C2CCN(C(C3(C)CCS(=O)(=O)CC3)=O)CC2)C1 50722,N1(C(Cc2cccc(C)c2C)=O)CC2CCN(C(c3cn[nH]c3)=O)C2C1 50723,c1(C(=O)NCCC(C)N(C)C(c2ccnn2CC2CC2)=O)cc(C(F)F)ccn1 50724,c1(OC)cscc1C(=O)NC(C(N1CCCC1CN(C)C)=O)C1CCCC1 50725,c1(OC)ccc(CC(=O)NC2(C)CCCN(C(c3ccc(F)c(O)c3)=O)C2)cc1C 50726,C(=O)(CCC(CC)CCC)N(C(CNC(c1cc(OCC)ncc1)=O)C1CC1)C 50727,C1(C(=O)NCc2cc(C)ncc2)COCCN(C(=O)CN(C)C(=O)C2CC2)C1 50728,c1(CC(=O)N(C2CC(NC(=O)C=CCO)C2)C)ccc2c(c1)OCO2 50729,C(=O)(C1CCCc2n[nH]cc21)N1CC(CCCNC(CC=CCC)=O)OCC1 50730,CC(C)(CCC(=O)NC1CCN(C(c2ccc(Cl)cc2)=O)C12CCC2)[N+](=O)[O-] 50731,C(=O)(C1=C(C)OCCC1)NC(C)CNC(=O)C(C)ONC(=O)OC(C)(C)C 50732,c1(C(=O)NCCCC2(NC(C(CC)NC(N)=O)=O)CC2)nn2ccccc2c1C 50733,CC(C)(CC(=O)NCC1CN(C(c2csc(Cl)c2)=O)C1)C1CC1 50734,C1(O)(CC=C)CCN(C(=O)NCC2CCC2NC(=O)OC(C)(C)C)CC1 50735,c1(CC)cc(C(=O)NC2CN(C(C3(CO)CCCO3)=O)C2)ccc1C 50736,Cc1c([N+](=O)[O-])c(C(=O)NCC(C)(CO)NC(=O)CCC(C)(C)C)nn1C 50737,Cc1cc(C(=O)NC2CCCC(CNC(C3CNC(=O)O3)=O)C2)n(C2CCC2)n1 50738,CC(O)CC(=O)NC1CC(C)(NC(C2(c3cncs3)CC2)=O)C1 50739,N1(C(C(C2CC2)OC)=O)CCOCC(F)(CNC(C2C3CCC4C(C3)CC24)=O)C1 50740,CC(C)CCCCC(=O)NCC1CN(C(=O)CC2OCCC2(C)C)CC1C 50741,N1(C(CN(CC(C)(C)C)C)=O)CCC(C(=O)NOC2CCC(F)(F)C2)CC1 50742,N1(C(C(CC)SCC)=O)CCC12CN(C(=O)COCC1CCCO1)C2 50743,C=C(C)c1cccc(NC(C2CCN(C(c3cscn3)=O)C23CCC3)=O)c1 50744,C(=O)(CCCCC(N)=O)NCC1(C)C(C)CN(C(C(C)OCC)=O)C1 50745,C1(CC)CCCCN1C(=O)C(CCN(C)C)NC(=O)C(CN(C)C)CC 50746,N1(C(C(C2CC2)OC)=O)CCN(C(c2cnc[nH]2)=O)C(C2CCCC2)C1 50747,c1(C(=O)NCCN(C(c2cnn(CCF)c2)=O)CC)cc2cccc(C)c2nn1 50748,C(C(C)C(C)C(=O)N(C)CC1(O)CCN(C(c2cn(C)cn2)=O)CC1)OC 50749,C(=O)(C1=CCC(F)(F)CC1)NC12CCN(C(c3ccc(C=C)cc3)=O)CC1C2 50750,C1(N(CC(N2CC(OCC(=O)NC3CCCC3)C2)=O)C)CC2(CCC2)C1O 50751,C(=O)(CCCC(C)(C)C)N1CCC(C)CC1CNC(=O)CCc1cccnc1Cl 50752,C1(CC)CN(C(C23CC(F)(C2)C3)=O)CCC1NC(c1ccccc1O)=O 50753,N1(C(C2(C(=O)OCC)CC2)=O)CC(C(=O)NC(=O)CSCC)C2(CCCC2)C1 50754,CC(C)C(O)C(C)C(=O)N1CC(C)(NC(=O)CCc2ccc(F)cc2)C1 50755,CC1CN(C(C2(O)CCCC2)=O)CCC1CNC(c1cc(N(C)C)ccn1)=O 50756,n1(CC)nccc1-c1cn(CCCOCCNC(c2cnc(Cl)[nH]2)=O)nn1 50757,C(=O)(CS(=O)(=O)C1CC1)NC1C2(CN(C(c3c(C)cc(O)nc3)=O)C2)CC1 50758,c1(C(N2CCN(C(c3occ(OC)c(=O)c3)=O)C(C)C2)=O)c(C)ccc(F)c1N 50759,C1(CC=C)(N(C(=O)CC(=C)Br)CC)CCN(C(=O)C(C)(C)C2CCCCO2)C1 50760,C=C1CCN(C(C2CCN2C(C)(C)C)=O)C(C(=O)N(C(CCO)C(F)F)C)C1 50761,N1(C(=O)Cn2cc(C3CCCOC3)nn2)CCCC2(C1)C(O)CC2O 50762,N1(C(CCCC#C)=O)CC2CCC(C1)N(C(c1ncc(Br)cc1OC)=O)C2 50763,Cc1cc(F)c(S(=O)(=O)N2CCC3CC2(C(=O)O)CC3)cc1C(=O)O 50764,N1(C(CN(C(C)=O)C)=O)C(CC(N2CCC2C2CCCCC2)=O)C2CCCC12 50765,C1(C(=O)NC2CCN(C(=O)OC)CC2)CCC(C)(C)CC1 50766,N1(C(c2c(C)snc2)=O)CC(CCNC(C2CCC(CO)CC2)=O)C(C)C1 50767,CC(C(=O)NC1C2CN(C(=O)CCc3cccc(C(F)(F)F)c3)CC12)C(C)(F)F 50768,c1(C(=O)NCC2CC(NC(=O)C(=Cc3cccnc3)F)C2)ccc2nsnc2c1 50769,CCC(C)C(O)CC(=O)NC1C2CC(NC(C3(C#N)CC3)=O)CC12 50770,C1(CC)CN(C(=O)CN2CCC(O)CC2)CCN1C(=O)CNS(N)(=O)=O 50771,c1(C(=O)NC(CCNC(C(CC=C)C)=O)C)cnc2c(c1)N(C)CCO2 50772,c1(OC)ncccc1C(N1CCC(CC(=O)NC(C)(C)CN2CCCC2)C1)=O 50773,CCC(CC)C(=O)NCC1CC(F)(CO)C1.n12cc(nn1)C1CCCN1C(=O)C2 50774,C(CC(=O)N1CCn2ccnc2C1)(C(F)(F)F)NC(C(C(CC)C)=O)=O 50775,N1(C(Cc2nnc(C)o2)=O)CC2C(CN(C(=O)CSC(F)F)C)C2C1 50776,c1(C(N2CC(CNC(C3CC(OC)C3)=O)C(O)C2)=O)cc2cccnn2n1 50777,CCCCC(O)CC(=O)N1CC(C(=O)NC23CCC(CO)(CC2)C3)C(C)C1 50778,CCCC(CCCNC(c1cnc(OC)cc1C)=O)NC(c1cnccc1Cl)=O 50779,Cc1ccc(C(N2CC(C(N3CCCC3C(F)(F)F)=O)C2)=O)c(O)c1 50780,C1(C(=O)NC(CC=C)CNC(=O)CSS(C)(=O)=O)CC(=O)N(CC)C1 50781,C1(NC(C(CC)N(CC)CC)=O)CCN(C(c2cc(C)cs2)=O)C(C)C1 50782,c1(C(=O)NC2C(NC(c3ccc(C)n3C)=O)CCC2)cc(N)c2ncccc2c1 50783,CC1CCC(CO)CN1C(c1cc(CNC(c2ccoc2)=O)cs1)=O 50784,C(=O)(C(O)CCCNC(c1ccccc1)=O)N(CC)Cc1ccoc1 50785,CC1(C)CCCC(C(=O)NC(CNC(=O)CCc2ncco2)C2CC2)C1 50786,c1(C(=O)NCCC(=C)CNC(C2(OC)CS(=O)(=O)C2)=O)ccc(-n2cccn2)nc1 50787,C(c1cnccn1)=CC(=O)NCCCC1CN(C(=O)Cn2cnnc2)CCO1 50788,C1(C(N(C)Cc2ncco2)=O)CCC2(CC2)N1C(=O)C(F)CC1CCOC1 50789,CCCC(CCC)C(=O)NCC1CC2(CC2)CN1C(c1[nH]ccc1COC)=O 50790,Cc1c(C(=O)NC2(C#N)CCN(C(c3ccon3)=O)C2)cncc1Br 50791,N1(C(C)(C)C)CC(C(=O)NC2CCC(CNC(C3(CF)CC3)=O)CC2)CC1=O 50792,C1(C(=O)NCC(C(C)C)(C)F)CCCC(NC(C2CCCSC2C)=O)CC1 50793,N1(C(c2cc(C)on2)=O)CC(N(C)C(c2nn(C)cc2C)=O)C(F)C1 50794,C(=O)(C(CCF)NC(=O)CC=CC(C)(C)C)N(CC(O)CO)C 50795,N1(C(CNS(CC)(=O)=O)=O)CC(CO)C2(C1)CN(c1cc(C3CC3)ncn1)C2 50796,N1(C(CCCSC)=O)CC(NC(=O)C(C)(C)c2cccnc2)CC1C 50797,C1(C(N(C(C)C)CCNC(C2(CO)CC(F)(F)C2)=O)=O)CCCCCN1C 50798,C(=O)(C(O)C1=CCCCC1)N(CC(=O)NC(c1csnn1)C)C(C)C 50799,Cc1cc(Cl)nc(Cl)c1NC(C1CC(O)CCN1Cc1cc(F)c(F)cc1Cl)=O 50800,C1(C(=O)NC2CC(NC(c3ccc(C)cc3)=O)C(O)C2)CC2CCC(C1)C2(F)F 50801,Cc1cc(C)c(C(N2CC=C(CNC(=O)CC3CCOC3(C)C)CC2)=O)cc1N 50802,N1(C(CC2(C(=O)OC)CCC2)=O)CCN(C(c2cnoc2C2CC2)=O)CC(O)C1 50803,C(=O)(CC1CCCc2ccccc21)NC(CNC(C(CC#C)C)=O)(C)C1CC1 50804,c1(C(=O)NCCC(CC)(CC)NC(C2CCC(C#N)C2)=O)cc2ncccc2[nH]1 50805,CC(C)CC(CNC=O)CC(=O)N1CC(C)C(=O)N(C)C1 50806,c1(CNCC(C(=O)NC(CCC)C)N2CCCC2)ncccc1C 50807,c1(SCC)nc(C(=O)NC2CC(C)N(C(=O)CCC3CCCC3)C2)cc(=N)[nH]1 50808,CS(=O)(=O)CCC(=O)NCCCC1CCCN1C(=O)CCc1cncc(F)c1 50809,N1(C(C(C)SCCCC)=O)CC(NC(C2CN(C(=O)NCC)C2)=O)C2(CCC2)C1 50810,c1(CC)ccc(C(=O)NC2CCC(NC(c3ccc(C(C)C)cc3)=O)CC2)cc1 50811,C1(C(=O)NC2(CC=C)CN(c3nc4ccccc4o3)C2)CCc2nncn2C1 50812,c1(OC)ccc(CO)cc1NC(C12CC(CNc3cc(C)cc(Cl)c3)(C1)C2)=O 50813,Cc1c(CN(C(=O)CCCCNC(c2ccncc2)=O)C)cnn1C 50814,C#CCCC(=O)N(CCC(=O)NC1CCOC1=O)CCCO 50815,Cc1ccc(NC(C2CCCC2CNC(c2ccc(C(C)C)[nH]2)=O)=O)c(C)n1 50816,C1(CCOC)(C(=O)NC2CC(O)(CNC(=O)C(O)C3CCC3)C2)CCCC1 50817,C12(C(N3C(C)CC(CC(=O)NC4(CCC)CCC4)C3)=O)CCCN1CCC2 50818,C(CCC(C)C(=O)N(CCCCC(=O)N(C)Cc1ocnc1C)C)OC 50819,Cc1c(Cl)sc(Cl)c1C(=O)N(CCCN(C)C(c1cccc(=O)o1)=O)C 50820,Cc1cc(C(=O)N(CC(=O)NCC2CC(O)C23CCC3)CC2CC2)cnc1O 50821,N1(C(C)=O)CCOCC1NC(=O)C(C)N(C)C.C1(C2CNC(=O)N2)CCOCC1 50822,Cc1cc(C(F)(F)F)nn1CC(=O)NCCC1CCN(C(c2cncs2)=O)C1 50823,N1(C(C(C)NC(c2ccco2)=O)=O)CC(C)(C)CC1C(=O)NCC1(C)CC1(F)Cl 50824,C1(CC)C(C(N2CCC2(C)CCO)=O)CCN1C(=O)Cc1ccc(C)o1 50825,C1(CNC(C2(CC=C)CCCC2)=O)CN(C(=O)Cc2ccnc(O)c2)CCN1C 50826,C1(C2CCCO2)(C(=O)NCC2CC(C)N(C(=O)Cc3ccnn3C)C2)CCCO1 50827,C1(NCc2c(C)ncs2)CCN(C(=O)CC2(O)CCCC2)CC1C 50828,C(=O)(CC(=O)NCCC1(C(=O)NCCC(O)CO)CCCC1)N(C)C 50829,C(=O)(CC(O)C(=O)N1CC2CC2(CNC(c2coc(Cl)c2)=O)C1)OC(C)(C)C 50830,Cc1cnc(C(=O)NCc2nocc2C(=O)N(C2CCCCC2C)C)cc1C 50831,N1(C(CCC(C)(C)NC(=O)C=Cc2cscn2)=O)Cc2ccccc2C1 50832,C1(CNC(CN(C)C(N)=O)=O)CC(F)(F)CN1C(c1cccnn1)=O 50833,c1(C(=O)NCCCN(C)C)ccc2c(c1)CN(C(=O)C(=O)NCC(F)F)C2 50834,C1(NC(C(C)=C2CCC2)=O)CN(C(c2nn(C)nc2C(F)(F)F)=O)CCC1CO 50835,C(=O)(CCCCCC(C)O)NC1C=CCN(C(C(CC(C)C)O)=O)C1 50836,C1(C(=O)NCCCCNC(c2cn(C)nc2O)=O)CS(=O)(=O)CC1C(F)(F)F 50837,C1(C#N)(C(=O)NCC2CC(NC(C3N(C(C)=O)CCCC3)=O)C2)CCCOC1 50838,CN1CC(C(N2CCC(F)(C(=O)NCCC(F)=C(F)F)C2)=O)CC1=O 50839,N1(C(=O)C(F)=CCCF)CCCC(CCNC(C2(O)CCCC2)=O)CC1 50840,CC1CN(C(c2ccc([N+](=O)[O-])[nH]2)=O)CCC1NC(=O)CC12CCC(CC1)CC2 50841,c1(CC(=O)NCC2C(NC(c3ccncc3)=O)CC2)ccc(F)cc1C(F)(F)F 50842,c1(CC)conc1C(=O)NC(CNC(C1(SC)CC1)=O)C1CC1 50843,CCC(CC)CC(F)C(=O)NCc1ccoc1C(=O)N(CC(O)C(F)(F)F)C 50844,c1(C(=O)NC(c2c(F)cccc2F)C2CCCC2)cnc(O)c2ccsc12 50845,C1(C(N(C2CCOC2)CC)=O)CCC(NC(=O)C(C)=O)CC1 50846,N1(C(Cc2c(C)non2)=O)CCN(C(c2nnc(O)nc2O)=O)C(C)C1C 50847,C1(NC(CC(C2CC2)NC(C)=O)=O)CCCC(CNC(=O)C=C(C)C(C)(C)C)C1 50848,C(CC(C)C(=O)N(CCNC(c1cnc(O)o1)=O)C1CC1)=CCC 50849,C1(CCCC)CN(C(=O)CNC(=O)C(F)(F)F)CCN1C(C1CC(C(C)C)C1)=O 50850,CC(CCNC(=O)C(C)Cc1ccco1)CCNC(=O)CCc1cn[nH]c1 50851,N1(C(c2ccc(CSCCC)o2)=O)CC2=C(C1)CN(C(=O)C=C1CCOCC1)C2 50852,C1(C(=O)NC(CC(=O)OC)C)CCCCCN1C(=O)CN1CCCC1=O 50853,C(C)(CN=c1ccn2ncc(S(=O)(=O)NCc3ccccc3Br)c2[nH]1)OCC 50854,c1(OC)cnc(C(N2CCCC(NC(=O)CC3CN(C)C3)CC2)=O)c(OC)n1 50855,C1(NC(COCCC)=O)CC2(N(C)C(C3CCN3CC)=O)COC1C2 50856,C(C)(C(=O)N(CCCCC(=O)NC1CC(=O)N(C2CC2)C1)C)(C(C)C)OC 50857,c1(C(=O)NC(CC=CC)C(N2CCS(=O)C(C)C2)=O)ncc(F)cc1C 50858,CCC1=NOC(C(=O)NC(C)(C)CNC(c2ccc(C(O)CF)cc2)=O)C1 50859,c1(C(N2CCC(O)(C(C)NC(=O)C(C3CCCCC3)O)C2)=O)cc2sccc2s1 50860,C1(OC)CC(NC(c2cc(C)nn2C)=O)C12CCN(C(c1scnc1C)=O)CC2 50861,c1(OC)cc(C(=O)Nc2ncc(-c3ccc(C)nc3F)cc2C)cc(Cl)n1 50862,CC1(NC(c2ncoc2CN)=O)CCC(NC(=O)Cc2ccccc2)CC1 50863,CC1CC(CCNC(=O)CCCc2ccccn2)CCN1C(c1cccn1C)=O 50864,c1(C(=O)NCC2CCN(C(=O)C=Cc3cnc[nH]3)C2)coc2c1CSC2 50865,c1(C(=O)NCC2CC2NC(C2CCC2)=O)ccc2nc(O)nc(O)c2c1 50866,N1(C(C(COC)OC)=O)CCC(CCC(C)(C)NC(c2cnc(S)[nH]2)=O)CC1 50867,C1(CN=C(NCC(N(C)C)C2CC2)NC2CCOCC2)CCS(=O)(=O)C(C)(C)C1 50868,N1(C(CCOC)=O)CCCCC(N(C(=O)CC(C(C)C)c2ccccc2)C)C1 50869,C1(NC(CCc2ccc(C)s2)=O)CCN(C(C2CN(C(C)C)C2)=O)CC1 50870,Cc1c(O)ccc(CNC(C2(Cc3coc(C#N)c3)CCC2)=O)c1O 50871,O=C(CC(C(F)(F)F)NC(=O)CNC(=O)C1CC1)NC1(C2CCC2)CC1 50872,N1(C(CC(C=C)(C)C)=O)CCN(C(=O)CCC(CC)OC)C(C)C1C 50873,C(=O)(C(C(C)CC)N(C)C(c1ccc(SC)o1)=O)NCCSCCCC 50874,c1(SC)c(NC(C)=O)cccc1F.C1(C2CNC(=O)N2)CCCO1.C1(CO)CC1 50875,CN1CCC(C(=O)NCc2nc(CNC(=O)C3=CCCC3)cs2)S1(=O)=O 50876,Cc1cnc(NCC2CCCCC2NC(C2(O)CCOCC2)=O)nc1O 50877,C1(NC(CCCn2c(C)ncc2)=O)CC2(C(=O)O)COC1C2 50878,N1(C(COCc2cccc(C)c2)=O)CCC(CNC(c2ncnn2C)=O)C(O)C1 50879,N1(C(c2c(C)[nH]cc2)=O)CCC(O)(CCNC(C2CCN(C3CC3)CC2)=O)CC1 50880,CC(C)C(C)C(CNC(=O)C=Cc1ccoc1)NC(=O)CCCCCN(C)C 50881,c1(C(=O)NCC2CC(F)(CNC(CCC#C)=O)C2)cc([N+](=O)[O-])n[nH]1 50882,CC(C)C(C(=O)NC12CC1CN(C(=O)CN(C)C(=O)C1CC1)C2)NC=O 50883,C1(NC(CSc2cc(C)on2)=O)CC2CN(C(=O)C3=CCCO3)CC12 50884,C1(C(N2C(CNC(CC3CC(=C)C3)=O)CC(C(F)(F)F)C2)=O)CCCCC(=O)N1 50885,C12(C(=O)OC)CC(c3nnc(C(=O)NC(C)C(OC)OC)o3)(OC)CC1C2 50886,C1(C2CCOCC2)(C(=O)NC2CC(NC(C(C(C)C)OCC(C)C)=O)CC2O)CC1 50887,C(=O)(C(O)CC(C)(C)C)NCC(C1CCCC1)NC(c1cc(C)[nH]c1)=O 50888,C=C1CCN(C(c2nonc2N)=O)C(C(=O)Nc2cnc(F)nc2)C1 50889,C(=O)(CC1=CCCC1)OC(C(C(=O)OCC)=O)C 50890,c1(C(N2CCC(N(CC#C)C(c3cscc3OC)=O)C2)=O)oc(C)nc1C 50891,C(c1cc[nH]c1)=CC(=O)NCC(C1CCOC1)NC(c1cn(CC2CCCO2)nn1)=O 50892,c1(OC)cccc(NC(c2sccc2CNC(=O)N(C)C)=O)c1.C1(C)C(=O)N1 50893,N1(C(c2[nH]ccc2C2CCNCC2)=O)CCC(n2cn[nH]c2=O)CC1 50894,C1C(=O)N2CCCN(CC(F)(F)F)N2C(CO)CC(C)CC1 50895,CC1CCN(C(c2cnccn2)=O)CCN1C(c1cccc(=O)n1C)=O 50896,C1(CCCNC(=O)CSC(F)(F)F)CCCN1C(C1COCCO1)=O 50897,N1(C(C23CC(NC(c4ccc(F)c(O)c4)=O)(C2)C3)=O)CC2CCC(O)C(O)C12 50898,C(C(C)(CC(C)C)NC(c1ccc(C)c(O)n1)=O)NC(CCCC(C)=O)=O 50899,C1(C(=O)Nc2ccnc(CO)c2)CCN(Cc2ccc(O)c(F)c2F)CC1(F)F 50900,C1(CNC(c2ccc(CC)cn2)=O)CCC2(CCC2)C1NC(=O)C=C1CCC1 50901,CC(C)CC(CNC=O)CC(=O)NCC(C1CCC1)NC(=O)C(=O)C(C)(C)C 50902,N1(C(c2c(C)nc[nH]2)=O)CC(C)C(NC(=O)C=CCO)C(C)C1 50903,c1(CC)ccc(NC(=O)COCC(C)(C)C)cc1F.N12CCCC1C1(CC1)C2=O 50904,C(=O)(C1COc2ccc(Cl)cc21)N1CCC(CN(C)C(C2CC3CC3C2)=O)C1 50905,c1(C(=O)NC(CC)(CNC(C2(CO)CCCC2)=O)CC)cccc(N)c1Br 50906,c1(C(N2CC3(CCN3C(=O)C=CCF)C2)=O)cc(N2CCC2)cc(Br)c1 50907,CC(C)C(F)C(=O)NCCC1CCC(NC(=O)CC2CC=CC2)C1 50908,N1(C(c2cn(C)c(=O)cn2)=O)CCC(NC(=O)CNS(N)(=O)=O)CC(O)C1 50909,C1(N(C)C(c2c[nH]cc2Br)=O)CCCC(NC(=O)Cc2nc(C3CC3)cs2)C1 50910,C1(NC(C=C(COC)C)=O)CN(C(c2cc(CC(C)C)c[nH]2)=O)CC1N=[N+]=[N-] 50911,c1(C(=O)NCC(C(C)C)NC(C2COCCO2)=O)sc(N2CCOCC2)nc1Cl 50912,c1(NC(C(=O)NC(C2CCN(C(c3cc[nH]n3)=O)C2)C)=O)cc(Cl)ccc1Cl 50913,C=Cc1ccc(C(=O)NCC2(O)CCN(C(=O)CSc3nncs3)C2)cc1 50914,c1(CCC(=O)NC23CCN(C(=O)CN4CCOCC4)CC2C3)ccc(Cl)cc1Cl 50915,N1(S(CCC(=O)OCC)(=O)=O)CC2(CCN(S(=O)(=O)c3cnc(OC)s3)C2)C1 50916,c1(OC)cc(C(=O)NC(C)CN(C(=O)CC(C)SC)C)c(O)c(Cl)c1 50917,c1(C(=O)NC2(C)CN(C(C3(CC(C)C)CCC3)=O)C2)nn(C)c2ccccc12 50918,CCC(C)C(C)C(=O)N(CC(=O)NC1CCN(CCOC)CC1)CC 50919,c1(C(N2CC(O)CC(NC(CNC(=O)OCC)=O)C2)=O)cnc2c(c1)CCOC2 50920,Cc1ccc(C(=O)NC2CCN(C(=O)C(C)N(C)C)CC2(C)C)cc1[N+](=O)[O-] 50921,NS(=O)(=O)c1ccc(C(=O)N(CCC(F)(F)F)CCNC2CC2(F)F)o1 50922,C1(NC(N2CC(NC(=O)C(F)F)C2)=O)(Cc2cccc(F)c2)CCCCC1 50923,c1(NC(C)(C(c2ccc3c(c2)CCC3)=O)C2C(C)C2)nc(Br)c2c(F)cccn12 50924,C1(C(=O)NC2CN(C(CC3CCN(C)C3=O)=O)CC2(C)C)CC2(CCCC2)CO1 50925,C1(CN(C(=O)CCCOCC)CCN(C(=O)CSC(F)F)CC)CCCC(=O)N1 50926,c1(C(N2C(C)(C)CC(NC(=O)C(O)C3CC3)C2)=O)cc(N)cc([N+](=O)[O-])c1 50927,c1(NCc2scc(CNC(C(C)OCC#C)=O)n2)cc(C#N)c(F)cc1[N+](=O)[O-] 50928,N1(C(=O)Nc2c(OC)nsc2)CN(C)C(=O)N(C)C1 50929,CCCC(C(=O)OC)C(=O)NC1COCCC1NC(c1ccc2n[nH]cc2n1)=O 50930,c1(C(N2CC3CC(NC(CSCCC)=O)CC3C2)=O)cc2c(s1)CCC(C)C2 50931,CCCCC(O)CC(=O)NC(CC(F)F)C(=O)N1CCOC2CC12 50932,N1(C(c2c(CC)csc2)=O)C(C(=O)NCCOC(C)=O)CCC12CC2 50933,C1(C(N(C)Cc2cnc[nH]2)=O)CCCCC1(C)NC(=O)C(N)=O 50934,c1(NC(C2C(CNC(=O)C=CCF)C2)=O)ccc(Cl)cc1O 50935,CC1CN(C(C2(CC3CC3)CCCO2)=O)CCN1C(=O)CCc1cc(Cl)cs1 50936,c1(OCC(=O)OC)ccccc1CN1CCC(Cc2n[nH]cc2C(F)F)C1 50937,C1(NC(CCc2cc(C)no2)=O)(CO)CCCN(C(C2CC23CC(C)(C)C3)=O)C1 50938,c1(C(=O)NCC(CC)NC(c2ccc(C)n2C)=O)c(C)coc1C(C)(C)C 50939,N1(C(C)=O)CCN(C(C)C(=O)NC2CC(NC(C3CC34CC4)=O)C2)CC1 50940,c1(C(=O)NCC(CNC(c2cc(C)c(C)[nH]2)=O)C)ncc(Cl)cc1Cl 50941,N1(C(c2cn(CC)nc2)=O)CCN(C(=O)C(F)C(F)(F)F)CC1c1ccccn1 50942,N1(C(CC=C(C)C)=O)CCCC2(CCC(NC(=O)C=CC3(C)CCOCC3)C2)C1 50943,C=C(C)CC(C(=O)NCC)OCC(C(C)C)NC(=O)CN1CCOCC1=O 50944,CC1CN(C(=O)CCC#N)CCCN1C(=O)C1=CCCCCC1 50945,C1(C2CNC2)CN(C(C(C)(C)OC)=O)CCO1.C12(CCOCC1)C(F)(F)C(=O)N2 50946,C(CC(=O)N1CC(F)(F)C1)(C(F)F)NC(c1n(C)c(S)nn1)=O 50947,CCCS(=O)(=O)CC(=O)NC1CN(C(c2ccc(O)nc2)=O)CC1CO 50948,c1(OC)ccc(C(N2CC(NC(C3CC(OC(F)F)C3)=O)C(O)C2)=O)cc1 50949,c1(C(=O)NCC(F)CNC(C2CC(F)C(=O)N2)=O)cc2cccc(O)c2[nH]1 50950,c1(C(N2CC3C(CNC(C(CC=C)CC=C)=O)(C3)C2)=O)ncccc1S(C)(=O)=O 50951,C(=O)(C(C)S(=O)(=O)N(C)C)N1CCC(C(C)NC(CCC(C)SC)=O)CC1 50952,C=C1CC(CN(C(C(=O)OC)C2CN(C(=O)NC(C)(C)CC)C2)C)C1 50953,CCCS(=N)(=O)c1cccc(CNc2cccc(C#N)c2F)c1 50954,C=CC(CC)CC(=O)N(C1CCCC1)CCCNC(C12CCN(CC1)CC2)=O 50955,C=C(C)CCCC(=O)N1CC=CC(NC(C2(Cc3cccc(F)c3)CC2)=O)C1 50956,C1(C(N2C(C)CCC(NC(CN(CCOC)C)=O)C2)=O)CC2(C1)CC1(CCC1)C2 50957,CC1(C)CN(C(C2(S(C)(=O)=O)CC2)=O)CC(C)(C)C1NC(=O)C(F)CC1CCC1 50958,c1(C(N2CC(NC(C(CSCC=C)c3ccccc3)=O)C2)=O)[nH]c(C)cc1C 50959,N1(C(C(C#C)(C)C)=O)CCN(C(=O)CC2CCNC2=O)C(CC(F)(F)F)C1 50960,C(C(COC)C(=O)N1CCC(CCC(=O)NC2CC(OC)C2(C)C)C1)OC 50961,C(C(=O)NCCCCC(C)C)(C(C)C)NC(CCCNC(C)=O)=O 50962,Cc1cc(C(N2CCC(C3CC3)(NC(=O)C(=O)N(C)C)C2)=O)c(N)c(Cl)n1 50963,CC1CC(NC(=O)CCc2cnn[nH]2)CN1c1nnco1 50964,c1(CCCC)ccc(C(=O)NC(C)C(C)NC(c2ccsc2SCC)=O)cc1 50965,C1(O)(CC(=O)NC2C(C(=O)NCC(C(=O)NC)O)CCC2)CCCCC1 50966,CC1(C)C(NC(=O)C(CC2CC2)CC2CC2)C(C)(C)C1N 50967,C=CC(CC(=O)N(c1ccccn1)CCNC(=O)COCC)c1ccccc1 50968,Cc1ccnn1C(C)C(=O)NC1CCCCC1.C12CC(C1)CNC2=O 50969,c1cn2c(n1)C(Nc1cc(NCCCC3CC3)ncn1)CCC2 50970,N1(C(c2cn(C3CC3)nn2)=O)CCN(C(=O)CCN2CCCS2(=O)=O)C2CCC12 50971,C(CC)(C(=O)NC(C1CN(C(=O)CC2CC2C)C1)C)=CC 50972,N1(C(c2c(C)noc2N)=O)CCN(C(C2CCC(=O)N(C(C)C)C2)=O)C(C)C1 50973,c1(OC)cccc2c1CCCC2NC(=O)C(=O)NCC(c1ccc(F)cc1)(F)F 50974,c1(C(=O)NCC(F)CNC(C2CCCCO2)=O)ncc(C(F)F)cc1Cl 50975,c1(C(=O)NCC(CC(C)C)NC(CC2CC(CC)C2)=O)c(F)cncc1Br 50976,c1(C(N(CC(CC)NC(=O)C(C)SC)C)=O)nccn1C 50977,c1(C(c2ccccc2)CNC(CC)C2CC2)ccccc1Br 50978,C1(CC)CN(C(=O)CC2CC(C)C2)CCN1C(C1CN2CCN1CC2)=O 50979,c1(CCCC(=O)NCC2CC(OC)CN2C(=O)C(F)F)c(F)cccc1F 50980,N1(C(COCCC)=O)CCN(C(=O)CCc2cc(C)n(C)n2)CC2(CC2)C1 50981,CCCCCCC(C(=O)OC)NC(CCC(=O)OC)C(=O)O 50982,N1(C(C(C)(C)c2cncnc2)=O)CCC(CNC(=O)C(=O)Nc2ncc[nH]2)CC1 50983,C(Nn1cccn1)c1ncc(-c2n(C(C)C)ccn2)s1 50984,c1(C(N2C(C(=O)Nc3nccs3)CC(F)C2)=O)c(F)cccc1F 50985,C1(C(=O)NCC2(C)CCN(C(c3cnco3)=O)C2)(CC)CNC(=O)C1 50986,c1(C(=O)NC2CN(C(c3nc(C)nn3C)=O)CC2C)cnn2ccn(C)c12 50987,Cc1cccc(C(=O)C=CC(=O)NC(C)CNC(C2CC2C(F)F)=O)c1 50988,C#CC(N(C)N(C)Cc1ccc(-c2ccc(F)cc2)cc1)C1CC1 50989,Cn1cc(S(N)(=O)=O)c(C(=O)NC2CC(C)(NC(=O)CC3CCC(=O)N3)C2)n1 50990,CC(C)(C)C(CO)C(=O)N1CCCC1CN(C(=O)CCc1ncccn1)C1CC1 50991,CCCC(C)(CC)C(=O)NCC(C1CC1)NCC.c12cnc(c(Cl)c1)oc2=O 50992,N1(CCCNC(C)=O)CCC(C(=O)OCc2nc[nH]n2)C1 50993,Cc1c(C(=O)N(C)CCOCCCNC(C2(O)CC(F)(F)C2)=O)cccc1F 50994,N1(C(CCN(CC#C)C(C2CC2(F)Cl)=O)=O)CC(=O)NCC1C 50995,N1(C(CC(=C)C)=O)CCN(C(=O)COc2ccccc2C#N)CC1C1CC1 50996,C1(C(=O)NCCC(C)N(C)C(c2ccnc3[nH]nnc23)=O)CCOCC12CCC2 50997,c1(OC)ccc2c(c1)CCN(C1=NC=CC(=NC3CCN(C4CCCC4)C3)C1)C2 50998,C=CCC(C)(O)C(=O)NCCC(=O)N(C1CC(O)C1(C)C)C 50999,CCCC(CCC)C(=O)N(CC(N1CCC(C)(C)C1C)=O)C1CC1 51000,c1(OCCC)c(NC(c2ccn(-c3ccccc3)n2)=O)cccc1C 51001,c1(-c2cccc(CC)c2)c(C(=O)NCCc2cc3sccc3s2)[nH]c(C)c1CC 51002,C(C)(C)(CCC(=O)NC1CC(CO)C2CC12)NC(C(CC)NC1CCCC1)=O 51003,C1(CC)CC(C(=O)N(C2CCC2C)C)CCN1C(c1nn(C)cc1Cl)=O 51004,N1(C(C2=NOC(C)C2)=O)CCC(C2(NC(=O)C=Cc3ncc[nH]3)CC2)C1 51005,C1(OC)CN(C)CC1NC(=O)C=CCC(C)(C)NC(c1cnccn1)=O 51006,c1(C(C(=O)NCCOC)N(C)CCOCC2CCCO2)ccc(F)c(Br)n1 51007,C(=O)(CCCC(C)=O)NCC(CC=C)NC(=O)C=Cc1ccco1 51008,CC1(C)CCCC(C(=O)NCCC(C)(C)NC(C2C3CCCCC23)=O)C1 51009,C1(C(N(C)CC2N(CC)CCC2)=O)(COCC)CCCCC1.N1(C=O)CC(O)C1 51010,C(=O)(C(CC)C(C)C)N1CC(C=C)(C(=O)NC(CO)CC=CC)C1 51011,N1(C(c2n(CC=C)ccc2)=O)CCC(CC(C)NC(=O)Cc2[nH]cnc2C)CC1 51012,N1(C(C=CC(C)(C)SC)=O)CCN(C(=O)CCNC2CCCC2)C(CF)C1 51013,CCCC(C(=O)N(CCCN(C(=O)CCc1cc(C)sc1C)C)C)NC(N)=O 51014,Cc1nn(C)c2[nH]c(=O)c(CCC(=O)NC(C)CNC(=O)CC(C)(C)C)c(C)c12 51015,CC1COCCC1NC(=O)C(=O)N(CCCC1CC2CCC1C2)C 51016,CN1CCC(CCNC(=O)CC2C=CC(NC(c3cncn3C)=O)C2)C1 51017,Cc1cc(CC(N2CC(NC(C3COC(=O)N3)=O)C(C(F)F)C2)=O)ccn1 51018,C12(C(=O)NCC3C(C)(C)N(C(c4csc(F)c4)=O)CC3)CCC(N=[N+]=[N-])C1C2 51019,Cn1nnc2cc(C(N3CCCC(CCNC(=O)CC4CC4(C)C)C3)=O)ccc12 51020,C1(NC(c2c(COC)noc2)=O)C2CCN(C(c3ccoc3C3CC3)=O)CC12 51021,c1(CN(C)C)ccc(C(=O)NC2(CNC(=O)CC3CCOC3)CCC2)cn1 51022,C1(C(N2CCC(CCNC(c3ccc(C)s3)=O)C2)=O)C(Cl)(Cl)C12CC2 51023,N1(C(COC)=O)CC(NC(C2(C)CCC(=O)NC2)=O)CC(C)(C)C1 51024,C(=O)(CCCCCCC(=O)OC)NC1CN(C(C2C(CC)C2)=O)CC(F)C1 51025,Cc1ncc(C(=O)NCC(C)CNC(=O)CC(C)n2ccnc2)c(Br)c1Cl 51026,Cc1cccc2c1OC(C(=O)NC1CCCCN(C(=O)CCS(C)=O)C1)C2 51027,C1(C(N(CCNC(c2ccc(OC(C)C)nc2)=O)CC)=O)CCC(F)(F)C1O 51028,C(CN=C(NCC(=O)N(C)C)NCC1CCC(=O)N1)c1cccc(NC)c1 51029,C1(NC(C(c2ccc(C)cc2)C)=O)CCCC12CN(C(=O)Cc1cncn1C)C2 51030,CC(CC(=O)N1CCC(CNC(C2COCCOC2)=O)CC1)C(C)(C)C 51031,c1(C(=O)NCC2(OC)CN(C(c3nocc3C)=O)C2)n[nH]c(C(C)C)c1Br 51032,NS(=O)(=O)c1n[nH]cc1C(N1CC2CCC1C2NC(=O)Cn1cnccc1=O)=O 51033,CCCC(CCC)C(=O)NC(C)CN(C)C(c1onc(OC)c1Br)=O 51034,c1(C(=O)NC2CN(C(c3ccc(C(C)C)o3)=O)C3C2C3)cc(F)cc(F)c1 51035,c1(OC)ccncc1C(=O)N(C1CCN(C(=O)CCc2cc(Cl)cs2)C1)CCO 51036,c1(C(=O)NC(CNC(C2C(C)CC2)=O)(C)C)ccc(C(F)F)cc1Cl 51037,C(CN=c1ccc(Br)c(S(=O)(=O)NCc2c(F)cc(Br)cc2F)[nH]1)C1(C)CC1Br 51038,Cc1ccc(SCC(=O)NCC2CC(O)(CNC(=O)C(C)NC(N)=O)C2)c(Cl)c1 51039,CC1CN(C(C2C(F)(F)C23CCC3)=O)CCC1CNC(=O)CC1OCCC1(C)C 51040,C1(OC)CCC(CC(=O)NC(C)CNC(c2sccc2CC#N)=O)CC1 51041,C(C)(C)(C(=O)NCCCC1(NC(=O)CC2CC(F)C2)CC1)OCC 51042,C1(C(=O)NCC2N(C(Cc3nn(C)c(C4(Cl)CC4)c3)=O)CC2)C2CC3C(C2=O)C13 51043,CC1Oc2ccc(C(=O)NCC(C)NC(c3cc(C(C)(F)F)on3)=O)cc2C1C 51044,N1(C(CN2CCC(C)C2)=O)CC2CCC1CN2C(=O)C(C1CCCCC1)O 51045,CC1CN(C(c2nc(C(F)(F)F)cn2C)=O)C(C(=O)O)CC1C 51046,c1(CC(=O)NCCN(C)C(C2CC2(C)C(F)F)=O)cnn(C)c1 51047,C(=O)(C1CCc2c[nH]nc21)N1CCC(C(C)NC(c2cnsc2)=O)CC1 51048,C12N(CCCC1(C)C)C2=O.C12CCc3cnn(c3C1)CC1CCN2CC1.COOC 51049,C#CCC(CC#C)C(=O)NCC(CO)NC(=O)CNC(=O)Nc1ccccc1C 51050,CC(C(=O)N1CC(NC(C2CNC(=O)N2C)=O)C(C)C1)C(C)C1CCCCC1 51051,c1(CCCC)ccc(C(c2nnnn2C)NCCc2csc(C)n2)cc1 51052,C(C(=O)NCC1(NC(c2c(Cl)cnn2C)=O)CCC1)(C(C)C)SC 51053,C1(C2CCN(S(=O)C3CC4C(C3)C4(F)F)CC2)(C(=O)O)CC(F)(F)C1 51054,N1(C(=O)NCCOC(=O)OC2CCCC2)CCN(c2ccccc2)C(=O)C1 51055,c1(C(=O)NC(CNC(c2ccc(SC)cc2)=O)C2CC2)cncc(Cl)c1C 51056,Cc1ccc2c(=NC(C)c3nccs3)[nH]c(=NCc3c(F)cccc3Cl)[nH]c2c1 51057,CC1CN(C(c2cccc(C(N)=O)c2)=O)CCCN1C(c1ccc(Cl)s1)=O 51058,N1(C(CC(C)C(F)F)=O)CCC2CCCC12C(=O)NCCC1CCC1 51059,CCC(F)(F)C(C)(C)C(=O)N1CC2CC1CN2C(c1ccc2oc(C)nc2c1)=O 51060,c1(C(N2CCN(C(=O)CCn3ccnn3)C(CF)C2)=O)ccc(O)cc1Cl 51061,C12(C(=O)NC3CC(CNC(c4ncc(OC)cc4F)=O)C3)CCCCC1OCC2 51062,C#CC1CC2CCC1N(C(C1CCN(C(=O)CCC3CCCN3C)C13CC3)=O)C2 51063,c1(C(N(CCNC(C23CCC(C2)C3C(=O)O)=O)CC)=O)ccc(CO)c(Cl)c1 51064,c1(CNC(CC2(OC)CN(C(c3cnnn3C)=O)C2)=O)cc2ccccc2[nH]1 51065,c1(C(N(CC)CC2CCCN2C(C2OCCC2C(C)C)=O)=O)cccc(=S)n1O 51066,CC(C)(C(=O)NCCN(C1CCCC1)C(C1OCCOC1C(F)(F)F)=O)C(N)=O 51067,N1(C(CCC=C)=O)CCN(C(=O)C(c2ccccc2F)C)CC1CCO 51068,CCC(C)(COC)C(=O)N1CC(C2CC2C(N2CCOC(CCO)C2)=O)C1 51069,N1(C(CCP(C)(C)=O)=O)CC(CNC(=O)Cc2cc[nH]c2)CC12CCC2 51070,c1(OC)ccc(Cl)cc1CC(=O)N(C1CC(NC(=O)CC2(O)CCCC2)C1)C 51071,c1(C(=O)NCC(C)(O)CNC(=O)Cn2cnnc2)cc2c(F)cccc2[nH]1 51072,C1(CCC)CN(C(c2oc(CO)cc2C)=O)CC1NC(c1ccsc1SC)=O 51073,N1(C(CCC)=O)CCN(C(c2cc(C)nn2C)=O)C(CCO)C1 51074,C1(C(=O)NCC(CNC(=O)CN2CCS(=O)(=O)CC2)O)CC2C=CC1C21CC1 51075,c1(C(N2CC(CNC(C(C(CC)O)(F)F)=O)C2)=O)cc2ccccc2c(=O)n1C 51076,CC1CCN(C(C2CNC(=O)O2)=O)CCN1C(c1ccnn1CC(F)F)=O 51077,N1(C(c2ccc(C(CC)=O)cc2)=O)CCN(C(c2coc(C)n2)=O)CC1C1CC1 51078,Cc1ccc(C(=O)NCC(=O)NCCOCC(C)(C)O)c(F)c1 51079,c1(C(N2C(CN(C(=O)Cn3nnc(C)n3)CC)CCC2)=O)cc(C)nc(O)n1 51080,N1(C(CC=CC=C)=O)CCCC(N(C(=O)CCOc2cccc(C)c2)C)C1 51081,C1(C#N)(C(N(CC(C(=O)NC(CCOC)CO)C)C)=O)CCCOC1 51082,N1(C(C(C)(C)C)=O)CCC2CCCC12C.C(=O)(CCF)NC1(NC(CN)=O)CC1 51083,CCC(C)(C)CC(=O)N1CC(N(C(=O)C(C)OC)C)C(O)C1 51084,C1(CNC(C=CC=CCC)=O)CN(C(=O)C(=O)NC(C)C)CCC1C 51085,N1(C(CCN(CC)CC)=O)CCCN(C(c2sc(S(N)(=O)=O)cc2C)=O)CC1C 51086,N1(C(C2C(NC(c3c(COC)onc3)=O)CC=CC2)=O)CC(C)N(C)C(C)C1 51087,N1(C(CNS(CCCC)(=O)=O)=O)CCc2nc[nH]c2C12CCN(C(=O)C(N)=O)C2 51088,c1(NC(=O)NCC=CCCOC)cnc2ccccn2c1=O 51089,Cc1ccc(C)c(C(=O)NCc2nocc2C(=O)NCCCO)n1 51090,c1(CN(C(C(=O)OC)CC2CCOC2)C(C(C)CCC(C)C)=O)ccc(F)cc1 51091,C1(CC(=O)NC(C)CCCCNC(c2ccsn2)=O)CCC(=O)NC1=O 51092,c1(NC2CC(C)N(C(c3cc([N+](=O)[O-])c[nH]3)=O)CC2)ncc2c(c1C#N)CCC2 51093,C1(C)(C(=O)Nc2cc(NC(C3C(NC(=O)OC(C)(C)C)C3)=O)[nH]n2)CNC(=O)C1 51094,c1(C(N2CC(CNC(C(C)c3ccsc3)=O)C2)=O)ccc(-c2ccco2)o1 51095,N1(C(C2C(C)(CC)C2)=O)CCC(N=c2cc(C(=O)OC)nc(Cl)[nH]2)(CO)CC1 51096,Cc1cc(O)ncc1C(=O)N(CCCN(C(=O)CC1CCC(=O)N1)C)C 51097,N1(C(C(C)C(C)(F)F)=O)CC2(COC(CNC(=O)C(C)N(C)C)C2)C1 51098,Cc1ccc(C(N2CCC(C(N3CCC(C)(C(N)=O)CC3)=O)(CO)C2)=O)nc1C 51099,N1(C(=O)Nc2cn(C(=O)OC(C)(C)C)nc2)Cc2ccccc2OC(C)C1 51100,C1(C(=O)OCC)CCCN(C(C2(C)CCN(C(C3CC3C(N)=O)=O)C2)=O)C1 51101,Cc1ccc(C(=O)NC(C)CN(C(=O)C(C(C)O)N(C)C)C)cc1I 51102,c1(C(C)C)cc(C(=O)NC2CCN(C(c3ccc([N+](=O)[O-])[nH]3)=O)C2)cc(Br)c1 51103,C1(NC(=O)C(F)CC2CC2)CN(C(=O)C=CCOc2ccccc2)CC(F)(F)C1 51104,CC(C)(CCNC(=O)C(O)C1CC1)NC(C1C(c2ccccc2)C1(F)F)=O 51105,C1(C2(O)CCC2)(C(=O)NCC(C)NC(C2CC3CC2C3)=O)CC1 51106,c1(CC)cnc(C(=O)NCC2(NC(C3CCC34CCC4)=O)CCCC2)cn1 51107,N1(C(=O)C(c2cccnc2)O)CC2CC(C(N3CCCC4CC34)=O)(C2)C1 51108,c1(C(N2C3C(NC(C(C(CC)CC)C)=O)C(C3)C2)=O)nc(N)cc2ccccc12 51109,N1(C(C(CC)(F)F)=O)CCC(C)C(NC(c2ccc(CNC(C)=O)o2)=O)C1 51110,C1(NCC2CCCN(C(Cc3c(C)cccc3)C)C2)CCC2CC2CC1 51111,C1(OC)(NC(c2cc(Br)ccn2)c2nnnn2Cc2cccs2)CCOCC1 51112,C1(NC(C(CC#C)O)=O)C2CCN(C(C3C(C(=O)OC)C3(C)C)=O)CC12 51113,c1(OCC)ccc(NC(c2nc(C)c(C)o2)c2nnnn2C2CCOC2)cn1 51114,CC1(C)CN=C(N2CCN(S(C)(=O)=O)CC2)S1.c12ccccc1CN2 51115,c1(C(=O)NC(CC=C)CNC(c2cnc(C)n2C(F)F)=O)cnc(CO)nc1C 51116,CCC(C)C(CN(C)C)NC(=O)Nc1ncccc1C(F)(F)C(F)(F)F 51117,N1(C(c2ccc(NCC)cc2)=O)CCCC(C)C1CNC(c1ccccc1)=O 51118,c1(-c2ccc(C(=O)NC(CNC(C3CCSC3)=O)CO)s2)cccc(F)c1 51119,C1(C(=O)NCC(CN(C(COCC(C)C)=O)C)C)CCC(N(C)C)CC1 51120,C1(C(N2C(C)CN(C(c3csc4nccn34)=O)CC2)=O)CCCC2CCCN12 51121,C1(CC(=O)NCC2(O)CN(C(Cc3cnn(C)n3)=O)C2)CC2C=CC1CC2 51122,C1(CC(=O)NCC2CC(CNC(C=CC(C)C)=O)C2)CN(C)CC1O 51123,O=C1NC(Sc2ccc(O)c(Cl)c2)C(=O)N1CCCc1ccc(Br)cc1 51124,C1(C(=O)NCCn2cc(NCCO)nn2)CC2CCC1C2 51125,CC(=O)N=c1nc(C2CCN(C(C3CCN(C(=O)C(C)C)CC3)=O)CC2)[nH]n1C 51126,N1(C(C=Cc2c(OC)cccc2)=O)CCCC(C)(NC(c2scnc2C)=O)C1 51127,C(C)(CCC(=O)NCCCCCO)NC(C1ON=C(C)C1)=O 51128,N1(C(C2CC2F)=O)CCC2(CCN(S(=O)(=O)c3ccc(Br)cc3)CC2)C1 51129,c1(NC(C(=O)NC2C(NC(C(C)(C)O)=O)CCOC2)=O)ccc(C#N)c(Cl)c1 51130,Cc1cccn2cc(C(=O)NCCC3CCN(C(C4CCO4)=O)CC3)nc12 51131,C1(C(N(CC(C)NC(=O)C(C)(C)N(C)C)CC)=O)CCC(O)CN1C 51132,Cc1ccc(C(C)C(=O)NC2(CN(C)C(c3nc[nH]c3C(F)(F)F)=O)CC2)cc1 51133,C1(C(C)NC(c2ccc(C)o2)=O)CN(C(=O)CC23COCC(C2)C3)CCO1 51134,c1(OCC)cc(NC2CCCC(CNC(C3(C)CNC3)=O)C2)ncn1 51135,C1(C(=O)NC(CC=CC)CO)CN(C(c2cc(C(F)F)[nH]n2)=O)C(C)(C)C1 51136,C1(NC(CC(C)C2CCCO2)=O)CCC(C)N(C(=O)Cc2cnn(C)n2)C1 51137,N1(C(CCCc2onc(C)n2)=O)Cc2nccn2CC(NC(=O)C(C)(F)F)C1 51138,O(NC(=O)C(c1ccnn1C)c1ccoc1)CCOCCOCC 51139,Cc1nccn2c(C(N3CCNC(=O)C3c3ccccc3Cl)=O)cnc12 51140,c1(C(=O)NC(CNC(C(CC=C)C)=O)CO)cccc2[nH]c(C)cc12 51141,c1(NC2(C3CCCO3)CCC2)ccc(Br)c(S(=O)(=O)N2CC(CCC)OCC2)n1 51142,c1(C2(NC(=O)NCc3cc(Cl)cs3)CC2)ccc(F)c(F)c1 51143,N1(C(C)C)CCCC(O)(Cc2nc(C3CCC3)ns2)C1.N12CCC(CC1)C2=O 51144,N1(C(CN(C2CCSC2)C)=O)CCOC(CCCNC(=O)C=CC=C(Cl)Cl)C1 51145,C1(CNC(C(c2ccccc2F)C)=O)COC(C)(C)CN1C(=O)C(O)C(F)(F)F 51146,C12CCCCC1C(=O)NC2.n1(CC)nncc1-n1ccc(C(C(=O)NC)(C)C)n1 51147,C(=O)(C1=NOC2(CCC2)C1)N1CC(C)C(C(=O)NC2(c3nn[nH]n3)CC2)CC1 51148,N1(C(C(F)=C(C)C)=O)CC(C2CCCCN(C(C3CCc4n[nH]cc4C3)=O)C2)C1 51149,c1(CC)cc(C(N2CC(F)(CNC(=O)Cc3cc(C4CC4)no3)C2)=O)nn1C 51150,C1(C(N2CCC(c3scc(CC)n3)CC2)=O)CCN(C2CC2)C1(C)C 51151,C(=O)(C1=CCOC1)N(c1ccccc1)CC.CC1CNC1=O.C(C)(C)(C)O.C1(=O)OC1 51152,c1(C2C(NC(C3NCCC3C(F)(F)F)=O)C2)ccc(Cl)cc1 51153,c1(C(=O)NCCN(C(=O)C(O)C(C)SC)CCCCCC)cnc(N(C)C)nc1 51154,C1(C(=O)NC2C(NC(c3cscc3C3CC3)=O)CC2)CCS(=O)(=O)N1 51155,c1(C(=O)NC2(COC)CCCN(C(=O)CC(C)F)C2)ccc(C)c([N+](=O)[O-])c1 51156,C(=O)(C1=CC2C=CC(C1)C2)NCC1C(C(N(CC(C)(O)C2CC2)C)=O)C1(C)C 51157,c1(NN)cccc(CCC(=O)NCC2CCCN2C(=O)CCF)n1.C(F)(F)F 51158,C1(NC(c2c(C)ccc(Cl)c2)=O)COC2(C1)CN(C(=O)C(c1ccccn1)C)C2 51159,Cc1cccc(C(C)C)c1-n1nc(CC2CC2)nc1C(c1cnn(C)c1)C 51160,C1(C(=O)NCC(=O)N(CC)CC)CCN(C(c2n[nH]c(C(C)(C)C)n2)=O)C1 51161,c1(C(N2CC(C)C(NC(=O)Cc3cnn(C)c3)CC2)=O)ccn2nccc2n1 51162,C(C)(C)(CC(F)C(=O)NCC1CCOC(C)(C)C1)NC(C(C(=O)OC)OC)=O 51163,CN1CCN(C(=O)CN2CCCC2=O)CC1C(=O)NOCc1ccncc1 51164,C1(C(N2CC(O)(CCNC(C(C)SC(F)(F)F)=O)C2)=O)CC2(C1)CC2(F)F 51165,CCCC(C)(O)C(=O)NCC1CCC1NC(c1ccc(N)c(CC(C)C)c1)=O 51166,CC1CC(NC(=O)CC2CCN(C(C3CC(F)CN3)=O)C2)C(=O)O1 51167,N1(C(C(=O)NC2CC(CSCC)C2)=O)CCC(CNC)C(F)(F)C1 51168,CN1CCC(C)(CNC(=O)COC2CCN(C(=O)CSCC(F)F)CC2)CC1 51169,C=CC(CC)CC(=O)NCC1CCN(C(c2cc(C(F)(F)F)ccc2O)=O)C1 51170,c1(OC)c(C(=O)NCC(C2CCCC2)NC(c2c(Cl)cnn2C)=O)ccnc1Cl 51171,Cc1ccnc(O)c1C(=O)N(CCNC(C12CCCCC1C2)=O)C1CC1 51172,Cc1c(C(N2CC(F)(C(=O)NC3(C)CCCC3(F)F)C2)=O)cccc1O 51173,C=CCCCC(C(=O)NCCCCC(C)(F)F)NC(C1C2CCCCC12)=O 51174,c1(C(N2CCC(N(C(C(CCC)F)=O)C)C2)=O)nccc(OC)c1C 51175,C(CCCCC(=O)NCCC1(O)CCN(C(=O)CCn2ccnc2)C1)NC(N)=O 51176,C1(C(=O)NC(C2CN(C(c3ncoc3-c3ccon3)=O)C2)C)C(C)(C)C1(C)C 51177,c1(OC)ccccc1C(CNC(C1CCC2CC12)=O)NC(C12CC(CO1)C2)=O 51178,C=CC1(CC(N2CCC(C(C)C)CC2)=O)CN(C(C2CCCN2C(C)C)=O)C1 51179,C(=O)(CC(C)CNC(C1CC(NC(=O)C(CC2CC2)OC)CCO1)=O)NC 51180,CCCS(=O)(=O)CC(=O)NCC(C)(O)CNC(C1CC2(CCC2)CO1)=O 51181,N1(C(c2c(C)nc(N)cn2)=O)CCC2(CCC(NC(=O)C#CC3CCOC3)C2)C1 51182,c1(CC)ccc(CC(=O)NC(CNC(c2cc(=O)n(C)cn2)=O)C2CC2)cc1F 51183,C1(CNC(C(F)=CCC)=O)CC2CCCC(C1)N2C(=O)C=C1CCCCC1(C)C 51184,c1(C(N2CC(CNC(C(C=C)O)=O)OCC2)=O)ccc(C)c(S(=O)(=O)CCO)c1 51185,Cc1ccc2cccc(C(=O)NCC3CN(C(c4cc(C(F)F)cs4)=O)C3)c2n1 51186,N1(C(C(CC=C)CC=C)=O)CC2COCCC2(NC(c2ccc(Cl)nc2N)=O)C1 51187,c1(CNC(CC2OCCN(C(C3CC(C)(F)C3)=O)C2)=O)ccc(F)c(O)c1 51188,N1(C(c2cncnc2)C(=O)NCCCCSCC)CCC(C2CCCC2)C1 51189,C(C(CC)CO)NC(C1(C(C)NC(COCCC=C)=O)CC1)=O 51190,c1(NC(CN2CCC(OC)C2)=O)sc(C)nc1C.C1(=O)C(C)CN1 51191,CCCCC(O)CC(=O)NCC12CCCN1C2=O.c1(CSC)ccc(F)c(O)c1 51192,c1(-c2nc(NC(C(C)SC3(F)CCS(=O)(=O)C3)=O)sc2)ccc2c(c1)OCO2 51193,C1(C)(C(=O)NCC(CNC(C2(CC#C)CCCC2)=O)O)Cc2ccccc2N1 51194,C1(C(N=S(C)(C)=O)=O)CCCC2(CCCC2)O1 51195,CC1CN(C(c2nn(C(C)(C)C)cc2Cl)=O)CCN1C(C1CC(=O)NC1(C)C)=O 51196,c1(OC)c(F)cc(Br)c(CS(C)(=O)=NC(=O)c2c(F)cccc2Br)c1F 51197,c1(C(=O)NCC(C2CC2)NC(c2cnns2)=O)cc([N+](=O)[O-])c2nsnc2c1 51198,c1(OC)nccc(C(N2CC(OC)CC2)=O)n1.C(CN(C)C)(CO)NC=O 51199,Cc1nn(C)cc1C(=O)NC1CC(NC(=O)C(C2CCCCCC2)C)C1 51200,c1(C(=O)NC2CCC(NC(C(N3CCCCCC3)C)=O)C2)cncc(N)n1 51201,c1(N(C2CCCOC2)C)cc(Br)ccc1S(=O)(=O)NC1(C2CC2)CC1 51202,Cc1cccc(CN2CCC(C)(CN)C2)c1Br 51203,N1(C(C=NOC)=O)CCCCC1CNC(=O)CC(C)O 51204,C(C(CC(=O)NC(CC1CCC1)CO)NC(C1(C)COC1)=O)OC 51205,C1(C(=O)NCCCCC(C)NC(C2(C(=O)NC)CCC2)=O)C(F)(F)C12CCC2 51206,c1(C(N(CCCCNC(C(C(CC)C)O)=O)C)=O)cc2ncn(C)c2cn1 51207,CCC(COC)C(=O)NC1CN(C(c2ccc(-c3csnn3)cc2)=O)CC1O 51208,C(=O)(C(F)C(C)(C)O)NCC1C(C)CN(C(=O)C=CCN2CCCC2)C1 51209,C1(C(NOC(c2nc[nH]n2)C)=O)N(C(c2csnn2)=O)CCCC1(C)C 51210,N1(C(=O)CCc2ccccc2)CCC(C2CCCN(C(c3ccco3)=O)C2)C1 51211,Cc1sc(C(F)(F)F)nc1C(=O)NC1CCC(NC(=O)C(C)C(F)F)C1 51212,c1(C(=O)NC2CC(CNC(C3(C)N(C)CC(O)C3)=O)C2)ccc2nc(=N)[nH]n2c1 51213,C1(NC(c2n(C)ncc2)=O)CC2CN(C(=O)Cc3c(Cl)cnn3C)CC12 51214,C#CCC(C)(C)C(=O)NC1CC(NC(=O)C(c2cnn(C)c2)C)C(O)C1 51215,C1(C(=O)NCC2C(NC(C3CC(C(C)(C)O)C3)=O)CCC2)CCc2nc[nH]c2C1 51216,CCCCCCCCC(C)C(=O)NC(C1(O)CN(C(c2cccnc2O)=O)C1)C 51217,N1(C(c2c(C)nsc2)=O)CCC(NC(C2(c3ccc(F)cc3)CC2)=O)C(F)C1 51218,Cn1cc(C(C(=O)NCC2(F)CCC2)NC(=O)CC2(O)CCC2)nn1 51219,N1(C(CCOCC#C)=O)CC(CNC(c2c(NC(C)=O)c[nH]c2C)=O)CC1C 51220,c1(C(=O)NC(CC(=O)N2CCC(CC#C)C2)COC)coc2c1COC2 51221,c1(NC)ccc(F)cc1C(=O)NC1CC(NC(C2CC2OC(C)(C)C)=O)CC1O 51222,N1(CCCCCC=C)CCC(O)C(C(N2CCOC(CC(N)=O)C2)=O)C1 51223,C1(O)(CNC(c2c(C)coc2)=O)CCN(C(c2cc(Br)ns2)=O)C1 51224,N1(C(CCC(C)N(C)C)=O)CCCCC(CNCc2cccc(Br)c2)C1 51225,CCCC(O)C(=O)NCC1(CNC(=O)C(C)SC)CCOCC1 51226,N1(C(Cc2n(C)ncc2)=O)CC2CC(O)C1C2NC(c1ccc(CO)cc1F)=O 51227,c1(C(=O)NC2C(C#N)CN(C(c3ccno3)=O)C2)ccc2ccccc2n1 51228,CCC(CC(=O)NC(C(=O)N1CC(NC(N)=O)C1)C1(C)CC1)C(F)F 51229,C1(CNC(COC2(C#C)COC2)=O)CN(C(=O)CC2C(C)(C)C2(C)C)CC1(C)C 51230,N1(C(C(C)C2CCC2)=O)CCCC(C2CN(C(c3cccc(C4CC4)n3)=O)C2)C1 51231,N1(C(C2COCCN(C(c3c(CC)ncs3)=O)C2)=O)CCCc2ccccc21 51232,c1(C(N2CCC(NC(c3n(C)ccn3)=O)C(F)C2)=O)cncc2[nH]ccc12 51233,C1(OCC(=O)NC2(CO)CN(C(c3cnc(CC4CCC4)s3)=O)C2)CCCOC1 51234,C1(C(C)(C)C)CC(C(=O)N2CC(CNC(=O)CCC3CC3)C(C)C2)=NO1 51235,c1(C(=O)NC2(c3ccccc3)CCN(C(c3c(C)nc[nH]3)=O)C2)ccc(N)cc1Cl 51236,c1(C(=O)NCC2(F)CCN(C(C3CCOCC3)=O)C2)ccc2c(=O)ccoc2c1 51237,C(=O)(C#CC1(C)CCCO1)N1C2CC(CN(C(C3CCCN(CCC)C3)=O)C2)C1 51238,c1(C(=O)NCCCCC2CN(C(C(C(CC)O)C)=O)C2)ccc2nnc(O)n2c1 51239,c1(OC)cc(CN2CCCC2CC(N2CCC(CO)CC2)=O)ccc1O 51240,N1(C(C2(NC(CNC(CC)=O)=O)CCN(C)C2)=O)CCCN(C=O)CC1 51241,c1(CC)noc2ncc(C(N3CCN(C(C4CCC=CCC4)=O)C(C)C3)=O)cc12 51242,c1(C(=O)NC2CCN(C(C3OCCN(C)C3)=O)C2)ccc2c(n1)OCC(=O)N2 51243,S(=O)(=O)(C1CN(C(c2nccn2C)=O)C1)N1CCN(C(C2C(C(C)C)C2)=O)CC1 51244,C(=O)(C(C#N)C(C)C)N1CCC(C(C(=O)NC(c2nccn2C)CC)F)C1 51245,C(=O)(CCCCCN)C(C(C(=O)C1(C(C(=O)NCC)OCC)CC1)OC)=O.OC 51246,c1(NC(CC=CC)=O)cc(C(=O)OC)ccc1C 51247,N1(C(c2c(CC)nco2)=O)CCOC(CCNC(=O)C(C)CF)C1 51248,c1(OC)cccc(C(=O)NC(C2CCN(Cc3cnc(C)s3)CC2)C)c1O 51249,C1(C(=O)NC(C(C)NC(C(CC=C)(F)F)=O)CO)CN2CCN1CC2C 51250,Cc1nc(N(C)C(c2ccc(F)c(F)c2)C)ncc1Br 51251,C=CC(CCC)CC(=O)N1CCOC(C)C1C(N1CCC(OCC)C1)=O 51252,S(=O)(=O)(c1ccc(OC2CCOCC2)cc1C)NCCc1c(C(N)=O)cccc1 51253,N1(C(c2n(CC)nc(Br)n2)C(=O)NC(C)(C)CC)CCC(C)(C)CC(C)(C)C1 51254,N1(C(c2cc(CC)[nH]n2)=O)CC(CNC(=O)C(CC2CC2)OC)CC(C)C1 51255,c1(OC)cc(N)c(F)cc1C(=O)N(C)CC1CCCN1C(C1C(C)C1C)=O 51256,Cc1ccc(Cl)cc1C(N1CCC(CNC(c2ncncc2Br)=O)CC1)=O 51257,C1(CC(=O)NC2CC2O)CCCCN1C(c1ccc(Cl)o1)=O 51258,C1(NC(CCc2c(C)cccn2)=O)CCN(C(C2(C)CCCC2)=O)CC1(C)C 51259,c1(OC)n[nH]cc1C(=O)N(C)CCOCCCNC(=O)Cc1nnc(O)s1 51260,CC1C(NC(=O)Cc2cccs2)C(C)CCN1C(c1cnc2n1CCC2)=O 51261,C1(OC)CC(C(=O)OC)CN(C(=O)C(CC)(CC)OC)C1 51262,C=CC(C(=O)NC1CC(C(=O)NCC2(CC)CCCC2)C1)OC 51263,C1(F)(NC(C(C)OCC2CC2)=O)CCN(C(C2CCN(c3ccccc3)C2)=O)C1 51264,N1(C(C(n2cc(C(C)O)nn2)C)=O)CCN(C(=O)CCn2ccnc2)C(C)C1 51265,C1(O)(CN(C)C(c2occc2Cl)=O)CCN(C(=O)CCCF)C1 51266,c1(NCC)cncc(C(=O)N(C)CCOCCNC(=O)CCc2cn(C)nn2)c1 51267,c1(OC)ccc2cc(C(=O)NC3CC(N(C(=O)CC(C)C(F)F)C)C3)[nH]c2n1 51268,c1(NCCC2(COC)CC2)nc(N2CCC3(CC(=O)NC3=O)C2)nc2scnc12 51269,N1(C(C2C3COCC23)=O)CC2(C(=O)NCCCC(F)(F)F)CC1CO2 51270,c1(C(=O)NCCCN(C(=O)CC2CC3(CC3)C2)C)sccc1C#N 51271,C1(F)(CNC(c2c(CC)noc2)=O)CCN(C(=O)CNC(c2cccs2)=O)CC1 51272,C#CCCCC(=O)NC1CC2C(NC(c3ccn(C4CC4)c3C)=O)C2C1 51273,c1(OC)cc(C)c(C(=O)NC2CN(C(=O)CCc3cnc(O)[nH]3)CC2O)c(C)c1 51274,n1(CC)nc(C)cc1C(N1CC(F)CC1C(N1CCC(O)(C(F)F)C1)=O)=O 51275,C1(CN(C(=O)CCc2nccs2)C)CCCN(C(c2cnsn2)=O)C1 51276,N1(C(C(C(C)NC(c2cc[nH]n2)=O)(C)C)=O)CC(O)C2(CCCC2)C1 51277,c1(C(=O)NC(C2CCN(C(C(F)=CCC)=O)C2)(C)C)cc(C)c(C)o1 51278,CCC(C)(C)C(C(=O)N1CC(CC(=O)NCC2(OC)CCC(C)C2)(OC)C1)OC 51279,N1(C(CS(CC)=O)=O)C(C)CC2CN(C(C3(n4cccn4)CCC3)=O)CC12 51280,Cc1sc(C(=O)NC2CC(O)CN(C(c3ccc(O)nn3)=O)C2)cc1S(N)(=O)=O 51281,C1(OC)CN(C)C(C)(C(=O)NCC(CO)NC(c2ccsc2SC)=O)C1 51282,N1(C(C(C)(F)F)=O)CCN(C(=O)CN2CC(C(N)=O)C2)CC(CO)C1 51283,N1(C(c2cc(SC)oc2)=O)CCN(C(=O)CNS(=O)(=O)N(C)C)C(CC2CC2)C1 51284,C1(NC(CCN(C(=O)C(C)=CCC)CC#C)=O)(CO)CCSC1 51285,CCC(C)(C)C(=O)C(=O)N(CC(=O)NOCCCC1CC1)C 51286,c1(-c2ccc(C(=O)NCCN(C(=O)CCCc3ncco3)C)[nH]2)ccccc1F 51287,c1(C(=O)NC(CC=C)CNC(c2cccnc2C2CC2)=O)ccc(C)nc1OC 51288,Cc1ccc(C)c(CN(C(c2cccc(Br)c2)C(=O)O)C)c1 51289,c1(C(=O)OC)cc(C#N)cnc1NC1CCC2CN(C(C3C=CCCC3)=O)CC12 51290,c1(C(N2CC(C)(NC(C3CC(C#N)C3)=O)C2)=O)nnn2c1CSCC2 51291,c1(CC)ccc(C(N2CCOC(CNC(c3cnn(C(C)C)n3)=O)C2)=O)c(C)n1 51292,Cn1ncc2c(N3CCC4(CC4)C3)nc(=NCCOCc3ccccc3F)[nH]c12 51293,C1(NC(=O)C(F)CC2CC2)CN(C(c2cccc(Br)c2)=O)CC2(CCC2)C1 51294,c1(C(=O)NC2CN(C(CC(CCC)O)=O)CC(C)C2)cc2ccc(F)cc2[nH]1 51295,C1(COC)(CNC(=O)C2=CCSC2)CCCN1C(c1ccc(C#N)s1)=O 51296,C[S+](C)CCC(O)C(=O)OCCCNC(=O)C1CC1 51297,CCCC(CCCO)C(=O)N1CC(C)CN(C(c2cccs2)=O)CC1C 51298,CN1CCC(CC(=O)NCCNC(c2ccc(F)cn2)=O)CC1 51299,c1(CC(=O)NCCCOC(C(=O)NCCCNC)OCCC#C)cnccn1 51300,c1(C(=O)NCC(C2CCN(C(C(C(CC)O)C)=O)CC2)C)cc2cccnc2o1 51301,CCCCCC(O)CC(=O)N1CCCC(C2CCCCN2C(c2cnsc2)=O)C1 51302,CC(C)CC(O)C(=O)N(CC(CO)C(C)C)C1CC1 51303,C1(NC(c2cnc(COC)s2)=O)CC(N=c2[nH]c3c(C)cccc3o2)C12CCC2 51304,c1(CNC(C2(C)CN(C)C(=O)C2)=O)ccc2c(c1)CN(C(=O)CS(C)(=O)=O)C2 51305,c1(CCC(=O)NC2C(NC(C(CC)C)=O)C2)c(OC)cc(OC)cc1OC 51306,C1(CC2CC(=C)CN2c2ccccc2F)N(C(=O)C2=C(C)OCC2)CC12CCCC2 51307,c1(C(=O)NC2C(CNC(c3c(COC)nn(C)c3)=O)C2)cc2occc2n1C 51308,N1(C(c2cn(CCNC(COCC=C)=O)nn2)=O)CCC(N=[N+]=[N-])CC1 51309,CC(C)CC(C)N(C(=O)CCN(C(=O)CC1OCCO1)C(C)C)C 51310,CCC(C)(CCNC(=O)C(C)SC)NC(=O)Cc1ccn(C(C)C)n1 51311,C1(N(C(=O)C(C)Cc2ccco2)CCC)CCN(C(C2COCCO2)=O)CC1 51312,C1(C(=O)NC2(CN(C)C(C3CC3C3(C)COC3)=O)CC2)CCC(O)CN1C 51313,c1(C(=O)NC2C(CNC(C3(CC#C)CC3)=O)C2)cnc2[nH]ncc2c1 51314,N1(C(Cc2cc(=N)[nH]cc2)=O)CCCC(NC(c2cccc(CO)c2)=O)CC1 51315,c1(NC2CCC(C(=O)OC)NC2)ccc2[nH]c(C)cc(=O)c2c1 51316,c1(CCOC)nc(CC(C)Sc2nncn2C)n(-c2cccnc2)n1 51317,c1(N2CC(C)(C)C(NC(=O)COc3ccsn3)C2)cc2nncn2cn1 51318,c1(OC(C)C)nc(C(=O)N(CCCNC(C2CCC(=O)N2)=O)C)cc(O)n1 51319,N1(C(c2nc[nH]n2)=O)CCC2(CC1)CN(C(C1COCCN1C(C)=O)=O)C2.CCS 51320,c1(NCC(C)OC(CSCC=C)=O)cc(C)ccc1Cl 51321,CCC(C)C(C(=O)NCC1(NC(c2ccc(C)cc2Cl)=O)CC1)NC(C)=O 51322,Cc1nc(Cl)ccc1S(=O)(=O)N1CCC(F)C(NC(c2cc(Cl)ncn2)=O)C1 51323,c1(OCCCOC)ncccc1CNC(c1nnc(C2CCNCC2)s1)=O 51324,C1(C(=O)NC(CN(C)C)C(=O)N2CC(N(C)C)C2)CCC2(CC2)C1 51325,Cc1ccccc1C=CC(=O)NC1C2CC3C(C2)C13 51326,c1(C(=O)NC(CC=C)CNC(=O)CC2(C)CC(F)(F)C2)ccc(S(N)(=O)=O)cc1 51327,C1(NC(C(CSC)C)=O)CC12CCN(C(c1n[nH]cc1[N+](=O)[O-])=O)CC2 51328,CN1C(=O)CCC1CNC(=O)CC=CCNC(c1ocnc1C1CC1)=O 51329,N1(C(c2cccc(NCC)c2)=O)CCN(C(C2CC2(C)C(F)F)=O)C(CCO)C1 51330,c1(C(=O)NC(C2CN(C(C3CC3C3CCC3)=O)C2)C)ccc2cncn2c1 51331,C=CCC(F)(F)CNC(=O)CNC(C1CCN1C(C)(C)C)=O 51332,C1(C(=O)NCC2C(C(=O)NC(C)CC3CC3)CCO2)C2CN(C)CC12 51333,c1(NC(C)=O)ccc(Cl)c(C(N2CCOCC2CNC(=O)CNS(N)(=O)=O)=O)c1 51334,c1(-c2ccc(CN3CC(C(=O)OC)C(C)CC3)s2)cccc(F)c1C#N 51335,C=C(C)CC(=O)NCC(C(C)C)NC(C1CCCN1Cc1ccccc1)=O 51336,C(=O)(CC(C)CC(F)(F)F)NCC(CN(C(C(C(C(C)C)O)C)=O)C)O 51337,c12ccccc1C(=O)NC2.c1(SC)cc(C(=O)NC(C)CCCO)co1 51338,C1(NC(C=Cc2c(C)ccs2)=O)CN(C(=O)C(=C2CCCCC2)F)CC12CCC2 51339,C1(C)(NC(C=CC=CC(CC)C)=O)CC(NC(C2CCC(C(F)(F)F)O2)=O)C1 51340,c1(C(N2CCC(NC(C3(C)CCC(=O)N3)=O)C(O)C2)=O)cc2ccc(F)cc2s1 51341,c1(C(=O)NC2CC(CNC(C3CC(F)(F)C3)=O)C2)nccc(Br)c1O 51342,CC(C)C(C(=O)NC(CO)C(C)NC(=O)C=CC1CC1)n1cc(Br)cn1 51343,CCCC(C(=O)NCCCN(CCC)C(C1CCN(C)C1C)=O)NC(N)=O 51344,c1(C(N2CC3CC3(CNC(C3(Br)CCC3)=O)C2)=O)ccc(OC(F)(F)F)nc1 51345,c1(C(N(C2CCCN(C(C(C)N(C(C)=O)C)=O)C2)CCO)=O)ccc(F)c(C)c1N 51346,c1(C(c2onc(Cc3cn(C)nc3-c3ccnn3C)n2)=O)ccc(F)c(F)c1 51347,CC1CN(C(C2CCN2S(C)(=O)=O)=O)CC1(C)CNC(=O)CN(S(C)(=O)=O)C 51348,Cc1cnc2c(C(=O)NC3CN(C(=O)CO)CC34CC4)cccn12 51349,C1(C(N(C(C)COC)CC)=O)(CNC(=O)C(N)=O)CCCCC1 51350,c1(C(=O)NC2(C)CCN(C(C3CCC3)=O)C2)nc(Cl)ccc1N 51351,N1(C(=O)NC(c2cc[nH]n2)C)CCC(CCc2cn[nH]c2)CC1 51352,N1(C(C2C(CCCC)CCC2)=O)CCN(C(=O)Cc2ccsn2)CC1 51353,c1(CCC)cccc(C(N2CCC(C)(CNC(=O)CCS(C)=O)C2)=O)c1 51354,N1(C(C2CN(C(C)=O)C2)=O)CC(C(=O)NCC(C)(F)C(C)C)C(F)(F)C1 51355,c1(CC(=O)NCC2(CCNC(=O)C=C3CCC3)CC2)ccc(F)cc1F 51356,C(c1ccccn1)=C(C)C(=O)NC(C)C(C)NC(=O)CN(CC(C)(C)C)C 51357,CCCCC(F)C(=O)NC(C)CCN(C)C(c1ccc(CCF)cc1)=O 51358,N1(C(CC2(OC)CCC2)=O)CCC2CC12C(=O)N(C(CO)C(C)C)C 51359,C#CCC(CC(=O)NCC#CC1CC1)NC(=O)CN1CCC(C)C1 51360,C(C)(c1cnccn1)=CC(N1CCCC(CN(C(CCC(C)OC)=O)C)C1)=O 51361,C1(NC(c2n(CCSC)nnn2)c2conc2C)CC2(C1)NC(=O)NC2=O 51362,c1(C(N(CCN(C2CCCCC2OC)C(=O)CCF)CC)=O)c(C)cc(C)cc1O 51363,C1(F)(C(N2CCC(OCC=C)C2)=O)CCCN(C(=O)CCc2ccn(C)n2)C1 51364,c1(NC(C2COCCN(Cc3nccc(OC)c3)C2)=O)cc(F)c(C)cc1Br 51365,c1(C(=O)NC2CC(c3ccccc3)(NC(=O)C3CC3)C2)ccc(=O)n2c1COCC2 51366,C1(C(=O)NC(C23CCC(CC2)C3)CNC(COC(CC)C)=O)CCOC(=O)CC1 51367,c1(OCCN(C)C)ccc(C(N2CC(NC(=O)Cc3ccsn3)C(O)C2)=O)cc1N 51368,c1(C(N2CC(N(C)C(C3(F)CC=CCC3)=O)C(O)C2)=O)cc(O)nc(O)n1 51369,C1(NC(C2C(C)(CC)C2)=O)CC2CCC(C1)N2C(C1(N(C)C)CC1)=O 51370,c1(C(=O)NCC(CC=C)NC(C2CCCC(O)C2)=O)cccc2c1CCCN2 51371,C1(C(=O)NC2CC(N(C(C(C)OCC=C)=O)C)C2)CCC2(CC1)CC2(F)F 51372,Cc1cc(C(=O)NCCC(O)CNC(=O)CC(C)C)n(C2CC2)n1 51373,CCCC(C)(O)C(=O)NCCOCCNC(=O)Cc1ccc(Cl)cc1Br 51374,C1(NC(=O)NC(c2ccc(OC)nc2)C)(CO)CCCCC1C 51375,N1(C(C2C(C)CCO2)=O)CC=CC(C(=O)N(C)CC2CC2)C1 51376,CC1CN(C)CC(C(=O)NCC23CC(NC(C4CC=CC4)=O)(CCO2)C3)O1 51377,C(c1cccc(Br)c1)=CC(=O)NC(CC)CNC(=O)Cc1ncn(C)c1C 51378,C(CC(C)C)(C(=O)Nc1cncnc1C1CC1)ONC(C(C)NC(C)=O)=O 51379,c1(COc2c(NC)cccc2C)nn(C)c(Cl)c1I 51380,C(=O)(C(O)CC[S+](C)C)NCc1cn(CC(C)NC(c2cc[nH]n2)=O)nn1 51381,n1(CCC(=O)OCC2CCCCc3ccccc32)nc2ccccn2c1=O 51382,Cc1nnccc1C(=O)NCC(C1CCOC1)NC(=O)CN1CCOCC1 51383,c1(OC)c(C)cc(C(N2CCCC2CNC(=O)C=C2CCC(C)C2)=O)cc1C 51384,Cc1c(C(=O)NCCc2n[nH]cc2C(=O)NC2COCC2C)nnn1C 51385,C1(C(N2C(C)CC2)=O)CC(F)CN(C(c2cc(C(F)(F)F)ccn2)=O)C1 51386,C1(NC(C2CCC(=C)CC2)=O)CCN(C(=O)Cn2cc(C(F)(F)F)nn2)C(C)C1 51387,C1(C(N2CC(CC(C)(C)CNC(=O)C(C)(Cl)Cl)C2)=O)C(C)(C)C1(F)F 51388,C1(F)(C(=O)NC2C(SC)CCCC2)CCN(C(c2ccccc2)=O)CC1 51389,C1(CNC(=O)CSC(F)F)CN(C(C23CC4CC2C3C4O)=O)CCC1(F)F 51390,N1(C(c2cnc(CC)s2)=O)CC2(CC(CNC(C3SCCC3C)=O)C2)C1 51391,c1(OCC(=O)NC(c2ccccc2)C(C)NC(=O)CC2CC2)ccc(F)cc1O 51392,N1(C(C(C)n2cncn2)=O)CC2(C1)CN(C(=O)CC1(C#N)CCOCC1)C2 51393,CC1(c2cn(CC3CCC(C(=O)O)O3)nn2)CCCN1C(=O)COC1CCCC1 51394,N1(C(c2[nH]cc(CC)c2)=O)CC2C(CN(C(=O)C=CCCC=C(C)C)C)C2C1 51395,C1(NC(C2N(C(C3C(OC)CC3)=O)CCN(C)C2)=O)CCCC(C2CC2)C1 51396,c1(C2C(C(C(=O)NCCC#N)N(C)CCC3CC3)C2)ccc(F)c(F)c1 51397,C(=O)(C(CCN(C)C)NC(=O)CC1CC1(C)C)N1CCC(C(CC)CC)C1 51398,c1(C(=O)NCC2(O)CC(NC(c3cccc(N)n3)=O)C2)cc2ccc(O)nc2s1 51399,CC1C(NC(c2cscn2)=O)C(C)CCN1C(c1ccc(C#N)cc1F)=O 51400,Cc1nnc2n1CCCC2C(=O)c1cn(-c2cc(F)ccc2F)nn1 51401,N1(C(C(NOC)=O)=O)CCC(C=CC(=O)N(CCN=[N+]=[N-])C)CC1 51402,C1(C(C)NC(CC(C)OC)=O)CCCN(C2CCCNC2=O)C1 51403,C1(NC(C(=O)NCCOC)=O)CCCCN(C(=O)Cn2cccn2)C1 51404,CC(C)(CC(F)(F)F)C(=O)NCC1(F)CCN(C(C2CCC3(CCC3)C2)=O)CC1 51405,C1(O)(CN(C)C(c2ccnn2CCF)=O)CCN(C(=O)COC2CCOC2)C1 51406,C1(C)(C(=O)NC2C(CNC(CCSCC)=O)CCCC2)Cc2ccccc2N1 51407,CC1CN(C(c2cscc2Cl)=O)CC1NC(c1cccc(OC(F)(F)F)n1)=O 51408,c1(OC(C)C)c(F)cc(-c2ccccc2C(N2CC3CCC2C(O)C3)=O)cc1F 51409,C1(N(C(COCC(C)C)=O)C)CCN(C(=O)Cc2cncn2C2CC2)CC1 51410,N1(CCNC(c2ccc(C)o2)=O)CCCN(C(=O)CC2CC3CCC2O3)CC1 51411,C(=O)(C(C)CC(C)C(C)=O)NC1C2OCC(NC(c3c(CC)n(C)nc3)=O)(C2)C1 51412,c1(C(=O)OC)cncc(C(=O)NC2CN(C(C3(SC)CC3)=O)CC2O)c1 51413,C1(CNC(c2c(C)coc2)=O)CN(C(=O)C(O)C2CCCC2)CC1(F)F 51414,C(=O)(CCN=c1[nH]ccs1)N1CCN(C(C(CC)(C)C)=O)CC1CO 51415,N1(C(Cc2scc(COC)n2)=O)CCCC(C)(NC(=O)C(O)C(F)F)C1 51416,c1(NC(=O)NC(CC=CC)C(=O)N2CC(NC(C)(C)C)C2)nnc2n1CCC2 51417,C1(NC(Cc2c(C)con2)=O)CC=C(C(=O)N2CC(C)C(C)C2C)C1 51418,N1(C(CCC#CC)=O)CCC2(CC(NC(=O)Cc3nc([N+](=O)[O-])n[nH]3)CO2)C1 51419,c1(C(=O)NC(C2CCN(C(c3c(SC)csc3)=O)C2)C)n[nH]cc1[N+](=O)[O-] 51420,Cc1cc(Cl)cc(C(N2CC(NC(=O)CSc3ccncc3)CC(C)C2)=O)c1N 51421,C(=O)(CP(=O)(C(C)C)C(C)C)NC(CN(C(c1cc(COC)[nH]n1)=O)CC)C 51422,c1(C(N(c2ncc(F)s2)C)=O)cccn2ccnc12 51423,c1(C(=O)OC)cc(C(=O)NC2(C)CN(C(=O)CC3CC3C)C2)cc(C)c1 51424,C(=O)(C(C)S(N)(=O)=O)NC1(C(C)NC(c2ccc(CN3CCCC3)cc2)=O)CC1 51425,N1(C(C2(C)CCCN(S(=O)(=O)CCBr)C2)=O)C2CCCC1COC2 51426,CCCCCC(CC)C(=O)NC1COCCN(C(c2cc(N)cnc2C)=O)C1 51427,C1(NC(CCCCOC)=O)(CO)CCCN(C(C2CC3CC3C2)=O)C1 51428,C1(C(N2CC(CNC(C=Cc3nc(C)sc3)=O)C(O)C2)=O)Cc2ccccc2O1 51429,c1(CSCC(=O)NC2CCC2NC(C2CC23CC3)=O)ccccc1Cl 51430,c1(-n2cc(C(N(C(COC)(C)C)C)=O)nc2)cccc(Br)c1 51431,CN1CCC(CC(=O)N(C(=O)C(N2CCC(O)CC2)C)CC2CC2)CC1 51432,CC(C)(CC(F)(F)F)C(=O)N1CCN(C(=O)CCCCC(N)=O)C(C(F)F)C1 51433,c1(CNC(N(C)Cc2cncc(NS(C)(=O)=O)c2)=O)ccc(F)c(F)c1 51434,N1(C(C(C=C)O)=O)CC(OC)C(OC)C1CNC(=O)CCS(C)(=O)=O 51435,c1(N2CCN(C)CC2)cc(CNC2CCC2c2ccc(F)cc2)[nH]c(=N)n1 51436,c1(CC(=O)N(C(C)C)CCN(C)C(C2CCOC2C)=O)cnc2n1CCCC2C 51437,N1(CCC)C2CCC1CC(NC(C1(C)CC3CCC(C1)S3)=O)C2 51438,Cc1cc(=NCCCN2CCC(C)CC2)[nH]c(N2CCC(c3nncs3)CC2)n1 51439,N1(C(C(CC(=C)Cl)NC(=O)Cc2ccn(C)n2)=O)CC(=O)NC(C)(C)C1 51440,c1(C2C(C(=O)NCC(CNC(c3cc(OC)ns3)=O)(C)C)C2)cccc(C#N)c1 51441,C1(C(N2CC(OC)C(C(=O)NC3C(C)(C)C3(C)C)C2)=O)CCCCNC1=O 51442,c1(N(C)Cc2cccc(OC)c2OC)nccc(=NC2CCCC2S(C)(=O)=O)[nH]1 51443,C1(C(C#C)NC(=O)CCN(C(=O)CC2CC(F)C2)C2CC2)CCOCC1 51444,N1(C(CCCSC)=O)CCC2(C1)c1[nH]cnc1CCN2C(=O)CCc1nccs1 51445,N1(C(COCC)=O)C(C(N2CSCC2C(=O)O)=O)CCC12CC2 51446,C1(C(N(C(C#C)C)C)=O)C2CCC(C2)C1NC(C1CCC1C#N)=O 51447,C=CCCCCC(=O)NCc1ccc(CCNC(=O)CC(F)(F)F)cc1 51448,Cc1occc(=O)c1OCC(=O)NCCCN(C)C(c1ccc(NC=O)cc1)=O 51449,N1(C(c2c(C)nn(C)c2)=O)CCC2(CC(C(=O)N3CCOCC3C)=NO2)C1 51450,c1(CC(C(=O)N(C2CCN(C(c3cnc(CC)[nH]3)=O)C2)C)C)c(C)n[nH]c1C 51451,N1(C(C=NOC)=O)C(C)CC2CN(C(=O)CC3CC=CCC3)CC12 51452,C1(CCC(=O)NCC(C2CCCC2)NC(C(C)N(C)C)=O)CCN(C)CC1 51453,C12(C(=O)NC(CCCC)CNC(=O)C(F)n3ccnc3)C3CC(CC13)C2(F)F 51454,N1(C(c2c(OC)cncn2)C(=O)NCCCSC)CC(N(C)C)C(C2CC2)C1 51455,c1(CN(CCF)CC)cn(CCNC(C)C(=O)Nc2ccc(C(=O)O)o2)nn1 51456,C1(C(=O)NC(CC=C)CNC(c2cnc(C)[nH]2)=O)CCC(n2ccnn2)CC1 51457,c1(C(N(C2C(NC(CC(CC)C3CCC3)=O)CCCC2)C)=O)ncnc(C)c1C 51458,C(CC(C)(C)NC(=O)Cc1ccccc1)NC(CN(C)C1CC1)=O 51459,C1(NC(CS(CC)=O)=O)CCCCN(C(c2cc(C)n(C3CC3)c2C)=O)C1 51460,N1(C(c2c(C)nn(C)c2)=O)CCc2c(C(N3CCCCC(O)C3)=O)csc2C1 51461,CCCCCC(O)CC(=O)N1CC2CCCC2C1C(=O)NCC1(C)COCCO1 51462,c1(C(=O)NC2C(C)N(C(=O)CCc3ccc(Cl)nc3)CC2)ccc2c(c1)COC2 51463,c1(OC)cncc(C(N2CCOC(CNC(C3CC(=O)N(O)C3)=O)C2)=O)n1 51464,Cc1ccc([N+](=O)[O-])cc1C(=O)NCC1(CNC(=O)C(CO)C(F)(F)F)CC1 51465,C(CNC(C1CCCCCC1)=O)(CC(C)C)NC(C1(C(=O)OC)C(=C)CC1)=O 51466,C1(NC(CC2(COC)CC2)=O)CCCN(C(c2ccc(C3CCC3)cc2)=O)C1 51467,C12(CCNC(C3(NC(CCC4C(C)(C)C4)=O)CSC3)=O)CC(CO1)C2 51468,c1(C(N2CC(C(C)Nc3ncc(C(=O)OC)cn3)OCC2)=O)ncc(Cl)cc1F 51469,c1(CCC)nc(C(=O)NC(CNC(=O)Cc2nc[nH]n2)C2CCC2)cs1 51470,c1(CC(=O)NC(CCNC(CC(CC)SC)=O)C)ncn2c1CCCC2 51471,CC1CCC(C(=O)NCCn2ccc(C(=O)NCC(F)(F)C(N)=O)c2)CC1 51472,c1(C(N(C2CN(C(Cc3c(C)ccs3)=O)C2)C)=O)ccc2[nH]ccc(=O)c2c1 51473,C1(C(=O)NC(CN(C(C2(COC)CCCO2)=O)C)(C)C)CC2CCC(C1)C2 51474,C12(C)NC(=O)N(C1=O)C2.C12(C)CN(C1)C(=O)Cc1nc2no1.C(=O)(C1CC1)OC 51475,c1(CC(C(=O)N2CC(CNC(CCNC(=O)OCC)=O)C2)C)c(C)nn(C)c1C 51476,Nc1cccc(C(=O)NC2COCC2CNC(=O)Cc2ccc(O)nc2)c1 51477,c1(OC)noc(C)c1C(=O)NC1CCC(CC(=O)NC2CC2c2cncs2)CC1 51478,c1(OC)ccccc1S(=O)(=O)NC1CC1C(=O)Nc1ccc2cc(C)[nH]c2c1 51479,Nc1ccc(F)c(C(N2CCC(NC(=O)Cn3ccnn3)C(F)C2)=O)c1 51480,C(CC(C)C)(C(C(=O)NCC(F)F)N1CCSCC(C)C1)OC 51481,c1(C2C(CN(C)C(C3COCCN3C(=O)C(C)(C)CO)=O)C2)ccc([N+](=O)[O-])cc1 51482,c1(OC)cc(C)c(C(N2CCC(CNC(=O)C3=CCOCC3)C(C)C2)=O)c(C)c1 51483,n1(CC(=O)OCC)nc(C)c(S(=O)(=O)N2CC(O)CC2C(=O)OC)c1C 51484,c1(C(=O)NCC(F)CNC(C2(C(F)F)CC2)=O)cccc2ccnn12 51485,c1(C(=O)NCC2C(C)CN(C(C3CC(O)C3)=O)CC2)nc(Cl)c(=O)[nH]c1N 51486,C1(C(=O)NC2CC(CNC(C(Cn3ccc(C)n3)C)=O)C2)CC(=O)N(C(C)C)C1 51487,c1(C(=O)NC(CN(C(c2cnc(OCC)nc2)=O)C)CC)ccc(F)cc1C 51488,c1(C(=O)NCC2C(NC(c3cnc4cc[nH]c4c3)=O)C2)nc2cc(O)ccc2[nH]1 51489,N1(C(CCCCC#C)=O)CCS(=O)(=O)C(CCNC(=O)C(O)P(C)(C)=O)C1 51490,N1(C(CC(CC)OC)=O)CCC(CNC(C2CC=CC(O)C2)=O)C(C)C1 51491,C1(O)(C(=O)NC2CCC(CNC(C(N3CCOCC3)C)=O)C2)CCCC(C)(C)C1 51492,c1(OC)ccnc(NC(=O)C(N2CCNCC2C#N)=O)c1F 51493,S(=O)(=O)(c1cc(Br)c(Br)s1)n1ncc(-c2nnc(-c3cncc([N+](=O)[O-])c3)o2)c1 51494,C(=O)(C(Cn1cncn1)NC(=O)C(=O)NC(C)C)NCCSC 51495,C1(N(CCCCCO)C(c2cccc(C#N)c2)=O)CCCC12CCNCC2 51496,c1(CC(=O)NCC(O)CCN(C(=O)CC2CC2(Cl)Cl)C)csc(Cl)c1 51497,C(C(=O)N=c1cc(C)nc(-c2cccc(F)c2)[nH]1)n1ccc(C)n1 51498,C(C(CNC(c1ccc(SC)cc1)=O)C(F)(F)F)NC(CCCC#C)=O 51499,c1(C(N(C)CC2N(C(CC(C=C)C)=O)CCCC2)=O)cc(C)cc2cccnc12 51500,C1(NC(c2nsnc2O)=O)C=CCCC1C(=O)NCC1CCCS1 51501,c1(OCC(=O)N(C(CNC(c2c(C)c[nH]n2)=O)C)C)ccccc1C(F)(F)F 51502,c1(NC(c2scc(CNC(C(CC)n3ccnc3)=O)c2)=O)ccc2c(c1)COC2 51503,C(Cc1ccccc1)(CCCO)NC(c1n(CCOC)nnn1)c1csc(Cl)c1 51504,c1(SC)ncc(C(=O)NCC(C)N(C)C(C2CCCN2C(=O)OC(C)C)=O)s1 51505,c1(SCC(N2CCN(C(C3CC(C)(C)C3)=O)CC2)=O)ccc(F)c(F)c1 51506,N1(C(C(c2ccc(C)cc2)CC)=O)CC2(CCC(CNC(=O)CC(C)F)O2)C1 51507,N1(C(C2(SC)CCC2)=O)CCN2CCN(C(=O)C3=COCCC3)CC2C1 51508,N1(C(c2c(COC)cccn2)=O)CCC(NC(=O)C(F)CC(C)(C)C)C(C)(C)C1 51509,c1(NC2CC(OC)C23CCNCC3)nc2c(cc1C#N)CCOC2 51510,CCS(=O)(=O)CCN(CC(=O)NCc1cccc(Oc2ccccc2)n1)C 51511,C1(CNC(c2[nH]cc(CC)c2)=O)CN(C(=O)CC(F)(F)F)CC1C(F)(F)F 51512,C(=O)(CCCCCNC(C)=O)N1CC(OC)C(NC(=O)C(C)(C)c2cncs2)C1 51513,C(C(O)CN(C(=O)COCCF)C)NC(C=CC)=O 51514,N1(C(C)C(=O)NC(c2ccc(F)cn2)Cc2ccccc2)CC(C)OC2(CCC2)C1 51515,C#Cc1ccc(C(N2CCC(CNC(c3cncc(C)n3)=O)CC2C)=O)c(F)c1 51516,CCC(C(=O)N1CC=CC1CNC(c1ncccn1)=O)NC(N)=O 51517,c1(C(=O)NC(CC)CNC(c2ccn(CCF)n2)=O)cc(OC)c(Cl)s1 51518,c1(C(N2CC(CCNC(Cc3n(C)ccc3)=O)OCC2)=O)cnc2[nH]ccc2n1 51519,Cc1oc(C(=O)NC2CC3CCC2N3C(=O)C(O)C(C)(C)C)cc1S(N)(=O)=O 51520,C1(NC(C2(CC)CC2)=O)CCCC(NC(=O)C(c2ccc(O)cc2)=O)C1 51521,N1(C(C(C)OCC)=O)CCC(F)(CNC(c2ccc(N)cc2Br)=O)CC1 51522,c1(COCC(=O)NCC(C2CC23CC3)NC(=O)Cc2ccno2)nc[nH]n1 51523,Cc1c(C(N2CCC(C(=O)N(O)Cc3ccccc3)C2)=O)cc(F)cc1Br 51524,c1(C(C)C)nc(NCC(C)(C)OCCO)cc(=NC2CCCC(O)C2)[nH]1 51525,C1(C(N(c2cc(COC)on2)C)=O)CN(C(=O)CN2CCC(=O)CC2)CC1(F)F 51526,N1(C(C2N(CC#C)CCC2)=O)CCCC2(CC(NC(C3CC(F)(CO)C3)=O)C2)C1 51527,N1(C(C(CO)NC(c2ccc(F)nc2)=O)=O)CC2CC1CO2 51528,C(CN=c1[nH]c(=NC2COCC2CO)[nH]c2c1COC2)SCCOCC 51529,N1(C(C(C=C)CC)=O)C2CC1CN(C(=O)Cn1ccc(C(F)F)n1)C2 51530,C1(NC(CC=CC)=O)CC2CC1N(C(=O)CC(C(F)F)c1ccccc1F)C2 51531,c1(N(CC(=O)OCc2ccccc2)C(C2CCCC2)=O)ccc2ccnn2c1 51532,C1(C2CC2)(NC(COCC)=O)CCN(C(=O)C(Cc2ccccc2)SC2CC2)C1 51533,C(=O)(CCCC(F)F)N1CCC(CN(C(C(C(C)C)C)=O)C)CC1 51534,C1(OC)CCCC(C(N2CCCC2CCCNC(=O)Cc2c(Cl)cnn2C)=O)C1 51535,N1(C(CCC(C)N(C)C)=O)CC(C)N(C(C2CCCN2C)=O)C(C)C1 51536,C(C(=O)N=c1ccn(CCCNC(C23CCCC2OCC3)=O)[nH]1)N(C1CC1)CC 51537,c1(SC)ccccc1CCNC(=O)NC1CCOC(C(F)(F)F)C1 51538,c1(N2CCC(N3C(=O)CC(OC)C3)CC2)ccnc(C2CC2)c1O 51539,C(N=c1[nH]c(=N)[nH]c(=NCc2ccc(Br)o2)[nH]1)C1(N(C)C)CCCC1 51540,C1(C(C)=O)CC1(Cl)C(=O)NC1CC1NC(=O)COc1cn[nH]c1 51541,CCC(C)CC(C)C(=O)N1CC(CC(N2CC(O)C(N=[N+]=[N-])C2)=O)(OC)C1 51542,c1(OC)ccc(C(C)C(=O)NC2CC3CC(NC(=O)CP(C)(C)=O)CC23)c(C)c1 51543,N1(C(CC(CC)(F)F)=O)CCN(C(c2c(C)ccnc2O)=O)CC2CCCCC12 51544,N1(C(CCc2ncc(C)[nH]2)=O)CCCCC(CNC(C2CCCN2C(C)C)=O)C1 51545,C1(NC(C2(C#C)CN(C(c3cc(C)sn3)=O)C2)=O)CCCOC12CCC2 51546,N1(C(C(=O)NCCNC(C)=O)=O)CCN(C(=O)CC(C)P(C)(C)=O)CCC1C 51547,C(C)(CC(C)C(F)F)NC(C(CN(C(c1cc(CC)[nH]n1)=O)C)C)=O 51548,C1(O)(CC(C)C)CCN(C(C2(NC(=O)C(C(C)C)C3CCC3)CCOCC2)=O)C1 51549,CC1=C(C(=O)N2CCC(C3CCCN3C(c3[nH]c(O)nc3C)=O)C2)SCCO1 51550,Cc1ccc2cc(C(=O)NC3CN(C(=O)COCCCF)C(C)(C)C3)[nH]c2c1 51551,C1(CNC(C=CC(=O)NC2CC2)=O)CCCC1C(=O)NC1CCC1(F)F 51552,N1(C(c2n(C)cc(Br)c2)=O)CCC2CN(C(C3CC(C4CC4)=NO3)=O)C2C1 51553,C(C(C)(C)C#CC(=O)N(CCF)CC)NC(C(CC)N(C)C)=O 51554,C1(NC(C2N(CC)CC2)=O)CC2(CCC(CNC(c3cocc3C)=O)OC2)C1 51555,C1(C(=O)NCC2(C)CC3CC3C2)CN(C(C2(C)CC(C#N)C2)=O)CC1(F)F 51556,N1(C(CCc2n(C)ccn2)=O)CC2(CC(CNC(=O)C(O)Cc3cnc[nH]3)C2)C1 51557,c1(C(=O)NCC2N(C(CCCCCOC)=O)CCN(C)C2)ccc(F)c(C#N)c1 51558,c1(C(N2CC(NC(C(C3CCCCC3)OC)=O)C2)=O)ccc(=NC)[nH]c1 51559,C1(NC(=O)COCCOC(C)=O)CC(C(CC)=O)CCO1 51560,N1(C(C2C(=C)C2)=O)CCC2(CC(NC(c3c(-c4ccccc4)coc3C)=O)C2)C1 51561,N1(CC(=O)NC2C=CCN(C(C(c3cccnc3)C)=O)C2)CCCCS1(=O)=O 51562,N1(C(C(C)SC)=O)CCC(C2CCCN(C(c3c(Cl)nn(C)c3Cl)=O)C2)C1 51563,C1(C)(C(=O)NC2CN(C(c3sc(CC)c(C)c3)=O)C3C2C3)CCC(C)CC1 51564,C1(CC2CCC2)CC2CC(C1)C(=O)NC(=NC)NC(CCCC)C2=O.OC 51565,N1(C(C)CN(C)CCO)CCC(CO[Si](C)(C)C)CC1 51566,CC(C)S(=O)(=O)C(C)C(=O)NCC1(O)CCCN(C(=O)C(O)C2CCC2)CC1 51567,N1(C(CCOC)=O)CCN(CCN(C)C(C2CCCC(CF)C2)=O)CC1 51568,c1(C(N2CC(NC(CCCCN(C)C)=O)(CO)C2)=O)cccc2[nH]cc(Cl)c12 51569,C(=O)(CC(O)C(C)C)NCc1ccn(CC)n1.C1(=O)C(CC2CC2)N1C 51570,CON1CC(C(=O)NCC2CCCC2C(=O)NC2(C)CC=CC2)CC1=O 51571,C(C)(CCC(C)(C)C)(c1n(CCOC)nnn1)NCC1(C)COCCO1 51572,c1(N(CC(C)NC(c2csc(CN(C)C)n2)=O)C)nc(O)c2ccc(Cl)cc2n1 51573,N1(C(c2c(CC)cnnc2)=O)CC2CC(C)N(C(c3cccc(F)c3C)=O)C2C1 51574,c1(NC(C(CCOC)C)=O)ccc(NC(=O)C(C)(C)n2ccc(C)n2)cc1C 51575,N1(C(CC(CC)OC)=O)CC(N(C(=O)CCOC)CC)C2(CC2)C1 51576,c1(C(N2CCC(F)(C(=O)Nc3c(C)cccc3)C2)=O)cc(C)c(C)cc1I 51577,O=C(CCCn1cc(-c2ccccc2F)nn1)NNC(=O)C1CCCS1 51578,C1(C(=O)NCC2CC(NC(=O)COc3cccnc3)C2)CCCC(=O)O1 51579,Cc1cc(N2CCOc3ccc(F)cc3C2)nc(=NCC(C)(C)C2CCCC2)[nH]1 51580,C1(CC#C)(NC(=O)C=CCNC(=O)CC2CCCO2)CCC1 51581,c1(CN(CCO)CC)cc(-c2coc3ccccc23)c(OC)c(Cl)c1 51582,C(CC(C(C)(C)C)NC(C1CC12CCC2)=O)N(C(c1cn(CCCC)nn1)=O)C 51583,N#CC1(C(N2CCCC(F)(C(=O)NCC(O)C(F)(F)F)C2)=O)CC(F)(F)C1 51584,c1(C(=O)NC(C)CC(C)NC(C2CCCC2c2ccccc2)=O)ccc(O)nc1 51585,C1(C(=O)NC(CN(C(c2c(C)nc(C)[nH]2)=O)C)(C)C)CC2COCC2C1 51586,C(CC(C)CC)(C(=O)NCCCc1ccnn1C)NC(CC(C=C)(C)C)=O 51587,c1(CNCCN(C2CCC3CC23)C)ccc(C2CCC2)cn1 51588,C1(C(N(CC#CC)C)=O)CCCCC1(C)NC(C1CCOCC1)=O 51589,C1(C(=O)NC(C)C(C)NC(C2CC(F)(F)C2)=O)CCCN1C(c1ccccc1)=O 51590,c1(CC)c(Cl)nc[nH]c1=NCC1CCCCN1C(C1CCN(C(C)(C)C)C1)=O 51591,N1(C(CC(CC)C(C)C)=O)CCC2(CC1)OCCC2NC(=O)CC(C)C(F)(F)F 51592,N1(C(C(C=C)(C)C)=O)CCC2(CC1)CC(NC(=O)C(CC)n1nccc1C)CO2 51593,N1(C(C(c2ccccc2)N)=O)CC=CC(NC(c2cc(C(F)(F)F)ncn2)=O)C1 51594,c1(CN2CCCC(CC(=O)N(CCCCC=C)C)C2)cc(O)cc(Br)c1 51595,Cc1cccc(CC(=O)NC23CC2CN(C(c2cnn(C(C)C)c2F)=O)C3)c1Cl 51596,N1(C(c2ccccc2)CCNC)CCC(S(=O)(=O)N2CCCC2)C1 51597,N1(C(CCC(=O)OC)=O)CC(C(=O)O)C2(C1)CN(C(c1n[nH]cc1Cl)=O)C2 51598,c12cc3n(n1)CCCN(C3)C2=O.c1(CNC(=O)C(F)Cl)ccc2nc(O)oc2c1 51599,c1(CC(N2C(CC)C(NC(=O)CC#N)CCC2)=O)c[nH]c2cc(C)ccc12 51600,C12(CNC(C3CC(C)(CC)C3)=O)CCCC1N(C(=O)C(C1CCC1)OC)CC2 51601,N1(C(c2cnsc2)=O)CCOC2(C1)CN(C(c1cc(Br)c3nccn3c1)=O)C2 51602,N1(C(C2(C=C)CC2)=O)CCC(NC(c2sc(SC)cc2C)=O)C(F)C1 51603,C12(C(N(CCCNC(C(C)NC(C)=O)=O)CC3CCCC3)=O)CC(C#N)(C1)C2 51604,N1(C(C(C=C)(C)O)=O)CCCC(C)(C(=O)NC2CCOCC2F)C1 51605,CCC(C(=O)NCC(C)N(C)C(C1(C#N)CC1(C)C)=O)C(C)C 51606,c1(C(N2CCCC(C(=O)Nc3c(C)ncn3C)C2)=O)cc(Br)cc2c1OCC2 51607,N1(C(CCCCOCC)=O)CCC2CN(C(=O)CCC(CF)CF)CCC12 51608,Cc1ccc(NC(c2nccn2C)c2nnnn2CCN2CCOCC2)c(C)c1Br 51609,c1(C(=O)NC(CCNC(c2c(C)snc2)=O)C)nn(-c2ccon2)cc1Br 51610,c1(C(N2CCC(CC(N)=O)C2)=O)ccc(NCCN(C)C(c2nc[nH]n2)=O)cc1 51611,C1(CNC(C(CC(C)C)O)=O)CN(C(c2ccccc2O)=O)CCC12CCC2 51612,c1(SC)ccc(C=CC(N2CC(C(C)NC(C3CCCCC3O)=O)C2)=O)s1 51613,C1(CC(=O)NC2(C=C)CCC2)CCN(C(C2CCCN2CCC)=O)C1(C)C 51614,c1(C(C)C)ccc(C(=O)NCC(=C2CN(C(=O)C(C#N)=CC3CC3)C2)F)c(F)c1 51615,Cc1ccc(Cl)c(C(=O)NCCn2cc(CC(=O)NCCNC(N)=O)nn2)c1O 51616,CC(C)CC(C)(O)C(=O)N1CC(O)(CNC(c2cc3c(s2)COCC3)=O)C1 51617,C1(OC(=O)NC(C)CC2CN(C(=O)CC3(O)CCOC3)C2)CCCCC1 51618,c1(C(=O)NCC2CC(OC)CN2C(=O)COCC(F)(F)F)c(F)ccc(F)c1Cl 51619,C12(CNC(Cc3ncc(C)s3)=O)CCC(C1)N(C(=O)CN(C)S(N)(=O)=O)C2 51620,C1(CC)(CC)CC(C(=O)NC(C2(CNC(c3ncnn3C)C)CCCO2)=O)C1 51621,c1(C(=O)NC(c2cn(C)nn2)C(=O)NCC(CC)N(C)C)cncc(C)n1 51622,Cc1cc(C(=O)N(CCC(=O)O)CCCC(C)N=[N+]=[N-])c(Br)s1 51623,S(=O)(=O)(c1cccnc1NCC1(CCOC)CCCC1)N1CC(C)N(C)C(C)C1 51624,C(=O)(C1CCOc2ccccc21)N1CC(NC(c2nocc2C)=O)CC(OC)C1 51625,C=C1CC2CCCC(C1)N2C(C1CCCN(C(c2csc(=N)[nH]2)=O)C1)=O 51626,C(=O)(C#CC1(C)CCCO1)NCC(C)N(C(c1cc(Cl)ccc1O)=O)CC 51627,c1(-c2n(CC=C)c(CC(C)(C)C)nn2)c(Br)ccc2c1OCCO2 51628,CCCCC(O)C(=O)N1CC(CNC(c2ccc(C(N)=O)nc2)=O)C2(CC2)C1 51629,C1(C(=O)NC2(CF)CCN(C(C3CCC(C)(C)C3)=O)C2)CC2(CC(=O)N2)C1 51630,N1(C(c2ncc(CC)cn2)=O)CCC2CCCC12C(N1CC2C(C1)C2(F)F)=O 51631,c1(C(=O)NC(C2CCCCN2C(=O)CC2CSC2)C)ccc(S(=O)(=O)N(C)C)cn1 51632,C1(C2CC2)(NC(C2C(NC(c3cc(CO)[nH]n3)=O)CC2)=O)CCCC1 51633,C(=O)(C1CC(=O)Nc2ncccc21)NC(CC(C)C)CNC(=O)C(C)C(C)O 51634,Cc1nn(C)c(F)c1C(N1CCC(CNC(c2ccnc(OC(F)F)c2)=O)C1)=O 51635,CCC(CC(=O)N1CC(C)(C)CC1CC(=O)N(C)Cc1cnnn1C)CC(C)C 51636,CC(CC(=O)N(C)CCc1ccccc1)NC(=O)CC1(C#N)CC1 51637,C(CC(C)C)(C(=O)NCC1CN(C(=O)COc2cccc(C(C)C)c2)C1)OC 51638,CCCCS(=O)(=O)N1CCC(COC(=O)NC2CCOC2=O)CC1 51639,C(=O)(C#CC1(CC)CC1)N(CCNC(c1ccncc1N(C)C)=O)CC 51640,CC1CN(C(=O)Cn2ccnn2)CCN1C(C1(C(F)(F)F)CCOCC1)=O 51641,N1(C(C(=O)NCc2c(CC)noc2C)=O)CCC(C)(c2nc(C)no2)CC1 51642,c1(C(N2CCC(NC(c3cc(C(C)C)no3)=O)C(O)C2)=O)ccc2snnc2c1 51643,N1(C(C(CCC)N(C)C)=O)CC(N(C(=O)C=Cc2ccco2)C)C2(CC2)C1 51644,CC1(C)CC(C(N2CCC(C(C)(C)O)CC2)=O)CN(C(C2C3CCCCC23)=O)C1 51645,C12(C(=O)NCC=CCNC(c3c(C)occ3)=O)COCC(C1)C2 51646,CCC(CCC(=O)NCCC1(CO)CC1)NC(=O)CC1(C)CCCCC1 51647,C(=O)(C(C)CC(F)(F)F)NCCN(C(C(CSC)(C)C)=O)C1CC1 51648,C12(NC(CCCC#N)=O)CCC(CC1)N(C(=O)CCN1CCC1)C2 51649,NS(=O)(=O)c1cc(C(=O)OCC2C3CCCCCC23)c(F)c(Br)c1 51650,c1(CC)cnc(C(=O)N(CCNC(C2CCC(C(N)=O)CC2)=O)C(C)C)cn1 51651,c1(CCC)cnnc(C(=O)NC(C)(C=CC=NC(=O)C=C(C)C(C)(C)C)CO)c1 51652,N1(C(C2C(COC)C2)=O)CCN(C2CCCN(C(=O)C=C(C)C(F)F)C2)C(=O)C1 51653,c1(OC)cc(C(=O)NCC(C)CN(C(=O)C(=O)NCC(F)(F)F)C)ncn1 51654,c1(C(=O)NCC23CC(NC(C=C(C)C(F)F)=O)(C2)C3)c[nH]c2ncc(Br)cc12 51655,C(c1ncc(C)[nH]1)=CC(=O)ON(C1CC(F)(CC)C1)C(C1(c2ccno2)CC1)=O 51656,Cc1cc(=O)c(-c2nc(CO)nn2C(C)C(C)(C)C)cn1C 51657,C1(NC(c2c(COC)cco2)=O)CN(C(C2CCCC2(C)C)=O)CC1C 51658,C(CCO)(C(F)F)NC(C(Cn1ccnn1)NC(C=CCN(C)CC)=O)=O 51659,CCCCC(C(=O)N1CCN(C(=O)CSC)CC1c1ccccc1)NC(N)=O 51660,c1(CC2CC(CC(=O)NCc3occ(C)n3)C2)cnn2cccc(C)c12 51661,N1(C(C2=C(C)CC2)=O)C(CC(N2CC3CCCCC23)=O)C2CCCC12 51662,c1(OC)nc(C)cc(C)c1CN1CCN(S(=O)(=O)c2sccc2C)CC1 51663,c1(CC(=O)NCCC2CC(NC(CCc3ccc(C)s3)=O)C2)cn(C)nc1C 51664,c1(CC)csc(CNC(n2cc(CNC(=O)CCN3CCOC3=O)nn2)=O)n1 51665,N1(C(C(CC=C)CNC(=O)C(C)CC)=O)CCN(C)C2(CC2)C1 51666,C=CCC(Cc1ccccc1)C(=O)NC1CCCC1NC(=O)CC(F)F 51667,c1(NCCc2cc(C)ns2)ccc(S(=O)(=O)NC2CN(C)CCC2O)cc1C#N 51668,N1(C(C(C(C)C)OCC)=O)CCN(C(c2ccc(C(N)=O)[nH]2)=O)C(C(F)F)C1 51669,c1(C(N2CC3C(CNC(C4(C)CCN(C)C4)=O)(C3)C2)=O)cc(F)ccc1C1CC1 51670,S(=O)(=O)(c1ccc(F)cc1)NCC(F)(F)F.n12cc(nn1)CNCC2C 51671,C1(NC(c2cc(F)cc(F)c2)=O)CC(NCCC2CCCC2)C12CCC2 51672,C(C(=O)N(C(C)CCNC(=O)C(C)Sc1ccccc1)C)(C(C)C)NC(C)=O 51673,CC1C(=O)N(CC(=O)NC2(CNC(=O)Cc3nncs3)CCC2)C(=O)C1C 51674,c1(CN(C2CCCCNC2)C)n[nH]c2c1COCC2 51675,N1(CC)CC(C(=O)NC2CCCN(C(C3CN4CCN3CC4)=O)CC2)CCC1=O 51676,n1(CC)cc(C(=O)NCC2CCCN2C(=O)Cc2c[nH]nc2O)c(C(C)(C)C)n1 51677,C(C(C)(C)C(F)F)NC(C(C1CCN(C(=O)C=Cc2ccccc2)C1)C)=O 51678,c1(NC(c2ccc(NCc3ccncc3Br)cc2Cl)=O)ccc2ccccc2c1 51679,c1(C(c2nnnn2CC2CCOC2)Nc2cn(CC)nc2)nc2c(s1)CCC2 51680,N1(C(C(C)N(C)C)=O)CCC(CNC(=O)C(C)CC(N)=O)C12CCC2 51681,c1(OC)ncccc1C(=O)NC(C)(C)CN(C(=O)Cn1ccc(C)n1)C 51682,c1(C(=O)NCC(C2CCCCC2)NC(CC(C)SC)=O)cc2n(n1)CCCN2 51683,C1(NC(C(CSC)C)=O)CCCOC12CCN(C(c1coc(CO)c1)=O)CC2 51684,C1(NC(C(C)NC(N)=O)=O)(CNC(c2cnn[nH]2)=O)CC2CCC1CC2 51685,Cc1cc(C(C)C(=O)N2CC(CNC(c3nc(C(C)(F)F)cs3)=O)C2)c(C)o1 51686,C1(NC(c2ncc(CC)s2)=O)COC2(C1)CN(C(=O)Cc1ccc(O)cc1)C2 51687,c1(CC)nc(C)[nH]c1C(=O)NC(CNC(=O)C(C(C)C)SC)CC(C)C 51688,CC(C)(C(=O)NCC1CCCN(C(=O)CCOCC(F)(F)C(F)F)C1)C(F)(F)F 51689,C(N=c1ncc(C(C)(C)O)c[nH]1)C1CCC(NC(c2c(C)ocn2)=O)CC1 51690,N1(C(C(CC)CC)=O)CC2CCCC(NC(=O)C(COC)N(C)C)C2C1 51691,c1(C(=O)NCCCN(C(CC(CC)O)=O)C)coc2cc(F)cc(F)c12 51692,c1(OC)ncnc(OC)c1C(C)NC(C1CC1C(F)(F)F)=O 51693,CN1CCN2CC1C2=O.c1(C(C(=O)OC(C)(C)C)F)ccc(F)cc1F 51694,CCCCCC(=O)NCC(=O)NC1CCN(C(=O)C(C)CCOC)C1 51695,C1(CSC)CCCN(C(C2CC=CCC2)C(=O)NCCc2cccc(OC)c2)C1 51696,CC(CC(=O)N1CC(C)C1C(=O)N=c1ccn(C(C)C)[nH]1)CC(C)(C)C 51697,C1(NC(c2c(C)nn[nH]2)=O)CCC2CC1CN2C(=O)CCCCCC#N 51698,c1(NC(=O)NCC(C)(C)CC2CCC2)cccc2c3c([nH]c12)CCCCC3 51699,C1(C(=O)NCC(CCNC(c2ccc(C(=O)OC)s2)=O)O)CCCCCN1C 51700,C1(NC(c2c(C)ccs2)=O)CCCCN(C(c2cnc(C(C)(F)F)s2)=O)C1 51701,C1(NC(c2c(CC)n[nH]c2)=O)CC2(CNC(=O)CCC3CCOCC3)CC1CO2 51702,C(=O)(C(C)C(F)(F)F)NCc1c(C(=O)NC(CCCCC)C)[nH]cc1 51703,C(c1cn(C)nn1)=CC(N1C(CNC(c2c(C(C)C)scn2)=O)CC1)=O 51704,c1(CNC(N(C2CCC3CC23)C)=O)cccc(Br)c1F 51705,C(=O)(C1=CCC(F)(F)CC1)N1CCC(C2(NC(c3cc(C)no3)=O)CC2)C1 51706,C#CCCC(=O)NCCn1ccc(C(=O)NCC2(SC)CC2)c1 51707,C12CC(C1(C)C)NCCN(C)CC(=O)NC2.C(C(=O)NCC(=O)NC)=CC 51708,c1(NC(C(=O)NC2CC(C=C)C2)=O)c(OC)cccc1C 51709,c1(NC(C2CCCN(CCCC(=O)NC)C2)=O)c(O)nc(=O)n(CCSC)c1N 51710,C(=O)(CS(=O)c1ccc(Cl)cc1)N1CCC(N(C(C=CC(C)(C)SC)=O)C)C1 51711,C1(C(c2nnnn2CCSC)NC(c2ccccc2)COC)CCS(=O)(=O)CC1 51712,N1(C(C(=O)NCC=C)C(C)C)CCOC(C)(C(F)(F)F)C1 51713,C(C(F)(C(=O)NCCC1CCCCO1)C(C)C)NC(c1c(C)nsc1C)=O 51714,CCC(CCC(=O)NC1CC2(C1)CC2C(=O)N(C)CCOC)OC 51715,N1(C(c2c(NC)scn2)=O)CCC2CCC(C1)N2C(=O)CC1CCSC1 51716,C12(CC(=O)NCCC(C)S(C)(=N)=O)CCC(CC1=O)C2(C)C 51717,C1(CNC(CC)=O)CCC2(CCN(C(c3ccccc3COC)=O)CC2)O1 51718,CON1CC(C(=O)NCC2(O)CCN(C(=O)Cc3ccn(C)n3)C2)CC1=O 51719,C12(CNC(CCc3onc(CSC)n3)=O)CCCN(C(=O)CSCC(C)C)C1C2 51720,c1(N)cnc(Cl)c(N)c1.c12ccc(cc1)OO2.C12CCCN1C(=O)N(CC)C2.CC 51721,C1(NC(C)=O)CN(C(=O)CCc2cc(Cl)cc(Cl)c2)CC12CC2 51722,c1(CN(CCC(C)(C)C)C(c2ccccc2)C)nn(C)cc1Cl 51723,c1(NC(C2C(C(N(CC)Cc3ccccc3)=O)C2)=O)ncc(C)cc1Br 51724,CCCCCC(O)C(C)C(=O)N1CCCC(CCNC(c2ccoc2Cl)=O)C1 51725,c1(C(=O)NCC23C(CN(C(C=CCCC)=O)C2)CC3)cc2c(Cl)c(Cl)ccc2[nH]1 51726,CCCC(CC)C(=O)NC(CC(=O)NCC1(C#N)CCCCC1)C(C)OC 51727,n1(CC(N2CC(O)CC(F)C2)=O)cc([N+](=O)[O-])cc1-c1nn[nH]n1 51728,c1(CNC(c2c(C(C)C)occ2)=O)cc(F)cc(O)c1F 51729,Cc1cnn(CCNC(=O)C(c2ccccc2)NC(c2csc(Cl)n2)=O)c1 51730,C12(C(=O)NC(C(C)NC(c3cncn3C)=O)C)CC(CCO1)C2 51731,C1(CNC(C(c2cncnc2)C)=O)COC(C)(C)CN1C(c1ccoc1C)=O 51732,c1(N(C)CC2(c3ccncc3)CC2)cc(-c2cccc(F)c2)ncn1 51733,C12(c3n[nH]c(=NCC4(C)C(C)CN(CC(C)(C)C)C4)o3)CC3CC(CC(C3)C1)C2 51734,c1(C(N2CCC(N(C(=O)CCC(F)F)CCC)C2)=O)ccc2c(c1)CCOC2 51735,c1(C2(C(=O)NC3CC4CN(C(=O)COCC5CC5)C3C4)CC2)c(Cl)cccc1Cl 51736,Cc1[nH]ccc1C(=O)NC1CCC(NC(C2(CC(C)C)CC2)=O)C1 51737,c1(CC)ccnc(C(=O)NCc2ccoc2C(=O)NC2COC(C3CC3)C2)c1 51738,N1(C(C2(C)COCCO2)=O)CCC2(CC1)CC2C(=O)NCCCCc1ncc[nH]1 51739,C=C=CC(C)C(=O)NCC(C)(C)C(=O)NCCC(C)(C)C=C 51740,c1(N(C(c2nc(OC)sn2)=O)C)cccc([N+](=O)[O-])c1 51741,CC(CCCNC(=O)CCc1cnoc1)NC(=O)CSc1nncs1 51742,C1(NC(C2(C(N)=O)CC2)=O)CC2CC(NC(c3cc(CC4CCC4)ccn3)=O)CC12 51743,c1(CCC(=O)NC23CC2CN(C(c2ccnn2C2CC2)=O)C3)nnc(O)nc1O 51744,Cc1ccc(O)cc1C(N1CCC(N(C(=O)C(C)n2cccn2)C)C1)=O 51745,C#CC1(C(=O)NCC2CC(n3cccn3)C2)CCN(C(=O)C(CSC)OC)C1 51746,c1(C(N2CC(CC(=O)NCc3n(CC)ncn3)C2)=O)cc2cccnc2[nH]1 51747,N1(C(c2ccc(C)nc2)=O)CCC2C(CCCN2C(c2c[nH]cc2C(C)C)=O)C1 51748,CC(C)(C)C(O)C(=O)NC1CCN(C(=O)C(F)(F)Cc2ccc(F)cc2)CC1 51749,c1(C(=O)OCC)c(C)[nH]c2ccc(OCC3C(c4ccccc4)C3C3CC3)cc12 51750,CCC(CC(=O)NCC1CC1C(=O)NCC1CC2(CCC2O)C1)CC(C)C 51751,N1(C(C2C(C(=O)OC)CC2)=O)CC(NC(c2ccn(C3CC3)n2)=O)CC(F)C1 51752,Cc1cnccc1-c1ccc(C(N2CC=CC2N(C)CC2CC3CCC2O3)=O)s1 51753,C#Cc1cccc(OCCC(=O)NC2CCOCC2NC(C2(COC)CC2)=O)c1 51754,c1(C(N2CC(CN(C)C(C3CCCS3)=O)C2)=O)csc2nccn12 51755,C(C1=CCN(C(c2cc(CCCO)on2)=O)CC1)NC(=O)C(F)=CC1CC1 51756,C1(CC=C)(C(=O)NC(COC)CCO)CCCN1C(=O)CNc1cccnc1 51757,C1(NC(c2cc(C)nc(C)c2)=O)CN(C(=O)CC2CCCN(C)C2)CC(C)(C)C1 51758,C(C(C)(C(=O)N1CC2C(C)C2C1)NC(c1cccc(C)n1)=O)SC 51759,c1(NC(CCCCCCNC(=N)N)=O)nc2ccc(Br)cn2c1F 51760,C(CC(C)CO)(C(=O)NCCOCC(F)(F)F)NC(C(C=C)(C)C)=O 51761,C1(CC)CN(C(C2(C)C=CCC2)=O)CCN1C(=O)COc1cc(C)on1 51762,C12(C(N(CC(=O)N(C)C)CCC)=O)CC(C)(CN1C(=O)Cc1nc(C)no1)C2 51763,N1(C(C2C(CNC(C3CC4(CCC4)C3)=O)CCO2)=O)CCC(=C(F)F)CC1 51764,C=CCCC(C(=O)Nc1cn(C)nc1OCC)NC(c1ccccc1F)=O 51765,Nc1cc(C(N2CC3CC2C3NC(=O)CCc2cscn2)=O)c(Cl)c(F)c1F 51766,Cc1ncnc(N2CCC(CNC(=O)COC(F)(F)F)C2)c1Br 51767,c1(C(=O)NC(CC)(C)CNC(=O)COCP(C)(C)=O)ccc(Br)cc1 51768,N(C(=NCC(C)CN1CCOCC1)NCc1ccco1)CC(C(=O)OC)F 51769,c1(C(=O)NCC(CC)NC(C2(C)CCNC2=O)=O)c(C)nc2ccccc2c1C 51770,c1(OC)cncc(C(=O)NCCC(C)(C)CNC(=O)C(C2CCCCCC2)C)n1 51771,C(=O)(CC(C)COC(C)CNC(=O)CC1CCOC1=O)OCC=C 51772,N1(CC(=O)NC2C(CCC)CN(C(=O)COCC(F)(F)F)C2)CCC(=O)NC1=O 51773,N1(C(c2cc(=O)cc[nH]2)=O)CCN(C(C2CC3COCC3C2)=O)C2COCC12 51774,C(C(C(C)C(C)C)NC(=O)C=CCO)NC(c1cn(CC)nc1C(C)C)=O 51775,C1(CC(N2CCC(NC(c3cnc4n3CCS4)=O)C2)=O)CN2CCC1CC2 51776,n1(CC(N2CC(OC)C(NC(C3CCC=CCCC3)=O)C2)=O)c(C)c(C)sc1=O 51777,C1(CNC(CNC(=O)NC)=O)CCCN(C(C2CC(C)(C)C2)=O)C1 51778,C12(CNC(c3cc(C)sn3)=O)CC3CC(CC(C3)C1NC(C1CNC(=O)C1)=O)C2 51779,CC(CN=c1[nH]nco1)(C1CC1)NC(c1cc(S(N)(=O)=O)co1)=O 51780,CCC(CC)C(=O)NCC(CNC(c1ncccc1F)=O)CO 51781,C1(C(C2N(C(CCC(=O)NC)=O)CCCC2)CNC(C)=O)C2(CCC2)C12CCC2 51782,C(=O)(C(C(CC)CC)OC)N1CCC(CCC(=O)NCCC(CCC)O)CC1 51783,n1(CCC)nc(C)cc1C(=O)N(C)CCN(C(=O)C(C1CC1)OC)C 51784,C1(NC(c2c(C)ncn2C)=O)CCN(c2nnc(C(C)(C)C)s2)CC1C 51785,N(C1CCCn2ncnc21)C(C(C)(N(C(COC)=O)C)C1CC1)=O 51786,c1(NC(N(CCOCCCOCC)C)=O)cc(Cl)c(Br)cc1C 51787,C(=O)(CC1=CCOCC1)NCC(CC)NC(C1CC(C)(C)OC1(C)C)=O 51788,N1(C(C(CC(C)=O)(C)C)=O)CCC2(CCCN2C2CCCNC2=O)C1 51789,N1(C(CCCC(=O)OC)=O)CCCC2CCN(C(c3cc(C4CC4)cs3)=O)CC12 51790,N1(C(C(c2ccccc2)N(C)C)=O)CC2CC(C1)N(C(=O)C=C(Cl)Cl)C2 51791,C(C(C)(C)CC(=O)NC1CCOCC1NC(=O)COCC(C)(C)C)OC 51792,C(C(C(=O)Nc1cnn(CCF)c1)C(C)(C)C)NC(c1c(C)n[nH]c1C)=O 51793,c1(NC(C)C)ncc(Br)c(C(=O)NCCOCc2ccccc2F)n1 51794,N1(C(C(N2C(=O)CCC2=O)C)=O)CC2CN(C(C3C(C)(C)C3(C)C)=O)CC2C1 51795,c1(CC(N2C(CCNC(C(CC)C)=O)CCCC2)=O)cc(C)cc(F)c1 51796,Cc1nc(CC(=O)NC2C=CCN(C(c3cc(C4CCOC4)[nH]n3)=O)C2)[nH]c1C 51797,CC1(C)CCC(CNC(c2ccccn2)=O)N(C(=O)CC=C(Cl)Cl)C1 51798,N12CC3CC3(C1)NCC2=O.CC(C)(C)NC(=O)N(CCCO)CCO 51799,C1(C(=O)NCCOCCCNC(c2ncsc2C2CC2)=O)CCC(C2CC2)C1 51800,C1(C(=O)NCC(C2CCN(C(C3(O)CCC3)=O)CC2)(C)O)COC2CCCCC12 51801,N1(c2nncc(C)c2C)CCCC(O)(C2CC2)C1 51802,c1(C(N(CC(C)NC(=O)C=CCN2CCSCC2)C)=O)ccc(CN(C)C)cc1 51803,N1(C(C2N(C(c3c(CC)cno3)=O)CC=CC2)=O)CCCC(O)(C(C)C)C1 51804,c1(OC)c(C)csc1C(=O)NC1CN(C(=O)Cc2cn[nH]c2)CC1C 51805,CC1CCCc2ncc(C(=O)NC3CC34CCN(C(=O)Cc3cnoc3)CC4)n21 51806,C1(CC=C)(NC(C2CCCN(CC)C2)=O)CCCN(C(=O)Cc2ccnn2C)C1 51807,C12(CNC(C3(C#C)CCC3)=O)CCC(CC1)N(C(c1coc(C)c1)=O)C2 51808,c1(C(c2n(CC)nnn2)NCc2conc2C(F)(F)F)ccccc1OCC1CC1 51809,C1(CC)CC(CNC(C2CC3(CC3)CO2)=O)N(C(c2cc(OC)no2)=O)C1 51810,S(=O)(=O)(c1ccc2ccccc2c1)Nc1cccc(NC(C(C(CC)C)O)=O)c1 51811,c1(C(=O)NC(CCOC)CNC(=O)C(C)(C)c2ccsc2)nccc2cc[nH]c12 51812,C1(CC(=O)NCCc2ccccc2O)CN(C(c2cccnc2)=O)CC1(F)F 51813,c1(CCCNC(N2CCCC2c2ncno2)=O)cccc(Br)c1 51814,N1(C(CC2(COC)CCCC2)=O)CC2CCN(C(=O)Cc3csc(C)n3)CC12 51815,N1(C(CCCCCCC)=O)CCN(C(c2cc(C(=O)OC)sn2)=O)CC2(CC2)C1 51816,CCC(CCC(=O)OC)N=C(NCCCCC(C)(C)C)NC(C)C 51817,C1(NC(c2ncn(CC)c2)=O)CCC(N(C(=O)COc2cn[nH]c2)C)CC1 51818,C1(C(=O)NCCN(C(=O)C(F)n2ccnc2)CCOC)CCC=CCCC1 51819,Cc1cccc(C(=O)NC(CNC(=O)CN2CCOCC2=O)C(C)C)c1F 51820,c1(C(=O)NC(C2N(C(c3cc(C)c(O)nc3)=O)CCC2)C)ccc(C)n(C)c1=O 51821,c1(C(N2C(C)CN(C(=O)CCC#N)CCC2)=O)cc(=O)c2cc(Br)ccc2o1 51822,Cc1csc(C(N2CCCC2C=CC(=O)NCC(C)(O)C(C)C)=O)c1C 51823,CC(N=c1nn[nH]n1C)C1C(NC(=O)CCC(F)(F)F)C1(C)C 51824,N1(C(CC(C=C)C)=O)CC2CC(C1)CN(C(C1CCCC(NC3CCC3)C1)=O)C2 51825,N1(C(C(C=C=C)C)=O)CCC(CC(=O)NCC(C2CCCC2)C)C1(C)C 51826,CCC(C)C(O)C(C)C(=O)NCC1CC(C(=O)NCC2CCCC(C)(C)C2)C1 51827,CN1CCC(C(N2CCOC(C3CC3(F)F)C2)=O)C(c2ccccc2)C1 51828,N1(CC(c2nccs2)=O)CC(n2cc(C(c3ccccc3)O)nn2)C(O)C1 51829,C1(C(=O)NC2CC(CCNC(c3ncncc3Cl)=O)C2)CC2(CCCCC2)CO1 51830,c1(OC)ccsc1C(=O)NCC1CCCC1C(=O)NOCc1nc[nH]n1 51831,c1(C(N2CCC(NC(C3CCC34CCC4)=O)C2)=O)cccc(C#CCO)c1 51832,c1(C(=O)NCC2C(C)CCN(C(=O)CSC(C)(C)C)C2)cc2ccccn2n1 51833,C1(NC(CC2CCC(C)O2)=O)CCN(C(C2(C3(C)CC3)CC2)=O)CC(O)C1 51834,C1(CNC(C=CSC)=O)CCN(C(=O)CCc2ccccn2)CC1(F)F 51835,c1(C(=O)NCC2(C(=O)NC(c3ccccc3F)C)CC(=C)C2)nccnc1O 51836,CC1CC(C#N)CN1C(=O)Cc1ncc(-c2cccc(Br)c2)[nH]1 51837,N1(C(CC(C)(C)OC)=O)CCC2CCCC12C(N1CC2C=CC1CC2)=O 51838,C1(NC(=O)CC2CC=CCC2)CCC2(CC1)CCN(c1nc3ccccc3o1)C2 51839,c1(C(N2CCOCC(CNC(COCC=C)=O)C2)=O)ncc2ccccn12 51840,CC1(C(N2CC3(CCC3NC(=O)Cc3ccccc3F)C2)=O)CCCCCC1 51841,CC(C)C(N=[N+]=[N-])C(=O)N1CCC(C)(C)C1C(=O)NC1CC2CC1CC2(C)O 51842,C1(CNC(Cc2c(C)nc(C)s2)=O)CC2(CO1)CN(C(=O)C(C)CS(C)(=O)=O)C2 51843,N1(C(C=Cc2ccc(C)s2)=O)CCCCCC1CNC(=O)CC1CCSC1 51844,CCCC(O)CC(=O)N(CCNC(=O)C(F)C(C)(C)O)CCOC 51845,C=CCN=c1ccc(S(=O)(=O)N2CCCCC2c2ncc(Br)cn2)c[nH]1 51846,N1(C(CCCC)=O)CC(CNC(c2cc(C(C)(C)C)n(C)c2C)=O)CC1(C)C 51847,C1(CC(=O)OCC2(C)CCCC2O)(NC(=O)OC(C)(C)C)CCCCC1 51848,CCC(CNC(c1cc(C#N)oc1C)=O)(CC)C(=O)NC12CCCCC1C2 51849,CCCCS(=O)(=O)CC(=O)NCC(CO)NC(c1csc(C)n1)=O 51850,Cc1ccc(C)c(C(=O)NC2CCCC2(C)CNC(=O)CC2CCCO2)n1 51851,C(=O)(C1=CS(=O)(=O)CCC1)NC1CCC(CNC(C2(C#C)CCCC2)=O)C1 51852,N1(C(CSc2ccc(C)cc2C)=O)CC(CNC(=O)CC#N)C2(CCC2)C1 51853,C1(NC(c2nccc(C)c2)=O)CCN(C(c2cncc(C(C)(C)C)c2)=O)CC1O 51854,C(C(=O)NC(C(=O)N(C)CC1CCOC1C)C1CCOC1)(C(C)(C)C)OC 51855,N1(C(C(C)=C(C)C)=O)CCC(C(=O)NCc2ncsn2)=C(F)C1 51856,c1(NC(=O)OC(C)(C)C)nc2ccc(NC(N3CC(O)CC(F)C3)=O)cc2s1 51857,C(C(C)(C1CC1)NC(=O)CNS(C)(=O)=O)NC(COC(CC)C)=O 51858,c1(CN(C)C)csc(C(C(=O)NC(C)(C)C)N(C2(c3cc[nH]n3)CC2)C)c1 51859,Cc1cc(C)n(CCC(N2CC3CC2C3NC(c2ccc(C(F)F)cn2)=O)=O)n1 51860,c1(OC2C(NC(N3CCCC3C3CCCOC3)=O)CCC2)ncccc1O 51861,C1(NC(CCCC)=O)CC(F)(F)CC1NC(=O)CS(=O)(=O)NCC1CCCO1 51862,Cc1cc(C(=O)NCCNC(c2ccccc2Cl)=O)ccc1-c1ccncc1 51863,C#CC1CC2CCC1N(C(=O)CC(C(F)(F)F)NC(c1cc(C)ccc1C)=O)C2 51864,Cc1nsc(CNC(c2nnnn2CCN2CCOCC2)(C2CC=CC2)C)n1 51865,C1(C(=O)NCC2CCCCC2C(=O)Nc2cn[nH]c2)CCCC2(CCC2)C1 51866,c1(CC)nc(C)c(C(=O)NC(C)CCN(C(=O)COCC2CCCO2)C)s1 51867,C(C1COc2ccccc21)NC(NC(c1ccc(Br)cc1)C#C)=NCCF 51868,C(=O)(CC(=O)N=c1ccn(-c2nccc(=NCCCN3CCOCC3)[nH]2)[nH]1)OC 51869,c1(OC)ccc2c(c1)CC(C(=O)NC1CCCC1NC(C1(CCO)CC1)=O)CO2 51870,CCCC(C)(O)C(=O)N1CC(NC(c2ccc(C(C)=O)c(F)c2)=O)C(C)C1 51871,C1(C(=O)NC2CC(CNC(c3cc(C4CCC4)no3)=O)C2)CC2(C1)OCCO2 51872,C12(C(N(CCNC(c3nn(CC)nc3C)=O)C)=O)CCC(C(F)F)(CC1)C2 51873,c1(C(=O)NCC=CCNC(c2occ(C)c2C)=O)c(O)cc(=O)n2c1CCCC2 51874,N1(C(C(C)N(C(=O)CNC)CCC)=O)CCC(CC(=O)O)C(C)C1 51875,c1(OC)cnc(Cl)[nH]c1=NC1CC2CCC1N(C(=O)CC1CC(C)OC1C)C2 51876,c1(C(N2CC(F)(C(=O)NCC3(CCO)CCC3)C2)=O)ncccc1Cl 51877,CC1COc2c(C(=O)NCCn3cc(CO)nn3)cnn2C1 51878,C1(CNC(c2cnc(C(C)C)s2)=O)CN(C(C2CSCCS2)=O)CC1O 51879,c1(C(=O)NC2(CNC(=O)C(Cl)=CCl)CC2)cccc(CO)n1 51880,C(=O)(CCCCCC(C)C)NCC1N(C(c2c(C)ccc(Cl)c2)=O)CC(F)C1 51881,N1(C(c2n(C)nnc2Br)=O)CCCC(C)(NC(=O)CC2C=CCC2)C1 51882,C1(CSC)CCCN1C(C1COCC1NC(C1(CF)CC1)=O)=O 51883,N1(C(C(c2cccc(O)c2)C)=O)CCC(F)(F)C(CNC(=O)CCF)C1 51884,N1(C(C=NOC)=O)CCC(N(CCO)C(C2CC2OC(C)(C)C)=O)CC1 51885,CCC(C(=O)N1CCN(C(c2ccnnc2O)=O)C(CO)C1)C(C)(C)CC 51886,CC1(C=CC(N2CCC(F)(CNC(C3CC4(CCC4O)C3)=O)C2)=O)CCOCC1 51887,S(=O)(=O)(c1cc(Br)ccc1Br)NS(CC1C(=O)CC1)(=O)=O 51888,C(=O)(C(C)C(O)CC)N(C)CC1CCN(C(c2nc(C(=O)OC)oc2)=O)CC1 51889,C(=O)(C(F)(CNC(c1ccccc1C1CC1)=O)C(C)C)N(CC=C)CC 51890,C1(CNC(C(CC)C2CCC2)=O)CCC2(CN(C(=O)CC3CCC3)C2)O1 51891,c1(-n2c(C(C)OCC(C)C)nc(-c3cnccn3)n2)ccc(Cl)c(Cl)c1 51892,CCC(CC)C(C(=O)NC1(C(=O)NCC(C)CC2CC2)CSC1)OC 51893,C(N=c1[nH]cnc(Cl)c1F)C1CN(C(C2(N(C)C)CCCCC2)=O)CC1(C)C 51894,c1(CC)nc2c(C(=O)NCC(C)(CO)NC(=O)C(C)C3CC3)ccnc2[nH]1 51895,CC1(C)CC(Cc2ccccc2)CN(CC(C2CC(F)CN2)C)C1 51896,CCC(CN=c1[nH]c(=NCCC(C)CCO)c2[nH]ccc2[nH]1)n1cccn1 51897,Cc1nnc2c(C(N3CCCOC(CNC(=O)C(C)(C)C)C3)=O)cccn12 51898,C1(C(C(=O)NC(c2cccnc2)C(=O)N(C2(CC)CC2)C)C)CCOCC1 51899,c1(OCC)cncc(C(=O)NCCCC(C)(C)NC(c2cccn2C)=O)c1 51900,c1(OC)cc(Cl)c(Br)cc1CN=c1[nH]c(-c2cccnc2C)cs1 51901,c1(C(=O)NC2CC(Nc3ncnc4scnc34)C2)cc2c(nc1O)CCOC2 51902,N1(C(c2c(SCC)cncc2)=O)CCC2(NC(c3cnc(Cl)s3)=O)CCCC12 51903,C(c1ccnn1C)=CC(=O)NC(C(=O)NC(c1n(CC)ncc1)C)c1ccoc1 51904,c1(C(C)=O)ccc(C(=O)NCC2(O)CC(NC(C3CCC(O)C3)=O)C2)o1 51905,CCCC(C(=O)N(CCNC(=O)Cn1cn[nH]c1=N)C(C)C)c1ccccc1 51906,C1(C(=O)NCC(CSC)OC)CCC(O)CN1C(=O)Cc1nocc1C 51907,N1(C(C2N(CCC)CCC2)=O)CC2CC(C(=O)NCc3cc(C)sc3C)(C2)C1 51908,C1(NC(c2cc(OC)n(C)n2)=O)CN(C(=O)CC2CCCS2(=O)=O)CCC1CO 51909,CC1CCN(C(=O)Cc2ccc(Br)o2)CC1NC(=O)Cc1ccccc1CO 51910,c1(C(=O)NC(C)CCCNC(c2cncc(Cl)n2)=O)nc2c(s1)CCCC2 51911,c1(COC)ccc(C(N2CC(NC(=O)CC3COC(=O)C3)CC2C)=O)cc1 51912,c1(C(N2CCSC2c2ccc(Cl)s2)=O)cccnc1NC(=O)Cn1cccn1 51913,CC(CC(F)F)C(=O)N(CCCCCCNC(C1(F)CCC1)=O)C 51914,C12(C(N3CCCC(CCC(=O)N(C)CCC4CCCC4)C3)=O)CCCC1C2(F)F 51915,n1(CC(=O)O)cc(C#N)c(O)nc1=O.c12cccc(c1[N+](=O)[O-])NCC2 51916,C(=O)(C(C)(C)C(c1nnnn1C1CCC1)NC1CC(=O)N(O)C1)OCC 51917,Cc1c(CC(=O)NCC2=CCN(C(C3(C#N)CC3C)=O)CC2)sc2ccccc12 51918,C(=O)(C(C)(C)C(=O)NCC(O)CN(C(=O)CCn1cc[nH]c(=O)c1=O)C)OC 51919,C1(CC=C)(NC(C2CC2(C)C)=O)CCN(C(=O)Cc2c[nH]ccc2=O)C1 51920,C1(F)(C(=O)NCC2(C(C)(C)C)CCN(C(C(C)SC)=O)C2)CC2(CCC2)C1 51921,c1(CC(=O)NCC2CC(NC(CCP(C)(C)=O)=O)C2)ccc2nsnc2c1 51922,c1(C(N2CC3C(NC(C(C)S(N)(=O)=O)=O)(C3)C2)=O)cccc2cc(O)ccc12 51923,N1(C(CC2(OC)CC2)=O)CC2OCCN(C(c3ccc4c(c3)CCN4C)=O)C2C1 51924,C(=O)(CCCCCCCCCO)NCC1C(C)(C)CN(C(C2C=CCCC2)=O)C1 51925,Cc1nc(N2CCC(NC(=O)C(C3CC3)C3CC3)CC2C)cc(C#N)n1 51926,c1(C(CC)N(C2C3CN(C(=O)C(OC)OCC)CC23)CC)ccc2c(c1)OCCO2 51927,C1(O)(CNC(C(CCOC)OC)=O)CCCN(C(=O)Cc2cnc(C)s2)CC1 51928,c1(CC(=O)NCC=CCNC(=O)CCCCc2cnc[nH]2)c[nH]c2ncccc12 51929,c1(C(=O)NCC2(CNC(CC(COC)(C)C)=O)CC2)cc(OC)c(OC)cc1N 51930,N1(CC)CCCCCC(N=c2[nH]c(N3CCC4(CC(F)C4)C3)nc3[nH]ccc23)C1 51931,CCCCCC(O)C(=O)N1CCCC1Cn1cc(CNC(C2(F)CC2)=O)nn1 51932,N1(C(C(C=C)O)=O)CCOC2(CCN(c3ccc(F)cc3[N+](=O)[O-])CC2)C1 51933,c1(C(=O)NC2CCCC(NC(CNS(NC)(=O)=O)=O)CC2)cn2ccccc2n1 51934,N1(C(CC2C(CC)C2(F)F)=O)CCC(NC(C2(C)CCCC2)=O)CC(O)C1 51935,CCC(O)CC(=O)NCC1CCC(NC(=O)CC2CSC2)CC1 51936,CCCC(CCCNC(c1ccc(=O)n(C)c1)=O)NC(c1sc(C)cc1C)=O 51937,c1(C(N(CC(C)NC(c2cc(CC)[nH]n2)=O)C)=O)ccc2cnsc2c1 51938,N1(CCN(C(=O)CCc2ccc(C(F)(F)F)cc2)C)CCN(C(=O)C2CC2)CC1 51939,c1(C(=O)NC(CC)CNC(=O)C(=O)N(C)C)cc2ccc(Cl)cc2o1 51940,C(=O)(C1CCCn2ncnc21)N(C)CC1CCCCN1C(=O)CCC[N+](=O)[O-] 51941,CC(C)(CO)C(=O)NC1(C)CCN(C(=O)COc2cccc(Br)c2)C1 51942,N1(C(C(C)Cc2ccc(Cl)cc2)=O)CC(NC(C2(O)CC2)=O)Cc2ccccc21 51943,C1(CNCC(=O)Nc2cn(C)c(-n3c(C)cc(C)n3)n2)CCn2ncnc2C1 51944,C1(COC)(CNC(=O)C(C)n2cccn2)CCCN1C(C1CC(CCO)C1)=O 51945,N1(C(CCC2(C)CC2)=O)CC(C2(NC(=O)Cn3cc(Br)ccc3=O)CC2)C1 51946,CC1CCOCC1C(=O)NCc1cccc(C(=O)NC2(CO)CCC2C)n1 51947,C=CC1(CNC(C2(C)CC(O)CN2C(=O)C(C)c2cccs2)=O)CCOCC1 51948,C1(C(=O)NCC2(C)CCN(C(=O)CCCCCF)C2)(COC)CCCNS1(=O)=O 51949,C1(C2(O)CCC2)(C(=O)NC2C(CNC(c3cnc(C(C)(C)C)[nH]3)=O)C2)CC1 51950,n1(CC(=O)NCCF)cc(CCc2ncc(C(=O)O)s2)nn1 51951,C1(COC)CC(O)CN1C(C1COCCC1NC(c1cc(Cl)n[nH]1)=O)=O 51952,C1(C(N2CC(NC(C=C(C)C(F)F)=O)C3(C2)CC3)=O)CCOCC12CCCCC2 51953,N1(C(c2c(C)nc(C3CC3)s2)=O)CCC(CNC(c2ccc(Cl)nn2)=O)C(C)C1 51954,C(=O)(C1CCCc2ncnn21)N1CCN(C(c2[nH]nnc2C2CC2)=O)CC(C)C1 51955,N1(C(c2c(C)c[nH]n2)=O)CCC(O)C(C(=O)NCc2ccccn2)C1 51956,c1(OC)ncc(CNC(=O)C(C2CCC(=O)N2)C)s1 51957,Cc1cc(C(=O)NC23CCCN(C(c4ccsn4)=O)C2C3)ccc1Br 51958,c1(CC2CCN(N(C)Cc3ccc(OCCCl)cc3)CC2)ccc2c(c1)OCO2 51959,N1(C(CCC(=O)NCC)=O)CCC(O)(CCNC(=O)CC23COCC(C2)C3)CC1 51960,c1(C(=O)NC2CCCC(N(C(=O)Cc3ccoc3)C)C2)ccc2ccn(C)c2c1 51961,c1(OC)cc(CNC(c2ccc(-c3ccnn3C)cn2)=O)ncc1C 51962,c1(C(=O)NC2CCC(NC(=O)C(F)=CC3CC3)CC2)cc2c(cn1)OCCC2 51963,N1(C(c2c(N)ncc(O)c2)=O)CCCC2(CCCCC2NC(C2CC23CC3)=O)C1 51964,C1(CNC(c2n(C=C)ncc2)=O)CC2CCC1N2C(C1SCCCS1)=O 51965,C1(NC(=O)CCCN2C(=O)CNC2=O)CC2CC(C1)N(C(c1nccs1)=O)C2 51966,C(C(O)CCNC(C1(n2nccn2)CC1)=O)N(CC(=O)NC(=O)C1CC1)C 51967,c1(C(=O)NC(CNC(C(c2ccc(CC)cc2)C)=O)C2CC2)cc(C)cc(N)c1 51968,N1(C(C(C(CC)CC)C)=O)CCC(NC(=O)CC2(C(=O)OC)CC2)C2(CCC2)C1 51969,CC1CN(C(C2(N=[N+]=[N-])CC2)=O)CCC1CNC(c1ccc(N)cc1F)=O 51970,C1(CNC(C(C)NC(N)=O)=O)CN(C(=O)CC2CC(F)(F)C2)CCC1(C)C 51971,N1(C(C2CC(C#N)(OC)C2)=O)CC(NC(c2ccc(OC)s2)=O)C2(CCC2)C1 51972,C=C(C)C(O)CC(=O)N1CC(C(N)=O)(CNC(c2ccnnc2C)=O)C1 51973,CN1CC(C(=O)NCc2occc2C(=O)NC(C2CCCO2)(C)C)CC1=O 51974,Cc1ncc(C(N2CCC(C(C)C(=O)NCCSCCO)C2)=O)n1C 51975,Cc1cc(Cl)ncc1CC(=O)NC1CCC(C(=O)NCC23CCCNC2C3)CC1 51976,CC1(NC(=O)N(CC(=O)NC2CCSCC2)CCCNC(=O)CSC)CCCC1 51977,C(C(CC(C)C)NC(=O)C(O)CCc1nccn1C)CC(CCC)OCC 51978,c1(-n2c(C(CC=C)CC)nc(-c3occc3C)n2)ccc(C)c(F)c1 51979,C=C=CCCC(=O)N1CC(CNC(C2CN(C)C(=O)N2)=O)C1 51980,c1(C(=O)NCC(C)CNC(c2nnn3c2CCC3)=O)nccc2ccncc12 51981,c1(C(N2C(CCNC(C(CC#C)O)=O)CSCC2)=O)cccc(F)c1C 51982,Cc1nc(CCC(=O)NC2CCCC2NC(c2cc(F)n(C)n2)=O)[nH]c1C 51983,CCC(F)(F)C(=O)NCC1CC(NC(c2cnc(C)nc2)=O)C1 51984,c1(C(N2CC3C(CNC(=O)C4=CC5CCC4C5)(C3)C2)=O)cc(Cl)cc([N+](=O)[O-])c1 51985,CC(C)(C)C(C#N)C(=O)N1CC=CC(C(=O)NCC2(N(C)C)CCC2)C1 51986,C1(CNC(c2c(SCC)cco2)=O)CCn2nccc2C1.N12CCC(C1)C2=O 51987,C(=O)(C1=NOC2COCC12)NC(C(C)C)CCNC(C1CC(n2cnnc2)C1)=O 51988,C1(C(=O)NC(C=C)(C)C2CC2)CC2(CCO2)C1 51989,N1(C(C(C)CC2CCCC2)=O)CCCCC(NC(c2cc(C(N)=O)ccn2)=O)C1 51990,C1(CC(=O)NC(c2c(C)nns2)C)CC2(CC2)CN1C(c1nnn(C)c1N)=O 51991,C(=O)(C(C)(C)CC(C)(C)C)NC1CCCCN(C(C(C(CC)CC)C)=O)C12CC2 51992,c1(N2CCC(CCNC(C(C)c3ccsc3)=O)C2)cc(=O)n(C)cn1 51993,C1(C(=O)OCC)CCN(C(=O)CN(C)CCOC(C)=O)CC1(C)C 51994,C1(C(N2CCOC(C(N3CC(O)(C4CC4)C3)=O)CC2)=O)CC2CCC1CC2 51995,CN=c1cc(C(N2CCC(N(CCO)CCO)CC2)=O)cc[nH]1 51996,CC(C)(CNC(C1CC1NCc1cccc(-c2ccccn2)n1)=O)C(=O)OC 51997,c1(CC(=O)NC(C)C(C)(C)NC(=O)CCCN2CCCC2)ccc2c[nH]nc2c1 51998,c1(C(=O)NC(C(N2CCCC(C=C)C2)=O)C2CCOC2)coc2ccccc12 51999,C1(NC(C2(CCOC)CCC2)=O)CCOC(C(=O)NCCC2CCN(C)CC2)C1 52000,N1(Cc2cncc(C)c2)CCC(C)(NC(C2CC2Cc2ccccc2)=O)CC1 52001,CC1CN(C(=O)CC2CC2CNC(=O)C=Cc2cccnc2)CCS1=O 52002,c1(OCCC)ccc(C(=O)NC2(CO)CCOC2)cc1OC 52003,C1(C(=O)NCCC(C)NC(c2cc(OC)n[nH]2)=O)Cc2cc(OC)ccc2O1 52004,C1(C(N(CCNC(=O)CCc2ccc(N)cn2)CC)=O)CCc2nn[nH]c2C1 52005,c1(C(N2CC(NC(C(C)SCCCC)=O)C(C)C2)=O)sc2nccnc2c1NC 52006,C(=O)(C1=CCCOCC1)N1C(C)CC(CCOC(C)(C)C)CC1 52007,C1(NC(C2CN(C(C)(C)C)C(=O)C2)=O)CN(C(c2cncc(Cl)c2)=O)CCC1F 52008,C(=O)(C1CCc2ccccc21)N1CCC(N=[N+]=[N-])(C(=O)NCC(C#C)C(C)C)C1 52009,N1(CC)CCOCC1C(=O)NCCCCC(C)NC(=O)C(C)(C)C1CCCCC1 52010,C1(C(N(C(C)C2CC2)C)=O)CCN(C(=O)C(CO)NC(N)=O)C(C)(C)C1 52011,CC1OCCCC1C(=O)NC1CCC(C(=O)NCC(F)CN(C)C)CC1 52012,C(c1ccccc1)=CCC(=O)NC1C(C(N(CCCC(C)C)OC)=O)C1(C)C 52013,C(=O)(C(O)C(C)(C)C)NCC(COC)NC(CC1(CCC#C)OCCO1)=O 52014,Cn1cc2c(n1)CCCC2C(=O)NC1CC(F)CN(C(=O)CC(C2CC2)C2CC2)C1 52015,C(=O)(C1=CCCOCC1)N1CC(COC)N(C(=O)C(n2cc(C)cn2)C)CC1 52016,CC1(C)CCC=C1C(=O)N1CCCCC1CNC(c1cn2cnnc2cn1)=O 52017,C(CC(F)(F)F)N(C)C(C1(CNC(=O)CC2CCOCC2)CC1)=O 52018,Cc1cccc(CC(N2CCC(NC(=O)CC3(c4ccccc4)COC3)C2)=O)c1 52019,c1(N2CC(C(C)NC(c3csnn3)=O)C2)c(F)cc([N+](=O)[O-])cc1F 52020,c1(C(=O)NCCCCNC(C(N)=O)=O)ncccc1Br 52021,c1(C2(CNC(c3n(CCCC)nnn3)(C)CCOCC)CC2)cc(C)cc(F)c1 52022,C1(NC(C=COCC)=O)CN(C(=O)C(=O)Cc2ccccc2)C2CCCCC12 52023,c1(C(=O)NC2(CNC(C(CSC)C)=O)CCCCC2)[nH]cc2c1CCS2(=O)=O 52024,c1(CC(=O)NC2CN(C(C(C)=C3CCC3)=O)CC(C)C2)ccc(S(N)(=O)=O)cc1 52025,CC1CN(C(=O)CCc2ccccc2)CC1NC(=O)CC1CCCN1C(C)C 52026,C1(CNC(c2scc(C(C)=O)c2)=O)CN(C(c2csnc2C)=O)CC1C 52027,CC(CCNC(C1CCN(C(C2(C#N)CC2(C)C)=O)CC1)=O)C(F)F 52028,c1(C(=O)NCC(C)N(C(=O)C(C2CCCCC2)F)C)cscc1C(N)=O 52029,c1(C(=O)NCCNC(C2(C(C)C)CNC(=O)C2)=O)cc2c(Cl)cccc2s1 52030,CC1CN(C(c2ncncc2Cl)=O)CC(C)N1C(=O)CCC1CCOCC1 52031,c1(C(N(C)CC2CCCN2C(C23CCC(C2)C3)=O)=O)cncc(S(C)(=O)=O)c1 52032,C1(C(=O)NCC(CNC(C2CCC(C(=O)OC)CC2)=O)(C)C)Cc2nncn2C1 52033,C1(NC(c2cccc(-n3cccn3)c2)=O)CC(F)CN(C(c2n[nH]cc2Cl)=O)C1 52034,c1(CC(N2CC(CNC(CC3C(C)C3)=O)OCCC2)=O)c(C)[nH]c2ccnn2c1=O 52035,CCC(C)(CNC(C1(NC(=O)CC2CCCCO2)CC1)=O)OC 52036,C=CCCC(CC(C)C)C(=O)NCCN(C(=O)CCC1(C)CC1)C(C)C 52037,c1(C(N2CCN(C(COCCC#C)=O)C(C(C)C)C2)=O)cc(Cl)cc2c1CCC2 52038,c1(C(N(CCCCCNC(C(CC=C)CC)=O)C)=O)ccc2c(c1)nc(C)n2C 52039,C(C1CN(C(=O)C(O)Cc2ccccc2)CC1C(=O)NCC(C)(O)C1CC1)=CC 52040,C1(c2cn(CCF)nn2)(C(=O)OC)CCN(C(c2ncc(Br)s2)=O)C1 52041,c1(C(=O)NCCOC2CCN(C(C3(CCCC)CCCC3)=O)C2)nccnc1C 52042,C1(CCNC(C2=CC(C)(C)C2)=O)CCN(C(C2CCCO2)=O)CCC1(F)F 52043,CCC(C(=O)OC)C(=O)N(CCC(=O)NC(c1nc(C(=O)NC)co1)C)OC 52044,C(C1CCN(C(c2nccn2C2CC2)=O)CC1)=CC(=O)NCc1c(C)cnn1C 52045,c1(C(c2n(C(CC)(C)C)nnn2)NCc2cnc(C)cn2)nc(C)c(C)[nH]1 52046,CN1CCN(C(C2CC(F)(CO)C2)=O)CC1CNC(C1CCS1(=O)=O)=O 52047,N#CC1CCC(CNC(=O)C(CCOCCO)NC(=O)CCF)CC1 52048,C1(c2cn(C3CC4(C3)CC4CO)nn2)(NC(CCC(=C)Cl)=O)CCCC(C)(C)C1 52049,c1(CCNC(=O)NCC2CCCCS2)ccc(Cl)cc1 52050,N1(C(C2N(C(CN(C(c3ccc(Br)cc3)=O)CCl)=O)CCC2)=O)CC2CCC1CO2 52051,c1(CNC(=O)CCOC2CC2)cnn2c1CN(C(=O)CC13CC(C1)C3)CC2 52052,C(=O)(C(C)(C)CS(C)(=O)=O)NC1CCCC(NC(c2cnc(C(C)C)nc2)=O)C1 52053,N1(C(c2cc(OC)n[nH]2)=O)CCCC(NC(c2ccc(F)c(C)c2)=O)CC1 52054,CN1CCN(C(c2cc(C3CC3)no2)=O)C(C(=O)N(C)Cc2ncnn2C)C1 52055,N1(C(Cc2cc(C)no2)=O)CC2CC1CN2C(c1cc(N(C)C)ccc1Br)=O 52056,Cc1cc(C(=O)NCC(O)CN(C(=O)Cc2c(C)noc2C)C)sc1Br 52057,C(C)(C(C)C(=O)NC(C)C)NC(C1(CC)CCC1)=O.C1CN(C(C)C)C1 52058,C(CC(C(C)(C)C)NC(c1cc(F)ccc1F)=O)N(C)C(c1ccc(F)o1)=O 52059,C1(NC(C(CC)n2cncn2)=O)CCC2(CC1)CN(C(=O)CC1CCC1)CCO2 52060,C=CC1(C(=O)C(=O)O)CCN(C(C2CCCCN2)=O)CC1 52061,C1(C(=O)Nc2n(COC)ncc2)(OCC)CCN(C(C2CCC(=O)N2)=O)C1 52062,N1(C(c2cc(C#N)no2)=O)CCOC2CN(C(=O)COc3cccc(F)n3)CC12 52063,O(NC(=O)CN=c1nc(OC(F)F)cc(C)[nH]1)CC 52064,CC(C)(C)C(CO)C(=O)N(C1(CNC(=O)CCCCCO)CCOCC1)C1CC1 52065,c1(C(=O)NCCC2CCN(C(C3CC3F)=O)C2)csc2cccc(F)c12 52066,C1(C(=O)NCC=CCNC(c2c(C)c[nH]n2)=O)CCc2nnc(O)n2C1 52067,CC(O)C(C(=O)NCC1(NC(c2csc(-c3cn[nH]c3)n2)=O)CCCCC1)N(C)C 52068,c1(C(N2CC3CN(C(C)=O)CC3C2)=O)cc2cc[nH]c(=O)c2s1 52069,C1(CNC(=O)Nc2cnc(C)o2)CCCN(Cc2ccccc2Cl)C1 52070,c1(NCC2CCC23CC3)c(Cl)cc(NC(=O)NC(C2CCCO2)C2CC2)cc1Cl 52071,CC1CN(C(=O)C=CC2COC(C)(C)O2)CCN1C(c1cncs1)=O 52072,C(=O)(CC(F)(F)C(F)F)NN1CCCN(CCNC(=O)CCC2CCOC2)CC1 52073,C1(CC(=O)N(CC(=O)NC)C)CC(C)N(C(c2ncsc2C)=O)C1 52074,C1(C(=O)NCCCCN2CCC2)CN(C(C2COCOC2)=O)CC12CCC2 52075,C(N=c1cc[nH]cc1S(=O)(=O)N1CCC(CN(C)C)C1)c1nnc(COC)s1 52076,c1(C(N(CCN(C(C2(CCC)CC2)=O)C)C)=O)nc(O)c(C)s1 52077,CCS(=O)(=O)CC(C)NC(c1cc(N(C)C)ccc1C)c1nnnn1CC(F)F 52078,c1(OCC(=O)NC2CCC(N3CCN(C(=O)C(F)F)CC3)CC2)ccc(F)cc1 52079,c1(C(=O)NCC(CO)NC(=O)Cn2cc(C3CC3)nn2)cc(C(F)F)ccc1F 52080,Cc1nc(C(N2CCC(C(=O)Nc3ccnc(F)c3Cl)CC2)=O)ccc1F 52081,c1(CC)ccc(C(=O)NCCC(C)NC(=O)CCC2CCC(=O)NC2)cc1 52082,C1(NC(c2c(C)nc(COC)s2)=O)CCN(C(=O)C=C(C)C(C)C)CC1C 52083,c1(CC)cccc(C(N2CCOCC2CNC(c2nnc(C)s2)=O)=O)c1N 52084,C1(C(=O)NCCC2(C)CCN(C(C=Cc3cn(C)nc3)=O)C2)CCCCN1N=O 52085,C12(C(N3C(C)(CC(=O)NC4(CCOC)CCC4)CC3)=O)CCCC1OCC2 52086,C12(NC(c3cnco3)=O)CC(CNC(c3cnn[nH]3)=O)(C1)C2 52087,O=S(=O)(c1ccc(Br)cc1N1CCSC1)N1CC2CC2C1 52088,C(=O)(C1=C(C)CCCC1(C)C)NCCC(CNC(c1cc(C)oc1)=O)O 52089,c1(C(=O)NCCN(C(COCC)=O)CC(C)O)sc2c(Br)csc2c1C 52090,c1(C(=O)NCC2N(C(Cc3cncc(C)c3)=O)CC2)ccc(C)cc1Cl 52091,CC1=NOC(=O)C1CCC(=O)NC1CC1CNc1cc(C(N)=O)ncn1 52092,c1(SC)ncc(CN2CCC(C(=O)Nc3nc(C(C)C)cs3)C2)c(Cl)n1 52093,C1(C(N(CCC(F)(F)F)CC)=O)CC2(CCC2)CN1C(=O)Cc1cnnn1C 52094,c1(C(=O)NCC(C)(C)OCCNC(CC2C(C)CCOC2)=O)cnn2c1CCC2 52095,C1(C(N(C(C)C)CCNC(c2cc(Cl)ncc2N)=O)=O)CCC2C1C2(F)F 52096,C1(C(N2CCN(CC(C)O)CC2)=O)CCN(C(=O)C2(C)CC(N=[N+]=[N-])C2)O1 52097,N1(c2c(C(C(=O)OC)=O)cccn2)CCCC2(C1)CN(C(=O)C(C)OC)CCO2 52098,C1(c2n(C)cnn2)CCCN(CCN2CCCCC2)C1 52099,CC1(C)CCC(CNC(=O)C(C)(C)C(N)=O)C(CN=c2nc[nH]s2)C1 52100,Cc1cc(C(N2CC3CC3C2C(N2CC3C(CO)C3C2)=O)=O)ncn1 52101,c1(C(C)C)cccc(C(N2CC(NC(C3CC4CCC4C3)=O)C(C)C2)=O)n1 52102,n1(CC)cnc2nc(=NC3C(C)C(OC)CC3C)[nH]c(NCc3ccc[nH]c3=O)c12 52103,c1(NC(C2CCN(Cc3cccc(F)c3Cl)C2)=O)ccc(I)c(Br)c1 52104,C1(NC(C(C2CC2)OC)=O)CCC(N(C)C(c2nnn(C)c2N)=O)CC1 52105,Cc1sc(O)nc1C(=O)NC1CCCCC1N(C)C(c1cc(C(F)F)ncn1)=O 52106,C(=O)(C1=CCC(C)(C)CC1)NC1(C(=O)NCC2(C(N)=O)CCCC2)C(C)CCC1 52107,N1(C(=O)OC(C)(C)C)CCC2(CCC2)C(NC(C2(S(N)(=O)=O)CCCC2)=O)C1 52108,c1(CNC(C2C(C(C)NC(C3CC34CCOC4)=O)C2)=O)cnccc1Cl 52109,Cc1ccnnc1C(N1CCCC1C(C)(C)C(=O)N(C)Cc1ncco1)=O 52110,c1(OC)nc(N2CCC2(C)C(=O)NCCN2CCCCCC2)ncc1Br 52111,N1(C(C2=CCCC2C)=O)CC(CO)C2(C1)CN(C(c1sccc1Cl)=O)C2 52112,C1(CC(=O)NCC(C)CNC(=O)Cc2cccc(N)c2N)CC2CCC(C1)C2 52113,c1(C(=O)NC2CCN(C(C3(C)CCCOC3)=O)C2)cccc(S(C)(=O)=O)c1 52114,CCC(CN=c1cccc(S(=O)(=O)NCCN(C2CC2)CC)[nH]1)N(C)C 52115,N1(C(c2cc(C)sn2)=O)CCC(C)(CC(N2CCC(F)CC2)=O)C1 52116,n1(CC)nc(C(=O)NC2CN(C(C3(Br)CC34CCC4)=O)C2)cc1C 52117,c1(OC)nc(C(=O)NC(C)(CNC(=O)CCc2nccs2)C2CC2)sc1C 52118,c1(CNC(C(CC=C)NC(C)=O)=O)nnn(C)c1C(=O)NC(CO)C(O)CCC 52119,c1(C(N(C2CCN(Cc3c(O)cccc3Br)C2)C)=O)ccc(O)c([N+](=O)[O-])c1 52120,C1(CC(N2CCC(NC(CCSC)=O)C2)=O)CCCC(C)C1 52121,N1(C(=O)Cc2cnoc2)CCC2CN(C(=O)Cc3cccc(F)c3F)CCC2C1 52122,c1(COC(C(OCC)NCC(C)(C)Cc2nc[nH]n2)=O)ccc(C(C)C)c(F)c1 52123,N1(C(c2ccc(CSCC)cc2)=O)CCC(O)C(NC(=O)CC(C)C(F)F)C1 52124,N1(C(CS(CC)=O)=O)CCC2(CC1)CC(NC(c1cnc(O)cc1C)=O)CO2 52125,C12(C(N(CC(C)O)CCNC(=O)CC(F)(F)F)=O)CCCC(CCC1)C2 52126,C1(C(=O)NCC(=O)OCC)(CC)CCCN(C(C2CC3CCCC3C2)=O)C1 52127,C(=O)(CCCCC(N)=O)NCC(CC)N(C)C(C1CCC2(CCC2)CC1)=O 52128,n1(Cc2n(CCCCC)nc(-c3ccnc(Cl)c3)n2)cc(Br)ccc1=O 52129,C1(C(=O)NCC(C)NC(=O)CC2CN3CCC2CC3)CCC2CC1C2(C)C 52130,CC1(C)COC(CCC(=O)NCCC2(O)CN(C(c3cc(O)cs3)=O)C2)C1 52131,c1(C(=O)NC)cccc(OCC(=O)NC2CCCC2NC(C2(C)CCCO2)=O)c1 52132,CC1(C)COc2cc(NC(C3CC4(CO)CC3C4)=O)ccc21 52133,N1(C(CC2(OC)CC2)=O)CCOCC1CC1CCN(C(=O)C(C)NC(C)=O)CC1 52134,N1(CC(=O)NC2CN(C(CCCCC#C)=O)CC2O)C(=O)NC(C)(CC)C1=O 52135,c1(NC)ncccc1C(=O)NC1CCCCC1NC(C1CC(C(=O)OC)C1)=O 52136,N1(C(N)=O)CC(O)CC1C(N1CCSCC1CCC(=O)NC(=O)CC(F)(F)F)=O 52137,C1(C(=O)NCC2(N3CCOCC3)CC2)CCOCCN1C(C1CC1F)=O 52138,Cc1cc(CCC(=O)NCC(C)NC(C2CCCC2C2CC2)=O)cc(C)n1 52139,N1(CCS(CC)(=O)=O)CC(=O)N(CC(C)(C)C(=O)OC(C)(C)C)C1=O 52140,CCCC(O)C(=O)NC1CN(C(c2ncncc2Br)=O)CC1C 52141,N1(C(CN(C(Cn2c(C)ccn2)=O)C(C)C)=O)CCC2CCN(C)C2C1 52142,N1(C(C(CCCC)O)=O)CCC(CNC(c2cccc(C)c2F)=O)C(F)(F)C1 52143,Cc1coc(C=CC(=O)NC2CN(C(=O)Cc3nn(C)cc3Br)CC2O)n1 52144,C(=O)(C(C)(C)C(=O)NCc1c(Br)nnn1C)NC 52145,CCCCC(CN=c1[nH]cnc(Cl)c1Br)NC(=O)C1CCc2ccccc21 52146,C(=O)(C(C)(O)CC(C)C)N(CCCNC(c1cc(OCC)cc(=O)o1)=O)CC 52147,CCCCCCC(=O)NCC1CN(C(C2CC3(c4ccc(F)cc4)CC2C3)=O)C1 52148,C1(C(NOC(C)C)=O)CN(C(C2CC(C)(C)CN2C)=O)CCN1C 52149,C(=O)(CC(C)CC(F)(F)F)NCCC1N(C(c2nc(C)[nH]n2)=O)CCOC1 52150,c1(C(=O)NCC2CCN(C(C(C)CF)=O)C2)cnnc2ccccc12 52151,N1(C(C2CC(C#C)(O)C2)=O)CC2CC(NC(=O)C(C)OCC(C)C)CC1C2 52152,Cc1ccc(N)c(C(N2CC(NC(c3cnn(CCO)c3C)=O)C3(CC3)C2)=O)c1 52153,N1(C(C(C2CCC2)OCC)=O)CCN(C(c2cccc(N)c2F)=O)CCC1C 52154,CCC(C)CC(C(=O)N1CC(C(N)=O)(N(C)C)C1)NC(=O)CCc1cccn1C 52155,Cc1cccc2oc(C(=O)NC3CC(O)CN(C(c4ncc[nH]c4=O)=O)C3)cc12 52156,CC1(C(=O)NC2CCCN(Cc3ccccn3)C2)CCCN(CCCl)C1 52157,c1(C(=O)NC2CC(C)CN(C(=O)CSCCC(F)(F)F)C2)cc2ccccn2c1 52158,c1(C(C(=O)N(CCCNC(=O)CNS(C)(=O)=O)C2CC2)OC)cnn(C)c1 52159,CN1CC2CC1CN2C(C1CC(NC(c2ncn3c2CCC3)=O)C1(C)C)=O 52160,c1(NC(CC(=O)Nc2cccc(OC)c2C)C)ccc2c[nH]nc2c1 52161,C(=O)(C(O)CC(=O)OC(C)(C)C)NCCC(C)(C)NC(c1cnc[nH]1)=O 52162,C(c1cnccn1)=CC(=O)N(C1CCCN(C(=O)C(C(C)C)C2CCC2)C1)CC 52163,N1(C(C2CCC(C)(CC)O2)=O)CCN(C(=O)CCCn2cccn2)C2COCC12 52164,N1(C(C=C(C)c2ccccc2)=O)CCNCCC12CC2 52165,N1(C(C(C)n2cccc2)=O)CCCCC(C2CN(C(=O)CCC(C)(C)C)C2)C1 52166,C1(NC(c2c(OC)cccn2)=O)CCN(C(=O)C(O)Cc2[nH]cnc2C)CC1F 52167,Cc1cc2nc(N3CCC(NC(=O)C(F)(F)c4cscn4)CC3C)cc(=O)n2o1 52168,c1(C(C(=O)NCC(CC=C)NC(=O)CCCOC)C)ccc(CC(C)C)cc1 52169,C1(NC(CCN(C)C)=O)CCCC1CC(=O)N(CC(F)Cl)C 52170,N1(C(C)=O)CCC(C2CCN(C(=O)Cc3ncc[nH]3)CC2)C1 52171,Cn1c([N+](=O)[O-])cnc1C(=O)NCC1(C)CC(NC(=O)CCc2ccoc2)C1 52172,N1(C(c2nc(=O)o[nH]2)=O)CCC2C(C1)OCCN2C(=O)CCc1ncc[nH]1 52173,C=CC1CN(C(=O)CCN(C)CC)CC1NC(C1CCN(C2CCCCC2)C1)=O 52174,c1(C(=O)NCC(CNC(c2cn(CCC)nc2C)=O)CO)coc2ccccc12 52175,c1(C(=O)NCCCN(C(C(CC=CC)C)=O)C)cc(OC)cc2ccoc12 52176,CC(C)(CC(F)C(=O)NCC1CC2CCC2C1)NC(=O)CP(C)(C)=O 52177,C1(CCNC(CCCc2c(C)ccs2)=O)COCCN1C(=O)Cn1cnc(=N)[nH]1 52178,N1(C(c2cncc(OC)c2)=O)CCC(NC(=O)CSCC(C)C)C(CO)C1 52179,C(=O)(C(CC)CC(F)(F)F)NCCCCC(CO)NC(c1cc(CCC)on1)=O 52180,CC(C)(CNC(C1CCC1C#N)=O)CC(=O)N1CCCCC1C1(O)CC1 52181,N1(C(C2(C(C)C)CCN(C(C3CC3Cl)=O)C2)=O)CCCCC(CO)C1 52182,C=C1CC2(C1)CC(C(=O)N(C(CNC(c1ncccc1F)=O)C1CC1)C)C2 52183,N1(C(C2C(C)(C(C)C)C2)=O)CC2(CCN2C(=O)CCN(S(C)(=O)=O)C)C1 52184,C1(NC(C(CC=C)CNC(C2(O)CCC(C)CC2)=O)=O)C2CCN(CC2)C1C 52185,C1(CN2C(CNC(CCn3cc(CCOC)nn3)=O)CCC2)CN(CC)C(=O)O1 52186,N1(C(c2n(C)ccn2)=O)CC=C(C(=O)NCc2ccc(F)c(F)c2)CC1 52187,CN1CCC(C(=O)NC2CS(=O)(=O)CC2NC(C23CC(C2)C3)=O)c2ccccc21 52188,c1(C(=O)NCC2C(NC(c3c(N)c(F)ccc3)=O)C2)cccc2c1OC(F)(F)O2 52189,C(=O)(CC1=NN(C)C(=O)C1)N(CCCNC(c1n(C(C)C)ncc1)=O)C 52190,C1(Nc2c(SC)scc2)CCCN(c2ccc(C(F)(F)F)cc2)C1 52191,C1(c2onc(C)n2)CCCCN1C(c1ncnn1C)C(=O)NC1(C)CC1 52192,c1(C(=O)NC2CCC(NC(C3(C#C)CC3)=O)C2)cc(OC)cc2c1NC(=O)CO2 52193,c1(C(=O)NC(C(C)C)CNC(c2coc(CO)c2)=O)cc(Cl)cn1C 52194,Cc1cccc(C(N2CCCC(C(C)Nc3nccnc3C#N)C2)=O)c1Cl 52195,C1(C(C)NC(CCCSC)=O)CCN(C(C2CCCC2SC)=O)CC1 52196,CCC(C)CC(C)NC(=O)C=CCNC(=O)COC1CCOCC1 52197,c1(OC)ccc(C)c(CN2CCC3(CC3C(=O)N(CC#N)CC#N)C2)c1 52198,N1(C(CC=C)=O)CC2CC(C)N(C(=O)CCOc3ccc(Cl)cc3)C2C1 52199,c1(OC(C)C(=O)N(CC(C)NC(C2(CN(C)C(C)C)CC2)=O)C)cccnc1 52200,c1(C(=O)NCC2C(NC(C3(CC)CCNC3=O)=O)C2)cnc(Cl)cc1N 52201,C12(C(=O)NCc3c(CC)nco3)CC(CO)(CN1C(C1(CC)CCNC1=O)=O)C2 52202,CCCCC(C)CCC(=O)NC(Cc1cnn(C)c1O)C(=O)NCC[Si](C)(C)C 52203,c1(CCCSCC)nc(-c2cccc(CCO)c2)n(C2CCCCC2C)n1 52204,c1(CCC)c(C(=O)NC2CC(CNC(c3cnnn3CC)=O)C2(C)C)cnn1C 52205,C1(C)(NC(C(CNC(CCOC(C)C)=O)(F)C(C)C)=O)CN2CCC1CC2 52206,N1(C(C(=Cc2cn[nH]c2)C)=O)CC2CCN(C(C3CCCCO3)=O)C2C1 52207,C(=O)(NNC(=O)C1OCCn2ccnc21)c1c(CN=[N+]=[N-])cc[nH]1 52208,N(C1COc2c[nH]nc21)C(CCC(CC)NC(c1cccc(F)c1N)=O)=O 52209,CCC(C)C(O)CC(=O)NCC(C)(F)CNC(c1ccnc2cc[nH]c12)=O 52210,O=C(CCCCCCBr)N1CCN(CNc2c(Br)cc(F)cc2Br)C2CC12 52211,C(CCO)(C(=O)N1CC(NC(C2CCN(C)C2=O)=O)C1)N(C)C 52212,C(CCC(C)C)(C(=O)NC1CN(C)CC1OC)NC(CN(C)CC)=O 52213,N1(C(C2(CC#C)CC=CCC2)=O)CCC2(CC1)CN(C(c1nccnc1C)=O)C2 52214,CC(CCC(=O)NCC1COC(C)(C)C1)NC(=O)C(F)C1CCC1 52215,c1(CF)cccc(CNC2CCCCC2OC(F)F)c1 52216,Cc1ncc(C#N)c(N(C)CC2CN(C(c3c(C)cc(O)cc3O)=O)C2)n1 52217,C(CC(F)F)(C(=O)NC1CN(C)NC1=O)NC(C1CCC(=C)CC1)=O 52218,C1(NC(=O)NCCC(C)N(CCC)C)CSC(c2ncccc2O)=N1 52219,N1(C(c2cc(OC)no2)=O)C2CCC(C2)C1Cc1cc(C(=O)OC)ccc1F 52220,C(c1cncn1C)=CC(=O)NC1CC(CNC(CSCCC)=O)C1 52221,CC(C)CCC(O)C(=O)NCC(C1CCN(C(c2cc(Cl)nnc2O)=O)CC1)C 52222,n1(CC(=O)NCC2N(C(COCC(=C)C)=O)CCC2C)cccc(C)c1=O 52223,CCC(CN(C)C)CC(=O)NC(C)(CSC)C(=O)NCCCCN(C)C 52224,CC1C2CC(C2NC(=O)CSc2cccc[n+]2[O-])N1C(=O)CSC1CCCCO1 52225,C1(CC)CCN(C(C2CN(C(=O)C=C3CCOCC3)CCO2)=O)CCO1 52226,C1(C(N2CC(CC(=O)NC3CCCC3CCO)(OC)C2)=O)CC(O)C(F)C1 52227,N1(C(CSc2ccc(OC)cc2)=O)CCN(C(c2ccccc2Br)=O)CC1C 52228,N1(Cc2ccc(C3CN(C(c4ccc(OC)cc4)=O)C3)cc2)CCCC(C)(O)C1 52229,C1(C(=O)NC2CCCC(N(C(=O)C=CBr)C)C2)CC2(CCC2=O)C1 52230,C(=O)(C#CC1CCCCO1)NC1CCCN(C(C(C)=C2CCCC2)=O)C1C 52231,Cc1[nH]c(C#N)cc1C(=O)NC(C)(CNC(C1CC2CC2C1)=O)Cn1cccn1 52232,c1(CCNC(CC2(OC)CCC2)=O)cnn(CC(=O)N(CCC(=O)OC)C)c1 52233,N1(C(CC2N(C)CCC2)=O)CC2N(CCSC3CCCO3)CCC1C2=O 52234,CCC(CC)C(C)C(=O)N(C(C)CCNC(c1cccc(COC)c1)=O)C 52235,CC(C)(CCC(=O)N1CCC(=CCNC(=O)CC2CCC(=O)N2)CC1)[N+](=O)[O-] 52236,C1(CN2CCC(C(C)C)C2)CCC2(CCC3(CC2)OCCO3)O1 52237,C=CC1(C(=O)N(C)Cc2cscn2)CCN(C(c2cc(CCC)on2)=O)C1 52238,N=c1cc(C(=O)NCC2(CNC(=O)C=Cc3ccc(Cl)s3)CC23CCC3)cc[nH]1 52239,C1(CNC(c2c(CC)c[nH]c2)=O)CCCC(CNC(=O)CCC2CCCCO2)C1 52240,CC(CC(C)(C)C)C(F)C(=O)N(C)CC1(O)CN(C(C2CCC3CCC2O3)=O)C1 52241,c1(CC)nc(C(N2CCC(C(C)NC(C3(CO)CCOC3)=O)CC2)=O)c(N)s1 52242,c1(CC)cc(C)ccc1C(=O)NCC(C(C)(C)C)NC(=O)C=Cc1cocn1 52243,N1(C(C=CCC)=O)CCOCC(CNC(C2CCC(=O)N(C(C)C)C2)=O)C1 52244,c1(NC)ccc(C(=O)NC2CC2CNC(c2sc(F)cc2C)=O)c(Cl)c1 52245,C1(C(=O)NCC2(OCC)CN(C(=O)CC3C=CCC3)C2)CCn2ccnc2C1 52246,C1(F)(C(=O)NC2CCCCN(c3c(C(=O)O)cncn3)C2)CCCCC1(F)F 52247,N1(C(CCC=CCC=C)=O)CC(C)CCC1CNC(=O)Cc1cnsc1 52248,C1(NC(c2ccncc2F)=O)CCCC12CN(C(c1sccc1F)=O)C2 52249,CC1CCN(C(C2(O)CC2)=O)C1CNC(c1cnn(C2CC2)c1)=O 52250,N1(C(c2cnc(OC)s2)=O)CC2CC(C)N(C(C3(F)CCCCC3)=O)C2C1 52251,CC1(C(N2CCOC(CNC(=O)CSCc3ccncc3)C2)=O)CC(C#N)C1 52252,C(=O)(C(C)(C)S(C)(=O)=O)NC1CCC(NC(c2c(NC)ccc(F)c2)=O)C1 52253,C1(C)(CNC(C2C=CC(NC(C3C(C)C3C)=O)C2)=O)NC(=O)NC1=O 52254,C(C(C)(C)CC(=O)NCC1(C)CCN(C(c2ccc(C3CC3)c(F)c2)=O)C1)OC 52255,c1(N2CCC(NCc3cn(C(C)(C)C)nc3)CC2)ncccc1C#N 52256,CC(C)CC(CNC(C1(P(C)(C)=O)CC1)=O)NC(C1CCCC(CF)C1)=O 52257,N1(C(CN(C(C)=O)C)=O)CC2CC(C1)CN(C(=O)C(c1ccc(F)c(F)c1)O)C2 52258,c1(CC)cccnc1C(=O)NCC1C=CC(NC(=O)CC2CCSCC2)C1 52259,O=C(C(=O)N=c1nc[nH]n1-c1ccccn1)N1CCC(C(O)CO)CC1 52260,n1(CC)nc(C)c(C(c2nnnn2C(C)C)Nc2cncc(Br)c2C)c1Cl 52261,c1(CNC(C2CCCNC2=O)=O)ccccc1F 52262,C12C(C1(C)C)C(=O)NC2=O.C(=O)(C(=O)NC1CC1)NC(c1nn[nH]n1)C 52263,c1(C(=O)NC(CNC(C(CCCC#C)C)=O)C)cc(C)c2occc2c1 52264,CC1CC(C)N(C(c2nccc(N)c2Cl)=O)CCN1C(c1cnns1)=O 52265,n1(CC(=O)NC2CC(CNC(=O)CC3(CC4CC4)CC3)C2)nnc2c1CCCC2 52266,N1(C(C2ON=C(C)C2)=O)CC(NC(=O)C(C)N2CCC2)C(CO)C1 52267,C12(C(=O)NC(C(C)NC(=O)C=CC3CCCCC3)C)CC3CC(CC(C3)O1)C2 52268,O=C(C#CC1CCC1)NC1CC(NC(=O)C=CCN2CCCCC2)C12CCC2 52269,C1(CNC(Cc2c(C)nc[nH]2)=O)CCCCCN1C(c1cnn(CC2CC2)c1)=O 52270,c1(CN2C3CN(C(=O)Cn4cc(Br)cn4)C(C3)C2)cc(F)c(F)c(Cl)c1F 52271,N1(C(c2cc(OC)ncn2)=O)CC2(CCN(C(c3ccc(Cl)nc3Cl)=O)C2)C1 52272,C12CCCC1(C)N2.n1(C(CN(C(CSSC)=O)C)C)nccc1CN1CCCC1 52273,C1(CCC(=O)NCC2CCCC2C(=O)NCC2CCCO2)CC(F)(F)C1 52274,c1(C2OCCN(C(c3cc(Br)cc(Br)c3)=O)C2)cc(F)c(Cl)cc1Cl 52275,CC(C)C(C(=O)NCCCS(N)(=O)=O)NC(=O)Cn1cnnn1 52276,c1(C(=O)NC2CC2C(N2CC3CCCCC3C2)=O)cn2c(Br)cccc2n1 52277,C1(CC(=O)NCC(CCNC(C2C(COC)(COC)C2)=O)O)CCS(=O)(=O)CC1 52278,c1(OC)cc(C2CC2)ccc1C(=O)NC1CN(C(C23CCC(C2)C3)=O)CC1C 52279,N1(C(CC(=O)OCC)=O)CC2(CCC2NC(=O)C(O)CCSC)C1 52280,CC(CO)C(=O)NCC(C(=O)NC(c1cnn[nH]1)C)N(C)C 52281,C1(C(NOCCC(C)C)=O)CCOCCN1C(=O)CCc1ncccn1 52282,c1(N(C(C)CNC(C2(C3CCCCO3)CC2)=O)C)ncnc(Cl)c1CO 52283,C(C(O)C(=O)NCCCCCNC(=O)C(C)OC1COC1)=CCCC 52284,c1(OC)ncc(C(F)(F)F)cc1C(N1CCC(CN(C)C(C)=O)CC1)=O 52285,CCC(C)(C)CCCC(=O)NCCN(C(c1cc(O)n(C)n1)=O)C(C)C 52286,c1(NCc2c(OC)cccn2)cc(=NC(C)c2c(F)cccc2Br)[nH]c(C)n1 52287,C(=O)(C1=CCC(C)CC1)NCC1CCC(C(N(C)CC2CCN(CC)C2)=O)CC1 52288,n1(C(C(N2CCC(CCNC(C=CCCC)=O)CC2)=O)C)nc([N+](=O)[O-])cc1C 52289,c1(NCC(N2CCN(C(=O)CC3C=CS(=O)(=O)C3)CC2)=O)cccc(F)c1 52290,c1(C(N2C(CNC(CC(C)SC)=O)CCC(C)(C)C2)=O)cnc2sc(C)c(C)n12 52291,C(=O)(C(C)(C)CCC#N)NCCC1CCN(C(c2c(C)nc(Cl)cc2)=O)C1 52292,c1(CC(N2CC(NC(C3CCOC3)=O)CC(C)C2)=O)cccc2cccnc12 52293,c1(C(=O)NC2C(NC(c3c(CC)n[nH]c3)=O)COCC2)n[nH]c2c1CCC2 52294,S(=O)(=O)(c1ccc(N2CCN(C(C3CC3(C)C)=O)CC2)nc1)NCCCCCC 52295,c1(C(=O)NCC2(C)CCN(Cc3c(C)c(F)ccc3)C2)cc2[nH]ccc2cc1Cl 52296,C=CC1CN(C(c2c(C)nn(C)c2C)C(=O)NC2CCC2)CC1O 52297,C#CCCC(O)C(=O)NC1(CO)CCCN(C(c2c[nH]nc2CC)=O)C1 52298,C1(CCOC)CN(C(C2CC(C)(C)O2)=O)CCN1C(=O)C=C1CCCC1 52299,c1(C(N2CC(NC(Cc3c(C)non3)=O)C(C)C2)=O)cnc2sccc2c1 52300,N1(C(c2c(C)nn(C)c2C)=O)CCN(C(c2cccc3c2CCC3)=O)CC(O)C1 52301,C1(NC(c2c(C)cns2)=O)CN(C(C2CC(F)C(=O)N2)=O)CC2(CCC2)C1 52302,C(=O)(CCCC(=O)N1CC=CC(NC(=O)C(C)C(C)O)C1)NC 52303,c1(OC)ccnc(NCC(=O)NC2CC2CNC(c2cc(Cl)cs2)=O)n1 52304,N1(CCNCc2nc(CC)sc2)CCN(C(c2ccnc(CC)c2)=O)CC1 52305,C1(C)(C(=O)NCC(C2(O)CCN(C(C(C)OC(C)=O)=O)C2)C)CCCN(C)C1 52306,N1(C(CC(CN(C)C)O)=O)CC=C(CC(=O)N2CCCC(CCO)CC2)CC1 52307,N1(C(c2ccc(NC)cc2)=O)CC2CCCC2C1C(=O)NCc1ccncc1 52308,c1(N(C(C)=O)C)ccc(NC(C2CCCN(Cc3ccncc3)C2)=O)cc1 52309,c1(C(=O)NCCCOCCC(=O)N(C(C)CCO)C)cnn(C)c1 52310,C1(C(=O)NC2CC(CCNC(Cc3c(C)cc(C)s3)=O)C2)CC2CCCC2C1 52311,CCC(C)C(O)C(C)C(=O)N1CCOC(CN(C(=O)CCC(C)C)C)C1 52312,C(=O)(C1Cc2ccc(Cl)cc21)N1CCCC(NC(c2cc(F)c(F)cc2O)=O)C1 52313,c1(OC)ccc(CC(N2CCC2CNC(C2C(Cl)(Cl)C23CC3)=O)=O)cc1OC 52314,N1(C(C2C(NC(c3c(C)[nH]c(C)c3C)=O)COCC2)=O)CCCC2(CC(O)C2)C1 52315,c1(C(=O)NCC(CNC(C(C)OC)=O)CO)c(Cl)ccc(Br)c1F 52316,c1(C(=O)NCCC2N(C(C#CC(C)C)=O)CCCC2C)ccn2ccnc2n1 52317,Cc1ccc(C(N2CCCC2CNC(=O)CNC(c2ccc(Br)o2)=O)=O)nn1 52318,C(=O)(CCCCCC(C)(C)C)NC1CN(C(c2c(C)oc(Cl)n2)=O)CC1F 52319,C1(CNC(c2nc(C(N)=O)sc2)=O)CC(F)CN1C(C1CC(N2CCOCC2)C1)=O 52320,C1(NC(CCCc2onc(C)n2)=O)COCCN(C(C2CC(N=[N+]=[N-])C2)=O)C1 52321,CC1(C)CN(C(C2CC(F)C(=O)N2)=O)CC(C)(C)C1 52322,C#CC1CCCC(NC(C2CCOC2CNC(=O)Cc2c(C)cnn2C)=O)C1 52323,C(=O)(CC1=CCOCC1)NC(CC(=O)NCC1(CCO)CCC1)C(F)F 52324,N1(C(CC2(CC)CC2)=O)CCC(O)(C(C)NC(C2CCCC(O)C2)=O)CC1 52325,N1(C(c2c(C)cco2)=O)CCC(NC(c2cnc(-c3cccs3)s2)=O)C(F)C1 52326,C=CCC(C)(C)CC(=O)NC1CC2CC1N(C(c1coc(OCC)n1)=O)C2.CN 52327,c1(OC)ccc(C(=O)NCC2CC2NC(c2ccnc(C)c2)=O)c(Br)n1 52328,C1(C)(NC(C(n2c(C)ncc2)C)=O)CCN(C(C2(C(C)C)CCCO2)=O)C1 52329,C(=O)(C(C)=Cn1ccnn1)NCc1ccc(CCNC(CC(=O)OCC)=O)cc1 52330,C(=O)(C1CCCc2ncccc21)N1CC(OC)(CNC(=O)C=C2CCOCC2)C1 52331,C1(CNC(c2cncc(C)n2)=O)CCC2(CCN(C(=O)C3=CCC3)CC2)CO1 52332,C(=O)(CC(O)CC(C)C)NC(CCSC)C(=O)NCC1(C)CC(C)C1 52333,N1(C(C(CC)C)=O)CCC2(CCCC2CNC(=O)CCOCC(F)(F)F)CC1 52334,C1(CC(=O)NCc2cccc(F)n2)C2CCC(C2)N1C(=O)C(c1ccccc1)F 52335,C(=O)(CCC(O)C(C)(C)C)N1CC(CNC(C2(CC#C)CCCO2)=O)C(C)C1 52336,C(=O)(C(O)CCc1ccccc1)NC1C(CNC(=O)C(c2ccccc2)O)COC1 52337,n1(CC(=O)OC)cc(C2(O)CN(C(C3CC3c3ccccn3)=O)C2)nn1 52338,CC1(C)CC(NC(=O)CCc2ccc(F)cc2Cl)CN(C(=O)Cc2nc[nH]n2)C1 52339,c1(C(N2CCC(NC(c3c(C)[nH][nH]c3=N)=O)C2)=O)ccc(C)c2c1CCC2 52340,Cc1nc(NCC(C2CC2)NC(=O)CC(O)C(C)C)c(C)c(O)n1 52341,n1(CC)ncc(C(=O)NCc2ocnc2C(=O)NC2(C)CCOC2C)c1C 52342,N1(C(CC(C)F)=O)CCN(CC(C)(C)NC(c2cc(CCO)on2)=O)CC1 52343,N1(C(=O)CCOC2CC2)CC2CC1CN2C(c1ccc(Br)c(Br)c1)=O 52344,c1(C(=O)NC(CN(C(c2n[nH]cc2Br)=O)CC)C)ccc(C)cc1 52345,C1(NC(C=CSC)=O)C(C)CCN(C(c2cnc(C3CC3)o2)=O)C1C 52346,CC1CCCCC1(C)C(=O)NC1CCCN(C(c2csc(O)n2)=O)C1C 52347,N1(C(CS(CC)=O)=O)CCCCC2(CCN(C(c3ccc(C4CC4)nc3)=O)C2)C1 52348,N1(C(C(CC(=O)OC)N(C)C)=O)CC2CCC1CN2C(c1coc(N(C)C)n1)=O 52349,N1(C(=O)Cc2cccc(F)c2)CCCN(C(C2(F)CCC2)=O)CC1CO 52350,C1(CCCC(N2CC(O)(CCNC(CCC3(C)CC3)=O)C2)=O)CCCC(=O)N1 52351,N1(C(C=CC=CC)=O)CCCCC2(C1)CN(C(c1ccc(OCOC)cc1)=O)C2 52352,c1(C(=O)NC2CC3CN(C(C(C)OC)=O)CC2C3)cc2cccc(C)c2o1 52353,C1(C)(CNC(c2ccc(C)o2)=O)CCCN(C(C2CC3(CC3)CN2C)=O)C1 52354,C1(C(N2CCC(NC(c3c(C)[nH][nH]c3=N)=O)CC2)=O)CCC2(CCC2)O1 52355,C(=O)(C(C(C)(C)C)n1cc(C2(C(=O)O)CCCC2)nn1)NC1(C(C)=O)CCC1 52356,c1(C(=O)Nc2scc(CN(C)C)n2)ccc2cc(I)ccc2n1 52357,Cc1cc(C(=O)NC(C(=O)N(C)Cc2nc[nH]n2)C2(C)CC2)ncc1N 52358,N1(C(C2(C)CCCN2C(c2cnn3ccncc23)=O)=O)CCn2cccc2C1 52359,CCCCC(CC(=O)NCC(F)(F)C(C)C)NC(c1cc(C)ncn1)=O 52360,C=CCCCCCCCCC(C)NC(=O)CNc1ccccc1CC(=O)OC 52361,CCCC(C(=O)NCC(F)CNC(c1ccccc1Cl)=O)NC(N)=O 52362,Cc1ncnc(C)c1CC(N1CC(O)(CNC(C2(F)CCCN(C)C2)=O)C1)=O 52363,C=CC(CC)CC(=O)N1CC2CC2(CNC(=O)CN(C)Cc2ccc(C)cc2)C1 52364,CC1(C)NC(=O)CCC1NC(C1CC(NC(=O)C=Cc2ccco2)C1)=O 52365,CCCC(CC)CCC(=O)N1CC(C(=O)OC)C1.c12cc(cs1)C(=O)NC2 52366,CC1CN(C)CCN1C(C1CC2(CC2)CN1C(=O)Cc1nccn1C)=O 52367,n1(CC(=O)NC(C)C(C)NC(=O)Cc2cccc(F)c2)nnc2c1CCCC2 52368,O=C(C1=CCSC1)NC1CN(C(=O)Cc2ccccc2O)CC1c1ccccc1 52369,C12(C(=O)NCCCN(C(C3CCCC(=O)N3C)=O)CC)CCC(C)(CO1)C2 52370,C(C1CCc2nccn21)NC(C1=NOC(CNC(C(CC)OC)=O)C1)=O 52371,c1(SC)ccccc1C(=O)NC1CN(C(=O)COc2ccsc2Cl)CC1F 52372,C1(CN(C(CC(C)C2CC2)=O)C)CCC(NC(C2COC(=O)O2)=O)CC1 52373,C1(NC(CC2C(C)OCC2)=O)CC(C(=O)NCC2CC2CCN=[N+]=[N-])C1(C)C 52374,Cn1ncc2cccc(-c3nc(C4CCOC4)nn3-c3ccnc(O)c3)c12 52375,N1(C(Cc2c(C(=O)OC)csc2)=O)CCCC(CNC(=O)COCC(F)F)CC1 52376,N1(CC(=O)NCC(CN(C(=O)C(C)C2CCOC2)CC)(C)C)CC(=O)N(C)C1=O 52377,c1(C(N(CC(C)NC(=O)COc2cn[nH]c2)C)=O)c[nH]c2nccc(Cl)c12 52378,C1(CCNC(c2cn(C(C)C)nc2)=O)CCCN(C(=O)Cc2ccsc2)CC1 52379,c1(C(=O)NCC(CC(C)C)NC(C(CC)(C)C)=O)ccc2c(c1)CCCC2 52380,CCCCC(O)C(=O)N1CCCC1CNC(=O)CCc1ncc(F)cn1 52381,Cc1cnc2cc(C(=O)NC3CC(CNC(=O)COC4(C)CCCC4)C3)nn2c1 52382,CCC(CC1CCCC1)C(=O)NC1CCOC(CNC(=O)C=C2CCCCC2)C1 52383,N1(C(C2CCC(C)C2)=O)CCC2(CCN2C(=O)NCC(F)(F)F)C1.C(C)(C)(C)O 52384,C(CCCC(=O)NCC(C)NC(=O)Cn1nnc(-c2cccs2)n1)OCC 52385,N12CCC(C1)CC(=O)N(C(CCO)c1ccsc1)C2=O.C1(C(C)(C)C)CCCC1 52386,c1(CNC(c2ccn(CC)c2)c2nnnn2CCOC)ccc(S(C)(=O)=O)cc1 52387,N1(C(CN(CCC)C(c2ccc(C#N)cc2)=O)=O)CCS(=O)C(C)C1 52388,c1(OC)ccc(N(C2(C(=O)Nc3nc(C(C)(C)C)co3)CNC2)C(C)=O)cc1 52389,C1(CNC(c2cnc(C)[nH]2)=O)CCN(C(=O)Cc2ccc(C(F)F)cc2)C(C)C1 52390,c1(NC(c2nnc3ccccn23)CC)nccc(=NC2CCN(S(C)(=O)=O)C2)[nH]1 52391,C1(C(C)NC(=O)Cc2ccon2)CN(C(=O)CC2NC(=O)NC2=O)CCO1 52392,N1(C(CC2CCN(C(C(C)CO)=O)CC2)=O)CCCCCC1CO 52393,c1(CC(C)C)ccc(C#N)c(N2CC(CN(C)C(C3C=CC=CC=C3)=O)C2)n1 52394,c1(C(N2CC(CCNC(C3C(OCC)C3)=O)OCC2)=O)cnc2c(n1)CCCC2 52395,c1(C(=O)NCC2(CNC(Cn3ccc(C)n3)=O)CC2)c(C)cc(Cl)cc1C 52396,Cc1ccccc1C(=O)NCCCCCNC(C1CCC(C(F)(F)F)C1)=O 52397,c1(C(=O)NC(CC2CCC2)C(=O)NCc2cncs2)cccc[n+]1[O-] 52398,N1(C(c2nc(CC)[nH]n2)=O)CC(NC(=O)C(C)CCOC)C(C)(C)C1 52399,c1(CC)ccc(C(=O)NCC(C2CCC2)NC(=O)CC(=O)OC)cc1[N+](=O)[O-] 52400,c1(C(=O)NC2CC(C)(CNC(C3(C=C)CC3)=O)C2)c(C)nc2sccn12 52401,c1(C(=O)NC(CN(C(C2C(OCC)C2)=O)C)(C)C)cnc(Cl)s1 52402,c1(C(N2CC(NC(=O)Cn3nccn3)C(O)C2)=O)ccc(Cl)c2ccccc12 52403,C(=O)(CCCC(C)NC(=O)C(C)COC)N1CC(CC)N(C)CC1 52404,C(=O)(C(O)CCCNC(=O)CCCc1ncco1)N(CCC(=O)NC)CC 52405,C(=O)(C(C#N)C(C)C)NCCCCNC(C(C(C)C)SC)=O 52406,CC1(C)CCCN(C(=O)COc2cccc(F)n2)C1CNC(=O)Cc1ccoc1 52407,c1(N(CCC)CC2CC(F)(F)C2)cc(OC)c(OC)c(Cl)c1 52408,n1(CC)nc(C)cc1C(=O)NC(C(=O)NCC1(CC)CCC1)C1(C)CC1 52409,c1(C(N2CC3C(NC(C4(C)CN(C)C(=O)C4)=O)C(C3)C2)=O)cc2c([nH]1)CCCC2 52410,C12(C(=O)NCC3(NC(CNC(N)=O)=O)CCCCCC3)CCCCC1C2(F)F 52411,c1(C(CN2CCC(NC(=O)NCc3n(C)ccn3)CC2)=O)c(Cl)cccc1Cl 52412,CN1CC(C)(C(N2CC(N(C(=O)CSc3nncn3C)C)C2)=O)CCC1=O 52413,C1(NC(CCC2CC(OC)C2)=O)CC2CCC1(C(N1CC(C3CCCO3)C1)=O)C2 52414,C1(CC(N2CC(N(C)C(c3ccncn3)=O)C2)=O)NC(=O)CN(C)C1=O 52415,N1(C(=O)Nc2cn(C(C(=O)OC)(C)C)nc2)CCC(=O)N2CCCCCC12 52416,C1(CCC)CN(C(=O)CC(F)(F)CC)CCN1C(c1cc(F)ccc1OC)=O 52417,C1(CC)CC(O)CCN1C(C1CCOC1CNC(c1cnnn1C)=O)=O 52418,CCC(CC)C(=O)NC(Cc1cnn(C)c1O)C(=O)NCCc1noc(=O)n1C 52419,c1(SCC(=O)NCC(F)CNC(=O)CCN2CCOC2=O)ccccn1 52420,C1(NC(C(C(C)C)O)=O)CCC(C)N(C(C2C3CCC2(C)C3(C)C)=O)C1 52421,C=C(C)C1OCCC1CNC(=O)CC1CC(C(=O)OCC)C1 52422,C1(C(CNC(C2C(CC)C2)=O)(C)O)CCN(C(C2(C(N)=O)CC2)=O)CC1 52423,Cc1ccn2c(C(N3CCOC(CCNC(c4ccccn4)=O)C3)=O)cnc2c1 52424,C1(NC(c2cc(CC)nn2C)=O)CC2CC1CN(C(=O)CCNC(=O)COC)C2 52425,C1(CNC(C2CCS2(=O)=O)=O)CCN(C(c2csc(C(F)(F)F)c2)=O)C1 52426,c1(C(N2CC(C)C(CNC(c3cc4c[nH]nc4s3)=O)C2)=O)cc(N)c(Cl)c(O)n1 52427,C(=O)(C1=NOC(C)(C)C1)N(C1CCCC(NC(c2c(CC)[nH]cc2)=O)C1)C 52428,c1(CNC(c2c(C)c[nH]n2)=O)cccc(C(=O)NC(C)CN2CCCC2=O)n1 52429,C#Cc1cccc(CC(=O)NCC2(NC(c3[nH]c(C)nc3C)=O)CCOCC2)c1 52430,c1(C(=O)NCC(CC)NC(=O)C(F)(F)c2csc(Cl)c2)n[nH]c2c1CC(C)CC2 52431,S(=O)(=O)(c1cccc(NC(=O)COCCOCCN)c1)NC 52432,C#CCCCC(C)C(=O)NC1CC(C(=O)NC(C)CN2CCCC2)C1 52433,Cc1cc(C(N2CCC3(NC(c4ccon4)=O)CC3C2)=O)cc2c1NCCC2 52434,C1(C(=O)NCC2COC3CC2C3)CCC2(CCOCC2)C1 52435,c1(C(=O)NCC2(NC(CCC3CCC(C)O3)=O)CC2)nc(N(C)C)nc(=N)[nH]1 52436,C(=O)(C(C1CCCC1)NC(=O)CN(C)C(C)=O)NCC(C)OCC#C 52437,N1(CC(=O)NC(C(C)C)CNC(c2cc(Cl)n[nH]2)=O)CCC(=O)NC1=O 52438,C1(N(C(C(F)=CC)=O)CCF)CCCN(C(c2ccn(CC)n2)=O)C1 52439,n1(C(C)C)ncc(C(=O)NCC2(NC(C3C(C)C3C)=O)CCOC2)c1Cl 52440,O=S(=O)(c1ccc(Cl)cn1)NC1CCN(Cc2cccc(Br)c2F)C1 52441,C(=O)(CCCCCOC)N(C(C)C(=O)NCC(C1CCCCC1)C)CC 52442,CC1CC(NC(=O)C(C)(F)F)CCN1C(C1(c2ncccn2)CCC1)=O 52443,c1(CC(N2CCC(O)(CNC(C)=O)C2)=O)ccc2nc(Cl)sc2c1 52444,c1(CN2CC(CNC(C(CC)c3ccccc3)=O)OCC2)nc2ccccc2[nH]1 52445,N1(C(C#CC(C)C)=O)CCCC(C2CC2NC(=O)CC2CCCCCC2)C1 52446,c1(C(N2C(CN(C(=O)C=CC3CC3)C)CCC2)=O)c(O)nc(=O)n2c1CCC2 52447,n1(CCC(=O)NCC=CCNC(c2c(OCC)cccn2)=O)nc(C)c(C)c1C 52448,c1(C(c2n(CC(=C)C)nnn2)NCC2CCO2)c(Cl)ncn1C 52449,O=S(=O)(c1[nH]cc2c1CCS2(=O)=O)Nc1ccncc1C(F)(F)F 52450,Cc1ccnc(N(C)CC2CCCN2C(=O)C(C)Oc2ccccc2)c1[N+](=O)[O-] 52451,C12(N(C)C(C3CCCC3CNC3COCCO3)=O)CCC(CC1)CC2 52452,c1(OCC)ncc(NC(=O)CCCN(C(=O)C(c2ccccc2)F)C)cn1 52453,C1(F)(C(=O)NCC2C3CN(C(c4scc(C)c4)=O)CC32)CC2(CCC2)C1 52454,C(=O)(C(CCOC)NC(=O)Cc1nc(C)no1)NCCC=CC=C 52455,N1(C(C(C)(C)OCC)=O)CC2CC(NC(=O)CNS(=O)(=O)CCOCC)C1C2 52456,CC1CC(C(=O)NC23CC(c4ccccc4)(C2)C3)N(c2ccncn2)C1 52457,N1(C(C2(C)CC2Br)=O)CCC2(CCCCN(C(c3ccc4cnnn4c3)=O)C2)C1 52458,c1(C(N(CCCOCCNC(C(C)OCCC=C)=O)C)=O)cc(Cl)c(Cl)[nH]1 52459,C(=O)(C(O)CC(F)(F)F)N1C2C(CNC(CCN(C)CC)=O)C(C2)C1 52460,C(=O)(CCCCCCS(N)(=O)=O)N1C(C)CN(C(=O)CCC2OCCO2)CCC1 52461,c1(N2CC3(C(NC(C4CC5C=CC4C5)=O)CCC3)C2)c(Cl)cc([N+](=O)[O-])cc1Cl 52462,Cc1cc(C(=O)NCCCOCCNC(=O)C(O)CC(F)F)nc(O)c1 52463,C#CC1(C(=O)NCc2cc(C)c(C(=O)NC(C)C(C)CO)o2)CCCC1 52464,C1(CNc2ncc(C(=O)OC)nc2)(SC)COCCN1C 52465,C=CCCC(C(=O)N1CCC(CC=C)C1)NC(c1ccc(C)cc1)=O 52466,CN1CC=C(c2ccc(NC(=O)N(CC(=O)OCc3ccccc3)C)cn2)CC1 52467,C1(CNC)CC(OC)CN1C(C1CCC1C(C)(C)C)=O.C12(CC=CC1)C(=O)NC2 52468,c1(-c2onc(C)n2)cccc2cc(CNCCCCS(=O)CCO)oc12 52469,c1(CC(=O)NCC2C=CC(NC(C3CNC(=O)N3)=O)C2)cccc(C(F)(F)F)n1 52470,C1(C(=O)NCC(C)NC(=O)C(C2CC(F)(F)C2)O)CCCN(C)C1 52471,CN1CCC(C2CCN(C(=O)C(C)(C)CCC#N)C2)C1 52472,N1(C(CCC=CC)=O)CCC(C2CCN(C(c3c[nH]nc3CC)=O)C2)C1 52473,C(=O)(C(F)(F)CN1CCCC1)NCCCN(C)C(C1(F)CCCCC1)=O 52474,c1(C(=O)NC2CCC(C)N(C(C3CC(N(C)C)C3)=O)C2)ccc2cnoc2c1 52475,N1(C(C=CSC)=O)CCC2CCC(C1)N2C(c1cccc(N2CCCC2)c1)=O 52476,Cc1c(C(=O)NC(C2CCN(C(c3ccc(=O)oc3)=O)C2)C)c[nH]c1C1CC1 52477,C1(C(CNC(Cc2nc(NC=O)sc2)=O)C)CCN(C(=O)C(Cl)=CCl)CC1 52478,C1(OC)(OC)CC(C(=O)N(C2CCN(C(=O)CCC3CCCOC3)C2)CCO)C1 52479,c1(C(=O)NCC(CO)NC(=O)CCC2NC(=O)NC2=O)ccc2c(c1)OCCN2 52480,C(=O)(C(CCF)NC(=O)CC(=O)NC1CC1)NC(C)CCCO 52481,C(=O)(C(O)CCC(C)C)N1CCCC(CN(C(=O)Cc2ncccc2C)CC)C1 52482,N1(C(CC2CC(CC)C2)=O)CC2(C(=O)N(C)CC3CCSC3)CC1CCO2 52483,C(=O)(C1=CCCCCC1)NCC(CC=C)NC(C1CC(Cl)(Cl)C1)=O 52484,C1(O)(CNC(c2cc(C)c(F)cc2)=O)CCCN(C(C2C=CCS2)=O)CC1 52485,C1(NC(C(C2CCC2)OC)=O)CC2(CNC(=O)C(C)=C(C)C)CC1CO2 52486,n1(CC)cnc(C(=O)NC(C)C(C2CCCCC2)NC(C2CC(C)(F)C2)=O)n1 52487,N1(C(c2c(C)ocn2)=O)CCN(C(C2(C3CCC3)CC2(F)F)=O)C2COCC12 52488,c1(C(=O)NC(CC2CC2)C(=O)NCC2(CCO)CC2)c[nH]c(=O)cn1 52489,N1(C(C2CCN(C(C)=O)CC2)=O)CCC2(CCCN2C(=O)Cn2cc(C)cn2)C1 52490,Cc1cccc2[nH]cc(CCC(N3CCC(CN(C(=O)CSC(C)C)C)C3)=O)c12 52491,c1(C(N2C(CNC(C3CCN(C)CC3)=O)CC2)=O)cnc2c(n1)CCCC2 52492,N1(C(C=CCCC)=O)CC(NC(=O)C(C)(C)C#N)C(c2ccnn2C)C1 52493,CCCCC(=O)C(=O)NC1CNC1=O.c1(CC(C)SCC)ccncc1 52494,C1(c2ccc(CC)s2)CCCN(CC(N2CCC(C)(NC(=O)C(C)CCC)C2)=O)C1 52495,N1(C(c2cc(N)c(F)c(F)c2Cl)=O)C2CCCC1CN(C(c1ccsc1)=O)C2 52496,C1(NC(C(C(C)O)(C)C)=O)CCCCN(C(=O)CC(=O)OC(C)(C)C)CC1 52497,CCC1(CNCCCCCCl)OCCc2ccccc21 52498,N1(C(C)=O)CC(C)(C)CC1C(=O)NCC1CC(F)(F)CN1C(=O)COC(F)F 52499,c1(NC(C(n2cc(CCCC(C)=O)nn2)C)=O)n[nH]c2c1CC(C)CC2 52500,CCC(O)C(C)C(=O)N1CCCC(CCNC(c2cc(C3CC3)n(C)n2)=O)C1 52501,c1(C(N2CCCCC(CNC(CC3CN(C)C3)=O)C2)=O)cnn2c(=N)[nH]cnc12 52502,N1(C(C(CC)C(C)C)=O)CC2(C1)SCCC2NC(c1cccn2cncc12)=O 52503,C1(C(=O)NCC(c2ccccc2)C)CC(O)CN1C(=O)CC1CC(=O)NC1=O 52504,C#Cc1cc(C(=O)NCCC(O)C(=O)NC(C)CC(=O)NC(C)C)ccc1C 52505,C1(C2CCCCO2)(C(=O)NCC(C)CN(C)C(c2ccc(CO)o2)=O)CCCO1 52506,n1(CC(=O)NCC2(CNC(CCSC)=O)CCC2)cc2ccccc2n1 52507,N1(C(COCCSC)=O)CCC(NC(C2Cc3nccn3C2)=O)C(C(N)=O)C1 52508,C1(C(N2CCCC(N(C(CCN3CCN(C)CC3)=O)C)C2)=O)CC(C2CC2)=NO1 52509,CC1CN(C(c2nccc3nn[nH]c23)=O)C(C)CN1C(c1n[nH]c(O)n1)=O 52510,C1(NC(C2C(=C)CC2)=O)CN(c2ncnc3scc(C)c23)CCC12CCC2 52511,c1(CC)ccc(C(=O)NC)nc1.c12ccc(o1)CNC(=O)C1(F)CC(C1)C(=O)N2 52512,c1(C(=O)NCC2CCN(C(CCOCCOC)=O)C2)nc(C)c(C)nc1C 52513,N1(C(CCc2n(C)cnc2)=O)CCC2OCCN(C(C3CCCS3(=O)=O)=O)C2C1 52514,c1(C(N2CC(O)CC(NC(Cn3ncc(C)c3)=O)C2)=O)n[nH]c2c(C)cccc12 52515,c1(CC(=O)NCC(C2CC2)NC(CC=CC)=O)nc(C)cs1 52516,CCC(C)C(C(=O)NC1C2CC3C1C3C2C(=O)N(CCCO)C1CCC1)N(C)C 52517,C1(CN(C(COCC=C)=O)C)C2CN(C(=O)CCCc3nc(C)no3)CC12 52518,c1(OCC)ccc(F)cc1NC(c1cc(=O)n(-c2ccc(C)cc2)[nH]1)=O 52519,N1(CC)CCC(C(=O)NC23CC(C(=O)NCC(O)C(F)F)(C2)C3)C1 52520,CCC(C)C(C)C(=O)NC1COCCN(C(=O)CC(O)C(C)C)C1 52521,C(=O)(C(CC1CC1)NC(c1ccoc1C(C)C)=O)N1CC(C(N(C)C)=O)C1 52522,N1(C(c2cc(C)sc2C)=O)CC(CNC(=O)C(O)C2CC2)CC(C)(C)C1 52523,N1(C(C2C(C)CC=CC2)=O)CCOCCC1C(=O)N(C1CCC(F)(F)C1)C 52524,N1(C(C(C)N(C(c2cnnn2C)=O)CC)=O)CCN2C(=O)NCC2C1 52525,N1(CCOCC)C(=O)CCN(CC2CCN(c3ccc(C)cc3)C2)C1=O 52526,CC(=O)C(C)CC(C)C(=O)N1CC2(CC(C(=O)NCC3(C)CC3)CO2)C1 52527,N1(C(=O)NCC(N2CCCCC2C)C)CCC2(CCCCC2)CC1 52528,N1(C(c2c(C)cno2)=O)CC2CC(NC(=O)Cn3ccc(C(F)F)n3)C2C1 52529,CC1(CC(=O)NC(CO)C(F)(F)F)CCN(C(c2nccs2)=O)C1 52530,CCC(C)CC(C(=O)N(CC(O)C(F)(F)F)C)NC(=O)CN(C)CC 52531,C1(C(=O)NCCC2(OC)CN(C(c3ccnnc3O)=O)C2)CCC(C)NC1=O 52532,C1(=CCNC(C(C)(O)C2CCOCC2)=O)CCN(C(=O)CSC(F)F)CC1 52533,C1(NC(C2CCC2c2nc[nH]n2)=O)CC2CC(C1)N(C(=O)Cc1cc(Cl)no1)C2 52534,CCC(F)(F)CC(=O)NC(CC1CC1)CC(=O)Nc1cnn(C(C)(C)C)c1 52535,C1(NC(C2N(C(Cc3cc(C)on3)=O)CC3CC32)=O)CN(C)C2(CCC2)C1 52536,c1(CC(=O)NCC(=C)CCNC(c2cc[nH]n2)=O)nc(C2CC2)nn1C 52537,c1(CN(C(N(C2CCCSC2)C)=O)C2CC2)cccc(Br)c1Br 52538,c1(C(=O)NCC(C(C)C)NC(=O)COC2(C)CCCC2)cc2cc(Cl)ccn2n1 52539,C(=O)(C1=COc2ccccc2O1)N(CC(C)NC(C1(CCOC)CCC1)=O)C 52540,C(=O)(CCS(=O)(=O)CC(C)C)N1CC(C(=O)NC(C=C)CO)C1 52541,C1(CN(C(C)C)C)CCCN(C(=O)CCOCCNC(=O)Cn2cnnn2)C1 52542,C1(NC(CCN(CCC)C)=O)CCCCCC1NC(=O)CC1CCC(F)(F)CO1 52543,c1(C(=O)NCC2(O)CCCN(C(C(C)=C(CC)C)=O)C2)cc2c(=O)[nH]ccn2n1 52544,C(=O)(C(F)C(C)(C)O)NCC1(C(=O)NCC=CC2CC2)CC(=C)C1 52545,c1(CNC(C(C)c2ccsn2)=O)ncoc1CCNC(C1CC1Br)=O 52546,Cc1cc(F)ccc1C(=O)NC(C)CCc1ccc(F)cc1 52547,N1(C(c2c(C)n(CC(C)C)nc2)=O)CCC(CNC(=O)C(O)C2CCC2)C1(C)C 52548,C(=O)(C=CSc1ccccc1)N(CCN(C(C)C)C(c1nscc1N)=O)C 52549,Nc1ccc(C(N2CCCCC(C(=O)NCC(O)CNC(N)=O)C2)=O)nc1F 52550,N1(C(C2C(CC)CCN2C(c2cc(C)oc2C)=O)=O)CCSC2(CCC2)C1 52551,N1(C(c2n(CC)ccn2)=O)CC2CCN(C(=O)CC3CCCC(C)(C)C3)CC12 52552,N1(C(c2c(OC)nccn2)=O)CC(C2CCCCN(C(=O)COC3CCC3)C2)C1 52553,C1(CC(=O)NC(CSC)C(=O)N2CC(OCC(F)F)C2)C(=O)NN=C1C 52554,N1(C(CS(=O)(=O)NC)=O)CCCC(C)(C)C1C(=O)NC1CN(C)C(C)(C)C1 52555,C1(NC(c2cn(CC(C)C)nc2)=O)COCCN(C(c2ccc(=O)n(C)n2)=O)C1 52556,c1(C(=O)NC2CCC(CNC(c3nocc3Cl)=O)C2)ccc(F)c2occc12 52557,c1(CC(=O)NCCCNC(C2C3CCC(=O)C23)=O)ccc(F)cc1Br 52558,N1(C(CNC(=O)OCC=C)=O)CCCC1C(C)NC(C1(C(F)F)CC1)=O 52559,C1(NC(C(C2CCN(OCCO)CC2)C)=O)C2CCC(C2)C1Cc1ccncc1 52560,C(CNC(=O)C(C)CC1CC1)(C(C)(C)C)NC(c1c(OCC)scc1)=O 52561,C(=O)(C(C)Cn1ccnc1)N.C1(C(=O)OC)CC(CC(=O)N(C2CCCC2)CCO)C1 52562,C(c1ccc(OC)cn1)=CC(=O)NCC1CCN(C(c2cnn(CC)c2Cl)=O)C1 52563,c1(C(N(c2ccccc2)CC=C)=O)cc(CNC(c2cccc(O)n2)=O)ccn1 52564,Cn1nc(Cl)c(C(=O)NCC2CCCC2NC(c2cncc(F)c2)=O)c1Cl 52565,C1(S(N)(=O)=O)(C(=O)NC2C(CNC(c3cc(C)oc3)=O)C2)CCC1 52566,C1(C(N(CCCCN(C(C(CCN(C)C)N(C)C)=O)C)C)=O)CCCC(=O)CC1 52567,C1(CNC(CCC)=O)(CNC(=O)C(c2ccc(Cl)cc2)(C)C)CC12CCC2 52568,C(=O)(C(C)(C)C1CCC1)NC(C(=O)N(C1(CC)CC1)C)C 52569,C1(C)(CC(=O)N(C)CC2CCCN2C(C2(C)COC2)=O)CCCCC1 52570,CC(C(=O)N1CCC(C)(C(=O)NCCOC2CCCC2)CC1)S(C)(=O)=O 52571,S(=O)(=O)(c1cc(Cl)ccc1F)N1C(C(=O)Nc2ncc(OC)cc2F)COCC1 52572,CS(=O)(=O)c1ccc(C(=O)NCC(C2CC2)NC(C2(CO)CC2)=O)o1 52573,C#CCC(CC(=O)NCCCCC(N)=O)NC(C1(Cl)CC1)=O 52574,C1(NC(c2c(C)cccc2)=O)CN(C(=O)CC2CNC(=O)C2)CC(C)(C)C1 52575,C1(NC(C=CC=CC)=O)CC2CCC1CC2NC(c1ccncc1O)=O 52576,N1(C(CSC)=O)CCN(C(C2CC3CC2C3)=O)C(CS(C)(=O)=O)C1 52577,CCS(=O)(=O)c1ccc(CC(=O)NCC2CN(C(=O)C(C)N(C)C)C2)cc1 52578,C=CCCC(F)(F)C(=O)N1CCC(N(C(=O)CCN(C)CCO)C)C1 52579,C(=O)(C(O)CCNC(C1CCCC(=O)N1)=O)NCC1CN(C(N)=O)C1 52580,c1(C(=O)NCC2C(C)(C)CCN(C(CCCOC)=O)C2)cnn2c(Cl)cccc12 52581,N1(C(C2CCC(C)CC2)=O)CC2(CO)CC1(C(=O)NC1CCN(C(C)(C)C)C1)C2 52582,N1(C(c2c(C)nsc2C)=O)CC(CC(N2CC(N(C)C)C(C)C2)=O)C2(CC2)C1 52583,Cc1ccc2c(C(=O)NCCC3CCCN3C(c3c[nH]c(=N)s3)=O)c[nH]c2c1 52584,C(CC(C)(C)C(=O)CNC(=O)CCc1cnco1)N(C(=O)CC)C 52585,C(=O)(C(C(C)C)C(C)C)N(C)CC1N(C(C2CC(OC)C(OC)C2)=O)CCC1 52586,CCCC(CCO)NCC1CCCN(c2cccnn2)C1 52587,N1(C(c2c(CC)scc2)=O)CCOC(CCNC(=O)CCCn2cccc2)C1 52588,C12(NC(CCC=C(C)C)=O)CCC(C(N3CCN4CCC3CC4)=O)(CC1)CC2 52589,C(C)(C)(CCC(=O)NC1(C(=O)NC2CCCC2CN(C)C)CC1(C)C)OC 52590,Cc1cc(NCc2ccc(S(N)(=O)=O)cc2)ncc1S(=O)(=O)NCCS(C)=O 52591,c1(C(=O)NC(C2CCOC2)CNC(=O)CCC(F)(F)F)cc2c(Cl)nccc2o1 52592,CS(=O)(=O)C=CC(=O)NCC1(O)CCN(C(C2CC3(CCC3)C2)=O)C1 52593,c1(C(=O)NC2C(C)N(C(c3cn4c(n3)SCC4)=O)CC2)cc(F)c(Cl)cc1Cl 52594,CC(C(C)C(=O)NC(C)C(C)C(=O)OC)NC(c1nc(=N)cc[nH]1)=O 52595,c1(C2N(C(=O)Nc3cncc(OC(C)C(C)C)c3)CCC2)ccc(F)c(F)c1 52596,C1(CNC(C=CC)=O)CC(CNC(C2C=C(C)CS2)=O)C1 52597,Cc1ncc(C=CC(=O)NC2CCC(CCNC(=O)CCS(N)(=O)=O)C2)c(O)n1 52598,C(CCCC(CO)NC(C1ON=C(C)C1C)=O)NC(c1c(C)nc(CCC)o1)=O 52599,Cn1ncc2c(NCC3CCC4(CCC4)O3)[nH]c(=NCC3=CCCCC3)nc12 52600,c1(C(=O)NC2C(NC(Cc3c(C)scc3)=O)CCOC2)ccc(N)c(Cl)n1 52601,c1(OC)cccc(NCCCC2CCCO2)c1C(c1ccccc1)OC 52602,Cc1ncc([N+](=O)[O-])cc1C(=O)N(C)CC1CCCN1C(C1CC2CC2C1)=O 52603,C1(C(=O)O)CC(F)(CNC(C2C=CCCN2)=O)C1 52604,CC1C(C(=O)NC(CCO)C2CCC2)CCN1C(c1cccs1)=O 52605,N1(C(CN2CC(C)(C)C2)=O)CCCC(NC(c2cncc(N(C)C)n2)=O)CC1 52606,C1(NC(c2cc(C)[nH]n2)=O)COC2(CCN(C(C3(CO)CCOCC3)=O)C2)C1 52607,CCCS(=O)(=O)CC(=O)NCC1CC2(CO1)CN(C(c1c(C)ncn1OC)=O)C2 52608,c1(-c2n(-c3cccc(C)c3)nc(C3CCOC3)n2)cn(C)cc(Br)c1=O 52609,c1(C(=O)OC)ccc(CN(C)Cc2cc(-c3ccccc3)n[nH]2)cc1 52610,C(=O)(C1=CCCN(C(C2CCCC(O)C2)=O)C1)NC1(C)CCCC1O 52611,N1(C(C2CN(S(CC)(=O)=O)C2)=O)CC(O)(C2(CNC(=O)CC(C)(C)O)CC2)C1 52612,c1(NC(C)C)ccc(C(=O)NCC2(O)CN(C(C3CC3(C)Br)=O)C2)cn1 52613,c1(N(C(CNC(CC(=O)NC)c2ccccc2)=O)C)ccc(OC)c(C#N)c1 52614,c1(NC(CNC(c2ccn(C(CC)CC)n2)=O)C2CC2)cc(O)nc(O)n1 52615,C1(NC(c2cc(CC)sn2)=O)CC12CCN(C(=O)C(C)C1CCCC1)C2 52616,N1(C(C2(C3N(C(c4ccc(OC)o4)=O)CCC3)CC2)=O)CC(=O)NCC1C 52617,N1(C(c2cc(C)oc2)=O)CC(NC(=O)C(C)Cc2cnc[nH]2)C(N=[N+]=[N-])C1 52618,C(C(F)(C(=O)NC(CC)C(N)=O)C(C)C)NC(c1ccn(CCC)n1)=O 52619,c1(NCC(CNC(C2CC=CC2)=O)O)cc2nncn2cn1 52620,n12cc(nn1)CCCNC(=O)CC2.C(=O)(C(C)(C)O)N(S(C)(=O)=O)C 52621,c1(-c2n(-c3c(CC)cccc3)nc(C(O)CC)n2)ccc(F)c(Cl)c1F 52622,c1(C(=O)NCC2C(C)(C)CN(C(C3(CCF)CC3)=O)C2)cn2cc(Cl)cnc2n1 52623,N1(C(C=NOC)=O)Cc2nccn2CC(NC(c2cccc(C(F)(F)F)n2)=O)C1 52624,c1(C(N2C(CCCNC(=O)C=CCO)CCC2)=O)ccc2ncncc2c1 52625,C1(C)(CC(=O)NC(c2ccccn2)CC)CCN(C(=O)CCN2CCOC2=O)C1 52626,Cc1cc(CN2CC(NS(=O)(=O)c3cnoc3C)C(CO)C2)c(O)c(C)c1 52627,N1(Cc2ncc(C(=O)NCC(C)NC(C3CC3C)=O)s2)CCNC(=O)C1 52628,c1(OC)cc(Br)c(CNC(=O)C(C2CCS(=O)(=O)CC2)F)cc1C 52629,c1(N(C(=O)NC)CC)ccc2cc(-c3ccc(F)cc3OC)n(C)c2c1 52630,N1(C(c2c(C)nc(CO)nc2)=O)CCN(C(c2ccccc2O)=O)CC12CCC2 52631,C1(CCC(=O)NCC2(Cl)CCC2)CCCCN(C(c2ccc[n+]([O-])c2)=O)C1 52632,C(=O)(CCCCC(F)F)N(CC(C)CNC(C1(C(F)F)CCOCC1)=O)C 52633,N1(C(CC2C(C)(C)C2)=O)CCCC(C)(C(N2CCOCC2C(N)=O)=O)C1 52634,CC1CC(NC(c2ccnn2C)=O)CN1C(=O)Cc1csc(-c2cccs2)n1 52635,N1(C2CCC(NC(C(F)=CCC)=O)C2)CCN(C(c2cc(Cl)cnn2)=O)CC1 52636,C(F)(F)(C(F)(F)F)OCC(=O)Oc1ccc(N2CCC(N(C)C)C2)cc1 52637,c1(C(=O)NC(CNC(c2nc(OCC)sn2)=O)(C)C(C)C)ccc(N)c(F)c1F 52638,n1(CC)nc(C(=O)NC(C2CN(C(=O)Cc3ccncc3Cl)CCO2)C)cc1C 52639,Cc1[nH]nc(CO)c1C(=O)NC1CC(C)N(C(=O)CCN(C2CCCCC2)C)C1 52640,C1(C(=O)NCC23CC(CNC(C4CC4(Cl)Cl)=O)(OC2)C3)Cc2cscc2C1 52641,C1(NC(Cc2cn(C)nc2)=O)CN(C(c2cc(Br)no2)=O)CC1N=[N+]=[N-] 52642,c1(C(N2C(C(N3CC(O)(CCC)C3)=O)C(C)CC2)=O)ccc([N+](=O)[O-])[nH]1 52643,CC(CN(C)C)CC(=O)NCCCCCNC(=O)CCc1nncnc1O 52644,C1(C(=O)NCC(C)OCC#C)CCOCCN1C(c1nc(C)ccc1F)=O 52645,N=c1cc(CC(N2CCN(C(=O)CCc3nccs3)C3CC23)=O)cccn1 52646,C1(C)(C(=O)NCC(CC)NC(C2CC2C2CCC2)=O)SCCCS1 52647,C#CC1C(C(N2CCCC2CNC(=O)CN2CCCS2(=O)=O)=O)C1(C)C 52648,C(=O)(CC(O)CC(C)C)N(CCOC)CCNC(=O)Cn1nc(C)nc1C 52649,Cc1c(C(=O)NC23CC(C2)N(C(c2cc(Br)c[nH]2)=O)C3)nn(C)c1N 52650,Cc1c(Br)csc1C(N1CCCC1Cn1cc(C2OCCO2)nn1)=O 52651,n1(CC(=O)NCC2C(NC(C=C(C)C3CC3)=O)COC2)ncn2nccc2c1=O 52652,c1(CCC(=O)NC2C(CNC(CN3C(C)CCC3)=O)C2)ccccc1C(F)(F)F 52653,N(C(=NCCC1CCC2(CCC2)O1)NCc1ccccn1)C1CCCC1 52654,C1(NC(=O)Cc2cncnc2)CC12CCC(NC(c1cc(Cl)cs1)=O)CC2 52655,c1(OC)ccn2ncc(-c3cnc(NC(=O)C(F)(F)C(O)c4cccs4)s3)c2c1 52656,CC1(NC=O)CCOC1.C(C)(CN)(CO)NC(=O)CCF 52657,N1(C(CCSC)=O)CC2CC2(C(=O)Nc2sccc2I)C1 52658,c1(C(N(CCCCCNC(=O)C(C)c2cncs2)C(C)C)=O)ccc(Cl)cc1 52659,c1(SC)cc(C(=O)NCC2CCCN2C(c2cn(CCO)nc2C)=O)ccn1 52660,C12(C(=O)NC3CC(NC(Cn4ncc(C(=O)OC)c4)=O)C3)C=CC(CC1)C2 52661,c1(OC(C)C(N2CCC(O)(CNC(=O)C(F)F)C2)=O)c(Cl)cc(Cl)cc1Cl 52662,CCCC(C(=O)N1CC(NC(c2cc[nH]n2)=O)CC(O)C1)S(N)(=O)=O 52663,C1(NC(=O)C(O)C(F)(F)F)CN(C(C2CC3(C2)CC2(CC2)C3)=O)CC12CCC2 52664,C(=O)(CC(C)(C(F)F)N(C)C)NCCN(C(C1(C)CCC(=O)N1)=O)CC 52665,CC12CCC(C(=O)NC3COCC3CNC(=O)Cc3ccc(Cl)cc3)(CC1)CO2 52666,CC1CC(C)C(C(=O)NC2CCN(CC3CC3)CC2)CN1C(=O)C1=CCCCC1 52667,c1(CNCCCc2ccc(F)cc2)ccc(F)c(F)c1Br 52668,c1(NC(COc2c(CC)n[nH]c2)=O)cn(CC(C)C)nc1C(F)(F)F 52669,C(CC(=O)N(C)CC1CCCCC1O)(C(C)(C)C)NC(c1cc(C)c(=N)[nH]c1)=O 52670,c1(C(=O)NCC(C)N(C(C(CC)CCOC)=O)C)cc2c(OC)ccc(C)c2[nH]1 52671,C(=O)(CCN(CCCO)C(C1CC1CCCC)=O)N(C(C#C)C)C 52672,CN1CCC2C(CCCN2C(Cc2ccccc2)C(O)c2ccccc2)C1 52673,C12CCCN(C1)N1CC(C(OC)C(=O)N2)C1.C(=O)CCC1(C)CC1 52674,O=[N+]([O-])c1ccsc1COC(c1cc(Br)ccc1F)=O 52675,c1(C(=O)NC(CC)(CNC(C2CC(=C3CC3)C2)=O)CC)ccc(C)c(OC)c1 52676,c1(OC)cnc(C(=O)NCC2(OC)CCC23CCC3)c(C)c1 52677,c1(SC)cn(C)nc1C(=O)NC1CC1CNC(c1ccc(CN(C)C)cc1)=O 52678,c1(C=O)nnc(O)cc1O.C1(C)CCCN(N(C)NC(CCOCCC)=O)C1 52679,c1(COC)ccccc1COCC(=O)NC(C)CNC(C1CCC1)=O 52680,C1(C(=O)NC(CNC(c2c(OC)noc2C)=O)C)CCCCCC1(F)F 52681,N1(C(C=Cc2ncn(C)c2)=O)CC(C2CC2C(=O)NCCC2CCCC3CC23)C1 52682,c1(CC(=O)N(C)CC2N(C(C(CCC)N(C)C)=O)CCC2)ccc2ocnc2c1 52683,c1(C(=O)NCC2(NC(CCNC(C)=O)=O)CCCCC2)cc2c([nH]1)CCOC2 52684,C(=O)(C1=CC(C)(CC)C1)NCC1CN(C(CN(C(=O)OCC)C)=O)CC1O 52685,n1(CC)c(N(CC)CC2CCCCC2)nnc1-c1noc(C)n1 52686,C1(NC(C=COCC)=O)(CNC(C2CCCS2)=O)CCC(C)(C)CC1 52687,CC1(C)CCN(C(C2CCO2)=O)CC1NC(=O)CCCOCc1ccccc1 52688,O=C1CC(C(=O)NC(c2cccc(F)c2)c2ccccc2)=NN1 52689,N1(C(c2ccc(C#C)nc2)=O)CCN(C(C2CC2(F)F)=O)CC(O)C1 52690,C1(NC(Cc2nc(C)[nH]n2)=O)CC(=O)N(C2CN(CCC(=O)NC3CC3)C2)C1 52691,CN1CC2(C1)N=C1C=CN=C(N1)NC(CN1CCCCC1)C(=O)C2 52692,CC(C)C(C(=O)N1CC(NC(=O)CC2CC2)C(n2cccn2)C1)n1cncn1 52693,Cc1ccc(C(O)C(=O)NCC2CCC2NC(c2cnc(S)n2C2CC2)=O)cc1 52694,C1(C(N(C(CC(=O)OC)C)C)=O)(NC(=O)CCn2ccnc2C)CC(F)(F)C1 52695,C12(C(N3C(CO)CC(NC(Cc4n(C)nnc4)=O)C3)=O)CCCC1C2(F)F 52696,CCCCCCCCC(CCCCCC)C(=O)NCC1CCN(C(=O)CC)C1 52697,c1(C(N2C3CCC(NC(c4cc(F)n[nH]4)=O)(C3)C2)=O)ccc2cccnc2c1O 52698,N1(C(C(C)NC(c2cnc[nH]2)=O)=O)CCC2CN(C(c3cccc(F)c3)=O)CC12 52699,c1(OCC(=O)NCC(=O)NCc2cnc(C(C)C)nc2)ccc(S(N)(=O)=O)cc1 52700,Cc1ccc(C2CC2NC(=O)Cc2nc(C(C)(C)C)ns2)cc1C 52701,N1(C(c2cc(CC)ncn2)=O)CC(CNC(=O)C(F)n2cccn2)C2(CC2)C1 52702,c1(C(=O)NCCN(C(CS(CC)=O)=O)CC2CC2)cc(C#N)cc(C)n1 52703,C(c1ccc(Br)s1)=CC(=O)N(C(CC)Cn1cncn1)c1ccco1 52704,C1(C(=O)N(CCCCN(C)C)C)(COC)CCN(C(=O)Cc2cccnc2)CC1 52705,CN1CCn2nc(C(=O)NCC3CCN3C(c3cccc([N+](=O)[O-])c3)=O)cc2C1 52706,Cn1cc(C(N2CCCC2CCCNC(C2CC(C)(O)C2)=O)=O)nn1 52707,CCC(C)(C(=O)NC1CCC(NC(c2ccnc(C)n2)=O)CC1)C(N)=O 52708,c1(C(N(C(CCNC(c2c(CC)nns2)=O)C)C)=O)ccc(C)n1C 52709,N1(C(C2C(C)=C2)=O)CCN(C(c2ccc(C)c(O)c2)=O)CC1C 52710,N(C1CCCn2ccnc21)C(CC1CCN(C(C2CC(=C)C2)=O)C1(C)C)=O 52711,C1(C2CCN(C)CC2)(C(=O)NC(CC)(C)CNC(=O)Cc2c(C)n[nH]c2C)CC1 52712,CC1(C)CC(CC(N2CCCC2CNC(C2(c3ccsc3)CC2)=O)=O)C1 52713,Cc1c(COC(=O)CNC(C2(F)CCCCC2(C)C)=O)oc2ccc(Cl)cc12 52714,C(C)(C(=O)NC(C)(C)CN(C(=O)CC1CC1CC)C)OCCC=C 52715,c1(C(N2CCC(C(NOCC=C)=O)C(C)C2)=O)cnn2cccc2c1 52716,Cc1c(C(=O)NCC(F)CNC(=O)C(C)(Cl)Cl)oc2c(F)cccc12 52717,C(=O)(C1=CCCCC1C)NCC(C(=O)NCC1CC(SC)C1)C 52718,N1(C(CCN(CCC)C)=O)CC2CCCC2(C(=O)NCC(C)C(C)(C)C)C1 52719,C1(NC(C(C)Cn2cccn2)=O)C2CC3C(C2)C13C(=O)NCCCSC(F)F 52720,c1(OC)ccc(C(=O)NCC2(NC(=O)C=C(C)Cl)CC2)c(O)c1F 52721,C1(NC(C(C2CC2)OCC)=O)(CC)CCCN(C(=O)C(C)(C)CCOC)C1 52722,N1(C(CSCC(C)C)=O)CCOC2(CCN(C(=O)CC3CN4CCN3CC4)C2)C1 52723,c1(C(=O)NC(CC=C)CNC(C2CC(=O)OC2(C)C)=O)c(C)c(C)nn(C)c1=O 52724,S(=O)(=O)(c1ccc(NCCC2(C)OCCO2)cc1Cl)NCCCC 52725,c1(OC(C)C(=O)NC2CCCN(C(=O)CCCF)C2)ccccc1Br 52726,C1(NC(C(C)C2CC2)=O)CC2(CCN(C(c3cccc(F)c3Br)=O)CC2)C1 52727,N1(c2nc(C)c(Br)cn2)CC(C)CN(C(C2CN3CCC2CC3)=O)CC1C 52728,N1(CC)CCOCC1CC(=O)N(C(C)CCNC(=O)CCc1cn(C)cn1)C 52729,N1(C(C2CCN(C(C=CCC)=O)C(C)C2)=O)CCCN(C=O)CC1 52730,c1(C(N2CC3C(CN(C(C(CC=C)NC(C)=O)=O)C)C3C2)=O)ccc(O)nc1Cl 52731,N1(C(CCCn2cc(-c3cn(CC)nc3)nn2)=O)CCCC(CC(N)=O)CC1 52732,N1(Cc2c(C)nn(C3CCOCC3)c2Cl)CC=C(c2ccnn2C)C1 52733,c1(N2C3CN(C(C(CC)(C)CC)=O)CC2CC3)ccc([N+](=O)[O-])c(O)n1 52734,c1(NC)snc(C)c1C(=O)NC1CCN(C(C2(F)CCOC2C)=O)C1 52735,N1(C(C=CCC)=O)CC(OC)CC1(C)CNC(c1ccc(C)cc1N)=O 52736,N1(C(=O)NC(C)(C)C)CCC(CN(c2nccc(Cl)c2O)C)C(C)(C)C1 52737,N1(C(C(CC=C)NC(c2ncncc2OC)=O)=O)CCC2CN(C(C)=O)CCC12 52738,c1(CN2CCCC(NC(=O)COC(F)(F)C(F)(F)F)CC2)cc2ccccc2o1 52739,Cc1cc(C)c(C(N2CC(NC(c3ccsc3)=O)C(O)C2)=O)c(Cl)n1 52740,C(=O)(C1=CC2(CCOC2)C1)NCCC1(NC(c2c(C)c(Br)no2)=O)CCC1 52741,CC(C)C(F)(F)CC(=O)N1CC(CNC(c2c[nH]c(C(N)=O)c2)=O)CC1C 52742,c1(SCC(=O)NCC(C)(O)CNC(c2c[nH]ccc2=N)=O)ccsc1[N+](=O)[O-] 52743,N1(CC(=O)N(CCC(=O)NCC2CC2C#N)CC)CCCC1C 52744,CC(C)CCCCC(=O)N1CCC2CN(C(=O)CS(=O)(=O)CC3CCCO3)C2C1 52745,CCCCC(O)CCC(=O)NCC1CCN(C(=O)OC(C)(C)C)CC1(C)O 52746,CCCC(O)CC(=O)NCCN(C(=O)Cc1ccc(CC(C)C)cc1)C 52747,N1(C(CCSCCCC)=O)CCC(NC(C2CC(N3CCCC3)C2)=O)CC1 52748,CC1(NC(c2ncc(Cl)nc2Cl)=O)CCCN(C(=O)Cc2cscn2)C1 52749,N1(C(c2c(C)cn(C)n2)C(=O)NCC(C)C)CCC(O)C(CC(C)C)C1 52750,C1(C(=O)NC2C(C)CN(C(C3(O)CCOC3)=O)C2)CCC2(CCC2)CO1 52751,C(=O)(C(C)(C)CC(F)F)NCC(CC)(C)NC(=O)C(Cc1ccccn1)=NO 52752,N1(C(C(C)SC(F)(F)F)=O)CCOCC(NC(C2(c3ccno3)CCC2)=O)C1 52753,c1(C(=O)NCc2ccc(C(C)NC(=O)C(O)C(C)C)cc2)cnc(O)n(C)c1=O 52754,N1(C(C(C)CC2CCC2)=O)CCC(C2CC2)(CNC(=O)COCCF)C1 52755,Cc1c(C(=O)NCCC2(NC(=O)C=Cc3ccoc3)CC2)cc(F)cc1Br 52756,c1(NCc2c(C3CN(C(c4cc(C)on4)=O)C3)ocn2)ncnc2sccc12 52757,C1(C(=O)NCCN(C(C2CC2F)=O)CC)(CO)CCCC1 52758,Cc1nnc2cc(NCCCCNC(=O)C(c3cccc(Cl)c3F)(C)C)ncn12 52759,C1(NC(CCCN(C(C)=O)C)=O)CCC12CCCN(C(=O)C(C)P(C)(C)=O)C2 52760,C1(NC(CS(C)(=O)=O)=O)CN(C(=O)C(=Cc2cccc(F)c2)F)CCC1O 52761,C1(NC(C2CCC(N=[N+]=[N-])C2)=O)C2CC3CN(C(C4CCCN4C)=O)C1C3C2 52762,CC(CC(=O)N(CCCNC(=O)CCC1CC(F)(F)C1)CCO)C1CCCO1 52763,c1(CC(=O)NCCCC(C)NC(C2COCC2(C)C)=O)c[nH]c2cnccc12 52764,Cc1ccc([N+](=O)[O-])c(C(=O)NC2COCCC2NC(c2ccncc2C)=O)c1 52765,C(=O)(C1=CCCCC1)N1C(CN(C(c2ncc(C=O)nc2)=O)C)CC(F)C1.CO 52766,c1(C(=O)NC(c2cn(Cc3ccc(Cl)nc3)nn2)CCC)cn2ccccc2n1 52767,c1(NCc2ccc(C(C)(C)C)c(Br)c2)ccc(C#N)c(F)c1.N12CCCC1C2=O 52768,C1(C(=O)NCCCNC(=O)CC2CCCO2)(Cc2cccs2)CCCCC1 52769,C(CNC(N1CCCC(C(=O)Nc2ccccc2)C1)=O)(C(F)(F)F)OC 52770,c1(C(N2CC(C(C(=O)NC(C(C)C)C3CC3)OC)C2)=O)cc(O)cc(=O)o1 52771,C1(C(N2C3CCC2CN(C(C2(C4CCCO4)CC2)=O)C3)=O)COC2CCCCC12 52772,N1(C(C(C)(C)C2CCCC2)=O)CCC(CNC(=O)CCc2csnn2)C(O)C1 52773,CC1(C)CCC(CNC(C23CC=CCN2CCC3)=O)N(c2nnccc2C#N)C1 52774,C1(F)(C(=O)NC2CN(C(C(C)N3CCC3)=O)CC2C)CCCCCC1 52775,Cc1ccc(F)cc1C(N1CCN(C)CC1CNC(c1nccn1C(C)C)=O)=O 52776,n1(CC)ccc(C(=O)NC(C)CCNC(=O)CCCNC(c2ccccc2)=O)n1 52777,C12(CNC(CCCN(C)C)=O)CCC(CC1)CN2C(=O)C(c1ccc(F)cc1)O 52778,c1(SCCC(=O)NC23OCCC(C(=O)OC)(C2)C3)nc2ccccc2s1 52779,N1(C(c2c(Cl)ccc(C)c2)C(=O)NC2CCOC2)CCCC1C1CCCO1 52780,C(C(F)CN(C(=O)OC(C)(C)C)CC1CC1)OC(C)(C)C 52781,C1(NC(Cc2ccc(SCC)cc2)=O)CC2CCC(C1)N2C(=O)C(C)(Cl)Cl 52782,Cc1ccc2[nH]c(C(=O)NCC(O)CCNC(=O)CCC(C)(C)C)cc2c1 52783,C1(NC(C(C)SC)=O)CCN(C(=O)CC2CCCCO2)C(C)C1 52784,N1(C(Cc2c(C)n(C)cn2)=O)CCCC(C)(C)C1C(=O)NCCc1nncn1C 52785,C1(N2CC(C)C(NC(=O)C3=CCCC3)C2)CCc2ccccc2NC1=O 52786,c1(C(N2CCCC(C)(NC(C(CCC)N(C)C)=O)C2)=O)cncc2ccsc12 52787,c1(C(N2CCC(CO)C2)=O)ccc(N2CCSCC2)cc1Cl 52788,N1(CC(=O)N(C)CCc2ccc(O)c(O)c2)CC(N(C)CCO)CC(F)(F)C1 52789,c1(NC(c2[nH]cc(COC)c2)=O)cccc(NC(C2(C)CCCO2)=O)c1 52790,N1(C(c2ccc(OCCO)c(F)c2)C(=O)NC)CCOC(C(F)(F)F)C1(C)C 52791,c1(Nc2cc3c(cc2)OC(C)C3)nccc(=NC2CCCn3nccc32)[nH]1 52792,N1(C(C2CCCN3CCCCC23)=O)CC2OCCN(C(=O)C=CCF)C2C1 52793,C1(NC(C2(CNC(C(C)=C3CC3)=O)CCCCC2)=O)CC(O)C12CCC2 52794,C1(C(=O)NC2CC(NC(CC(C)NC(N)=O)=O)C2)CC12CCC1(CC1)CC2 52795,c1(C(=O)NC(C(=O)NCC(CC=C)NC(=O)CC)COC)cccc(N(C)C)c1 52796,C1(C(=O)OC)CC2CN(C(=O)C(N3CCCC(O)C3C(=O)OC)=O)CC12 52797,c1(OCC(=O)NC)ccc(CN2CCC(c3ccccc3F)C2)cc1 52798,C1(C(N2CCC(NC(Cc3cc(C)no3)=O)C2)=O)CCCCC1c1nncn1C 52799,N1(C(c2[nH]cc(C#N)c2)=O)CCCCC(CNC(=O)C=CC(F)(F)F)C1 52800,c1(C(N(CC(CC)NC(c2cc(C)c(Cl)cn2)=O)C)=O)cc2[nH]nc(C)c2cn1 52801,C12C(C3CC3)CCN1C(=O)c1cncc(c1)NC2=O.CN1CCC2(CCC2)C1 52802,N1(C(c2n(CC)cnn2)=O)CCC2(CCCC2NC(c2ccc(C)s2)=O)C1 52803,C(C(CC(C)C)NC(=O)CC(O)C1CC1)NC(c1c(NC(C)=O)cccn1)=O 52804,c1(N(CCOCC)C)nnc(Cc2ccc(F)cc2)n1CC(C(C)C)SC 52805,C1(OC)CN(C(=O)Cc2cccc(F)c2)CC1NC(=O)CC1CCC(C(N)=O)O1 52806,C1(C(=O)NCCNCCN(C)Cc2ccccc2Cl)COc2ccccc2O1 52807,N1(C(c2n(C)cc(Cl)c2)=O)CC2(CCC(NC(C3CCCCS3)=O)CC2)C1 52808,C(=O)(CC(C)CC(F)(F)F)NC1CCC(NC(c2nn(CC)c(C3CC3)c2)=O)C1 52809,c1cc(Br)cnc1I.N12CCN(CC1)C(=O)C1C(C1)C2=O.C1CC1 52810,c1(CNC(C2(Cl)C(C(C)C)C2)=O)ccc(SC(F)F)cc1 52811,C(=O)(CC1CCc2ccccc21)NCC1C2CN(C(c3c(C)nsc3N)=O)CC21 52812,C(=O)(CS(=O)(=O)C1CC1)N1CCC(NC(CC2C=NN(C)C2=O)=O)C1 52813,CCCC(C(=O)NCCCCCNC(=O)C=Cc1cn[nH]c1)S(N)(=O)=O 52814,C(=O)(C(C)(C)CCCC(=O)NCC1(O)CN(C(c2c(C)nn(C)c2F)=O)C1)OC 52815,C1(CNCC(c2ccc(Br)cc2)C)CCC2(C1)CC2(F)F 52816,C1(N(CCCCC)C(c2cccnc2)=O)CC(F)CN(S(=O)(=O)CC2CCC2)C1 52817,C1(CC(=O)NCc2c(C)n[nH]c2C)CN(C(=O)CC2CCCO2)C(C)(C)C1 52818,Cc1nc(C(N2CCN(C(c3c[nH]cc(F)c3=O)=O)CC2C(C)C)=O)cc(O)n1 52819,c1(C(=O)NCC2CCN2C(=O)CC2CC3CCC2CC3)c(F)cc(F)cc1Cl 52820,CC(N=c1ccc(C#N)n[nH]1)C1CCCCN1C(=O)CC(O)CN(C)C 52821,N1(C(C(CC)(C)O)=O)CCCC2(C1)CN(Cc1cccc(Cl)c1)CCO2 52822,N1(c2nnc(C)o2)CCC2(CC1)OC1(C)CC2(NC(=O)CC2NC(=O)NC2=O)C1 52823,C1(CNC(C(CCC)F)=O)CN(C(C2CCCCC23CC3)=O)CC12CCC2 52824,N(C(=NCCCF)NCCC(C)(C)C)C1CC(OCC)C1 52825,C#Cc1cccc(C(N2CCC(C3CCN(C(=O)CN(C)C)CC3)C2)=O)c1C 52826,c1(N2C3CC(CNC(c4c(C)cns4)=O)CC2CC3)cc2nnc(C)n2cn1 52827,C(=O)(C1=CC(C)(C)C1)NC1C=CCN(C(C(c2ccc(N)cn2)C)=O)C1 52828,C(CS(=O)(=O)CC(=O)NCCC1CCCN1C(=O)CC1CC2CCC1CC2)OC 52829,Cc1cc(C(=O)NC(Cn2ccnn2)C(=O)NCC2(C)CCCC2O)nn1C 52830,C(CC(C)(C)CBr)(c1n(CCCCCC)nnn1)NC(C)COCC1CC1 52831,C1(CC)COCC1NC(=O)C(C)(C)NC(=O)C(C)=CC(C)(C)C 52832,c1(C(=O)NCC2N(C(C(CC)OC)=O)CC2)ccc([N+](=O)[O-])cc1C(F)F 52833,N1(C(C(C)Cc2cnc[nH]2)=O)CCC(C)(CNC(=O)CCc2nncs2)C1 52834,C1(NC(c2c(CC)cco2)=O)CC1C1CCN(C(=O)COCCCN(C)C)CC1 52835,c1(OCC)nc(C(=O)NC(C)(C)C(C)NC(=O)C(C)CN2CCCCC2)ns1 52836,C1(F)(C(=O)NC(CC)CSC(F)F)CCCN(C(C2(n3cccn3)CC2)=O)C1 52837,C1(C(=O)NC(C(=O)OC(C)C)C)CC2(C1)CC(N=c1ncnc3[nH][nH]c(I)c1-3)C2 52838,C12(CNC(=O)Cc3ccco3)CC1CN(C(=O)C(F)n1ccnc1)C2 52839,c1(C(N(c2nc(OC)c(F)cn2)C2CCNCC2F)C2CC2)cc(Br)c(F)cc1Cl 52840,c1(C(N2CCC(C(C(=O)NCC(CC)(C)C)F)C2)=O)nn(C)cc1C 52841,C1(NC(N(C2CCCC2C#N)CC(C)C)=O)CC2C=CC1CC2 52842,c1(OC)ccc(Br)c(C)c1C(N1CC(N(C)C(c2cc(C)c(C)s2)=O)C1)=O 52843,C(=O)(C1=CC(C)CC1)N1CCC(N(CCOC)C(c2cc(C)ccn2)=O)CC1 52844,C1(C(N2CCCC(N(C)C(c3scnc3Cl)=O)C2)=O)CCc2cncn2C1 52845,c1(COC)cc(CC(=O)N(CC(C)NC(c2c[nH]nc2C(C)C)=O)C)no1 52846,C(=O)(CC1=CCCCC1)NC(C(=O)NCC1(OC)CCC(C)C1)C(C)C1CC1 52847,c1(NCC(=C)Cl)cc(N2CCCC(OCC)C2)nc(C(F)(F)F)n1 52848,N1(C(c2n(C)nnc2)=O)CC2(CC2)CC1CC(=O)NCCC1(C)CCCC1 52849,CC1CN(C(=O)CN(C)C)CC2(CCN(CC(=O)N(C)C)C2)O1 52850,N1(C(C(C2CCN(C(C(C)=C(CC)C)=O)C2)F)=O)C2CCC1CC1(C2)N=N1 52851,C(=O)(CCCN(C)C)N(C(C)C(=O)N(C)CC1(CO)CCCC1)C 52852,CC(C)C(O)CC(=O)NC12CC(NC(=O)CCC3(C)CC3(F)F)(C1)C2 52853,c1(C(C)(C)OC)nc(=NC(CNC(C2CCCCCC2)=O)CO)s[nH]1 52854,CC1(C(=O)NC2C3CCC(C3)C2C(=O)Nc2cncc(CO)c2)CCC(O)CC1 52855,c1(CC(=O)N(CC(CC)NC(=O)C#CC2CCC2)C)cn2ccccc2n1 52856,c1(-c2nccc(NCc3c(CC)c(C)ccc3)c2)c(F)cc(CO)cc1F 52857,c1(C(C(=O)N(C2CN(C(=O)OC(C)(C)C)C2)C)O)cc(F)c(F)c(Cl)c1 52858,C1(N(C(c2c(COC)ncs2)=O)C)CC2CCC(C1)N2C(c1ccc(F)s1)=O 52859,C1(CNC(CC2(CSC)CC2)=O)CN(c2ncns2)CCC12CCOC2 52860,C(=O)(N=c1cc[nH]cc1I)N(C)CC1(F)CCOCC1 52861,N1(C(CC=CC=C)=O)CCCC2(C1)CN(C(=O)CC1CCCOC1)CCO2 52862,CC(C(=O)NC(CNC(=O)CCCn1c(O)nnc1O)C(C)(C)C)C(C)(F)F 52863,C1(NC(C2CC(CC)(CC)C2)=O)CN(C(=O)CNC2(SC)CCOCC2)CC1F 52864,c1(C(N2CCCC(CNC(c3ncc(C(F)F)s3)=O)C2)=O)ccnc2[nH]nnc12 52865,c1(CC)nn(C)c(Cl)c1C(=O)NCC1CCN(c2nc(C(F)(F)F)ns2)C1 52866,Cc1cc(C(=O)NC2CC3CCC2(NC(C2CC(C)(C)C2)=O)C3)nc(O)c1 52867,C1(C(N2CC(C)=C(C)CC2)=O)N(C(c2cn(C3CC3)cn2)=O)CC12CCCC2 52868,O=C1C2C(O)CCN2C(=O)N(c2cccc(Cl)c2Br)C(=O)C1CC1CCCC1 52869,C1(CNC(CC2CC(C)OC2C)=O)CC2(CO1)CN(C(c1nc(=O)n(C)[nH]1)=O)C2 52870,N1(C2(c3c(Cl)ccc(Cl)c3)CC2)CCc2c(-c3nn[nH]n3)cccc21 52871,CC1=C(C(=O)NC2CCN(C(=O)CCc3cc(C)cc(C)c3)C2C)CCC1 52872,C12(CCCC1)C(=O)NC1CCN(C1)C2=O.C1(CN(C)C)CN(c2nncs2)C1 52873,C(=O)(CC(C)CN(C)C(=O)NCc1cc(C)nn1C)OC 52874,C1(C(=O)NC(C)Cc2ccc(Cl)cc2)CCC(=O)C(C)C1 52875,C(CCCCCNC1OC2CCC1C2)n1cc(-c2nnc(C(=O)OCC)s2)nn1 52876,c1(CN(C(=O)Cc2cnoc2)CCNC(=O)CCSC(F)(F)F)ccc(Cl)nc1 52877,N#CC1CCCC1N.N(S(=O)(=O)NCC)CCCO[Si](C)(C)C 52878,CC1CN(C(C23CC2COC3(C)C)=O)CCN1C(c1[nH]cnc1C#N)=O 52879,CCCCC(C)C(=O)N1CC2(CC2)CC1CNC(=O)CCCN1C(=O)CNC1=O 52880,C1(CC)CCCCC1C(=O)NCc1ccc(CNC(C2CCCC(=O)N2)=O)cc1 52881,C1(SC=CC(=O)N2CC(c3cc(OC)c(F)cc3)(F)C2)CC2CC1CC2(F)F 52882,c1(C(C(=O)OC)NC(CCCCN(C(=O)OC)C)=O)ccc(F)c(Cl)c1 52883,C1(CNC(c2c(CC)nccc2)=O)CN(C(C2CCC(C)CO2)=O)CCN1C 52884,Cc1cc(C(=O)NC2CCN(C(=O)CSc3n[nH]c(=N)s3)CC2C)nnc1C 52885,C(=O)(C1CCCc2nncn21)NCCN(C(=O)C(C)n1ccnc1)CC 52886,C1(NC(C2(CN(C)C)CCCC2)=O)CCCN(C(=O)CCC2CNC(=O)N2)CC1 52887,C1(NC(C2(C(C)C)CCC2)=O)CN(C(c2ccc(N)c(Cl)c2)=O)CCC1CO 52888,C(=O)(C(O)CC(C)C)NC(C(=O)NC(c1c(C)cccc1)C)c1ccoc1 52889,C1(NC(C2CN(C(C(N3CCN(C)CC3)=O)=O)C2)=O)CN2CCC1CC2 52890,C1(NC(CC2(NC)CCC2)=O)CCC(CNC(=O)C=Cc2nc(C)cs2)CC1 52891,C(=O)(C1CNC(=O)c2ccnn21)N(CCCNC(=O)CN(C)S(=O)(=O)N(C)C)C 52892,C1(N(C(=O)COC2CCCCC2)C)CCCN(C(=O)CCC2CC2(C)C)C1 52893,N1(c2n(C)nnn2)CC2CC(NC(C3CN(C4CCOC4)C3)=O)C2C1 52894,C(=O)(CCCC(F)F)N1C(CNC(=O)CCc2nc(C3CC3)no2)CC(OC)C1 52895,c1(CN2CCC(CNC(=O)C=CCBr)C2)ccc2ccc(Cl)cc2n1 52896,C(C)(C(O)C(F)F)NC(C(CNC(c1cc(C(C)=O)[nH]n1)=O)OC)=O 52897,C1(CC(C)NC(C2(CC)CCOC2)=O)CCN(C(c2cccn2COC)=O)CC1 52898,c1(C(=O)NCCN(CCOC)C(c2cc(O)cs2)=O)csc(-c2ccoc2)n1 52899,C1(C(C)C)CCCN(C(=NCC2CCN(C)C(=O)C2)NCC2CCCCO2)C1 52900,c1(CCNC(c2c(CC)noc2)=O)cc(F)ccc1C 52901,c1(C(=O)NCCOC2CCN(C(CCNC(C)=O)=O)C2)c(Cl)ccc2c[nH]nc12 52902,Cc1c(C(=O)N(C)CCOCCNC(=O)CN2CCC(C)CC2)cccc1Cl 52903,N1(C(C(C)CN2CCOCC2)=O)CCC2CN(Cc3cc[nH]c3)CC12 52904,c1(CN(C(C)C)C)ccc(C(=O)NC(C)(C)C(C)NC(c2cnco2)=O)cc1 52905,CCS(=O)(=O)CC(=O)N(CC(CC(C)O)c1ccccc1)Cc1cccc(C)c1 52906,c1(CNCCC(=O)N(C(c2ccccc2)C)C)ccccc1-c1cnc(F)cn1 52907,CC1CC(C(=O)NCCCN2CCN(c3ccccc3)CC2)C1(C)C 52908,c1(C(=O)NC(C(C)=C2CCCN2)=O)cc(C)ccc1C 52909,C1(C(CC)C(=O)N2CC(N(C)C(C3CCCO3)=O)C2)CCC(C)CC1 52910,C1(NC(N2CC(C(C(=O)O)OC)C2)=O)C2Cc3ccc(Br)cc3C12 52911,C1(C(=O)NC(C2(O)CCN(C(C3(C)CC(F)C3)=O)C2)C)CCCOCC1 52912,N1(C(CC2CCCN(C(CCCC(=C)C)=O)C2)=O)CCn2ccnc2C1C 52913,c1(C(c2n(CC)nnn2)NC2CCCC2COC)cccc(C)c1C 52914,c1(-n2cc(C(N3CC=CC(NC(C4(C)CC(=C)C4)=O)C3)=O)s2)ccc(F)cc1C 52915,c1(C(=O)NCC(C)(C2CC2)NC(c2csc(=N)[nH]2)=O)cnc(-c2ccccc2)o1 52916,N1(C(CCCNC(N)=O)=O)CC2CCC(C1)N2C(C1CC1c1ccc(Cl)cc1)=O 52917,C1(c2n(C(C(=O)OC)C)nnn2)(NCCS(=O)(=O)CCO)CC2(C1)OCCO2 52918,Cc1cc(F)c(N)cc1C(=O)NC1CC(F)CN(C(c2cc([N+](=O)[O-])c[nH]2)=O)C1 52919,CC(C)CC(C)C(=O)NCC(C)(C1CCC1)NC(=O)Cc1nnc(S)n1C 52920,CCCCC(C)CCC(=O)NC1CC2CNC1C2 52921,N1(C(C2CC2COC)=O)CCC(OCC)C(CNC(C)=O)C1.c12cc(on1)C2 52922,C(C(C(=O)N1CCCC1CN(C)C)C(C)(C)C)NC(CC(=O)OCC)=O 52923,N(C(=NCCCCl)N1CCCC2(CC2)C1)CCNC1C(C)Cc2ccccc21 52924,CCCCC(C(=O)OC)NC(c1cc(C)[nH]n1)=O.C1(=O)C(O)C2CC(C2)N1 52925,CN1CCC(C(=O)N(C2CCCN(C(=O)CCc3nncs3)C2)C)C1=O 52926,S(=O)(=O)(c1cccc(F)c1C)N1CCCC(CNC(c2ccc(C(C)N)cc2)=O)C1 52927,C(=O)(CC(C)CC(F)(F)F)N(C1CCCCN(C(c2cc(C(C)=O)sc2)=O)C1)C 52928,c1(CC)ccc(C(N2CCNC(=O)C2)C(=O)NCCC2CC2)nc1 52929,C1(NC(CC(C)N2CCCC2=O)=O)C2CC1CN(C(c1ccc(Cl)c(Cl)c1)=O)C2 52930,c1(NC(C2C(CNC(C(COC)COC)=O)CCC2)=O)cnc2ccccc2c1 52931,C1(NC(=O)CC(F)F)CC2CC(C1)N(C(=O)CC1CCS(=O)(=O)C1)C2 52932,N1(C(C2(O)CCSCC2)=O)CCC(O)(NCCC(F)Cn2cc(CO)nn2)CC1 52933,c1(C(=O)NCCC2CCCN(C(c3cc(OC)ncc3)=O)C2)cc(C#N)[nH]c1C 52934,c1(C(=O)NCCCCC(C)NC(c2c(CC)cco2)=O)cc(C)ccc1C 52935,CN1CCN(C(C2C3CCC(=O)C23)=O)C(CNC(c2ccno2)=O)C1 52936,C1(NS(CC(C)C)(=O)=O)CC2CCC(C1)N2C(=O)C(C)(C)C 52937,c12ccc(o1)C(=O)NC1CN(C1)C2C.n1(CC)cc(C2(N(C)C)CCOC2)nn1 52938,c1(C(N2CC(O)(CN(C(C(CC)CC)=O)C)C2)=O)cnc(C(F)F)cc1C 52939,c1(SC)cc(C(=O)NCCC(C)NC(c2ccc(C)c(F)c2)=O)c(Cl)cc1Cl 52940,CCC(C)CC(C)NC(=O)C(CCOC)N(C(=O)CCOC)C 52941,c1(C(C(=O)N(CCNC(C(C=C)c2ccccc2)=O)C2CC2)C)cccc(O)c1 52942,c1(SC)cccnc1C(=O)NCC(C)CN(C(=O)C(C#N)=CC(C)C)C 52943,C(CC(C)C(=O)NC(CNC(c1coc(C(C)C)n1)=O)CO)=CCC 52944,C1(C(=O)NC(C(C)C)CNC(c2cc(-c3cccs3)on2)=O)CCC(C)(C)OC1 52945,N1(C(CC(COC)C)=O)CCCC2(C1)CN(C(=O)CC(C)CN(C)C)C2 52946,C12CCC(CC1)C(=O)N2.N1(CC)CCCC1CNC(=O)COC1CCOCC1 52947,c1(C(N2CCCC3(CN(C(COC)=O)C3)C2)=O)cc(O)nc2c(OC)cccc12 52948,CN1C(=O)C(=O)N(CC(=O)NC2CCN(C(=O)Cc3nncn3C)C23CC3)C1=O 52949,c1(NCc2[nH]nc(C(C3CCCO3)OCC)n2)cccc(F)c1.c12nnnn1C2 52950,C(=O)(C(C)CC1CCC1)NCC(CC)N(C(=O)CSCc1cccs1)C 52951,CCC(CCC(=O)NCC1(CC2CCC2)CC1)NC(C1CCCC(=O)N1C)=O 52952,n1(C(CC)C)ccc(=NC(=O)C2C3CC2N(C(=O)C(c2ccn(C)c2)C)C3)[nH]1 52953,n1(C(C(=O)NCCCN(C(C(C)=C(C)C)=O)C2CC2)C)nc(C)cc1C 52954,O=C(CC1CCCN1C(C12CCC(CC1F)C2)=O)N=c1ccn(C2CCC2)[nH]1 52955,C1(C(=O)NCCN(C(=O)C=NOC)CCC)CCN(c2cnccn2)CC1 52956,N1(C(C2C(C)C2C)=O)CCC(NC(C2(c3ccno3)CCC2)=O)C1C 52957,c1(NC(N(C2CCCN(C3CC3)C2)C)=O)ccc(F)c(Br)c1F 52958,c1(NC(C2C3(CN(Cc4cc(C)nc(C)c4)C3)C2)=O)cc(Cl)c(C)cc1[N+](=O)[O-] 52959,C=CCC(CC=C)C(=O)N1CCCC(C)C1CNC(c1cnc(S)nc1)=O 52960,C(Cc1ccoc1)(C(=O)NCC1CCCN1C)NC(CCC1(C)CC1)=O 52961,c1(OCC(N2CCC(NC(CC(n3c(C)cc(C)n3)C)=O)C2)=O)ccc(Cl)c(F)c1 52962,Cc1c(Cl)ccc(C(=O)NC2CCC(N(C(=O)COCC(C)(C)C)C)C2)c1N 52963,c1(CN(C)CC2CCCN(C(c3cnc(Cl)cc3I)=O)C2)cc(Br)cc(O)c1O 52964,Cc1nc2ccc(C(=O)NC(CNC(C3CC(=O)N(C)C3)=O)C(C)C)cc2s1 52965,c1(CNCC2N(C(C3C(C)(C)CCC3)=O)CC2)cc(Br)cn2ncnc12 52966,C12(NC(C(C3CCCOC3)OCC)=O)CCCC1N(c1nc(CC)ns1)CC2 52967,c1(C(N2CC3(CN(C(C(CC)CCOC)=O)C3)C2)=O)[nH]c2cc(C)ccc2c1C 52968,C(CCS(=O)(=O)NC(C)C(=O)NCC1(OC)CN(C(=O)C(F)F)C1)OC 52969,C#Cc1ccc(OCC(=O)NCCNC(=O)CC2CC(CC)=NO2)cc1 52970,N1(C(C2OCCN(C)C2)=O)CC2CC(C1)C2NC(=O)CCN(S(C)(=O)=O)C 52971,CC(CCCO)N=c1[nH]c(N2CC(C)(C)OCC2CCO)nc2c1SCC2 52972,c1(C(=O)NCC(C)(C2CC2)NC(c2ccnc(C3CC3)n2)=O)cc(F)cnc1O 52973,C1(NC(C(C2CCCC2)OC)=O)CCN(C(C2CCCC(OC)C2)=O)C1(C)C 52974,CC1(C)CC(NC(C2COCC2C(N)=O)=O)CN(C(c2ccon2)=O)C1 52975,Cc1cc(C(=O)Nc2nc(Cl)cc(Cl)n2)cc2nc[nH]c12 52976,c1(OCC)ccccc1C(=O)NCC(F)CNC(C1CC12CCC2)=O 52977,c1(C(=O)OC)cc(C(=O)NCC(C)(C)CNC(=O)CC2CCOC2C)c(F)cn1 52978,c1(-n2cc(NC(N3CCC(CC4CCCC4)C3)=O)nn2)ccc(C(=O)O)c(F)c1 52979,n1(CC(=O)NCCC(CC)(CC)NC(C(CC)C)=O)ccc(=O)c2ccccc12 52980,Cc1c(C(=O)NCC(C)CNC(C2(C(C)C)CCCO2)=O)cnc2ncnn12 52981,CC(C)(O)C#CC(=O)NCC1CN(C(=O)CC(C)(C)CN(C)C)CC1(C)C 52982,N1(C(C=C(C)C(C)C)=O)CCCCC(CNC(=O)Cc2nc(C(C)(C)C)cs2)C1 52983,Nc1cc(F)c(C(N2CC=CC(NC(=O)C3=CCCC3)C2)=O)c(F)c1 52984,CC1(C)CN(C(c2ccn(C3CCC3)n2)=O)C(CNC(=O)CNS(N)(=O)=O)CO1 52985,c1(C(=O)NC(CC)CN(C(=O)CCC(=O)N(C)C)CC)coc2c(F)cccc12 52986,CCCCC(CC(=O)NC(COC)CCO)NC(C1(C2(C)CC2)CC1)=O 52987,C12(C(N3CC(NC(C4(C)CCO4)=O)C3)=O)CC3CC1(CO)CC3C2 52988,c1(C(=O)NCC2C3CN(C(CCC(N)=O)=O)C2CCC3)cc2cccc(F)c2o1 52989,c1(C(=O)NCCCC2N(C(c3cc(C(=O)OC)[nH]n3)=O)CCC2)n[nH]c(C)c1C 52990,c1(C(N2C(CNC(CC(=O)N(C)C)=O)CC2)=O)cc(CO)ccc1Cl 52991,N1(C(c2cn(CC=C)nn2)=O)CCN(C(=O)Cn2cc(C)cn2)CC(O)C1 52992,c1(CC(=O)NCC(CC)NC(c2cc(O)cc(N)c2C)=O)ccc([N+](=O)[O-])cc1 52993,N1(C(C(C(C)C)NC(C)=O)=O)CCCN(C(c2sc(F)cc2Cl)=O)CC1 52994,c1(CCC)cccc(C(N2CC(NC(=O)C3=C(Cl)CC3)C(O)C2)=O)c1 52995,C1(O)(CNC(CCn2ccc(C)n2)=O)CCCN(C(=O)CCCCCC#N)CC1 52996,c1(OCC(=O)NC(C(C)NC(=O)C(C)(C)N(C)CCO)CO)cccc(C#N)c1 52997,c1(C(=O)OC(C)CC(C)(C)O)cc2c(s1)CCCC2 52998,Nc1ccc(C(=O)NCC2(NC(C3CCOC3C3CC3)=O)CCC2)cc1Cl 52999,c1(OCC)ccc(-c2cc(C(=O)Nc3c(C)ncnc3C)ccn2)c(F)c1 53000,CC(CCO)C(=O)N1CC(N(C(=O)C(c2ccc(Cl)cc2)C)C)C1 53001,C=CCC(C(=O)NCC1CCC2(CN(C(C3(CO)CC3)=O)C2)O1)C(C)(C)C 53002,N1(C(C(=O)NCC)=O)CCC(NC(c2cn(CC(N)=O)nn2)=O)C(F)C1 53003,C1(C(=O)NCCCN2CCC(NC(C(C(C)C)O)=O)C2)C2CCC(F)(F)C12 53004,CCCC(CCC)CC(=O)N1CCC(O)C1C(=O)NCC(O)C1(Cl)CC1 53005,C1(CC)CCCN(C(=O)C(COC)CNC(C2CCC=CCCC2)=O)CC1 53006,c1(NC(C(CC)CCOC)=O)cc(C#N)cnc1C 53007,c1(C(=O)NC(CNC(c2nnc(C)s2)=O)C(C)C)cccc(S(=O)(=O)CF)c1 53008,C1(c2ccccc2)(NC(CC2CC(C)C2)=O)CC(NC(=O)C(C)CO)C1 53009,C1(C(=O)NC(c2cnc(C)s2)C)CC(O)CN1C(c1cn[nH]c1)=O 53010,C1(NC(C(C=CC)O)=O)C(C)(C)C(NC(=O)Cc2cccs2)C1(C)C 53011,C=C(C)CCCC(=O)N1CCCC1c1cn(-c2cc(CC)ccc2C)nn1 53012,c1(C(=O)NC2CCN(C(CCOCCC)=O)CC2C(N)=O)cc(N)c(F)cc1F 53013,S(=O)(=O)(c1ccc(NCCC2CC2C)cc1Br)N1CCC(NC(C)=O)CC1 53014,c1(C(=O)Nc2nc(C)c(Cl)c(Cl)c2)cn2c(n1)CN(C(C)(C)C)CC2 53015,N1(C(CC2(C=C)CCC2)=O)CC2(C1)CN(C(c1ccc(Cl)cc1C)=O)CC2CO 53016,N1(C(c2cc(OC(C)C)no2)=O)CC(C)OC2(CCOC2)C1 53017,C1(C)(C(N(C)CC2CN(C(=O)CCN3CCCC3)CCO2)=O)CCCCNC1=O 53018,c1(-n2cc(C3(C)CN(C(Cc4scc(CC)n4)=O)C3)nn2)ccc(Cl)cc1 53019,c1(C(N(C)CCN(C)C(c2cc(C(N)=O)c[nH]2)=O)=O)cc(C(C)(C)C)n(C)n1 53020,CC1=C(C)CC(C)(C(N2CCCN(C(c3cnc[nH]c3=N)=O)CC2)=O)CC1 53021,N1(C(CCCC=C)=O)CC2(CCN(C(C3CC3c3cscn3)=O)CC2)C1C(C)C 53022,Cc1c(C(=O)NCCc2cn(-c3cccc(F)c3)nn2)oc2ccccc12 53023,C1(C(N(CC)CC2CCCN2C(=O)CP(C)(C)=O)=O)OCC2CCCC12 53024,c1(CC)nc(CC(=O)NC2CC(N(C(=O)C(C)n3cccc3)C)C2)co1 53025,C(=O)(C(O)CC(C)C)N1CC(N2CCN(C(c3c(C)nns3)=O)CC2)C1 53026,C=CC(C)(C)C(=O)NCC(C)(C1CC1)NC(=O)CC1CC1C1CC1 53027,c1(C(=O)OC)cc(C(=O)NCC(O)CN(C)C(c2ccn(C)n2)=O)c(C)s1 53028,C=CCC(CC)C(=O)N1CCCOC(CCNC(=O)C=Cc2cccc(Cl)c2)C1 53029,c1(C(=O)NC2CN(C(COC(C)(C)C)=O)C3C2C3)cc(S(N)(=O)=O)ccc1Cl 53030,N1(C(c2cnc(CC)nc2)C(=O)NCc2ccccc2)CCCC2C1CCN2C 53031,C1(C(=O)NC(CCCC)CNC(c2cc3cscc3s2)=O)CCCC(F)(F)CC1 53032,C1(C)(CNC(c2sccc2C(=O)NC)=O)CCN(C(=O)Cc2cc[nH]c2)C1 53033,C1(N(C(C(CC)n2ccc(C3CC3)n2)=O)C)CCN(C(=O)CCNC(N)=O)CC1 53034,C1(CNC(c2nc(C)sc2)=O)CC2CCC1N2C(=O)C(C)NC(c1ccco1)=O 53035,c1(SC)nn(C)cc1C(=O)NCc1ccc(C(C)NC(=O)CC(C)F)cc1 53036,C=CC(C)(O)CC(=O)NCCOC1CCN(C(C2CCC(=O)NC2)=O)CC1 53037,N1(C(C(CC)F)=O)CC(C)(C)OC2(C1)CN(C(c1nn(C(=O)OC)cc1Cl)=O)C2 53038,C1(NC(C(CC)n2cccn2)=O)CCCCCN(C(=O)C=Cc2cnc[nH]2)C1 53039,Cc1ccc(F)c(C(=O)NCC2CC(C)N(C(=O)CSCc3ccncc3)C2)n1 53040,c1(CC)nc(C(N2CCC(O)(Cn3cc(-c4csnn4)nn3)C2)=O)c(C)o1 53041,c1(C(=O)NC2CCN(C(c3[nH]c(=NCC)sc3)=O)C23CC3)cnc2ncccn12 53042,C(CN=c1nc(-c2ccccc2)nc[nH]1)(N(C(=O)C(C)(C)C1CCC1)C)C1CC1 53043,c1(C(NNC(C2CC3CC(C(=O)O)C3C2)=O)=O)nc2ccccn2n1 53044,N1(CC(N2CC(CNC(=O)Cc3ccsc3Br)C2)=O)CCCNC1=O 53045,N1(C(C(C)OC)=O)CCCCC2(C1)CN(C(=O)Cc1csc(S)n1)C2 53046,CCC(CC)C(F)C(=O)N1CCC(CC(N2CCCNC(=O)C2)=O)C1(C)C 53047,c1(OC)cc(C#N)ccc1C(N1CCC(CS(N)(=O)=O)CC1)C(=O)NC(C)(C)C 53048,C1(C(C)NC(C2N(CC)CC2)=O)CCN(C(=O)CC2CCC(=O)C2)CC1 53049,C1(NCC2CCCN(C(C)(C)C)C2)CC(c2ccccc2[N+](=O)[O-])=NO1 53050,C(C(=O)NNC(=O)c1coc(-c2ccc(C)cc2)n1)SC(CCC)C 53051,N1(C(c2c(C)cno2)=O)CC(NC(c2c(Cl)cncc2Cl)=O)CC(O)C1 53052,C(CC1CC1)(C(=O)NCCCNC(C)=O)OCC.C12(CCC1)CC(=O)N2 53053,N(C1CCc2c(Cl)ccc(F)c21)CC1N(C)CCN(C(=O)OC(C)(C)C)C1 53054,C1(NC(C=CSC)=O)CCCC(N(C)C(c2cc(N(C)C)ccn2)=O)C1 53055,C1(CC)C(NC(C2CCCN2C)=O)CCN1C(=O)CCC(=O)OC(C)(C)C 53056,N1(C(=O)CC2CCCO2)CCC2(C1)CN(C(c1ccc(Cl)c(F)c1)=O)CCO2 53057,c1(CC)nc(C)cc(=NC(CCN(C)C(C2CC3(CCOCC3)C2)=O)C(C)C)[nH]1 53058,C1(NCc2c(OCC)cccc2)CCC(N=c2ccn3ncc(Br)c3[nH]2)CC1 53059,C1(CCC(=O)NCC(CC)N(C)C(C2CC(=O)N(C)C2)=O)CCCCN1C 53060,NS(=O)(=O)c1ccc(CN2CC3CC3(C(N3CCCC4(CCO4)C3)=O)C2)cc1 53061,C1(C)(C(N2CCOCC(NC(CSCCC)=O)C2)=O)CCCNS1(=O)=O 53062,C(=O)(C1CCCc2scnc21)N1CC(O)CCC(NC(c2c(C)nc(C)s2)=O)C1 53063,N1(C(C(CSC)OC)=O)CCCC(N(C(=O)Cc2cc(C)cs2)CCO)C1 53064,Cc1oc(Cl)nc1C(=O)NCCCCC1CN(C(=O)C(=O)NCC(F)(F)F)C1 53065,C1(C#N)(C(=O)NCC2CN(C(c3c(C)n(C)nn3)=O)C2)CCOCC1 53066,c1(CNC(c2c(C(N)=O)coc2)=O)c(F)cc(F)cc1F 53067,C1(CC)CN(C(C2(C(N)=O)CC2)=O)CCC1NC(=O)CCc1ncc[nH]1 53068,CC(C)C(F)(F)CC(=O)NC(C)(CNC(c1cc(Cl)ccc1F)=O)CO 53069,c1(C(=O)OC)ccsc1COC(=O)C(N1CCCC1CSCCOC)=O 53070,c1(OC)c(C(N2CCC(C(N3CC(O)C3)=O)C2)=O)cnn1-c1ccccc1 53071,Cc1nc(CCC(=O)NCCC2CCN(C(c3c[nH]nc3C(C)(F)F)=O)C2)cs1 53072,c1(OC)ccc(CC2CCCOC2C2CCN(C(=O)SC3CC3)CC2)c(OC)c1 53073,C1(NC(c2ccccc2OC(F)F)=O)C2CCN(C(=O)C3=COCC3)CCC12 53074,C1(CCNC(C2C3CCN2CC3)=O)CCCCN1C(C1CCCCC1O)=O 53075,CC1CN(C(=O)C(C)(C)C(F)(F)F)CC(C)C1NC(=O)Cc1ccc(F)cc1 53076,N1(C(C(C)NC=O)=O)CCC(CCNC(c2cc(CCO)on2)=O)C1 53077,c1(C(N2C(C)CC(CNC(CC3CC(=C)C3)=O)C2)=O)ccc2nccn2n1 53078,n1(CC)ncc2c(C(=O)NCCC3(NC(=O)CC(C)(C)O)CCC3)cc(C)nc12 53079,C1(CC(=O)NC2CCN(C(CN(CC)CC)=O)C2)CCCN(C(C)COC)C1 53080,N1(C(C2(C#N)CC2)=O)CCC2CCN(C(C3CC3c3ncccc3Br)=O)C2C1 53081,C1(C2CCN(C(C3CC3C(C)O)=O)CC2)(NC(CC2CC(C)C2)=O)CC1 53082,C1(C(=O)NCC(CN(C(C2(CC=C)CC=CC2)=O)C)O)CC(F)(F)C1(C)C 53083,c1(C(N2C(CNC(=O)Cn3cc(Br)cn3)C=CC2)=O)ccc(O)c(F)c1F 53084,c1(C(N2CCC(N(C(C=CSC)=O)CC(C)C)CC2)=O)cc(S(N)(=O)=O)c[nH]1 53085,c1(OCC)cnc(CC(N2CC=CC(NC(c3nc(C)oc3C)=O)C2)=O)cn1 53086,CC1(C)C(C(N2CC(O)(CNC(=O)C(F)=C3CCC3)C2)=O)C1(F)F 53087,C1(NC(c2scc(OC)c2)=O)COCCN(C(=O)C(F)(F)c2cnccn2)C1 53088,C(=O)(C(O)C(F)F)N(CC(C)N(C(=O)CCCNC)C)C.CC(C)CC(C)NC(N)=O 53089,N1(C(c2ccc(CC)nc2)=O)CCCC(NC(c2cn[nH]c2)=O)C1C 53090,c1(NCc2c(C)nc(C)c(C)n2)nc(=N)[nH]c(=NCC2=COCCO2)[nH]1 53091,N1(C(C2=CCCC2C)=O)CCC(C(=O)NCC2CC3CCCC3C2)C12CCC2 53092,c1(C(=O)NC(C)C(C)NC(C2(CCO)CC2)=O)cnc(-c2ccccc2Cl)nc1 53093,N1(C(CCc2cn(C)nc2)=O)CCCC1(C)CNC(C1CC1c1ccco1)=O 53094,C#Cc1ccc(C(=O)N(CCC(=O)NCC2CC2C(N)=O)C)c(C)c1 53095,N1(C(C23C(C(=O)OC)(CCC2)C3)=O)CCCCC(NC(C2(C)CC(C)(C)C2)=O)C1 53096,c1(OC)c(C(=O)NCCC(C)NC(C2(C)COC(=O)C2)=O)cnn1C 53097,C1(NS(=O)(=O)CC2CCC3(CC2)COC3)CCCC12CCOCC2 53098,N1(C(CC=CC=C)=O)CCCC2(CNC(C34CCC(C)(C3)OC4)=O)CCCC12 53099,C(CCC(=O)NCCCC1CC1)(C(C)C)NC(c1ccc(C)c(F)c1)=O 53100,Cc1ccc2c(N3CCC3(C)C(=O)Nc3ccc(Cl)cc3CO)ncnc2c1 53101,c1(C(=O)NC(C(C)C)CCNC(=O)Cc2cscn2)cccc2nc(CO)[nH]c12 53102,n1(CC)cc(C(=O)NC2CCN(C(C3CCOC3)C)C2)c2ccccc12 53103,c1(C(=O)Nc2c(C(=O)NC)cc(Br)cc2)cn2c(n1)CN(Cc1cc[nH]c1)CC2 53104,N1(C(CSCC)=O)CCc2ccccc2C(NC(=O)CC2(COC)CC2)C1 53105,c1(CNC(=O)CC2(O)CNC2)ccc(CNC(=O)C(c2ccccc2)F)cc1F 53106,CCC(C)(C)C(C(=O)NCC12CC1CN(C(c1ncc[nH]c1=O)=O)C2)OC 53107,c1(C(C)NC(c2c(C#C)c[nH]n2)=O)cc2ccccc2n1C 53108,C1(CC(=O)NCC2N(C(c3ccc(OC)cc3)=O)CC=C2)NC(=O)CN(C)C1=O 53109,C1(F)(CNC(C2Cc3nncn3C2)=O)CCCN(C(C2(CO)COC2)=O)CC1 53110,c1(N2CCC(CCC)C2)nc2ccccc2c(=NCC(F)(F)Br)[nH]1 53111,C1(C(=O)NCCOC2CCN(C(c3cc(F)cs3)=O)C2)CCc2nc[nH]c2C1 53112,N1(C(CCC=C)=O)CCC2CCCN(C(=O)CN(C)CCc3ccccc3)C2C1 53113,Cn1cc(C2CC(C(N3CCC(N4CCOC4=O)CC3)=O)C2)c(C2CCC2)n1 53114,N1(C(COCOC)=O)CCCOC(CNC(=O)CC2CCCCO2)C1 53115,N1(C(CC(C(C)C)C)=O)CC2OCC(NC(C3(CCN(C)C)CC3)=O)C2C1 53116,c1(C(C)NC(=O)CC2(C(=O)NC3(O)CCCCC3)CCC2)cc2ccccc2o1 53117,Cn1nc(C(N2CC3(CNC(c4ccsc4)=O)CC2CO3)=O)cc1C#N 53118,N1(C(C(=O)Nc2cnc(OC)nc2)=O)CCn2c(C(C)(C)C)nnc2C1 53119,C(=O)(C(CCC)=CCC)NCC(C1CCCCC1)NC(C1(C=C)CC1)=O 53120,c1(SCCC)ccc(C(=O)NCC2(CNC(=O)C(OC)SC)CC2)o1 53121,c1(CC2(Nc3c(C(=O)O)occ3)CCC2)ccc(Cl)cc1 53122,c1(C(=O)NCC2(CNC(CCN(C(CCC)C)C)=O)CC2)csc(Cl)c1Cl 53123,c1(CC(C)C)ccc(C(C)C(=O)NCCCCNC(C2CCOC(=O)N2)=O)cc1 53124,Cc1cc(S(N)(=O)=O)oc1C(=O)NCCC1CCCCN1C(C1COC(=O)N1)=O 53125,N1(C(C(C)(N(C(C2CCC(C)(CC)O2)=O)C)C2CC2)=O)CCCC(C)(COC)CC1 53126,c1(C(N2CC(CCNC(CC)=O)C(C)C2)=O)cc2cc(Cl)cnc2[nH]1 53127,c1(NC(C(c2ccccc2)NC(C2CC(=O)NCC2)=O)=O)cccc2c1CCO2 53128,C1(CNC(CCCCN(C)C(c2ccn(C)c2)=O)=O)CCCC(C)(C)C1 53129,C1(OC)(OC)CC2(CC(NC(N3CCN(C4CCCCCC4)C(=O)C3)=O)C2)C1 53130,CC(CCNC(C1CCC(C(N)=O)CC1)=O)CCNC(=O)C(c1ccnn1C)C 53131,C(C)(C)(CC(=O)NCCN(c1cn(C2CCOC2)nn1)CC1CC1)NC(COC)=O 53132,c1(C(=O)NCc2nc(CNC(C3C(C)(C)C3)=O)sc2)cc(S(N)(=O)=O)ccn1 53133,C1(C(N2C(CNC(CCS(C)=O)=O)CCC2)=O)CCOCC12CCC2 53134,C1(C(=O)NC(CCN(C(c2cnc(C(C)C)s2)=O)C)C)CCC(=O)N(C)C1 53135,N1(C(c2cn(CCC)nc2)=O)CCC(C(=O)NCC2CC(C)=NO2)C12CCC2 53136,N1(C(c2c(CC=C)c[nH]c2)=O)CC(C)N(C(=O)C=CC=CCOC)CC1C 53137,c1(OC)ccc(OCC(N2CC(NC(c3cnn[nH]3)=O)CC2CO)=O)cc1C 53138,N1(c2nc(SC)c(C)cn2)CCC2CC(C(=O)NCCN(C)C(=O)C3CC3)C2C1 53139,O=C1CC2CC(CC(N3CCCC(O)(CNC(C4CCC(=O)NC4)=O)C3)=O)C1C2 53140,CC1CN(C(=O)C(C2CC2)NC(=O)C(F)C(C)(C)O)Cc2c[nH]nc21 53141,CCCC(C)CC(=O)N1CCCC(CNC(c2ccc(-c3cc[nH]n3)s2)=O)CC1 53142,Cn1c(O)nc2c(N3CCCN(CCC(F)(F)C(F)(F)F)CC3)ncnc12 53143,c1(C(N2CC(COC)(CNC(=O)C(F)(F)C3(O)CCC3)C2)=O)ccnc(C)c1O 53144,C1(NC(C(C)=CC2CC2)=O)CCC(C)(NC(C2CNC(=O)N2)=O)CC1 53145,C1(CC)CCN(C(=O)C(F)F)C(C(=O)NCC2(C)CCCOC2)C1 53146,N1(C(c2c(C)ocn2)=O)CCN(C(=O)CNC(c2ncn(C)n2)=O)CC1 53147,c1(CC)cc(NC2CC(NC(=O)CCC(F)F)C2(C)C)ncn1 53148,C(=O)(C(O)C(F)(F)F)N1CC(OCC)C(CNC(=O)CCc2ccoc2)C1 53149,c1(C(N2C(CNC(=O)C(O)C3CC3)CC(O)C2)=O)cnn2c1OCCC2 53150,C1(C(=O)NC(C)CN2CCCC2CC(C)O)CCN(C(=O)C2CC2)CC1 53151,N1(C(c2cnc(CCC)s2)=O)CCCC(N(C)C(c2ccn(C(C)C)n2)=O)CC1 53152,C12(C(=O)NC3(CNC(c4cc(C)c(Cl)s4)=O)CC3)C3C4C1C1C2C3C41C(N)=O 53153,N1(C(C(C)C2CCCC2)=O)CC2CCC1C2NC(c1ccc(Cl)c(O)c1)=O 53154,Cc1ccc(C=CC(=O)NC2CCN(C(C3CS(=O)(=O)C3)=O)CC2F)nc1 53155,c1(OC(C)(C)C)nccnc1NC(N1CCC1Nc1cccnc1)=O 53156,C=CCCCC(C(=O)N1CCn2ncnc2C1)Oc1cc(C(=O)NCC)on1 53157,Cc1c(CC(=O)NCCCNC(=O)CC2C=CCC2)cccc1[N+](=O)[O-] 53158,c1(C(=O)NCCC(CNC(C(C)OCC)=O)=C)cc(N(C)C)ncn1 53159,CC12CCN(C1)C2=O.C1(OCC(=O)NCC(F)(F)F)CC(=O)N1 53160,C1(NC(=O)CCc2cn[nH]c2)CC2CN(C(c3cccc(Cl)c3Cl)=O)CC12 53161,C1(NC(C2CCN(C(c3cn(CCC)nc3)=O)C2)=O)CCN(C)CC1C#N 53162,C1(C(=O)NC(C2CCOCC2)C#C)CCC(C)N1C(=O)CC1CCOC1 53163,C(CCN=c1[nH]c(N2CCOC(CF)C2)nc2c1SCC2)OCC(C)C 53164,c1(OC(N2CC(N(C(COC)=O)C)C(F)C2)=O)cc(C(C)=O)ccc1SC 53165,Cc1cccc(C(=O)N(C)CC2CCCC2NC(C2(O)CCC(C)CC2)=O)c1N 53166,N1(CC(N2CC(O)(CNC(C3(c4ccc(Cl)cc4)CCC3)=O)C2)=O)CCCCC1=O 53167,C1(NC(C2C(C)CCC2)=O)(CNC(C2CC(F)(F)C2)=O)CCOCC1 53168,C1(O)(C(C)NC(=O)CC2CSCCO2)CCN(C(=O)C(C)(C)C2CCCC2)CC1 53169,C(c1cccnc1)=C(C(=O)NC(CCOC)CNC(=O)CCc1cc(C)no1)F 53170,C1(CN(C(=O)CCN2CCC2)C)CCN(C(c2cn(C3COC3)nn2)=O)CC1 53171,C1(C(=O)NCCCn2cnnc2)CCC2CCC1N2C(=O)Cc1ccsc1 53172,N1(C(C)=O)CC2=C(C1)CN(C(=O)Cc1sccc1-n1cccc1)C2 53173,CC(CC(=O)NOCCCCC1CC1)NC(=O)C(CO)NC(N)=O 53174,C(=O)(CC(C(F)(F)F)NC)NC1CN(C(C2(CC#C)CCCCO2)=O)CC1C 53175,N1(C(C2(CC#C)CCCCO2)=O)CCC(Nc2ncnc(=N)[nH]2)C(F)(F)CC1 53176,C(=O)(C1=CC2CCCC12)NCC(C)CNC(c1c(O)cc(F)cc1F)=O 53177,N1(C(C(CCF)NC(C(CC=CC)C)=O)=O)CCCNC(=O)C1 53178,C1(NC(C2CC3CC2C2CC32)=O)CCC2CN(C(=O)C=Cc3cscn3)CC2C1 53179,N1(C(C(CC2CC2)NC(Cc2cccc(C#C)c2)=O)=O)CC(F)(F)CCC1C 53180,c1(OCC)ccc(NC(=O)NCCOC2CC2(F)F)cc1OC 53181,Cc1sc2ncnc(N3CCC4CCC(C3)N4C(=O)NC3CCC(C)C3)c2c1C 53182,c1(C(N2CCC(CNC(CC(C)OC)=O)CC2)=O)ccc2c(c1)CC(C)(C)C2 53183,c1(CNC(=O)CCN2CCOC2=O)ccc(-c2ccccn2)cn1 53184,Cn1cc2c(n1)CCCC2C(=O)NCC(C)(O)CNC(=O)CCC1CCCCC1 53185,N1(C(c2cnn(CC)n2)=O)CCCC(NC(c2ccnc(Cl)c2O)=O)C1C 53186,C#CC1(CC)COCCN1C(c1nc(CC)cs1)C(=O)NC1CC(F)(F)C1 53187,C1(C(N2CCSCC2C2CC2)C(=O)NC2(C)CC2)CCOC2(CCOCC2)C1 53188,N1(C(CC(CC)O)=O)CC(C)CN(C(c2[nH]ccc2C2CC2)=O)CC1C 53189,Cc1c[nH]c(=NCCC(C)NC(C2CCCC2)=O)nc1S(C)(=O)=O 53190,C1(NC(CCC(C)CN(C)C)=O)CCCCC12CCN(C(=O)CNS(N)(=O)=O)C2 53191,c1ccc(CNC=O)cc1.C1(CN(C)C(C2CC(N(C)C)C2)=O)CCCO1 53192,CC1CN(C(c2cnc(C3CC3)s2)=O)CCCN1C(=O)CC1CCCCC1O 53193,Cc1sc(O)nc1C(N1CCCC(NC(c2cnc(Br)s2)=O)C1)=O 53194,C(=O)(CCCCC(N)=O)N(C1CCN(C(c2cnc(C)s2)=O)CC1)CCOC 53195,N1(C(CC2CC(C)(C)C2)=O)CC2CCCC(NC(c3nc(Cl)c(Cl)s3)=O)C2C1 53196,C1(C(N(C)CCNC(c2cccc(=O)o2)=O)=O)CC(C)(C)OC1(C)C 53197,C(=O)(C(C)(C)S(C)(=O)=O)NC1CN(C(c2c(OC)c(F)ccc2)=O)CC(C)C1 53198,CC(C)CCC(=O)NCCN(C)C.C12CC1C(=O)N(C)C1(CC1)C(=O)N2 53199,C1(C#N)(C(=O)NC(C)(C)CNC(C2CCCN(CC(F)(F)F)C2)=O)CC12CCC2 53200,N1(C(CCc2n(C)cnn2)=O)CCN(C(=O)CCc2cccc(F)c2Br)C2CC12 53201,C1(C(=O)NCC2(CNC(CC(C)C)=O)CC2)CC(C)CC(C)(C)C1 53202,N#Cc1ccc(=NCC(=O)N2CCCOC(CNC(c3n[nH]cc3Cl)=O)C2)[nH]c1 53203,C(CN=C(NCC(COCC)C(=O)OC)N1CCC(N2CCCC2=O)C1)OCC 53204,N1(C(CC(CC)SC)=O)CCC2(C=C(C(=O)N3CCN4CCCCC4C3)C2)C1 53205,c1(CC(N2CCCC(N(C(=O)CC(C)(C)F)C)C2)=O)noc2ccc(O)cc12 53206,Nc1c(C(=O)NCC(=O)NCC2CCOC2)cccc1F 53207,C1(C(=O)N(C)CC2(CNC(=O)CC3(C(=O)OC)CC3)CC2)(OC)CS(=O)(=O)C1 53208,c1(CC)cc(N)c(C(N2CCCC(C)CC2)=O)cc1F 53209,c1(C(N2CCCC(CNC(C(CC)C(C)O)=O)CC2)=O)cnc2c(F)cccn12 53210,CC1(C)CCCCC1(CO)NC(C1CCC1C1CC1)=O 53211,c1(OC)ccc(CC(=O)NC2(C)CCN(C(C34CCC(OC)C3C4)=O)C2)cc1Cl 53212,C1(C(N(C2CCN(C(C3CC3C#N)=O)CC2)CCC)=O)CN(C)CCO1 53213,c1(C(=O)NCCC2CCN(C(CC3ON=C(C)C3)=O)C2)cc2cccnc2s1 53214,c1(COC)ncc(C(=O)NCCC2COCCN2C(=O)C(F)C(C)C)c(O)n1 53215,Cc1nc(N2CC(NCc3ccccc3Br)C3(CC3)C2)c2c[nH]nc2n1 53216,C1(NC(C=CC=CC)=O)CS(=O)(=O)CC1NC(C1(S(C)(=O)=O)CC1)=O 53217,C1(C(N(c2cccc(O)c2)CC)=O)CCC2CCC1N2C(=O)C(O)CC(C)C 53218,C1(C(N2CCC(CNC(COCC(C)(C)C)=O)C2)=O)CCNC(=O)C1 53219,C(=O)(C(CC(C)C)OC)NC1CC(C(=O)NCC(=O)OCCCC)C1 53220,CCCCC(=O)C(=O)N1CC(C)CC1C(N1CCCC(COC)C1)=O 53221,C1(C(N(C)CC2CCCN2C(c2ccc(Cl)o2)=O)=O)CC2CC1C1CC21 53222,C1(CNC(C=COCC)=O)COCC2(CCN(C(=O)CCc3ncccn3)C2)O1 53223,CCCCCC(=O)N1CCC(F)(CNC(=O)C(C(C)C)c2cnn(C)c2)C1 53224,C(=O)(C1CCCc2cn(C)nc21)NC(C)CCC(C)(C)O 53225,C1(C2CCN(C(c3cncc(Cl)c3)=O)C2)(NC(Cc2c(C)noc2)=O)CC1 53226,C(=O)(CCC(C)S(C)(=O)=O)NC1CN(C(c2c(C)nc(C3CC3)s2)=O)CC12CC2 53227,c1(C(N2C(C(=O)NCC34COC(CF)(C3)C4)CCC2)=O)ccc2ncncc2c1 53228,N1(C(C(CCC)C(C)C)=O)CCC2(CC1)COC(CNC(c1cscn1)=O)C2 53229,c1(OC)cc(C(N2CCC(C)(NC(C3CCS(=O)(=O)N3)=O)CC2)=O)cc(F)c1 53230,CC(C)CCC(O)C(=O)N1CCCC(F)(C(=O)NC2CCC(N=[N+]=[N-])CC2)C1 53231,N1(C(c2c(C)scc2)=O)CCCC2(NC(=O)Cc3ccccc3[N+](=O)[O-])CC2C1 53232,Cc1oc(Br)cc1C(N1CC(C)(NC(C2CC23CC(O)C3)=O)C1)=O 53233,N1(C(C=COCC)=O)CCOCC1CN(c1ccccc1)C(=O)C(C)=C(C)C 53234,Cc1c(F)ccc(C(N2CCOCC2)C(=O)N(C2CC2)Cc2ccccc2)c1Cl 53235,c1(CCC(=O)NCC(CC2CCCO2)OC)cc(C)nc2c(F)cccc12 53236,C1(CC(N2CCCC(C)C2CNC(=O)C=C2CCCC2)=O)Cc2ccccc2N1 53237,N1(C(c2cn(C)nc2C(F)(F)F)=O)CC2CCC(C1)N2C(=O)CC1CCC1 53238,C1(C(=O)N)CC2CCC1C2.C1(CC=C)(N)CN(C(C2(CF)CC2)=O)C1 53239,N12CCOCC1NCCc1ccc(o1)C2.C(=O)(CCc1nccs1)NS(C)(=O)=O 53240,Cc1coc(C)c1C(=O)NCC(C)CN(C(=O)CSCc1csc(=N)[nH]1)C 53241,n1(C(=O)NCC2CCCN2Cc2c[nH]c3ncccc23)c(=O)oc2ccccc12 53242,CCC(O)C(C)C(=O)NCC(C)(C(C)C)NC(c1oc(C(F)(F)F)nc1C)=O 53243,c1(CC)nccnc1CNC(=O)C(C)(CSC)NC(=O)C=CC1(C)COC1 53244,Cc1cn2c(n1)C(C)CC(C(=O)NC1CCC1NC(=O)CCC(C)(C)C)C2 53245,N1(C(Cc2c(F)ccc(C)c2)=O)CC2CCC(C1)N2C(c1cc(C(N)=O)co1)=O 53246,c1(C(N2CCC(C)(NC(c3n(C)c(Cl)c(Cl)c3)=O)C2)=O)nc2c(s1)COCC2 53247,C(=O)(CCC(F)(F)CN=[N+]=[N-])NC1C(C)(CNC(C=CCOCCOC)=O)CCC1 53248,CC1(C)CCN(C(C2(C(N)=O)CC2)=O)C1CNC(C1CCCC(=O)N1)=O 53249,C(=O)(CC1CCCc2ccccc21)NC1CC(CNC(C2(C)CC=CCC2)=O)C1 53250,C(=O)(C1=COCCC1)NCC1CCN(C(C(C(C)C)OCC(C)C)=O)C1 53251,N1(C(Cc2c(C)con2)=O)CC(NC(=O)CCC2CCC(=O)N2)C(C)C1 53252,n1(CC(=O)NC2(CC=C)CN(C(=O)C(F)CCC)C2)nc2c(n1)CCCC2 53253,c1(CC(N2CCCN(C(C(C(C)C)F)=O)CC2CO)=O)ccc(S(N)(=O)=O)cc1 53254,C1(OC)CC(CNC(=O)C(C)(C)c2cccs2)N(C(C2CCOC2C2CC2)=O)C1 53255,C(=O)(C1=CCCN(C(c2ncccc2F)=O)C1)NC(c1ccc(O)nc1)C 53256,C1(C(=O)NCC)CN(C(=O)C(c2ccn(C)n2)C)CC12CCC2 53257,c1(OC)cc(NC(=O)C(C)N(C(=O)CC(C)n2ccnc2)C)ccc1F 53258,c1(C(N2CC(CNC(CCSCCCC)=O)OCC2)=O)cccc(C)c1Cl 53259,N1(C(C=CC(C)C)=O)CC2CN(C(=O)C=CC3COC(C)(C)O3)CC2C1 53260,c1(NC(CC)CN(C(=O)CC2=NNC(=O)C2)CC)cnc2cc(F)c(F)cc2n1 53261,n1(C(C(=O)N(CC(C)C)CCN(C)C)C)cc(CN)nn1 53262,C1(OC(C)C)CCN(c2nnc(Cc3ccccc3Cl)n2CC2CCN2C)CC1 53263,C#CCC(C)(C)C(=O)N1CC(O)(C(F)C(=O)NCC(CC)C(C)(F)F)C1 53264,CC1=NN(C)C(=O)C1CC(=O)NCC1CC1CNC(=O)COCC1CC1 53265,C1(C(=O)NCC(C)NC(=O)CC2COCCO2)CCCCN1C 53266,N1(C(C2C(COC)C2)=O)CCC(C(C(C)C)NC(C2C(C(F)F)C2(C)C)=O)CC1 53267,C1(NCc2ccc(C(=O)OC)cc2)CC2(C1)CC(NC(c1cccnc1)=O)C2 53268,c1(OCC)ccc(C(N2CCN(C(=O)CSC)CC2)C(=O)NCCC(C)O)nc1 53269,C1(C(=O)NC(C)CNC(=O)Cn2ccnn2)CCCC(=O)C1 53270,c1(C(=O)OC)cc(C(=O)NC2CCC2NC(=O)COC2CC=CC2)ccc1F 53271,N1(C(c2ccc(Cl)c(F)c2)=O)CCCC2(CCN2C(c2ccoc2I)=O)C1 53272,c1(NC(C2CCN(C(C=CCN(C)CC)=O)C2C)=O)cc(C)cnc1O 53273,C1(CC)CC(C(=O)NC2CN(C(=O)Cc3cnc(CC)[nH]3)CC2C)CCO1 53274,CC#CCCC(=O)NC(CC1CCC1)C(=O)NCC(N1CCCCC1)C 53275,c1(C(=O)NC2CC(CNC(c3cnc(Cl)[nH]3)=O)C2)nnc2ccccc2n1 53276,N1(C(Cc2cc(C)[nH]n2)=O)CCCCC1CCNC(C1(CC(C)C)CCC1)=O 53277,Cc1cc2c(CC(=O)NC3COCCC3NC(C3(C)CC=CCO3)=O)csc2s1 53278,N1(C(CC2N(C(c3c(C)nc(C)[nH]3)=O)CCC2)=O)CC=C(c2ccccc2)CC1 53279,C(=O)(C1=C(C)OCCC1)NC1C(NC(c2nc(OC)c(F)cn2)=O)CCC1 53280,c1(SC)cncc(NC(=O)C(c2ccccc2)NC(=O)CC2CCC(=O)CC2)c1 53281,Cc1ccnc2sc(-c3nc(CCN(C)C)nn3CCF)c(C)c12 53282,c1(COC)ccc(OC)cc1C(=O)NC1(CO)CN(C(=O)CC2CC2)C1 53283,Cc1nnc(O)c(C(=O)NCC2C3CCCC2N(C(=O)Cc2ccco2)C3)c1C 53284,N1(C(Cc2c(C)nc(C)s2)=O)C2CCC1CC(NC(c1ccc([N+](=O)[O-])s1)=O)C2 53285,c1(CC)ccc(C(=O)NCC(C)(C(C)C)NC(=O)C(c2cccnc2)C)cc1 53286,C1(C(=O)NCC(C)C(F)(F)F)CCC(C)(C)N(C(C2(C3CC3)CC2)=O)C1 53287,N1(C(C(COC)NC(=O)Cc2cccc(C)n2)=O)CCCCC1CC(N)=O 53288,Cc1cc(NC(C2CC(CCNC(c3[nH]ccc(=O)c3C)=O)C2)=O)ccc1F 53289,C1(NC(C(CC)N(C)C)=O)CCC12CCN(C(c1oc(SC)cc1C)=O)CC2 53290,N1(C(C2C(NC(c3ncc(OC)cn3)=O)C2)=O)CCCC2(COC2)C1 53291,N1(C(C(=O)NCC=C)Cc2ccccc2)CCOCC1(C)c1ccccc1 53292,C1(C(C)C)CN(C(=O)CN2CC=CC2)CC1C(=O)N(C1CCOC1)CCO 53293,c1(C(N2C(C#C)COCC2)C(=O)NCCOC)nn(C)c2c1CCC2 53294,C1(C(=O)Nc2nc(C)ncc2Br)(OC)CCN(C(C2CC2F)=O)CC1 53295,N1(C(C=CCC)=O)CCN(C(=O)CC2C(C(F)F)C2(C)C)C(C2CCCC2)C1 53296,C1(N(C(C(C)OCC2CCCO2)=O)CCO)CCN(C(=O)CCc2ccc[nH]2)C1 53297,C1(CC=C)(NC(c2cccnc2OCC)=O)CCN(C(c2[nH]ncc2C#N)=O)C1 53298,c1(CCCSCC)cn(CCCC(=O)NCc2ccsc2C(=O)O)nn1 53299,C(C(CC(=O)NCCSC)NC(=O)CC1CCC(C)(C)O1)OC 53300,N1(C(C(C)OCC2CCCCO2)=O)CC2CN(C(C3CCC4(C3)N=N4)=O)CC2C1 53301,C(=O)(CCC(C)N(C)C)NCC=CC(=O)NCC1(COC)CCCO1 53302,c1(CC(N2C(C)(COC)CCC2)=O)ccc2c(c1)CC(C)O2 53303,C(=O)(CCP(C)(C)=O)N1CCC(N(CC#C)C(c2nc(C)oc2C)=O)C1 53304,CC1CCC2(CC2)N(C(c2cc(NS(N)(=O)=O)ccc2Cl)=O)C1 53305,C(C(=O)N1CCN(C(C2CCCCN2CC(F)F)=O)CC1C)(C(C)(C)C)SC 53306,Cn1ccc(C(=O)NCCCCC2CCCN(C(C3(C)CC=CC3)=O)C2)cc1=O 53307,c1(C(C)(C(=O)NCC(CNC(=O)CCCC2CC2)CO)N(C)C)ccc(F)cc1 53308,N1(C(c2cc(N)c(Cl)cn2)=O)CCOC2CN(C(=O)CC3C=CCC3)CC12 53309,C(C(CC(F)(F)CNC(=O)CC1CCOC1C)OC)OC 53310,n1(CC=C)cc(C(=O)NCC2CC(NC(c3cc(CC)c(CC=C)s3)=O)C2)cn1 53311,N1(C(CCC2(C)CC2)C(=O)NCC2CC2)CCC(S(=O)(=O)C(F)F)CC1 53312,C1(CC(=O)N(CC(=O)NC(c2ccc(F)cn2)C)C(C)C)CC2C=CC1C2 53313,N1(C(c2cccc(C(N3C(CN)CCCC3)=O)c2)C)CC2ON=C(C(F)F)C2C1 53314,c1(C(=O)NCC2C(NC(c3cnc4[nH]cncc3-4)=O)C2)ccc(Cl)c(F)c1F 53315,N1(C(C=CCCC)=O)CC2CC(C(N3CCC(CO)C(C)C3)=O)C(C2)C1 53316,Cc1ccccc1C=CC(=O)NC1CC2(C1)CC2NC(C1CCC(=O)O1)=O 53317,N1(C(CC(CC)(C)C)=O)CC2CC(CNC(=O)C(C)(C)SC)CC1C2 53318,CCC(CC(=O)NC(C)(CNC(c1nc(C(F)(F)F)oc1C)=O)CO)C1CC1 53319,c1(CC)ccccc1NC(=O)C(c1cnn(CC(F)F)c1)N(C1CCC(C)C1)C 53320,C(=O)(C(O)CC(F)(F)F)NCCCOCCOCCC(=O)NCN1CCC1 53321,Cc1cc(OC(F)(F)F)c(CNc2ncccc2Br)cc1Cl 53322,C1CCC2(C1)COC(CNCC1(c3nnnn3C3CC3)CC3(CCC3)C1)C2 53323,CCC(CC)N(C(=O)COC(C1CC1C1CCCO1)=O)CC 53324,C1(C(N2CC(OCCOC)C2)=O)CCC(CNC(=O)CCCF)O1 53325,C1(C(N(CCC(CC)(F)F)C)=O)CCCN(C)C1c1ccnn1C(C)C 53326,N1(C(C2CNC(=O)N2)=O)CC(NC(c2ccoc2Br)=O)C2(CCC2)C1 53327,c1(CN2C(C(=O)NC3CC(O)C3)C(O)CC2)c(Br)ccc2c1OCO2 53328,C1(CC=C)(C(=O)NC2CCN(CCOC)C2)CCN(C(c2conc2CC)=O)C1 53329,N1(C(C2CC(NC(C(CC)n3ccnc3)=O)C(O)C2)=O)CC2CC2C2CC12 53330,c1(C(=O)NCCCN(C)C(c2cnc3ccoc3c2)=O)cncc(P(C)(C)=O)c1 53331,C(C1=NOC2CCCC12)NC(N1CC(OC(C2(CS(N)(=O)=O)COC2)=O)C1)=O 53332,C1(O)(CC(=O)NC2C(NC(=O)C(F)=C3CCCC3)C2)CCCOC1 53333,c1(N2CCN(C)CC2)cncc(C#N)n1.N12CCCC1C2=O.C1CCN1C(=O)CO 53334,c1(CNC(N2CC(C)(C#N)C2)=O)ccc(N=[N+]=[N-])cc1 53335,C1(CNC(c2ccc(OC(F)(F)F)c([N+](=O)[O-])c2)=O)CCC2COCCC2C1 53336,c1(C(N(CC(CC)NC(C2(CF)CCC2)=O)CC)=O)ncn2ccc(C)cc12 53337,CCC(C)CCC(O)CC(=O)N1CCCC1C1CCN(C(=O)CCCOCC)C1 53338,C1(CNC(C2C(C(N)=O)C2)=O)C2CC1N(C(C1CCCC1F)=O)C2 53339,c1(C(=O)NC2C(CNC(Cc3n(C)nc(CC)c3Cl)=O)C2)nc2c(s1)COCC2 53340,C1(CNC(=O)C2CC2)C2CN(C(C3CC(n4cncn4)C3)=O)CC12.O=C1CCN1 53341,c1(C(N2C(C)CN(C(=O)Cn3nnc(C(C)(C)C)n3)CC2)=O)cc2sccc2[nH]1 53342,CCC(C)(C)C(C)CC(=O)N1CCN(C(c2nocc2C(C)C)=O)CC1CO 53343,c1(C(=O)NCC(CNC(c2c(C)onc2O)=O)F)ccc(S(=O)(=O)C(F)F)cc1 53344,c1(CN2CCN(CC(=O)NC(c3ccc(CC)cc3)CC)CC2)cc(Br)ccc1Cl 53345,C(=O)(CC(N)C(C)(C)O)NCC(C(=O)OC)(C)O 53346,N#Cc1ccc(-c2cccc(C(=O)N(C3CCCC3)CCc3nn[nH]n3)c2)cn1 53347,c1(C2(CNC(c3cc(F)c[nH]3)=O)CC2)ocnc1-c1cn(CCO)nn1 53348,CC1(C#CC(=O)N2CCC(CC3COCCO3)CC2)CN(Cc2ccccc2)C1 53349,c1(C(=O)NC2CC(N(C)C(C3CCCCCC3)=O)C2)cc(F)c(F)c(Cl)c1F 53350,N1(C(C2(CC)CCNC2=O)=O)CCCN(C(=O)C2CC2)CC1 53351,n1(CC)ccnc1C=CC(N1CCOC(CCNC(C2CCS2(=O)=O)=O)C1)=O 53352,C(=O)(C(F)C1=CCCCC1)NC(C1CCCC1)CNC(c1c(CC)n[nH]c1)=O 53353,c1(C(C(=O)NC)N(CC(F)(F)F)CCCO)cc(C(C)(C)C)no1 53354,N1(C(C(C)SCC)=O)CCCC(C)(CNC(=O)CCc2cc(C)nc(C)c2)C1 53355,C1(NC(CCN(CCCO)C(C2(OC(C)=O)CC2)=O)=O)CCCC2(C1)N=N2 53356,C1(NC(C(C=C)C)=O)CCCCC1NC(=O)CCc1cc(C)no1 53357,c1(C(N2CCCC(C)(c3cn(C4CCCC4O)nn3)C2)=O)nc2c(s1)COCC2 53358,CC(C)CCC(F)C(=O)NC(CC1CCCC1)C(=O)NCC1CCC(=O)N1 53359,c1(C(=O)NC(CNC(C2(C)CC2Br)=O)CO)cncc2sccc12 53360,O=C(N=c1cc[nH]cc1F)C12CC1CN(C(=O)Nc1ccc(Cl)c([N+](=O)[O-])c1)C2 53361,N1(C(C(=O)NCCc2ccc(OC)cn2)=O)CCC(C)C(C)C1 53362,c1(C(N(C)CC2CCCN2C(=O)C(F)CC2CC2)=O)c[nH]c2cccc(C#N)c12 53363,c1(CC(=O)NC2CC(C)(NC(C(C3CCC(=O)N3)C)=O)C2)csc(Br)c1 53364,C1(C(=O)NCC(CNC(C2C(c3n(C)ncc3)OCC2)=O)O)CC2(C1)CC(O)C2 53365,C(C(C)(O)CC(=O)N1CCN(C)CC1CNC(c1cc(C2CC2)n(C)n1)=O)OC 53366,CCCC(C)(C)CC(=O)N1CCC(NC(=O)C(C)(C)CC(C)C)C(C)C1 53367,c1(C(N2CCN(C)CC2CNC(c2ccnnc2O)=O)=O)cc2c(o1)CCCC2 53368,C1(NC(c2cc(N)sc2)=O)CC2(NC(c3cnc(C4CCOC4)s3)=O)COC1C2 53369,C(CC(C(C)C)NC(=O)Cc1csc(C)n1)NC(c1ccc(COC)o1)=O 53370,N1(C(C2CN(C(c3ccc(C)o3)=O)CC(C)C2)=O)CCC2(CC1)CC(O)C2 53371,c1(CC(=O)NC2C(C)N(C(=O)Cc3cnoc3)CCC2)ccc2c(c1)ncn2C 53372,N1(C(C(C2CCN(C(CS(CC)=O)=O)CC2)C)=O)CCc2nn[nH]c2C1 53373,c1(C(C)(C)C)cccc(CC(N2CC(F)CC2C(N2CCOC(CO)C2)=O)=O)n1 53374,N1(C(c2c(CC)nc(C)o2)=O)CC(NC(=O)C(C(C)C)C2CCC2)CC(F)C1 53375,c1(C(=O)NC2CC3(C2)CC3(F)F)n[nH]c2c1CN(C(=O)CN1CCCC1)C2 53376,c1(CNC(CN(C(CCCOCC=C)=O)CC)=O)cc(Cl)ccn1 53377,c1(C(C(=O)NCCCN(C(C23CCC(CC2)O3)=O)CC)=O)cc(F)cc(Cl)c1 53378,N1(C(Cc2ccn(CC)n2)=O)CCC(NC(=O)Cc2cc(C3CC3)on2)C12CC2 53379,C1(NC(C(CSC)O)=O)CCCC(C(=O)N(C2C3CCCC23)C)CC1 53380,N1(C(C(C)(Cl)Cl)=O)CCC(CCC(=O)NC2(CCF)CC2)CC1 53381,c1(OC)ccc(CC(=O)NC(C)(C)CNC(c2cc(CN(C)C)on2)=O)c(C)c1 53382,c1(C(=O)NC(CC)(C)CNC(C2CC2(C)C(F)F)=O)ccc(F)cc1OC 53383,C1(C(=O)NCCC(CCC)O)CCCCN(C(c2cnn(C)c2OC)=O)C1 53384,C=CC(C)C(=O)N(CCC(=O)N(C1CCC1)CCO)C 53385,C1(C(=O)NCc2cn(C3CCN(C(CC)=O)CC3)nn2)CCS(=O)(=O)C1(C)C 53386,N1(C(C(C)(C)CC2CC2)=O)CCC2(CCN(C(c3csc(CO)n3)=O)C2)C1 53387,Cn1ncc(NC(C23CC(CN2C(C2CCCC(F)C2)=O)C3)=O)c1C(N)=O 53388,Fc1cncc(ONC(N2CCN(c3ccccc3)CC2)OC2CCNCC2)c1 53389,C(N=c1[nH]c(=NC2CCOCC2)[nH]c2c1CCC2)C1(S(C)(=O)=O)CC1C(F)(F)F 53390,C1(C(=O)NCC(CC)(CC)CO)CN(C(c2ncn3ccccc23)=O)CC(C)O1 53391,C1(C(N(CCCNC(=O)C(C2CC(F)(F)C2)OC)CCC)=O)CC2CC(=O)C1O2 53392,C1(NC(c2n(C(C)C)ncc2)=O)(CO)CCCN(Cc2ccc(Br)s2)C1 53393,C(=O)(C(C)P(C)(C)=O)C(C(n1cc(Br)cn1)NCc1c(C(=O)OCC)occ1)=O 53394,C1(C)(CC(=O)NCc2snc(C)n2)CCN(C(c2sccc2F)=O)C1 53395,N1(C(C(C)c2cccs2)=O)CCOCC1CNC(c1cc(-c2ccco2)no1)=O 53396,C=CC1(C(N2CCC(CC)(CO)CC2)=O)CCN(C(=O)C(C)CC=C)C1 53397,c1(-c2ccc(C(=O)NC3C(N)CC3)s2)cc(OC(F)(F)F)cc(F)c1 53398,n1(CC)nc(C(N2CC(O)CC2C(=O)NC(C23CCC(CC2)C3)C)=O)c(C)n1 53399,CC(C)CC(O)C(=O)NC1CCCC(CC(=O)N(CCCCCO)C)C1 53400,c1(OC)ncnc(N2CCOC(C(C)NC(c3cnccn3)=O)C2)c1OC 53401,N1(C(c2nccc(OC)c2)=O)CC2CCN(C(=O)CS(N)(=O)=O)C(C2)C1 53402,C(=O)(C(C)(C)S(C)(=O)=O)NCC1C(C)CCN1C(=O)Cn1ccc(C(F)F)n1 53403,N1(C(=O)NC(C(C(C)C)C)CN2CCCS2(=O)=O)c2ccc(Cl)cc2OCC1C 53404,N1(C(C2(CCC=C)CN(C(c3cccc(C)c3O)=O)C2)=O)CC2CCCC2C1 53405,C12(C(=O)NCC3(NC(c4cocn4)=O)CCCC3)COCC1CS(=O)(=O)C2 53406,C=CC(CCC)CC(=O)N(C)CC1CN(C(c2ccccc2)=O)CCO1 53407,CC1(NC(c2cc(CNS(C)(=O)=O)cs2)=O)CCN(C(=O)CCC2CCOCC2)C1 53408,C=CCC(C)(CC)C(=O)N1CCC(NC(c2ccnc(C(F)(F)F)n2)=O)CC1 53409,C1(C#N)(C(N2CC(NC(c3ccc(OC)s3)=O)C(C)C2)=O)CCSCC1 53410,c1(C(N2CC(CCCNC(=O)C=CC3CC3)OCC2)=O)cccc2[nH]cc(Cl)c12 53411,C=CCC(C)(C)CC(=O)NC(CCF)C(=O)NC(CO)CC#CC 53412,C1(C(N2CC(N(C)C)C2)=O)CC1C1CN(C(=O)CCC2CCCCO2)C1 53413,c1(C(=O)NC(CCCC)CNC(C2(F)CCOC2)=O)cc2c(C)cc(C)nc2s1 53414,N1(C(C(C)(C)C)=O)CC(NC(=O)CCc2nc3ccccc3s2)C(C2CC2)C1 53415,N1(C(C(C)N=[N+]=[N-])=O)CC2COCC2(C(N2CCSC(C)C2)=O)C1 53416,C(=O)(C1OCCc2ccccc21)NCC(CN(C(c1c(COC)nn[nH]1)=O)C)O 53417,CC1(C)CC(COC(c2ccc(F)c(CO)c2)=O)OC1=O 53418,C#CC1(C(=O)Nc2ccc(SC)cc2)CCN(C(=O)CSc2nncn2C)CC1 53419,N1(C(CN(C2CC2)CC)=O)CC=CC(NC(c2cccc(C(C)(C)C)n2)=O)C1 53420,CCCCCCC(CNC(c1nc(C)c(C)nc1C)c1nnnn1C)CC 53421,CN1CCN(C(=O)CCc2nccs2)C(C(=O)NC2C3CCC(F)(F)C23)C1 53422,c1(N2CCC(NC(c3c(C)ncs3)=O)C2)cc(-c2ccc(Cl)cc2)ncn1 53423,c1(C(N2C(CNC(=O)CC3(O)CCC3)CC2)=O)n[nH]c2c1CC1CC21 53424,C1(NC(C2C(=C)C2C(=O)OC)=O)CN(C(=O)COCCN(C)C)CC2CCCC12 53425,c1(-c2ccc(C(=O)Nc3ccc(C(=O)OC)cn3)nc2)cc2cc[nH]c2cc1F 53426,N1(C(CC(C=C)C)=O)CC2(CC(NC(c3c(C)cc(C)nc3S)=O)CO2)C1 53427,c1(CNC(c2nnc(C)n2C)c2n(CCOC)nnn2)cccc(Br)c1 53428,C(=O)(C(CCC(C)C)NC(=O)CC(C)C(C)C)NC(C(=O)NC)CC(C)C 53429,C1(NC(C=C(COC)C)=O)CCCC12CN(C(=O)C=Cc1ccccc1F)C2 53430,Cc1cncc(C(=O)C(=O)NC2C=CCN(C(c3sccc3C(C)C)=O)C2)c1 53431,C(C(C(F)(F)F)N1CCOCC1)NC(=O)CCCn1cc(-c2cccs2)nn1 53432,N1(C(C2C3CN(C)CC32)=O)CCC(C(N2CCC(F)(F)CC2)=O)C(C)(C)C1 53433,c1(C(N2CC(Cn3cc(CN(S(C)(=O)=O)C)nn3)C2)=O)cc(Br)sc1Cl 53434,Cc1cccc(C)c1NCC(N1CCCN(C(C2CCC(C)O2)=O)CC1)=O 53435,NC1CN(C(=O)C(=O)NCC2(C(c3ccc(F)cc3)=O)CC2)CCc2ccccc21 53436,C1(C(=O)NC2CCN(C(CCCC)=O)C23CC3)CCn2nccc2C1 53437,C1(C(=O)NCC2CN(C(C3CCC(C)S3)=O)C2)(OC)CCC(F)(F)CC1 53438,c1(C(=O)OCC(ONC(C(=O)OCC)=O)(C)C)csc(=NC2CC2)[nH]1 53439,c1(C(N(C(C)C)CCC2CCOC2C2CC2)=O)ccccc1OC(F)F 53440,CC(C)C#CC(=O)N1CCC(O)(C(C)NC(=O)C(C)(C)c2ccn(C)n2)C1 53441,C1(C(=O)NC(CCCNC(CC(CCC)C)=O)C)CCc2cnn(C)c2C1 53442,Cc1[nH]c2ccccc2c1C(N1CC(C)CN(C(=O)CCOC(C)C)C(C)C1)=O 53443,c1(C(=O)NCCCN(C(C2(n3nccn3)CC2)=O)CC)ccc[nH]1 53444,C(C(F)(F)C(=O)NC1CCC(NC(=O)C(c2cccc(Cl)c2)C)C1)OC 53445,CN=c1[nH]nc(CC(=O)NCC2(O)CCN(C(=O)Cn3ccccc3=O)C2)s1 53446,C1(C(=O)NC2(CC=C)CCCC2)CC(C)CCN1C(=O)CCCN(C)C 53447,N1(C(c2c(C)n(C3CC3)cc2)=O)CCN(C(=O)C(C)OCCN(C)C)CCC1C 53448,c1(CN2C(CNC(=O)C=CCN3CCCCC3)CSCC2)c(Cl)ccc(F)c1F 53449,C(=O)(C(C)(C)S(=O)(=O)C1CC1)C(c1cccc(C)c1)=O.CC(=O)N(C)CCNC 53450,N1(C(C2C(C#N)C2)=O)CC2CC2(CNC(c2cn(CCO)nn2)=O)C1 53451,N1(C(Cc2c(C)ocn2)=O)CCC2CCC(NC(c3c(Br)nnn3C)=O)C12 53452,C(c1ccc(N)c(N)c1)=CC(=O)NC1(CNC(c2cccc(CC)n2)=O)CC1 53453,n1(CC)nc(C(=O)NCC(C)(CO)NC(C2CCN(C)C2=O)=O)cc1C 53454,c1(CC)nn(C)c(C(=O)NC(C)C(CO)NC(C2CCCS2)=O)c1Cl 53455,N1(C(=O)C(O)C(F)F)CCC2(CCCN2C(c2ccc(N3CCCC3)nc2)=O)C1 53456,c1(C(N2CCC(CN(C)C(c3csn3C3CC3)=O)C2)=O)cc2c(s1)CCC2 53457,N1(C(CSC(C)(C)C)=O)CC(C(C)(C)O)(CNC(=O)Cc2cc[nH]c2)C1 53458,c1(C(=O)NC(C)CCNC(=O)CC2CN(C)C2)n[nH]c2ccccc12 53459,C1(O)(C(=O)NC2CN(C(C(COCC)N=[N+]=[N-])=O)CC2C)CCCC(C)CC1 53460,C1(O)(CNC(C=CCC)=O)CCN(C(=O)CCC2CCOCC2)C1 53461,N1(C(CC(CC)CC)=O)C(C)CC2CN(C(=O)Cn3ncc(Br)n3)CC12 53462,CC#CCC(C(=O)NCC1CC1(F)F)NC(c1c[nH]c(C)c1)=O 53463,C1(C(=O)NCC(N2CCC(NC(c3cscc3Cl)=O)C2)=O)CCC(F)CC1 53464,c1(C(=O)NC2CCN(C(=O)C3=CCCC3)C(C3CC3)C2)ccn2cccc2c1 53465,N1(C(c2c(CC)ccs2)=O)CC2CCC(CNC(c3cncnc3CC)=O)(C2)C1 53466,c1(CC(=O)NC2CC(C)(NC(COCC=C)=O)C2)c(CSC)oc2ccccc12 53467,N1(C(C(C)C2CCC2)=O)CCc2sccc2C1CNC(=O)CC(C)(C)CC(F)F 53468,N1(C(C(=Cc2cccs2)C)=O)CC2CCOCC2(NC(C2SCCCS2)=O)C1 53469,CC(C)CS(=O)(=O)CC(=O)NCCCc1cn(-c2cnc3nc(O)nc-3[nH]2)nn1 53470,C(=O)(C(CCCCC(=O)OC)N(CCc1cccc(F)c1)CCN(C)CC)NCC 53471,Cc1ncc2c(n1)CCC(C(=O)NC1CN(C(=O)C#CC3(C)COC3)CC1C)C2 53472,N1(C(C2CCOC2)=O)CC2OCCN(C(c3cc(C4CCOCC4)[nH]n3)=O)C2C1 53473,C(=O)(CCN1CCC1)NC(C)CC1CN(C(=O)C(C)OOC2CCCC2)C1 53474,c1(CC)nocc1C(=O)NCCN(C(=O)C(C)COC)C 53475,C(=O)(CC(C)(O)CCC)NC1C(C)CCN(C(C(C=C)c2ccccc2)=O)C1 53476,c1(C(=O)Nc2ccc(OC3CCNCC3)cc2)cccnc1N1CCOCC1 53477,N1(C(c2cn(C3CC3)nn2)=O)CCCCC(C2CN(C(C3CCSC3)=O)C2)C1 53478,N1(C(CCCC=C)=O)CCC(CO)C(NC(c2ccc(Br)c(C)c2)=O)C1 53479,c1(C(=O)NC2CC(F)(CNC(C(CC=C)CC)=O)C2)cc2nn[nH]c2cc1F 53480,c1(C(=O)Nc2cc(Cl)cc(Cl)n2)ccc2c(c1)CCN(c1ncccn1)C2 53481,c1(NC(C(c2cccs2)N(CCSC)CC)=O)nc(O)c2c[nH]nc2n1 53482,N1(CCNc2ncc(-c3ccc(Br)cc3)o2)CCC2CCCC(C1)N2 53483,c1(OCC(N2C(C)CC(NC(=O)CC(C)(C)C)C2)=O)nc(O)nc(O)n1 53484,c1(CC)[nH]nc(Cl)c1C(=O)NC1CC2C(NC(c3ncsc3C)=O)C2C1 53485,N1(C(C)=O)CCCCC1C(=O)NC1(C)CC(NC(C2CCNC2=O)=O)C1 53486,Cc1cc(C(N2CCC(N(C(=O)Cc3cnns3)C)C(C)C2)=O)cc2c1CCC2 53487,C(=O)(CCN=C(NC(C)C)NCc1cncc(C(C)(C)C)c1)NCCC 53488,c1(C(=O)NC(CNC(C=C(CCC)C)=O)CO)ccc(CCC)c(Cl)c1 53489,c1(C(=O)OC)c(OC)ccc(S(=O)(=O)N2CCN(C=O)CC2)c1OCOC 53490,c1(N(CC(C)C(=O)N2CCCCC2)Cc2cccs2)ncnc2ccc(Cl)cc12 53491,C#Cc1cc(F)c(C(=O)NC2CCN(C(C3CCC(C)(C)CC3)=O)C2)c(F)c1 53492,c1(C(=O)NC2C(NC(C(C)(C)OC)=O)CCCC2)ncc(Br)cc1N 53493,Cc1ccc(-c2cc(C(=O)NC3CC(C)(NC(=O)CN(C)S(N)(=O)=O)C3)n[nH]2)s1 53494,CCCC(C#N)C(=O)N1CC(C)(C)CC1C(=O)NCCc1n[nH]c(CC)n1 53495,c1(OC)cc(NC(C2C3CC2N(Cc2cc(Cl)ccc2I)C3)=O)ccc1C 53496,c1(C(=O)NCC2CCCN2C(=O)CSc2nc[nH]n2)cccc(-c2nccs2)c1 53497,c1(C(=O)NCC(C2CCCC2)N(C(=O)CC(C)(C)O)C)cc(Cl)cc(Cl)c1 53498,N1(C(CCCN(C(C)=O)C)=O)CCC(C)(C)C1C(=O)N(C1CC(O)C1)C 53499,C1(N(C(=O)CC2CSC2)CC)CCN(C(=O)C(C2CCOCC2)F)CC1 53500,C(CC(CC)C(=O)NC1CC(C)(NC(=O)C(CC)C(=O)OCC)C1)=CC 53501,c1(NC(CN(C(=O)CN2C(C)CCC2C)CCC)=O)ccc(F)c(O)c1 53502,C(=O)(CCCCCCC(=O)N1CCN(Cc2c(O)cccc2Br)C2CC12)OC 53503,Cc1cc(C(=O)NC2(CNC(=O)C(O)CCN(C)C)CC2)cc(S(N)(=O)=O)c1C 53504,C(=O)(C(C(C)C)NC(=O)C(C1CCCCC1)C)NCC#CCC 53505,N1(CC(=O)NCCCN(CCCCNC(=O)C(O)C2CCCC2)C)CC(=O)N1 53506,Cc1nc(=O)c2c(C)c(C(=O)N(CCC(C)NC(=O)CN3CC(C)C3)C)sc2[nH]1 53507,C1(CCOC)(C(=O)Nc2cncnc2C)CCN(C(=O)C(C(C)C)SC)C1 53508,C(=O)(CS(=O)c1ccc(Cl)cc1)NCC(C1CC1)NC(=O)Cc1cnsc1 53509,Cc1oc(C#N)cc1C(N1CCCC(C(=O)NC2(CC(N)=O)CCC2)C1)=O 53510,c1(-n2c(C)ncc2)ccc(C(=O)NCC2CCCC2NC(=O)CC(C)C)cc1 53511,C(=O)(N=c1[nH][nH]c2ncccc12)C1C(NC(c2cccc(C)c2)n2cncn2)C1 53512,C(N=c1[nH]c(=NCCCn2cnnc2)[nH]c2cc[nH]c12)c1cn(C)nc1C(F)F 53513,CC12CN(C(=O)CNC3CCC(O)C3)C(C(=O)O)(C1)C2c1ccccc1O 53514,c1(C(N2C(C(C)NC(=O)CC3OCCCO3)CCC2)=O)cncc(C2CC2)c1 53515,CC1(CNC(C2(F)CCCC2)=O)CCCN1C(C1CCCCO1)=O 53516,CS(=O)CCC(=O)NCC1(NC(=O)CCNC(c2ccoc2)=O)CC1 53517,N1(C(CC=CCC)=O)CCN(c2ncncc2C)CC1C 53518,C1(C(=O)NC2CCSCC2)(NC(C2C(C)(C(F)F)C2)=O)CC1(C)C 53519,C(=O)(C1CCCc2scnc21)NC1CCC(CNC(c2coc(Br)c2)=O)C1 53520,C(=O)(CC(C)C(C)C)N(C(C(=O)NCCc1c(C)noc1C)(C)C1CC1)C 53521,C(=O)(CC(F)(F)C(F)F)N(CC(CC)NC(c1cc(Br)n[nH]1)=O)CC 53522,C1(NC(C(C2CC2)SC)=O)CCC(CC(=O)NC(CO)CCO)C1 53523,N1(C(CC=CCC)=O)CC(NC(c2cc3n(n2)CCC3)=O)C(C#N)C1 53524,c1(C(=O)NC2CN(C(C(C)(C)c3ccc(Cl)s3)=O)CC2F)ncc(F)cc1F 53525,C1(NC(Cc2c(C)con2)=O)CCCCC1NC(=O)C(C)(C)c1ccn(C)n1 53526,N1(C(c2scc(OC)c2)=O)CCCCC1CNC(=O)C1=CCSC1 53527,N1(C(Cc2nc(C)[nH]n2)=O)CCC2(CC1)CN(C(=O)C(C)(O)Cl)C2 53528,c1(C(=O)NC2CCC(C)N(C(=O)CCc3cncs3)C2)ccc2c(ccn2C)c1 53529,c1(C(N(C2CCCC(NC(c3ccc(C)s3)=O)C2)C)=O)cc(C)c(C#N)cn1 53530,c1(C(C(=O)NCCSCC(=O)NCC(C)Cc2ccco2)O)cccnc1 53531,C(=O)(C#CC1CCCCC1)NCC(C1CCCC1)NC(C1C(C)OCCC1)=O 53532,N1(C(C(C)Cc2ccco2)=O)CC(C(N2CCS(=O)CC2)=O)CC(F)(F)C1 53533,N1(C(c2n[nH]c(CC)c2Cl)=O)CC2(CCCC(CNC(c3oncc3C)=O)O2)C1 53534,C1(CNC(C=Cc2cc(OC)ns2)=O)CC2CC(C1)N(C(=O)CC(C)C)C2 53535,C1(CC)CN(C(=O)C(C)(C)C)CCN1C(=O)CN(CCC(C)C)S(C)(=O)=O 53536,N1(C(CC(C=C)C)=O)CC2(C1)CN(C(c1[nH]nnc1C)=O)CC2CO.C1(CO)CC1 53537,CC(C)CC(C)(CNC(=O)CCc1cnc(O)[nH]1)NC(c1cnn(C2CC2)c1)=O 53538,c1(C(=O)NC(C(=O)OC)Cc2cn(C)cn2)cnn2c(Br)cccc12 53539,C(=O)(C(C)C(O)CCCC)NCCCCCC(=O)N(C1(CCC#C)CC1)C 53540,N1(C(c2cc(Cl)cc(Br)c2F)=O)CCCC2(CCCO2)C1 53541,Cc1cc(N(C)C)ccc1CN1CCCC(OC(=O)N(C)C)C1 53542,C1(NC(c2c(C)sc(O)n2)=O)CCN(C(=O)C(C)Cc2ccco2)C(C2CC2)C1 53543,c1(CN(c2ccnc(CC3CCCO3)n2)C(C)C)cc(Cl)ccc1Cl 53544,Cn1cncc(C(=O)NC2COCCN(C(c3cnn(C4CCC4)n3)=O)C2)c1=O 53545,N1(C(CC(C=C)C)=O)CC2CN(C(=O)CC(=O)OCCC(C)C)CCC12 53546,Cc1cc(NC(C2CC3CC3N2C(=O)C(C)OC(C)(C)C)=O)c(C)cc1Br 53547,CCCS(=O)(=O)C(C)C(=O)N(CCCNC(=O)Cc1c[nH]nc1O)C 53548,c1(OC)ccc2c(c1C(=O)N(CCNC(=O)C1=CCC(C)CC1)C1CC1)CCC2 53549,c1(C(N2CC(C)(NC(c3ccc(N(C)C)c(F)c3)=O)C2)=O)cc(F)cc(Cl)c1N 53550,N1(c2nccc(N3CC=C(C)C3)n2)CCCC2(CC=CCO2)C1 53551,c1(C(=O)NCCN(C(=O)CCn2ccnn2)C)ccc2cc(F)c(F)cc2n1 53552,C1(C(=O)NC(CCN(C(c2c(OCC)ccs2)=O)C)C)CCCC2(CCC2)O1 53553,C1(C(N2CC(C)C(C)(CO)C2)=O)CC(C)(C)OC1(C)C 53554,c1(C(=O)NCCC(C(=O)N2CC(O)(C(F)(F)F)C2)OC)ccc2nccn2c1 53555,c1(C(=O)NC2C(CC)N(C(=O)Cc3nc(=N)[nH][nH]3)CC2)cnn2c(C)cccc12 53556,c1(C(NNC(c2cccc(-n3cc(C(=O)O)nn3)n2)=O)=O)onc2c1CCCC2 53557,c1(C(=O)NC2CCC(C(C)NC(c3cnc(Cl)nc3)=O)CC2)ccc(I)cc1Cl 53558,C(=O)(CCCC(F)F)N(c1nnc(C(C)C)s1)Cc1ccc(-c2nn[nH]n2)cc1 53559,C(CCCCC(=O)O)N1CC(SC(C)(C)C)C1 53560,c1(C(=O)NC2(CC=C)CN(C(C3SCCC3C)=O)C2)ccn2ncc(C)c2n1 53561,C1(CC(=O)NCCNC(=O)NC)CN(C(=O)CC(C)(C)C)CCO1 53562,C1(C(=O)NCC(C)(C2CC2)NC(c2cocn2)=O)CC1[N+](=O)[O-] 53563,C1(C(=O)NCC(c2ccccn2)C)C2Cc3ccc(Cl)cc3C12 53564,C(=O)(C(F)(F)CC=C)N1CCC(C2C(NC(C3(OCC)CCC3)=O)CCO2)CC1 53565,N1(C(C2C(CC)C2)=O)CCCN(C(c2c(OC)cccc2C)=O)C(C)C1 53566,O(C1CCc2ccc(C(=O)O)cc21)C(c1cccc(C(C)(C)C)c1)=O 53567,N1(C(CC2(C)CC2(Cl)Cl)=O)CC2C3CCC(C2C1)N(C(=O)CN1CCCC1=O)C3 53568,N1(C(C=CC=CCC)=O)CC(N=[N+]=[N-])CC1C(=O)NC1CCC(CCO)CC1 53569,Cn1[nH]c(C2CCNCC2)nc1=NC(=O)NCc1nnc(CCO)s1 53570,C1(CNC(CC=CC(C)(C)C)=O)CC2CCC1N(C(=O)CSc1ccccc1)C2 53571,C1(OC)CC(NC(=O)Cn2ccc([N+](=O)[O-])n2)C12CCN(C(=O)C(F)=C(C)C)CC2 53572,c1(CNCC(=O)NCCCOC=C)ccc([N+](=O)[O-])o1 53573,C1(NC(C=C(C)C)=O)CCOC(CNC(c2ccc(F)cc2)=O)C1 53574,C(CCCC(C)(C)C(=O)NNC(=O)C(C)(C)O)NC(CCC(=O)NS(C)(=O)=O)=O 53575,CCC(CC(=O)N(C)CC=CC(=O)N(C1CCOC(C)(C)C1)C)C(C)(C)C 53576,N1(C(C2C(C)N(C)CC2)=O)CCCC(C)(NC(=O)CCc2ccc(Cl)nc2)C1 53577,Nc1c(C(N2CCC(NC(C3CC3(F)Cl)=O)CC2)=O)ccc(F)c1F 53578,C(C(O)C(=O)N(C)CC1CCCN1C(c1cc(C(C)(C)C)on1)=O)SC 53579,N1(C(CC2(OC)CC2)=O)CCC(C2CC2C(=O)NC2CC2CC(C)(C)C)CC1 53580,N1(C(Cc2c(SC)cccc2)=O)CC(C)CN(C(=O)C=C(C)C)C(C)C1 53581,C1(CNC(c2ncn(CC)c2)=O)CN(C(=O)CCc2cncnc2)CC1C 53582,c1(C(c2nnnn2C2COC2)NCC(CCC)C)cc(S(N)(=O)=O)ccc1F 53583,c1(C(N(C(C)CC2CC2)C)=O)cc(CNC(C2(C3CC3)CCC2)=O)ccn1 53584,C1(NC(CC(=C)Br)=O)CCC(C)N(C(=O)CCC=CC)C1 53585,N1(C(c2n(CCC)ccc2)=O)CC(C(=O)NC2(C(=O)NC)CC2)CC(C)C1 53586,C1(CNC(CC(OC)OC)=O)CCCN(Cc2ccnn2C)C1 53587,C(=O)(C1=CCCOCC1)N1CC(O)(CN(C(C=CC(=O)OCCCC)=O)CC)C1 53588,C1(C)(CC)CC(C(N2CCCC2(C)CNC(=O)C(C)(C)C2(O)CCC2)=O)CCO1 53589,C(C(CCCC)NC(=O)C=CBr)NC(CC=CCC)=O 53590,S(=O)(=O)(CC(=O)NC1(C)CN(C(=O)C(C)(C)N2CCCC2)C1)N(C)C 53591,c12cnn3c1CN(CC3)C2=O.CN.CC1(O)CCN(c2ccnc(C(=O)O)n2)C1 53592,N1(C(C2C(OCC)C2C)=O)CC2(CCN(C(C3CC4(C)CC3CO4)=O)C2)C1 53593,CCCCC(C(=O)NCCC1(C(C)(C)O)CC1)N(C)C.C12(CC1)C(=O)NC2 53594,Cc1cc(C(=O)NC2CC(NC(=O)C(C)Sc3ccc(Cl)cc3)C2)c(C)s1 53595,C(=O)(C(F)C(=O)NC(C)CCCCNC(=O)C(C)(C)C1CCCC1OC)OCC 53596,c1(C(=O)NC(CC)CNC(c2c[nH]c(=N)o2)=O)sc2cccc(F)c2c1Cl 53597,c1(NC(N2CCN(c3cncs3)CC2)=O)nc2ccccc2[nH]1 53598,N1(C(Cc2nc(C)[nH]n2)=O)CCC2(CNC(c3ccccc3F)=O)CCCCC12 53599,Cc1ccc2ccnc(NCc3nc(C(=O)O)c(C)s3)c2c1 53600,N1(C(C(C)C#N)=O)CCCC(F)(C(=O)N(C)Cc2ccccc2)C1 53601,c1(CC(N2CCCC(N(C(=O)Cn3cccn3)C)CC2)=O)ccc2c[nH]nc2c1 53602,N1(C(N(C(CC)C)CC)=O)CCC(CO)C1CO 53603,C(=O)(C(O)C1=CCCCC1)N(C1(C(=O)NCCC(CCCCC)O)CC1)C 53604,C1(C(N2CCC(N(C(=O)CCC(F)(F)F)CC)C2)=O)CCC(=O)C(C)C1(C)C 53605,c1(C(=O)NCC(C)N(C(C(C)n2ccnc2)=O)C)cc(S(N)(=O)=O)sc1Cl 53606,C12(C(N(C3CCC3)C)=O)CCCC(CN1C(=O)C(O)CN1CCCC1)C2 53607,C1(CC)CCCCCN1C(=O)CC1CCCCN1C(c1cccn1CC)=O 53608,N1(C(C=COCC)=O)CCCC2(CCN(C(=O)C(C)CCC(C)(C)C)CC2)C1 53609,C1(NC(c2ccc(F)cc2O)=O)C2COCC1CC(NC(C1CCCCS1)=O)C2 53610,c1(CN)cccc(C)c1C.C12(CSC)CCC1Cn1c2nnn1.c1ccccc1 53611,C1(NC(CC2(C=C)CCC2)=O)(CO)CCN(C(C2CN(CC)CCO2)=O)CC1 53612,N1(C(C(CC2CCCC2)OC)=O)C2CCC1CC(CNC(C1(CO)CCC1)=O)C2 53613,C1(CCNC(C2(C)CC(=C)C2)=O)CCCN(C(c2cc(CCC)[nH]n2)=O)C1 53614,N(C(=NCCN(C)C)NCc1ncccc1C(N)=O)CC(C)(C)OCC 53615,N1(C(c2cc(C)n(C)n2)=O)CCCN(CCNC(C2CC2CF)=O)CC1 53616,CC1(CCCC(=O)NCC2(O)CCN(C(=O)Cc3ccco3)C2)NC(=O)NC1=O 53617,c1(CC2C(C(=O)OC)CN(C(=O)CSc3ccncc3)C2)cccc([N+](=O)[O-])c1 53618,C12(C(N3CC(NC(CCc4ccc(C(C)C)cc4)=O)C3)=O)CC(C)(C1)OC2(C)C 53619,c1(N2CCCC(NC(c3n(CCC)ccc3)=O)C2)ncnc2sc([N+](=O)[O-])cc12 53620,C1(NC(c2c(N)ccc(Cl)c2)=O)CCC12CCN(C(C1CC3(C1)CC3F)=O)CC2 53621,C(=O)(C(F)CC(CC)CC)NC1(C(=O)NCCC=CCCC)CC(F)C1 53622,N1(C(C(C)Sc2ccc(OC)cc2)=O)CC2CC(C)N(C(=O)C=CC(C)C)C2C1 53623,N1(CCCNC(=O)NC(C(=O)OC)C)CCN(S(=O)(=O)Cc2ccccc2)CC1 53624,c1(CCC)cc(C(=O)NCCNC(=O)C(C)NC(=O)OC)no1 53625,C1(CN(C(=O)CC2(CC(=O)OC)CC2)CC)CCCCN1C(=O)CC=C(C)C 53626,c1(C(=O)NC23CC2CN(C(=O)COCC2CCCO2)C3)ccc(OCF)c(F)c1 53627,CC1c2ccccc2CC1N(C(=O)C(=O)NC1CC(c2cccc(Cl)c2)C1)C 53628,Cc1cc(C)c(CC(N2CCC(NC(=O)C(F)(F)C(C)O)CC2)=O)c(C)c1 53629,Cc1nncc(C(=O)NC2CC(c3cn(C4CCCC(C)C4)nn3)C2)c1C 53630,N1(C(CC(C)n2ccnc2)=O)CC(C(=O)N(C2CC3CCC2CC3)C)C2(CC2)C1 53631,c1(C(=O)NCC2OCCN(C(Cc3nc(C)oc3)=O)C2)cc2nccnc2[nH]1 53632,CCC(CC(=O)NCC(c1ccccc1)NC(C12CC(C)(CO1)C2)=O)C1CCC1 53633,C(=O)(C(C)CC(C)(C)C)N(CCCNC(C1CCC(C)C(C)C1)=O)CCO 53634,N1(C(c2cc3n(c2)CCSC3)=O)CCC2CN(C(=O)C3=CCOCC3)CC2C1 53635,c1(NC(=O)NCCn2cc(C3(C4CC4)CC3)nn2)cn2cc(F)ccc2n1 53636,C(C)(C(=O)N1CC(O)(C(C)NC(=O)C=Cc2cnc[nH]2)C1)(C1CC1)OC 53637,C(CC(CO)NC(=O)C(c1cnn(C)c1)NC(c1ncoc1C(C)C)=O)OC 53638,CC1(C)CC=CCN(C(C2(NC(C3CC3(C)C(F)F)=O)CCCC2)=O)C1 53639,C12(NC(c3cc(C)sc3C)=O)CCCC1CN(C(=O)CC1CC3CC3C1)C2 53640,C(N=c1ccnc(N2CC(CO)OC(C3CCCC3)C2)[nH]1)c1ccc(C#N)cc1 53641,C1(CCNC(=O)NOC2CC2)CCCCO1 53642,c1(C(C(=O)NCCCCCNC(=O)CSC(C)(C)C)N(C)C)ccccc1Cl 53643,Cc1cc(C(=O)NC2CC(C)CN(C(=O)CC3CCCO3)C2)nc(O)c1 53644,c1(OC)cccc2cc(C(c3nnnn3C)NCc3cnc(C)cc3C)oc12 53645,C1(C2CC2)(CNC(CC2CCC(C)(C)CO2)=O)CCN(C(=O)C(Cl)=CCl)C1 53646,C(C1=NOC2CCCC12)NC(C1OCCN(C(C2CCC(=C)CC2)=O)C1)=O 53647,C(=O)(CC(C)C(C)C)NC(C(=O)NCCCC(=O)NC)C1CC1 53648,CCC(C(=O)OC)C(=O)NC1CC(F)CN(C(c2[nH]ccc2COC)=O)C1 53649,C1(C(=O)NCC(C)NC(=O)CCc2ccn(C)c2)CCC2(CC1)NC(=O)NC2=O 53650,CC1(CNC(C2CC2C(C)NC(=O)CNC(C2CCC2)=O)=O)CC2(CC2)C1 53651,C1(NC(c2c(CC)occ2C)=O)CC(C2CCN(C(C3(O)CCOCC3)=O)C2)C1 53652,c1(OC)nccc(C(=O)NC(C)(C)CN(C)C(c2occc2Br)=O)n1 53653,N1(C(CN2CCN(C)CC2)=O)CCCC2C1CCN2C(c1csc(C2CC2)n1)=O 53654,n1(CC)cccc1C(=O)N(CC(=O)N(C1(CO)CC1)C)CC1CC1 53655,C1(C(N(C(CC(C)C)C(=O)NCCN2CCCC2=O)C)=O)CC(=O)CC12CCC2 53656,c1(NCC(=O)OCCCC)ccc(OC(=O)CC2CCC2=O)cc1 53657,C12COC3(C1)CN(C3)C2=O.c1(NC(C(N2CCC(C)C2)=O)=O)ccc(C#N)[nH]1 53658,C(=O)(C1=CC2C=CC1C2)NCC#CC(=O)NCc1c(O)ccc(C)n1 53659,C1(NC(C(C)n2ccnc2)=O)CCCC12CCN(C(C1CCC1)=O)CC2 53660,N1(C(C(C)OC2CCCC2)=O)CCOCC(CNC(C2(O)CC(C)(C)C2)=O)C1 53661,C(CCF)(C(=O)NCCC1CC(C)C1)NC(C1CC(OCC)C1)=O 53662,C1(C(=O)NCC(=C)C)C(C(F)(F)F)CCN1Cc1ccc(CC)nc1 53663,c1(CC)cc2c(CC(N3CC(NC(=O)COCC4CC4)C(O)C3)=O)csc2s1 53664,N1(C(CCC(N)=O)=O)CCC(C2(O)CCN(C(C3CC(=C4CCC4)C3)=O)C2)CC1 53665,C1(COCC)CCCN(CC(=O)NCCc2cccc(C)c2)C1.C1(C)C(=O)N1 53666,c1(C(=O)O)cc(Br)c(C(=O)NC2CC(CO)(CF)C2)cc1F 53667,c1(CC)ccc(C(=O)NC2CC2NC(C2(C3CCCO3)CCOCC2)=O)cc1N 53668,CCCC(C)CC(=O)N(C(C)(C(=O)NCC(C)(C)CCO)C1CC1)C 53669,N1(C(C2C3CC2N(Cc2ccc(N4CCCC4)[nH]2)C3)=O)CCC2(CCCO2)C1 53670,N1(Cc2n(C(C)C)ncc2)CC2CC1CN2C(C1CC1(F)F)=O 53671,C(CC(N)CC)NC(=O)NC(c1nc(CC2CCOC2)cs1)CC 53672,C1(NC(C2CCCC23CC3)=O)CCCN(C(=O)Cc2cscc2Br)CC1 53673,C(CCC(=O)NC1CCC(CNC(=O)C(F)=CC2CC2)C1)OCC 53674,c1(CC)ccc(C(=O)N(CCNC(c2ccc(C)o2)=O)CC2CC2)c(F)c1 53675,C1(COC)CCCN(C2=NCCC3N2CCCCO3)C1.N1(CC)CCCCC1 53676,CCC1=NOC(C(=O)NCCCCC(C)NC(c2cncnc2C(C)(C)C)=O)C1 53677,CCCN=C(NCCC(C)(C)O)NCc1cc(-c2ccco2)on1 53678,CC1CCN(C(=O)CC2CSCCO2)CCN1C(=O)CC1C=NN(C)C1=O 53679,C(C(=O)NNC(=O)CCCN)N(c1cccc(C(c2cccc(Cl)c2)(C)O)c1)C 53680,C1(C(=O)NCCC(CNC(c2cnc(CC)[nH]2)=O)O)CCC(F)(F)CO1 53681,N1(C(c2cnc(CCC)s2)=O)CCN(C(C2CCC(C)(F)CC2)=O)CC(C)(F)C1 53682,c1(C(=O)NCCC(CNC(C2C(=C)C2)=O)O)ccc(OC)c(S(=O)(=O)NCC)c1 53683,CCC(CC)C(F)C(=O)N1CC(C(=O)NC(C2CCC2)C)C2(CCC2)C1 53684,c1(C(=O)NCCNC(c2c(N)c(C(F)(F)F)ccc2)=O)cccc2c1COC2 53685,c1(C(=O)NCC2COCCN(C(C3CCCS3(=O)=O)=O)C2)ccnc2c1CCO2 53686,C1(CC=C)(NC(=O)CCC2CC2)CCCN(C(=O)CC(N2C(=O)CCC2=O)C)C1 53687,C1(C(N2CCC(C)C2)=O)C2C=CC3(CN(C(N4CCc5ccccc54)=O)C(=O)C13)O2 53688,c1(C(N2C(CN(C(C3(OC)CS(=O)(=O)C3)=O)C)COCC2)=O)ccc(O)nc1Cl 53689,C(c1cnn(C)c1)=CC(=O)NC1(CO)CN(C(c2c(OC)csc2)=O)C1 53690,c1(CC(C)C(=O)O)ccc(-c2cc(NC(C3CCOCC3)=O)ccn2)cc1 53691,C1(NC(CC2CC(=O)C2)=O)CN(C(C2CCCCC2(F)F)=O)CC12CCC2 53692,O=C1COC(CNC(C2CCN(C(=O)C(O)C3CCC3)CC2)=O)CN1 53693,c1(NC(CCNC(C(CC#C)C)=O)=O)cc(-c2ccc(OC)cc2)ccc1F 53694,c1(C(=O)NC)ccc(CC(=O)NCC(C)NC(c2cnn(C)c2C(C)C)=O)cc1 53695,N1(C(c2ccn(C(CC)CC)n2)=O)CC(CNC(=O)Cc2cc(OC)no2)C2CC12 53696,c1(CNCc2ccc(-c3ccc(OC)cc3)s2)n[nH]c2ccc(C)cc12 53697,C(=O)(CCCCNC(C)=O)NCCN(C(C(C)(C1CCOCC1)OC)=O)C1CC1 53698,C(c1ncco1)=CC(=O)NCC1CCN(C(c2ccoc2C2CC2)=O)C1 53699,CC(C)(C)C1=NOC(C(=O)NCCOCCNC(=O)C(F)CC2CCOC2)C1 53700,C1(OC)CN(C(=O)C(CO)c2ccccc2)CC1NC(=O)CCc1cn[nH]c1 53701,Cn1cc(C(N2CCC(CO)C(NC(=O)CC3CC4CC4C3)C2)=O)c2sccc12 53702,C1(CC(N)=O)(NC(c2c(C)cc(C)[nH]2)=O)CCN(C(c2sc(F)cc2C)=O)CC1 53703,C1(C(=O)NCC2=CCCCC2)C2CCN(C(c3ccsc3Cl)=O)CC12 53704,C1(CC)(NC(c2coc(CS(C)(=O)=O)n2)=O)CCCN(C(C2COC(=O)N2)=O)C1 53705,c1(NC)ccc(C(=O)Nc2c(CC(CC(=O)O)C(C)C)cccc2)cc1F 53706,C1(C(=O)NCCCCNC(C(CN(CC)CC)F)=O)CCC(C)CC1 53707,N1(C(c2cnn(C(CC)CC)c2C)=O)CCC(C)C(NC(c2csc(=N)[nH]2)=O)C1 53708,NS(=O)(=O)CCC(=O)NCCNC(C1CCCN(C(c2ccc(F)s2)=O)C1)=O 53709,c1(C(N2CC(O)(CNC(CC3C(C)C3)=O)C2)=O)cc2c([nH]1)CCCC2=O 53710,C=C=C(C)CC(=O)NC1C2CN(C(=O)CC3(CC(=O)OCC)CC3)CC12 53711,C#Cc1ccccc1CNC(C1CCN(C(=O)C(C)CC2CC2)CC1O)=O 53712,c1(C(=O)NCc2c(C(N(CC(CC)OC)C)=O)cco2)cncnc1C 53713,N1(C(Cc2c(C)ccnc2)=O)CCCC(C(=O)NCc2ncn(C)c2C)CC1 53714,c12ccncc1CNC2c1nnnn1-c1ccccc1.c1(CCC)cccn1C 53715,N1(C(C(C)N(CC)CC)=O)CCN(C(c2cc(C(C)=O)cn2C)=O)CC(O)C1 53716,Cc1nccc(C(=O)NCC2(F)CCN(C(c3ccc(N(C)C)cc3)=O)C2)n1 53717,N1(C(CN(C(=O)CCC(F)(F)F)CC)=O)CCCC(C)(N(C)C)C1 53718,C1(CC(N2CCC(N(C(c3c(C)cncc3)=O)CCO)C2)=O)CC2(CCNCC2)O1 53719,N1(C(C2(C)CCCC2)=O)CC2(CCCCN2C(=O)CCCCCF)C1 53720,C(CC(C(N)=O)NC(C1(NC(C2CC2(F)Cl)=O)CCOCC1)=O)OC 53721,N1(C(c2cn(C)nc2O)=O)C2CCC1CN(C(C1CCCC3(CC3)C1)=O)C2 53722,c1(CNC(C2CCCNC2=O)C)ncccc1Cl 53723,c1(C(=O)NCCCCCN(C)C(C2C=CCC2)=O)cnn2c1OCC(O)C2 53724,CCCCCC(F)C(=O)N(C(C)C(=O)NOCCCO)C 53725,Cc1nsc2ncc(C(=O)NCC3(F)CCN(C(=O)CCCC(C)(C)C)C3)cc12 53726,c1(C(N2CC3C(CNC(COCC(C)C)=O)C3C2)=O)nn(C)cc1S(C)(=O)=O 53727,C12(C(N3C(CNC(c4ccccn4)=O)C4CC4C3)=O)CCC(F)(CC1)CC2 53728,Cc1cc(C(=O)NCC2CCCC2NC(c2ccn(C)c2C)=O)cc(=O)n1C 53729,c1(C(=O)OCCC2CCC(NC(=O)OC(C)(C)C)C2)cc(Cl)c(Cl)cc1N 53730,C(=O)(C(C)(C)C(F)(F)F)NC1CCCN(C(C(C2CCCO2)OC)=O)CC1 53731,C1(C2CC2)(NC(CC(C)N(C)C)=O)CCN(C(c2coc3c2CCCC3)=O)C1 53732,CN1CCN(C(=O)Cc2cnns2)C(CNC(=O)CC2CCCCC2(C)C)C1 53733,C12(CNC(CCCOCC)=O)CC1CN(C(=O)C(C)Cc1ccccn1)C2 53734,C(N=c1[nH]c(=NCC#CC2CC2)c2c(F)cccc2[nH]1)c1nccc(CC)c1 53735,c1(N(CCCCCCCC)C)nc2c(c(=NC(C)c3ccco3)[nH]1)COCC2 53736,c1(C(N(C(CNC(C2(C)CCC(C)C2)=O)C2CC2)C)=O)occ2c1CCOC2 53737,CS(=O)(=O)c1nccc(N2CC(F)(F)CC2C(=O)Nc2ccc3sccc3c2)n1 53738,N1(C(=O)Nc2n(C)ncc2C2CCC2)CC2C3CCC(C(O)C3)C2C1 53739,C(CCC(C)C(=O)N(CCCN(C(=O)Cn1cnc([N+](=O)[O-])n1)C)C)OC 53740,c1(C(=O)NC)ccccc1NCc1cscc1Br 53741,C1(NC(C=CC)=O)CN(C(=O)C=CC2CCCCC2)C(C)(COC)C1 53742,C1(C(=O)OC)CC(C(=O)NCCCCNC(=O)C(C)(C)C2CC2)C1(C)C 53743,c1(OC)cc(F)cc(C(N2CCOCC(CNC(=O)C3=NOCC3)C2)=O)c1N 53744,c1(C(=O)NC23CCN(C(=O)Cn4cnnn4)CC2C3)c[nH]c2nccc-2c1 53745,c1(CC(=O)NC2(CCCC(=O)NCCC=C=C)CCC2)ccc(C)c(F)c1 53746,C(=O)(C(C)(C)C(C)O)NC1C(SC)CN(C(c2ccc(C(C)(C)C)cc2)=O)C1 53747,c1(C(C)OC)nc(C)c(C(N2CC(CNC(=O)C=C(Cl)Cl)C(O)C2)=O)s1 53748,CC(C(=O)NC1COCCC1NC(c1cn(C(F)F)cn1)=O)S(N)(=O)=O 53749,C1(C(N2CC3CCN(C(CC)=O)CCC3C2)=O)CC(c2cccc(Br)c2)=NO1 53750,C(=O)(C#CC1CCCO1)N(C)CC1(O)CCN(C(c2nn(CC)c(O)c2)=O)C1 53751,Cc1ccc(-c2csc(NC(CNC(C3(N(C)C)CC3)=O)CO)n2)cc1 53752,C(=O)(C(C)CC(C)(C)C)N1CC(CNC(CSSC)=O)C(C(F)(F)F)C1 53753,C=CCCCCCC(=O)N(C1CCCCN(C(=O)C(C)(C)OCCC)C1)C 53754,N1(C(C2(C)CCCC2O)=O)CC2(CC(CNC(c3cccn3C3CC3)=O)C2)C1 53755,C1(NC(C=C(CCC)C)=O)CC1C1CCCN(C(=O)Cc2ccccc2OC)C1 53756,N1(C(c2c(C)cco2)=O)CCC(C)C(NC(c2cncc(C(F)(F)F)n2)=O)C1 53757,c1(C(=O)OC(C)(C)C)c[nH]c(=NC2CCC3CC23)cn1 53758,C1(C(N(CCC(=O)NCC(C)(O)CO)CC)=O)CCCCC1F 53759,c1(C(=O)NC(CNC(CCC(C)(F)F)=O)C2CC2)cc(N)c(Cl)c(O)c1 53760,N1(C(C2ON=C(C)C2)=O)CCCC(C(N2CCCCC2CCCO)=O)C1 53761,C1(C(=O)Nc2nc(N(C)C)oc2)CN(C(=O)CCc2nncs2)CC12CCC2 53762,C=CCCCC(C)NC(C1C=CCCN1C(c1cc(C)oc1C)=O)=O 53763,c1(OC)cccc(S(=O)CC(=O)NCC(O)CNC(C2(COC)CCCC2)=O)c1 53764,NC(=O)CCN=c1ccn2ncc(S(=O)(=O)N3CCCC(C#N)C3)c2[nH]1 53765,c1(NC2C(C(=O)Nc3nc(Br)ccc3O)CCCC2)ncc2ccc(F)cc2n1 53766,C1(C(N(CC(=O)NC(C#C)CC2CC2)C)=O)CCCOC1 53767,C1(NC(C)=O)CCN(C(c2ccc(OCC(=O)OCCN(C)C)cc2)=O)C1C 53768,c1(C(=O)NC2CCC(CNC(C3ON=C(C)C3)=O)C2)ccc2c(c1)CC(C)O2 53769,N1(C(C(F)=C(C)C)=O)CCCCC1CN(C)C(c1nocc1C(C)(C)C)=O 53770,Cn1cc(C(=O)NCC(CNC(c2ncccc2N)=O)CO)c(C2CCCC2)n1 53771,C1(CNC(C(C)C)=O)(NC(=O)C=CC(C2CCCCC2)=O)CCCCC1 53772,c1(C(N2CCC(CC(C)NC(C3CC(F)C3)=O)CC2)=O)ccc(Cl)c(C#N)c1 53773,Cc1cc(C(=O)NC2CCOCC2C(=O)N(CCC(C)C)C2CC2)c(C)n1C 53774,Cc1nc(CC2CC2)sc1C(=O)NCC1CCCC(NC(c2c[nH]nc2F)=O)C1 53775,C1(NC(c2ccccc2F)=O)CN(C(c2ccc(C3CCOC3)s2)=O)CC1F 53776,C1(C(=O)NC(CN(C)C(C2(C(C)(F)F)CC2)=O)(C)C)CC12CCOCC2 53777,C(=O)(C1=CSCCO1)NC(CC(C(=O)N1CCCC1CO)OC)(C)C 53778,c1(C(N(C2CC(NC(C3CC3c3ccn(C)n3)=O)C2)C)=O)nccnc1N 53779,CC1CC(N(C(=O)C(F)C2CC(NC(c3c[nH][nH]c3=N)=O)C2)C)CCO1 53780,c1(C(=O)NC2CC(CNC(C(C)OC)=O)C(O)C2)ncc(Cl)cc1F 53781,C12(C(=O)OCCCONC(=O)OC(C)(C)C)CCCC1C2(F)F 53782,C(=O)(C1=COCCO1)NCC1N(C(c2cn(CC(CC)O)nn2)=O)CC=C1 53783,CC1(C)CCC(CNC(C2CC(C(=O)O)C2)=O)CC1 53784,C(=O)(CC(C(F)F)c1ccccc1)N(C(C)(C)C(F)F)CCO 53785,c1(C(N2C3CC(NC(=O)COCCF)CC2CC3)=O)ccc(F)c2[nH]ccc12 53786,C1(C(=O)NCCCN(C(=O)CCSCCOC2COC2)C)(OC)CCC(C)C1 53787,N1(C(c2c(CC)con2)=O)CC2(CCN2C(=O)CCN2CCC(F)C2)C1 53788,c1(C(=O)NCC(=O)NC2C(NC(C3(C#C)CCC3)=O)CC2)ccccc1F 53789,c1(CC)onc(C)c1C(=O)NCC1(F)CC(CNC(C2(C)CCCC2)=O)C1 53790,N1(C(C(C)(C)C)=O)CCC2(CC1)CC2C(N1CC2C(CO)CC2(C(F)(F)F)C1)=O 53791,N1(C(CC2(OC)CN(C(C3(C)COCCO3)=O)C2)=O)CC(C2=NOCC2)C1 53792,C1(C(N(C2CC(F)(F)C2)C)=O)CN(C(c2ccn(CCF)n2)=O)CC1(F)F 53793,C1(O)(CN(C)C(C2CC2(C)C)=O)CCN(C(C2(CC)CC2(F)F)=O)C1 53794,C1(n2cc(CNC)nn2)CCN(C(C23CCCC2CC3)=O)CC1 53795,C(=O)(C1CCCn2cncc21)NCC(C(C)C)NC(COC(C)C)=O 53796,CC(CC(C)(C)C)C(=O)N1CCC1CNC(c1ccncc1Br)=O 53797,Cc1ccnc(Cl)c1C(=O)NCC1CCCCC1NC(=O)CCC1CC1(F)F 53798,N1(C(CC2C(C)C2)=O)CCC2(CC1)CCN(C(C1CC13CC(C)(C)C3)=O)CC2 53799,c1(-c2cn(CCCCNC(C3CC(C(=O)OC)C3)=O)nn2)cc(F)ccc1Cl.C1CC1 53800,c1(C(N2CC(CNC(C(CCO)N(C)C)=O)C2)=O)ccn2ncccc12 53801,C(CCOC)(C(=O)NC1(CSC)CCC1)NC(C(C)OCC=C)=O 53802,C(=O)(C(CCC(C)C)NC(=O)C1=CC2C=CC1C2)NCc1c(CC)n[nH]c1 53803,CC(C)C(CCN(C)C(=O)Nc1ccc(-c2ccccn2)nc1)N(C)C 53804,Cc1cc(C(=O)NC2CC3C(NC(=O)Cc4sccc4Cl)C3C2)c(C)n1C 53805,c1(CC(C(=O)N(CCNC(C2(C(=O)NC)CCCO2)=O)CC)C)ccc(F)cc1 53806,Cc1ccc(S(=O)(=O)NCC2CCN(c3ccccc3)CC2C)cc1Cl 53807,C1(CNC(C(C)Cc2ccncc2)=O)CC2(CC2)CN1C(c1nccnc1N)=O 53808,CCC(CC)CC(=O)NC1CC2(C1)CC2NC(c1sc(F)cc1C)=O 53809,c1(C(=O)NC2CC3CN(C(CSCCCC)=O)C(C2)C3)cccc2nc(O)[nH]c12 53810,C(N=c1[nH]c2c(c(=NC3CC=CC3)[nH]1)CCC2)c1c(N)c2c(s1)CCCC2 53811,C1(NC(C=CC(C)(C)SC)=O)CN(C(=O)CCc2ncc[nH]2)CC1C(F)F 53812,C1(CN(C(=O)C(C)(C)c2nncn2C)C)CCN(C(c2cnoc2C2CC2)=O)C1 53813,Cc1ccc(C(=O)Nc2cn(C)c(C(=O)Nc3nc(Cl)nc(Cl)n3)n2)c(C)c1Br 53814,Cc1ccc(CCNC(=O)C(C)CNC(=O)C(n2ccnc2C)C)cc1 53815,c1(C(N2CC(CCNC(c3ncc(C(F)F)s3)=O)(OC)C2)=O)ncc(C)cn1 53816,c1(C(=O)NC2C(C=C)CN(C(=O)CCCn3cncn3)C2)cccc(S(C)=O)c1 53817,N1(C(COC)=O)CCC(NC(c2ccc(C(O)CF)cc2)=O)C(F)C1 53818,c1(C(N(CC(C)N(C(=O)Cc2cccc(F)c2F)C)C)=O)cc(F)ccc1F 53819,c1(C(=O)NC2CN(C(CC3C(=O)NCC(=O)N3)=O)CC2O)cc2cn[nH]c2cn1 53820,c1(N(CCCN(C(=O)CCC2CCC(C(N)=O)O2)C)C)ccc(S(N)(=O)=O)cc1Cl 53821,CC1(C)OC2(CO)CCC1(NC(c1ccc(F)c(O)c1)=O)CC2 53822,CC(O)C(C(=O)N1CCC(C)(NC(c2cnn(-c3cccnc3)c2)=O)C1)N(C)C 53823,c1(NC(C(CC2CC2)NC(C(CC2CCC2)OC)=O)=O)cnc(C)c(Cl)c1 53824,c1(CC(=O)NC2CCC(N3CCN(C(=O)COC)CC3)C2)cc(Cl)cc2c1OCC2 53825,C(CN=c1[nH]c2cccc(C)c2s1)(C1CCCC1)NC(C(C(CC)C)O)=O 53826,CS(=O)(=O)c1ccccc1C(N1CCCCC(NC(=O)C2=COCCC2)C1)=O 53827,C1(C(N2CCC(NC(=O)Cc3ccnnc3O)C2)=O)CC2(COC(=O)N2)C1 53828,C1(CNC(c2nc(CC)oc2)=O)CCCCC1NC(C1CC(=C2CCC2)C1)=O 53829,C1(OC)CN(C(c2cccc(F)c2)=O)C(C)(CNC(c2cccc(C)n2)=O)C1 53830,CN1C(=O)OCC12CN(C(=O)NCc1ccnc(OC3CCCC3)c1)C2 53831,CC(C)C(O)CCN=c1[nH]c2c(c(=NCC3CC(F)(F)CO3)[nH]1)SCC2 53832,N1(C(CCC(C)SC)=O)CC2CCCC2(NC(=O)Cc2ccn(C)n2)C1 53833,N1(CC)CCCC(C(N2CCCCC2CNC(=O)CCc2cn[nH]c2)=O)C1 53834,c1(NC2CN(C(c3c(C)[nH]nc3C(F)(F)F)=O)C2)cc(=O)n(C)cn1 53835,N1(C(C(C)NC(COC)=O)=O)CCC2CCN(C(=O)Cc3cncnc3)CC12 53836,c1(C(=O)NC(c2ccc(OC)cc2)c2nccn2C)coc2c1COC2 53837,C(=O)(CC(C(F)F)NC(c1c(C)n[nH]c1C)=O)NC1C(CC=C)CCC1 53838,N1(C(c2cccc(NCC)c2)=O)CCC(C2CC2)(CNC(C2C(C)C2C)=O)C1 53839,CC(C)CCC(=O)NCC(=O)NC1CC(CNC(c2ncn(C)n2)=O)C1 53840,C(=O)(CC(COC)NC(=O)C(C)n1cccc1)NCC1(COC)C(C=C)C1 53841,N1(C(C=CC(C)NC(=O)Cn2nccn2)=O)CCC(C2CCCC2)C1 53842,C(=O)(C(C)CCN(C)C)N1CC(CNC(CC(=O)OCC)=O)(OC)C1 53843,c1(CC)ccc(C(=O)NCC2(O)CC(CNC(=O)Cc3ncc(C)o3)C2)o1 53844,N1(C(c2cncc(C(C)C)c2)=O)CC(C)CCC1CNC(=O)Cc1cnnn1C 53845,C#CC1(C(N2CCC(CC(F)F)C2)=O)CCN(C(=O)C(C)c2ccsc2)CC1 53846,c1(COC)nc(C(=O)NC(C)CN(C(=O)C=C2CCC2)C)n[nH]1 53847,C1(C(=O)NCC(F)(F)C(F)F)(CC)CCCN(C(c2ccccc2O)=O)C1 53848,N1(C(CC=C=C)=O)CCC(CC(=O)NC2C=CCCC2)C1(C)C 53849,CCN(Cc1ccc(Br)cc1)N1CCN(CC(=O)NC2CCCCC2)CC1 53850,Cc1c(C(=O)N(C2CCCCN(C(C3CCCS3(=O)=O)=O)C2)C)cccc1F 53851,c1(C(=O)NCCCC2(NC(CC3C(C)CCC3)=O)CC2)c(F)cc(F)cc1Cl 53852,C1(CC)(CC)CC(O)CN1C(=O)C(C1CCN(C(c2cc(F)n(C)n2)=O)C1)F 53853,n12nnnc1C2(C1CC1)NCCOC1CCCCC1.c1(SCC)cc[nH]n1 53854,C1(CNC(C2(CC)CC2(F)F)=O)CN(C(=O)CCc2cccn2C)CCC1(C)C 53855,C1(N(C(C(CC#C)C2CC2)=O)C)CN(C(c2ccc(C(N)=O)cc2)=O)CC12CC2 53856,C1(NC(C2C(C)(CC)C2)=O)CCN(C(=O)Cc2ccc(F)cc2)CC1 53857,C1(CNC(c2nc(CC)sc2)=O)CC(NC(C2CC(N3CC(O)C3)C2)=O)C(O)C1 53858,C1(C)(C(N(C2CCC(C)CC2)C)=O)CCN(C(=O)CC2CCCC(=O)C2)CC1 53859,Cc1nc2cccc(C(C3CC3)NC(C(C)S(C)(=O)=O)c3ccccc3Cl)c2[nH]1 53860,CC1CCOC1C(=O)NCc1cn(C2CC(NC(=O)CO)C2)nn1 53861,N1(C(C(C)CC2CCC2)=O)CCCCCC1CNC(=O)CC(C)(C)CN(C)C 53862,N1(C(C2C(CC)C2)=O)CCCCC(CNC(c2csc(C3CCCO3)n2)=O)C1 53863,c1(CC)nccnc1C(=O)NCC(C)CC(=O)NC1CC2CCC1O2 53864,C(=O)(C1=CC2CCCCCC12)N1CCC(C(C)NC(c2ccc(C(C)=O)s2)=O)C1 53865,C(c1ccc(S(=O)(=O)NCC2CC2)cc1)=CC(=O)NC(C(CC)C)=O 53866,C=CCCC(C(=O)OC)NC(=O)C(C)CSC.C12(CCSC1)C(=O)N2 53867,C1(NC(=O)CSCC(N)=O)CCN(C(=O)CCOC(CC)C)CC1.C(COC)O 53868,Cc1nsc(C(N2CC(CNC(=O)CCCN(C)C)CC2C)=O)c1N 53869,O(C1CCSc2ccccc21)CC(C)(C)C1CCCO1 53870,N1(C(C2(F)CCN(C(C(C=CC)O)=O)C2)=O)CC(C)OC(C)(C)C1C 53871,C1(C)(C(=O)NCCN2CCN(C(C3OCCC(C)C3)=O)CC2)CCS(=O)(=O)CC1 53872,c1(C(N2CCC(C(C)C(N3CCCCC3CCO)=O)CC2)=O)cc(N)cc(O)c1 53873,c1(C(N2CC(CNC(C3C(C(=O)OC)C3)=O)C(C)C2)=O)cc2c(cn1)CCCC2 53874,Cc1nsc(N)c1C(N1CCC1CNC(c1cc(Br)n(C)n1)=O)=O 53875,N1(CCN(CC)CCC(=O)NC(C)C)N(CCCCC)C(COC)(C)CNC1=O 53876,Cc1c(NC(c2sccc2NCc2ccnc(O)c2)=O)ccc(Br)c1Cl 53877,C1(CNC(CCCCC#C)=O)CCCC2CN(C(=O)Cc3ccc(F)nc3)CC12 53878,n1(CC(=O)N(C2CN(C(=O)COCCN(C)C)CC2F)C)cnc2ccccc12 53879,Cc1cnn(CCN(C(=O)CN(C(=O)CNc2cccnc2)CC(C)C)C)c1 53880,CCC(CC(=O)NCC1OCCC1C(=O)NCc1cc(OC)ns1)C(F)F 53881,N1(C(C2C(C=C)OCC2)=O)C2CCC1CC(NC(=O)C(C)(C)c1cncnc1)C2 53882,N1(C(C=CCSC(C)(C)C)=O)CC2CC1CN(C(=O)CSc1ccccn1)C2 53883,C1(C(=O)NCCCNC(c2ccn(C)c2)=O)CCNC(=O)C1 53884,C(=O)(C1=Cc2ccccc2C1)C(C(C)N(C(C1COCCC1O)=O)CC)=O 53885,C(=O)(C1=C(Cl)CC1)N.C(C(O)COCC(=O)NCC=CCOC(C)(C)C)N(C)C(N)=O 53886,N1(C(C(C(C)C)OC)=O)CCC2(CNC(=O)CCCn3cccn3)CCCC12 53887,C=C(C)C1CC=C(C(c2nnnn2C(C)C)NCCC(C)C(C)(C)C)CC1 53888,N1(CC(=O)CCNC(=O)C(c2ccc(Br)cc2)(F)F)CCC(C(O)C(F)F)CC1 53889,c1(C(=O)NCCCN(C(=O)CCC2CCCCCC2)CC)cc[nH]c(=N)c1 53890,Cc1ccc(CNC(C2CCN(C(=O)COCC3CCCOC3)CC2)=O)c(C)c1 53891,N1(C(CCN2C(C)CCCC2)=O)CC2=C(C1)CN(C(C1CCS(=O)(=O)N1)=O)C2 53892,C12(C(=O)NCC(C(C)C)O)CCC(NC(=O)CC(C)O)(CC1)C2 53893,CC(C)CC(CNC(=O)CCC(C)(F)F)C(=O)NCC1=NOC2COCC12 53894,C(=O)(CC(O)CNC(=O)CNC(=O)OC(C)(C)C)N(C1CCCC1O)C 53895,Cn1nc(CNC(=O)CC2CCOC2=O)c2c1CCN(C(c1ccon1)=O)C2 53896,c1(CNC(COC)=O)ccc(CNC(=O)CC(C)C2CCC2)cc1 53897,C(=O)(C(CC(C)C)N(C)C)NCC1(OC)CCN(C(c2ccn(C3CC3)n2)=O)C1 53898,C(=O)(C1=CCCC1(C)C)N1CC2C(NC(C3C(C(=O)OC)CC3)=O)(CC2)C1 53899,c1(C(N(CCCNC(=O)Cc2ccnn2C)CC)=O)cnc(Cl)c(F)c1N 53900,c1(COCC)nnc(N2CCCC2CCNC(=O)C2CC2)s1 53901,CC1CC(NC(c2cc(C#N)n(C)n2)=O)CCN1C(c1cnc(C2CC2)[nH]1)=O 53902,C=CCN(OC)C(=O)CCC1CCCN(C(=O)CC2CC(F)(F)C2)C1 53903,C(C1=NOC2(CCC2)C1)NC(C1CCN(C(C(CC)N(C)C)=O)C1)=O 53904,Cn1nc(C(F)F)c2cc(C(=O)NC3CC(NC(=O)CCSC(F)(F)F)C3)sc12 53905,C1(C(=O)NC(c2nccn2C)CC)CCCN(C(c2nn(C)cc2C)=O)C1 53906,C1(CNC(C(C)n2ccnn2)=O)(NC(=O)CCNC(=O)C=CCl)CCCC1 53907,c1(C(=O)NCCN(CCC)C(C2(C)CC(C)=NO2)=O)nc(C)n(C)n1 53908,Cc1nc(CC(=O)NC(Cc2cc[nH]n2)C(=O)NCC2CC(F)(F)C2)n[nH]1 53909,C1(NC(CCc2nc(C)c(C)[nH]2)=O)CN(C(=O)CC2CCCCC2)CCC1C 53910,c1(-c2cc(NC(C3CCCCCC3)C)sc2)ccc(F)cc1 53911,c1(C(=O)NC(C)CNC(C2CCN2S(C)(=O)=O)=O)cnc2n1CCS2 53912,C1(C(N(c2cn(CC)nc2)C)=O)C(C2CC2)CCN1C(C1C2CC3C(C2=O)C13)=O 53913,CCCCC(CC)CC(=O)NC1CCC(C)N(C(=O)C(C)CC)C1 53914,c1(CC(C(=O)NC2(CNC(CCN(CC)CC)=O)CCOC2)C)ccccc1Cl 53915,C1(C(=O)NCC2N(C(c3cc(C)sc3C)=O)CC(F)C2)CCCC2(CC2)C1 53916,C1(NC(=O)CC2CCCC23CC3)C2CCC(C2)C1C(=O)NC1CCC(C2CC2)C1 53917,C1(CC)CC(C)CN(C(=O)C(=O)N(C(c2ccccc2)C)Cc2cccs2)C1 53918,Cc1cc(Br)ncc1NC(C1CC(O)CN1C(=O)Cn1ccncc1=O)=O 53919,N1(C(C2CN(C(Cc3nc(C)sc3C)=O)CC(F)C2)=O)CCC(O)C(C)(CO)C1 53920,c1(OC(C)C)ncccc1CC(=O)NC1CCCC1NC(=O)CCc1cscn1 53921,c1(N2CCC(NC(COCC)=O)C2)cc(C)ncc1C(=O)OCC 53922,Cc1cc(F)ccc1CC(=O)NC1CN(C(=O)C(C)NS(C)(=O)=O)CC1(C)C 53923,C(C)(C)(CC(F)C(=O)N(C1CCOC(C)(C)C1)C)NC(C1C(C)OC(=O)N1)=O 53924,CC1(C)CC=C(c2cn3cnc(C(=O)NCc4ccc(Cl)cn4)c3s2)CC1 53925,C1(CNC(c2c(CC)nns2)=O)CCN(C(C2CN(C)CCO2)=O)C12CC2 53926,C1(NC(CCN(C(=O)C(C)CC2CC2)C(C)C)=O)CC1C1CC1 53927,N1(C(CN(C(C)=O)C)=O)CCCC2(CCN(C(c3c[nH]nc3C(F)(F)F)=O)C2)C1 53928,C1CCCCN1C(C(C)(C)C)=O.c12ccc(cc1)CNC(=O)N2.C(=O)(C1CC1)OCC 53929,C1(CNC(N2CC(CC)OC(C)C2)=O)CC2(CO1)CC1(C2)OCCO1 53930,C1(CC)CN(C(c2sc(CC(C)C)nc2C)=O)CCN1C(=O)C(C)C(C)(C)O 53931,S(=O)(=O)(CC(=O)NC(C(C)NC(=O)CCCNC(N)=O)C(C)C)NCC 53932,C1(NC(=O)CSCC(N2CCCC2)=O)CC2CC1N(C(C1C3CCCOC13)=O)C2 53933,CN1CC(C(=O)NCC(C)(C)NC(=O)COC(F)F)c2ccccc2C1=O 53934,C1(NC(c2n(C)nc(Cl)c2)=O)CC12CCN(C(C1CCc3nn[nH]c3C1)=O)CC2 53935,N1(C(C(CC=C)C)=O)CCC2(CC1)CC2(CO)CNC(c1ccc(C)cn1)=O 53936,C1(NC(c2c(F)ccnc2F)=O)CC1C1CCCN(C(=O)C2=C(Cl)CC2)C1 53937,N1(c2nc(OC)nc(OC)n2)CC2CCCC(C1)C2C(N1CCCC(F)C1)=O 53938,C(=O)(C1=C(C)CCCC1(C)C)N(C1CCC(OC)C1)C(c1cccc(N)c1)=O 53939,c1(C(N2CCN(C(c3ncsc3Br)=O)C(CO)C2)=O)ccc(F)cc1Cl 53940,Cc1nc(CNC(=O)CCC(=O)N(C)C)oc1C(=O)NC(c1nc[nH]n1)(C)C 53941,C1(C(N2CCC(N(C(=O)C(C)(C)NC(=O)C(F)(F)F)CC)C2)=O)CCC2(CCC2)O1 53942,Cc1cc(C(N2CC(F)(F)CC2CNC(=O)CCc2cnc[nH]2)=O)cc(N)c1O 53943,C1(NC(C(CCSC)OC)=O)C2CCC1N(C(c1nc(C)ncc1Br)=O)C2 53944,c1(NCCCCC(C)NC(c2ccc(OC)c(C)c2)=O)ncnc2[nH]ccc12 53945,N1(C(N2CC(C#C)(F)C2)=O)CCOCCc2ccc(F)cc21 53946,C(C(C)(C)CC(=O)NC(C1CC=CCC1)C(=O)Nc1ccccc1CCO)OC 53947,c1(C(=O)NCC2CCN(C(C3C(C)(Br)C3)=O)C2)coc2ccc(F)cc12 53948,Cc1ccccc1C(F)(F)C(=O)NC1CCC(NC(=O)C(N2CCCC2)C2CC2)C1 53949,C(C(C)CN=c1cc(C)nc(CO)[nH]1)NC(C=Cc1cccc(OCC)c1)=O 53950,c1(OC)cccc(OC(F)(F)F)c1S(=O)(=O)NC1COC2(CNC2)C1 53951,C1(CNC(C2CC(F)(F)C2)=O)CC2(CCC2)CN1C(c1cccn2nnnc12)=O 53952,CC12COC(C(N3CCC(O)(CNC(c4ccns4)=O)C3)=O)(C1)C2 53953,c1(OCC(=O)NC2C(C)CN(C(=O)CCCF)CC2C)ccc([N+](=O)[O-])c(Cl)c1 53954,c1(CC(N2CC3C(C2)N3C(c2ccc(O)c(Cl)c2)=O)=O)cc(Br)ccc1I 53955,c1(C(N2C3CC(NC(Cc4c(C)non4)=O)C2CC3)=O)nn(C)c2c1CSCC2 53956,Cc1nn(C)c(Cl)c1C(=O)NC12CC(CNC(c3ncccc3O)=O)(C1)OC2C 53957,N1(C(CCC)=O)CC2(CNC(c3[nH]nc(OCC)c3Cl)=O)CCC1CC2 53958,c1(OCCN(C(=O)CCCn2cc(C)nn2)CC)ccc(C)c(C)c1.C(CO)O 53959,c1(OC)cc(O)c(NCCc2ccc(OCCOC)cc2)cc1S(=O)(=O)OC 53960,C1(CNC(c2cc(C)on2)=O)CC2COCC2N1C(C1CC(C)(C)CN1C)=O 53961,Cc1c(C(N2CCN(CCNC(=O)C=CC(F)(F)F)CC2)=O)cnn1CC(F)F 53962,C(=O)(Nn1ccccc1=O)C1CC(NC(C(C2CC2)OC)=O)C1 53963,N1(C(CC2CCC(C)CO2)=O)CC(NC(c2cccn2CC2CC2)=O)CC1(C)C 53964,C(C(=C)CCN)NC(CC1(OC)CCC1)=O.C(=O)(C(C)(C)OC)NCCC 53965,c12cccc(n1)NC(=O)C(C)N(C)CC(=O)N(CC)C2.C1(C(N)=O)CCCCC1 53966,C1(C(N2CCC(NC(=O)Cc3ccc(Cl)nc3)C(F)C2)=O)CN=C2N=CNN2C1 53967,N1(C(CCOC)=O)CCOC(CC2CN(C(=O)CC3CCC4CC34)C2)C1 53968,C(CCCCCF)NCCC.C(C(F)(F)F)=CC(=O)C(=O)C=C.N 53969,Cc1cn2c(CC(N3CCC(C4CC4)C3C(=O)NCC=CC3CC3)=O)csc2n1 53970,c1(C(=O)OC)cc(OC(C)C(c2ccccc2Br)OC)cc(Cl)c1 53971,N1(C(c2cc(C)cc(C)c2C)=O)CCOC2(CCN(C(C3CCN3C)=O)C2)C1 53972,c1(C(=O)NC2CC(C)N(C(c3cc(Cl)n(C)n3)=O)C2)ccc2ncsc2c1 53973,c1(C(N2CCN(C(C3CCC(C)CC3)=O)CC2)=O)cc2cc(Cl)ccc2n1C 53974,c1(C(N2CC(C(C(N3C(C(=O)OC)C=CC3)=O)OC)C2)=O)ccnnc1C 53975,S(=O)(=O)(c1c[nH]c(C(=O)NCC(O)CNC(C2CC(C(F)F)C2)=O)c1)NC(C)C 53976,C(=O)(CCCCSC)NCCN(C(=O)C(C)C1CCCO1)CCOC 53977,N1(C(C(CCC)C)=O)CCN(C(c2ccc[nH]2)=O)CC1c1cn[nH]c1 53978,N1(C(C(COCC)C)=O)CCC(C)(C(=O)Sc2cn(-c3ccccc3C)nn2)C1 53979,N1(C(c2cnc(CC)nc2)=O)CCN(C(c2cocc2C)=O)C(C)C1C 53980,C12(CNC(=O)CC3CCN(C(C4COCO4)=O)C3)CCN(CC1)CC2 53981,N1(C(C2C(C(C)C)C2)=O)CC(C)(CNC(c2onc3c2CCCC3)=O)CC1(C)C 53982,CC(C(=O)NCCCCCCNC(=O)CC(C)(C)N(C)C)C(F)(F)C(F)F 53983,c1(OC)cncc(C(=O)NC2CCCC(C(N3CCC(F)CC3)=O)C2)c1 53984,C1(NC(CN(C2CC2)CC)=O)C2CC(O)C1N(C(=O)Cc1cscn1)C2 53985,c1(NC(C2CN(c3ccncn3)CCO2)=O)ccc2c(=O)[nH]ccc2c1 53986,c1(C(N2CC(C#C)(C(=O)O)C2)=O)cc(Br)c(O)c(Br)c1 53987,C1(c2scc(C(=O)OC)n2)CN(N2CCCC2c2cc(C)cs2)CCO1 53988,C1(S(N)(=O)=O)(C(=O)NC(C)CN(C(=O)CCC#N)C)CCCC1 53989,CCCC(CNC(=O)CC1(O)CCCC1)NC(=O)CC1CCOC1C 53990,C(=O)(C(C(C)O)N(C)C)NCC1(NC(C=C(C)I)=O)CC1 53991,N1(C(NC2CCc3cccnc32)=O)CC2(CCOCC2)c2ccccc21 53992,c1(CN(C(c2n[nH]c(C)n2)C(=O)NC2CC2)CC=C)ccccc1 53993,C(=O)(C1=CCCCO1)NC(C)CNC(C1(Oc2ccccc2)CC1)=O 53994,CCCCC(CCCC)CC(=O)N1CCOCC1CS(N)(=O)=O 53995,c1(C(C(=O)N(C2CCN(C(=O)C(N)=O)C2)CC)N(C)C)c(F)cccc1F 53996,N1(C(C(c2ccc(Br)cc2)C)=O)CCC(F)C(NC(C2CS(=O)(=O)C2)=O)C1 53997,c1(C(=O)NC2CC(CNC(CC(CCC)O)=O)C2)cc(F)cc2nccnc12 53998,c1(CCC(=O)N(C)CC2N(C(CCSC)=O)CCC2)ncc(F)cn1 53999,N1(C(c2c(CN=[N+]=[N-])noc2)=O)CCN(C)C(C(=O)NCC2CCCCN2)C1 54000,O=C(C1Cc2c(Cl)cccc21)NCC1(F)CC(NC(c2c(F)cccc2F)=O)C1 54001,C1(C)(C(N(C)Cc2ccc(CNC(=O)Cc3cccs3)cc2)=O)CCCCNC1=O 54002,c1(C(=O)NCC(CO)NC(=O)CC2(O)CCC2)cccc(-n2ccnc2)c1 54003,c1(C(=O)NC2CCC(N(C)C(c3ccccc3Cl)=O)CC2)cc(F)ccc1F 54004,c1(SCCOCCNC(CC2CC(CC(C)C)OCC2)=O)ccc(Cl)cc1Cl 54005,CC(C)CC(C(=O)NC1CCN(C(=O)C(C)SCC#N)CC1)N1CCCCC1=O 54006,N1(C(COC)=O)CCC2(C=C(C(=O)NCC3(C(C)(F)F)CC3)C2)C1 54007,C1(C(N2C(CF)CC(OC)C2)=O)CC2CCC(C1)N2C(=O)Cc1cnns1 54008,N1(C(C(CCCC)O)=O)CCCC(C2CCCN(C(=O)CC3CC(OC)C3)C2)C1 54009,c1(C(=O)NCC2C(CNC(CCC(=C)Br)=O)C2)cc2ccccc2n1C 54010,N1(C(C2CC3C=CC2CC3)=O)CC2CCN(C(c3cnc4cccnn34)=O)C2C1 54011,C(=O)(CCCC(=O)OC(C)(C)C)NC1CCC(NC(=O)NCc2n(C)cnc2)C1 54012,c1(CCC)onc(C)c1C(=O)NC(CNC(c1cc(C(F)F)ccn1)=O)C1CC1 54013,N1(C(C2CSC2)=O)CCC2(CC1)CC(NC(C13CCC(CF)(CC1)CC3)=O)C2 54014,c1(C(N2C(C)C(NC(=O)CC3CCC(=O)N3)CCC2)=O)ccc(F)c2[nH]ccc12 54015,C12(NC(CC(=C)C)=O)CCC(CNC(=O)CCCOc3ccccc3F)(C1)OC2 54016,c1(C(N2C(C(CNC(c3ccc(C)s3)=O)(C)O)CCC2)=O)cn2ccccc2n1 54017,C1(NC(CSCCC)=O)CCN(C(=O)C=C(C)C(C)(C)C)CC1O 54018,C(c1cn(C)cn1)=CC(=O)NC(C1CCN(C(=O)C=Cc2ccnn2C)C1)C 54019,C1(CNC(C2CN(C)C(=O)C2)=O)CC(C(=O)NCc2cn[nH]c2)=NO1 54020,CCCC1CC(=O)C2CC3C(C(Nc4cc(C)cnc4OCC)C2C3)C(=O)N1 54021,CCCCCCC(C(=O)NCC(C)NC(C1(C#N)CCCC1)=O)NC(C)=O 54022,C1(CC(N2CC(NC(CC3N(CC)C(=O)CC3)=O)C(OC)C2)=O)CC2C=CC1CC2 54023,c1(-c2scc(C(C(=O)NCc3ccco3)N(CC(C)C)CC#N)n2)cccc(C)c1 54024,c1(CC)c(C(=O)NC2CN(C(=O)CCc3ccn(C)c3)CC23CC3)cccc1C 54025,C1(CNC(C(CC)OC)=O)CCC2(CN(CCOc3c(C)cc(Cl)cc3C)C2)O1 54026,N1(C(Cc2c(C)occ2)=O)CC(NC(c2cocc2C(N)=O)=O)CC(F)C1 54027,c1(C(=O)NCC(=C)CCNC(=O)C(Cc2cnc[nH]2)NC(C)=O)ccc(F)cc1 54028,c1(C(=O)NCCNC(CS(CC)=O)=O)ccn(CC(F)(F)F)c(=O)c1 54029,N1(C(c2cc(C)ns2)=O)CCCN(C(C2CCn3nccc3C2)=O)C(C)C1 54030,c1(C(N2C3CN(C(c4ccc(C(N)=O)cn4)=O)CC2C3)=O)ccc([N+](=O)[O-])cn1 54031,N1(CC(=O)NCC(C)N(C(c2c[nH]c(=N)s2)=O)CC)CCCCCC1 54032,N1(C(C(CC(C)C)CNC(c2ccoc2)=O)=O)CC(C)c2ncccc21 54033,N1(C(C2(C)CC(=O)NC2=O)=O)CC2(CCCC(CNC(=O)CC3CCC3)O2)C1 54034,N1(C(CC2ON=C(C)C2)=O)CCC(O)(CNC(c2cc(C(F)(F)F)cs2)=O)CC1 54035,CC(C)CCCCC(=O)NCCCC(O)C(=O)NCc1cc(Cl)ccn1 54036,C1(NC(CCN(C(C)C)C(C2C=CCS2)=O)=O)C(O)CC1O 54037,c1(C(C(=O)NC)NC(c2c(CC)ccs2)c2nnnn2C(C)C)ccccc1Br 54038,c1(NC(C2CCCC2NC(=O)CNC(=O)C(F)(F)F)=O)cnncc1Cl 54039,C(=O)(CCCCCCCCN)N1CCN(CC(=O)Nc2c(OC)cccc2)CC1 54040,c1(NC(C2CCN(C(C3CCC(C(=O)OC)C3)=O)C2)=O)ccc(O)cc1O 54041,CC1(NC(c2c(OC(F)(F)F)cccc2O)=O)CCN(S(N)(=O)=O)CC1 54042,C1(CNC(COCC=C)=O)CN(C(=O)C(C2CCC2)SC)CCC1(C)C 54043,C1(C(=O)NC2CC(NC(c3n(CC)ccc3)=O)C2)Cc2cc(F)ccc2O1 54044,Cc1c(C(=O)NCC(C)CNC(=O)C(C(C)C)NS(C)(=O)=O)ccc2c1CCC2 54045,N1(C(CN(C(C)=O)C)=O)CCN(C(=O)CC2CN(CC(F)(F)F)C2)C2CC12 54046,c1(NCCN(c2cc(C(C)C)nc3n2ncn3)C)ccc(C(N)=O)cc1[N+](=O)[O-] 54047,C1(C(C)NC(c2ccn(C)n2)=O)CCCN(C(c2cnc(=N)[nH]c2)=O)C1 54048,c1(CNC(c2cnn(C)c2C)c2n(CC)nnn2)cn(C)c2ccccc12 54049,C12CC(C1C)CC(=O)O2.C1(OCC)C(OC)O1.CS.C(C)OC.CC 54050,N1(C(c2c(C)nccc2)=O)CCN(C(=O)CCc2ccccc2F)CC1CO 54051,C#CCC(C(=O)NCC(C(=O)OC)OC)NC(c1cc(C(N)=O)co1)=O 54052,c1(CC)cccc(F)c1C(=O)NCC(C(C)C)NC(=O)CC1COC2CC1C2 54053,C1(CC(=O)NC2C(NC(c3cc(=N)[nH]cc3)=O)C2)CCC2(CC1)OCCO2 54054,c1(C(C(=O)NCCCCCN(C(C2CC(C)C2)=O)C)O)ccc(F)c(Cl)c1F 54055,c1(C(=O)NCCC(C)(C)NC(C2CCOC2(C)C)=O)ccccc1C#N 54056,C(=O)(N1OC2CCC1CC2)C1C=CC(C#C)(OC)C1 54057,Cc1cc(C(=O)N(CC(C)N(C)C(C2CCCN2C)=O)C)ccc1C(F)(F)F 54058,CCCCC(CC)C(=O)NC1CCCC1NC(=O)C(C)(C)c1cnco1 54059,C1(NC(c2cc(-c3nc(C)sc3)oc2)=O)CCN(C(c2ccoc2Cl)=O)CC1C 54060,C=CCC(C)(O)C(=O)NC(C)C=CC(=O)N(CC(F)(F)CO)COC 54061,c1(CCCC(=O)NCC2CC(NC(=O)C(F)C3CCC3)C2)nc2ccccc2s1 54062,c1(N2CCOCC(CNC(Cc3cccc(OC)n3)=O)C2)cc2nncn2cn1 54063,C1(NC(CC2C(C)C2)=O)CN(C(=O)C(C)S(C)(=O)=O)CCC12CCC2 54064,CC1(C)CCC=C(C(=O)NC2CC(CNC(=O)CCC3CCC(=O)N3)C2)C1 54065,Cn1nc(CNC(=O)C(C2CCOC2)NC(=O)OC(C)(C)C)cc1C(F)(F)F 54066,N1(CC(=O)NCC(C2CCC2)NC(c2cccnc2O)=O)CCS(=O)(=O)CC1 54067,C(=O)(C1=CC(O)C(NC(c2ccc3c(c2)CCC3)=O)C1)N1CCN(C(C)=O)CC1 54068,C(C(C)C)(C(O)C(=O)NC(CNC(c1cc(C)ns1)=O)CO)OC 54069,c1(C(N2CCCCC2c2ccccc2)C(=O)N(CC=C)CC)cn(C(C)C)nc1Br 54070,CCCCC(C(=O)NC1CCN(C(C2CC2(C)C(C)C)=O)CC1F)NC(N)=O 54071,C1(CC(=O)N(C)CC2N(C(C(F)OC)=O)CCC2)CCCN(C(C)C)C1 54072,Cc1cccc(C(N2CC=CC(NC(C3CC(N=[N+]=[N-])C3)=O)C2)=O)c1F 54073,C(=O)(CCCC(C)(F)F)N(C1CCCN(C(C(C=CC)O)=O)C1)CCF 54074,N1(C(COCCC=C)=O)C2CCC1CC(NC(=O)CN1Cc3ccccc3C1)C2 54075,C(=O)(CC(C)(C)CC(F)(F)F)N1CCC(COC)(NC(=O)C(F)=CCCF)C1 54076,C1(NC(c2cc(CC)n(CCO)n2)=O)CN(C(C2CC(=O)N(C)C2)=O)C(C)(C)C1 54077,N#CCCCC(=O)N1CC(F)CC1CNC(c1cccnc1-n1nccn1)=O 54078,c1(OC)c(Cl)ccc2[nH]c(C(N3CC4CC(O)C3C4NC(=O)CC(C)F)=O)cc12 54079,C=CC1(CC(=O)NCCC(C)NC(=O)CCc2c[nH]c(=N)[nH]2)CCCCC1 54080,CCC(CO)CN=c1cc(C)c(S(=O)(=O)N2C3C=CCC2CCC3)c[nH]1 54081,c1(C(N2CCCC(N(C(C(C=C)(C)C)=O)C)C2)=O)c(C)ccn1C 54082,C1(C2CCC2)(CNC(C(CSC)OC)=O)CCN(C(c2ccncn2)=O)CC1 54083,N1(C(c2c[nH]c(=NC)o2)=O)CCC2(NC(=O)C3=C(C)CCC3)CCCCC12 54084,N1(C(C2OCCN(CC)C2)=O)CC2(CCN(C(=O)CCC(C)C)CC2)CC1C 54085,N12CCCC(C)(C)C1C(=O)NOCC(O)CC2=O.C(COCCF)OC 54086,N1(C(C(F)=C(C)C)=O)CCN(C(=O)C(CC(F)F)c2ccc(F)cc2)C(CO)C1 54087,c1(C(=O)OC(c2c(C)n(C)nc2)C)cc(OC(F)F)nc(C(C)C)n1 54088,C(C(C)C(C)C(=O)N1CC(O)CC1CNC(=O)C(C)=CC1CC1)OC 54089,C(=O)(CC(C)CC(C)C)NCCC(C(=O)N(CCCOC)C)(C)C 54090,c1(CC)cc(C(=O)NCCNC(=O)C(=O)NC(c2cccc(C)c2)=O)ccc1Cl 54091,N1(C(CNC(=O)NC)=O)CCC(C)(C)C(CNC(=O)C(=O)NC2CCCCO2)C1 54092,N1(C(C2(C)CCCO2)=O)CC2(NC(=O)CCC3(C#N)CCC3)CC1C2 54093,C=CCC(C(=O)NC1(CC(=O)NC(C)Cc2ccncc2)CC1)C(C)C 54094,C1(CN(C(=O)COCC2CCC2)CC)CCN(C(C2CCC(C)S2)=O)CC1 54095,c1(C(N2C(C(=O)Nc3c(C)ccnc3C)CC2)=O)n[nH]c2cccnc12 54096,c1(SC)nc(=NC(C)C(c2ccccc2)NC(c2cc(C)co2)=O)s[nH]1 54097,C12(CNC(C(CC#C)(C)C)=O)CCCC(CN1C(=O)CNC(=O)OCC)C2 54098,C1(CCC)CN(C(=O)Cn2ccc(C)n2)CC1C(=O)N(C12CC(C1)C2)C 54099,C1(C(=O)NC(c2cn(C)nn2)C(=O)NC(C(C)C)(C)C)CC2(CCC2)CO1 54100,C1(C(=O)NCC2N(C(c3c(OC)c(C)ncn3)=O)CCC2)CCCC1S(C)(=O)=O 54101,CC1COCCN1C(C1CC1(c1cccc(Br)c1)F)=O 54102,C1(NC(C2CC=CCO2)=O)CCOC12CCN(C(=O)Cc1ccccc1F)CC2 54103,C12(C(=O)NCC(CC(=O)N3CC(COC(C)=O)C3)OC)C(=O)C3CC1C2C3 54104,C#CC1(C(N2CC(OC)CC(NC(c3cccc(F)c3C)=O)C2)=O)CCOCC1 54105,c1(C(N2C3CCN(C(C(CC=C)(C)C)=O)CC3C2)=O)nc2ccc(CC)cc2[nH]1 54106,c1(C(N2CCCN(C(C(C=C=C)C)=O)CC(O)C2)=O)ccc(CC)c([N+](=O)[O-])c1 54107,c1(CC(=O)NC(c2cnn(C)c2)C(=O)NCC(CSC)(C)C)ccc(C)c(C)c1 54108,N1(C(C2CCN(CC)C2)=O)CCN(C(=O)COc2ccc(F)cc2F)CC1CF 54109,N1(C(c2c(CC)c[nH]n2)=O)CC(O)CC1(C)C(=O)NCC(C)C(C)(F)F 54110,N1(C(N2CCCS2(=O)=O)=O)CC2CCN(C(=O)CCN3CCC3)CC2C1 54111,C(=O)(C(O)CCS(C)=O)NCCCCCNC(C(C)Cc1cccc(Cl)c1)=O 54112,c1(NC(CCN(C(=O)CC(C)=C(C)C)CC#C)=O)ccc(CSC)c(F)c1 54113,CC1(C)CCCC(NC(C2(CSc3cncnc3)CCOC2C2CC2)=O)O1 54114,C1(NC(=O)C(O)CN2CCOCC2)CN(C(=O)CCOCC(F)(F)F)CC1F 54115,c1(N2CCC(c3scc(CC)n3)CC2)ccc(S(=O)(=O)N(c2ccns2)C)cn1 54116,c1(C(N2CC(CNC(C3N(C)CCC3)=O)C2)=O)cnc2c(c1)CNC(=O)N2 54117,c1(C(=O)NCCCN(C(C2CC23CCC3)=O)CC)scnc1C(F)F 54118,c1(CC)ccc(CN(C(C(CNC(=O)CC2CC2(Cl)Cl)C2CC2)=O)C)o1 54119,C1(CC(C)NC(c2cncc(F)c2)=O)CC2CCC(C1)N2C(C1CCCCCO1)=O 54120,N1(C(c2[nH]cc(OC)c(=O)c2)=O)CC2CCCC(C1)N(C(c1[nH]nnc1C)=O)C2 54121,c1(C2C(NS(C3(c4cn(CCN(CC)CC)nn4)CC3)(=O)=O)C2)cccc(F)c1 54122,O=C(CCCCCCCC1CC1)NC1COCC1NC(=O)C(O)CC1CC1 54123,Cc1nocc1C(N1CC(O)(CCNC(=O)CC2C=CCCC2)C1)=O 54124,N1(C(c2nc(CNC(C(CCC)CC)=O)oc2C)=O)CCC(C)C(F)(F)C1 54125,C1(C(N2CC(OCCNC(C3CC=CCC3)=O)C2)=O)COCC1O 54126,C(=O)(C1=CCC(NC(c2ccc(F)c(O)c2)=O)C1)NCC(C)CC1CCC1 54127,c1(N2CC(OC)C(O)C2)nc2cc(Cl)ccc2s1.c1(CC=C(C)C)csc2c1NC2=O 54128,C1(CN(C(C2CC(N(CC)CC)C2)=O)C)CCCN(C(=O)CC2COCCO2)C1 54129,c1(OC)ccc(F)c(CC(=O)NC2CCN(C(=O)CCF)CC2O)c1 54130,C1(NC(CC#N)=O)CCCOC1C1CCN(C(=O)CNC(C2CCC2)=O)CC1 54131,C1(C(N(C(CNC(c2ccc(C(C)=O)cc2)=O)C)C)=O)CC12CCS(=O)(=O)CC2 54132,c1(CCC)cc(C(=O)NCCC(C)(C)NC(C2CCC2(OC)OC)=O)n[nH]1 54133,C1(CNC(CCN(CCC)C)=O)CCCCC1NC(c1cccc(C(F)F)n1)=O 54134,C#CC1(C)CCCN(C(C2OCCC2NC(=O)CCSCCC)=O)C1 54135,C1(C(N(CCCNC(=O)CCc2nccs2)CC)=O)CNC(=O)CC12CCOC2 54136,c1(C(C)NC(c2cccc(Br)c2)c2nccn2C)ccc(F)c(F)c1F 54137,Cc1cc(CNC(C2COCCN2Cc2cnc[nH]2)=O)nn1C 54138,CCC(C)(C(=O)NCCCN(C(=O)C(F)(F)C1(OC)CCCC1)C)C(F)F 54139,N1(CC(=O)N(CCCNC(c2ncsc2C2CC2)=O)C2CC2)CSCCSC1 54140,CCC(C)C(O)C(=O)NC1CC(OC)CN(C(=O)C(C)(C)CC#N)C1 54141,C1(NC(c2nc(C(C)(C)C)sc2)=O)C2CN(C(C3(CCN(C)C)CC3)=O)CC12 54142,CC1CN(C(c2ccncc2N(C)C)=O)CC1NC(=O)C(c1ccccc1)=O 54143,C#CC(CC)(CC)CCC=C.C1(=O)C(C)C(C)N1.C1(=O)CO1 54144,n1(CCC)cc(C(=O)NC2CCC(CCNC(c3cnc(C)s3)=O)C2)nn1 54145,C#CC1CC2(CC(C(N3CC(CNC(=O)CCC)OC(C(F)(F)F)C3)=O)C2)C1 54146,S(=O)(=O)(c1ccc(C#N)cc1)NC(CC1(C)CN(CC2CNC(=O)C2)C1)=O 54147,N1(C(c2cccc(N)c2N)=O)CCN(C(c2ccc(CO)s2)=O)CC(O)C1 54148,c1(C(=O)NC2CN(C(C(C3CCCOC3)OC)=O)C2)nonc1N 54149,C1(NC(=O)CC2CCC(F)(F)C2)CN(c2ccncc2[N+](=O)[O-])CCC12CCC2 54150,C1(CC)(CC)C(N2CCOC(c3cccc(O)c3)C2)CC1OCC 54151,C1(F)(C(=O)NCC2(O)CN(Cc3c(OCC(=C)C)cccc3)C2)CCC(F)(F)CC1 54152,C(=O)(N=c1ccn(CCCO)[nH]1)C1N(C(c2ccc(COC)cc2)=O)CC=C1 54153,C1(C(=O)NC(c2n(CC)ncc2)C)(CC)CCCCO1.C1(C(=O)N)CCC(CO)CC1 54154,N1(C(c2cc(C)c(O)cc2)=O)C(C(N2CCC([N+](=O)[O-])CC2)=O)C2CC(O)C1C2 54155,C(=O)(CC(CNC(c1c[nH]cc1C(C)C)=O)C1CCC1)NC(COC)CO 54156,c12ccc(cc1Br)NC(=O)NC(C)CN(CC)C(=O)CCCO2.OC.OC 54157,C(=O)(C1=CCC(C)(C)CC1)NCC(CNC(c1c(C)c(C(N)=O)ccc1)=O)O 54158,C1(C)(C(N2CC(CNC(C3OCCC(C)C3)=O)OCC2)=O)CC(=O)N(C)C1 54159,C(=O)(C1CCCc2ncnn21)N1CCCC(N(C(=O)CCCN=[N+]=[N-])C)C1 54160,c1(C(=O)NC2CCCCC2CC(N2CC(N3CCC3)C2)=O)ccc(F)nc1 54161,c1(C(N2C(CNC(C(C(C)C)C)=O)CCCCC2)=O)coc(S(C)(=O)=O)c1 54162,C1(CNC(C(CC)C)=O)CC(F)CN1C(=O)CC1CCC1(OC)OC 54163,Cc1cc(C(N2CC3C(CNC(C4CCC(=O)N4)=O)C3C2)=O)c2sc(=N)[nH]c2n1 54164,CCC(C)CN(C)N1CC2C(c3nc(-c4ccc(C(C)(C)C)cc4)no3)C2C1 54165,N1(C(CCC=C(C)C)=O)CCC(NC(C2CC(=C(F)F)C2)=O)C(F)C1 54166,c1(CCOCC(=O)NCCCN(C(=O)CC2C=CCCC2)C(C)C)ccccc1 54167,Cc1cc(Cl)c(C(N2C3CCC2C(NC(=O)C(C)O)C3)=O)cc1N 54168,C1(COC)CC(O)C(O)CC1C(=O)NC1(C)CCCO1 54169,CCC(CC(C)C)C(=O)N1CC2CC(C(=O)N(C(C)CN(C)C)C)CC2C1 54170,C(C)(CN=c1[nH]c2c(c(=NCCCN=c3cc[nH]c4ccccc34)[nH]1)SCC2)SC 54171,C(=O)(CCCCCO)NCCOC1(CNC(C2CC(C)OC2)=O)CCOCC1 54172,CCC(C)(C(=O)N1CCCC(CO)(NC(c2ccc(OC)c(C)c2)=O)C1)C(F)F 54173,C1(C(N2CCC(NC(c3ccnn3C3CC3)=O)(CF)C2)=O)CN2CCC1CC2 54174,c1(OC)cc(N)ccc1-c1cn(CCC(=O)NCC(CO)OC)nn1 54175,N1(C(C=CC)=O)CCCC2(CCCCC2NC(c2cc(C)c(C)cn2)=O)C1 54176,c1(C(C)NC(C(c2scc(C)n2)C)=O)cc(Br)ccc1Cl 54177,c1(C(=O)NC2C(NC(Cc3c(C)ncs3)=O)C2)cc([N+](=O)[O-])cn1C 54178,N1(C(CCCC(C)=O)=O)CC2(CC(NC(=O)CN3CCS(=O)(=O)CC3)CO2)C1 54179,C1(NC(CN(C(CCOCCC)=O)C(C)C)=O)CCOC(CC)C1 54180,C1(C(N(C(CNC(C(CC(=O)OC)C)=O)C)C)=O)Cc2cccnc2C1 54181,c1(N2CCC(C(=O)NCc3c(OC)c(Cl)c(Cl)cc3)C2)nc(C)nc2occc12 54182,N12CCC(C(O)C1)SCC2=O.N1(CC(=O)Nn2cnnn2)CC2CC2C1 54183,c1(C(=O)NC(C(C)NC(C2(O)CCCCC2)=O)CO)ccc(Cl)c(C#N)c1 54184,CC(C(=O)N1CCCC(CNC(=O)CNC(N)=O)CC1)C(C)(F)F 54185,c1(C(N2CC(C(Cn3cc(CS(C)(=O)=O)nn3)F)C2)=O)cc2sccc2s1 54186,C1(C2CCC2)(C(=O)NC2C(NC(C3(C(F)F)CCCO3)=O)CCC2)CC1 54187,N1(C(C(C)OC)=O)CCCN(C(c2cc(C)n(C(C)(C)C)n2)=O)C(C)C1 54188,CC(C)C(CC(=O)NC12CC(NC(c3ccnc(S)c3)=O)(C1)C2)C(C)C 54189,C1(NC(CC2C(C)(C)N(C(C3NC(=O)OC3(C)C)=O)C2)=O)CCCN(CCO)CC1 54190,O=C(CCN1C(=O)CSc2ccccc21)NCCNC(c1ccc(Cl)[nH]1)=O 54191,c1(CNC(CCCN(C(C(CSC)C)=O)C)=O)nn(C)cc1C 54192,c1(C(=O)NC(C2CCCCC2)CNC(C(C=C)(C)O)=O)nccc(C)c1F 54193,C1(CC(=O)NCC2(CNC(C(C)(C)C3CCCCC3)=O)CCC2)CC(=O)NC1=O 54194,N1(C(C23N(C(CCN(C)C)=O)CCC2C3)=O)CCc2nnnn2CC1 54195,c1(C(N2C(CC)C(NC(C3CCS(=O)(=O)N3)=O)CC2)=O)csc2nccn12 54196,c1(CC)ccc(C(N2CCN(C(=O)C3CC3)C3CC23)=O)cc1[N+](=O)[O-] 54197,c1(C(=O)NCC(CCNC(Cc2cn(C)nc2)=O)(C)C)c[nH]c2ncccc12 54198,C1(NC(CCC2C(C)C2)=O)CCN(C(c2ccc(NC=O)cc2)=O)C1(C)C 54199,N1(C(c2ccn(CC(F)F)n2)=O)CCN(C(c2cnc(O)o2)=O)C(C2CC2)C1 54200,c1(OCCC(=O)NC(CC)CN(C(=O)COC2CC2)C)cccc(OC)c1 54201,c1(C(=O)NC2(CC(=O)N(C3CCSC3)C)CCC2)cc(OCCOC)n[nH]1 54202,CCCC(CC)CC(=O)NC1CCN(C(c2ccc(C)cc2)C)C1 54203,C=C1CC(C(=O)N(C2CC(C)C2)C)(CNC(c2cc(Cl)cs2)=O)C1 54204,N1(C(C2C(NC(CCCCC#C)=O)CCOC2)=O)CC(O)CCC(C)(C)C1 54205,c1(N(CCC(C)(C)SC)C)cc(C)c(S(=O)(=O)NC(C2CC2)C2CC2)cn1 54206,C#Cc1ccc(CNC(CC(=C)Br)C2CC2)c(O)c1 54207,C1(CC(=O)NCC(=O)OCc2ccccc2)OCC2CCN(C(=O)CCBr)CC12 54208,CC(F)(F)C(F)C(=O)NCC1CN(C(=O)CSCC(F)F)CC12CC2 54209,c1(C(=O)OC(C(N2CCN(C(C)=O)CC2)=O)C(C)C)cc2cc(Cl)ccn2n1 54210,C#CCCC(O)C(=O)NC1COCCN(C(c2ncc(C)cc2C)=O)C1 54211,C(CCCCNC(c1c[nH]nc1F)=O)N(C)C(c1cnn(CC2CCCC2)c1)=O 54212,N1(C(c2occ(C)c2)=O)CC(NC(=O)CC2CCC(=O)NC2=O)C2CCCC12 54213,C1(C(=O)NCC2CCCN2)CC(O)CN1C(c1ccsc1)=O 54214,C(C1CCCN1C(C1CC(C)(O)C1)=O)=CC(=O)N(C)CC1CCN(CC)C1 54215,C(N=c1ccc(Br)c(S(=O)(=O)N2CCC(C(C)(C)C)C2)[nH]1)c1nccc(C)n1 54216,C(c1ccc(F)cc1Cl)=CC(N1C(C(C)C)CN(C(c2ccn(C)n2)=O)CC1)=O 54217,C1(NC(=O)NCCCN2CCCC2=O)CC1C1CC1 54218,c1(C(=O)NC(c2ccccc2)C(C)NC(=O)C(C)(C)O)cccc(CO)c1 54219,N1(C(C(C)O)=O)CC(C)(C)OC2(C1)CN(C(C13CCCC1C3(F)F)=O)C2 54220,c1(C(N2CC3(CN(C(CC(=O)NCC#C)=O)C3)C2)=O)cc(S(N)(=O)=O)cs1 54221,N1(C(CCC(CC)C)=O)CCCN(C(c2cnc(C3(C)OCCO3)s2)=O)CCC1 54222,N1(C(c2cc(CCC)n(C)n2)=O)CCC(C)C(NC(c2ocnc2CCC)=O)C1 54223,c1(-c2cc(C)c(OC(C)C)nc2)ccc2[nH]c(C(N3CCCC3CO)=O)nc2c1 54224,C1(C(=O)NCc2cnsc2)(CNC(CC(C)n2ccnc2)=O)CCCCC1 54225,C(=O)(C(F)CC(C)(C)NC(c1ccns1)=O)NC1CCN(C)C1=O 54226,c1(C(N2CCC(N(C(C3CC3c3cnc[nH]3)=O)CC)C2)=O)ccc(Cl)c(F)c1 54227,c1(C(=O)NC(C2CN(C(C(C)OCC(F)(F)F)=O)C2)C)ccc2scnc2c1 54228,Cn1cc(Br)c(C(C(=O)NC(C)(C)C)N(CCC=Cc2ccccc2)C)n1 54229,N1(C(C(CO)N(C)C)=O)CCN(C(=O)Cc2ccccc2)C2CNCC12.N 54230,CC1CCC(NC(c2cc(Cl)no2)=O)CN1C(=O)CN1CCN(C)CC1 54231,[N-]=[N+]=NCCCOCC(=O)NC(C(=O)NCCC(O)C1CC1)C1CC1 54232,C(=O)(CCCCC(=O)N1CCN(C(c2cccc(OC)c2)=O)CC1C1CC1)NC 54233,CCCC(C)(O)CC(=O)N1CCCCC(N(C)C(c2nc(C(F)(F)F)cs2)=O)C1 54234,N1(C(c2nnn(C)c2N)=O)CC2(CCN(C(C3CCCOC3)=O)C2)C1 54235,CCCCCC=CCC(=O)NC.c1(NCC(=O)NCC2C(C(=O)OC)C2)cscn1 54236,n1(CC(N2CC(N(C)C)C2)=O)cc(CNC(=O)C(O)C2CCCC2)nn1 54237,N1(C(=O)NC2(c3nc(C)on3)CCC2)CCC2C(CCCN2C2CC2)C1 54238,n1(CC(N2CCC(CNC(CCCCCC)=O)C2)=O)cc(C)c(O)nc1=O 54239,c1(CC(=O)N(C(CNC(C(C2CCCCC2)OC)=O)C)CC)ccc(O)c(F)c1 54240,C1(NC(CSCC=C)=O)CCN(C(=O)CN2CSCC2=O)CC1F 54241,C1(C(C)NC(=O)COCC2CCC2)CCN(C(=O)Cc2csnn2)CC1 54242,C1(NC(CCC=C)=O)CCN(C(c2cc(-c3ccco3)[nH]n2)=O)C(C2CC2)C1 54243,c1(Cn2c(C(O)CO)nc(-c3cccc(CC)c3)n2)c(F)c(F)cc(F)c1F 54244,C(CCCC(=O)NC1C(C)CCN1C(=O)C1=CCOC1)n1cc(CSC)nn1 54245,CC1CC2CC2CC1C(=O)NC1CCCCCN(C(C2(C(F)F)CC2)=O)C1 54246,C1(N(C(CC(=O)NCC)=O)C)CS(=O)(=O)C12CCN(C(C1CCCCC1)=O)CC2 54247,N1(C(c2ccc(OC)o2)=O)CCN(C(=O)C(C)SC(C)C)C(c2cccnc2)C1 54248,C(=O)(C1=NOC2(CCC2)C1)NC1(C)C(C)(C)CCC1 54249,C(CCCCCCNC(c1ccco1)=O)n1cc(COCC)nn1 54250,C1(C(N2CCC(CC(C)NC(C(C=C)O)=O)CC2)=O)Cc2ccccc2C1 54251,C1(CNC(CC2N(C)CCC2)=O)CN(C(c2ncncc2Cl)=O)CCN1C 54252,C(=O)(C(F)CC(C)(C)NC(=O)CC(C)(C)CN(C)C)Nc1c(CC)noc1 54253,C1(c2n(CC)ccn2)CC1N=c1[nH]c(=NCCC(C)O)[nH]c2c1SCC2 54254,c1(C(=O)NCC2N(C(CCC(C)OCC)=O)CCC2)ccc(S(N)(=O)=O)cn1 54255,C1(C(=O)NCC2CC(F)CN2C(C23CC(F)(C2)C3)=O)CCN(c2nncs2)CC1 54256,N1(C(CSCCOC)=O)CCCCC(C2CN(C(c3cc(C(C)=O)cs3)=O)C2)C1 54257,Cc1n[nH]c2cc(C(=O)NC3CCCC3NC(c3ncccc3F)=O)ncc12 54258,c1(N2CCC(N(C)C(C3(c4ccc(F)cc4)CC3)=O)C2)c(Cl)cncc1[N+](=O)[O-] 54259,CC1CCN(CCNC(C2(c3nn[nH]n3)CC3(CC3)C2)=O)CC1 54260,c1(N(C)NCc2cc(C)on2)nc2c(c(=NCc3ncn(C4CC4)n3)[nH]1)CCC2 54261,Cc1cc(N2CC(F)(F)CC2(C)CNC(C2CC23CCCOC3)=O)ncc1C#N 54262,C1(C(=O)NC(CC(C)C)c2ccccc2)(CF)CCN(C(=O)OC(C)(C)C)CC1 54263,C1(OC)CN(C(C2C(C)CCN2C(=O)CSc2cn[nH]c2)=O)CC12CC2 54264,C(=O)(C1CN(C(=O)NN2C3CCC2CC3)c2c(C)cccc21)OC 54265,N1(C(C(CCCNC(CC2CC(C)C2)=O)O)=O)CCc2c(F)cccc21 54266,N12CCC3(CCC(C3)NC(=O)NC3(CCCC3)C1=O)C2.c1(C(=O)NC)ccoc1 54267,N1(C(C2C(C)CCC2)=O)CCCC(CCNC(=O)COCC2CCOCC2)C1 54268,c1(C(N2CC3CC(NC(C4C(C)=C4)=O)C3C2)=O)cc(F)c(C)cc1F 54269,c1(NC)ncccc1C(N1CC(NC(=O)Cc2ccsc2Cl)C(C)C1)=O 54270,C#CC1(C(N2CCC(O)C(O)C2)=O)CCN(C(=O)CNc2cccnc2)C1 54271,C1(NC(c2nc(COC)oc2)=O)CC(NCC2CCCC(C)(C)C2)C12CCC2 54272,c1(-c2cn(C(CNC(C(C3CCCC3)SC)=O)C)nn2)c(F)cccc1Cl 54273,n1(C(C)C)ncc(C(=O)NCC(C2CC2)NC(C2(O)CC2)=O)n1 54274,c1(C(N2C3CC(NC(COC4(C)CCC4)=O)C(C3)C2)=O)ccc2c(C#N)c[nH]c2c1 54275,c1(C(=O)NCC(C2CCOCC2)(F)F)cc2c(s1)CCCNC2=O 54276,CC1CN(C(=O)CCNS(C)(=O)=O)CC1CNC(=O)CC#N 54277,C(C(C(=O)NCC(O)C(=O)OC)C(C)C)NC(C(C(=O)OC)OC)=O 54278,N1(C(CCC2CNC(=O)N2)=O)CC2CCC(C1)N2C(C1CNC(=O)N1)=O 54279,c1(C(=O)NCC(CNC(c2cccs2)=O)OC)cc2ccc(F)cc2o1 54280,c1(OC)ccc2[nH]c(C(=O)NCC3CCN(C(=O)CCF)CC3(F)F)c(C)c2c1 54281,N1(C(C(c2cnn(C)c2)C)=O)CC(NC(c2cc3sccc3[nH]2)=O)CC(F)C1 54282,C1(C2CN(C(C(C3CC3)OC)=O)C2)CCCN(C(=O)Cn2cccn2)C1 54283,CC(C)CC(C(=O)NC(C)(CNC(c1ccc(Cl)nc1Cl)=O)C1CC1)C(C)C 54284,C1(C(=O)NCCN(C(C2CC(OC)CN2CC)=O)CC)CC(=O)N(C(C)C)C1 54285,c1(C(c2nnnn2CCCSC)NC2CC(OCC)C2)nc(CC(F)(F)F)cs1 54286,C1(N(S(=O)(=O)Cc2ccc(F)cc2)Cc2ccccc2)CCc2ncnn2C1 54287,CN1CCC(O)(CNC(=O)CNC(=O)CNC(C2CCC(N(C)C)C2)=O)C1 54288,C1(NC(=O)C2CC2)CC2(CCN(C(C34CC(CO3)C4)=O)CC2)C1 54289,C1(C(=O)NC(C)CC(C)NC(=O)C(C)Oc2cccnc2)CCN(C(N)=O)CC1 54290,c1(C(=O)NCC2CCC(NC(=O)C=Cc3ccncc3)C2)ccc2cncn2c1 54291,C1(O)(CNC(C(CC)(C)C)=O)CCCN(C(=O)CC2CCCC(C)(C)O2)CC1 54292,O=C(N1CCCc2nccn21)C1CC2(C1)CC(c1cn(CC(F)(F)F)nn1)C2 54293,C(C1=CCCN(C)C1)NC(C(C(C)NC(c1cnc(N)cn1)=O)C)=O 54294,C1(N(C(Cc2nc(C(C)C)sc2)=O)C)CCN(C(c2csc(=N)[nH]2)=O)CC12CC2 54295,N1(C(COCCCCC)=O)CCN(C(C2CCCN2CC(C)C)=O)C(C2CC2)C1 54296,CC1CC(C)N(C(c2nnn3c2CCC3)=O)CCN1C(c1cc(N)c(Cl)cn1)=O 54297,c1(N(C2C(OC)COCC2)C)ncnc2c([N+](=O)[O-])cccc12 54298,C1(c2nnnn2-n2ccnn2)(COC(CC)CC)CCC(SC)C1.C1CN1 54299,c1(CONC(C2(CCNC(COCC(=O)OC)=O)CC2)=O)cccnc1 54300,C=C(Cl)CCC(=O)NC1(CCNC(C2CCS(=O)(=O)C2)=O)CCOCC1 54301,C(=O)(C1=CC(c2ccc(F)cc2)=NS(=O)(=O)N1)N(CC(=O)OC)C 54302,C1(O)(NC(=O)Nc2cccc(N3C(C)CC3)n2)CCN(C(=O)OC(C)(C)C)CC1 54303,C=C=CCCC(=O)NC(C1CCN(C(c2cc(C)cs2)=O)C1)C 54304,N1(C(COCC(=O)NC)=O)CCCC(C2CCCCN2C(=O)C(O)CNC)C1 54305,n1(CC=C)cc(C(=O)NCC2(CC(=O)NCC3CC34CCC4)CC2)nn1 54306,Cc1ccc2c(C(=O)NCC(C)CNC(=O)CCc3ccc(F)nc3)coc2c1 54307,c1(NC(c2c(CNC(c3c(NC)csc3)=O)ocn2)=O)ccc2c(c1)COC2 54308,Cc1cc(C(=O)NC2CCN(C(c3cnc(Cl)[nH]3)=O)C2C2CC2)cn(C)c1=O 54309,C(=O)(C(C)(F)C(C)(C)F)N1CC(CN(C)C(c2cn3cnnc3cn2)=O)OCC1 54310,n1(CC)cc(Cl)c(C(=O)NCC2CCCN2C(c2sc(C)cc2C)=O)n1 54311,c1(C(N(C2(C3CCCN3C(=O)C3=CCC3)CC2)C)=O)cc2ccccc2o1 54312,C(=O)(C(CC1CCCC1)NC(=O)C=CCN1CCC1)N(C(CCSC)C)C 54313,C(=O)(CCCCCF)N(CCN1CCN(C(C2(C(=O)NC)CCC2)=O)CC1)C 54314,CC(C)CC(C(=O)N1CCOCC1CC)ONC(c1ccc(CC2CC2)s1)=O 54315,C1(C(=O)NC(C)CC2(O)CCC2)C(CO)CCN1C(c1cnco1)=O 54316,N1(C(C2(NC(C(COC(C)=O)C)=O)CCN(C)C2)=O)CCC2OCCC2C1 54317,CC1CC(C(N2CCCC2CNC(c2cccc(C3CC3)n2)=O)=O)CC(C)C1 54318,c1(C(=O)OC)c(C)cc(C)nc1NC(C)CC(C)NC(=O)CC(C)CC(C)C 54319,C1(NC(C(C)N(CC)CC)=O)CN(C(c2ncc(C(F)F)s2)=O)CCC1O 54320,C(c1cncc(F)c1)=C(C)CNC(=O)N(C)CC1CCS(=O)(=O)CC1 54321,CC(C)C(C)(CNC(c1cnc(S)n1C)=O)NC(=O)C(c1ccc(Cl)s1)C 54322,c1(CCC(=O)NCC(C)(C2CCC2)NC(C(C)OCCCC)=O)c(C)n[nH]c1C 54323,c1(CNCC(CC(=O)N(CC(F)F)CCOCC)O)cnn(C)c1C#N 54324,C(CC(C)C)(C(=O)NCC(C(C)(C)C)NC(=O)CC(O)C1CCCC1)NC(C)=O 54325,C1(C(N(C(C)C(=O)NC(C)CC2CC2)CC)=O)CC2(CC2)CN1C 54326,N1(C(C(C)SCCCC)=O)CCC(CNC(=O)C(CO)OC)C1C 54327,N1(c2nc(C)c(C(F)(F)F)cc2)CCCC2(CCCO2)CC1 54328,C(CN=C(NCc1ncc(C)s1)N1CCC2(CCCOC2)C1)C1CC(OC)C1 54329,C(C1=CCN(C2CCC2)CC1)Oc1cncc(NC(C=CC(C)(C)SC)=O)c1 54330,C(=O)(C1CCCn2cnnc21)NC1(C)CCN(C(c2c(OC)cc(C)cn2)=O)C1 54331,C1(C(=O)NC2(CSC)CCC2)CC2CC2N1C(=O)CCc1nc(=N)[nH][nH]1 54332,Cc1nn(C)cc1C1CC1C(=O)NCCCNC(C1CC2CCC1O2)=O 54333,c1(C(N2C(CNC(CCc3c(C)n(C)nc3)=O)CC2)=O)nn(C)c2c1CCC2 54334,C(C(C)C)(C(O)C(=O)N1CCC(CF)(NC(=O)CN(CC(C)(C)C)C)C1)OC 54335,C1(C)(c2n(CC(F)(F)F)nc(CC3CC3)n2)CC(F)(F)C1(F)F 54336,C(=O)(C1=CC2CCC(C1)C2)N1CCC(C(=O)NCc2c(C)ccs2)C1C 54337,C1(C)(CN(C(C(C)NC(c2cc[nH]c2)=O)=O)C)CCCC1 54338,Cc1ncccc1C(=O)N(CCCNC(C12CC(O)C1C2)=O)C 54339,N12CC(C3CCCCC13)C2=O.C(=O)(C(O)CC1CC1N)NC(C)(C)C 54340,CC1=C(CNC(=O)C(c2ccns2)NC(=O)OC(C)(C)C)S(=O)(=O)CCO1 54341,S(=O)(=O)(c1c(Cl)cc(Br)cc1Cl)N1CC(C)(C(=O)Nc2cc(Cl)cc(Cl)c2F)C1 54342,C12CC(C)(C1)NC2=O.C(=O)(C(N)=O)NCCCN(C)C 54343,N1(C(c2c(F)ccc(F)c2Cl)=O)CC23CCCC2(C1)CN(c1ncc(Br)cn1)C3 54344,C1(c2n(C)cnc2)CCN(S(=O)(=O)N2CC=CCCC2(C)C)CC1 54345,c1(C(=O)NCC2N(C(C(C(=O)OC)C)=O)CC(C)(C)C2)cccc2c1cnn2C 54346,C1(C)(CNC(CNC(c2ccccc2)C)=O)CC(C#N)C1 54347,c1(NC(C(=O)NC(CC=C)CO)=O)ccc(OC(F)(F)F)c(Cl)c1 54348,C(=O)(CC(CC)C(C)(C)C)N1CCC(N(C(=O)CCc2ccc(O)nc2)CC)C1 54349,C(=O)(C(C)(C)C(N)=O)N1CCC(CN(C(c2c(NC)cncc2)=O)C)C1 54350,CCC(C)C(C)C(=O)NC1(C)CC(NC(c2cnn(CCO)c2N)=O)C1 54351,N1(C(C(C)OCC)=O)CCC2CN(C(=O)C=Cc3cnccn3)CCC12 54352,c1(C(=O)OC)cccc(C(=O)NCC(C)(C)CNC(=O)CCF)c1C 54353,c1(SCC(=O)NCC2(NC(C(CC)N(C)C)=O)CCCC2)ccc(C)cc1 54354,CCC(C)(C)CCCC(=O)N1CC(NC(c2cnc(S)[nH]2)=O)C2(CC2)C1 54355,C1(n2nc(C(N(CC(C)CNC(=O)CCF)C)=O)c(O)c2)CCC(F)(F)CC1 54356,c1(CCNC(c2nnnn2CC)CCOCC=C)c(C)cc(Br)cc1C 54357,CCC(CNC(=O)CCN1CCCS1(=O)=O)(CC)NC(=O)Cc1cnco1 54358,CC(CNC(c1ccccc1O)=O)C(F)C(=O)NCc1c(F)cncc1F 54359,N1(C(C2C(C)(C)C2)=O)CC2CCC(CNC(c3n[nH]c4c3CCC4)=O)C2C1 54360,CS(=O)(=O)CCC(=O)NC1CCN(C(c2csc(-c3cccnc3)n2)=O)C12CC2 54361,n1(Cc2nc(-c3scc(C)n3)nn2C(C2CCOCC2)C)cccc(C)c1=O 54362,CCCCCC(F)C(=O)NCC(c1ccccc1)NC(C12CC(C)(C1)OC2C)=O 54363,CC1(C)CC(CCNC(=O)C(CC2CC2)NC(c2cncnc2)=O)CO1 54364,C1(C(=O)NCC2(NC(=O)Cn3cc(Br)cn3)CC2)CCC(=O)N2CCCC12 54365,Cc1coc2ccc(C(=O)N(CC(C)NC(c3cc(Cl)cc(F)c3F)=O)C)cc12 54366,c1(CC(C2CCCC2)OC)nnc(SCC2COCCO2)n1CC(C)C 54367,N1(C(C2(C)CCN(C(c3cc(C)oc3C)=O)C2)=O)CCCC2C(O)CC12 54368,Cc1[nH]c2ncccc2c1C(=O)NCC1CN(C(=O)CCC2CCOC2)CCO1 54369,C1(CCOC)(NC(=O)C(C)Cc2cnco2)CCN(C(=O)CSS(C)(=O)=O)CC1 54370,C1(C(N2C(CNC(C3(C(C)C)CCNC3=O)=O)CCC2)=O)CS(=O)(=O)CC(=O)N1 54371,c1(C(N2CC(F)CC(NC(C(C)c3ccco3)=O)C2)=O)c(N)c(F)cc(F)c1F 54372,C(C(C)C)(C(O)C(=O)NC1CC(N(C(=O)CCc2cc(C)no2)C)C1)OC 54373,N1(C(c2c[nH]c(=N)o2)=O)CC(NC(=O)CCCC2CCOCC2)C2(CC2)C1 54374,C1(C)(C(N(CC=C)CCOC)=O)CN(C(C2CCC(C(N)=O)C2)=O)CC1C 54375,n1(CCC)nnnc1C(c1cc(C)[nH]n1)NCCc1cnoc1 54376,CC(CNC(=O)COCC1CC1)C(=O)NC(CO)CCC1CC1 54377,C1(C(=O)OC)C2CCC(C2)C1NC(C)COC(C)(C)C 54378,CCC(CC(=O)N1CC(=CCNC(=O)NC)OC(C)C1)C(F)F 54379,CCCC(CC)C(=O)N1CC2CC2(NC(c2cc(C(C)(C)C)c[nH]2)=O)C1 54380,C1(NC(CCSC)=O)CCN(C(c2ccc(CF)cc2)=O)CC1C 54381,C(=O)(C(CCCC(C)(F)F)N(C)CC1(NC(=O)OC(C)(C)C)CCOCC1)NC 54382,C(=O)(CN=c1cc[nH]cc1)N1C(C(=O)NCC2N(C(C)=O)CCC2)CCCC1 54383,C(=O)(C(C)C(=O)NC(C)CC(=O)Nc1cncnc1O)OC 54384,C(=O)(C1CNC(=O)c2ccccc21)N1C(CNC(C2(C(C)C)COC2)=O)CCC1 54385,C(=O)(CCCCCS(N)(=O)=O)NC1C(NC(c2ccnc(OC)n2)=O)CCC1 54386,C1(CNC(CN(c2nccs2)C)=O)CN(C(c2ccc(F)cn2)=O)C2CCN1C2 54387,c1(C(N2CC(CNC(CNc3nccc(OC)n3)=O)C2)=O)cc(C)cc(O)c1 54388,CC(CCCCCO)N=c1[nH]c(=NCC(F)CO)c2ccc(C(F)(F)F)cc2[nH]1 54389,c1(C(N2CC3C(CNC(C(CC)(C)O)=O)(C3)C2)=O)cc2cscc2s1 54390,Cc1c(N)c(C(=O)N(C)CCNC(=O)CN(C)C)cc(F)c1Br 54391,C(CCCCCF)NC(C1CC(NC(=O)CC2CCC2)C1)=O 54392,c1(C(C)C)ncc(Cl)c(C(=O)NCC2CCN(C(C3CCC3C(F)F)=O)CC2)n1 54393,N1(NC(c2ccc(COCC)o2)=O)CCC(Cc2cnc(O)c(OC)c2)C(C)C1 54394,C1(NC(C(C2CCCC2)NC(CC=C)=O)=O)CCCCCC1F 54395,C1(CNC(C(c2cc(C)sc2)(C)C)=O)CC2(C1)CN(C(C1(C)CC1(C)C)=O)C2 54396,C1(C(=O)NC2(CCCC(=O)NC(CCCCC)C)CCC2)CC(=O)CC(=O)N1 54397,C1(F)(C(=O)NC2C(SC)CN(C(=O)C=C3CCN(C)CC3)C2)CC2(CCC2)C1 54398,CC1CCN(CCC(=O)NC2CCCC(NC(C34CCC3CC4)=O)C2)CC1 54399,C(=O)(C(C)(C)C(=O)N1CCC(F)(CNC(C(C)OCC=C)=O)CC1)NCC 54400,Cc1cc(C(=O)N(C2C3CN(C(C4CN(C)CCO4)=O)CC23)C)c(Cl)cc1F 54401,CC1Cc2ccc(NC(=O)NCCOc3ccc(F)c(F)c3)cc2C1 54402,c1(C(N2CCC(NC(CCOc3ccc(C)cc3)=O)CC2)=O)cc(C#N)cn1C 54403,C1(C(N2CCN(C)C(=O)C2)=O)CC(C)(C)CCN1C(C1CN2CCC1CC2)=O 54404,N1(C(CCCN)=O)CCC(=CC(N2CCC2CO)=O)CC1 54405,N1(C(C(C)N(C(C)=O)C)=O)CC2(CCN(C(c3cn(C)c(=O)cn3)=O)C2)C1 54406,C1(CC=C)(NC(c2c(C)noc2C)=O)CCN(C(=O)COCCCOCC=C)C1 54407,c1(C(C)=O)cnc[nH]c1=NCC1CC2(CC(NC(=O)COCC3CCCO3)C2)C1 54408,N1(C(C(CCCC)O)=O)CCC12CCCN(C(=O)C(=C)CC)C2 54409,C1(=O)N(CCOCC(=O)NCC(C)O)CCN1.C(CO)OCC 54410,c1(SCC(=O)NCC2N(C(C(COC)(C)OC)=O)CCC2)cc(Cl)ccc1Cl 54411,CCC(C)C(O)CNC(C1(CNC(=O)CCOC2CCC2)CCCC1)=O 54412,N12CCOC(C1)CCCNC1(CC1)C2=O.C1(OC)CN(C(=O)COC(C)C)C1 54413,CC(C)CC(CC(C)C)C(=O)NCCC1CC(NC(c2cn(C)nn2)=O)C1 54414,c1(C(=O)NCCNC(c2c(C)cc(C)cc2O)=O)sc2[nH]c(C)nc(=O)c2c1C 54415,CC1(C(=O)NCCCC2CCCN2C(c2cnc[nH]2)=O)CCCC1(F)F 54416,C1(C(C)C)(C(=O)NCC2CC2CNC(c2coc(CO)c2)=O)CCCO1 54417,c1(CCC)onc(C)c1C(=O)NCC(CCOC)NC(C1(C(C)(C)O)CCC1)=O 54418,C1(CC(=O)NC(C)CCNC(=O)CCc2ccccn2)CCCCC12CC2 54419,Cc1[nH]nc2c1CC(C(N1CCCC(F)(CNC(=O)C(C)(C)C(F)F)C1)=O)CC2 54420,N1(C(CN2CC(C)(OC)C2)=O)CC=C(C(=O)NCC2CCN(C(C)=O)C2)CC1 54421,c1(C(=O)NCC(O)CCNC(C2(N(C)C)CC2)=O)cccc2[nH]ccc12 54422,c1(C(=O)NCC(C(C)C)NC(C2C(C=C)CC2)=O)cccc(S(N)(=O)=O)c1F 54423,N1(C(c2cnc[nH]2)=O)CC(C2CCN(C(C3CCCN(C(N)=O)C3)=O)CC2)C1 54424,c1(OC)csc(C(=O)NCC2COC(CNC(c3cccnn3)=O)C2)c1 54425,CC#CCCCC(=O)NC(CNC(c1nnsc1C(F)F)=O)CC(C)C 54426,c1(C(N2C(C(=O)NC(c3cscn3)C)CCOCC2)=O)cccn2ccnc12 54427,N1(C(C2CCC(C)(C)C2)=O)CCc2[nH]nc(CNC(C3CCOC3)=O)c2C1 54428,CC1CCc2onc(C(=O)NCCN(C)CCNC(=O)C3CC3)c2C1 54429,c1(OC)cc(OC)nc(NC(CC2N(C(C3CCN(C)C(=O)C3)=O)CC2)=O)n1 54430,c1(C(CC(=O)NC2C(CNC(CCCc3onc(C)n3)=O)C2)O)cccc(F)c1 54431,N1(C(C(C)c2ccco2)=O)CCOC(CNC(C2CC2(C)Br)=O)C1 54432,Cc1nn(C)c2c(NCCCn3ccnc3C)nc(=NC3CCCOC3)[nH]c12 54433,c1(OC)cncc(C(N2CC(CCNC(=O)C(=O)N(C)C)C(C)C2)=O)n1 54434,C(=O)(CC(C=C)CCC)NCC1CCCC(NC(CSCC#C)=O)C1 54435,C1(C(=O)Nc2c(C)ccnc2)CN(C(c2cccc(Cl)c2I)=O)CC(F)(F)C1 54436,C1(OCC#C)CCCN(C(=NCC(C2CCCC2)N(C)C)NC(C)C2CC2)C1 54437,c1(CC(=O)CN2CCCCC2C(N2CC3(CCC3)C2)=O)ccccc1Br 54438,N1(C(=O)Cc2ccccn2)CCCC(CO)(NC(C2CC3C=CC2O3)=O)C1 54439,c1(N(c2ccccc2)C(=O)NC(c2ccccc2)CF)ccnc(C(F)(F)F)c1 54440,Cc1[nH]c(C)c(C(=O)NCC(C)(C2CC2)NC(=O)CCC(=O)NC2CCCC2)c1C 54441,N1(C(C(CCCC)F)=O)CCC2(CC(C(=O)N(C3CC(C(N)=O)C3)C)C2)C1 54442,N1(C(C(C=C)O)=O)CCCN(CCNC(=O)C(C)c2cncs2)CC1 54443,C1(C(N(Cc2ccccn2)C)=O)CCCN(C(=O)OC)C1.C(c1cnc(C)s1)=CC 54444,CCCC(CCC)CC(=O)N(C1CC2CC1N(C(c1ccc(F)c(C)c1)=O)C2)C 54445,N12CC(CC(O)C1)NC(=O)NCC2=O.N1(C2(C(=O)NCCCC)CC2)CCCC1 54446,C1(C(N2CCC(N(C(C(F)=CCC)=O)CC)C2)=O)Cc2nn(C)cc2C(=O)N1 54447,c1(C(=O)NC2CCC(NC(=O)CCN3CCCC3=O)C2)n[nH]c2c1CCSC2 54448,c1(N2CCC(=CC)C2)cc(C)c(S(=O)(=O)N2CCOC(c3ccccc3)C2)cn1 54449,C1(CNC(CN(CCOC)C)=O)(NC(=O)C(C)CO)Cc2ccccc2C1 54450,CC(C)CC(CNC(=O)CC1CC2(CCC2)C1)NC(=O)CCc1cccc(Cl)c1 54451,N1(C(C2CC(C)(C)C2)=O)CCN(C(C2CCC(C(F)(F)F)CC2)=O)CC(O)C1 54452,N1(CC(c2ccccc2)NC(=O)NCCC(CC)O)CCSC(C)(C)C1 54453,Cc1cccc(CCC(=O)NCC=CCNC(C2CCCN(C)C2)=O)c1 54454,N1(C(c2cn(CC(C)C)nc2)=O)CCC(N(C(=O)CN2CC=CC2)C)C(C)C1 54455,N1(CCN(C(c2ccc(C(=O)OC)o2)=O)C2CC2)CC(N(C)C)C2(CC2)C1 54456,CC(C)C(CNC(C1(C)CC(C)(C)C1)=O)C(=O)N1CC(C)(F)C1 54457,c1(CC(CNC(C2CCC(n3cccc3)CC2)=O)CO)cccc(NC(N)=O)c1 54458,c1(C(c2nnnn2CCCSCC)NCCC(CC)C)nc(C)[nH]c1Br 54459,Cc1cc(C(N2CCCC(C(=O)NCCn3cnc(C)c3C)CC2)=O)c(C)cn1 54460,n1(C(C)C)ncc2c1CC(NC(=O)NC1CCCC1C(N)=O)CC2 54461,c1(C(=O)NC(CC)CNC(=O)CC(O)CN(C)C)cc(C(C)C)nc(O)c1 54462,C1(NC(C(C2(O)CCC2)NC(C=C(C)C)=O)=O)COC(C(F)F)C1 54463,N1(C(c2n[nH]c(CC)c2Cl)=O)CC(C)C(NC(=O)CN(S(=O)(=O)CC)C)C(C)C1 54464,C1(C(=O)NCC(C)N(C)C)CC1C1CN(C(C2CCCN2C2CC2)=O)C1 54465,c1(-c2n(C)cnc2)cccc(F)c1C(N1CC(NC(c2ccno2)=O)CC(F)C1)=O 54466,CCC(C)C(O)C(C)C(=O)N1CC(OC)CC1C(=O)NCc1ccc(F)c(Cl)c1 54467,C1(C(=O)NCc2cccs2)(CC)CCN(C(=O)CC2CC3(CCC3)C2)C1 54468,C(CCC)(C(=O)N1CCCC1C(N1CCCC1CCCC)=O)=CCC 54469,c1(CNC(CC2CC(OC)C2)=O)nc(CNC(=O)CC2CC(C)C2)cc(O)n1 54470,C1(CCC(=O)NC2CN(C(C(N)=O)=O)C2)CCC(=O)NC1 54471,c1(NCCCCc2onc(-c3ccc(C)cn3)n2)cc(N(C)C)nc(C)n1 54472,c1(-c2ccnc(N(C)Cc3n(CC)ccn3)n2)ccc(O)c(C)c1C 54473,c1(NCC2C(C)CN(C(=O)C(F)(F)c3cscn3)CC2)ncnc2c1cnn2C 54474,C#CCC(C(=O)NCc1nn(C)cc1Cl)NC(=O)CCCCN(C)C 54475,Cc1nc2ccc(CN3CC4(CC4C(=O)Nc4nc5c(s4)COCC5)C3)cc2[nH]1 54476,c1(CC(=O)NCC(C)NC(c2ccc(C(C)=O)cc2)=O)c(C)[nH]c2ccccc12 54477,c1(C(N(C)CC2(O)CCN(C(C3CC(O)C3)=O)C2)=O)ccc(Cl)c2cccnc12 54478,N1(C(c2cnc(CC)[nH]2)=O)CC(NC(=O)CC2CC(C)(C)CO2)C2(CCCC2)C1 54479,c1(C(=O)NCC(CNC(c2cnccn2)=O)O)ccn2ccccc12 54480,C1(C(N2CCC(N(C)C(C3CCOC(=O)N3)=O)CC2)=O)CCC2C(C1)C2(F)F 54481,C1(c2ccn(C)n2)CCCN(C(c2cnc(-c3cccc(CO)c3)cn2)=O)C1 54482,CCC(CC)CC(F)C(=O)NC1C2CC3C1C3C2C(N1CC2(CCC(O)CC2)C1)=O 54483,C(C(C)(O)CC(=O)NCC=CCN(C(c1ocnc1-c1ccccc1)=O)CC)OC 54484,C1(C(=O)NCC2(COC)CN(C(C3CC=CC3)=O)C2)CNC(=O)CC1C 54485,N1(C(c2c(C)ccc(O)c2)=O)CCC2CN(C(C3CC3(F)F)=O)CC2C1 54486,N1(C(CC(C=C)C)=O)C2CCC1CC(O)(CNC(=O)CC1=CCCC1)C2 54487,c1(C(N(CCCNC(C2(C)CC2Br)=O)CC)=O)c[nH]cc1COC 54488,C1(CC)(CNC(C2CN(C(=O)CCCC3CCCC3)CCO2)=O)CCOCC1 54489,c1(CC(=O)NCC(C)(C)NC(C2CCC(C(=O)OC)C2)=O)cc(F)ccc1OC 54490,CC1(C)CN(C(=O)C(c2cscn2)NC(=O)OC(C)(C)C)Cc2ccccc21 54491,c1(OC)ccc(CC(=O)NC2CCN(c3nccnc3C)CC2)cc1 54492,C1(CC(=O)NCC2CN(C(c3c(C)snc3)=O)CC2C)CC(C)CC(C)(C)C1 54493,Cc1ccc(S(=O)(=O)NCC(N2CC3(C2)CN(C(C2CNC(=O)N2)=O)C3)=O)cc1 54494,C1(CC)CN(C(C2CCN(C)CC2)=O)CCN1C(=O)C=CCOC 54495,C1(c2nnnn2CC(F)F)(Sc2ccc(C)cc2)CCC1C1CCC1.CCO 54496,C12(C(N3CC(C)C(NC(c4cnn[nH]4)=O)C3)=O)CCC(C1)C2(C)C 54497,c1(OC)cc(CC(N2CCC(CN(C)C(C3C(C)CC3C)=O)CC2)=O)ccn1 54498,C1(NC(c2cc(C)ncn2)=O)CC(C2CCN(C(c3cccc(C#N)c3)=O)C2)C1 54499,C1(CNC(C2(C#C)CCCC2)=O)COCC2(CCN(C(c3cn[nH]c3)=O)CC2)O1 54500,C12(CCN(CC(=O)NCCCN(c3cnccn3)C)C)CCCN(CC1)C2.C 54501,C1(NC(CCOCC)=O)CC2C1CCN2C(c1ccc(C(C)(C)C)c(Cl)c1)=O 54502,N1(C(c2c(CC)cc[nH]2)=O)C(C(=O)NC(c2snnc2C)C)CCC1C1CC1 54503,CON=CC(=O)NCC(O)CCNC(c1cncnc1)=O 54504,C1(C(=O)NCC2N(C(=O)Cn3nccc3C)CC(OC)C2)CC1C1CC(F)(F)C1 54505,c1(C(N2C(CNC(CC=C)=O)C3CCC2C3)=O)cc(C)cc(OC)c1C 54506,c1(NC(=O)NC2(C)CCCN2Cc2sccc2C(=O)O)c(Cl)cc(Cl)cc1Cl 54507,C1(C(=O)Nc2ccc(CNC(=O)CCCCC3CC3)cc2)(NC(N)=O)CCCCC1 54508,N1(Cc2cc(CC)no2)CCC(C(C)C(=O)NC2CCOC2)CC1 54509,CC1(C)CC(=O)NCC1C(=O)NC1CC(NC(=O)CN2CCOC2=O)C1 54510,c1(C(=O)NCC(C)NC(C2(c3ccccc3)CC2(F)F)=O)cc2cccn2cn1 54511,C(C(CO)CC(C)C)NC(C1(C)N(C(c2cc(C)sc2N)=O)CCC1)=O 54512,Cc1nc(NC(C)(CNC(C2(CC3CC3)CCCO2)=O)C2CC2)cc2nncn12 54513,C1(CNC(=O)CCc2cccs2)CCCN(C(C2CCC(F)(F)CO2)=O)CC1 54514,c1(OCC(N2C(N(CC#C)C(=O)OC(C)(C)C)CC2)=O)ccc(Br)cn1 54515,c1(C(=O)NCC(CN(C(=O)CC2COC(=O)N2)C)(C)C)cn2ccccc2n1 54516,N1(C(c2ncoc2Br)=O)CC2CCN(C(c3cnn(CCF)c3)=O)C2C1 54517,Cc1cc[nH]c1Cc1cn(C2CCCC2C(=O)NOC(=O)C2=CCC2)nn1 54518,c1(CC)ccc(C(N2CCC(CNC(=O)CN3CCCC3=O)C(C)C2)=O)cc1N 54519,Cc1nc(NC(C2CCCC2)CC2CN(C(=O)C(C(C)C)NC(N)=O)C2)[nH]c1C 54520,S(=O)(=O)(c1cccc(S(C)(=O)=O)c1)Nc1c(C(=O)NCC(C)OC)cccc1 54521,C1(C)(CC)CC(NC(c2c(OC)cccc2O)=O)CN1C(c1cnoc1C)=O 54522,N1(C(c2c(C)c(N)ccc2)=O)CCCC(C2CCCN(C(C3CCCO3)=O)C2)C1 54523,C12(NC(c3cc4occc4s3)=O)CCCN(C(=O)Cc3ccoc3)CC1C2 54524,c1(-c2ccc(CNC(c3nccnc3Cl)=O)cn2)cnc2sccc2c1 54525,CC1COC2(CCC2)CN1C(=O)CSCCNC(=O)CC(O)CN(C)C 54526,c1(C(N2CC3CC(NC(c4cc(C(C)=O)on4)=O)C3C2)=O)cc2oc(Cl)cc2[nH]1 54527,C(=O)(C1=COCCO1)N1CCC(F)(CNC(c2cc(C)ncn2)=O)C1 54528,C1(C2CC2)(C(N(CC(C)NC(c2cc(C(N)=O)[nH]n2)=O)C)=O)CC=CC1 54529,c1(N2CC(N(C)Cc3ccc(C#N)cc3)C2)ncc(I)nc1Cl 54530,CS(=O)(=O)CCC(=O)NCC1(O)CCCN(C(=O)CC2CCCS2(=O)=O)C1 54531,N#CC1(NC(c2ccc(I)cc2O)=O)CCN(C(c2ccc(Cl)nc2Cl)=O)C1 54532,c1(C(=O)NC(CCCCNC(C2(c3cc(C)no3)CC2)=O)C)occ2c1CCC2 54533,Cn1ncc2nc(O)c(C(=O)NC(CNC(C3NC(=O)OC3(C)C)=O)CO)cc12 54534,CC(C)(CCC(=O)NCC1CCN1C(c1ccc(F)c2[nH]ccc12)=O)[N+](=O)[O-] 54535,CC1CCN(C(c2sccc2C2CC2)=O)CC1NC(c1nscc1N)=O 54536,c1(C(=O)OC)cc([N+](=O)[O-])cc(S(=O)(=O)NC2(CN)C3CCCOC3C2(C)C)c1 54537,c1(N(CC(N2CC(C(C)NC(=O)C(C)C3CCCC3)C2)=O)C)ccncc1 54538,C(C(C(=O)NCCC(C)O)C(C)(C)C)NC(c1ncc(CC)cn1)=O 54539,C(CC1CCCC1)(C(=O)NCc1n[nH]c(C)n1)NC(C(c1ccn(C)n1)C)=O 54540,C(=O)(C(F)C(C)CC(C)(C)C)N1C(C)CN(C(C2C(OC)CCCC2)=O)C(C)C1 54541,C(=O)(C1CCc2cccnc21)N(CC(C)NC(=O)C(C(C)C)n1cnnc1)CC 54542,N1(C2c3cnc(s3)C(C)NC2=O)CC2C(C(N)=O)C2C1.c1(CC)ccc(Cl)cn1 54543,N1(C(C23OCC(C(C)C)(C2)C3)=O)CCN(c2ccc(C(=O)O)cn2)C(C)C1 54544,c1(C(N2CCC=C(Br)C2)C(=O)NCC)cccc(C(=O)OC(C)(C)C)n1 54545,C1(C(N2CC(CC(C)C)OCC2)=O)CC2CCCC2N1C(=O)C(F)C(C)C 54546,c1(C(=O)NC(CNC(Cc2nnc(C)s2)=O)C(C)C)c(Cl)cnn1C 54547,c1(CC)cc(C(=O)NCC(C2CC2)NC(=O)CCCC2OCCO2)ccn1 54548,c1(C(=O)NCC(CC=C)NC(=O)Cn2ccccc2=O)cc[nH]c(=NCC)c1 54549,C(CC(=O)NC)(C(F)(F)F)Oc1c(C)ccc(C(=O)NCC2CC(OCC)C2)c1 54550,c1(CC(=O)N(CC(C)NC(c2n(COC)ncc2)=O)C)cccc([N+](=O)[O-])c1C 54551,C1(C(=O)NCC=CCNC(C2(c3cccs3)C(C)C2)=O)CCC(F)(F)CC1 54552,C=Cc1cncc(C(C(=O)NCC2CCCO2)N(c2cccc(C)c2Br)C)c1 54553,C=Cc1ccc(C(N2CC(CNC(=O)Cn3nnc(-c4ccsc4)n3)C2)=O)cc1 54554,c1(N2CC(OC)(CNC(=O)CCc3nc(C)cs3)C2)cc(=O)n(C(C)C)c(O)n1 54555,C(COC(C)C)(C(=O)NCC1(CCNC(C2CCCCS2)=O)CC1)NC(C)=O 54556,c1(NC(c2cccc(OCC)c2)(c2ccccc2)C2CC2)ccc(S(N)(=O)=O)cc1 54557,c1(OCC)nc(Cl)ccc1C(=O)NC1CCCN(C(C2CC3(CCC3O)C2)=O)C1 54558,CC1CC(C(=O)Nc2ncccc2CO)N(C(=O)CO)C1 54559,C12(C(N(CC(C)NC(C3CN(CCC)C(=O)C3)=O)C)=O)CCOC(C)(C1)C2 54560,C(=O)(CCCCC(=O)N1CCC(NC(=O)CCn2nc(C)c(C)c2C)C1)NC 54561,c1(C(N2CCC(CNC(c3n(C=C)nnc3)=O)C2)=O)cc(Br)ccc1O 54562,N1(C(=O)CC2CC2(Cl)Cl)Cc2ccccc2C(Nc2ncc([N+](=O)[O-])cc2Br)C1 54563,n1(C(C)C)cnc(N)c1.C1(C(N2CC(OCC=O)C2)=O)CCC(CO)C1 54564,C=CCC(C(=O)N(CCCNC(c1cc(F)ccc1C(F)(F)F)=O)CC)C(C)C 54565,Cc1ccc(C(N2CC(NC(c3ccsn3)=O)C(O)C2)=O)cc1O 54566,Cc1cccc(C(=O)NCC2CC(NC(C3(C#N)CC3)=O)CC2O)c1Br 54567,N1(C(c2ccoc2Cl)=O)CCC2(CC1)CCN(C(C1(CC3CC3)CC1)=O)C2 54568,c1(OC)ccc(Cl)c(Cl)c1C(=O)NCC1CCN1C(C1CC1c1ccco1)=O 54569,O=C(C#CC1CC1)NCC1CC(F)CN1C(C1CCC1Cc1ccc(Cl)cc1)=O 54570,C1(C)(C(c2n(CCC(=O)OC)nnn2)NCCNC(C)=O)CCC(C)(C)CC1 54571,N1(C(CC2CCN(C)C2)=O)CCN(C(c2cnoc2-c2cccs2)=O)CC(O)C1 54572,N1(CC(C)C)CCC(C(=O)NCC2CCCC2NC(=O)C2=CCOC2)CC1 54573,C(=O)(C(C)CS(C)=O)NCC1(OC)CN(C(=O)Cc2cnoc2)C1 54574,N1(C(c2ccc(OC)cc2)=O)CCC(F)C(NC(c2cccnc2OC)=O)C1 54575,C(CC1=CCN(C(C2CCOC2C)=O)CC1)NC(c1cc(C)sc1)=O 54576,C=C1CON(C(=O)C2CC(NC(c3cnn(C)n3)=O)CCO2)C1 54577,O=C(N=c1ccn(CCCO)[nH]1)C1CC2(CC2)CN1C(=O)CC1CS(=O)(=O)C1 54578,c1(C(=O)NCC2(NC(=O)COc3ccncc3)CC2)cnn(C2CC2)c1Cl 54579,C1(NC(=O)CCc2cccs2)CC2(C1)CC2NC(=O)CCCn1cccc1 54580,C(C(=O)NC(CC(=O)NCCCc1ncc[nH]1)C1CC1)(C(C)C)N(CC)CC 54581,c1(C(=O)NC2C(NC(C(C)(C)SC)=O)CCC2)cc2c(C(C)C)nn(C)c2s1 54582,c1(SCC(=O)N(CC(C)CNC(C2CCNC2=O)=O)C)ccc([N+](=O)[O-])cc1 54583,N1(C(C(CC(F)F)NC(C(CC2CCC2)OC)=O)=O)CCC(F)(F)C(F)C1 54584,C1(C(N2CC(OCC#C)C2)=O)CC(=C)CCN1C(=O)OCC.C1(=O)CO1 54585,N1(C(CN(CCC)C)=O)CCOCC1CN(C(=O)C(F)C(C)C)C 54586,S1(=O)(=O)c2cccnc2N1.CC1C(C)N(C)CCN1CCCCN(C)C 54587,c1(OC)cnc(OC)c(C(=O)NNC(=O)C2CC2(Br)Br)c1 54588,CCC(C#N)C(=O)N1CCC(C(=O)N(CCCCCO)C)(OC)C1 54589,c1(CC)ccc(C(=O)NC2CC(N(C(=O)C=C(C)C)C)C2)c(F)c1 54590,C1(NC(c2onc(C)n2)C2CCOCC2)CCn2nnnc2C1 54591,C1(C(N(C2CCN(C(c3c(Cl)cn(CC)n3)=O)C2)CCO)=O)CC12CCCCC2 54592,c1(C(=O)NC(C)(C)CCNC(=O)CC2(O)CCOC2)cc2ccncc2cc1F 54593,CC1(C)CCC(C(=O)NC2(CO)CC2)CN1C(C1CN(C2COC2)C1)=O 54594,c1(NC(CC)CC(C)CO)ccc(S(=O)(=O)NCc2csc(C)c2C)cc1C#N 54595,C1(COC)CN(C(=O)CC2CCC(=O)NC2)CCN1C(c1nocc1C)=O 54596,C1(NC(C2CN(C(N)=O)C2)=O)CN(C(c2ccc3n[nH]cc3n2)=O)CC2(CC2)C1 54597,N1(C(c2n(CC)cc(Cl)c2)=O)CCC2(COC)CCCC12 54598,C1(NC(c2cnc(OCC)s2)c2nnnn2CCCF)CCCCC1OC 54599,O=S(=O)(c1ccc(=NCC2(C3=CCOCC3)CC2)[nH]c1)N1CCC(OCCO)C1 54600,C12(NC(C3CCC4CC34)=O)CC(C(=O)N(CCn3ccc(CO)c3)C3CC3)(C1)C2 54601,C1(CNC(c2c(CC)[nH]cc2)=O)CC2(CCC2)CN1C(=O)CC1(CSC)CC1 54602,C(=O)(CS(=O)(=O)NC(N)=O)NC1(CN(C(C2(CCC=C)CC2)=O)C)CC1 54603,C(=O)(C(C#N)C(C)(C)C)NC(C(NOC(C)C)=O)Cn1cccn1 54604,c1(C(=O)NCC(CNC(C2(S(N)(=O)=O)CC2)=O)OC)ccc2c(c1)NCCC2=O 54605,C1(C)(C(=O)NCCC2(CO)CN(C(c3c(C)oc(CO)c3)=O)C2)CCCS1(=O)=O 54606,N1(C(c2cn(CCC)nc2)=O)CC2CCC(NC(c3oc(C)nc3C)=O)CC2C1 54607,N1(C(c2ccc(C(N)=O)o2)=O)CCOCC1Cc1cccnc1 54608,C1(COC)CC(CNC(C2CCC(C)O2)=O)N(C(c2[nH]c(O)nc2C)=O)C1 54609,C1(F)(C(=O)NCC2C(NC(C=NOC)=O)C2)CCCOC1 54610,CC1C(O)CC2CCC1N2C(c1cccc(N(C)NC(C2CCCS2)=O)c1)C 54611,c1(C(=O)OC)cc(C)nn1CC(=O)NC(C)CC(C)NC(=O)C(C)CC1CC1 54612,c1(C(=O)NCC2N(C(Cn3c(C)cnc3)=O)CCOC2)ccc(Cl)cc1Br 54613,c1(C(=O)NCC2N(C(C3N(C(N)=O)CC(O)C3)=O)CCC2)ccc(N)cc1Cl 54614,CON(C(=O)CCC1CCCN1C(C1C(C)(C)C1(F)F)=O)C1CCC1 54615,CCC(CC)(CO)C(=O)NC1CCN(C(=O)C(c2ccc(F)cc2)C)CC1 54616,C(C(C)C)(C(O)C(=O)N1CC(C(C(=O)NCC2CCOC2=O)OC)C1)OC 54617,C1(OC(C)C)CCN(C(=O)C(CC2CC2)NC(=O)CC2CN(C(C)=O)C2)CC1 54618,C(C(C)(C)C(=O)NC1CCCC1CC(=O)NOC(c1ccncc1)C)N(C)C 54619,c1(C(N(CCCNC(C(CCC#C)O)=O)C)=O)cc(F)c(F)c(Cl)c1F 54620,Cn1ncc(NCc2cccnc2P(C)(C)=O)c(Cl)c1=O 54621,c1(C2(c3nnc(CN4CCC(O)C4)o3)CC2)ccc(Cl)cc1 54622,c1(C(=O)NC(CNC(CCC(C)OCC)=O)CO)cc(=O)n(C)cc1Br 54623,C1(C(N2C(CC(=O)OC(C)(C)C)CC(OC)C2)=O)CC2(CCCCC2)N1C(C)=O 54624,C1(COCC)CCN(C(c2nonc2C)C(=O)NCc2ccccc2)C1 54625,N1(C(=O)NCc2ccn(C(C)C)n2)CCN(C2CCCOC2)CC1 54626,N1(C(Cc2ccc(C)s2)=O)CC=CCC1C(N1CCCC1CCO)=O 54627,N1(C(c2ccc(CC)s2)=O)CCCC2CN(C(=O)Cc3ccc(C)c(C)c3)CC12 54628,c1(C(C)C(N2CCC(N3CCN(c4ccncn4)CC3)C2)=O)ccccc1Cl 54629,c1(-c2nc(C3(O)CN(C(c4c(C)nco4)=O)C3)on2)ccc(F)cc1 54630,c1(CCN=C(NCC2CCC(C)C2)NCc2ccccc2)c[nH]c2ccccc12 54631,C1(CNC(=O)Cc2nc(C(C3(C(=O)NC)CC3)=O)n[nH]2)(CO)CC(OC)C1.C1CC1 54632,C1(CNC(C=C(CCC)C)=O)CCCCC1NC(=O)C(C)(C)C1(O)CCOC1 54633,c1(OC)cc(C(N2CC3(CC(NC(=O)CC4CCC5CC5C4)C3)C2)=O)cc(F)c1 54634,C(C(C)C(F)C(=O)NCC1CC(C)C1)NC(c1c(C)cc[nH]1)=O 54635,C(=O)(C(CC)(CC)CC)NC1C(C(=O)NC(CCC=C)C(=O)OC)CCC1 54636,N1(C(c2n(CC)ccc2)=O)CCCC(C)(NC(=O)Cc2ccc(OC)cc2C)C1 54637,c1(-n2ccc(C(=O)NCC3C(NC(C4(SC)CCC4)=O)C3)n2)cnccc1C 54638,c1(C(=O)NCC2C(C)CN(C(=O)Cc3csc(Cl)c3)C2)cc(Cl)cc(F)c1N 54639,CC1(C(N2CC(CCNC(=O)C#CC3CCOC3)C2)=O)CCCCC1(F)F 54640,N1(C(C(CCSC)O)=O)CCOCC(C(=O)NCCC(=O)N(C)C)C1 54641,C(c1cccc(Cl)c1)=CC(=O)NCC1CCC(NC(c2cn(C)[nH]c2=N)=O)C1 54642,C1(NC(=O)C=CCN2CCC2)COCCC1C(=O)NCc1ncc(CO)o1 54643,n1(CC(N2CC3C(C(=O)OCC)C(CC3)C2)=O)cc(C#N)ccc1=O 54644,c1(C(=O)NC2CN(C(CCCOCC)=O)C2)ccc2ccc(Br)cc2n1 54645,N1(C(C2(C(=O)O)CCC(F)(F)CC2)=O)CCN(C2=NCCCN2)CC1 54646,C(C)(CCC(=O)N1CCC(C)(CCNC(c2cc(F)n(C)n2)=O)C1)SC 54647,C#CCCCC(C)C(=O)NCC(C(C)C)NC(=O)Cc1cccc(SC)c1 54648,C1(C(=O)NC2CC23CCN(C(c2cc(F)c[nH]2)=O)C3)CC12CCCCCC2 54649,N1(Cc2n(CC)ccn2)C(=O)NC2(CCCCC2)C1=O 54650,C(=O)(NNC(=O)C(C)Sc1cn2c(COC)cccc2n1)c1ccc(OC)cc1 54651,C1(SC)CN(C(C2CCC(N(C)C)CC2)=O)CC1NC(C1CC(C)(O)C1)=O 54652,C1(NC(CCc2ccc(OC)c(OC)c2)=O)CCNC12CCOCC2 54653,N1(C(C(CSC)C)=O)CCC(C)(CNC(c2c(C)coc2-c2ccccc2)=O)C1 54654,C(=O)(CN=c1cc[nH]cc1)N1C(CNC(C2C(C)(C)OCC2)=O)CCC1 54655,CC(C)C(O)C(C)C(=O)N(C1CC(c2ccc(F)cc2)C1)C.n12cc(nn1)CC2 54656,CC1(O)COCCN(C(c2cc(CNC(=O)C(c3ccccc3)F)no2)=O)C1 54657,N1(C(CCC#CC)=O)CC(NC(C2(OC)CCOC2)=O)C(C2CC2)C1 54658,N1(C(C(CC#C)C2CC2)=O)CC2CC1CN2C(=O)CN(C)CCO 54659,Cc1[nH]nc(Cl)c1C(=O)NC1CN(C(c2cnn(C(C)(C)C)c2C)=O)C1 54660,Cc1c([N+](=O)[O-])c(C(N2CC(NC(=O)C(=O)N(C)C)CC3(CC3)C2)=O)nn1C 54661,C1(CNC(=O)CCc2ccccn2)C(C2CC2)CCN1C(=O)Cn1cccn1 54662,c1(NC(=O)NCC(CNC(=O)OC(C)(C)C)OC)ccc(OC)c(C)c1 54663,C(=O)(C(=O)NNc1cc(C)c(Cl)cn1)NC1CC(C(=O)OC)OC1 54664,C1(CC(C)NC(C)CC2CCCO2)CCN(C(=O)OC(C)(C)C)C1 54665,C1(C2CC2)(CNC(CC2C(C)(C)C2)=O)CCN(C(c2nccnc2N)=O)C1 54666,N1(C(c2ccc(N)c(C)c2C)=O)CCN(C(C23CCCCC2C3)=O)CC(C)(C)C1 54667,C(C(CC(=O)N1CCCC1CN(C)C)NC(=O)C(C)CCN(C)C)OC 54668,N1(C(c2cc(CCC)c(C)s2)=O)CC(NC(=O)CCNC(C)=O)C(C)(C)C1 54669,C1(c2cn(CC3CCN3C(C3CN(C4COC4)C3)=O)nn2)(OC)CCCC1 54670,N1(C(C(CCC)CC)=O)CCCC2(C1)CN(C(C1(CCO)CC1)=O)C2 54671,C1(NC(C(CSC)O)=O)CC2CCC1CN(C(C1(F)CCCCC1)=O)C2 54672,c1(C(=O)NCC(CC)NC(=O)CCOCC2CCC2)cnoc1C(C)C 54673,N1(C(CCCN(C(C2ON=C(C(C)C)C2)=O)CCO)=O)CCCN(C=O)CC1 54674,O=C1NC2(CCO1)CN(C(=O)C(c1ccoc1)NC(C1CCC=CCCC1)=O)C2 54675,C1(C)(C(=O)NC2(CC)CC2)CC(O)CN1C(=O)C(CC1CCC1)OC 54676,CN1CCCC(O)(CNC(=O)NC2CCCCN(Cc3ccc(F)cn3)C2)C1=O 54677,C(=O)(C(C)(F)C(=O)OC)N1CC(C)(NC(C(CC=CCC)C)=O)C1 54678,C1(NC(C2(SC)CC2)=O)CN(C(c2n[nH]c(C)c2Br)c2ccccc2)CC1C 54679,C(=O)(C(CO)C(C)(C)C)N(CCC(C)(C)NC(C(c1ccccc1)OCC)=O)C 54680,c1(N2CC(O)(CCNC(C(CCC)C)=O)C2)ncc(C)c(SCC)n1 54681,Cc1sc(C(N2CCC(CC3(O)CC3)CC2)=O)c(Br)c1C 54682,c1(C(C(=O)NC2(CCNC(COCCOC)=O)CC2)(C)C)cc(OC)cc(F)c1 54683,c1(C(C)C)nccc(C(=O)NC(c2cccc(Cl)c2)CNC(C2CC2C)=O)n1 54684,NS(=O)(=O)c1ccc(C(N2CCN(C(C3CC(F)C3)=O)CC2CC2CC2)=O)nc1 54685,c1(CN2CCCC(C(=O)Nc3cccc(O)c3Cl)C2)c(O)ccc2ccccc12 54686,c1(SC)nc(C(=O)N(CCCN(C)C(C2CC(F)CN2C)=O)C)c2ccccn12 54687,c1(C(N2C(C(C)NC(C3(C)CCC(=O)N3)=O)CCC2)=O)cc2nc[nH]c2cn1 54688,N1(C(C(F)OC)=O)CCC(NC(c2ccccc2N2CCCCC2)=O)C(C)C1 54689,C(C(C(=O)NC1CC(N(C)C(c2cnn(C)c2CC)=O)C1)C(C)(C)C)OCC=C 54690,N(C1CCCc2c(Br)cccc21)C(N1CC2(C(F)(F)F)CCC2(CO)C1)=O 54691,CC1(C)CCCC(C(=O)NCCCc2cn(C3CCCC=C3Br)nn2)C1 54692,c1(OCOC)cc(-c2cnc(C(F)(F)F)cc2C)ccc1OC 54693,N1(C(c2cc(C)sc2)=O)CCN(C(c2cc(C3CC3)ns2)=O)CC1CCO 54694,C12(OC)CCC(NC(=O)CC3CCN(C(=O)C(F)=CC4CC4)CC3)(CC1)C2 54695,C(=O)(CCC(=O)C1CC1)NC(C(C)NC(c1n[nH]cc1CN(C)C)=O)CO 54696,c1(C(N(CC(N2CCN(C(C(C)C(C)O)=O)CC2)=O)C)=O)cc(F)c(Cl)cc1Cl 54697,C1(NC(C2(SC)CCC2)=O)CCCC(CC(=O)NC23CC(C)(C2)C3)C1 54698,c1(CC)cncc(C(=O)NCCCCNC(=O)Cc2ccnc(Br)c2)c1 54699,c1(NCC(N2CC(c3c(CNC(C(CSC)O)=O)nco3)C2)=O)ccc(O)cc1 54700,c1(C(CNC2N(C(=O)OC(C)(C)C)CSC2)(C)O)ccc2ccccc2c1 54701,N1(C(c2cc(C)sn2)=O)CCC2(CCN(C(c3cc(F)c4cn[nH]c4c3)=O)C2)C1 54702,c1(C(=O)NC(CNC(COCC=C)=O)C)ncc(C)cc1C 54703,c1(N(CCNC(=O)CC(C)C2CCCCC2)CC)ncnc(Cl)c1Br 54704,N1(C(c2c(C)cccn2)=O)CCCC(N(C)C(C2COC(=O)N2C)=O)CC1 54705,N1(Cc2ccn(CC)n2)CCC(NC(=O)CCC(=O)N2CCCC2)CC(C)(C)C1 54706,C12(C(N3C(C(C)NC(Cc4nc(C)oc4)=O)CCC3)=O)CCC(F)(CC1)C2 54707,C1(C(=O)NCC(N(C(=O)CO)C)C2CC2)C2CC3C(C2)C13 54708,c1(NC(C)=O)sc(Cl)cc1C(=O)NCCCNC(=O)CCC1CCCOC1 54709,C1(NCc2cnn(C)c2Cl)COC2(CCN(C(c3cnnn3C)=O)CC2)C1 54710,C1(CN(C)CCC2C(CC)CCCC2)CC12CCOCC2 54711,n1(CC=C)nnnc1C(c1csc(Br)n1)NC(c1nnc(CO)s1)C 54712,c1(CC(N2CCN(C(c3cc(C)c(N)cn3)=O)CC2)=O)ccc(S(N)(=O)=O)cc1 54713,O(NC(=O)C(C)NC(c1scnc1C)=O)C(CC)CC 54714,C1(F)CC(CNC=O)C1.C1(C(C)(C)C)(C2CC2)CCCO1.C12CCC1C(=O)NC2 54715,Cc1nc(NC(C)Cn2cnnc2)cc(NC(C2CCC(F)(F)CC2)C)n1 54716,C#CCCCCC(C)C(=O)N1CCC(C(=O)NC2CC2)(CF)C1.C1CO1 54717,S(=O)(=O)(c1ccc(NCCCCn2cnnc2)cc1Br)N(CCCC(=O)NC)C 54718,N1(CC(N2C(CCNC(CCC=CC)=O)CCC2)=O)C(C)CCC1C 54719,CC1(C)C(CN)CN1c1nc(-c2ccccc2Cl)no1 54720,C1(C(=O)NC(C)(C)CS(C)(=O)=O)CN(C(=O)CC2CCC(=O)NC2)CC12CC2 54721,CC1(C(=O)NCC2CCN(C(=O)CCCc3ccccc3Br)C2)CC(F)(F)C1 54722,Cc1c(N2CCOCC2)ncnc1N1CCC(NC2COCC2C)CC1 54723,C1(NC(C2CC2c2c(OC)cccc2OC)=O)CCCN(C(C)=O)C1C 54724,C1(C(=O)NCCOCC(NOCC)=O)(NC(c2ccc[nH]2)=O)CCCCC1 54725,c1(NC(C(CCOC)NC(=O)C=CC(=O)N(C)C)=O)cn(CC)nc1C#N 54726,c1(C(N2CC(CNC(c3cc(C)ns3)=O)C2)=O)c(C)ccnc1O 54727,c1(C(N2CCC(CO)C2)C(=O)OC)cccc(Cl)c1F 54728,S(=O)(=O)(CCC(=O)NCC1C=CC(NC(=O)C(c2ccccc2)F)C1)NC 54729,c1(CNC(c2c(CC)cc[nH]2)=O)ccc2c(c1)CCN(C(C1C=CCC1)=O)C2 54730,c1(NC(C2CC2C(N2C3COCC2C3)=O)=O)cnc(I)cn1 54731,N1(CCC)CCCC(C(=O)NC(C)CCNC(c2cc(CC)no2)=O)C1 54732,C(N=c1[nH]c(=NC2CCCC(F)(F)C2)c2ccccc2[nH]1)c1nc(C)c(C)[nH]1 54733,c1(C(=O)NCCC2N(C(CCC#CC)=O)CCC2)ccc2c(c1)OCCO2 54734,Cc1nc([N+](=O)[O-])cn1CC(=O)NC1CC2CCC1CC2NC(=O)C=CS(C)=O 54735,c1(C(=O)NCC(C(C)(C)C)NC(c2ccc(F)c(N)c2)=O)cc2c(s1)CCCC2 54736,Cc1cn2c(CC(N3CCC(CNC(C4(C)C(C)(C)C4(C)C)=O)C3)=O)csc2n1 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54753,c1(OC)c(F)cc(C(=O)NC(C)(C)C(C)NC(=O)CC2CC=CCC2)c(N)c1F 54754,c1(C(N2CCC3CN(C(=O)COc4ccsn4)CC32)=O)coc2c1C(=O)CCC2 54755,c1(C(N2CCC(C(C)NC(c3cc(CCO)on3)=O)CC2)=O)ccc(O)cc1Cl 54756,C1(C(N(C2CCCC(C)(C)C2)C)=O)CN(C(=O)C(F)n2ccnc2)CC(C)(C)C1 54757,N1(C(CCN(C(CCC(C)CN(C)C)=O)CC2CC2)=O)CCOCC(C)(O)C1 54758,CCC(C(=O)N1CCC(NC(C2CCCN2CC)=O)C1(C)C)C(C)(F)F 54759,C(N=c1[nH]c(N2CCCC3(CC2)CC3)nc2cc[nH]c12)C1(F)CC1 54760,C(C1CCCN1C(=O)C(c1ccccc1)C)=CC(=O)N(C1C(C)CC1)C 54761,c1(OC(CC)C)ccc(CN2CC(C(=O)O)C(C(=O)O)C2)cc1Cl 54762,C1(C(=O)NCCN(C(=O)C(F)CSc2ccc(F)cc2)CC)CC2CCCC(C1)C2 54763,N1(C(C2C(C)CCO2)=O)CCC(F)(C(=O)NC2(C)CCCC2O)C1 54764,Cn1cc(C=CC(=O)Nc2ccnn2CC(F)F)cn1 54765,C1(CNC(c2ccc(F)cn2)=O)C(C2CC2)CCN1C(=O)COCC1CCC1 54766,c1(C(=O)NC2CCC(N(C(CC3CN(CCC)C3)=O)C)C2)cc(OC)nc(Cl)c1 54767,C(C1c2ccsc2CCN1C(=O)C(C)OCC=C)NC(CCCCCCC=C)=O 54768,C1(CC)(CC)CCC(NC(C2(CC(C)C)CCNC2=O)=O)CC1 54769,C1(CC(C(=O)OCC)F)CCCN(CC(c2ccsn2)=O)C1 54770,Cc1c(C(=O)NCC2(CNC(C3CCCC(=O)N3C)=O)CC2)[nH]c2ccccc12 54771,C(=O)(C1=NOC(C)C1C)NC1CC(CNC(Cc2c(C)nc(S)s2)=O)C1 54772,C1(CNC(C(C)CC2CCC2)=O)CCN(C(C23C(=O)C4CC2C3C4)=O)C1(C)C 54773,C1(C(N2CC(O)(C(C)C(=O)NC3CCCC(F)(F)C3)C2)=O)CCC(C)(C)CC1 54774,c1(C(N2CCC(N(CCC)C(C3CCC3OC)=O)CC2)=O)cc2sc(C)cc2[nH]1 54775,c1(CNC(C(CNC(=O)CCc2nc[nH]n2)OC)=O)ccc(CO)cn1 54776,C(CC(=O)NC1CCCOC1)(C(F)F)NC(=O)CC1CC2(CCC2)C1 54777,Cc1csc(CC(=O)NCCOC2CCN(C(=O)CCc3ccon3)C2)c1 54778,N1(C(C2CC(=C)C2)=O)CCC(C(=O)NC2CC(C(C)(C)O)C2)(CC)C1 54779,C(=O)(CCCCC(C)CC)N(C1CN(C(Cc2cc(CC)c(OC)cc2)=O)C1)C 54780,c1(C(=O)NCC(CN(C(=O)CN2CCCC2)C)O)cc2sc(Cl)cc2s1 54781,c1(C(N2CCCC(CNC(C(CC)CN(C)C)=O)C2)=O)ccc(C)nc1C 54782,c1(C(N2CC(N(C)Cc3ccc(O)cc3)C2)=O)cc(Cl)cc(Cl)c1O 54783,c1(C(=O)NCCNC(C=C(CCC)C)=O)ccnn1C(C)C 54784,c1(-c2cn(-c3ccc(CC(C)C(=O)NC(N)=O)cc3)nn2)cc(F)ccc1Cl 54785,CC1(CNC(C2(CNC(=O)CC34CCCC3C4)CC2)=O)CCCCC1O 54786,c1(C)nnc(O)cc1O.N1(C(CC2CCC(SC)CC2)=O)CCN(NC)C2CC12 54787,Cc1c(C(N2CC3(CCC3NC(C3C4CCCOC34)=O)C2)=O)cccc1C1CC1 54788,C1(C)(C(=O)NC(COC)CO)CN(C(=O)CC2C(C)(C)C2(C)C)C(C)(C)C1 54789,CCC(CC(=O)NCc1cc(C(=O)NCCNC(=O)NC)n(C)n1)N(C)C 54790,CC(C)(C)CC(O)CC(=O)NC1CC2(C1)CC2C(=O)NC1(C(O)CO)CC1 54791,CCC(CC)(C(=O)NC1CCC(CNC(c2ccc(=O)n(CC)n2)=O)CC1)OC 54792,C1(CNC(CC=CC=C)=O)(CO)CCCN(C(=O)C(F)C2CCOC2)C1 54793,C1(NC(c2c(CNC(c3cnco3)=O)nco2)=O)CCCCCC1 54794,C1(CCC(N2C(CNC(c3c(C)coc3)=O)CCC2)=O)CCCCN1C 54795,CCC(C#N)C(=O)N1CC(F)CC1CNC(=O)C(C)(C)c1cccnc1 54796,N1(C(=O)CCOCC(F)F)CCC2(C1)CN(C(=O)C(c1ccccc1)O)CCO2 54797,n1(C(C)(C)C)cc(C(=O)NC2CCC(CNC(=O)Cc3cc[nH]c3)C2)nn1 54798,N1(C(Cc2n(C)ccn2)=O)CCC2CN(C(C3OCC4CCCCC34)=O)C2C1 54799,Cc1cc(C(=O)NC2CCOCC2NC(=O)CCCn2cncn2)ncc1C#N 54800,N1(C(Cc2nccc(OC)n2)=O)CCOCC(CNC(=O)CCC2CC2(F)F)C1 54801,CCC(C)(CC)C(=O)NC(C1CCN(C(c2cc(C(C)(C)C)n[nH]2)=O)C1)C 54802,C1(NC(N2CC(COC)OC(C)(C)C2)=O)CCc2cc(OC)ccc2C1 54803,CCC(CCC(=O)N(CCC(=O)NC1CCN(C(C)C)CC1)C1CC1)OC 54804,c1(CC)cc(C(=O)NC(c2ccccc2)C(=O)NC2CCCC2C(C)C)on1 54805,C1(C(=O)NC2CCCN(CCC)C2)CCCCN(C(=O)C2=CCOCC2)C1 54806,N1(C(CCc2ccc(C)nc2)=O)CCC2(CC(NC(C3(C)CCOCC3)=O)C2)C1 54807,c1(CC)nn(C)cc1CN(C(C)C(=O)NC)C 54808,N1(CCCNC(C23CC(C2)C3)=O)CCN(C(c2ncoc2C2CCCO2)=O)CC1 54809,C1(NC(c2cnc(C(C)(C)C)s2)=O)CC(F)(F)CC1NC(=O)C1=CCSC1 54810,Cc1cc(C(=O)NC2CCOC(C(=O)NCc3ccccc3CO)C2)n(C)n1 54811,O(NC(=O)CCCN(C(=O)C(C)CN(C)C)CCOC)C(C=C)C 54812,c1(C(=O)NC2(CCCNC(CC(CC)OC)=O)CC2)c(C)cccc1Cl 54813,N1(C(C(CCC#C)O)=O)CCC(CCNC(c2sc(C)nc2C)=O)C(F)(F)CC1 54814,N1(C(C(C(=O)NC)(C)C)=O)CCN(C(=O)CCNC(C2CCCO2)=O)CC(O)C1 54815,CCCC(CC)CC(=O)N1CCN(C(c2c[nH]nc2-c2cccnc2)=O)CC1C 54816,C1(O)(C2CC2)CCCN(C(=O)C=CC(C)(C)N(c2nc3sccn3c2C)CC)C1 54817,C(N=c1nc2c(cnn2C)c(NCC(C)(F)F)[nH]1)C1(C(C)C)CC1 54818,N1(C(C2C(CC)CCO2)=O)CC(S(=O)(=O)N2CCN(C(C3CC3(F)F)=O)CC2)C1 54819,c1(CNC(C2(CC(=O)OC(C)(C)C)CCCCC2)=O)ccc2c(c1)CCCNC2 54820,N12CCCC(CC1)C2=O.N1(C(C(C)NC(=O)OC)=O)CC2CC2(CO)C1 54821,N1(C(c2nc(CC)[nH]n2)=O)CCC(C2CCCCN2C(C2CCSC2)=O)CC1 54822,c1(C(=O)NC2CC(F)(CNC(C3CC(C)N(C)C3)=O)C2)cccc(S(N)(=O)=O)c1 54823,Cc1c(C(=O)N(CC(C)NC(=O)COc2ccc(OC)cc2)C)cc(O)cc1N 54824,C1(C(=O)NCC2N(C(CN(C)C)=O)CC2)CCCC(=O)N1 54825,C1(C(=O)NC2CC2CNC(=O)C=CC2CCCC2)(COC)CC=CC1 54826,C1(N(C(Cn2cc(-c3cccc(C)n3)nn2)=O)C)CCCCC1(C)C 54827,C1(CC(=O)N(C2CCCN(C(CC(=C)C)=O)C2)CC)OCCOC1(C)C 54828,N1(CCNC(CCC2CCC(NC(c3ccn(C)c3)=O)C2)=O)CCCC(O)C1 54829,c1(C(=O)NCC23OCC(CNC(C(CC)(F)F)=O)(C2)C3)cc2ccccn2c1 54830,C(CNC(=O)Cc1csc(Cl)c1)(C(C)C(C)C)NC(c1cnc(C)[nH]1)=O 54831,C1(=O)CCCC(C(=O)O)N1.c1(OC)ccccc1COC(C)C 54832,c1(OCC)cccc2c(NC(=O)NC3CCC(SC)CC3)c([N+](=O)[O-])cnc12 54833,N1(CC(=O)NC2C=CCCC2C(N2CC3CC2(C(F)F)C3)=O)C(=O)CNC1=O 54834,C1(NC(C2(CC)CCC2)=O)C(C)(C)C(NC(c2ccc(O)c(C)c2C)=O)C1(C)C 54835,C(C)(CC(C)NC(c1cncs1)=O)NC(CN(C(COC)=O)C)=O 54836,C1(NC(C(COC)(C)C)=O)CCN(C(c2cccc(CCN(C)C)c2)=O)C(C)C1 54837,C=C(C)CC(C(=O)NC(c1cccnc1O)C)NC(=O)CCn1ccc(C)n1 54838,Cc1nsc(N)c1NC(=O)NC1CC=CCC1C(F)(F)F 54839,C1(NC(C(=Cc2cn[nH]c2)C)=O)CC(C)N(C(c2nnsc2N)=O)C1 54840,Fc1ccsc1C(c1nnnn1C1CCC1)NCCc1ccn(C(F)F)n1 54841,N1(C(CCc2c(C)noc2)=O)CCCC(CCC(=O)NCCCC(C)(C)C)C1 54842,c1(NCC(c2ccccc2Cl)C)nc(N2CCN(CCO)C(C)C2)nc2sccc12 54843,c1(C(=O)NCC2OCCN(C(COCC=C)=O)C2)cc2ccsc2c(O)n1 54844,CC(C(=O)NC1CC(CCNC(c2ccn(C3CC3(F)F)n2)=O)C1)C(F)F 54845,N1(C(C2N(C)CCC2)=O)CCCC2C1CCN2C(c1cc(Cl)ccc1[N+](=O)[O-])=O 54846,c1(NC)cc(Cl)ccc1C(=O)NC(C)CNC(=O)C(c1cc(F)cc(F)c1)O 54847,C1(CC(N2C(CC)CN(C(c3nc(C)sc3C)=O)CC2)=O)NC(=O)CN(C)C1=O 54848,N1(C(c2c(CC)nccn2)=O)CCCN(C(=O)C(O)Cn2cncn2)C(C)C1 54849,CCCC(C)(CCC)C(=O)NC1CCCCN(C(=O)C#CC(C)C)C1 54850,C(N=c1[nH]c(C)nc2[nH]ccc12)C1CC2(CC(NC(C3(C=C)CCC3)=O)C2)C1 54851,CCC(CC(=O)N1CCC(CNC(=O)CCn2ccnc2C)C1)C1CCC1 54852,C(=O)(CCCC(F)F)N1CC(CC(C)NC(c2cn(C(C)C)nc2)=O)C1 54853,C(CC1=CCN(C(=O)CCCF)CC1)NC(c1n(OC)cnc1C)=O 54854,C1(C(=O)Nc2scc(-c3ccc(OCC)cc3)n2)C2CCCCCN12 54855,CC1(C)CC(CNC(c2cnc(=N)[nH]c2)=O)N(C(=O)C(N)=O)C1 54856,C1(C(=O)NCCc2n(C)cnn2)CC2(CCC2)CN1C(C1CCSC1)=O 54857,C(=O)(C#CC1CCC1)NCC(c1cc(F)cc(Cl)c1)NC(C(CC)=CC)=O 54858,C1(NC(CC=C=C)=O)CN(C(c2nn(C)cc2C)=O)CC1C(F)(F)F 54859,N1(C(CN(c2ncccn2)C)=O)CCCC1C1CCCN1C(c1ccc(F)s1)=O 54860,N1(C(C23CC(NC(CC4CC(=C)C4)=O)(C2)C3)=O)CC(C)CC(C)(C)C1 54861,CCC(C)(C(=O)NC1CC(C)N(C(=O)C(=O)NOC)C1)c1ccccc1 54862,Cc1onc(CO)c1C(=O)N(CCCn1cc(CCc2ccccc2)nn1)C 54863,C1(NC(CC(C(F)F)NC(C=CC(C)C)=O)=O)CCn2ncnc2C1 54864,c1(OCC(=O)NC2(CNC(CN(c3ccoc3Cl)C)=O)CCC2)ccc(O)cc1 54865,c1(C(=O)NC(C(=O)NCCC(CCC)C2CC2)c2ccoc2)oc(C)nc1CC 54866,c1(C(=O)OC)cccc([N+](=O)[O-])c1N(C1CCNCC12CC2)CCCOC(C)C 54867,C1(C(N2CCC(N(C(Cc3ncc(CC)[nH]3)=O)C)CC2)=O)CCCCNC1=O 54868,O=S(=O)(c1nc(N2CCOC3(CCCCC3)C2)ccc1Br)NC1(CO)CC1 54869,C1(NC(=O)CC2CCCC3CC23)(CO)CCCN(C(C2CC3CC(=O)C2O3)=O)C1 54870,c1(CC(=O)OCCC(=O)N(CC(C)N(C(C)C)CC)C2CC2)cn(C)nn1.CC 54871,C1(COCCCC)(CN(C)C)CCN(C(C2CC(C)=NO2)=O)C1.C(CCC(=O)NC)OC 54872,N1(C(C(C)SCCCC)=O)CC2CC(NC(=O)CCc3ccncc3)CC1C2 54873,c1(-c2c(C)csc2)cccc(NC(=O)NCc2ccccc2Cl)c1 54874,C12(NC(CC3(C=C)CN(C(C4CC(N(C)C)C4)=O)C3)=O)CCC(CC1)C2(C)C 54875,C1(C(N(CCNC(=O)CN(C)C)CC)=O)CC(=O)C1C 54876,Cn1cc(C(c2nnnn2C)NC(c2cnn(CC(F)F)c2)C2CCC2)cn1 54877,C1(NC(c2c(C)cco2)=O)CC2CCC1CN2C(C1CCC(C)CC1)=O 54878,c1(CC(=O)N(CC(C)NC(COCCC)=O)CC)ccc(Br)nc1 54879,c1(C(N2CC(F)(C(N3CC4(C3)CN(C3CC3)C4)=O)C2)=O)cc(Br)c2ccccc2n1 54880,C(=O)(C1CN(C)C(=O)c2ccccc21)NC(C)CNC(=O)C=CCF 54881,c1(C(=O)NCC(C2CCC2)NC(C2N(CC)CC2)=O)cnccc1C(F)(F)F 54882,C1(C2CCN(C(c3ccc(S(C)(=O)=O)o3)=O)C2)(NC(CC(C)F)=O)CC1 54883,C1(NC(C(C=C)(C)CC)=O)CC2CN(C(=O)C(CCC)C(C)C)CC2C1 54884,CC1CN(C(c2cccc(C3CC3)c2)=O)CCC1CNC(=O)CC1(C#N)CCC1 54885,CN1CCCN(S(=O)(=O)CCNC2CC3CCC2N3S(=O)(=O)C2CC2)CC1 54886,C(CNC(c1c(C)n[nH]c1C)=O)(C(C)(C)C)NC(C(C)OCC=C)=O 54887,C12(C(N(CCN(C(=O)CCC3CCCCO3)CCC)CC)=O)CCC(OC)C1C2 54888,C(C(O)(C(F)(F)F)C1CCC1)NC(NC(CC)C(F)F)=NCc1ccnn1C 54889,N1(C(CCCC=C)=O)CCN(C(c2ccc(-c3ccccc3)[nH]2)=O)C(CCC)C1 54890,Cc1cccc(C(=O)NCC2(C)CCCN2C(=O)COc2ccccc2)c1F 54891,Cc1cc(C(=O)NCCCN2CCN(c3ccnc(Cl)c3)CC2)nnc1C 54892,c1(C(N2CCCCC(CNC(C3CC(C#C)(O)C3)=O)C2)=O)c(F)ccc(C)c1Cl 54893,C1(CC(C)C)CN(C(=O)CC(C)(C)C)CC1NC(=O)CC1C=NN(C)C1=O 54894,c1(OC)cc(C(=O)N(C2CCC(NC(c3[nH]ccc3C)=O)CC2)C)cc(F)n1 54895,CS(=O)(=O)c1cc(C(N2CCN(C(=O)C3=C(Cl)CC3)C(CCO)C2)=O)ccc1F 54896,c1(OC)c(Cl)cc(CN2CCC(O)C(C(=O)Nc3ncc(F)cc3Cl)C2)cc1Cl 54897,CCCC(CNC(C1(CC(=O)OC)CC1)=O)C(=O)NCc1nc(CO)n[nH]1 54898,c1(C(=O)NCC(CCCC)NC(=O)C(O)C(F)(F)F)ccc(C)c(C)n1 54899,C(=O)(CCC(N)C(=O)O)N1CCN(CC(=O)Nc2c(C)cccc2)CC1CCO 54900,c1(Cc2cn(C3CN(C(C)=O)OC3)nn2)ccc2c(c1)OC(C)C2 54901,c1(C(=O)NCC(N(C(CCOC(C)C)=O)C)C2CC2)cc(Br)c2cccnn12 54902,N1(C(c2ccn(CCCC)n2)=O)CCN(C(c2cnn3ccsc23)=O)C2CC12 54903,CC1(CNC(=O)CN2CC=CC2)CN(C(c2c(Cl)csc2Cl)=O)CCO1 54904,N1(C(c2cc(=N)[nH]cc2)=O)C(CNC(=O)CCc2cscn2)CC2COCC12 54905,C1(C2CN(C(=O)C(F)C3CCCC3)C2)(NC(=O)C(=Cc2cccc(F)c2)F)CC1 54906,C(N=C(NCC1CCCO1)N1CCC2(C1)OCc1ccccc12)c1cc(C)oc1 54907,c1(NCC(=O)Oc2cccc3[nH]ccc23)cc(F)c(N2CCCCC2)c(F)c1 54908,C1(C(=O)NCC(CCC)O)CC2CCC1N2C(=O)C(C(C)C)NC(C)=O 54909,C1(CC)(NC(c2nccn2C)=O)CCN(C(c2c[nH]nc2C)=O)CC1 54910,N(C1CCc2c(OC)cccc21)C(=O)NCc1c(C(=O)OC)sc2ccccc21 54911,CC(O)C(=O)NCC(O)CNC(=O)C(c1cccs1)N(C)C 54912,C1(CCC(=O)NC2C(C(=O)OCC)CC2)CCCN1C(=O)CCCN(C)C 54913,CCS(=O)c1ccccc1C(=O)NCCC1CCN(C(=O)C(C)(F)F)CC1(F)F 54914,C1(NC(Cc2cc(C)on2)=O)CCCC2CN(C(c3cccc(C#N)c3)=O)CC12 54915,Cn1nccc1C1OCCC1C(=O)NCC(C1CCC1)NC(C1CC(F)(F)C1)=O 54916,C(=O)(C(C)CON(C(N1CCCC1CCc1ccccc1)=O)C(C)C)OC 54917,C1(CC(=O)NCC(C)N(C(C(=O)NC(C)C)=O)C)CCC(C)(C)CC1 54918,N(C(=NCCC1(C)OCCO1)NCc1cnccc1Cl)CC1(OC)CCC1 54919,CCC1=C(C(=O)NC2(CNC(=O)C#CC3(C)CC3)CC2)SCCO1 54920,c1(NCc2cccc(NC(C3CN(C(CC)=O)C3)=O)c2)nc(O)c2ncnc-2[nH]1 54921,C1(NC(c2cn(CC(C)C)nc2)=O)CCCCCN(C(=O)CC(C)F)C1 54922,CC1(C(=O)NCC2(F)CN(C(C3CC3CF)=O)C2)CC(c2ccccc2Cl)=NO1 54923,CC1(F)CC2(CN(C(C3CC(F)(CF)C3)=O)C2)C1 54924,CCC(F)(F)CC(=O)NCC1CN(C(=O)C(c2ccccc2Cl)N(C)C)CC1C 54925,c1(C(=O)NC2CN(C(=O)COCCCF)CC2CO)c(O)cccc1F 54926,C1(OCC(=O)NC(C2CCCCN2C(=O)C2=CCSC2)C)CCCCC1C 54927,c1(C(=O)NCC(C)(C(C)C)NC(C(CCOC)C)=O)nc[nH]c2nccc1-2 54928,C1(C(=O)NC(C2N(C(C(C(C)C)F)=O)CCC2)(C)C)C2(CCC2)C12CCC2 54929,CCCCCCCCC(=O)NCC1(OC)CN(C(C2(n3cncn3)CC2)=O)C1 54930,C1(C(CNC(C2(OC)CCC2)=O)C)CCN(C(c2cncn2C(C)C)=O)CC1 54931,C1(NC(c2cnn(C)n2)=O)CCCCC12CCN(C(C1CCSC1)=O)CC2 54932,c1(NC(C(C(C)CNC(=O)CC2(C)CCC2)F)=O)cccc(N=[N+]=[N-])c1 54933,c1(Cn2cc(-c3cnc(OC)s3)nn2)cc2c(cn1)CCCC2 54934,C(=O)(CCC1CCc2ccccc21)NCCCn1cc(C(C(C)C)O)nn1 54935,N1(C(CCC(C)C)=O)CCCC(C)C1CNC(=O)CC1CCCCCCC1 54936,C(=O)(CCC(C)(C)NC(c1nccn1CCN)=O)NCCCc1cn(C)nc1 54937,C(=O)(C(CO)C(C)(C)C)N1CCCC(C(N2C(C)CC(CO)C2)=O)CC1 54938,c1(C(N(C)CC2C(NC(CCCN(C)C)=O)CCC2)=O)cc(O)cc(F)c1 54939,C1(NC(CCCCC=CC)=O)CCOC2(CCN(C(=O)CCCCC)CC2)C1 54940,Cc1ncc(C2CN(C(=O)CCCn3cc(CNC(=O)OC(C)(C)C)nn3)C2)o1 54941,N1(C(C2CCC3(CCC3)C2)=O)CCCC2(CCCN2C(=O)CC2CCCOC2)C1 54942,C1(N(C(C2(COC)CCCO2)=O)CC)CCCN(C(c2nc(Cl)sc2Cl)=O)C1 54943,Cc1cc(NC(C2CCCN2C(C2CCC(C)(C)C2)=O)=O)cc(O)c1 54944,C1(C(N2CC(CCNC(C(c3ccccc3Cl)C)=O)C2)=O)CCc2cnnn2C1 54945,n1(CCN(C(=O)NC2CC2)Cc2c(C)occ2)ccc2c(C)cccc12 54946,C(=O)(C1(C)OC(=O)c2ccccc21)NCCCNC1Cn2c(C)ncc2CC1 54947,C#CCCCCC(=O)N1CCC1C(N1CCCC(CCCO)C1)=O 54948,C(=O)(C(F)C(CC)CC)NC(CCC)C(=O)NCC(F)(F)C(F)F 54949,c1(CC(=O)NCC(C(C)C)NC(C23CCCC2C3(F)F)=O)cccc(Cl)c1F 54950,c1(SCCC(=O)N(C2CCN(C(C(CC)=CC)=O)C2)CC)cccc(Cl)c1 54951,Cc1c2cccc(NC(C3CC3C(=O)NCC3CCCOC3)=O)c2nn1C 54952,c1(C(=O)NCc2c(N3CC(C)OCC3)cccc2)cc(OC(F)(F)F)ccc1F 54953,CCCCC(O)C(=O)N(C1(C(=O)NCC(c2cccnc2)O)CC1)C 54954,c1(C(=O)NCCCNC(CC(C)SC)=O)ncc(Br)c(SC(C)(C)C)n1 54955,C1(CNC(CN(C2CCC2)C)=O)CC(NC(=O)C(C)(C)CF)CC1O 54956,O=C(CCCn1ccnn1)NC(C(=O)NC(CO)CCF)c1cccs1 54957,N1(C(CC(C)(C)N(C(c2nn(CC)c(C)c2)=O)C)=O)CCC2CCN(C)C2C1 54958,N(C(=NCC1CCCC12CC2)Nc1ccccc1Cl)CCNS(CC)(=O)=O 54959,N1(C(CCC2CCC(N(C(CC(=O)OC)=O)CC)C2)=O)CC(O)(C#C)C1.C#CCS 54960,c1(NC(N2CCC(C(=O)Nc3ncn(C)c3)C2)=O)c(C(F)(F)F)ccc(F)c1F 54961,c1(C(C)C(=O)NC(C)(CNC(=O)Cn2cncn2)CO)cccc(Cl)c1 54962,N1(C(C2C(C)=CCS2)=O)CCC2(CC2NC(C2CC2c2ccccc2)=O)C1 54963,N1(C(c2c(Cl)nc(N(C)C)s2)=O)CC2(CC(NC(C3CCC(F)(F)C3)=O)CO2)C1 54964,C1(NC(C2(CC)CCN(C(=O)CC3(COC)CC3)C2)=O)CCCCCC1C 54965,N1(N2CC(n3c(C(=O)OCC)ncn3)C2)CCC(CO)C2CCC12.C(=O)NC 54966,Cc1nc2ncc(C(=O)NCC3CCCN(C(C4CC4(Cl)Cl)=O)C3)c(=O)n2[nH]1 54967,c1(N2CCC(CCNC(CCNC(=O)C=CCl)=O)CC2)ccn2ccnc2n1 54968,C1(C)(CC)CCN(C(=O)CCN2CCC(NC(=O)C(N3CCOCC3)=O)CC2)C1 54969,c1(C(N2CCC(O)(CC(C)NC(COCCCC)=O)C2)=O)nc(Cl)c(=O)[nH]c1N 54970,CC(C)(F)C(=O)NCCCCNC(c1cc(-c2ccccc2)on1)=O 54971,c1(OC)cccc2c1CN(C(=NCCC1CCCS1(=O)=O)NC(C)C)CC2 54972,c1(C(N(CCNC(c2c(C#C)c[nH]n2)=O)CC)=O)cccc2c1ccn2CC#C 54973,c1(C(CC)C)cc(C(=O)NC2CC(NC(C3CCN(C)C3)=O)C2)on1 54974,n1(CCC)cc(C(N2CC(Cc3cn(-c4ccc(Cl)cc4)nn3)C2)=O)c(C)n1 54975,c1(NC(C2CCOC2)=O)cccc(CNC(=O)C(F)CC2CCOC2)c1 54976,Cc1nn(C)c(C)c1CC(=O)NCC1C(C)CCCN1C(c1cnco1)=O 54977,c1(C(=O)NCCN(C(=O)C(C)c2cc[nH]n2)CCOC)nc(O)sc1C 54978,C1(C(N(CCCN(C)C(c2nnn(C)n2)=O)C)=O)CC2CCC1CC2 54979,c1(CNC(CCCNCCN(C(c2cnnn2CC)=O)CC)=O)cccc(Cl)c1 54980,CC1C(OC(C)(C)C)CCCN1N(CCO)CCO 54981,Cc1sc(C)c2sc(C(=O)NC(CNC(C3CC4CCC3CC4)=O)C3CC3)cc12 54982,Cc1ccc(Br)nc1NC(C12CCC(NC(c3cnon3)=O)(CC1)CC2)=O 54983,n1(C(C)C(=O)N2CC(NC(C3C4COCC34)=O)C2)c(C2CC2)nc2ccccc12 54984,c1(CC)ccc(C(=O)NC2CCC2NC(=O)C#CC2(C)CC2)cc1[N+](=O)[O-] 54985,N1(C(=O)C=Cc2ccco2)CCCC(C2CN(C(=O)C3=CC4CCCC34)C2)C1 54986,N1(C(C)=O)C(C)CN(CC(=O)NC2CC3(C2)CC3(F)F)CC1C 54987,N1(CC(=O)NCC2(CN(C(=O)CN(C)S(N)(=O)=O)C)CC2)CCCCS1(=O)=O 54988,N1(C(c2ccc(SCC)nc2)=O)CCC(NC(C2(C(F)F)CC2)=O)C(C)C1 54989,N1(C(CN2CCC(=O)CC2)=O)CC(NC(=O)CCc2cnn[nH]2)C(C2CC2)C1 54990,C(=O)(C(C1CC1)OC)N(CC(=O)NC(C1CCOC1)CO)CCOC 54991,N1(CC(=O)NC2(C)CN(C(=O)CC3CCC(=O)O3)C2)CCC(F)(F)C1 54992,c1(C(C(=O)NCC2(CCNC(CN(CCC#C)C)=O)CC2)F)ccccc1 54993,c1(OC(CC(=O)NCCN(C(CC)=O)CC(C)O)C)cc(Cl)cc(Cl)c1 54994,N1(C(C(=O)NC(C)C)C2CC=CC2)CCOC2(CCCS(=O)(=O)C2)C1 54995,c1(CNC(N(CC(c2ccccc2)CC)C)=O)ccc2c(c1)OCC2 54996,c1(SCC(=O)N(CCCN(C(C2CN(S(CC)(=O)=O)C2)=O)C)C)ccccc1O 54997,CC(C)C(C(C)NC(=O)Cc1csc(-c2nc[nH]n2)n1)NC(=O)Cc1ccsc1 54998,N1(C(c2c(C(C)C)ccs2)=O)CC(NC(C2CN(C(N)=O)C2)=O)CC(F)C1 54999,C(=O)(C#CC1CCOC1)NC1C(NC(C2(OC)CCCC2)=O)CCC1 55000,C1(C)(CNC(C2C(C)CC2)=O)CCN(C(=O)C(O)C2CCC2)CC1 55001,N1(C(CC2(C)CCCC2)=O)CC(NC(C2CCS(=O)(=O)C2)=O)CC1CO 55002,c1(N2CC(CC)C(CC)C2)nc2ccc(OC(F)F)cc2c(=NC(C)C2CC2)[nH]1 55003,Cc1nc2ncnn2c(C)c1CC(N1CCC(NC(=O)C(C)(C)C(C)O)C1)=O 55004,c1(OC)ccc(C(=O)N(C)CCNC(c2csc3cncn23)=O)cc1C(C)(C)C 55005,c1(CNC(C(=O)NCC(CCCC)CCC)=O)nc2c(C(F)(F)F)cccc2s1 55006,c1(C(N2CC3C(NC(c4ccc(C(=O)OC)cn4)=O)(C3)C2)=O)cc(C)c(C)cn1 55007,C1(NC(COC(C)(C)C)=O)CC2COCC(C1)N2C(=O)C(O)C1CC1 55008,C(=O)(C1COc2ccc(Cl)cc21)N1CC(NC(CC2C(CC)C2)=O)C(C)CC1 55009,C(=O)(C(CO)C(F)(F)F)N1CCC(C(=O)NCc2ncc[nH]c2=O)(CC)C1 55010,c1(C(C)=O)c[nH]c(C(=O)NC(c2cn(C)nn2)C(=O)N(CCCF)C)c1 55011,N1(C(c2c(C)nco2)=O)CCC2(CCC2NC(C2CC23CCCCCC3)=O)CC1 55012,C(=O)(C(CC(F)F)C1CCC1)NCC(C)N(C(c1nc(OC)oc1)=O)C 55013,C1(NC(C(C(C)C)O)=O)CCN(C(=O)Cc2cn[nH]c2)CCC1CO 55014,c1(COC)nc(C(=O)NC2(CO)CN(C(=O)C(C)C3CCOC3)C2)co1 55015,C(=O)(C(O)CC(F)(F)F)N(CC)CC1CCCN(C(=O)CCn2cnnn2)C1 55016,C1(C(=O)NC2C(C(=O)NC(C3CC(O)C3)(C)C)CC2)CCCC1F 55017,N1(C(COC2CC(NC(C(CCCC#C)C)=O)C2)=O)CCN2C(=O)OCC2C1 55018,C1(NC(c2cc(C)c(C)o2)=O)CC2(C1)CC(CNC(=O)CC(C)(C)N(C)C)C2 55019,Cc1c(C(N2CCN(C(=O)CCc3ccoc3)C3CC23)=O)ccc2c1CCC2 55020,c1(C(=O)NCC(C(C)C)(C)NC(=O)C2=CCCS2)ccnc2ccc(N)cc12 55021,C1(CNC(c2c(C)onc2)=O)CN2CCCCC2CN1C(=O)C1=CCOCC1 55022,C1(NC(c2cc(C)oc2C)=O)CC(C)CN(C(C2(O)COC2)=O)C1 55023,c1(-c2c(F)ccc(C(=O)NC)c2)cnn2c1CN(Cc1cc(F)ccc1O)CC2 55024,Cc1c(CC(N2CC3CC3(CNC(C3CCCC3(C)C)=O)C2)=O)ncn1C 55025,c1(C(N2CCCC(N(C(C3C(C=C)OCC3)=O)C)C2)=O)cnc(CC)nc1O 55026,c1(CC)ccc(C(F)(F)C(N2CC(NC(c3cnc(O)n3C)=O)C(O)C2)=O)cc1 55027,C(=O)(C(C)(C)n1cc(Nc2ncnn2C2CCN(C(C)C)C2)cn1)OC 55028,C1(CC(=O)NCC(C)OCC)(CC2CCCC2)OCCO1 55029,N1(c2n(CC(C)(C)OCCC)nnn2)CCc2c(Cl)cccc2C1 55030,Cc1cccc(O)c1C(=O)NCC1(F)CC(CNC(=O)C=CCOC(C)(C)C)C1 55031,Cc1cc(C)c(S(=O)(=O)N2CCOC3CC23)cc1-c1ccc(C(C)C)cc1 55032,C=CCC(C)(C)CNC(=O)C(C(C)C)NC(=O)CC1COCC1O 55033,Cc1cccc(CC(=O)N(CCCNC(=O)C(C)Cn2cccn2)C2CC2)c1Cl 55034,C12(CC(N3C(C)CC(CNC(C4(F)CCC4)=O)C3)=O)CC3CC(CC(C3)C1)C2 55035,Cc1cc(N2CCCC(Oc3ccc(Cl)cn3)C2)ncc1[N+](=O)[O-] 55036,Cc1cc(Cl)cc(Cl)c1OCC(=O)N(C)CCNC(c1ncn(C)n1)=O 55037,C1(C(N2CCCC(NC(c3nc(CC)[nH]n3)=O)(CO)C2)=O)CCCCCS1(=O)=O 55038,c1(CC)ncc(S(=O)(=O)NCc2nc(CO)ns2)n1CC1CC1 55039,N1(C(C2OCC2(C)C)C(=O)NCC)CCC(C(=O)OC)C12CCC2 55040,c1(CNC2CCC(NC(c3c(CC)cccc3)=O)C2)cc(Br)cnc1C 55041,Cc1cnc2n1C(C(=O)N1CC(CO)(NC(c3cc(=O)cc(Cl)[nH]3)=O)C1)CCC2 55042,Cc1cc(C(N2CC(=C(F)CNC(c3ncccc3Cl)=O)C2)=O)c2c(c1)CCO2 55043,C1(C(=O)NCCCCC=C)CCC2(CC2)N1C(=O)Cc1n[nH]c(C)n1 55044,CCC(CC)C(F)C(=O)N1CCCC1CC(=O)N(C1CN(C(C)C)C1)C 55045,CCCC1C(=O)N2CC(C)(C2)O1.c1(CNC(=O)CSC)n[nH]c(O)n1 55046,C(=O)(CCC=O)NC.c1(OCC)ncc(C(N(C)CCOC2CC2(F)F)=O)cn1 55047,c1(NCC2CN(C(=O)Cc3csnn3)CC23CCC3)nc(Cl)nc2[nH]c(O)nc12 55048,N1(C(CC(C)CF)=O)CCCC(O)(CCNC(c2coc(CC3CC3)n2)=O)C1 55049,c1(C(=O)NCC(C2CCC2)NC(C2CCC(O)C2)=O)ccc2c(c1)OCCN2 55050,C1(O)(CCNC(c2ccn(C(C)C)n2)=O)CCN(C(C2CCCCC2F)=O)CC1 55051,CN1CC2CCN(C(C3CC(C)(NC(C4CC45CCC5)=O)C3)=O)CC2C1 55052,CC1(NC(=O)Cc2csc(-n3cccc3)n2)CC(NC(=O)CCSCC(N)=O)C1 55053,N1(C(CNC(C2CCC2)=O)=O)CCC2(CCN(C(C3CCSC3)=O)C2)C1 55054,N1(C(C(CN(C(C(C)(C2CC2)OC)=O)C)C)=O)CC2(CNC(=O)C2)C1 55055,c1(C(N(CC(CNC(Cc2nc(CC)sc2)=O)C)C)=O)cccc(NC(N)=O)c1 55056,C1(OCCC)CCCCC1C(=O)NCCCN1CCN(C(=O)CC(C)(F)F)CC1 55057,C1(C2(O)CCN(C(C3C4CCC(F)(F)C34)=O)CC2)(NC(C(P(C)(C)=O)O)=O)CC1 55058,CCCC(C(O)C(=O)NCC(C)(O)C(C)C)NC(c1ccc2c[nH]nc2c1)=O 55059,c1(OC)cc(C#N)ccc1CNCCC(C)(C)C(=O)NS(=O)(=O)CC1CC1 55060,Cc1ccc([N+](=O)[O-])cc1N1CCN(C2CC3CCC2C3)CC1 55061,Cc1cccc2ncc(-c3noc(-c4sccc4Cl)n3)n12 55062,C1(C(=O)NCCCCSC)CCC(NC(=O)Cc2ccc(Br)cn2)CO1 55063,c1(C(=O)OC2CCN(S(C)(=O)=O)C2)ccnc(Cl)c1Br 55064,Nc1ccc(C(=O)NC(Cc2ccccc2)CCNC(=O)CSCCO)cc1F 55065,C(=O)(CCC(C)(C)C#N)N1C(CNC(c2cnc(SC)s2)=O)CCCC1 55066,C12(C(=O)NCCN(C(C(CC)(C)CC)=O)C)CCCCN1CCC2 55067,c1(C(N(C(C)CNC(C2(COC)CCC2)=O)CC)=O)nc[nH]c1C(F)(F)F 55068,C12(CNC(C3(C)CC=CCC3)=O)CCC(CNC(C3CC(F)(F)C3)=O)(CC1)CO2 55069,N1(C(CSCCC)=O)CC2CCC(C1)N2C(=O)C=Cc1ccc(OC)c(C)c1 55070,C1(C(=O)NCC(C)CNC(=O)C(C)(C(F)F)c2ccccc2)CN2CCN1CC2 55071,CN1CCCC1CCCNC(C1(CC(F)F)CCNC1)=O 55072,N1(C(C(C)=C(C)C)=O)CCC2(CCN(C(=O)CC3COC(=O)C3)C2)C1 55073,N1(C(C(C)OCC2CC2)=O)CCC(F)(CNC(=O)C(=Cc2cccnc2)F)C1 55074,N1(C(c2c(SCC)cccn2)=O)CC(c2ccccc2)C(C#N)C1 55075,CCCCC(C)(CO)NC(C1CC=CC(NC(=O)CCc2cscn2)C1)=O 55076,c1(SC2CCC(NC(COC(C(=Cc3cnc[nH]3)C)=O)=O)C2)cccc(Br)c1 55077,C1(C(=O)NCCC#C)CN(C(C2(CN(C)C)CC2)=O)CCO1 55078,C1(NC(C(CC=C)(C)C)=O)CC1C1CCCN(C(=O)CCC2CCCC(O)C2)C1 55079,c1(OC)c(C(=O)NC2CC2C(=O)Nc2ccc(Cl)c(C)n2)cc(Cl)cc1Cl 55080,Cc1nncn1NC(=O)C1c2c[nH]nc2CN1C(=O)C1CCc2nccn21 55081,c1(OC)ccc(CN(C(=O)C(=O)Nc2csnc2C2CC2)C)c(C(F)(F)F)c1 55082,C(=O)(CC(CC)C(F)F)N1C(C(=O)NCCOCCC#C)CC1C 55083,C1(C(=O)NCC(C=C)O)N(C(C2CC(=O)N(OC)C2)=O)CC12CCCC2 55084,CCC(C)(CO)C(=O)NC(C1CCN(C(=O)C(C)NS(=O)(=O)CCC)CC1)(C)C 55085,C1(F)(C(=O)NC2(C(=O)NCC3(CC=C)CCCC3)CSC2)CCOC1C 55086,N1(C(CNC(CC)=O)=O)CCCCC(NC(C2(C(F)(F)F)CCCCO2)=O)CC1 55087,C12(CNC(C(CC)OC)=O)CCC(CC1)N2C(=O)C(c1cccs1)SC 55088,C1(NC(c2ccc(=O)oc2)=O)CC(F)CN(C(c2cnn(CC3CC3)c2)=O)C1 55089,c1(CC(C(=O)OC)NC(C2OCC3CCCC2C3)=O)c(F)c(F)c(F)c(F)c1F 55090,Nc1c(F)cc(C(N2CC3(CCCC3NC(c3cncnc3)=O)C2)=O)c(F)c1F 55091,C#CCCCC(=O)NCCC1CSCCN1C(=O)COC(C)(C)CC 55092,CC1C(O)CCCN1C(C1CCCC1NC(c1ccc(=O)oc1)=O)=O 55093,c1(C(N2CCC(NC(C3C(=O)NCC3)=O)C2)=O)cc2cccc(Br)c2s1 55094,c1(C(N2Cc3[nH]nc(-c4ccnnc4)c3C2)=O)ccn2ncc(Br)c2n1 55095,C12(NC(Cc3c(C)scc3)=O)CCC(CNC(=O)C(n3cc(Cl)cn3)C)(C1)OC2 55096,S(=O)(=O)(c1cc(Br)c(F)cc1F)N1CCC(C)C2(C1)CCCCC2 55097,c1(CC(=O)NC(CC)CNC(=O)CCC2CCC2)cccc(OC2CCOC2)c1 55098,N1(C(C(c2cccs2)SC)=O)CCCN(C(=O)CN2CCCC2)CCC1 55099,c1(NC(C)C)cccc(C(N2CCC(CN(C(=O)CCc3cnc[nH]3)C)C2)=O)c1 55100,C1(C(N2C(CCNC(CN(C(C(C)C)=O)C)=O)COCC2)=O)CCCC2(CC2)C1 55101,CCC(C)(F)C(=O)N1CCCC(NC(=O)NC2CCCC2)C1 55102,N1(C(C2(C=C)CC2)=O)C2CCC1CN(C(C1(C3CC3)CCC1)=O)C2 55103,C(=O)(CC(CC)C1CC1)N(CCCC(=O)Nc1noc(Cn2cnnn2)n1)CC 55104,O=S(=O)(c1ccc(-n2cc(-c3cccc(F)c3Cl)nn2)cc1)C(F)(F)F 55105,CCCCC(C(=O)N1CC2CC1CN2C(c1nn(C)cc1C)=O)N(C)C 55106,CCCCCCCCC(=O)NC(C1CCCCC1)C(C)NC(=O)C(=O)NCC 55107,C(=O)(C1=NOC2COCC12)NCC(CN(C(c1nn(CC)c(=O)cc1)=O)C)O 55108,O=C1Cc2c(N3CCCC3CCC(=O)Nc3ccc4nncn4c3)ncnc2N1 55109,c1(CNC(C2(C)CCN(C(C(CCC)OC)=O)C2)=O)cccc(F)c1F 55110,n1(CC)nc(C(=O)NC(C(=O)OC)C(C)O)c2c1CCOC2 55111,C1(CC(=O)NCc2n(C)ncn2)(NC(C2CC3CCC3C2)=O)CCCCC1 55112,CCCC(C(=O)NC1CCCC(NC(c2cc(C3CC3)on2)=O)C1)C(C)C 55113,C1(C(N(CCCNC(C2CC=CCO2)=O)C)=O)CC2(CCCCC2)S1(=O)=O 55114,c1(C(=O)NCC2(CNC(C3C(C)(COC)C3)=O)CCCC2)ccc(N)c(Cl)c1 55115,C1(C(=O)Nc2c(C(=O)OCC)csc2)CCN(C(c2csc(CO)n2)=O)CC1O 55116,C#CC1(C(=O)NCC2CCC(F)C2)CN(C(=O)CC2CC(N(C)C)C2)C1 55117,c1(N(C)C)ccc(C(=O)NCC)nn1.C1CCC(NC(=O)C(=O)NCC2CC2)C1 55118,c1(C(=O)NC(CNC(c2onc(C)c2C)=O)C2CCC2)cc2c(nc1N)CCC2 55119,N1(C(C(COC)C)=O)CC2CCCC(C1)N2C(c1ccnnc1O)=O 55120,c1(CN2CCN(CCC(=O)NC3CN(C)C3)CC2)c[nH]c2cccc(F)c12 55121,N1(C(C(C2CCN(C(CN(C)CC)=O)C2)F)=O)CCC12CC(CC(N)=O)C2 55122,c1(CNC(=O)Cn2cc(N3CCC3c3ccccc3)nn2)ccc([N+](=O)[O-])cc1 55123,CCC(CNC(C1CCCOC1CC1CC1)=O)(CC)NC(C1CC(F)(CF)C1)=O 55124,C(=O)(CCS(C)(=O)=O)N1C(C)(CNC(C2(CN(C)C)CCCCC2)=O)CCC1 55125,c1(C(=O)NCC(C)N(C(CCC(C)OC)=O)C)ccn2c(C(F)(F)F)nnc2c1 55126,CC1CCN(C(C23CCC(O)(CC2)CC3)=O)C(C)C1NC(=O)Cn1cnnc1O 55127,N1(C(c2c(CC)non2)=O)CCC(NC(=O)C=C2CCCC2)C(F)C1 55128,CC(C)CCN=C(NCC(C)(C)C1(O)CC1)NC1CC1F 55129,C(=O)(C1=CC2CCC(C1)C2)N(C1CCC(NC(C(C(C)C)C)=O)CC1)C 55130,N1(C(Cc2cc(OC)no2)=O)CC(C)N(C(=O)Cc2cc(Cl)ccc2Cl)CC1C 55131,O=C(C1=CCCCC1)NC1C=CCC(C(=O)NCCCC(O)CO)C1 55132,C1(C(=O)NC(CC#C)CC)CNC(=O)CN1C(=O)C(COC)N(C)C 55133,CC(C(=O)NCCCC(=O)N1CC(C(N)=O)(N(C)C)C1)C(F)F 55134,C1(NC(CCCCC=C)=O)CN(C(=O)C=CC2CCCN2C)CC12CCC2 55135,N1(Cc2n(CC)ncc2)CCC2(CC1)CC2NC(c1ccc(N)cc1OC)=O 55136,c1(-n2c(C(c3ccc(OC)nn3)NCC(Cl)Cl)nnn2)ccc(Cl)cc1F 55137,C1(C(=O)NC(CCC)C(=O)OC)CCCN(c2nnc(CC(F)(F)F)s2)CC1 55138,N1(C(c2nc(C)[nH]n2)C)CC=C(CNC(C2CCCCN2N=O)=O)CC1 55139,CC1(CC(=O)NC2CC(C(F)C(=O)NCc3conc3C3CC3)C2)CCCCC1 55140,c1(C(=O)OC)c(S(=O)(=O)NC2CCOC23CCCC3)n[nH]c1C 55141,c1(CCC(=O)OCCSc2c(C)cccc2)nc2ccccc2c(=O)n1C 55142,C(=O)(C(O)CNC(=O)C(C)CNC(C)=O)NCC1CC(C(=O)OC)C1 55143,c1(COC)ccc(C#N)cc1F.C1(=O)C(C)C(=O)NCCC(C(=O)NC)N1 55144,c1(CC)nc(C(N2CCC(C(C)C(=O)NCC(O)CF)CC2)=O)c(N)s1 55145,C(=O)(C(CN(C)C)C(C)C)NCC1(F)CN(C(c2ccnc(OC)n2)=O)C1 55146,Nc1cc(F)cnc1-n1cc(CC(CC(=O)O)NC(n2cc(C3CC3)cn2)=O)nn1 55147,c1(OCC)cccc(CC(=O)NCCOC2CCN(C(=O)CCCCSC)C2)c1 55148,N1(C(c2nc(CC)oc2C)=O)CCOCC(C(=O)NCC(F)CO)C1 55149,c1(CN(C2(CCCl)CCC2)C)cc(C2(F)COC2)n[nH]1 55150,c1(CC)onc(C)c1C(=O)NCC1CC1NC(=O)CCCN1C(=O)CCC1=O 55151,c1(C(C(=O)NC(C)C(=O)OC)N(C(C)(C)C)CC)cc([N+](=O)[O-])c(C)s1 55152,Cc1cc(C)c(C(=O)NC2CCNC2C2CC2)cn1 55153,CCCC(C(=O)N1CCC(N(C)C(c2cnoc2-c2ccc(C)o2)=O)C1)N(C)C 55154,Cc1nc(C)n(CC(=O)NC(C)(C)C=CC(=O)NCc2cc(C)n(C)c2)n1 55155,c1(C(N(CCNC(C2CC3(CCO2)CC3)=O)CC)=O)cnc2ccncc2c1 55156,N1(C(c2nn[nH]n2)CCOC)CCC(C#N)(c2ccc(C)cc2)CC1 55157,c1(C(C(=O)Nc2ccccc2)N(C2CCC3(CC2)CC3)C)cc2cnccc2o1 55158,CC1(C)CN(C(c2c(F)cncc2F)=O)c2cc(-c3cccc(O)c3)cnc21 55159,CC(C)CC(C(=O)NCC1(NC(c2cccnn2)=O)CCCC1)C(N)=O 55160,N1(C(C2C(C(C)C)OCC2)=O)CC=CC(C(=O)NCCCC2(C)CC2)C1 55161,c1(-n2c(CC3C(OC)COCC3)nc(C(C)C3CC3)n2)ccnc2ccsc12 55162,C1(CC)C(NC(c2ccn(C)c2C)=O)CCCN1C(c1ccc(=O)n(C)n1)=O 55163,C1(C(=O)NC2(CC(=O)NC(c3ccco3)CO)CCC2)CNC(=O)N1 55164,c1(CN2CCC(F)(C(=O)NCC(c3ccccc3)(C)O)C2)cnc2ncccn12 55165,C1(C(=O)OC)C2CC(CNC2)C1NC(=O)CCc1ccc(CC(=O)OC)cc1 55166,C1(F)(CNC(C2(C)CC=CCO2)=O)CC2CCC(C1)N2C(c1cnc(C#N)s1)=O 55167,CCC(C)CC(=O)C(=O)NC1(C(N2CCSCC2CO)=O)CC1C 55168,C(c1ccccc1F)=CC(=O)NCC1(CNc2nccc(OCC)n2)CC1 55169,c1(C(=O)NC2CN(C(c3c(Cl)cc(C)nc3)=O)C3C2C3)ccc2occc2n1 55170,C(c1csc(S(=O)(=O)N2CCCC2)c1)=CC(N1CC(C(=O)OC)C(F)(F)C1)=O 55171,C(=O)(C1=C(C)OCCS1)N1CCC(COC)(NC(C2CCC2(F)F)=O)C1 55172,c1(OC)ccc2ccnc(C(C)NC(c3cc(F)cnc3O)=O)c2c1 55173,C1(CC(=O)Nc2cc(C(C)(C)C)no2)CCN(c2ncncc2I)CC1 55174,N1(C(c2cc(OCC)n[nH]2)=O)CCCCC1C(C)(C)CNC(c1cnsc1)=O 55175,CC1(C=CC(=O)NCC2(O)CCN(C(C3(C)CCC(=O)N3)=O)C2)CCOCC1 55176,Cc1ccc(CC(=O)NCC2(C)CCCN2C(=O)C=Cc2ccncn2)cc1C 55177,c1(CNC(N(C(c2nccn2C)CO)C)=O)c(Cl)cc(OC(F)F)cc1Cl 55178,C1(C)(CNC(C2CC(OC)C2)=O)CCN(C(c2cnns2)=O)CC1 55179,N1(C(c2n(CC)ccc2)=O)CC2CCCC2(NC(c2cccc3ccnn23)=O)C1 55180,CC(O)(C(=O)NCCCOCCNC(=O)CC1CCC1)C1CCC1 55181,C1(NC(c2ccn(CC3CC3)n2)=O)CCOCC1NC(C1(CF)CCOCC1)=O 55182,c1(C(N2CCN(C(CCN(C)CC)=O)CC2C(C)(C)C)=O)cn2c(n1)CCCC2 55183,N1(C(C(CC)C)=O)CC(O)(C2(CNC(C3CCC(N(C)C)C3)=O)CC2)C1 55184,C(=O)(CCCCCF)N1CCC(NC(c2c(C)cc(CC)o2)=O)(COC)C1 55185,N1(C(C(CCCC)N(C)C)=O)CCCCCC(NC(=O)CC2(CO)CC2)C1 55186,C1(COC)(NC(=O)C(C)CN(C(=O)Cc2coc(C)n2)C)CCOC1 55187,N1(C(CCC=C=C)=O)CCCCC(CNC(C2CCCOC2)=O)C1 55188,C1(NC(=O)CNS(=O)(=O)N(C)C)CCNC12CCC2.n1(CC=C(C)C)[nH]cnc1=N 55189,C1(NC(c2cn(CC)nn2)=O)CN(C(c2coc(C(N)=O)c2)=O)CC1O 55190,C12(C(=O)Nc3cncc(SC)c3)CCC(NC(=O)CC3CCCN3C)(CC1)C2 55191,c1(NC(C(=O)NC(C)CCCNC(C23CC4CC2C3C4)=O)=O)ccc(Cl)c(F)c1 55192,c1(C(=O)NCCOC2CN(C(C3(SC)CCCCC3)=O)C2)cc(Cl)c(C)cn1 55193,O(N(C)C(=O)CN=c1[nH]c2c(c(=NC(C)c3ccncc3Br)[nH]1)COCC2)CC 55194,C(=O)(CC(C(F)F)C(C)(C)C)NCC1C2(CCN(C(CCCCSC)=O)CC2)C1 55195,c1(C(=O)NC(CC#C)C(=O)NCCCC2CCCCC2)cc(C)ccc1O 55196,c1(N2CCC(C(C)N(C)C)CC2)nc(=NC(CCO)C(F)F)[nH]c2ccc(Cl)cc12 55197,C(C1(O)CCc2ccccc21)NC(=O)Nc1c(C(F)F)cn(C(C)C)n1 55198,Cc1nn(C)c(Cl)c1C=CC(N1CC2CCC(C1)N2C(c1sccc1F)=O)=O 55199,c1(NC(C2CCC(C)N2C(=O)C2=CCCCO2)=O)cc(Br)cc(F)c1C#N 55200,Cc1nc(Cl)ccc1C(=O)NC(C)CNC(=O)CSC(F)F 55201,C(=O)(C1=CNS(=O)(=O)N=C1C)N1CC(CNC(CC(C(F)(F)F)OC)=O)OCC1 55202,c1(CNCC2OCCN(C(C3N(C)CCC3)=O)C2)ccc(Br)cc1C#N 55203,N1(C(C(C(C)C)C#N)=O)CC2CC(NC(=O)CSC(F)F)C(C2)C1 55204,N#Cc1cnn(CC(=O)NCCCCCNC(c2cc(C3CC3)on2)=O)c1 55205,C(=O)(CCC(C(C)C)NC(=O)C(F)C(C)(F)F)NCC(CC)C(C)C 55206,N1(C(CC2N(Cc3ccc(OC)cc3F)CCOC2)=O)C2COCC1CC(F)C2 55207,c1(C(=O)NCC2(O)CC(CNC(C(C)NC(N)=O)=O)C2)cn(C)c(=O)nc1O 55208,C1(NC(c2cncc(OC)n2)=O)CN(C(=O)C2=COCCC2)CC(F)(F)C1 55209,c1(CC(N2CCC(CNC(C3(CC(F)F)CCOCC3)=O)C2)=O)cccc(F)n1 55210,CCCCC(=O)C(=O)NC(C)(CNC(=O)C=CS(C)=O)C1CC1 55211,CCC(C(=O)N1CCCC1CCNC(=O)C=CI)C(C)C 55212,c1(-n2c(C(c3c(C)scc3)NCCCCF)nnn2)ccc(S(C)(=O)=O)cc1 55213,N1(C(C(C2CCCCC2)OC)=O)CCC(C2(O)CN(C(=O)C3=CSCS3)C2)CC1 55214,c1(CC(C(C)C)CN(C=O)Cc2ccccc2-c2cn[nH]c2)ccc(Cl)cc1Cl 55215,c1(CN(c2n(CCC=C)c(C3COCCC3(F)F)nn2)C)ccc2ccccc2c1 55216,CC(C)CC(C)CC(=O)N1CCC(C(=O)NCCc2c[nH]nc2O)CC1C 55217,S(=O)(=O)(c1c(C)cnn1CC)N1C(C#C)CN(C(=O)CS(=O)(=O)CC)CC1 55218,C1(COC)CN(C(c2cn(CC(N)=O)nn2)=O)CCN1C(=O)CN1CCOCC1 55219,c1(C(C)(C)C)cncc(C(=O)NCCC2CCN(C(=O)C(C)(C)C3CC3)CC2)c1 55220,N12CC3(CC3)CC1C2.CCC(C(=O)N1CC(OC(C)C(=O)NC)C1)n1ccnc1 55221,N1(C(CCC#CC)=O)CCCC(COC)(NC(=O)C=NOC)C1 55222,C1(NC(C2C(OC)CC2)=O)CCN(C(C2CC(C(F)(F)F)C2)=O)CC1(C)C 55223,C(=O)(C1=CC2CCCCC12)N1CC(NC(c2sc(CC)c(C)c2)=O)C(C)C1 55224,N1(C(c2c(CCC)[nH]cc2)=O)CCC(C)N(C(c2c[nH]nc2C)=O)CC1 55225,c1(C(=O)NC2CC(C)(NC(C3C=CCC3)=O)C2)cccc([N+](=O)[O-])c1O 55226,N1(C(c2c(C)cc(C)o2)=O)CCC2(COC(CNC(c3cc(C)c(C)o3)=O)C2)C1 55227,CCCCC(O)CC(=O)NC(COCC)CO 55228,CC1CN(C(C2COCCN2C=O)=O)CCCN1C(=O)CP(C)(C)=O 55229,N1(C(C2CCCC2NC(=O)CC2CC3CCC2C3)=O)CCc2nncn2CC1 55230,C1(C2CN(C(=O)C=CCO)C2)(NC(=O)COc2ccc(Br)cn2)CC1 55231,c1(C(=O)NCCC(CNC(C2CC2(C)C)=O)OC)ccc(C(C)C)cn1 55232,CC1C(NC(c2cnc(-c3cnn(C)c3)s2)=O)CCCN1C(c1ns[nH]c1=O)=O 55233,C1(C(N2C(CNC(C(CC)(C)CO)=O)C(C)CC2)=O)C2CCC1(C)C2(C)C 55234,c1(COC)ccoc1C(=O)NCC1COCC1NC(=O)C(C)n1ccnn1 55235,C1(F)(CNC(CCCC=C)=O)CCC(CNC(=O)C(F)(F)C2(O)CCCC2)CC1 55236,Nc1nc2ncccc2cc1C(=O)NCCCCNC(C1CCC12CCCO2)=O 55237,C1(CNC(c2c(C)onc2CO)=O)CC2CCC(C1)N2C(=O)C(C)C1CCCC1 55238,Cc1ccc(C)c(CC(=O)NC2CCC2CNC(=O)CN2CC(=O)N(C)C2=O)c1 55239,c1(CN2C(CNC(c3nc(C)c(F)cc3)=O)CCC2)cccc2cccnc12 55240,c1(CNC2CCC(C(=O)Nc3c(C#N)cc(F)cc3)C2)ccc(Cl)c([N+](=O)[O-])c1 55241,S(=O)(=O)(c1ccc(N2CCCC(S(N)(=O)=O)C2)c(Cl)c1)NC(C)(C)COC(C)(C)C 55242,Cc1cc(C(N2CCOC(CN(c3ccncn3)C)C2)=O)c(C(F)(F)F)o1 55243,c1(C(N2CCC(C(C)NC(=O)CC3C=CCC3)CC2)=O)cccn(C)c1=O 55244,C1(NC(c2ccc(C(C)C)o2)=O)C=CCN(C(=O)CNC(=O)CCCCO)C1 55245,N1(CC(=O)N(c2ccn(C)n2)C)C(=O)NC(C)(CNC(=O)OC(C)(C)C)C1=O 55246,Cc1cnc(O)n1-c1cccc(NC(=O)C(=O)N(C)CCN2CCCC2=O)c1 55247,c1(C(=O)N(C2CC2)OC)ccc(-c2cc(-c3nccn3-c3nc[nH]n3)c[nH]2)cc1 55248,CC(Cc1cccs1)N=c1cc[nH]c(=NCCCC2(C)CC2)[nH]1 55249,CC12CCC(C(=O)NCCC3=CCN(C(C4CSCC(=O)N4)=O)CC3)(CC1)OC2 55250,C(=O)(C1CCc2nccn21)NC1CN(C(C2(SC)CC2)=O)CC1C 55251,C1(C(=O)NCC(C)N(C)CCc2c(F)cccc2Cl)CC2CCC1CC2 55252,c1(C(=O)NCCOCCN(C)C(C2CCCC(C#N)C2)=O)cnc2ccccn12 55253,C=C1CCCN(C(=O)CSCCNC(c2ncn(CC)n2)=O)C1 55254,C(=O)(CCCCC(C)C)N1C(C(=O)NCc2ccc(C)s2)CC(C)(C)C1 55255,C(=O)(N=S(C)(=O)c1ccc(C)cc1)c1cc(N(C2(COC)CCC2)C)nc(C)n1 55256,C12(C(=O)NC3C(C)N(C(c4ccc(CO)o4)=O)CC3)CC=CC(C1)OC2 55257,N1(C2CCC(NC(C(=C(C)C3CC3)F)=O)C2)CCN(C(=O)C2=CCSC2)CC1 55258,Cc1ccc(CC(=O)NCCC(C)(C)NC(=O)CC2CC(C3CC3)C2)cc1Cl 55259,c1(CCC(=O)NCC2CN(CC(O)COc3cccs3)C2)ncc(F)cn1 55260,c1(C(N2CCCC(N(C(CCC#CC)=O)C)C2)=O)cnc2cc(OC)ccn12 55261,Cc1ccn2cnc(C(=O)NC3CN(C(C4(C)CCCC4)=O)CC3O)c2c1 55262,C1(CC(=O)NCCOCCN(C(C(C)n2cncn2)=O)C)CCOCC1(C)C 55263,C(=O)(C1CCc2cc(OC)ccc21)NC1CCC(NC(C2(COCC)CC2)=O)C1 55264,C1(N(C(C2CCCN(C(C3C(CC)OCC3)=O)C2)=O)C)CCCC(C)C1C 55265,C12(CNC(C3N(C(=O)NC)CCC3)=O)CCC(NC(c3cccs3)=O)(CC1)CO2 55266,C(CCCCC(=O)NC1CC(C(=O)NCC2(COC)CC2)C1)OC 55267,C1(C(C)(C)C)(C(=O)NCCOC2CN(C(CC3C(C)CCC3)=O)C2)CCCCC1 55268,c1(C(C)=O)cc(C(=O)NC(C(=O)NCCS(C)(=N)=O)C2CCC2)no1 55269,c1(CNc2c(CC(=O)Nc3ncc(C)c(F)c3)cccc2)ccc(F)c(C)c1Cl 55270,c1(CC(=O)NCCC(CNC(C(C(C)O)C)=O)(C)C)ccc(S(N)(=O)=O)cc1 55271,c1(C(=O)NCC2CC(F)(CNC(C(CC)OC)=O)C2)c[nH]c2cc(OC)ccc12 55272,c1(C(=O)NCC(C)NC(C(C(=C)Cl)(C)C)=O)snc2ccc(Br)cc12 55273,c1(OC)ccc(COC2CCC2C(=O)OCC(C)CC2CCCC2)cn1 55274,C1(C(=O)NC(CCC=C)C2CC2)C2CC1N(C(=O)C=Cc1ccncc1)C2 55275,CCC1=C(C(=O)N(CCC(=O)NCCCOC(=N)O)CCCO)CCCO1 55276,c1(OC)cccc2ccc(C(=O)N(C(C)CNC(=O)CS(C)(=O)=O)C)nc12 55277,S(=O)(=O)(c1ccc(NC23CC(CN=[N+]=[N-])(C2)OC32COC2)cc1)NC 55278,C(=O)(C(F)C(C)CC(C)(C)C)N1C(C(C)NC(=O)C(=O)N=S(C)(C)=O)CCCC1 55279,S(=O)(=O)(c1ccc(N2CCS(=O)(=O)CC2)c(Br)c1)NCc1ccc(OC)c(O)c1 55280,c1(CNC(C2CC(C)OCC2)=O)cnn2c1CN(C(C1CCN(C)CC1)=O)CC2 55281,C=CC1CN(C(=O)CCCn2ccnn2)CC1NC(=O)CC1CNC(=O)C1 55282,c1(N2CCN(C(c3cc(F)ccc3F)=O)C3C2C3)ncnc2cc(Br)ccc12 55283,Cc1nc(C)c(C(N2CCC(O)(C(C)NC(=O)Cc3nn(C)cc3Cl)C2)=O)s1 55284,Cc1cc(C)c(CN2CCN(C(=O)C=Cc3ccoc3)C3CC23)cc1C 55285,C=CC1(CO)CCN(C(C2CCOC2CNC(=O)CC(C)N(C)C)=O)CC1 55286,c1(C(=O)Nc2c[nH]nc2C(=O)Nc2cc(F)ccc2I)cc2sccc2[nH]1 55287,c1(CC(=O)NC2(CO)CCN(C(=O)C3=CCC3)C2)cccc(F)c1 55288,C(=O)(C(CC)C(F)(F)F)N1C(CC)C(C(=O)NCCNS(N)(=O)=O)CCC1 55289,C(=O)(C(C)(C)CSC)NC(CN(C(c1cnc(-c2ccccc2)o1)=O)CC)C 55290,N1(C(CC=CCC)=O)CCC2CCC12CNC(c1cncc(C(F)(F)F)n1)=O 55291,N1(C(CC)C(=O)O)CCC2(CC1)CC2(C)C(=O)NC1CCOC(c2cccs2)C1 55292,c1(CC)c(C(=O)NCC(C)CN(C)C(c2ncccn2)C)cnn1C 55293,c1(C(C)NCc2cc(C3CCC3)no2)coc2ccccc12 55294,c1(C(=O)NC(CCCC)CNC(c2cc(Cl)no2)=O)cc2cccn2cn1 55295,c1(NC2(CC=C)CCC2)nc(N2CC(OC)C(OC)C2)nc2sccc12 55296,CN1CCC(C)(C(=O)NCCC2(C)CCN(C(C34CCC3C4)=O)C2)CC1 55297,C1(C(=O)NC(C)Cc2cnn(C)c2)CC2CCC(C1)O2.C12CCC(CC1)C(=O)N2 55298,c1(C(=O)NCc2c(C(=O)NC3CC(C)(C)OC3)c[nH]n2)cc(O)ncc1F 55299,C(=O)(CS(=O)(=O)C(C)C)N(C1CCCN(C(CC2(C=C)CCOCC2)=O)CC1)C 55300,CN1CCN(C(c2cc(CO)[nH]n2)=O)C(C(=O)N(CC(N)=O)C)C1 55301,N1(C(C2CCC(C(F)(F)F)CC2)C(=O)NCCCC)CCC2C(O)C(C)(C)C12 55302,C(=O)(C#CC1CCCC1)NCCCCC(C)NC(C1(c2cccc(O)c2)CC1)=O 55303,C(=O)(C(C(C)CC1CCCC1)N(C1(C#N)CCC1)C)N(CCC)CCC 55304,c1(NC(=O)NC2C(C)OCC2)ccc(OC2CCCC2)cc1F 55305,c1(CC(=O)N(C2CCN(C(=O)C#CC3CCCO3)C2)CC)cccc2sccc12 55306,C1(NC(c2n(CCC)ccc2)=O)CCN(C(c2cn[nH]c2)=O)C1(C)C 55307,C#Cc1nc(C(=O)N(CC(N2CCN(C(=O)CCCCOC)CC2)=O)C)cs1 55308,N1(C(c2c(C)cno2)=O)CCC2(C1)CN(C(C1(C)CC1C(F)(F)F)=O)C2 55309,CC(=O)CCCC(C)C(=O)NC(CC(=O)N1CCCC(O)(CN(C)C)C1)CC(C)C 55310,CC1(C)COc2cc(C(=O)Nc3ncc(-c4cncc(F)c4)s3)nn2C1 55311,CCC(CC)C(C(=O)N1CC(C)(C(N2CC([N+](=O)[O-])C2)=O)C1)OC 55312,N1(C(c2ccc(C(C)C)o2)=O)CCCC(C)(CNC(c2cnc(O)c(Cl)c2)=O)C1 55313,Cc1cc(C(c2nnnn2CC(F)F)Nc2nn(C)cc2Br)cc(C)c1Br 55314,C#CC(C)(C)C(=O)N1CCCC1.c12nnc(N(C)C(C)C)n1CCC(=O)OC2=O 55315,C1(C(=O)NCC(CC(=O)N(CCCO)CC)O)CC2C(C1)C2(C)C 55316,N1(C(CCC2CC(C)C2)=O)CCCC(CO)(CNC(=O)CS(C)(=O)=O)C1 55317,C(=O)(C(C)(C)CCCNC(C1CCC(=O)C1)=O)NCC(n1ccnn1)C 55318,C1(CC(=O)NC)CN(C(C2CCC2(C)C)=O)CCN1C(C1CCC=CCC1)=O 55319,C#CC(CNC(=O)C(Cn1cncn1)NC(=O)CN1CC(C)(C)C1)CC(C)(C)C 55320,n1(CC)nc(C2CC2)cc1C(N1CCCC1C(C)(C)CNC(=O)CCC(N)=O)=O 55321,C(=O)(C(O)P(C)(C)=O)NCC(N(C(=O)CCCc1cncs1)C)C1CC1 55322,c1(NCC(C)(C)Nc2ccccn2)ccc(Br)cc1 55323,N1(C(=O)NCC(N2CCCCCC2)C)C2CCCC1CN(C)C2 55324,CC(C)CC(CCO)CN=c1[nH]c2c(c(=NCC3C(F)(F)C34CCC4)[nH]1)CCCC2 55325,C1(NC(C(N2CCCC(CNC(=O)OCC)C2)=O)=O)CC2(C1)CC(F)C2 55326,Cc1c(NCCCOCCCO)nc[nH]c1=NCc1ccc(CC(=O)N(C)C)cc1 55327,c1(C(N(C(C)C)Cc2cccc(C)c2C)=O)ccc2c(c1)OC(C)C2 55328,Cc1nccc(Cl)c1C(=O)NCCN1CCCN(C(=O)CC2CCCC2)CC1 55329,C12(C(N(C)CCNC(=O)C(c3ccc(O)cc3)=O)=O)CC3CC1C2C3 55330,CC1(C(N2CCC(N(C3CCCCC3)CCO)C2)=O)CCCN1CC(=O)NC1CC1 55331,C#CCC(CC#C)C(=O)NCCCC(CCC)NC(c1csc2c1CCCC2)=O 55332,C1(NC(=O)OC(C)(C)C)CC=C(C(=O)N2CC(Nc3occ4c3CCC4)C2)C1 55333,CC#CCCC(=O)N(CC(C)(C)CNC(c1cncnc1C1CC1)=O)CC 55334,c1(SC)cncc(C(=O)NC2CC(NC(=O)C=CC3CCOC3)C2)c1 55335,N1(C(C2(C)CNC(=O)C2)=O)CCC(C2CCN(C(=O)CC=C(Cl)Cl)C2)C1 55336,C1(C(=O)NC(C)(C)C=CC(=O)NC(C)(C)CCCF)CN2CCC1CC2 55337,N1(C(CCC=CCC=C)=O)CCC(C)(NC(=O)C(C)CC2CCC2)C1 55338,n1(CC)ccnc(NC(C2(C)CCN(C(=O)OC(C)(C)C)C2)=O)c1=O 55339,C(C)(CCCC(=O)N(C)CC1(O)CCCCC1)NC(COC(C)=O)=O 55340,C1(C(F)(F)F)(C(=O)NCC2N(C(c3n(C)ccc3)=O)CCCC2)CC2(CCC2)C1 55341,c1(NC(C(C(C)C)NC(C(CCC)NC(N)=O)=O)=O)cc(C#N)ccc1O 55342,N1(C(c2c(C)ocn2)=O)CCN(C(c2csc(CC(F)(F)F)n2)=O)CC1 55343,S(=O)(=O)(c1cccc(=NC2CCC=CCCC2)[nH]1)NC1CN(C)C2(C1)CCOCC2 55344,c1(N2CCC(N(C(=O)C(O)CCSC)CCC)C2)cc(C)c(C#N)cn1 55345,CC1CC(C(=O)NCC2CC3(CC3)CN2C(c2cc(O)cs2)=O)CCC1C 55346,c1(C(N2CCC(C3N(C(C(F)OC)=O)CCC3)C2)=O)ccc(F)nc1F 55347,C1(C(=O)NCC2CCC(C)O2)CCC(CNC2(CCN=[N+]=[N-])CC2)CC1 55348,CC(CC(=O)c1cccc(Br)c1)C(=O)NC(c1sccc1-n1cccc1)=O 55349,C1(NC(c2scc(OC)c2)=O)CS(=O)(=O)CC1NC(=O)C=CSC 55350,C(C)(C(=O)NC1CC(NC(c2cc(C)sc2C)=O)C(O)C1)(C(C)C)OC 55351,N1(C(C(C)OCCCC)=O)CC2(CCC(NC(C3C=C(C)CS3)=O)CC2)C1 55352,S(=O)(=O)(C=Cc1ccccc1)N1CCN(C(CC=CCC)=O)C2C1C2 55353,n1(CC=C)ncc2c(O)nc(=NCC(C)CNC(=O)C(C)CC(C)(C)C)[nH]c12 55354,C(=O)(NN1CCCC1C(=O)NC1(CCF)CC1)c1cc(C(=O)OC)[nH]c1 55355,N1(C(C(C)NC(=O)NC)=O)CCCC(CO)(NC(=O)CC2C=CS(=O)(=O)C2)C1 55356,C1(C(=O)NC2(C)CCN(C(C3(C)C(C(=O)OC)CC3)=O)C2)CCC(C)(C)CC1 55357,C1(NC(C2C(C(C)NC(CCCC3C(C)C3)=O)C2)=O)CCOC1(C)C 55358,C1(C(=O)NCCC2(CNC(=O)COC3CC(F)(F)C3)CC2)CCCCCS1(=O)=O 55359,c1(C(N2CCC(N(C)C(c3ccc(-c4ccco4)[nH]3)=O)C2)=O)coc(C(N)=O)c1 55360,C1(C(=O)NC(C)C(=O)O)CC=CC(n2cc(-c3ccc(F)cc3)nn2)C1 55361,c1(C(=O)NC(CCCNC(C(CC(C)C)C)=O)C)cc2n(n1)CCCC2=O 55362,C1(COCC(C(=O)N(CC=C)CC)F)CCN(c2ccccc2)C1.C1C(=O)N1CC 55363,C12(C(=O)NCC(CC)NC(=O)C(F)=CC3CC3)CCCC1C2(F)F 55364,CCC(c1ccnc(N2CCN(C(=O)CC=CCc3ccccc3)CC2)c1)=CC 55365,N1(C(C(C)(C)OCC)=O)CCOCC(CNC(c2nc(C)n(C)n2)=O)C1 55366,C=CC1(C(=O)NCC=CCC(=O)N(C(C)CC(C)C)C2CC2)CCCCC1 55367,N#CC1CN(C(C2CCOC2)=O)CCN1C(c1ccc(N2CCC2)cc1)=O 55368,N1(C(=O)C=Cc2cccc(Cl)c2)CCCC2(CCC(NC(C3(F)CC3)=O)C2)C1 55369,c1(CC(C(=O)NC(C(=O)OC(C)C)Cc2ccccc2)N)cccnc1F 55370,c1(NC2CCCCN(C(CC(CC)O)=O)C2)c(Cl)cc([N+](=O)[O-])cc1Cl 55371,C(=O)(CC(C(F)F)NC(c1ncc[nH]1)=O)Nc1cccc(C(C)C)c1 55372,c1(C(N2CCC(CC=C)C2)=O)cncc(OC(C)C)n1 55373,C1(CC)C(NC(C2CCC(CC)CC2)=O)CCCN1C(=O)CCn1ccnn1 55374,n1(CC(=O)N(C)CC2CCN(C(C3(COC)CCCC3)=O)C2)ncn(C)c1=O 55375,N1(C(Cc2c(C)noc2)=O)CC(C2CCN(C(C3COC(C)C3)=O)CC2)C1 55376,N1(C(CCC=C)=O)CCC(C(=O)NCC2(c3ccnc(Cl)c3)CC2)CC1 55377,Cc1ccc2c(c1)CCC(C(=O)NCC1CCCCC1NC(c1csnn1)=O)O2 55378,C(=O)(C#CC1CCOCC1)NC(CCC)CC(=O)NCc1cnccc1OC 55379,N1(C(C2C(C)CC=CC2)=O)CCC(F)CC1C(=O)NCC1(C#N)CC(C)(C)C1 55380,C(=O)(C(CNC(=O)C(CNC(c1c[nH]c(C(N)=O)c1)=O)N(C)C)OC)OC 55381,CCC(CN(C)C)CC(=O)N1CC(NC(=O)CC(C)(C)C#N)C(n2ccnn2)C1 55382,c1(CNC(c2cccc(CC3C(COCC)CCCC3)n2)=O)cccc(CO)c1 55383,C1(CC)CN(C(c2cc(=O)n(C)o2)=O)CCN1C(C1CCCOCC1)=O 55384,c1(OC)ccc(NC(=O)NNC(C)CNc2ccccc2Cl)c(F)c1Br 55385,C1(N(C(=O)C(=O)NCCOC(C)(C)C(F)(F)F)C)CCS(=O)(=O)C1 55386,Cc1cc(C(=O)NC2CCCC(NC(c3cc(O)cs3)=O)C2)nnc1C 55387,C1(C(N(CC(C)NC(=O)CNC(N2CCCC2)=O)C)=O)COC(C)CO1 55388,OC1COCCN(N2CCC2C2CCC2)C1.c1ccco1 55389,c1(C(=O)Nc2cc(C)c(NC(c3ccnnc3C)=O)cc2)ccn2cncc2c1 55390,C(CCC(=O)NC1CC(C)(NC(c2cc(C(F)F)cs2)=O)C1)OC(C)C 55391,O=C(C1=CCOC1)NCC1CCN1C(c1cn[nH]c1)=O 55392,CCCCCCC(CC)C(=O)N1CCCCC1Cn1cc(CNC(N)=O)nn1 55393,c1(CC(N2CCC(CCS(N)(=O)=O)C2)=O)cn2c(Cl)cc(Cl)cc2n1 55394,C1(CN(C)C(=O)N(C(C)(C)C)C)CC1C1CC1 55395,c1(C(N2CCC(C(=O)Nc3c(C#N)cccc3O)C2)=O)nccc2ccccc12 55396,Nc1ccc(C(=O)N2C3(CCCC3)CC2)c(O)c1.C1(N)CC(=C2CCC2)C1 55397,c1(C(=O)NCC(CNC(CCCOC)=O)F)cccc2c1ncn2C 55398,Cn1cc([N+](=O)[O-])cc1C(=O)NCC1(F)CN(C(c2cc(F)cs2)=O)C1 55399,c1(OC)cc(C)c(C(=O)NC2CCCC2CNC(c2c(C)coc2C)=O)cn1 55400,c1(C(=O)NC(CNC(C(CC)CC2CCCC2)=O)C)ccc(CCCCl)c(F)c1 55401,C1(C)(C(C)C)CCCN1C(C1N(C(=O)Nc2ccc(C(N)=O)cc2)CC1)=O 55402,C1(n2cnnn2)(C(=O)NC2(C)CN(C(c3cc(C4CC4)no3)=O)C2)CCOCC1 55403,N1(C(c2c(OC(C)C)n[nH]c2)=O)CC(NC(C23CCCC2C3)=O)C2(CCC2)C1 55404,c1(C(=O)NCC(CC)NC(C2C(CCC)CCC2)=O)ccc(C)cc1O 55405,Cc1ncccc1C=CC(=O)NC(C(C)NC(=O)CCCC1CC1)C(C)C 55406,c1(C(=O)NC(C(C)O)C(=O)N(C)C)cnc(F)c(F)c1 55407,CC1(C(=O)NCC2(C)CCN(C(c3c(Br)nnn3C)=O)C2)CC(C2CC2)=NO1 55408,C1(CC)(NC(=O)CN2CCCC2C)CCCN(C(c2ccc(Cl)c(OC)c2)=O)C1 55409,c1(C(N(CCN(C(C(CC)N(C)C)=O)C)C)=O)cc2c(OC)cc(OC)cc2o1 55410,CC1(C(=O)NC2(C3CCC3)CC2)CCN(C(=O)C=CCN2CCC2)CC1 55411,Cc1cc(C)c(C(=O)NC2(C)CN(C(C34COCC3C4)=O)C2)cc1C 55412,N1(C(C(COC)C)=O)CCC2(CCN(C(c3[nH]c(C)c(C(C)=O)c3CO)=O)C2)C1 55413,CC(C)C(C(=O)NC1CCC(N(C(=O)C(N)=O)C)C1)NC(c1ccccc1Cl)=O 55414,c1(C(N2CCN(C(C3CCCCC3CCCC)=O)C3(CC3)C2)=O)ccc2[nH]ccc2c1F 55415,c1(NC(C)=O)ccc(C(=O)NCC2(O)CC(NC(C3CCC3(F)F)=O)C2)s1 55416,c1(C(=O)NC(CC2OCC(C(=O)OC)C2)=O)ccnnc1S 55417,Cc1cc(C(N2CCCC(N(C(=O)C(C)C3=CCCC3)C)C2)=O)cc2nc[nH]c12 55418,c1(C(=O)NC2C(CC)N(C(C)=O)CCC2)c(Cl)ccc(Br)c1F 55419,Cc1[nH]c2ncccc2c1C(=O)NC(C)CCCNC(=O)CCC1CC1(F)F 55420,C(=O)(C1=CCCC1C)N1C(C(N(CC(C)C)C)=O)CC(=O)C1 55421,C(=O)(C1=CC=CN2CCS(=O)(=O)N=C12)OCCC(C)OC 55422,N1(CCN(C(=O)CC2CC=CCN2C)C)CCN(C(c2ccns2)=O)CC1 55423,C1(NC(CCc2ccc(CC)cc2)=O)CCC(C)N(C(C2C=CCCC2)=O)C1 55424,C(=O)(CC(C)n1cccc1)NCCCN(C(C1CC(O)C1)=O)CC 55425,CCCCCC(CCCCC)C(=O)NC1CC(NC(c2cc(C#N)oc2C)=O)C1 55426,Cc1cc(Br)c(N)cc1C(=O)NCCNC(=O)CCCC(F)(F)F 55427,c1(C(=O)NC(CCNC(c2cn(C)[nH]c2=N)=O)(C)C)cccc2nsnc12 55428,N1(C(c2ccc(C(N)=O)s2)=O)CCC2(CC1)CC(NC(C1C3CC4C(C3)C14)=O)C2 55429,c1(C(=O)NC2CC(C)N(C(c3cccn3C)=O)C2)ccc2c(c1)C(=O)C(=O)N2 55430,C1(NC(CCCCCOC)=O)COC2(C1)CN(C(=O)C=Cc1cn[nH]c1)C2 55431,c1(C(N2C(CNC(=O)C(O)c3ccco3)CCC2)=O)cnn2cccc(Cl)c12 55432,N1(C(c2cc(C)[nH]c2)=O)CCN(C(=O)CC(C)C(F)(F)F)CCC1C 55433,c1(C(=O)NCC(CNC(c2ncc(C)cn2)=O)O)c(N)sc2ccccc12 55434,c1(C(N2C3CC(CC(NC(COCCC)=O)C3)C2)=O)ccc2n[nH]cc2c1Cl 55435,c1(C(N2CC(NC(CCC)=O)C(O)C2)=O)cccn2cncc12 55436,C(=O)(C1=CCCN(C(=O)Cc2ccccc2C)C1)NC(C(C)SC)C 55437,N#Cc1cccc(C2(C(=O)OCc3cc(-c4ccc(O)cc4)on3)CCCCC2)c1 55438,Cn1cc(C(=O)NC2CCCCC2CNC(=O)C(C)(C)c2cscn2)n(C)c1=O 55439,c1(CC(=O)NC2(COC)CCN(C(C3(C)CC(C)(C)C3)=O)C2)ccc(C#N)cc1 55440,C1(C(=O)NC(Cn2ncc(C)c2)C)CC(C)(C)CN1C(c1cc(C)c(F)cn1)=O 55441,N1(C(C(C)OCCOC)=O)CCC(C)C(NC(=O)Cc2csc(C)n2)C1C 55442,CC(C)CC(C)n1nccc1C.C(=O)(C(C)(C)c1cncnc1)N.CCC1CC(=O)N1 55443,C(=O)(C1=CC2CCCCCC12)NC(=O)OCCCCC1(CO)CN(C(C)(C)C)C1 55444,N(C(=NCCCSC)NCCC1CC(=O)N(C)C1)Cc1ccc(OCC=C)cc1 55445,C(=O)(C(CC(C)C)n1ccnc1)NC(CC=C)CNC(C1(CN(C)C)CC1)=O 55446,c1(C(=O)NC2CCC(CNC(C3(C)CC4CCC3O4)=O)C2)ccc(Cl)c(N)c1Cl 55447,c1(C(N2C(CNC(CC(C)P(C)(C)=O)=O)CC2)=O)cc2c(cn1)COCC2 55448,CCCCC(CNC(=O)CCCN(C)C(C)=O)NC(C1CC(CC2CC2)C1)=O 55449,C1(OC)CC1C1CCN(C(C2(C#N)CCN(C(=O)OC(C)(C)C)CC2)=O)CC1 55450,Cc1nc(C(N2CCOC(C(C)NC(=O)C(C)C3CCCO3)C2)=O)[nH]c1C 55451,C1(C(C)C)(CO)CCN(C(=O)C=CC(C)NC(=O)C(C)C2CCC2)C1 55452,c1(C(=O)NCC2N(C(c3c(C)coc3)=O)CCC2)ccc([N+](=O)[O-])cc1Br 55453,c1(C(=O)NCC(CNC(c2ccc(C)s2)=O)CO)ccnc2c1CCO2 55454,Cc1ccc(C)c(OCC(O)CNC(c2ccc(N)cc2Br)=O)c1 55455,Cc1onc(Br)c1C(N1CC(CNC(c2ccc(O)nn2)=O)C(C)C1)=O 55456,c1(C(N(CC(C)C)CC#C)=O)cccc(CCCSn2cccn2)c1 55457,c1(C(N2CC(CC(=O)N(C(C)C3CC3)CC)OCC2)=O)ccn2ccnc2c1 55458,Cc1cc(C(=O)NCC2CC(NC(c3cc(Cl)sc3Cl)=O)C(O)C2)cn(C)c1=O 55459,C(=O)(CCC(C)(C)[N+](=O)[O-])N1C2C(CC1)CN(C(C)C)C2=O.c1(CC)ccco1 55460,C1(NC(C2C=CCS2)=O)CC2(CCCN(C(=O)COCC3CCCC3)C2)C1 55461,N1(C(C2(C#C)CN(C(=O)C(F)C(C)(C)O)C2)=O)C(CO)CC2OCCC12 55462,C(=O)(C(CO)C(C)(C)C)NCC(CCOC)NC(c1cc(C)c(O)c(C)c1)=O 55463,S(=O)(=O)(C(F)(F)F)CCC(N1CC(C2CCCO2)(OC)C1)=O 55464,c1(N2Cc3n(C)c(Br)nc3CC2)nc2c(c(=NCCS(C)=O)[nH]1)CSC2 55465,c1(SC)ccc(CCC(=O)NC2CC(CNC(c3oc(C)nc3C)=O)C2)cc1 55466,C12(NC(c3ncc(OC)cc3F)=O)CCC(CC1)N(C(C1(C(C)C)CC1)=O)C2 55467,C1(C(=O)NC2CCC(NC(c3cnc(Br)s3)=O)CC2)OCC2CCCC1C2 55468,C1(C(=O)NCCC)CC(C)NC(=S)N1.c12ccc(F)c(c1)NC(=O)C(=O)N2 55469,c1(OC)cc(C)cc(C(=O)NCC(C)N(C(=O)CC(O)C(C)C)C)c1N 55470,c1(CCC(=O)NCC(CC)NC(C2CCC(C(F)(F)F)O2)=O)c(F)cccc1F 55471,CC1(C)CC(C(=O)COC(=O)CCCC2CCSS2)CC(C)(C)C1 55472,Cc1cc(C(=O)NC(C(=O)N2CC(C(C)(C)O)C2)C2CCOC2)nn1C 55473,Cc1ncc(C(N2CCN(C(=O)Cc3ccnc(F)c3)CC2C)=O)cc1N 55474,N1(C(c2c(CC)cccn2)=O)CCC(CNC(=O)CCCOCCOC)C(O)C1 55475,C12(C(=O)NCC3N(C(C4CC5(C4)CC5F)=O)CCC3)CCCCN1CCC2 55476,CC1CC(NC(C2(C)CC2(F)F)=O)CCN1C(c1coc(O)n1)=O 55477,C1(C(=O)NCc2ccc(C#N)cc2)CN(C(=O)CCC(N)=O)CC12CCC2 55478,N1(C(c2cccc(CN=[N+]=[N-])c2)=O)CC2(C(=O)O)CCC2(C(=O)O)C1 55479,C(=O)(C1CC=Cc2ccccc21)NC(C)(C)CCCNC(=O)C(=O)NCC(F)F 55480,C(=O)(CCCC(C)(C)C#N)OC.C1(=O)C(C(C)C)NC(=O)OCC(OC)CN1 55481,c1(C(N2C(CC=C)CCC2)=O)cc2nccc(OC)c2cc1OC 55482,CCCC(C(F)(F)F)NC(=O)NCC(c1ccncc1)CCC1CC1 55483,CN1CCN(C(=O)NC2CCC(N3CCOCC3)C2)CC1CC1CCC1 55484,n1(CCNC(C(C2CC2)SC)=O)ccc(C(=O)NC(c2nncn2C)CO)c1 55485,N1(C(c2cccc(OC)c2N)=O)CCC(NC(=O)C(C)CC(N)=O)C12CCCC2 55486,C(CCC(=O)N1CCCC1CC(N1CC(N(C)C)C1)=O)N(C(C)=O)C 55487,C1(C(=O)NCCOCC)CC(NC(=O)COC(C)=O)C(O)C1.CCCCC 55488,N1(C(C=C(C)C)=O)CC(NC(C2CCOC2c2cccnc2)=O)CCC(O)C1 55489,C(c1ccc(O)c(OC)c1)=CC(=O)NC(CC)CNC(c1sc(CO)nc1C)=O 55490,C(=O)(CCCC1(OC)CC1)NC(CN(C(C(c1cccs1)OCC)=O)C)(C)C 55491,CC(CNC(c1cc(C(O)C2CC2)ccn1)=O)CC(=O)N(C(C)C(C)C)C 55492,CCCC(CNC(C1CCN(OC)CC1)=O)C(=O)NCCN1CC(C)(O)C1 55493,C1(C)(C(=O)OC)CCN1C(=O)CC1CCCN1C(=O)C=CCF 55494,c1(N(CCNC(=O)CC2CCC3CC3C2)CC)nc(C(=O)OC)nc(C)c1C 55495,C1(C)(NC(c2cc(C)ns2)=O)CCN(C(c2cc(CC3CCC3)c[nH]2)=O)C1 55496,C12(C(=O)NCC3(NC(CCOC(C)=O)=O)CCCCCC3)CC=CCN1CCC2 55497,c1(CCC(=O)NCC(C)NC(=O)C(C)OC2CCCCCC2)nnc(O)nc1O 55498,C(C)(C(=O)N1CCN(C(=O)COc2ccc(C)cc2F)CC1)(C(F)(F)F)OC 55499,N1(C(CC2(C)CN(C(c3cc[n+]([O-])cc3)=O)C2)=O)CCC(C)(O)C(O)C1 55500,C1(C(N(C2CCC2O)C)=O)CC12CCN(C(=O)Cc1cn[nH]c1)CC2 55501,CCC(C)(CC)C(=O)NCCCCN(C(C1CC1c1ccccn1)=O)C(C)C 55502,c1(C(=O)NCC(CN(C(c2c(C)cncc2)=O)C)O)c(Cl)cccc1[N+](=O)[O-] 55503,c1(C(=O)NC(CCNC(c2c(C)nc(C)[nH]2)=O)(C)C)cccc2oc(C)cc12 55504,c1(C(=O)NC2CC(C)(CNC(c3n(CC)ccn3)=O)C2)ccc(F)cc1C 55505,c1(C(=O)NC2COCCN(C(=O)C(O)C(F)(F)F)C2)cc2c(F)c(F)ccc2[nH]1 55506,c1(C(N(C)CC2CN(C(=O)Cc3nncn3C)C2)=O)cc2ccccc2[nH]1 55507,C1(NC(c2c(CC)csc2)=O)CC2CN(C(=O)CC(F)(F)CC)CCN2C1=O 55508,C12CCCCCC1C(=O)N2.N1(C(CCOC)=O)CCC(C(C)C)(CO)C1 55509,C(N=c1[nH]cnc(NCCC2COCCO2)c1C)c1cc(CC)c(F)cc1 55510,C(=O)(C1=NNC(=O)CC1)NCC1CCC(F)(CNC(C=CC(CC)C)=O)CC1 55511,c1(C(=O)NC2C(CNC(=O)C=CSc3ccccc3)C2)ccc(Cl)s1 55512,N1(C(C(C(=O)NC)OC)=O)CCCN(C(=O)C(C)CC(F)F)CC1 55513,CCC(O)C(C)C(=O)N1CC(C(=O)NCCNC(=O)C2=C(C)OCC2)C1 55514,c1(C(N2CCC(N(C)C(c3coc(O)n3)=O)CC2)=O)cccc(C2CC2)c1Cl 55515,C(=O)(C1=CC2(CN(C(C3(C)CC(=O)N(C)C3)=O)C2)OC1)NCCCOC(C)C 55516,N1(C(C(=O)OCC)=O)CCC2C(CCCN2C(=O)C(O)CC)C1 55517,CC1(C)CN(C(c2coc(C#N)c2)=O)CCC1NC(=O)CN1CCCCC1=O 55518,CC1(C)CCOC1C(=O)NC1C=CCN(C(c2cnc(-c3ccccc3)s2)=O)C1 55519,CC(C)C(=O)C(=O)Nc1ccc(-c2ccc(CO)o2)cc1.C12CCCN(C1)C2 55520,N1(C(c2cc(COC)oc2C)=O)CC2CC(NC(=O)C3=CCCC3C)C1C2 55521,C1(C(=O)NCC(n2ccnn2)C)CCCCC1CNC(c1ccccn1)=O 55522,N1(C(C(=O)N(C2(Cc3ccccc3)CC(CO)C2)C)=O)CC(O)C(N)C1 55523,C(CS(=O)(=O)CC(=O)NCC(C1CCC1)NC(C1(c2ccno2)CCC1)=O)OC 55524,C(=O)(C(C)(C)C(F)(F)F)N(CCCCCNC(c1c(C)cn(C)c1)=O)C 55525,C1(C(=O)NCC2OCCC2C(N2CC3(CCOC3)C2)=O)CC2(CCC2=O)C1 55526,O=C(CCCCCNC(c1ncncc1Br)=O)Nc1ccccc1 55527,C1(C)(CCC)CN(C(c2cccc(OC3CC3)c2)C(=O)NCC(C)C)CCO1 55528,C(CCF)(C(=O)NCC1CC1(Cl)Cl)NC(Cc1cn(CC)nn1)=O 55529,C(=O)(C#CC(C)(C)CNC(=O)C#CC(C)C)N1C2CC(OC)C2CC1 55530,CC(C)C(F)C(=O)NC1CCCCC1NC(=O)CCSc1ccccn1 55531,Nc1ccnc(C(N2CC3(CC3)CC2CNC(c2csc(O)n2)=O)=O)c1Cl 55532,c1(C(=O)NC2CC(NC(C(C)N(C)C)=O)C(O)C2)cc(F)cc(S(N)(=O)=O)c1 55533,c1(C(=O)NC(CNC(C2(NC(N)=O)CC2)=O)CO)cc2n(n1)CC(F)C2 55534,c1(CC)ncc(C(=O)N(C(CNC(c2ccnnc2O)=O)CC)C)cn1 55535,CC(C)CC(C)(CNC(=O)CC1CC1)NC(c1ccc(N2CC=CC2)cc1)=O 55536,C#CCCCC(=O)NCCOCC(N1CCCC1(CC=C)CO)=O 55537,C1(CNC(C2N(C(C)=O)CCC2)=O)CC2(CO1)CN(C(c1sccc1C)=O)C2 55538,C12(C(=O)NCC(CC)NC(C3CCCOCC3)=O)CCC(O)(CC1)CC2 55539,CC(C)CC(C(=O)N1CC(NC(C2(C)CCN(C)C2=O)=O)CC(F)C1)C(N)=O 55540,Cn1nc(O)cc1C(=O)NC1C=CCN(N2CCCC(NC)C2)C1.C(N)=O 55541,N1(C(c2c(C)ocn2)=O)CCC(NC(=O)Cn2cc(CO)nn2)C12CC2 55542,c1(N(C)C)cccc(C(N2CCC2CNC(C2CCN(C)C2=O)=O)=O)n1 55543,N1(C(C(CC)C)=O)C2CCC1C(F)C(NC(c1nc(Cl)ccc1Cl)=O)C2 55544,C=CCC(C(=O)NCC1CC1CNC(C1CC2(CC2)CO1)=O)C(C)C 55545,c1(OC(C(=O)NCCC(C)(C)NC(C(COCC)C)=O)C)cccc(F)c1F 55546,O=S(=O)(c1cnccc1N1CCCC(c2nncs2)C1)NCc1ccccc1 55547,C(N=c1cc(C)[nH]c(=NCCc2ccnn2C)[nH]1)c1c(NC)cccc1 55548,CC1(CC(=O)NCCCNCCCNC(=O)CCc2cscn2)CCCC1 55549,C1(O)(CC(N2C(C(CC)O)CCC2)=O)CCN(C(C2CCCC2O)=O)CC1 55550,CC(C)(C)C(CNC(c1cccn2nccc12)=O)C(=O)NCC1(O)CCCOC1 55551,CCCC(O)C(=O)NC1CC(F)(CNC(=O)CCC2CCN(C)C2)C1 55552,C(=O)(C(F)(F)CCn1cc(CCC(=O)N(C)C)nn1)N(CCC(C)N(C)C)C 55553,c1(CNc2ncc(-c3cc(C(=O)OCC)c(C)cc3)s2)cnn2cccc(F)c12 55554,Cc1cc(CC(=O)NC2CN(C(c3cccnc3C)=O)CC2C)cc(O)n1 55555,C1(C(N2C(CCCNC(c3ccc(F)s3)=O)CCC2)=O)CC1C1CCOCC1 55556,c1(CCCC(N2CC(O)(CCNC(CC(C)O)=O)C2)=O)ccc(CN(C)C)cc1 55557,N1(C(C2(OC)CC2(F)F)=O)CCCN(C(=O)CC2CSCCS2)CC1 55558,N1(C(C2(C)CCCOC2)=O)CCN(C(c2cc(CO)on2)=O)C(CCO)C1 55559,CC(c1cccnc1)=CC(=O)NC1(C)CCCN(C(=O)CC2C=CS(=O)(=O)C2)C1 55560,Cc1ccc(OCC(=O)NCCCC(C)NC(C2(S(C)(=O)=O)CC2)=O)cc1 55561,C1(C(=O)NC(CC)CNC(C2CCSC(C)C2)=O)Cc2ccccc2N1 55562,c1(C(=O)NC2C(CNC(CC=C(C)C)=O)CC2)coc2cc(F)ccc12 55563,C(=O)(CC1CCOc2ccccc21)OC(c1ncccc1C)C(=O)OC 55564,C(N=c1nc(N(C)CCN2CCOC2=O)c2ccc(C)cc2[nH]1)C1C(C)=C1 55565,c1(N(CCOCCN(C(C(CC(=C)C)NC(C)=O)=O)C)C)cnn2ncccc12 55566,C1(C(=O)NC2C(NC(C34CC(C(C)C)(C3)C4)=O)COC2)COC(=O)N1C 55567,N1(Cc2ncc(N(C)C)nc2)CC2(CCCC2)C1c1nnc(O)n1C 55568,c1(C(=O)NCC(C)(C2CC2)NC(C23CC(C2)C3)=O)ccc(C(F)(F)F)cn1 55569,Cc1cc(Cl)c(Cl)cc1C(N1CC2CC2(CNC(c2cn(C)cn2)=O)C1)=O 55570,C1(C(=O)NCC2(C)CC2)CC2(CCN(C(=O)Cc3cccs3)CC2)C1 55571,CC(C)(C)C(=O)CCC(=O)N1CC(C(=O)NC2CC(=O)N(O)C2)C(C)(C)C1 55572,c1(OCCNC(C2C(NC(C3(C)CCCC3)=O)C2)=O)ccc(Cl)c(F)c1 55573,c1(C(N(C)CC2CCCN2C(=O)CC2CC2(Cl)Cl)=O)cnc(N)cn1 55574,C=CC1(CC(=O)NCCC2(CNC(=O)C(C)COC)CC2)CCOCC1 55575,C(c1ccccc1)=C(C(=O)NC(COC)CNC(C1(CO)CCCC1)=O)C 55576,C(=O)(CS(=O)(=O)C1CCCC1)NCCCC(C)NC(c1c(OC)csc1)=O 55577,Cc1nc(=N)[nH]cc1C(=O)NCC1C2CN(C(=O)C(C)Cn3cccn3)CC12 55578,c1(-c2nc(Nc3ccc(C#N)cc3I)sc2)ccc(C#N)cc1[N+](=O)[O-] 55579,c1(OC)ncc(CNC2CCC(C(=O)Nc3cnc(C)nc3)C2)cn1 55580,c1(CC)cccc(C(=O)NC2CC23CC(NC(=O)CCNC(=O)CC(C)C)C3)c1 55581,C1(OCC)CCCN(C(C2CCC=CC2NC(C2CCOC2)=O)=O)C1 55582,c1(CC(=O)N(C2CCN(C(=O)C(F)CC3CC3)C2)C)ccn(C(F)(F)F)n1 55583,CC(C)CC(C(=O)NC1CN(C(c2cnn(C)c2C#N)=O)CC1O)NC(N)=O 55584,CC1(C)CN(C(c2ncoc2C(F)F)=O)CC(CNC(=O)CCC2(C)CC2)O1 55585,Cc1nc2cc(C(=O)NCC(C)N(C(=O)CC3CC(O)C34CCC4)C)ccc2o1 55586,c1(C(=O)OCC)ccc(C2CCCCN2C(C2COC(C)C2)=O)n1C 55587,C(=O)(C1(C)CCc2ccccc21)N1CC(F)CC(NC(COCC(=O)OC)=O)C1 55588,CC(O)C(C)(C)C(=O)NCCCC1CCCCN1C(=O)C(F)=CC1CC1 55589,C(=O)(C1CCc2nccn21)N1CC2N(C(c3cc(OC)cc(C)n3)=O)C(CC2)C1 55590,C(C(=O)N(CCC(=O)N1CC(c2ccccc2F)C1)OC)NC(CCOC)=O 55591,S(=O)(=O)(c1ccc(Cl)cc1F)NC1C(C#N)CN(C(=O)Cc2cccs2)C1 55592,c1(CCNC(N2CCOC(Cc3ccccn3)CC2)=O)c[nH]c2cc(F)ccc12 55593,C(CCc1ccccc1)(C(F)(F)F)NC(C(n1ccc(C2CC2)n1)C)=O 55594,Nc1cc(F)cnc1C(=O)NC1CC(CCNC(c2sccc2C2CC2)=O)C1 55595,N#Cc1ccsc1C(=O)NCc1ncccc1C(=O)NOCC1CCCCC1 55596,N1(C(C=Cc2ccc(CC)o2)=O)CC(NC(c2cnn3c2OCC3)=O)CC1(C)C 55597,C(=O)(C(CC(C)(C)C#N)N1CCC(CSC2CCC2)CC1)NCCCSC 55598,C1(CCC)CN(C(=O)Cc2nccn2C)CC1NC(c1nscc1C)=O 55599,C(=O)(C1(C)CCn2ccnc21)NCC1(CNC(C=Cc2cn(C)nc2)=O)CC1 55600,c1(C(N(CCNC(CC=CCC)=O)CCC)=O)cc(Cl)cn1CC 55601,N1(C(C2(CC=C)CN(C(=O)CCSC)C2)=O)CCC2(CCC(OC)C2)C1 55602,C1(NC(C(CCC)(C)C)=O)CN(C(c2cnn(C)n2)=O)C2(CCOC2)C1 55603,C1(C(N2C(C(=O)NC3C(C(C)(C)C)C3)C(O)CC2)=O)CC2CC(=O)C1O2 55604,CC1(C)CC(NC(=O)CCC2CCCCO2)CN1C(=O)CC1CCCCC1O 55605,C(=O)(C1c2c[nH]nc2CN1C(C1CC12CCCCC2)=O)NC1CC(C(=O)OC)C1 55606,c1(CC(=O)NCCC2CCCN2C(=O)C(F)=C2CCC2)cc(F)c(Cl)cc1F 55607,C=CCCCCC(=O)N(CC(C)NC(C1CCN(CC=C)CC1)=O)C 55608,C1(C(=O)NCC(C(C)C)NC(C2CCN(C3CCCCC3)C2)=O)CCCC2CC12 55609,c1(C(=O)NCC2C(NC(C(CCSC)O)=O)C2)occ2c1CCOC2 55610,c1(C(=O)NC2C(NC(C=NOC)=O)COC2)cnc2c(c1)NC(=O)CS2 55611,N1(C(C(CC=C)(C)C)=O)CCC2CCC(NC(c3csc(CC)n3)=O)C1C2 55612,C(=O)(CC(C)C(F)(F)F)NCC(C(=O)NCCc1nnc(C)o1)N(C)C 55613,c1(CCC(=O)NC2CC(NC(C(=Cc3ccccn3)C)=O)C2)cc(F)ccc1F 55614,N1(C(C(N2CCSCC2)C)=O)CCCOC(CCNC(=O)CC(C)CN(C)C)C1 55615,C=CCCC(C)(C)C(=O)N1CC(CNC(=O)CC(C)N(C)C)C(O)C1 55616,C1(C)(NC(C(C)SC)=O)CCN(C(c2c[nH]c(=N)nc2O)=O)CC1 55617,C(=O)(C(O)C(C)(C)C)NC1CCN(C(c2cc(C)[nH]c2C)=O)CC1 55618,c1(C(N2C(CC(=O)NCc3scc(C)c3)COCC2)=O)cccc2[nH]ccc12 55619,c1(C(N2CCC(NC(C=CC(C)C)=O)CC(O)C2)=O)ccc(F)c2occc12 55620,c1(C(N2CC(C)C(NC(C3CC4(CC4)CN3C)=O)C2)=O)cc([N+](=O)[O-])cn1C 55621,CC1c2ccsc2CCN1CCOc1cc(F)ccc1F 55622,N1(C(C(C(=O)OCC)F)=O)CCN(C(c2ccnn(C)c2=O)=O)C(COC)C1 55623,C(=O)(C1=C(C#N)CCC1)NCCCC(C(=O)NC(c1ccccn1)C)O 55624,C12(CNC(COC3CCN(C(CCC(N)=O)=O)C3)=O)CCCC1OCC2 55625,C1(c2nc(-c3cccc(C)c3)nn2CC2CCC2)CCC2(C1)CC2(F)F 55626,C(=O)(C(=O)C(C)CC)N(CCCC(=O)OC)CC=C.C1C(=O)N1 55627,C(C)(C)(C(=O)NO)NC(C(C)N(C)C(c1ccnnc1)=O)=O 55628,N1(C(CCC2OCC(C)(C)C2)=O)CCOCC(NC(c2cccc(Cl)c2Cl)=O)C1 55629,c1(CC(N2CCC(O)(CCNC(CC(CC)OC)=O)C2)=O)ccc(OC)cc1F 55630,C(C1=CCCSC1)(c1n(CCCOC)nnn1)Nc1ccc(-c2ccno2)cc1 55631,c1(C(N(C)CC2N(C(C3ON=C(CC)C3)=O)CCOC2)=O)ccc2ncnn2c1 55632,S(=O)(=O)(c1ccc(N2CCC(C)C2)cc1Cl)NCc1cccc(OC)n1 55633,C(=O)(CC(C)C(F)F)N(C1CCN(C(CCC2CCC(C(=O)NC)O2)=O)C1)CC 55634,CC1c2c[nH]nc2CCC1C(=O)NC1CCN(C(=O)C(=O)C(C)(F)F)CC1C 55635,c1(C(N(CC(C)NC(C(C(C)C)OCC)=O)C)=O)ccc(Cl)cc1[N+](=O)[O-] 55636,C(CCC(C)C(=O)N1CCC(OCCNC(C23CC(OC)(CO2)C3)=O)C1)OC 55637,C(=O)(C1SCc2cccnc21)N1CC(CNC(COCCC)=O)C(F)(F)CC1 55638,c1(CNC(C(C=C=C)C)=O)ccc2c(c1)CCCC2NC(=O)C(C)(C)CS(N)(=O)=O 55639,C(CC(C(=O)N(C)Cc1ccoc1)NC(c1c[nH]nc1C)=O)OCC 55640,N1(C(COc2cccc(C)c2)=O)CC(NC(=O)CC(F)F)CC(C)C1 55641,c1(OC)ccc(C(=O)NC2CCN(C(c3cn(C)c(O)n3)=O)CC2C)c(F)n1 55642,C(=O)(C#CC1CCCOC1)NC(C)CN(C(=O)CCC(F)(F)F)C1CCCCCC1 55643,C1(CC)CN(C(=O)C(C)OCC(c2ccc(O)cc2)=O)CCN1CC(C)O 55644,c1(OC)cc(CC(C(=O)O)NC(c2ccc(C(C)=O)o2)=O)ccc1O 55645,CCCCC(C(=O)N(C)CC1CN(C(C2CCC(=O)N2)=O)CCO1)C(C)C 55646,C(=O)(CCC(N)=O)NC1(C(N(C)OCc2ccccc2)=O)CC1 55647,CC1OCCC1C(=O)NC(C1(CNC(c2ccc(CCN(C)C)s2)=O)CC1)C 55648,Cn1ncc2cc(C(=O)Nc3ccccc3CC(N3CC4CC4C3C#N)=O)ccc12 55649,N1(C(=O)NC2(CO)CCCC2)CC2CC(C1)C2N=c1[nH]nc(-c2cccnc2)s1 55650,N1(C(C2OCCN(C(CC(C=C)CC)=O)C2)=O)C2CCCC1CN(C)C2 55651,N1(C(C(Cc2ccc(OC)cc2)C)=O)CCN(C(=O)CSC)C(C(F)F)C1 55652,c1(CC)c(C(=O)N(C)CC2CCN(C(=O)CSC)C2)nnn1C 55653,N1(C(c2cc(C(C)C)no2)=O)C(C(=O)NCCOC(F)(F)F)CC2CCCC12 55654,C(C(N=[N+]=[N-])C(=O)N1CC(NC(C2CC2C2CCCC2)=O)CCC1C)OCC 55655,CN1CCN(C(c2cscc2C(N)=O)=O)C(CNC(C2CCCCNC2=O)=O)C1 55656,C(CC(=O)N(C)C(C1CCC1)C)(C(F)F)NC(c1c(C)cncn1)=O 55657,c1(NC(c2c(-c3ccccc3)ccs2)c2ccccc2)ccc(C)cc1.c1(S)nn[nH]n1 55658,Cc1ccc(C(=O)NCC2CCCCN2C(c2cnsc2)=O)c(N)n1 55659,c1(C(N(C)CC2N(c3nccc(OCC)n3)CCOC2)=O)cc(F)cc(Br)c1C 55660,CCCC(CCC)=CC(=O)NCCOC1CCN(C(C2C3(CC3)C23CC3)=O)C1 55661,CC(C)C1=NOC(C(=O)NCC2(O)CCCN(C(=O)C=C(Cl)CCN(C)C)C2)C1 55662,Cc1ccnc(O)c1C(=O)NC(C)CNC(=O)Cc1nnc(-c2ccccc2)o1 55663,C(=O)(C1=CC2C=CC(C1)C2)N1C(C)(C(N2CCC=C(C)C2)=O)CC(O)C1 55664,N(C(=NCCC(F)F)NCC(=C1CCNC1)F)Cc1cccc(CCC)c1.C(C)=C 55665,C1(NC(CCCc2onc(C)n2)=O)CN(C(=O)CC23CCCC2C3)CC1C(F)F 55666,c1(C(=O)NCCC(C)N(C(Cc2cc(C)on2)=O)C)cccc(C(C)(F)F)c1 55667,C(CCN=c1[nH]c2ccc(Br)cc2s1)OCCNC(C1CC2C=CC1C2)=O 55668,c1(C(N2CC3C(C(=O)OC)C3C2)=O)ccc2cccc(OC)c2n1 55669,CC1(CNC(c2ncoc2-c2cccs2)=O)CCCN1C(=O)CSS(C)(=O)=O 55670,C#Cc1cnc(C(=O)N(CCC(C)NC(c2cccc(CC)c2F)=O)C)c(C)c1 55671,n1(CC(=C)C)c(SCCCn2cccnc2=O)nnc1-c1ccccc1 55672,c1(Nc2ccc(N(C3CCCC3)C(=O)NCC(=O)OC)cc2)cccc(F)c1[N+](=O)[O-] 55673,C1(CC)(CC)CC(NC(=O)CN2CCOCC2)CN1C(=O)C#CC(=O)N(C)C 55674,c1(C(=O)Nc2cnn(C)c2Cc2ccccc2)nn(C)c2c1CC(F)(F)CC2 55675,c1(C(=O)NC(C(=O)NCC(N2CCCC2)C)c2ccco2)cccc(O)c1F 55676,C1(OC)CCN(C(=O)CC2CCN(C(=O)C(N)=O)CC2)C1C 55677,C1(C(=O)OCCOc2[nH]cnc2C(=O)NCc2ccccc2)C(F)(F)C12CCC2 55678,C(=O)(C(C)CCCOC)N1C(CC(NOCC(CC)C)=O)CCC1 55679,C1(C(N(CCCNC(=O)CC2CC(O)C2(C)C)CC)=O)CC2(C1)CC(O)C2 55680,C1(CNC(c2cc(=N)[nH]cc2)=O)CCC2(CO1)CC(NC(=O)CNC(N)=O)C2 55681,C1(C(=O)NC(C2CN(C(CC=CCC)=O)C2)C)CCC(C)C1 55682,C12(CNC(C3CC(C#C)(O)C3)=O)CCCC1N(C(=O)Cc1occc1C)CCC2 55683,c1(NC(=O)NC2CC2c2ccc(-n3cnnn3)cc2)ccc(C(F)(F)F)cc1 55684,n1(CC(C)C)nc(CNc2cccc(F)c2)nc1-c1ccc(CC2CCC2)nc1 55685,C(CCCC(C)NC(=O)CC1CCC12CCC2)NC(c1cnc(OC)s1)=O 55686,C=C1CON(C(=O)CC2CCN(C(=O)COc3ccc(C)cc3)C2)C1 55687,N1(C(C(COC)(C)O)=O)CC(NC(c2ccc(OCCF)cc2F)=O)CC(O)C1 55688,N1(C(=O)NC(c2cc(C)ccc2C)CC)CCc2cc(Cl)ccc2C1 55689,C=CCC(C)C(=O)NC1CCC1CNC(c1cnn(C)c1COCC)=O 55690,C1(OCC(=O)N(CCN(C(CN(C)C)=O)CO)Cc2ccccc2)CCCCC1 55691,N1(C(=O)Cc2ccsc2)CCN(CC(N2CCC(c3cc(O)ns3)C2)=O)CC1 55692,C1(C(N(CC(C)O)CCNC(c2ccn(CC(F)F)n2)=O)=O)CC12CC(F)(F)C2 55693,C1(O)(C(C)NC(=O)C=CCn2cccn2)CCN(C(=O)Cn2cnnc2)C1 55694,CC(CC(=O)N1CCCC1C(C)(C)NC(=O)CC1CCCCCCC1)C(C)(C)C 55695,CC(C)C(CNC(=O)CC(=O)N(C)C)C(=O)N(C1CCCC(O)C1)C 55696,CCCC(CCC)=CC(N1CCC(CNC(=O)CSc2nnnn2C2CC2)C1)=O 55697,CC(C)CC(O)CC(=O)NC(C1CCCN1C(=O)CCC1CC1(F)F)C 55698,C1(NC(C2C(=C)C2SC)=O)CCN(C2CN(C(=O)CC(OCC)OC)C2)CC1 55699,C(=O)(CCCCCO)N1C(C)CC(NC(c2ccc(CN=[N+]=[N-])cc2)=O)C1 55700,N#Cc1c[nH]c(C(=O)NC2CCCC2C(N2CCC(CCO)CC2)=O)c1 55701,C1(CC(C)NC(C2(C=C)CCC2)=O)CC2CCC(C1)N2C(C1CCN(CC)C1)=O 55702,C1(C(=O)N([N+](C)(C)C)CCSC)CS(=O)(=O)CCO1.CO 55703,c1(C(C(=O)NC2CCCC2)N(CCOC)C)cc(OC)c(F)cc1F 55704,N1(C(C(=CC2CCCC2)C)=O)CCCC(CCNC(c2cc(C)ccn2)=O)CC1 55705,c1(C(=O)NCC2N(C(c3c(C)cn(C)c3)=O)CCC2C)cc2c(C)n[nH]c2cn1 55706,C12(C(=O)NCC(CC)NC(c3cc(C(N)=O)n[nH]3)=O)CC(c3ccccc3)(C1)C2 55707,c1(CN2C(C(=O)Nc3c(C(C)=O)cc(C)s3)CC(F)(F)C2)cc(Br)c(O)cc1O 55708,C#CCC(C)(C)C(=O)N1CCC(COC)(NC(C2CC2CC(C)C)=O)C1 55709,c1(CC(N2C(C)(CNC(C(C)OCCC#C)=O)CCC2)=O)cc(F)cc(Cl)c1 55710,c1(CCC(=O)NCCCCNC(C2CC3CC3C2)=O)ccc(F)c2ccccc12 55711,c1(NCC(C(C)C)O)ccc(S(=O)(=O)NC2CC3OCCCC23)c(Br)c1 55712,N1(C(C(CO)OC)=O)CCN(C(c2cc[nH]c(=N)c2)=O)CC1C1CCC1 55713,C(=O)(CC1CCCc2c1[nH]c1ccccc21)N1C2C(CN)C(C(=O)OC)C1CC2 55714,C1(COC)CN(C(=O)COC(F)(F)F)CCN1C(=O)CC1CCCOC1 55715,C1(CC(N2CCOC(CNC(C3(F)CCOC3)=O)C2)=O)C=CS(=O)(=O)C1 55716,N1(C(CC(=O)N(C)C)=O)CCCC(O)(CNC(c2ccc(=O)n(C)c2)=O)CC1 55717,C1(OC)CC2CC(NC(=O)NCCC(C)(C)CSC)CC12 55718,N12CCC3CN(CC13)CC(=O)C2=O.C(=O)(C(C)NC(C)=O)OC 55719,C1(C(N2CC(CC(C)(C)C)C(NC(C3CCOCC3)=O)C2)=O)COCC(C)(C)O1 55720,N1(C(C)=O)CCCCC1C(=O)NCC=CCNC(c1sc(F)cc1Br)=O 55721,c1(CCC)ncoc1C(=O)NC1CCC1.C(C)(CNC(=O)OC(C)(C)C)NC=O 55722,c1(NC(=O)CC2CN(C(c3csnn3)=O)CCO2)cc(C(F)(F)F)cc(Cl)c1 55723,C1(NCC(c2ccccc2)OC)CN(C(=O)C(=O)NC2CC2)CC1CC(C)(C)C 55724,C1(NC(CC2(C)CC2(Cl)Cl)=O)CC2CC(C1)N(c1ncc(Br)c(O)n1)C2 55725,Cn1cncc1CC(=O)NCc1ocnc1C(=O)NOCC1CCCCC1 55726,Cc1ccc(C(=O)NCCC2CCCN(C(c3ccn(C4CC4)n3)=O)C2)c(C)c1 55727,C1(O)(CCNC(=O)C(O)C2CCC2)CN(C(=O)CC2CCOC2=O)C1 55728,C(C(CC(C)C)C(=O)N1CCCC(NC(c2cnc(Cl)cc2N)=O)C1)OC 55729,c1(C(=O)NCC(C)N(C(c2cccc(CC)c2)=O)CC)cnc2n1CCC(C)C2 55730,Cc1cnc(CN2CCCC(C(N3CCCC(N(C)C)C3)=O)C2)cn1 55731,C(=O)(C1(C)OCCc2ccccc21)NCCN(C(=O)CCN1CCCC1=O)CC 55732,c1(C(N2CC3C(NC(C(CC)C(=O)OC)=O)C3C2)=O)cc(S(N)(=O)=O)ccc1F 55733,c1(OC(C2CCC(C)(C)CC2)C(=O)OC)cc(=O)c2cc(Cl)ccc2o1 55734,c1(CC)ccc(OCC23C(C(N(C4CCN(CC)C4)CC)=O)(CCC2)C3)cc1 55735,c1(OCC)cncc(C(=O)N(C)CCNC(=O)C(C2CCCO2)C2CC2)c1 55736,CCCCC(O)C(=O)NC(C1CCN(C(c2cccc(CN(C)C)c2)=O)C1)C 55737,C1(C(=O)NC(C2(O)CCN(C(=O)COC3CCC3)C2)C)COCCN1C=O 55738,C(c1ccc(Br)cc1)=CCN(c1n(CC(=C)C)c(-c2cccn2C)nn1)C 55739,c1(C(C(=O)NCCSC)N(CC=C)CC#N)nccc(Cl)c1F 55740,c1(C(C(=O)NC(C)C)N(CC=C)Cc2cccnc2)c(Cl)c(C)nn1C 55741,c1(NC(C=CCOCC)=O)ccoc1C 55742,c1(C(=O)NCC2CN(C(=O)C(F)(F)CC3CC3)CC2(F)F)cccc2c1CCO2 55743,N1(C(C(c2ccccc2)C)=O)CCC(CCCNC(C2CC2Cl)=O)CC1 55744,C(=O)(C(C)C1=CCCC1)N1CCCCC(N(C(c2cccc(C#C)c2)=O)C)C1 55745,CC(C)CCN=C(NCCC1C(O)CCN1C(=O)OC(C)(C)C)NC1CC1 55746,CCC(C)C(C)NC(C1(CCNC(=O)C(C)c2cccs2)CC1)=O 55747,CCC1=NOC(C(=O)NCC2CC(C)N(C(=O)CCc3cnccn3)C2)C1 55748,c12ccc(nc1)c(=O)[nH]2.CCC(C(=O)NCC(C)(O)C1(C)CC1)NC(C)=O 55749,c1(N(CC(=O)N(CC(=O)NCC)CC2CC2)C)cc[nH]n1.C1(=O)CCOC1 55750,C(CC(C)C(=O)NC1CC(N(C)C(c2cnc(N3CCOCC3)s2)=O)C1)OC 55751,c1(N2C(=O)CC(C(N3CCC(OC)C3)=O)C2)ccc(Cl)c(F)c1 55752,c1(C(C(N2CCC(C(=O)NCC(=O)N(CC)CC)CC2)=O)=O)ccc(F)c(C)c1 55753,CCCCCCC(C)C(=O)NC(CC1CCC1)C(N1CC2CCC(C1)C(=O)N2)=O 55754,CC(Cc1ccnn1C)C(=O)N1CCC1CNC(=O)CCc1ccccc1 55755,c1(N2CC(CC)OCC2)nc2c(c(=NCC(CC(C)C)OC)[nH]1)COCC2 55756,c1(C(C(=O)NCCC)N(C)CC2CCOCC2)cc(OC)c(Br)cc1OCC 55757,Cc1ccc2c(c1)C=C(C(=O)NC1CCOC(CNC(C3CC3F)=O)C1)CO2 55758,N1(C(C(CCC)O)=O)CC2CC(C1)CN(C(=O)C(F)C(F)(F)F)C2 55759,C(=O)(C(CC1CCCC1)C(C)C)N1CCC(N(C(Cc2c(C)onc2)=O)C)CC1 55760,C(CC(F)CN=[N+]=[N-])NC(C(CC=CC)NC(C1OC2CCC1C2)=O)=O 55761,c1(OC)[nH]c(=N)ccc1C(N1CCN(C(C)CNC(C2CCCCS2)=O)CC1)=O 55762,N1(C(C2C(C)C2C)=O)CCC(CNC(=O)C=CCn2cncn2)C1(C)C 55763,CC1CN(C(=O)CC(F)F)CC(CCNC(=O)C(c2ccccc2F)(C)C)O1 55764,CCC(C)C(O)C(=O)N1CCCCC1CNC(C1(O)CC1)=O 55765,CC(C)C(CCC(=O)NC(C)(C)CF)NC(=O)Cc1cn(C)cn1 55766,C#CC1(C(=O)NC(C)COCC)CCN(C(=O)C2=CCCSC2)CC1 55767,c1(CC)ccc(C)nc1N(CC(C)CNC(C1CCOC(C)(C)C1)=O)C 55768,C1(C(N2C3C(CNC(C4CC(=C)C4)=O)C(C3)C2)=O)CCC2CCC(=O)N12 55769,C1(F)(CNC(=O)C=Cc2ncco2)CC2CCC(C1)N2C(=O)CC1CC=CC1 55770,C(=O)(C(F)C(F)(F)F)N(C(CNC(c1cccc(CC)n1)=O)C)CC 55771,C(=O)(C1=NNC(=O)CC1)NCCN(C(c1ccc(Br)c(N)c1)=O)CC 55772,C=CCC(C(=O)NCCC1(CNC(=O)CN=S(C)(C)=O)CC1)C(C)(C)C 55773,CC1=C(C(=O)N2CC(NC(C3(C)CCCS3(=O)=O)=O)C(F)C2)SCCO1 55774,N1(C(C(CC)CO)=O)CCC(NC(C2(O)CCSC2)=O)C(C)C1 55775,[N-]=[N+]=NCC(C(=O)NCCOC1CCCC1)NC(C1CC2(CC2)CO1)=O 55776,c1(C(=O)NC2CC(NC(c3cncnc3)=O)C2)cnc(O)cn1.C1(S)CC1 55777,N1(C(C(CCC)C)=O)CCC2(CC1)CN(C(C1C=C1C)=O)C2C(C)C 55778,c1(OC)ccccc1CC(=O)N1CCC1CNC(c1oncc1C)=O 55779,c1(CC)cc(C(N2CCC(=CCNC(=O)C(C)SC(C)C)CC2)=O)c(C)nn1 55780,CCC(CC)C(C)C(=O)NC1CCN(C(c2ccnc3ccsc23)=O)C1(C)C 55781,C1(CC(=O)NC2(C#C)CC2)COCCN1C(=O)Cc1cnoc1 55782,C1(CC=C)(NC(c2cnn(C3CC3(F)F)c2)=O)CCN(C(C2CCSC2)=O)C1 55783,c1(CC)c(NC(CN(C(C)C)CC)=O)cnn1C(CC)CC 55784,c1(C(=O)NC2CN(C(C3(C(C)(C)C)CCC3)=O)CC2F)ccc(=O)n(CCF)n1 55785,CC1(C)CC(c2nnnn2CCOC(F)F)(NC2COC2)N=C1C#N 55786,C(CCCCC(=O)N1CC2CC(C1)C2NC(c1ncc(N)cc1Cl)=O)OC 55787,N1(C(C2N(C(C)=O)CC(O)C2)=O)CC2CCC2(NC(C2(CC3CC3)CCC2)=O)C1 55788,CC1(C)CCN(C(C2CCN(C(=O)CC3CCC(=O)N3)CC2)=O)CC1 55789,c1(CC(=O)N(C)CCNC(C2(Cc3cc[nH]c3)CC2)=O)ccc([N+](=O)[O-])cc1Cl 55790,C(C(=O)N1CCCO1)NC(C1(CC#C)CCN(C(=O)C(C)CC2CC2)C1)=O 55791,Cn1nc(Br)c2ccc(C(N3C4CN(C(C5CC5C5CC5)=O)CC34)=O)cc12 55792,C(=O)(CC(CC)C(C)(C)C)NCC(CN(C(=O)CC(C)C1CCCC1)CC)(C)C 55793,CC1(C)C2CCC1(CC(N1CCN(C(=O)C#CC3CC3)CC1C(F)F)=O)CC2 55794,N1(C(C(CC)SC)=O)CCCCC(NC(c2cc(CCOC)on2)=O)C1 55795,c1(NC(C2CC23CCN(C(=O)C=Cc2ccoc2)C3)=O)cc(I)ccc1CO 55796,N1(C(C2(C)CCN(C(CC(C(C)C)O)=O)C2)=O)CCC(C)C2(CCC2)C1 55797,c1(C(=O)NC2C(C)CN(C(c3ccn(C)c3)=O)C2)nnn2c1CSCC2 55798,N1(C(c2ccnc(C)c2C)=O)CCOC2(CCN(C(c3[nH]cnc3C#N)=O)C2)C1 55799,N1(C(C(C)N(C)C(C2CCC(CO)CC2)=O)=O)CCCC(CCO)CC1 55800,C=CCC(CNC(c1ccccc1CC#N)=O)C(=O)Nc1ccc(O)c(C)c1 55801,c1(CNC2(CC(=O)Nc3ccnc(Cl)c3I)CCC2)c(Cl)[nH]c2ccccc12 55802,C1(C(N2CCC(CC(C)C)CC2)=O)CC2(CC2)CN1C(C1CC(OC2CC2)C1)=O 55803,c1(C(=O)NCC2CC(OC)CN2C(c2cnccc2Cl)=O)ccc(=O)n(C)n1 55804,CC(C)CCCC(=O)N1CC(O)CCC1C(=O)NCc1cccnn1 55805,Cc1cc(C(=O)NC2CC2C(=O)NCCOc2ccc(Br)cc2)c(C)n1C 55806,c1(C(=O)NC(C(C)C)(C)CNC(C2(O)CC2)=O)ccn2cnnc2c1 55807,c1(CNCc2noc3c2CC(C)CC3)cc2c(cc1O)OCO2 55808,c1(NCCc2nc(C)oc2C)nc(N2CCc3sccc3C2)nc2sccc12 55809,C(=O)(CCCCC(N)=O)NC1CCC(N(C(COc2c(C)cccc2Cl)=O)C)C1 55810,C(C(CC(F)(F)F)NC(C1CC1C(F)(F)F)=O)NC(c1cnc(OCC)nc1)=O 55811,C(C)(CNC(=O)Cc1cnc(C(F)(F)F)s1)(CO)NC(C(C)OCCC(C)C)=O 55812,C1(C(C)NC(c2ccsc2C(F)F)=O)CCCCN1C(C1CCCCO1)=O 55813,Cc1coc(C)c1C=CC(=O)NC(C1CCCN(C(C2CC(F)(CO)C2)=O)C1)C 55814,c1(C(=O)NCC(CNC(CCC=CC)=O)CO)cnn(C(C)CC)c1C 55815,c1(OCC)nc(C(=O)NC(C)C(C)NC(c2ccn(C3CCOCC3)n2)=O)ns1 55816,c1(CC(=O)NCCC(=O)N2CC(=C(F)COC(C3C(C)=C3)=O)C2)cccc(F)c1 55817,c1(C(=O)NCC2CC2NC(c2coc(O)n2)=O)cc(Cl)cc([N+](=O)[O-])c1 55818,N1(C(CCC(CC)OC)=O)CCC(C2CCN(C(c3c(C)noc3C)=O)C2)CC1 55819,C1(F)(NC(C2C(CNC(CCCCOCC)=O)CCOC2)=O)CCCCCC1 55820,C12(CNC(C)=O)CC(CO1)N(C(c1sc(Br)cc1Cl)=O)C2 55821,C(=O)(CCC(C)CN(C)C)N1CCC(N(C(=O)CC2CC23CC3)CCC)C1 55822,CC1(C)CCCN(C(c2cncs2)=O)C1C(=O)NC(CCO)C1CC1 55823,C#CCCN=C(NCc1cnccc1Br)NC(C)CC 55824,c1(C(N2C(CNC(C3(C)CCOC3)=O)CC2)=O)ccc(Cl)cc1C(N)=O 55825,C1(C2CC2)(C(N2CCC(NC(c3sccc3F)=O)CC2)=O)CC=CC1 55826,c1(C(=O)NCC2(CCNC(CC)=O)CC2)cccc(C2(S(C)(=O)=O)CC2)c1 55827,C(=O)(C(CNC(=O)CCC1CCC1)CC(C)C)NCCc1ccc(C)s1 55828,C(=O)(C(CO)C(C)(C)C)NCC(CCC)C(=O)NCc1cccnn1 55829,N1(C(C2CC3(CC3)C2)=O)CCN(C(c2cccc(C)n2)=O)C(C)C1C 55830,Cc1cc(F)ccc1NC(C1CC2CC1CC2NC(c1cccc(F)c1F)=O)=O 55831,c1(CNC(N(C2C(C)CCC2)C)=O)cccc(C#CCC2CCCC2)c1 55832,C12(CNC(=O)NC(C)C(=O)Nc3cnn(C)c3)CCCC1CCC2 55833,c1(CNC(=O)Cc2cnoc2)ccnc(C(=O)NC2CCS(=O)CC2)c1 55834,C(CN=C(NCC(F)F)NCC1(CN(C)C)CCOCC1)=CC 55835,N1(C(C(C)n2cncn2)=O)CCOCC1CN(C)C(c1nccnc1C(N)=O)=O 55836,c1(NCC(C)S(C)(=O)=O)ccc(S(=O)(=O)N2CCOC(c3ccsc3)C2)cc1Cl 55837,O=C1CN(C(=O)CC2COCCO2)C(C(N2CC(CC(F)(F)F)C2)=O)CN1 55838,CC(C)C(F)C(=O)NCc1ncc(C(=O)NCC2COCC(C)O2)cn1 55839,C1(CCNC(C(C=C)(C)C)=O)CN(C(c2coc(N(C)C)n2)=O)CCCO1 55840,N1(C(CC(=C=C)C)=O)CC2(CCN2C(=O)Cc2ccc(C(=O)OC)nc2)C1 55841,C1(CN(C(C(Cn2ccc(C)n2)C)=O)C)CCN(C(=O)CSCC(N)=O)CC1 55842,CCC(C)CC(C)C(=O)NC(CNC(c1ccccc1CO)=O)(CC)CC 55843,c1(NCC2(O)CN(Cc3sc(C)c(Br)c3)C2)ccnc2ccnn12 55844,N1(C(C(Cc2ccc(C)cc2)NC=O)=O)CCCN(C(C2C=CCC2)=O)CC1 55845,N1(C(c2c(C)cn(C)c2)=O)CCCC(O)(CCNC(=O)C=C2CCC(C)C2)C1 55846,C12(CNC(c3nc(C)n(C)c3)=O)CCCC1CN(C(=O)C(F)(F)CC(C)C)C2 55847,C(N=c1ccnc(C(C2CC(F)(F)C2)C2CCCCC2)[nH]1)c1ccc(C)c(Br)c1 55848,C1(C#N)(CC(=O)NCCCN(C(C)C)C(C2CCCS2)=O)CC1 55849,c1(NC(c2nnn(C)n2)c2n(CC3CC3)nnn2)ccc2c(c1)CC(O)C2 55850,C(N=c1[nH]cncc1Br)C1(C)CCN(C(c2ccn(C)n2)=O)C1 55851,C=C=CC(C)C(=O)N1CCC(OCCNC(C2CCC(=O)N2CC)=O)C1 55852,Cc1nn(CC(=O)NC2CC(NC(=O)CC3(C(F)(F)F)CC3)C2)c(C)c1[N+](=O)[O-] 55853,c1(NC2C(C)COCC2)[nH]c(=NCc2sncc2Br)nc2c1ncn2C 55854,c1(C(N2CCCC(CCNC(CC(C)F)=O)C2)=O)ccn2ncccc12 55855,CC(C)(CNC(=O)CC1CCC1)CC1CN(C(c2cnc(C(C)(F)F)s2)=O)C1 55856,CCCCCC(=O)NC1COCCC1NC(c1cnc(C2CC2)[nH]1)=O 55857,C1(CNC(C(C)OCCC=C)=O)CCN(C(c2ccc(CC)[nH]2)=O)C(C)C1 55858,c1(C(C)NC(=O)Nc2cn(CC(=O)OC)nn2)cccnc1O 55859,C1(CC=C)(NC(c2cnn(C)c2OC)=O)CCN(C(=O)CC2CC2C)C1 55860,C(=O)(C1=NOC(C)C1C)NC(C1N(C(c2ccc(OC)cc2OC)=O)CCC1)C 55861,C(CC(C)(C)C)(C(=O)NCCC1(NC(=O)Cc2cn(C)cn2)CC1)OC 55862,c1(C(N(C)Cc2ccc(C)cc2Br)=O)n[nH]c2cccc(F)c12 55863,C1(NC(c2cn(C)nc2)=O)CN(C(C2CCCS(=O)(=O)C2)=O)CCC1F 55864,Cc1ccc(C=CC(N2CCC(NC(=O)CC3(C)CCCO3)CC2)=O)s1 55865,C(CN=c1[nH]c(=NC2CCC(C3CC3)CC2)[nH]c2c1SCC2)OCCOC 55866,C1(C(N(CCC(C)NC(c2ccnc(OC)n2)=O)C)=O)COc2ccccc2O1 55867,CN1C(=O)CCC1C(=O)NC1CC(C(=O)NCCC(N)=O)C1 55868,CC(C(=O)N1CCCC(NC(c2cnc(N)c(CO)c2)=O)C1)C(C)(F)F 55869,C(C(=O)N(CCCNC(=O)C=CC(C)C)C(C)C)(SC)SC.C1(N)CC1 55870,C1(C)(C(N(C(C)CNC(c2ccc(F)c(C(F)F)c2)=O)C)=O)CC(C2CC2)=NO1 55871,N1(C(C(CC=C)C(=C)C)=O)CCC2(CCC2C(=O)NCc2cc(Cl)ccn2)CC1 55872,c1(C(=O)NCC(CCCC)NC(=O)C(O)C(C)(C)CC)cccc2ccncc12 55873,Cc1c(C(N2CCC(Cn3cc(C(C)(C)C(C)C)nn3)CC2)=O)ccn1C(C)C 55874,c1(C(N2C(CNC(CC(C)N(C)C)=O)CC3(CC3)C2)=O)cccc2nccn12 55875,C1(NC(c2c(C)cc[nH]2)=O)CN(C(=O)Cc2ccccc2CS(N)(=O)=O)CC1O 55876,N1(C(C(N(C(CC(=O)OCC)=O)C)C2CC2)=O)CCOC(C)(C2(C)CC2)C1 55877,N1(CC(=O)NCCCCC2CN(C(Cc3c(C)ncs3)=O)C2)CCN(C)C(=O)C1 55878,N1(C(C(COC)C)=O)CC2(CCN(C(=O)C(C)Cc3ccncc3)CC2)C1 55879,N1(Cc2nc(C(C)C)on2)CCC(C)(CNC(=O)C(c2ccc(F)o2)C)CC1 55880,c1(C(C)OC(C)C)nc(-c2cc[nH]n2)nn1CC(C)(C)O 55881,C(C)(C(CC(=O)NC(CC1CC1)COC)NC(C1CN2CCN1CC2)=O)OC 55882,Cc1cnc(CC(=O)N(C2CCN(C(C3CCSC3)=O)C2)CCO)s1 55883,N1(C(C2CC=C(C)CC2)=O)CCCC(CCNC(=O)C=CC(C)C)CC1 55884,C1(C(N2CC(NC(=O)OC)C2)=O)CC2(CC(NC(c3c(C)nn(C)c3N)=O)C2)C1 55885,C1(C(C)NC(=O)C2=CCC2)CN(C(c2ccn(C)c2)=O)CCO1 55886,C(CC(C(=O)NCCC(F)Cn1cc(-c2cnsc2)nn1)OC)OC 55887,Cc1c(C(=O)NCC2CC2NC(C2CS(=O)(=O)C2)=O)cnn1C(C)(C)C 55888,Cc1c(C(=O)NCC2CCN(C(C3C4(CC4)C34CC4)=O)CC2C)sc2cncn12 55889,C1(C(=O)NC(CC)CSC)CN(C(c2ccc(CO)cc2)=O)CC(C)(C)C1 55890,C1(O)(CNC(C(C)(C)c2cccs2)=O)CCN(C(=O)CCOCC2CC2)C1 55891,c1(C(=O)NCCN(C(C2CC3OC(=O)OC3C2)=O)CC)nn(C)c2c1CCC2 55892,C1(NC(c2occ(C)c2)=O)CCCCC12CCN(C(c1cnc(F)c(C)c1)=O)C2 55893,C(=O)(C1CCCc2cccnc21)N1CCC(C)C1CNC(=O)CC1(O)CCCC1 55894,N1(C(c2c(C)nc(O)cc2)=O)CC(CNC(=O)C(C)n2cnnn2)CC(C)(C)C1 55895,C1(NC(C(C)NC(N)=O)=O)CCC(N(C(=O)Cn2cnc(Br)n2)C)CC1 55896,N#Cc1ccc(CN2CCCC(NC(c3ccnnc3O)=O)C2)c(Br)c1 55897,c1(C(=O)NC(c2ccc(Cl)c(Cl)c2)CN(C)C)nc2ccccc2s1 55898,N1(C(c2cnc(C)[nH]2)=O)CCC(NC(c2[nH]cnc2C)=O)C(CO)CC1 55899,C1(NC(C2CC(OC)C2)=O)C2CCC1N(C(=O)Cn1nc(C)cc1C(F)F)C2 55900,CN1CC(C(=O)NCCN(C(C2(CC(N)=O)CCCCC2)=O)CC2CC2)CCC1=O 55901,N1(C(C(C)=NOCC#N)=O)CCCC(CCNC(c2ccc(C)c(O)n2)=O)CC1 55902,c1(C(=O)NCC(C)N(C)C(C2CCC(C)(C)O2)=O)cccc(O)c1F 55903,C12C3CN(CC13)C2=O.CCC(C(=O)NCC1(C(F)(F)F)CC1)N(CC)CC 55904,N1(C(c2ccnc(OC)n2)=O)CCC(C)N(C(c2ccncc2C)=O)CC1 55905,c1(C(N(C(CNC(c2cc(C(=O)OC)no2)=O)C)C)=O)noc2c1COCC2 55906,C1(CC(=O)NC(CCC)CO)CN(C(=O)Cc2ccsc2)CCC1C 55907,C(=O)(CC(CCC)NC(C1(C2(C)CC2)CC1)=O)N1CCC(C=C)C1 55908,C1(C(=O)NCCC(C)N2CCCC2)(CC)CCN(C(C2CC2C(F)(F)F)=O)C1 55909,C1(C(C)(C)C)(C(N2CC(CC(C)NC(=O)CCc3cncs3)C2)=O)CCCC1 55910,C1(CO)CN(N2CC3CCCC(C3)C2)CC12CCOCC2 55911,N1(C(C2(C)CC(C)(C)C2)=O)CCN(C(C2CC=CCC2)=O)C(CC(F)F)C1 55912,c1(C(=O)NCc2cn(CCNC(CC=CC=C)=O)nn2)ccccc1C 55913,N1(C(c2scc(C(=O)OCC)c2)=O)CCC(N2CCC(N)C2)CC1 55914,n1(CC(=O)N(C(c2ccccc2)CO)CC2CCS(=O)(=O)C2)ccc([N+](=O)[O-])n1 55915,C1(NC(C2(C)N(C(C3C(C)CC=CC3)=O)CC=C2)=O)CCC2(CCC2)C1 55916,n1(CC)cnc(C(=O)NC2CCCC2CNC(C23CCC2C3)=O)c1 55917,N(C=CC(=O)C(F)(F)F)C(C1CCN(C(c2cccc(I)c2)=O)CC1)=O 55918,C12(CNC(c3c(C)ccc(N)c3)=O)CCC(NC(=O)CSS(C)(=O)=O)(CC1)CO2 55919,c1(CC(N2CC=CC(NC(CC3C(C)(C)C3)=O)C2)=O)cnc2ccccc2c1 55920,C1(NC(C2CCC3(CC2)CC3)=O)CS(=O)(=O)C12CCN(C(=O)CCC(F)F)CC2 55921,CC1(C)C(C(F)(F)F)CCN1C(c1cc(C(F)F)ncn1)=O 55922,N1(C(CCCC2C(C)C2)=O)CCN(CC(=O)N(C(C)(C)C)CCO)CC1 55923,N1(C(C(=O)NC(C(=O)OC)C)C(C)C2CCOC2)CCS(=O)(=O)CC1C(=O)OC 55924,CCCCC(C)(F)C(=O)NCC1CC(C)CCN1C(c1cccc(C)n1)=O 55925,c1(-c2cc(NCCN(C(C)C)CC)ncc2)c[nH]c2cc(C(=O)NC)ccc12 55926,C(=O)(C(C)S(N)(=O)=O)NCC1(C(N)=O)CN(C(c2c(C)cc(SC)o2)=O)C1 55927,c1(CC)ccnc(C(N2CCC(C(=O)N(C)CC3(O)CCC3)C2C(C)C)=O)c1 55928,C1(CN(C(C2C(C)(C)C2(C)C)=O)CC)CCCCN1C(c1ccnn1C(C)C)=O 55929,CCC(CC(=O)NCC(CO)NC(c1cnc(C2CC2)s1)=O)C1CC1 55930,N1(C2CCN(C(=O)C=CI)C2)CCN(C(=O)C(C2CCCCC2)O)CC1 55931,c1(C(=O)NNC(=O)N2CCC(O)CC2)ccc(S(=O)(=O)N2CCOCC2)cc1 55932,C=C1CC2CCC(C1)N2C(=O)C(F)C(C)CNC(C1(C(N)=O)CCC1)=O 55933,c1(CC)ccc2[nH]c(C(=O)OCC3(c4ccccc4)CCCO3)c(C)c2c1 55934,C1(CCNC(C2(OC)CCC2)=O)CCN(C(c2cc(C)ns2)=O)CCC1(F)F 55935,C1(O)(C(=O)NCC(C)(O)CNC(=O)Cc2ccns2)CN2CCC1CC2 55936,c1(NC(N2CCCC(n3cccc3)C2)=O)ccc(-c2ncc(C(F)(F)F)s2)cc1 55937,CCC(C)C(C(=O)NC1CC(C)(NC(=O)CCNS(=O)(=O)c2cccs2)C1)OC 55938,C1(C(N2CCC(CC=C)(NC(c3sc(F)cc3C)=O)C2)=O)C2CCCCCC12 55939,C1(NC(C(C)c2cccs2)=O)CC2CCC(C1)N2C(c1c[nH]nc1Br)=O 55940,c1(OCC(=O)N(C(C)C)C(C)C)ccc(C(=O)C(C)C)cc1 55941,c1(C(N2C(C(N(CCCO)CC#C)=O)CC(C)C2)=O)c(C)nn(C)c1C 55942,C=C(C)CN=C(NCC1NC(=O)CC1(C)C)N1CCC(F)(F)C(C)C1 55943,C1(CC(=O)NC(CNC(C=C(C)Cl)=O)C2CC2)CC(=O)c2ccccc2C1 55944,c1(C(=O)NCC23N(C(C4CC(CC)C4)=O)CC(C2)C3)cc2c(s1)CCC2 55945,c1(C(=O)NC23C(NC(CC4ON=C(C)C4)=O)CC(CC2)C3)nccc2n[nH]cc12 55946,C(c1ccc(O)cc1)=CC(=O)NC1(CO)CCN(C(C=CCN(C)CC)=O)C1 55947,C1(NC(C(COC(C)C)NC(c2ccc(C(C)C)o2)=O)=O)COCC1C1CC1 55948,c1(C(N2CCC(CN(C(C(F)=CC)=O)C3CC3)CC2)=O)c(C)nn(COC)c1C 55949,C1(CN(C)C)CN(C(=O)CCN(CCCO)C(c2cn[nH]c2)=O)CCO1 55950,C(=O)(CC(C(C)C)NC(=O)CC1CC2(CCC2)CO1)N1CCC(CCC)C1 55951,Cc1nsc(C(N2CCC3C(NC(c4ccnc(S)c4)=O)C23)=O)c1N 55952,c1(COC)ccnc(C(=O)NCCC2CCC(NC(=O)CP(C)(C)=O)C2)c1 55953,C(=O)(C(O)(C(F)(F)F)C1CC1)NCCC1(C)CC=CC1 55954,C1(C(=O)NCCC(C(C)C)NC(=O)C(C)CO)CCC(F)(F)CC1 55955,C1(CNC(c2c(C)nc(C)[nH]2)=O)CC(C(C)(C)C)CN(C(=O)CC(C)C2CC2)C1 55956,C1(CC=C)(C(=O)NC2CCN(C(=O)Cn3cc(C#N)cn3)C2CC)CCCCC1 55957,CCC(C(=O)NCC1CCCC1NC(=O)C(C)(C)F)NC(C)=O 55958,C1(C(=O)NC2C(NC(C3(C(=O)NC)CCC3)=O)CCOC2)CCC(F)(F)CO1 55959,C(=O)(C1=C(C)CCCC1)N(C1CCCCN(C(CCCC(=O)NCCC)=O)C1)C 55960,CCS(=O)(=O)C=CC(=O)NC1CCN(C(c2ccc3ncnn3c2)=O)C1(C)C 55961,C(C(=O)NCC(C1CC1)NC(=O)CCc1cnn(C)c1C)(C(C)C)OCC 55962,CCCCCC(O)C(=O)NCC1CCN1C(C1C(=C)C1C(=O)OC)=O 55963,N1(C(c2cn(CC=C)nc2)=O)CCC(C)(C)C1CNC(=O)CCN1CCC(F)C1 55964,Cc1nc2cccc(C(c3nnnn3CC(F)F)NC3COCCOC3)c2o1 55965,N12CCC(CC1)C(C(C)C)NC(=O)C2=O.C(C)(Cc1ccco1)(CO)OC 55966,C1(C(Cc2cccs2)OCC)CCCN(C(=O)CCN(c2cc(C)co2)C)C1 55967,c1(CNC(C2CCC(C)(CC)O2)=O)nc2c(s1)CN(C(=O)COC(C)(C)C)CC2 55968,N1(C(C(CCCC)O)=O)CC2CN(C(=O)CCn3c(C)cc(O)cc3=O)CCC12 55969,C1(C(=O)NCCN(C(=O)CC2CC(=O)C2)CCC)CCOC(C)(C)C1 55970,N1(C(C2(COC)COC2)=O)CC(C)CN(C(=O)Cc2c[nH]nc2C)C(C)C1 55971,C1(c2n(C(C(=O)OC)(C)C)nnn2)(N)CSC(C(C)(C)C)C1.c1cnn(C2CC2)c1 55972,C(=O)(N=S(C)(=O)CCO)NC(CC)Cc1ccc(Cl)cc1 55973,c1(-c2c(C(=O)NCC(CC)NC(C3COCCN3C)=O)c[nH]n2)cccc(Cl)c1 55974,c1(CNC(=O)OC(C)(C)C)occc1C(N1CCCC1C1CCCOC1)=O 55975,C(=O)(CC1=CCOCC1)N1CCC(CNC(c2c(Cl)c(C)n(C)n2)=O)C(C)C1 55976,C(=O)(CCCC(CC)NC(=O)CCCCCC)NC(C1CCOC1)C#C 55977,N1(C(=O)Cc2cc[nH]n2)CC2C(CNC(C3CCCOCC3)=O)C2C1 55978,N1(C(CC=CC=C)=O)CCC2CCN(C(c3cc(C(N)=O)co3)=O)C2C1 55979,N1(C(C2(c3ccc(OC)cc3)CCC2)=O)CCN(C(=O)C=CCN(C)C)CC1C 55980,Cc1cc(N)c(C)nc1C(=O)N(CCC(C(C)(C)C)NC(=O)CC(C)C(C)C)C 55981,c1(-c2c(C(=O)NCC(C)(C)O)cc(OCC)nc2)nc2ccc(CC)cc2s1 55982,NS(=O)(=O)c1cncc(C(=O)NC23CC2CN(C(C2CCCCC2)=O)C3)c1 55983,N1(CCC)CC(C(=O)NC(C)CNC(C2CCCN2N=O)=O)CC1=O 55984,N1(C(CCC#C)=O)CCC(C)C1CNC(=O)CCSc1nnnn1C 55985,CON(C)C(=O)OCC.c1(C(N2CCC2)=O)cn(C)nn1.C12(CC1)C(=O)NC2 55986,C(C(O)C(=O)NC1COCC1C(=O)NCC(O)CC1CCC1)N(C)C 55987,C1(NC(c2cncnc2)=O)CN(C(=O)CCN2C(=O)CCC2=O)C2(CCOC2)C1 55988,c1(CC=C)cccc(C(N2CC(CC=C)(NC(C3(CCF)CC3)=O)C2)=O)c1 55989,C1(CC(=O)NC2C3CN(C(C(C)OC)=O)C2CC3)Sc2ccc(Cl)cc2NC1=O 55990,C1(C(=O)NC(CCCNC(C=CC(C)(C)SC)=O)C)OCCOC12CCC2 55991,Cc1coc(C(C)C)c1C(=O)O.C(=O)(CC(C)(C)C)N(CCN(C(C1CC1)=O)C)C 55992,Cc1cc(C(c2nnnn2CC2CCCO2)Nc2cnoc2)c(Br)cc1F 55993,c1(C(N2CC(SC)C(NC(=O)CCC3CC(F)(F)C3)C2)=O)n[nH]c2c1CSCC2 55994,N1(C(=O)OC(C)(C)C)CCC(NS(=O)(=O)NCC2CC2c2ccncc2)CC1 55995,C1(CNC(C(CC)N(C)C)=O)CC2(CCN(C(=O)C(O)CCSC)C2)CO1 55996,C#CC1CCN1C(=O)C(C1CC1)NC(=O)CN(C)C(C)=O 55997,CCC(CCC(=O)Nc1ccccc1CCO)NC(C1CCCCC1O)=O 55998,C1(NC(C2CC2[N+](=O)[O-])=O)CC2C1CCN2NC(c1ccnc(S)c1)=O 55999,N1(C(=O)COCC(F)F)CCC(O)(CCNC(C2(c3ccc(F)cn3)CC2)=O)C1 56000,N1(C(c2c(NC)cncc2)=O)CCN(C(=O)C(O)C(C)C)C2COCC12 56001,N1(C(CC(=O)OCC)=O)CCC2(CC1)CC(NC(=O)CSc1cccc(O)c1)C2 56002,C1(C)(NC(CCOCCC)=O)CCCN(C(c2[nH][nH]c(=N)c2Br)=O)C1 56003,C1(CCN(C)C(C2CC(C(C)C)C2)=O)C(=O)N1.c1(NC(C)=O)nc(CO)cs1 56004,CC(C)C(C)(O)CNC(=O)C(C1CN(C(c2cc(CO)ccn2)=O)C1)OC 56005,CC1CN(C(=O)CCc2ccnc(Cl)c2)CCC1NC(c1c(Cl)n[nH]c1C1CC1)=O 56006,C1(C(=O)OC)CCC(C(N2CCC(CNC(=O)CC=C(C)C)C2)=O)CC1 56007,N1(C(=O)C(Cl)=CCl)CC2CC1CN2C(C1(C(=O)NC2CC2)CC1)=O 56008,N1(C(c2c(CC)nco2)=O)CC(C)OC2(CCN(C(=O)CSCC(C)C)C2)C1 56009,c1(C(=O)NCCOCCN(C(=O)CC2COC3CC2C3)C)ccccc1N(C)C 56010,C1(F)(CNC(Cc2ccn(C)n2)=O)CCN(C(C2CC(N3CCCC3)C2)=O)CC1 56011,C1(CC)CN(C(=O)CSc2n[nH]c(O)n2)CCN1C(=O)C(CC)NC(N)=O 56012,C(N1CCC(F)(F)CC1C)c1n(-c2cccc(OCCC(CC)C(F)F)c2)ncc1 56013,c1(-c2nc(CC3(C)CCCCO3)on2)ccc2nc[nH]c2c1 56014,CCC(O)C(C)C(=O)NC12CC(C(N3CC(c4ncc(C)[nH]4)C3)=O)(C1)C2 56015,C1(O)(CC)CCN(C(=O)C(C)(C)CN(C(=O)CCCN(C)C)C)C1 56016,N1(C(CCC(C)=O)=O)CCC2(CC(C(=O)Nc3cccc([N+](=O)[O-])c3C)=NO2)C1 56017,Cc1ncc2n1CC(C(=O)NC1CN(C(C3CCOC(C)(C)C3)=O)CC1C)CC2 56018,N1(C(CC=CC)=O)CC(NC(c2ccnn2CC(F)(F)F)=O)CC12CCCOC2 56019,C1(CCC(=O)NCC(CC)(C)NC(=O)COC(C)C)CCC(O)CC1 56020,N(C(=NCC(C)(CC)C(C)O)NCC1(C(C)(F)F)CCC1)CC(=O)N(CC)CC 56021,c1(CNC(C(N2CCC(N(CC(CN(C(C)C)C)O)C)C2)=O)=O)cccc(F)c1 56022,S(=O)(=O)(c1ccc(F)cc1Cl)NC(C(c1ccc(Br)cc1)(C)C)=O 56023,N1(C(COCC#C)=O)CCC(C)C(CNC(=O)C=CCCC(C)C)C1 56024,C1(CC(=O)NC(CCCNC(COCCOCCOC)=O)C)CCCC12CC2 56025,C12=C(Cl)N=CNC1=NCC1(CC13CCC3)CN2.c1(C(=O)OC)cncc(N(C)C)c1 56026,C1(CC)C(C(=O)NC2CC(C)(NC(=O)C3=CC(C)C3)C2)CCN1C 56027,Cc1ccn(C(C)CC(=O)NCC2(C)CC(NC(c3cc(F)cs3)=O)C2)n1 56028,N1(C(C(CC=CC)NC(=O)CCC(C)N(C)C)=O)CC(C)N(CC)C(C)C1 56029,C#CCCC(O)C(=O)NC(C)(C)CN1CCN(C(c2cccc(=O)n2C)=O)CC1 56030,C1(C(=O)NCc2oc(C)c(C(=O)NCc3cc[nH]n3)n2)CC2(CCC2O)C1 56031,c1(C(N2C(C(N3CCn4cccc4C3)=O)CC(C)C2)=O)ccc([N+](=O)[O-])cc1I 56032,CCCC(C(=O)NC(C)(C)CNC(c1cc(Br)cc(N)c1C)=O)C(C)C 56033,CC1=C(C(=O)N2CCC(C3(NC(c4sccc4F)=O)CC3)C2)CCCC1 56034,c1(C(=O)NC(C2CCOC2)CNC(C(C)=C2CCC2)=O)cc(F)cc(Cl)c1O 56035,c1(C(C)C)cccc(C(C)(C)ON2CCOC(c3cn[nH]c3)C2)c1 56036,N1(C(C2N(C(C(CC)N(C)CC)=O)CC=C2)=O)CCCCC1CC1(O)CC1 56037,CCCCC(COCCNC(=O)NC12CC3CC1C2C3)CC 56038,c1(C(N2CC(O)CC23CCC3)=O)ccc2ccccc2c1Br 56039,C1(NC(C2CC3CCC2O3)=O)C=CCN(C(=O)CCc2ccco2)C1 56040,CC1(C)CC(NC(C2CC3CC2C3)=O)CN(C(c2coc(OCC(F)(F)F)n2)=O)C1 56041,c1(CCC(=O)NC(CNC(CCOCC(C)C)=O)(C)C)cc(Cl)no1 56042,N1(C(C2(CCCC)CCC2)=O)CCCC(C)(NC(c2ccnnc2)=O)C1 56043,c1(OC(C)C)ccc(-c2nc(NC(c3cc(Cl)c(Cl)s3)=O)cs2)cn1 56044,CC(CC(C)(C)C)C(=O)NCCOCCCNC(=O)CSc1nncn1C 56045,c1(C(N2C(CCCNC(C(C)(C)OC)=O)CCCC2)=O)cnc2n(c1=O)CCS2 56046,c1(C(=O)NC2CN(C(c3c(C)nc(Cl)cc3)=O)C2)ccc2c(c1)CCCCN2 56047,N1(C(C)=O)CC2CC1CCC2NC(c1ccc(OCC2CC2)nc1)=O.OC 56048,Cc1c(Cl)c(C(N2CC(CNC(=O)Cc3ccc(O)cc3)CC2C)=O)nn1C 56049,C(=O)(CCCCC(F)F)NC(C)C(CO)NC(=O)Cc1cnccn1 56050,N1(CCC(=O)NCCNC(C(CC)F)=O)CCCCCC1 56051,c1(OC)ccc2c(c1)C(NC(=O)C(N1c3ccccc3CCC1C)=O)CC2 56052,c1(C(N2CC(F)(C(=O)Nc3cn(CC)nc3)C2)=O)cnc(C)cc1C 56053,C(=O)(CCc1ccsc1)OC(CCC(=O)NCCCOCCCN(C)C)=O 56054,Cc1nc(C)c(C(N2CC(NC(c3ccnn3C(F)F)=O)C(C)(C)C2)=O)nc1C 56055,CC(C)C(CNC(=O)CCCC1OCCO1)NC(=O)CC1(CO)CCCC1 56056,Cn1cc(S(N)(=O)=O)cc1C(O)C(=O)NCCC1CCCCN1C(=O)CC(F)F 56057,c1(OCC(=O)NC2CC(C)N(C(C3CC4CC3C3CC43)=O)C2)ccccc1C#N 56058,CCCCC(O)C(C)C(=O)NC(c1cnn(C)c1)C(=O)NCC1(O)CC1 56059,c1(C(N(C2CN(C(Cc3cnc(C)o3)=O)CC23CC3)C)=O)ccn2cccc2c1 56060,C12(C(=O)NCCN(CCC)C(C3C4CCC(F)C34)=O)CCC(CC1)OC2 56061,Cc1cccc(CC(=O)NC2CC2NC(=O)C(C)C2CCCC2)c1 56062,N1(C(CN(C2CC2)Cc2n(C)cnn2)=O)CCC2(CCOC2)C(C2OC(=O)N2)C1 56063,C(N=C(NCC(F)F)NC1CCN(C2CCCC2)CC1)C1(OC)CCC1 56064,C1(NC(c2cc(C)cc(C)c2)=O)CC2CC(C1)N(CCOCC(C)C)C2 56065,N1(C(C=C(COC)C)=O)CCN(C)C(CNC(C2OCC2(C)C)=O)C1 56066,C1(NC(C(C)(C)C2CCC2)=O)CC2CN(C(=O)C(c3ccccn3)O)CC2C1 56067,C1(NC(c2ccc(O)cc2)=O)CN(C(C2CCC3(CCC3)OC2)=O)CC2(CC2)C1 56068,Cc1c(C(=O)NC2CCCC(NC(=O)C(F)=C3CCCC3)C2)sc2ccccc12 56069,c1(C(=O)NC(CC)CNC(=O)CCOCC2CC2)cc(C2CCC2)[nH]n1 56070,O=C(C#CC1CC1)N1CCCC1C1(O)CN(C(=O)C(c2ccccc2)O)C1 56071,C1(C(=O)NC(Cc2cn(CCOC)nn2)C(=O)OC)CCC2(CC1)CC(O)C2 56072,C1(NC(CNC(=O)OCC)=O)CN(C(C2CCCCC(=O)N2)=O)C2(CCCC2)C1 56073,C(=O)(CCCCC#N)N1C(C(=O)NCC2(C)COCCO2)CC(F)C1 56074,N1(C(C(c2ccccc2)SC)=O)CC(NC(c2cc(C#N)oc2C)=O)CC(O)C1 56075,C1(C#N)(C(=O)NCC(C)CNC(=O)CCS(N)(=O)=O)CC2C=CC1C2 56076,C(CN=c1[nH]c(=NCc2cc(C3CC3)n[nH]2)[nH]c2cccc(F)c12)SC(F)(F)F 56077,c1(C(=O)NC2C3CN(C(c4ccc(CCC)[nH]4)=O)CC32)ncc2c(F)cccn12 56078,C=CCCC1C(=O)NCc2csc(c2)C(c2nnnn2C2CC2)N1.C(C)(C)OC 56079,C1(NC(C2C(C)(C)C2)=O)CCCCCC1C(=O)NCCC1(CO)CC1 56080,C1(CNC(c2c(C)nsc2)=O)CCCC(NC(C2OCC2(C)C)=O)C1 56081,C1(NC(c2ccc(COC)o2)=O)CC2CCC1N(C(=O)C(C)n1cnnn1)C2 56082,C(=O)(CC(C(F)(F)F)n1ccnc1)N1CCC(Sc2cc(C(C)=O)nn2C)CC1 56083,C1(C(=O)NC2(C#C)CCOC2)CCC2(CC2)N1C(C1CN2CCN1CC2)=O 56084,c1(OC)ccc(CCC(N2CC=CC2CNC(C2CCCO2)=O)=O)cn1 56085,N1(C(C2C3(CC(C(N4CCCC4OC)=O)C3)C2)=O)CC(CO)CC(C)(C)C1 56086,Cc1cccc(Br)c1C(C(=O)NC1CCNC(=O)C1)NC(c1ncc[nH]c1=O)=O 56087,C=CC(C)(O)C(=O)NCC1(CN(C)C(c2csc(-c3cocn3)n2)=O)CC1 56088,CN1CCOc2c(C(N3CC(NC(=O)C(O)C(F)(F)F)C3)=O)cccc21 56089,c1(C(=O)NCC(C2CCC2)NC(C2C(CC(C)C)C2)=O)nsnc1O 56090,C1(CNC(C2CCN(C(=O)NC)C2)=O)CN(C(c2conc2C)=O)C(C)(C)C1 56091,C(C(=O)NCCCN(C(=O)Cc1nc[nH]n1)C)(C1CCC1)OCC 56092,Cc1cnnc(O)c1C(=O)NCc1ccc(C(N2CCC(C)C2(C)C)=O)s1 56093,CC(CN=c1nc(N2CCC(c3ccnn3C)C2)c2c(ncn2C)[nH]1)N(C)C 56094,C1(C(=O)NC(CNC(CC2(C(=C)F)CCC2)=O)CC(C)C)CC(C)(C)CN1C 56095,c1(C(N2CC3C(CN(C(C(C=C)O)=O)C)C3C2)=O)cc(C)cc(C)c1 56096,CCCCC(C)(C(=O)OC)NCc1ccc(Cl)cc1C 56097,CC1CC=C(C(=O)NCC2CCC2NC(=O)CSc2nncn2C2CC2)CC1 56098,Cc1ccc2c(CC(=O)NC3CCCC3NC(C3CC3C3CCC3)=O)c[nH]c2c1 56099,c1(CNC(C(C)c2cccs2)=O)ccoc1C(=O)NCc1ccnn1C 56100,N1(C(C(C(=O)OCC)(C)C)=O)Cc2occ(C(=O)N(CCCN(C)CC)C)c2C1 56101,N1(C(C2C(C)CCC2)=O)CCC2(CC(NC(c3cccs3)=O)C2)C1 56102,CC1CN(C(c2cn(CCNC(=O)CC3CCCC(=O)N3)nn2)=O)CC(=O)N1 56103,C(=O)(C(C)(C)CCCCC)NC1CN(C(C2(CC#C)CC2)=O)CC(C)C1 56104,C1(NC(c2cc(CC)no2)=O)CC2CC1N(C(=O)C(C)(C)COCCOC)C2 56105,N1(C(C2(F)CCN(C(c3cc(C)ncc3C)=O)C2)=O)CCCC12CCCOC2 56106,N1(C(CSS(C)(=O)=O)=O)CCOCC1C1CC(F)C1 56107,c1(C(N2CCC(CC3CN(C(c4cocn4)=O)C3)CC2)=O)ccn2ccnc2c1 56108,c1(C(N2CCC3C(C(=O)OC)C3CC2)=O)cc2cccc(C)c2s1 56109,C(=O)(CCCCCC#N)NC(C(=O)NC(C#C)CC(C)(C)C)(C)C1CCC1 56110,Cc1cc2nc(C(=O)N(C3CC3)C(c3cccc(Cl)c3)C)ccc2c(=O)n1C 56111,C=CCCCCC(=O)N1CCN(C)C(C(=O)NC(CC)CO)C1 56112,Cc1cc2c(cc1C)OC(C(N1CCN(C(=O)CC3(CO)CCC3)C(C)C1)=O)C2 56113,C(=O)(C(C)C(=O)NCc1cc(C(=O)N(C)CCn2ccnc2)no1)OC 56114,c1(C(N(C(C)C)CCN(C(=O)CSCc2cccs2)C)=O)ccc2c(c1)COC2 56115,CC12CCC(C(=O)NCC3(C)CCN(C(=O)C(N)=O)C3)(CC1)C2 56116,N1(C(C(C2CN(C(C3C(OC)(OC)CC3)=O)C2)O)=O)C2CCC1CN(C)C2 56117,N1(C(C2(CC)CCN(C(C3CC34CCCC4)=O)C2)=O)CCC(C)(C2CC2)C1 56118,Cc1nc2ncnn2c(N2CC3C(C(=O)NC(C)C(C)F)C3C2)c1C 56119,c1(OC)cc(C(=O)Nc2ccc(C(=O)Nc3csc(C#N)c3)cn2)ccc1Br 56120,c1(CC)[nH]nc(C(N2CCCC2C2CCN(C(c3cn(C)cn3)=O)C2)=O)c1Br 56121,CN1N=CC(CNC(=O)NC2CC(NS(=O)(=O)N(C)C)CC2O)C1=O 56122,S(=O)(=O)(CC(=O)N(CCCNC(=O)Cc1cnn(CCO)c1)CC)NCC 56123,Cc1ccc(C(F)F)cc1C(N1CCC1CNC(c1cccc(C#N)c1)=O)=O 56124,C(C(=O)N=c1nc[nH]n2cccc12)CC1CNC(=O)O1 56125,c1(OC)cccc2c(N3CCCC(CC(C)C)C3)ccnc12 56126,c1(C(N(C)Cc2ncc(-c3ccccn3)[nH]2)=O)ccc(-c2cccs2)cc1 56127,C=C1CCC(C(=O)N(C2CCCCC2NC(=O)Cc2cnnn2C)C)CC1 56128,C(C(O)CC(=O)NC1CN(C(=O)C(C)(C)N2CCCCC2)CC1F)N(C)C 56129,C(=O)(CCS(C)(=O)=O)N1CCC(NC(c2occ(C(N)=O)c2)=O)CC1 56130,C(=O)(CCCC(C)(C)NC(=O)C(C#N)C(C)(C)C)NC1CCCN(C(C)C)C1 56131,Cc1ccc(C)c(C(N2CC(CCNC(C3CC(C(C)C)=NO3)=O)C2)=O)c1 56132,c1(N2CCC(C)C2)ncnc2c1ncn2CC1CCCCC1O 56133,CC1(C)COC1C(N1CCCC1CCNC(=O)CCC1CCCCC1)=O 56134,Cc1scc(C(=O)NCCOCCCNC(=O)CC2CC3CC3C2)c1C 56135,N1(C(CNC(CCC)=O)=O)CCC2CCN(C(=O)Cc3cccc(OC)c3)C2C1 56136,C1(CNC(CC(CC)(C)C)=O)CC2CCC(C1)N2C(C1(COC)C=CCC1)=O 56137,c1(C(=O)NC)ccc(NC(C2(C)CCCN2Cc2cnc(C)[nH]2)=O)cc1 56138,N(C1CCCc2c(Br)cccc21)C(C1N(C(=O)OC(C)(C)C)CC(C)(C)OC1)=O 56139,CC1CCN(C(=O)C(=O)NCCN(C)C(C2(C)CC2C(=O)OC(C)(C)C)=O)CC1 56140,C(=O)(C1=NOC(C)(C)C1)N1CCCC(NC(CCCCOC)=O)(COC)C1 56141,c1(CC)nncn1NC(=O)C(C)N(C(=O)C(C)=C1CCCC1)C 56142,C12(CNC(CCCCCC)CC)CNCC(=O)N1CCOC2 56143,c1(CSC)cc(NC(=O)NC2(c3ccccc3)CCOC2)cc(C)c1C 56144,C1(CC(=O)NC(CCNC(CC=CCC)=O)(C)C)CCCC(C)(C)C1 56145,c1(OC(C(NOC(C)(C)CO)=O)C2CCOC2)cc(C(F)(F)F)cc(C(F)(F)F)c1 56146,C1(CC)(NC(=O)CC2OCCC2C)CCN(C(=O)Cc2cccc(C)c2Cl)CC1 56147,c1(C(N2CCCN(C(CC(C=C)CC)=O)CC2)=O)[nH]c2ccc(F)cc2c1C 56148,N1(C(C(CC(C)C)(C)O)=O)CC2(C=C(C(=O)NCC3CCSC3)CO2)C1 56149,CC(C)(CCC#N)C(=O)N1CCN(C(=O)Cc2sccc2Br)CC1 56150,N1(C(c2c(CC)non2)=O)CC2CCN(C(c3cc(O)cc(O)n3)=O)CCC2C1 56151,C1(NC(C(C)CC2CC2)=O)CC12CCN(C(=O)C(c1cnn(C)c1)=O)C2 56152,C1(NC(c2cc(C)n(C)c2)=O)CCCCN(C(C2(Br)CC2(F)F)=O)C1 56153,C1(NC(c2c(CC)occ2)=O)(CC)CCN(C(C2(C)COC2)=O)CC1 56154,C1(NC(c2cc(CC)on2)=O)(CO)CCCN(C(C2(C)CCCO2)=O)C1 56155,c1(C(CNC(c2ccon2)=O)NC(C2CN(C)C(=O)C2)=O)ccc(F)cc1F 56156,C(=O)(C(F)(F)S(=O)(=O)N1CCCC1CCc1ccc([N+](=O)[O-])cc1)OCC 56157,c1(C(=O)NC(CC)CN(C)C(c2cc(C)cs2)=O)cc(N)c(Cl)c(O)c1 56158,C1(C(=O)N)CCCCC1CNC(=O)C(C(C)C)SC.N1(CCC)CCCC1C 56159,C1(C(=O)NCc2nc(C)sc2C)CC1C1CN(C(=O)C(F)CC2CCOC2)C1 56160,C1(CC(N2CC(C(C)NC(=O)Cc3cnco3)C2)=O)CC(C)(C)OC(C)(C)C1 56161,N1(C(C2C(C)=C2)=O)CCCCC1C(C)NC(=O)CCc1cnn(C)n1 56162,N1(C(C2(CC)COC2)=O)CC(CNC(=O)C#CC2CCCO2)C2(CCC2)C1 56163,C(=O)(C1=CCC2CCC1N2C(=O)CC1(C2CC2)CC1)N(CC(C1CCC1)OC)C 56164,C(=O)(C1CCCc2nn(C)cc21)N1CCN(C(CCc2cnc(C)s2)=O)C(C)C1 56165,c1(NCCC)ccc(C(=O)NCCCN(C(C2CC(CC)CO2)=O)CC)cc1 56166,C1(C(N2CCC(C(C)(C)C)C2)=O)(COC)CCN(C(=O)CN(C)C)C1 56167,O=C(C(O)CC(F)(F)F)NC1CC2CCC(C1)N2C(=O)Cn1cnccc1=O 56168,Cc1nnc2n1CC(C(=O)NC1C=CS(=O)(=O)C1)N(C)C2 56169,O=C(N=S1(=O)CCNC(c2ccccc2)C1)c1cc2c(s1)CCC2 56170,c1(C(N2CC3C(CNC(COCCCC)=O)(C3)C2)=O)nccc(Cl)c1C 56171,C(=O)(CCCC1CCCC1)NCC1(CNC(C(C)OCCC#C)=O)CC1 56172,N1(C(C2CNC2=O)=O)CCC(CO)C12CC2.c1(COCC)ccn(C(C)(C)C)c1 56173,N1(C(c2c(C)coc2C)=O)CCN(C(=O)Cn2nnc(=O)[nH]2)C(C)C1C 56174,C(CC)(C(=O)N1CCC(c2ncco2)C1)N(C(CSCCC)=O)C 56175,c1(OC)cc(C(=O)NCC2COC2)c(NC(c2ccccc2C)=O)cn1 56176,c1(C(=O)NCC(C)CN(C)C(c2nccn2C)=O)cc([N+](=O)[O-])n[nH]1 56177,C1(C(=O)NC(=O)CC2CC2)CCN(C(=O)C2CCC3(CCC3)O2)O1.C12CC(C1)C(=O)N2 56178,C(CC(=O)NC1CC2(C1)CC2(F)F)(C(C)OC)NC(c1cnc(CC)o1)=O 56179,C1(NC(=O)Nc2cc(OCC)c(C)cc2)CC(C(=O)OC)CC(C(=O)OC)C1 56180,c1(CNC(N2C(C)CSCCC2)=O)c(Br)ccc(Cl)c1F 56181,CC(CC(C)(C)C)C(=O)N1CC2CC(C1)N(C(=O)CNc1ncccn1)C2 56182,Cc1ccn2nc(C(=O)NCCN(C)C(C3CC4CC4C3)=O)nc2n1 56183,Cc1c(C(N)=O)cccc1C(=O)NCC1(F)CN(C(=O)C(F)C(C)(C)O)C1 56184,C1(C(=O)NC(C)Cn2cncn2)CCN(C(=O)CC2CCCC(=O)C2)C12CC2 56185,c1(OC)ncc(C=CC(=O)NC2CCCN(C(C3CCCN3C)=O)C2C)cn1 56186,c1(CCC)ccc2c(N)c(C(N3CC(C(=O)OC)C3)=O)sc2n1 56187,c1(C(N2CCC(NC(C)=O)C2)C(=O)NC)cc(C(=O)OC)cc(Br)c1 56188,C(=O)(CC=C(Cl)Cl)NC(CNC(C1(C(=O)OCC)CC1CO)=O)C1CC1 56189,N1(CCN(C(CCC)C)C)CC(C)OC(C)C1 56190,n1(CCC)cc(CNC(=O)CNC(=O)CNC(=O)C(C)CO)nn1 56191,CC1CC(C(N2CCN(C(c3nocc3Cl)=O)C(CO)C2)=O)CC(=O)N1 56192,N1(C(c2ccc(CC)[nH]2)=O)CC(NC(C2CC(OC(F)F)C2)=O)CC1C 56193,N1(C(CC(C)CF)=O)C2CCC1CC(NC(=O)CN1CSCCSC1)C2 56194,CCS(=O)CC(=O)NCC12CN(C1)C2=O.C1(NC(C)C)(CC)CCC(=O)N1 56195,C(=O)(C(C)(C)CN(C(=O)CC1CCC(O)C1)C)NC1(C(C)O)CC1 56196,C1(C(=O)NC2(C)CCN(C(C(N3CCOC3=O)C)=O)C2)CCCC(C)(C)O1 56197,c1(C(N(CC(CN(C(=O)CCc2cnc[nH]2)C)O)C)=O)cnc(C(C)(F)F)s1 56198,CC1CCCc2cc(C(N3C4CCC3CN(C(c3nccnc3N)=O)C4)=O)nn21 56199,CC1CC(N(C(C(=O)NCCC2CC2)c2cnc[nH]2)C)CCN1C 56200,C=C(C)CC(C)C(=O)NC(C)(C)CN(C(=O)C(Cl)=CCl)CC 56201,N(C(=NCCc1ccccc1F)NCCC1(O)CCCOC1)CC(C(C)C)N(C)C 56202,C(c1cncnc1O)=CC(=O)NCCC1CN(C(CCNC(=O)CO)=O)C1 56203,CC1CN(C(=O)CC2SC(=N)NC2=O)CCC1NC(C1CCC2(CC1)N=N2)=O 56204,Cc1cc(N)c(C(N2CCC(O)(CCNC(c3ccc(Br)o3)=O)C2)=O)c(F)c1 56205,C1(NC(=O)COCCCCCN(C(C(F)OC)=O)C)CCCCC1C 56206,C(=O)(CC(C)CC(=O)NC1CN(C(c2cc(C3CC3)no2)=O)C2(CCC2)C1)OC 56207,c1(C(=O)NC2C3(CC(NC(c4c(CC)nc(C)o4)=O)C3)C2)ccc(OC)nc1Cl 56208,Cc1cn(C)nc1C(=O)NC(c1cnn(C)c1)C(=O)NC(c1cnn[nH]1)C 56209,c1(OC)c(C(=O)NC2CCC(NC(=O)Cn3cccc3)C2)cccc1Br 56210,c1(C(=O)NCCCOCCCNC(=O)CC2C=CCC2)cscc1C1CC1 56211,C=CCCCCCCCC(C(=O)NCC=C)N1CC2CCCN2C(=O)C1C 56212,CC(CCC(=O)NC(C)C(=O)NCC(C)(F)F)N(C)C 56213,CC(C)CCCCC(=O)NC1C=CCN(C(=O)Cc2ccns2)C1 56214,NS(=O)(=O)c1cccc(C(=O)NC2C3CC2CN(C(c2ccc(CO)o2)=O)C3)c1 56215,N1(C(CCOC)=O)C(C(=O)NCC2CCC(C)(C)CC2)CCC12CC2 56216,CCC(CNC(=O)CSC1CCCCO1)(CC)NC(=O)CSC(F)(F)F 56217,C1(CN2CC(C)(C(C)C)OCC2)CNCCC12CCOCC2 56218,C1(O)(NC(CCONC(C2C(C)CC2)=O)=O)CCN(C(=O)OC(C)(C)C)C1 56219,N1(C(c2n(C)nc3c2CCC3)=O)CC(N)C2CCCC2C1.C(C)(COCC)(N)CSC.C1CO1 56220,c1(CC)nc(C(=O)NC2CC(CNC(=O)C(c3ccccc3)O)C2)c(C)o1 56221,N1(C(CC#C)=O)CC2COCC2(C(N2CCCC2C(C)(C)O)=O)C1 56222,c1(OC)cc(Br)c(C)nc1NC(=O)Cc1csc(=NCc2nc(Br)cs2)[nH]1 56223,N1(CC(=O)NC)CC(O)CC2(CCNCC2)C1.C12(CC1)C(=O)N2 56224,CCC(CC(C)C)C(=O)NCC1(C(N2CCC(OC(C)C)C2)=O)CCCCC1 56225,C1(CCNC(c2cc(-c3nc(C)sc3)oc2)=O)COC(C)(C)C1 56226,CCCCN=C(NC1CCC1C)N1CCc2nnc(O)cc2C1 56227,N1(C(C2N(C(c3c(C)ncc(Cl)c3)=O)CCSC2)=O)Cc2cccc(O)c2C1 56228,N1(C(CCn2cnc(=N)[nH]2)=O)CCC2CCN(C(=O)CCF)CC12 56229,CC(C)CC(C(=O)N1CCC(O)(CO)CC1)NC(=O)C(c1ccccc1)C 56230,C1(CNC(C(CC)SC)=O)CC2(CCN(C(c3ccc(SC)nc3)=O)CC2)C1 56231,C1(n2cc(C3(C(C)=O)CC3)nn2)CCCN(C(=O)SC2CCS(=O)(=O)C2)C1 56232,C(C(=O)NC1CCCCC1NC(=O)C#CC1CC1)(C(C)C)(C(C)C)NC(C)=O 56233,N1(C(CCC=CC(C)C)=O)CCC(C)(C)CC1C(=O)NCC12CCC(CC1)O2 56234,CCC(C)(CO)CN=c1cc(NCCc2nc(C3CC3)n[nH]2)nc[nH]1 56235,C1(NC(c2c(C)cc(C)cc2C)C2CC2)CCC2C3C=CC(C3)C12 56236,CC(C)CCC(F)C(=O)N1CCC(O)(CCNC(C2CCCCCC2)=O)CC1 56237,c1(OCC)cc(NC(c2nnnn2CCCF)C2(OC)CCSC2)cc(O)c1 56238,c1(N(CC(=O)NCC2(NC(C(C)NC(CC)=O)=O)CCC2)C)ccc(Cl)cc1 56239,c1(OC)ccc(F)cc1C(N1CC2CN(C(c3ccnc(C)n3)=O)C2C1)=O 56240,C1(C(N2CCCC(C(=O)NCC)CC2)=O)C(C2CC2)CCN1C(=O)OC(C)(C)C 56241,C1(C(=O)NCc2cncc(CC)c2)CCOCCN1C(=O)C(C1CC1)SC 56242,N12CCC(CC1)N(C)CC2=O.C1(OCC(=O)NCC2(C)CCOC2)CCCOC1 56243,C(=O)(C(CC(F)F)NC(=O)CCCCC1CC1)N1CC(COC)OCC1 56244,N1(C(C(C=C)(C)C)=O)CCC(C(F)(F)F)C(NC(c2nnc(C)cc2O)=O)C1 56245,CC(C)CCC(O)C(=O)N1CCC(C(C)C(N2CCN(C3CCC3)CC2)=O)CC1 56246,c1(C(N(CCOCCN(C(C2C(C=C)C2)=O)C)C)=O)cc(Cl)c(Cl)cc1O 56247,c1(OC)ccc(C2(NC(=O)N(C3CC3)Cc3ccnc(SC)n3)CC2)cc1OC 56248,c1(-n2c(C)ncc2)ccc(C(N2CCC(NC(C3CC(C)(F)C3)=O)CC2)=O)cc1 56249,N1(C(CCN(C)CC)=O)CCN(C(=O)CS(=O)(=O)CCO)C2COCC12 56250,c1(N2CCC(O)(c3ccco3)CC2)cc(-n2cccn2)n2nccc2n1.c1cccc(Br)c1 56251,C1(NC(=O)NCC2(OC)CC(OC)(OC)C2)OCC2COCCC12 56252,C1(C(N(C)CC2(O)CCC2)=O)CN(C(c2csnn2)=O)C(C)(C)C1 56253,c1(OC)cc(C2(NC)CC2)ccc1C.C1(N)CCC(CNC(=O)CC2CC=CC2)C1 56254,c1(CC)nc(C)c(C(=O)N(CCC(=O)NC(C(C)(C)O)C2CC2)C)o1 56255,N1(C(CCCC#C)=O)CCC(NC(C2CCCN(C(C)=O)C2)=O)C1(C)C 56256,CCC(C)(C)C(C(=O)NC1(CNC(c2cscc2C)=O)CCOCC1)OC 56257,C1(NC(CNC(CC(C)C)=O)=O)CCN(C(=O)COCC(F)F)C(C)C1 56258,c12ccc(F)cc1NC(=O)c1sccc1NC2=O.C1(S(=O)(=O)NC)(CC=C)CC1 56259,C1(C(=O)NC2(c3ccccc3Br)CCC2)CCc2ccncc2C1 56260,N1(C(C2=C(C)OCC2)=O)CC2(CCC(NCc3cc(F)cc(Br)c3)C2)C1 56261,C12(NC(c3csc(-c4ccoc4)n3)=O)CC1CN(C(c1cc[nH]c1C1CC1)=O)C2 56262,N1(C(C2N(C(C(C)CC(N)=O)=O)CC3CC32)=O)CC2(C1)NC(=O)NC2=O 56263,Cc1cc(C)cc(C=CC(N2CCCC2CN(C(=O)CCSCC(N)=O)C)=O)c1 56264,N(C1CCNc2ccc(OC)cc21)C(=O)NCc1ccc(CC)cc1 56265,c1(OC)ccc(OCCN(C(=O)C(C)OC)C)cc1.C123CCCC1(C2)C(=O)N3 56266,C1(C(N2CCN(Cc3cc(C4CCCC4)no3)CC2)=O)CC2(CSC2)C1 56267,c1(C(N(CCNC(C2CC(F)C2)=O)CC)=O)c[nH]c(=N)s1 56268,C1(C(=O)NC2(CC)CC2)C2CC1N(C(c1ccc(CO)s1)=O)C2 56269,C12(NC(c3cc(C)sc3)=O)CCCC1CN(C(c1cc[nH]n1)=O)C2 56270,C1(CNC(CC(C=C)(C)C)=O)CN(C(=O)CCc2nc(C)cs2)CC2(CCC2)O1 56271,C1(CC)(NC(=O)COc2cccc(C)c2C)CCN(C(c2snnc2C)=O)CC1 56272,CCC(CC(=O)N(C)CC1C2CN(C(=O)CC3CC4(CCO3)CC4)CC12)C(C)C 56273,c1(C(=O)NCC23CC(CO2)N(C(=O)CC=C(Cl)Cl)C3)c(F)ccc(Cl)c1F 56274,C1(NC(CC=C)=O)CC(C2CCN(C(c3ncnc(C)c3C)=O)C2)C1 56275,C1(C(C(=O)NCc2ccco2)C2CCCO2)CCC(F)(F)CC1 56276,C(C)(C)(CN=c1[nH]nc(C#N)s1)N(C1CCOCC1)C(=O)Nc1c(C)cc(Cl)cc1 56277,C12(NCC(=O)NCC3CC3)CCCC1(C(=O)O)C2 56278,Cn1cc(C(c2nnnn2C2CC(F)(F)C2)NCC2(C(O)C(C)C)CC2)cn1 56279,c1(OC)ccccc1NC(=O)C(Cc1cc[nH]n1)NC(c1cnns1)=O 56280,CC1CC(N(C(=O)C(C)(C)CN(C(=O)C(c2cncnc2)C)C)C)CC(C)O1 56281,N1(C(C2(c3cccc(OCCCO)c3)CCC2)=O)CC(NC2CC2)CC(O)C1 56282,N1(C(=O)CN2CCN(c3ccc(C(F)(F)F)cc3)CC2)CC2NCCOC2C1 56283,C(=O)(C(C)CC(C)C(C)=O)NC1C(C(=O)NCC2(CC(=O)OC)CC2)CC=CC1 56284,CCCC(CC)C(=O)NCCCNC(=O)C(O)Cc1c(F)cccc1Cl 56285,C(CN=c1[nH]c(=NC(C)c2ccccc2N)c2cc(Cl)ccc2[nH]1)OCCOC 56286,c1(OC)cc(C(=O)OCC2CCC(CC(F)(F)F)CC2)cc(C#N)c1 56287,c1(C(=O)NCC(c2cccc(Cl)c2Cl)F)cc(Cl)c([N+](=O)[O-])[nH]1 56288,n1(CC)c(C(N2CCC2c2nnc(C(=O)O)s2)=O)nc2ccc(Br)cc12 56289,N1(C(c2cc(C)n(C)c2)=O)CC(NC(C2CC3(CCCO3)C2)=O)CCC(O)C1 56290,c1(OCC)ccc(CNC2CC2C(=O)OC)c(OC(=O)Cc2cnn(C)c2C)c1 56291,c1(C(N2C(C(=O)Nc3ncc(O)cc3Cl)CC3CC32)=O)cc(Cl)cc(Cl)c1O 56292,C=CCC(C(=O)NC1CC1NC(=O)CN=c1[nH]c(C)cs1)C(C)(C)C 56293,C(=O)(C(C)(C)S(=O)(=O)C1CC1)N1C(Cn2cc(-c3c(C)nsc3)nn2)CC1 56294,C1(C#CC(=O)NCC(F)CNC(=O)C(c2ccc(O)cc2)(C)C)(CC)CC1 56295,N1(C(c2c(C)nc(O)s2)=O)CCN(C(=O)CCc2cn(C)nn2)CC(C)C1 56296,N1(C(COCC=C)=O)CC(NC(c2cnc(OC(F)(F)F)cn2)=O)CC2(CC2)C1 56297,c1(C(=O)Nc2ccc(F)c(F)c2F)n[nH]c2c1CN(Cc1cnc(C3CC3)s1)CC2 56298,C1(C(NOC(C)C)=O)CCC(NC(=O)COCCF)CC1 56299,Cc1cncc(C(=O)NCCC(C)CCNC(=O)C(F)Cc2ccccc2)c1 56300,CC1=C(Br)CN(C(c2ccc(C)c(Br)c2)C(=O)NC2COC2)CC1 56301,c1(C(=O)NCCN(C(=O)C(C)N2CCC2)CC)cc(C(=O)OC)c[nH]1 56302,c1(OC)cc(Cl)c(CN2CCCC(NC(c3sc(Cl)nc3Cl)=O)C2)c(Cl)c1 56303,c1(CN2CC(C)(CNC(c3c(C)cc(Cl)nc3)=O)C2)ccc(F)c(C#N)c1 56304,c1(SC)cc(C(=O)N(C)CC2(CNC(=O)CC3CC(=O)C3)CC2)c(C)o1 56305,c1(C(N2C3CCN(C(C(=O)OCC)=O)C3CCC2)=O)ccc2cc(O)ccc2c1 56306,C1(NC(CC2N(C(C(C)OC(C)C)=O)CC(O)C2)=O)CCC(C)(C)CC1 56307,Cc1cc(NC(=O)NC2(CCNC3CC4(C3)CC4F)CCC2)c(F)cc1F 56308,C(CC(C(=O)NCC(C)NC=O)NC(=O)CSCC(N)=O)SC 56309,C1(=O)CS(=O)(=O)CC(=O)C(CCC=C)(CC)C(=O)NCC(C)CN1C.OC 56310,CC1CC(C(=O)NCC2(F)CN(C(c3cc(O)cc(O)n3)=O)C2)Cc2nn[nH]c21 56311,C1(C(=O)NCCC(C)C(C)(C)C)(CC)CCCN(C(=O)CC2CCCC23CC3)C1 56312,N1(C(c2cc(C)nc(O)n2)=O)CC2(CCCN(C(c3ccc(CF)cc3)=O)C2)C1 56313,C1(C)(NC(c2ccc(C(C)C)nc2)=O)CCN(C(C2CCC(F)C2)=O)CC1 56314,N1(C(CCCC=C)=O)CCCC(C2CCN(C(c3cncc(C)c3)=O)CC2)CC1 56315,C(C(C)(C)C#CC(=O)NC1CN(C)CC1O)NC(Cn1c(C)ccc1C)=O 56316,Cc1cnc(C(=O)NC2CCC2NC(c2cc(Cl)nnc2O)=O)cc1Cl 56317,C1(NC(CCCCSC)=O)CCN(C(=O)CCOCC(C)(C)C)CCC1CO 56318,c1(C(=O)NC2C(NC(C(=Cc3cccs3)C)=O)CCC2)cc(Cl)ccn1 56319,N1(C(C2(NC(c3ccncc3O)=O)CC(OC)C2)=O)CCC2(C1)CC2(F)F 56320,N1(C(c2c(SCC)cccc2)=O)CCNCC1C(C)(C)C.C(C)(C)(C)O 56321,Cc1cncc(C)c1C(N1CCOC(CCNC(C2CCC(C)(C)OC2)=O)C1)=O 56322,CC1CCC2N(C1)C2=O.c1(CNC(=O)C=C(Cl)Cl)ccc(CO)cn1 56323,C1(N(C(C=C(C)c2cccs2)=O)C)CCN(C(=O)CCn2ccnc2)CC1C 56324,C1(O)(CCNC(C2C(C(C)(C)C)C2)=O)CN(C(C2CC(=C3CCC3)C2)=O)C1 56325,C1(OC)CCC(C(N2CC(N(C)C(c3cnn(C(C)C)c3F)=O)C(O)C2)=O)CC1 56326,c1(OC)cc(C(C(=O)NCCSC)N(C)Cc2cc(C)no2)c(OC)cc1C 56327,CCC(C)(CO)C(=O)N1CC2(CCN2C)C1 56328,CCCCCC(F)C(=O)NC1CCSC12CN(C(c1cnc(O)o1)=O)C2 56329,C1(NC(CCC=CC)=O)C(C)CCN(C(=O)CC)C1C 56330,CC1CN(C(C2(O)CCCCC2)=O)CC1(C)CNC(=O)C(F)(F)CN(C)C 56331,C(CC(C)C(=O)N(C(C)C(=O)NC1CC(C)(C)C1)C1CC1)=CC 56332,CC(O)CC(C)(C)CNC(=O)C=CCC1(NC(C2CC2C2CCCO2)=O)CCC1 56333,c1(C(=O)NC(CC)CN(C)C(c2coc(Cl)c2)=O)ncc2[nH]ncc2n1 56334,Cc1ncccc1NC(=O)C(C)CNC(=O)C(O)C1CCC1 56335,C(C(=O)NC)(C(C(C)C)OC)N1CCN(CC(c2nc(CC)on2)C)CC1 56336,N1(C(C(C)N(C(C)=O)C)=O)CCC(C(=O)NC2CCC(O)C2)C(C)C1 56337,C(CC(C)C(=O)NC(c1cccnc1)C(=O)NCc1cnc[nH]1)=CCC 56338,c1(C(N2C(CNC(C=CCCC)=O)CCCC2)=O)ccc2nc[nH]c2c1F 56339,C(=O)(C(CC)CC(F)(F)F)N1CCC(CNC(c2cc(CC)on2)=O)C12CC2 56340,c1(C(N(C2CCN(C(c3c(CCC)nns3)=O)CC2)CC)=O)cc(C)ccc1F 56341,c1(N2CCC(NC(C3N(CC)C(=O)CC3)=O)C(F)C2)ncc(C#N)cc1Br 56342,C(=O)(C1=C(C#N)CCC1)N1CCC(NC(c2ccc(-c3nc(C)on3)cc2)=O)C1 56343,c1(OC)cccc(NC(=O)C(c2ccon2)N(CCC(C)C)CC(C)C)c1 56344,N1(C(c2cc(C)oc2)=O)CCN(C(c2ncc3[nH]ncc3n2)=O)CC2(CC2)C1 56345,CC1CC(C(N2CC(C)(NC(=O)CC(c3cccc(F)c3)O)C2)=O)CC(C)O1 56346,c1(SCC(N2C(C3CCN(C(COC)=O)C3)CCC2)=O)ccc2c(c1)OCCO2 56347,C1(C)(NC(=O)NCCSCC(=O)NCCC#C)CC2CCC1C2 56348,Cc1ccnc(C(C)NC(=O)CC2CN(C(C3(CCCF)CC3)=O)CC2C)n1 56349,C=CC(C)(C)C(=O)N1CCC(CCCCCNC(=O)Cc2cc(C)n(C)n2)CC1 56350,c1(C(N(C(CNC(C(c2cccc(Br)n2)C)=O)C)C)=O)ccc(N(C)C)cc1 56351,C1(CNC(CCCN(C(=O)OC)C)=O)CCCCN(C(=O)CSC(C)C)C1 56352,C1(F)(C(=O)OCC)CN(C(c2cn[nH]c2-c2cnn(C)c2)=O)CC12CNC2 56353,N1(C(CN(C(=O)COCC(C)(C)C)CCOC)=O)CCC(CO)(CO)C1 56354,c1(C(N2CCC(F)(CF)C2)C(=O)NCCCSC)cccc2c1OC(C)(C)O2 56355,Cc1csc2c(C(N3CCCCC3C3CCCN(C(=O)C4CC4)C3)=O)cccc12 56356,C(=O)(C(C)CC(C)(C)C)NCC(CC)N(C(=O)CSC(F)F)C 56357,c1(CN(C2CCCN(C(c3nc(C)c(C)[nH]3)=O)C2)C(C)=O)nc(C)ccc1F 56358,C(=O)(C(F)CC(C)C)NC(CC=C)CNC(=O)COc1cccc(C(F)(F)F)c1 56359,C1(C)(N(C(=O)CC2CC(C)(C)CO2)CC)CCN(C(=O)CNC(=O)NC2CC2)C1 56360,c1(C(=O)NCc2cc(C(=O)NC(C(=O)OC(C)C)C)ncc2)ccc(=O)n(C)n1 56361,N1(C(C(C)OCC)=O)CC2(CCCC(CNC(c3nn(C)cc3[N+](=O)[O-])=O)O2)C1 56362,C(N=c1[nH]c(=NCC(=O)N=c2cc[nH]cc2)[nH]c2c1COCC2)C1(C)CC1Br 56363,Cc1cc(C=CC(=O)NCC2(O)CCCN(C(c3ccccn3)=O)C2)ccc1F 56364,N(C(=NCc1ncn(C)n1)NC(C1CCOCC1)COC)CC(COC)(C)C 56365,C=C(CNC(=O)Cc1ccsc1)CCNC(C1CCN1C(C)=O)=O 56366,C=C(C)C(C)(C)C(=O)NC1CCC(C)(CNC(=O)CNC(C)=O)CC1 56367,C(c1ccccc1F)=CC(=O)NCC1(NC(=O)Cc2cc[nH]c2)CCOCC1 56368,c1(OC)cc(CNC(C2CCCC2NC(=O)CCC2CC2)=O)cc2c1OCO2 56369,c1(C(=O)NC2C(CNC(CC(=O)OC)=O)CCC2)cc2cc(Cl)c(Cl)cc2[nH]1 56370,C1(NC(CC2(OC)CCCC2)=O)CCN(C(=O)CC(C)N(C)C)CC(O)C1 56371,c1(C(=O)NCCC(C)CCNC(=O)CC2CC(F)(F)C2)cc(F)c(F)cc1O 56372,c1(OC)cc(O)ccc1CN1CC(CC(=O)Nc2cc(I)ncn2)C1 56373,c1(C(=O)NC2CCC(C)(NC(c3n(C)ccn3)=O)CC2)cc2sccc2cn1 56374,c1(N(C(c2ccco2)=O)CC)ccccc1C 56375,C(=O)(CCCCCC#N)N1C(CNC(=O)C=Cc2ccccc2)CC(COC)C1 56376,Cc1cnsc1C(=O)N(C1CCC(NC(c2csc(C(C)N(C)C)n2)=O)C1)C 56377,N1(C(C(CCC)NC(COC2(C#C)COC2)=O)=O)CC(S(C)(=O)=O)C1 56378,c1(C(N2CC=CC(NC(C(C=C=C)C)=O)C2)=O)cc([N+](=O)[O-])n[nH]1 56379,N1(C2CCN(C(CC3(OC)CC3)=O)C2)CCN(C(C2CC3CC3C2)=O)CC1 56380,N1(C(c2cncc(C3CC3)c2)C(=O)NC(C(=O)OC)C)CCC(O)C2CCCCC12 56381,C1(CC)CN(C(=O)COCC2CC2)CCC1NC(C1CC(O)(C#N)C1)=O 56382,CCCC(C(=O)N(CCNC(=O)C(c1ccccc1)F)CCOCC)NC(N)=O 56383,c1(C(N2CCC(C(F)C(N3CC(F)C(F)C3)=O)C2)=O)cnnc(O)c1 56384,C1(NC(CN(C)Cc2nnc(C)n2C)=O)CC2CCC1(NC(=O)C(C)(C)O)C2 56385,N1(C(CC2C(C)(C)CCCO2)=O)CC2CC(C1)CN(C(C1C(F)(F)C13CC3)=O)C2 56386,Cc1ccccc1N=c1scc(-c2ccc(Br)o2)n1C1CC1(C)C1CC1 56387,c1(N2CC(CN(C)C(c3cc(SC)oc3C)=O)C2)nc(C)c(C)c(C)c1C#N 56388,Cc1nc2sccn2c1C(=O)NCC(C)CN(C(=O)CC1CCC(F)(F)CC1)C 56389,CC1(C(=O)NCC(c2ccc(O)c(O)c2)O)CCCN(CCN2CCCCC2)C1 56390,c1(C(=O)NC(CNC(C(COCC)(C)C)=O)(CC)CC)ccc(P(C)(C)=O)nc1 56391,c1(-c2cc(Cl)c(Br)cc2)nc(C2SCCc3ccccc32)no1 56392,c1(C(N(C2CCCN(C(=O)C=CC3CC3)C2)CCC)=O)cnc(CC)nc1O 56393,CCN=c1ccc(C(=O)NC(CO)C(C)NC(c2ccc3c(c2)COC3)=O)c[nH]1 56394,c1(CC)nccnc1C(=O)NC1CC(CNC(=O)COC2CC=CC2)C1(C)C 56395,C1(CC=C)(C(=O)N(C(C)C(C)SC)C)CCN(C(=O)C(CC2CCC2)OC)C1 56396,N1(C(c2c(SCC)nccn2)=O)CCN(C(=O)C2=CCCC2)C(C(C)C)C1 56397,C1(CC#C)CCCCN1C(=O)C(CCNC(=O)C(F)CC1CCOC1)OC 56398,C1(NC(c2cc(CC)nn2C)=O)CC(O)CN(C(=O)CCC2CCCO2)C1 56399,c1(C(=O)NC(CNC(CCNC(C)=O)=O)C(C)C)cc(C)c(C)c(S(N)(=O)=O)c1 56400,c1(OCC(=O)NC(CN(C(c2cnc(C(=O)OC)s2)=O)C)C)ccc(F)cn1 56401,CCC(C)C(O)C(C)C(=O)NCC(COC)NC(=O)C(O)CNC1CC1 56402,CC1C(NC(=O)C=Cc2nccs2)CCCN1C(=O)CC(C)c1ccccc1 56403,Cn1ncc(C(N2CCCC2CNC(c2cnn(C3CCC3)c2)=O)=O)n1 56404,c1(OC)c(Cl)ccc(C(=O)NC2(C)CN(C(c3cc(N(C)C)ccn3)=O)C2)c1N 56405,C1(C(N2C(c3c(C)ccs3)CCC2)=O)CC(F)(F)CCO1 56406,N1(C(C(C(=O)OCC)F)=O)CCC(NC(c2ccc(CO)cc2F)=O)C12CC2 56407,C(CCN=c1[nH]c(=NC(C)c2ncc3ccccn23)[nH]c2c1CSC2)OC 56408,C(C(C)(C)NC(C1CC(n2ccnc2)C1)=O)N(C(COCCOCC#C)=O)C 56409,N1(C(CNC(C)=O)=O)CC(O)CC1CNC(=O)C(C(C)C)c1ccc(F)cc1 56410,c1(OC)ccc(CC(O)C(=O)NC(C)CC(C)NC(=O)CN(C)C(C)=O)cc1 56411,C1(NC(c2c(C)scn2)=O)CCC(O)CN(C(=O)CN(C)C(=O)C2CC2)C1 56412,N1(C(C2(NC(c3cc(COC)on3)=O)CC(O)C2)=O)CCC(C)(O)C1 56413,N1(C(c2csc(C)c2C)=O)C(C)CC2CN(C(=O)CCC3(C)CC3(F)F)CC12 56414,Cc1ccc2oc(C(=O)NC3(C)CC(NC(=O)COC4CCCCC4)C3)cc2n1 56415,CCC(CC)(CC)C(=O)N1CC(CNC(c2nn(C)cc2N)=O)C1 56416,N1(C(C=CCN(C(C(C)(C)NC(C)=O)=O)C)=O)CCN(C)C2CC12 56417,C(=O)(CCCN=[N+]=[N-])N(CC(O)CNC(c1cc(-c2ccccn2)[nH]n1)=O)C 56418,C(N=c1[nH]c2cc(Cl)c(S(=O)(=O)NCC(Cl)(Cl)Cl)cc2s1)C1C(C)OCC1 56419,C1(NC(c2c(CC)ncs2)=O)COC2(C1)CN(C(C1(C)CCC(C)CC1)=O)C2 56420,C1(F)(CNC(C2CCC(=C)CC2)=O)CCCN(C(C2(F)CC=CCC2)=O)CC1 56421,N1(C(c2cccc(C)c2Br)=O)CC(NC(C2CC(O)C2)=O)CC12CCCC2 56422,c1(NC(N2CCCC2Cc2ccc(CC3(O)COC3)o2)=O)ccc(F)cc1 56423,C1(CN(C(C(CC)F)=O)C)CCCCN1C(=O)CCCSC 56424,C1(CNC(C2CC3CCC2O3)=O)CN(C(=O)CSc2ccccc2O)CC1(F)F 56425,CC1(C(N)=O)CCCN1C(=O)C(F)CC1CN(C(C2CC23CC3)=O)C1 56426,N1(C(C2C(C)=C2)=O)CCCCC(CNC(C2CNC(=O)CC2C)=O)C1 56427,c1(C(C)C(=O)NCC(C)N(C(=O)CCOCCOC)C)ccc(F)cc1.C=O 56428,N1(C(=O)OC(C)(C)C)CCC2CCN(CC(c3ccccc3)O)C2C1 56429,CCS(=O)(=O)c1ccc(C(=O)Nc2cnc(C3CCC3)s2)cc1 56430,c1(CC(N2CC(CC(C)NC(c3occc3F)=O)C2)=O)ccc(Br)cc1F 56431,C1(C(N)=O)(N)CCCCC1.c12c[nH]cc1NC(=O)CCN(C1CC1)C2=O.CC 56432,c1(C(=O)NC2C(NC(c3cn[nH]c3)=O)CC2)cc2ccc(Cl)cc2c(=O)o1 56433,Cc1c(C(N2CCC(O)(C(C)NC(=O)C(C)(C)CO)C2)=O)cc(Br)cc1N 56434,C(=O)(CC(C)(C)Cc1ccc(Cl)cc1)NC1N(C(C(C)NC(CC)(C)C)=O)CC1 56435,n1(C(C(=O)OC)C)nnnc1C(C1CCOCC1)(CC)NCc1ccc(O)o1 56436,c1(C(N2CCCC(CCC(=O)NCCCNC(=O)OC)C2)=O)ccc(C)c(O)n1 56437,C12(C(=O)OC)CC1CN(C(=O)C(CNC(=O)C(C(C)C)N(C)C)OC)C2 56438,CCCC(C(=O)NC(C(=O)NC)C1CCCC1)NC(c1cnn(C)n1)=O 56439,c1(N2CC(NC(CC(C(F)(F)F)OC)=O)C(C)CC2)nc(Cl)nc2c1ncn2C 56440,C#CC1CN(C(=O)CC2CCCCC2C)CCN1C(c1cccn1CC)=O 56441,c1(-c2cn(C(CNC(C=C(CC)CC)=O)C)nn2)c(F)cccc1F 56442,C1(NC(CCc2ccnc(C)n2)=O)CC2(NC(C3CC3C(N)=O)=O)COC1C2 56443,Cc1cc(=NCCCC(C)(C)NC(c2ncc(F)cn2)=O)[nH]c(C(C)(C)C)n1 56444,C1(N(C(=O)CC(CC(N)=O)C2CC2)C)CCN(C(=O)C(C#N)C2CC2)CC1 56445,C1(C(N2CC(O)(CC(C)C)C2)=O)CC2C=CC1N(C(=O)CCc1ccc[nH]1)C2 56446,C(=O)(C(F)C1=CCCCC1)N1C(CNC(COCCN(C)C)=O)CCC1 56447,c1(C(=O)NC2C(NC(C(Br)=C(C)C)=O)CC2)cc2ncccc2o1 56448,N1(C(c2ccnc(C)n2)=O)CC2CCCCN2CC1CNC(c1cnc(O)s1)=O 56449,N1(C(C(C=C)O)=O)CC2CCC1C1CN(C(c3c(F)cc(F)c(F)c3F)=O)CC21 56450,C1(OC)COCCC1(c1nnnn1CCSC)Nc1ccc2c(c1)COC2 56451,c1(C(=O)NC(C)CCCNC(=O)CC2CCCS2(=O)=O)ncccc1C#N 56452,O=C(C(F)C1=CCCCC1)NCC1CCN(C(C2CCOC2=O)=O)C12CC2 56453,C(=O)(C(C)C(C)CC)N1CC(CCCCNc2ccc(OCC#C)cc2)C1 56454,c1(C(=O)OC)ccc(CN(C)C(C2CCCN(C(=O)OC(C)(C)C)C2)=O)cc1Cl 56455,N1(C(c2ccc(OCC)cc2)=O)CCN(C(C2(C)CC2C)=O)CC1c1cn[nH]c1 56456,CCC(c1ccc(C)cc1)=CC(=O)NC(C)CNC(c1n[nH]cc1OC)=O 56457,c1(C(N(C)CCOCCN(C)C(C2(C)CC2F)=O)=O)ccc2c(c1)OCC2 56458,N1(C(C2(OC)CCOCC2)=O)CC2(CCN(C(c3ccc4c(c3)NCC4)=O)C2)C1 56459,C(=O)(CCC(=O)NC(C)(C)CC(=O)NC1CCN(C(C)C)CC1)NCC 56460,CC1(CNC(=O)NC2(c3cccc(F)c3)CCCC2)CCCCCC1 56461,C1(SC)CN(C(c2c(C)nsc2C)=O)CC1NC(=O)CC(C)(C)C1CC1 56462,c1(COC)ccccc1-n1nc(CO)nc1-c1cccc(C2CCC23CCC3)c1 56463,c1(C(c2nnnn2CC2CCCO2)NCCCS(C)=O)snc(OC)c1Br 56464,N1(C(CC(CC)(C)C)=O)CCC2(CCCN2C(c2sccc2C)=O)C1 56465,C1(C(N(C2CCCCN(C(c3coc(C(F)F)n3)=O)C2)C)=O)CC12CC(F)(F)C2 56466,CCCCC(C(=O)NCC1(F)CCN(C(=O)C(O)(C2CC2)C2CC2)C1)C(C)C 56467,N1(C(C=CCC)=O)CCC(C2CCCN(C(c3n[nH]c(CC)c3Cl)=O)C2)C1 56468,C12(NC(=O)CC3CC3)CC1CN(C(C1CCCOC1c1cc[nH]n1)=O)C2 56469,C1(CNC(CCSCCC)=O)COCCN(C(C2(Cl)CC2(F)F)=O)C1 56470,c1(C(N2CCSCC2(C)c2ccccc2)C(=O)NC(C)C)cc(Cl)c(Cl)c(Cl)c1 56471,C1(C(=O)NC(CC)(C)CC)N(C(c2c[nH]c(=NC)o2)=O)CCCC1(C)C 56472,N1(C(C(C)OC)=O)CC2(CNC(C34CCCC(CO3)C4)=O)CC1CCO2 56473,Cc1nc(Cc2ccccc2)oc1C(=O)NCC1CCN1C(C1CC1F)=O 56474,C1(NC(CC(CC)O)=O)CC2CCC(C1)N2C(=O)C(c1ccc(F)cc1F)C 56475,C(c1cccc(Br)c1)=CC(=O)N(CCC#C)C(C)(C)C 56476,C(=O)(C(F)C(F)(F)C(F)(F)F)NCCC(C(C)C)NC(Cc1c(C)cccc1)=O 56477,C(CNC(C1CC(C)=NO1)=O)(CC(=O)NCc1nnc(O)o1)OC 56478,C1(NC(CCNC(=O)NC)=O)CCN(C(c2c(C)ccoc2=O)=O)CCC1(F)F 56479,c1(C(N2CC(NC(C3(COC)CCCC3)=O)C2)=O)nn(-c2ccn(C)n2)nc1C 56480,c1(OC)cc(C(=O)NCC(COC)NC(C2(C)CCCCC2C)=O)cnc1C 56481,N1(C(C2C(C)(CC)CCC2)=O)CC2(C(=O)Nc3cn(C)nc3C#N)CCC1CC2 56482,c1(CN(c2ccc(OC)cc2)C)ccc(C)nc1O 56483,N1(C(=O)CCc2nc(O)n[nH]2)CC2CC(N=c3[nH]nc(C(F)(F)F)s3)CC1C2 56484,N1(C(c2cn(C)c(=O)cn2)=O)CC2CCN(C(=O)CC=C(Cl)Cl)CCC2C1 56485,c1(CC(=O)NCc2c(C3CN(C(c4cc(C)sn4)=O)C3)ocn2)ncccc1C 56486,c1(CN2CC=C(CNC(C3OCC(C)C3)=O)CC2)cccc2cc[nH]c12 56487,C1(NC(CC2C(CNC(c3cc(COC)no3)=O)C2)=O)CCN(C)CC1C 56488,c1(C(N2CC(NC(C3CC4CSCC(C3)C4)=O)C2)=O)ncc2[nH]ncc2n1 56489,N1(C(C(C)C)=O)CCC(NC(C2(C)CC2(F)F)=O)C(C)C1 56490,C1(OC)CN(C(C2CC3(CCC3)C2)=O)C(C)(CNC(c2ccc(F)cc2Cl)=O)C1 56491,N1(C(c2c(C)cns2)=O)CC(NC(=O)Cn2cc(C#N)cn2)C(CC2CC2)C1 56492,CC1CCC(Cl)=C(C(=O)Nc2nc(-c3cccs3)cs2)C1 56493,C(=O)(C1CCCc2scnc21)NC1C(C)CCN(C(C2C(C(=C)C)OCC2)=O)C1 56494,N1(C(C(C(C)C)OC)=O)CCC(CNC(=O)C(C)(C)O)C(F)(F)CC1 56495,c1(CN2CCN(CC#C)CC2)ccc(F)c(C)c1.c12cn(C)nc1n(C)c(=O)[nH]2 56496,N1(C(C=CC(=O)N(C)C)=O)CCC2(CC2)CC1C(=O)NCC1(C#N)CCC1 56497,CC(C)C(O)CC(=O)N1CC(F)CC1CC(=O)Nc1ccc(Cl)nc1 56498,Cc1ccc(C(=O)NCC(=C2CN(C(c3ncccc3Cl)=O)C2)F)cn1 56499,C1(CC(N2C(CC(C)=O)CCC2)=O)(N(C(=O)Cn2nccn2)CC)CCCCC1.O 56500,c1(NC2CC(C)N(C(c3cccc(OCCF)c3)=O)C2)ccccc1[N+](=O)[O-] 56501,C(c1cnc[nH]1)=CC(=O)NC(C1CCOC1)CNC(c1ncoc1C(F)(F)F)=O 56502,c1(C(N(C)CC2CCN(C(CCCCCC)=O)C2)=O)ccc2cccnc2c1 56503,c1(OC)ccc(C(=O)NCC(=O)NCC(C)CNC(C2(C)CC(C)(C)C2)=O)cc1 56504,CN1CCN(C(c2ccccn2)=O)CC1CNC(c1ncccc1F)=O 56505,CC(C)(F)CCC(=O)NCC1CCC(NC(=O)CC2COC(C)(C)CO2)CC1 56506,O=C1NCc2cc(C(=O)NC3CCCCC3Nc3ncncc3F)ccc21 56507,C1(NC(C2OCCN(C(C)C)C2)=O)(CO)CCN(C(C2(C(N)=O)CC2)=O)CC1 56508,C1(NC(c2ccccc2C2CC2)=O)CN(C(=O)CC2CCNC2=O)CC(F)(F)C1 56509,C1(NC)CCC(C(=O)N(CCC(N2CCC(C(C)C#N)CC2)=O)C)CC1 56510,N1(C(COCCCOC)=O)CC2CCC(C1)C(NC(c1conc1C)=O)C2 56511,N1(C(CCc2nc(C)c(C)[nH]2)=O)CCCC2CN(C(c3cnccn3)=O)CCC12 56512,C1(C2CCN(C(c3cccc(-n4cccc4)c3)=O)C2)(NC(CCC=C=C)=O)CC1 56513,CC1(C)CN(C(C2CCCCC2O)=O)CCC1NC(C1CC12CCSCC2)=O 56514,N1(C(C2(c3nn[nH]n3)CCC(O)CC2)=O)CC=C(c2cccc(Cl)c2F)CC1 56515,N1(c2nccc(OCC)n2)CCC(C)C(NC(C2CC(C)=NO2)=O)C1C 56516,Cc1ccc(C2=CCC(C)(C)CC2)c2nc(C(=O)NCc3ccnn3C)cn12 56517,c1(C(=O)NCCN(C(CSCCN(CC)CC)=O)C)ccc(O)c(F)c1 56518,C=CC1(C(N2CCOC(C#N)C2)=O)CCN(C(c2cc(CC)no2)=O)CC1 56519,C(=O)(C1=C(C)S(=O)(=O)CC1)NC(CCNC(c1c(CC)ncc(Br)c1)=O)C 56520,C(=O)(C(C)(Cc1ccncc1)N1CCNC(=O)C1)OC 56521,N1(C(=O)COC2CCCOC2)CCCC2C1CCN2C(=O)CN1CCS(=O)CC1 56522,C(CCCCC(=O)N1CCCC(C(=O)N(CC(C)O)CC2CC2)C1)SC 56523,c1(CC)ccc(C)cc1C(=O)NC1CN(C(c2cc(Cl)n(C)n2)=O)CC1C 56524,N1(C(Cc2c(C)noc2)=O)CCC2CN(C(c3cccc(=O)n3C)=O)CCC2C1 56525,C#Cc1cc(C(=O)NCC(C2CCCCC2)NC(=O)C=CC2CCCC2)ccc1C 56526,C(CCCOC)(C(=O)NCCCN(CC(C)C)C)NC(c1c(CC)cno1)=O 56527,c1(NC(=O)CNC(=O)NCCC2CCCN2Cc2cccnc2)ccc(F)cc1 56528,c1(C(N2CCC(C(CO)NC(C(C)O)=O)CC2)=O)cc2occc2s1 56529,c1(SCC(=O)NCC2C(CNC(C(N)=O)=O)C2)ccc(F)c(F)c1 56530,c1(CC)nnsc1C(=O)NCC(C)(F)CNC(=O)CC1CCCOC1 56531,C(=O)(C(C)(O)CC(F)F)NCC(CN(C(CCn1c(C)nc(C)n1)=O)C)(C)C 56532,c1(C(C(N2CCC(NC(C(C#N)C3CC3)=O)(CO)C2)=O)=O)ccc(F)cc1F 56533,O(N(CC)C(=O)CNC(=NCCSCC)NC1CCCOC1)CC 56534,CC(C)(CC(=O)NCC(CO)NC(=O)CCn1cc(Br)ccc1=O)C(F)F 56535,c1(CC(C)C)ccc(C=CC(=O)NCC2CC(CNC(=O)CO)CO2)cc1 56536,N1(CC(C)CNC(=O)C(Cc2cccs2)NC(N)=O)CCCCC1 56537,C(=O)(C(O)CC(F)(F)F)N1CC(CC(C)NC(=O)C(C)(C)C(F)(F)F)C1 56538,C1(NC(=O)Cc2ccnc(Cl)c2F)C2CCC1CN(C(C1CCCC1(F)F)=O)C2 56539,c1(NC(C2CC(CNC(C3C(C)=CCS3)=O)OC2)=O)cnc(C)c(C)c1C 56540,C=CCCCCC(=O)NCc1csc(CC)n1 56541,C1(C(N2CC3CC(NC(=O)C(C)c4ccco4)C2C3)=O)(CC)CCC(F)(F)CC1 56542,C(=O)(N=c1[nH][nH]c(-c2ccccc2)c1C#N)N(CC(C(C)C)C)C 56543,N1(C(Cc2c(C)cco2)=O)CCc2sccc2C1CNC(=O)C(Cl)=CCl 56544,N1(Cc2cc(OC)ns2)CC2(C)CN(C(C3CCC4(CC3)CC4)=O)CC2(C)C1 56545,CC1CC(C(=O)NCC2CC(C(=O)NC3(C)CC=CC3)C2)CCS1 56546,C1(N=[N+]=[N-])(C(=O)NC(CC)C(F)(F)F)CCN(C(C2CNC(=O)C2)=O)C1 56547,C1(CC(=O)N(CCC(=O)OC)CC#C)(NC(=O)C=CCOC)CCCCC1 56548,C1(NC(CCc2ncc(C)[nH]2)=O)(CO)CCN(C(c2occc2Br)=O)CC1 56549,S(=O)(=O)(c1cccc(C(F)(F)F)c1)N1CC2N(C(CCCN(C)C)=O)C2C1 56550,c1(C(=O)O)ccc2c(c1)CCC2NC(c1nc(F)ccc1Cl)=O 56551,C1(COC)(NC(=O)C(C)CC(N)=O)CCCN(C(=O)Cc2cccnc2O)C1 56552,c1(CC)ccc(C(c2nnnn2C2COC2)Nc2ccc(C)nc2)c(C)c1 56553,N1(C(COCCC=C)=O)CCC(Nc2nccc(CC#N)n2)C(C)C1 56554,Cc1nc(N(CC(C)CNC(c2cn(C3CC3)cn2)=O)C)c(C)c(C)n1 56555,C(=O)(NN1CCCC1C(=O)NCCCN(C)C)c1c(C)ncs1 56556,CC(C)CC(C(=O)NCC1(C)CSC1)ONC(c1ccc(N)cn1)=O 56557,C(=O)(C(O)CC(C)C)N1C(CCNC(c2c(OC)noc2C)=O)CSCC1 56558,c1(C(=O)NC2C(NC(C3(OC)CC3)=O)CCOC2)cnc(O)c(Br)c1 56559,N1(C(C(CCOC)(C)C)=O)CC2(CCC(NC(=O)CCNC(=O)N(C)C)CC2)C1 56560,c1(C(=O)OC)ccc(C2(C)CC2)cc1.N12CCC(C1)NC(=O)C2C1CC(OC)C1 56561,c1(NC)c(C(N2CCCC(CCF)C2)=O)sc2nccnc12 56562,C1(NC(c2nc(C(C)=O)sc2)=O)CCN(C(c2cnsc2)=O)CC1C 56563,C1(C2(O)CCOCC2)(C(=O)NC2CC3CC(NC(C(CC=C)C)=O)C2C3)CC1 56564,C=CCC(CC(=O)NCCOCCCC(=O)NC)NC(=O)CC1(OC)CC1 56565,N1(C(CCC(=O)NCC)=O)CCC2C(CCN2C(=O)CCCNC(C)=O)C1 56566,C1(C(=O)NCC(O)C(=O)NC2CC(CO)C2)CCC(O)CC1 56567,CN1CCN(C(=O)C2=CCCCO2)C(CNC(=O)C=Cc2ccc(=N)[nH]c2)C1 56568,C(=O)(CCCCCC#N)N1CCC(C(=O)NC(CCCC)C2CC2)C1 56569,C(=O)(C(CC(N)=O)NC(c1cn(C(C)C)nn1)=O)NCC(CC(C)C)O 56570,C1(C(=O)NC(CCC=C)C2CC2)(OC)CCN(C(=O)C=CC(=O)OCC)C1 56571,C(=O)(C1=CCCN(C(C2CCN(C(c3ccc[n+]([O-])c3)=O)CC2)=O)C1)OC 56572,c1(CONC(c2ccc(CNC(CC(C)(C)O)=O)o2)=O)ccc2c(c1)CC2 56573,c1(C(=O)NC2CC(O)(CNC(C3C(C)(C)C3C(F)F)=O)C2)cnc2[nH]nnc2c1 56574,CC1(CC(N2CCC(OCC3CC3)C2)=O)CN(C(=O)CCN2CCC2)C1 56575,c1(C(N2CCN(C(C(CC)C)=O)C(c3ccccn3)C2)=O)ccn2cncc2c1 56576,c1(C(=O)NCC(N(C(=O)CCn2cncn2)C)C2CC2)cccc(CF)c1 56577,N1(CC(C)C)CCN(C(C23CC(CN2C(=O)C(F)(F)CO)C3)=O)CC1 56578,c1(Nc2[nH]nc(SC)c2C#N)ccc2ncc(-c3cc[nH]n3)n2c1 56579,C1(NC(C(C)Cc2cccnc2)=O)COCCN(C(c2cc(F)ccc2N)=O)C1 56580,c1(C(=O)NC(CN(C)C(C2(Cl)CC2(C)C)=O)(CO)CO)ccc2ccoc2c1 56581,C(=O)(C1=CCC(F)(F)CC1)NCC1N(C(c2cnc(OCC)c(Cl)c2)=O)CCC1 56582,c1(C(N2C(Cn3cc(-c4n(CC)ncc4)nn3)CC2)=O)ncccc1OC(F)F 56583,C(=O)(C(O)C(C)C)NC(C(N1CC(O)(CC=C)C1)=O)CO 56584,c1(CCCCNC(=O)NC2(c3ccccc3)COC2)cccc(F)c1F 56585,c1(C(C)NC(=O)NC2CC(COC)C2)ccc(N2CCOCC2)c(F)c1 56586,N1(C(C2C(C)CC(=O)NC2)=O)CCC(C)C(NC(=O)CS(N)(=O)=O)C1C 56587,CN1CCC(CCC(c2cc(C(c3ccccc3)=O)n(C)n2)=O)CC1=O 56588,c1(C(N2CCCC2c2ccc(Cl)c(F)c2)C(=O)NCC)ccc(C(F)F)c(F)c1 56589,c1(C(N2C3C(NC(c4c(CC)onc4)=O)CC(C3)C2)=O)c(C)ccc2n[nH]cc12 56590,C1(C(C)(C)C)CC(=O)N1.C(=O)(N=c1ccn(C)[nH]1)C1C(C)C2CCC1C2 56591,N1(CCCC=C)CC2CCC1C1CN(C(=O)C(c3ccccc3F)OC)CC21 56592,C1(C(=O)NCC23CC(CNC(=O)CCn4cccc4)(OC2)C3)CC2OC1C1CC21 56593,N1(C(c2cc(C)c(F)cc2Cl)=O)CC(C)CN(C(=O)Cc2ccco2)C(C)C1 56594,N1(Cc2cc(OC)c(Cl)cc2)CCC(F)(F)C(C(=O)Nc2ncc(Cl)cc2Br)C1 56595,c1(OCC)nc(OCC2CCCC2)cc(N2CC(OC(C)(C)C)C(CO)C2)n1 56596,c1(C(=O)NC2C3CCN(C(CCSCCC)=O)C32)cc2ccc(OCC)cc2[nH]1 56597,C1(C(=O)NC2CCC(NC(=O)Cc3ccsn3)CC2)CN2CCN1CC2 56598,c1(CC(=O)N(C(C)CN(C(=O)C(O)c2ccco2)C)C)ccccc1C1CC1 56599,CC1CN2CC1CCNC(=O)CC2=O.C1(C)(CC(=O)NCC(F)(F)F)CCCO1 56600,C1(C(=O)NCCC(C)CO)(OC)CCN(C(=O)C(O)C(C)C)C1 56601,N1(C(COC)=O)CCC(CNC(C2COCCN2CC(F)(F)F)=O)C1(C)C 56602,C(=O)(C1=CCCCCC1)N1C(CNC(C2CC(OCC)C2)=O)C(C)CC1 56603,N1(C(CCC=C)=O)CCC(C2CCN(C(c3nc(CC)no3)=O)CC2)C1 56604,C1(C(CC)CC)CC(C(N2CCN(C(=O)CCO)CC2)=O)CCO1 56605,c1(NC(c2c(C(C)NC(CCC(CC)=O)=O)noc2)=O)cn(C)c(=O)cc1C 56606,C1(NC(c2ccc(CCC)[nH]2)=O)CC2CC(NC(C3(c4cc[nH]n4)CC3)=O)C2C1 56607,C1(C(=O)NCC(CC)(C)C(N)=O)CC(C)(C)CCN1C(C1CCOC1)=O 56608,C1(N(C(=O)CCC(=O)OC)C)CCCN(C(=O)COCCCF)CC1 56609,N1(C(c2c(COC)cc[nH]2)=O)CCN(C(=O)Cc2ccc3c(c2)CC3)C2(CC2)C1 56610,CCC(CC(F)(F)F)C(=O)NC12CCCC1N(C(=O)C(C)(F)F)CC2 56611,Cc1cc(C)c(CC(=O)NC2CCC2NC(C2CCC3(CCC3)O2)=O)c(C)c1 56612,C=CC(C)CC(=O)NCC(CO)NC(c1sc(=N)[nH]c1C)=O 56613,CCCC(O)CC(=O)N1CC(NC(=O)CC2=CCCC2)C(C)(C)C1 56614,c1(C(=O)NCC2C3CCC(C3)N2C(c2ccsn2)=O)ccc(Br)c2cc[nH]c12 56615,c1(C(=O)NCCNC(C2N(OCC)CCC2)=O)cccc2nc(N(C)C)oc12 56616,C(C)(C)(C(=O)N1CC(C(C(=O)NC2(C(C3CC3)OC)CCC2)OC)C1)OC 56617,c1(OC)ccc(OCC(C)=CC(N2CC(O)(CNC(=O)C(N)=O)C2)=O)cc1 56618,N1(C(c2c(C)cc(C)s2)=O)CCN(C(=O)Cc2c[nH]c3cnccc23)C2(CC2)C1 56619,S(=O)(=O)(c1ccc(C(=O)NCC23CCC2CNC3)o1)N(C)C 56620,c1(N2CCN(CC#C)CC2)nc(C2CCN(C(CC(=O)NCC)=O)C2)nc(=N)[nH]1 56621,CC1(NC(=O)CCNC(N)=O)CCN(C(=O)CCc2cccc(F)c2)CC1 56622,C(C(C)C(F)C(=O)NCCC(F)(F)C(C)C)NC(c1cc(C)ns1)=O 56623,C1(N(C(CCC(=C)Cl)=O)C)CCCN(C(c2nocc2Br)=O)CC1 56624,CC(=O)C(C)(C)CC(=O)NCCOCCCN(C)C(c1cc(C(N)=O)c[nH]1)=O 56625,C(=O)(C1=CC(O)CCC1)NCC(C)N(C(Cn1cccc(C)c1=O)=O)C 56626,c1(C(=O)NC2CC(NC(=O)CC3CCCC34CC4)C2)cc2ccc(Cl)c(F)c2o1 56627,C(=O)(C(CC(F)F)N(C)C(C1CCOC1C(C)C)=O)NCC(=C)CC 56628,C1(N(CCONC(c2ccccc2)=O)C(C2CCOC2)=O)CCSCC1 56629,C(=O)(C(C)(C)CC(C)C)NC1C(N(C(C(F)=CCC)=O)C2CCCC2)CC1 56630,Cc1ncc(C(=O)NC(C)C(C)(C)C(=O)NC2CC3(CCC3)C2O)c(=N)[nH]1 56631,C(=O)(CCC(F)(F)C(F)(F)F)N(CCC)CCNC(C1(C)CCOC1)=O 56632,C1(N(C)C)CC2CC1N(CC(N1CCCCC1NC(c1cc[n+]([O-])cc1)=O)=O)C2 56633,c1(C(=O)NCC2C(C)CN(C(C3C=CCC3)=O)CC2)cc2cc(F)ccc2s1 56634,c1(C(=O)NCCCNC(CC)=O)ccc(CNC(=O)C(C)CN(C)C)cn1 56635,N1(C(c2c(C#C)cnn2C)=O)CCC2(NC(=O)CCC(=O)NC)CCCC12 56636,C1(N(C(CCN(C(C)C)C)=O)C)CCOC(C)C1.C1C(=O)N1.C1C(=O)N1 56637,N1(C(C(COC)NC(C2(COC)CC2)=O)=O)Cc2[nH]nc(C(=O)N(C)C)c2C1 56638,c12ccc3c(c1)CCC3NC2=O.c1(C(=O)O)cccc(Cn2ccnn2)c1 56639,Cc1cc(C(C)NC(c2ncoc2C)c2nnnn2C2(C)CC2)ccc1F 56640,C1(C(=O)NCC)(OC(C)(C)C)CCN(C(C2(O)CC(F)(F)C2)=O)C1 56641,c1(C(=O)NCCCNC(c2c(NC)scn2)=O)cc(OC)cnc1F 56642,CC1CCCC(C(=O)NCCOC2CCN(C(=O)CCC3CCCC3)C2)C1 56643,CCC(CC)CC(=O)NC1CC1NC(=O)C(C)(C)C(C)C 56644,Cc1cccc(C(=O)NCCOC2CN(C(C3(CC(C)C)CC3)=O)C2)c1F 56645,c1(C(=O)NC2CCN(C(Cc3cncc(C)c3)=O)C2)ccc2c(c1)CCC2=O 56646,C1(C(=O)NCCC(C)N(CCC)C)C=CCCN1C(=O)Cc1ccsc1 56647,C(c1ccc(Cl)cc1Cl)=CC(N1C(C(=O)Nc2ccc(Cl)cc2O)CC(F)C1)=O 56648,N1(C(C(CC=C)OC)=O)CCCC(C(=O)Nc2cnc(F)c(C)c2)CC1 56649,c1(SC)cc(C(=O)N(CCNC(=O)C(C2CCCO2)SC)CC2CC2)co1 56650,c1(COC)cccc(C(=O)NC2CCCC(NC(=O)CSC(C)(C)C)C2)c1C 56651,C1(C)(NC(C(C)CC2CCC2)=O)CCN(C(=O)CCCF)C1 56652,CC1(C)CC(C(N2CCCC(O)(CNC(c3ccsc3Cl)=O)C2)=O)CC(C)(C)S1 56653,C12CC13CCC(CC3)N2.c1(C(=O)OC)sc(-c2ccc(Br)cc2)cc1Br 56654,c1(CC(=O)NC2(CCNC(Cc3cc(C)n(C)n3)=O)CC2)ccc(Cl)c(Cl)c1 56655,C12(CNC(=O)COC3CC3)CCC(CC1NC(=O)C(C1CCOCC1)O)C2 56656,c1(OC)cc(F)cc(F)c1S(=O)(=O)NC(C)(C)Cc1cc(F)cc(F)c1 56657,c1(-c2ccc(CC)cc2)cccc2c(C(N3CCC(C(N)=O)C3)=O)[nH]nc12 56658,N1(C(C(CC(=C)Cl)NC(=O)CCC2CCC2)=O)CCC12CCN(C)C2 56659,C1(C(N(CC(=O)N(C)C)CC)=O)CC12CCN(C(=O)CC(C)(F)F)CC2 56660,c1(C(=O)OC)cc(C(=O)NC2(NC(c3coc(C4CC4)c3)=O)CCOC2)cn1C 56661,c1(CCN)nnc2n1CCOC2.CCC(F)(F)CCC1(C)n2nnnc21 56662,c1(CC(=O)NCC2(F)CC(CNC(=O)C=CCN3CCC3)C2)csc2nccn12 56663,c1(C(=O)NCC2(COC)CN(C(C3CC4CC4C3)=O)C2)cnc2n1CCCC2 56664,C(CC(C(=O)NC(c1cn[nH]c1)C)NC(c1[nH]ccc1C)=O)OCC 56665,C(=O)(C(C)(F)C(=O)NCC(C)(F)CNC(=O)C(C)(C)c1cccnc1)OC 56666,S(=O)(=O)(c1ccc(I)s1)NCCC(Cn1cc(C(N(C)C)C2CC2)nn1)(F)F 56667,C1(NC(c2c(C)nccn2)=O)(CNC(C2CCCC2C)=O)CC2CCC1CC2 56668,N1(C(C(CC=CCC)C)=O)CC(NC(=O)CCC2CCCCCC2)CC(C)C1 56669,C(C(C)(O)CC(=O)NCC1CC(C)(C)CN1C(c1cc(Cl)ns1)=O)OC 56670,Cc1ccc(CN2CC(CC(N3CCOC(C)C3)=O)C2)cc1[N+](=O)[O-] 56671,c1(C(N(CC(C)CNC(=O)Cn2cnnc2)C)=O)cccc(CF)c1 56672,C(=O)(C1c2c[nH]nc2CN1C(c1cc(CO)on1)=O)N(CCCC)CCCC 56673,S(=O)(=O)(c1ccccc1N)N(c1ccc(NCCCc2ccccc2)cc1)C 56674,CC(O)CC(=O)NCCCCNC(=O)Cc1ccc(Br)s1 56675,c1(C(=O)NCCC2N(C(c3ccc(C(C)=O)o3)=O)CCC2)ccc2c(n1)CCC2 56676,C1(NC(c2n(CC#N)ncc2)=O)CN(C(=O)Cc2cnccn2)CC12COC2 56677,c1(C(N(C)CC2(CNC(C3CCC4CCC34)=O)CC2)=O)ccc(S(N)(=O)=O)s1 56678,N1(C(C2CCN(C)C2=O)=O)CCC(C)(NC(c2cc(O)nc(Cl)c2)=O)CC1 56679,O=C(CCC(=O)c1cccnc1)NC1CCCCC1NC(C1(CC2CC2)CC1)=O 56680,c1(C(=O)NCCCCNC(C2C(C)CCO2)=O)c(F)ccc(Cl)c1[N+](=O)[O-] 56681,C1(O)(CC(=O)N)CCCCC1.C1(C(C(C2CCCCC2)C)=O)CCC(N(C)C)C1 56682,C(C(=O)NCCOC1CCN(C(c2ccc(C)n2C)=O)C1)(C(C)C)OC 56683,C1(NC(c2c(C)coc2C)=O)C2CCC1N(C(c1cscc1Br)=O)C2 56684,n1(CC)nnnc1C(c1nc(C(=O)OC)co1)NC1CC1c1ccccc1 56685,C1(C(C)C)C(=O)N1.CCC(C(=O)c1nc(CNC(=O)COC2CC2)sc1)SC.C 56686,Cn1nccc1C=CC(=O)NCCCNC(c1cc(C(C)(C)O)ccn1)=O 56687,N1(C(c2scc(COC)c2)=O)CC(O)CC1(C)CO.c12ncccc1C(=O)NC2 56688,C1(C(=O)NC(C(=O)N(C2CC3CCC2O3)C)(C)C2CCC2)Cc2nccn2C1 56689,CC1(C)CC(C(=O)NCC(O)(CO)CO)CN(C(=O)Cn2cnnc2O)C1 56690,c1(-c2cccc(OC(C)C)c2F)c(C(=O)NCC2CCCOC2)[nH]c2ccccc12 56691,C(=O)(C(F)C(C)CNC(=O)CC1CC=CC1)N1CC(CSCC)C1 56692,CC1CC(NC(C2COCCOC2)=O)CN(C(c2ccsc2C(F)F)=O)C1 56693,N1(C(=O)C(C2CCCCC2)O)CC2(C=C(C(=O)N3CCOC4C(O)CC34)CO2)C1 56694,Cn1ccc(C2CC2NC(=O)Cc2csc(N3CCCC3)n2)n1 56695,CCCC(C)CC(=O)N(CCCNC(c1cc(C)nc(C)n1)=O)C(C)C 56696,N1(C(C(C)=CCC)=O)C2CCC(C2)C1CC(N1CCOC2CC12)=O 56697,N1(C(=O)C(F)F)CCCC2C(CCCN2C(c2cc(F)c[nH]2)=O)C1 56698,C1(CC)CC(c2nnnn2CCCOCC)(NCCC2CC2)CO1 56699,C(=O)(C#CC1(C)CCCO1)N1C(CN(C)C(c2cn(C)nc2C(F)F)=O)CCC1 56700,c1(C(N2CC3C(CNC(c4nc(C(C)C)sc4)=O)C3C2)=O)ccc(Cl)c(F)c1N 56701,c1(NC(C2N(C(c3ncc(C)nc3)=O)CCC2)=O)cccc(Cl)c1O 56702,C(=O)(CCCCCCCC)N1C(CNC(CC=CC)=O)CC2(CCC2)C1 56703,Cc1snnc1C(=O)NCC1CCC(NC(C2CC(O)C2)=O)C1 56704,N1(C(c2n(CC)ncc2)=O)CC2(C(=O)NC(COC)C(C)C)CCC1CC2 56705,C1(NC(C(C)(CO)NC(C(CN(C)C)N(C)C)=O)=O)CN(C)CC1(F)F 56706,C(C(C)(F)C(C)C)NC(c1c(CNC(CSCCC=C)=O)cco1)=O 56707,n1(CC(C)(C)CO)nc(C2CCCO2)nc1-c1ccc(Cl)o1 56708,C1(CC(C)NC(C2CCC(O)(c3ccccc3)C2)=O)CC(C)CC(C)(C)C1 56709,N1(Cc2cc(OC(C)C)cc(C(=O)OC)c2)CCC(C#N)CC12CC2 56710,C1(CC(N2C(CN(C(=O)Cn3cc(Br)cn3)C)CCC2)=O)COCC(C)(C)O1 56711,c1(CNC(C2CC(=C)CN2C(C2(O)CCC2)=O)=O)cc(C(F)(F)F)cc(Cl)c1 56712,C1(CNC(CCCOCCOCC)=O)CN(C(=O)C=C2CCN(C)C2)CC1C 56713,c1(C(=O)NCCCOCCN(C)C(c2sccc2C2CC2)=O)nn[nH]c1Cl 56714,C=C(C)CCC(=O)N1CCC(NC(C2CC(C)=NO2)=O)C1CC 56715,C1(CNC(C2CCCC2F)=O)COCCN(C(C2CCCOCC2)=O)C1 56716,N(C(=NCc1ccc[n+]([O-])c1)NCC1(N(C)C)CCOCC1)C(CC)CC 56717,N1(C(c2nn(CC)c(O)c2)=O)CCC(NC(=O)C2=CCCCC2)CC1C1CC1 56718,C(=O)(C(CC(C)C)C(N)=O)NC(C(=O)NCCOCC#C)C(C)C 56719,C(CNC(C1CC1C1CC1)=O)(C(C)(C)C)NC(c1n(CC)ncc1)=O 56720,C(c1cccc(F)c1F)=CC(=O)N(C1CCC(NC(CC(C)N(C)C)=O)CC1)C 56721,N1(C(c2c(C)cc(F)s2)=O)CCC2(CCCCC2NC(=O)CCc2cnco2)C1 56722,c1(CCC(N2CC(NC(C(CC)N(C)C)=O)C(F)C2)=O)cnc2ccccn12 56723,Cc1cc(Br)c(C(=O)NC2CCC(F)(F)C2)cc1Br 56724,C1(NC(CC(CC)C2CC2)=O)CCSC12CN(C(=O)CN1CC3C=CC1C3)C2 56725,CC1Oc2ccc(C(=O)OCC(=O)N(C)C(c3ccccc3F)C)cc2NC1=O 56726,c1(C(=O)NCCCCCNC(C2(C)CC=CCO2)=O)nnn2c1CCC2 56727,c1(C(=O)NCC2C(NC(COCC)=O)COC2)cc2ccccc2cc1OC 56728,C1(C(=O)NCCCN(C(c2c(C)snc2)=O)CCO)CCCOCC1 56729,N1(C(C2C(C)C2)=O)CC(CNC(=O)Cc2nc[nH]n2)C2(CCC2)C1 56730,c1(CN2CC(CC(=O)Nc3cc(Cl)cnc3Br)OCC2)cc(Br)c(O)cc1O 56731,C(=O)(C1SCCc2ccccc21)N1CC2(CN(C(C(C(C(C)C)O)(F)F)=O)C2)C1 56732,C(=O)(C1=NOC(CNC(=O)CCc2ccco2)C1)N1C(C#C)CCC1 56733,c1(C(=O)NC(C2CN(C(c3c(NC)cncc3)=O)C2)C)ccc2nc(O)cn2c1 56734,Nc1nonc1C(=O)NCC1(CC(N2CCC(F)C2)=O)CC1 56735,C1(NC(C2CC(C(=O)OC)C2)=O)CCCN(C(=O)C(C)C(C)O)C1 56736,CCN(Cc1ccoc1)N1CCc2cc(O)c(CC)cc2C1 56737,N1CC2C=CCC(C2)C1.c1(C2CC(N(CCC(=O)N(C)C)C)C2)ccccc1 56738,c1(CC(N2C(CN(C(C(F)=C(C)C)=O)C)COCC2)=O)c[nH]c2ccc(Cl)cc12 56739,Cc1cn(C)cc1C(N1C(C(N2CCOC(CN=[N+]=[N-])C2)=O)CCC1C(C)C)=O 56740,C(CCCCSC)N(C=O)C.C12(CC(=O)NCC3(C(C)(C)OC)CC3)CCCC1C2 56741,c1(C(=O)NC(CCC=C)C(=O)N2CCC(C)(CCO)C2)cccc2ccnn12 56742,c1(-c2ccn(C(c3nc(CCO)nn3CC(=O)O)C)n2)ccc(Cl)cc1Cl 56743,N12CCCN(CC1C)C(=O)c1nc(C)c(s1)C2=O.C1(OCC)(CSCC)CC1 56744,c1(CC(N2CC(n3cc(CCN(C)C)nn3)C2)=O)c(F)cccc1F.CC1CC1 56745,c1(C(=O)NC23CN(C(C(C=C)O)=O)C(C2)C3)ccc(C#N)cc1F 56746,C1(CC(=O)NCC2CCN(C(c3ncoc3C3CCC3)=O)C2)CC(=O)NC(=O)C1 56747,Cc1cc(C(=O)NCC2CC2CNC(=O)C(C)N(C)C)nc2ccccc12 56748,N1(C(c2nc(C)oc2)=O)CCC(CNC=O)(CO)CC1.c1(C23CC2C3)cnn(C(F)F)c1 56749,CS(=O)(=O)c1ccc(F)c(C(=O)NCC2(F)CC(NC(=O)C(F)F)C2)c1F 56750,c1(C(N(C2CCN(C(=O)C(O)CN3CCCC3)C2)CC)=O)ccc(=O)oc1 56751,C#CC1CC2(CC(C(N3CCN(C(=O)C(C)(C)NC(C)=O)CC3CO)=O)C2)C1 56752,CC(C)CC(C)(CNC(C1(Cl)CC1(C)C)=O)NC(c1cccc(C2(C)CC2)c1)=O 56753,Cc1cc(C(=O)NCC2CCN(C3CCN(CC4CC4)C3)C2)cc2nc[nH]c12 56754,CCC(C(=O)N1CCC(CC(=O)NCC(C)(O)Cn2cccn2)C1)C(C)(C)CC 56755,c1(OC)cccc(C(N2CC(NC(C3(OC)CCCOC3)=O)CC2CO)=O)c1N 56756,C1(C(=O)NCCN(C)CCF)CC2(CCC2)CN1C(=O)C(F)n1ccnc1 56757,c1(C(N2CCCC(N(C(C(CC)N(C)C)=O)C)CC2)=O)cc2n(n1)CCNC2=O 56758,N1(CCCC)CCCCC1C(=O)NC1CCOCC1NC(c1cc(CC)[nH]n1)=O 56759,N(C=CC(=O)C(F)(F)F)C(=O)CC1CN(Cc2cc3ncccc3[nH]2)CCO1 56760,C(=O)(C(=O)CCC(C)C)N1CC(CCC)C(NC(c2cn(C(C)C)nn2)=O)C1 56761,C1(NC(CN(CC(C)C)C(c2n(CC#C)cnn2)=O)=O)CCC2(CCC2)C1 56762,C#Cc1cccc(C(=O)NC2CC(CNC(=O)CN(C)C3CC3)C2(C)C)c1F 56763,c1(C2(CNC(c3c(CS(=O)(=O)NC)onc3)=O)CCCC2)cccc(F)c1 56764,N1(C(C2CCC(C)C2)=O)CCOC2(CCN(C(c3cc(Cl)ccc3N)=O)C2)C1 56765,C1(CC(=O)NC2(C(N(CCOC)C)=O)CC2)CCC(C#N)C1 56766,c1(C(=O)NCC2(F)CC(CNC(COCCC(C)C)=O)C2)ccc(F)c(N)c1F 56767,CCCC(C(=O)N1CCC(NC(c2cncs2)=O)C(O)C1)C(C)C 56768,N1(C(c2c(C)ncs2)=O)CCC2(CCCC2NC(c2cc(O)nc(O)c2)=O)CC1 56769,N1(C(c2c(OC)c(F)ccc2)=O)C2CCC1CN(C(=O)Cc1cccnc1)C2 56770,c1(SCC(=O)NC2CCC2NC(C2CNC(=O)N2)=O)c(F)cccc1F 56771,c1(OCCC(=O)NC2(C)CCN(C(=O)CC3CC3)C2)ccc(F)cc1Cl 56772,c1(-c2cccc(C(N3CCC(COC)CC3)=O)n2)csc2ccccc12 56773,C1(CCNC(=O)C(=O)Nc2ccccc2)(CSC)CCCC1 56774,CCC(CCOC)C(=O)N1CCCC(CC(=O)NCC2C=CCOC2)C1 56775,C1(F)(C(N2CCC(NC(=O)C(Cl)=CCl)C2)=O)CCN(C(c2ccccc2)=O)CC1 56776,C1(NC(c2n(C)nc(C3CC3)c2)=O)CC2CN(c3cnc(C#N)cn3)CC12 56777,N1(CC(=O)NCCCCN(C(=O)CCc2cn(C)cn2)C)CCn2nccc21 56778,c1(C(C)(CO)N(C(=O)C(C)(C)NC(=O)OC(C)(C)C)C)cccc(O)c1 56779,Cc1nc(=NCC(C)NC2CCN(C(=O)OC(C)(C)C)CC2C)s[nH]1 56780,C1(CNC(C(C)OC)=O)CCC(NC(C2CCOC2)=O)CC1 56781,C1(NC(C2CC(F)CN2C(=O)Cn2ncnn2)=O)CCn2ncnc2C1 56782,C#CCC(CC(F)F)C(=O)NC(CNC(c1nccnc1C(N)=O)=O)CC(C)C 56783,Cc1cccc(CONC(C2CC(C)N2C(=O)C(C(C)O)N(C)C)=O)n1 56784,N1(C(c2ncccc2CO)=O)CCC2(CC1)CCN(C(C1CC3(CC3)CO1)=O)C2 56785,C(=O)(CC(C)(C)NC(C1COCCC1C)=O)NCC(=O)NCCOC 56786,c1(CC(=O)NC2CC(CC)(CC)N(C(=O)CN(C)C)C2)cnn2ccccc12 56787,Cc1nn(C(C)(C)C)cc1C(=O)NCC(CO)NC(=O)C(C(C)C)N(C)C 56788,Cc1ccnc(C(=O)NCCC(C)NC(=O)CC2CCC2(F)F)c1N 56789,c1(C(N2CC(NCc3ncccc3Br)CC(F)C2)=O)cc(Br)c(O)c(Br)c1 56790,Cc1cncc(C(=O)NCCN(C(=O)Cc2cnc(C3CC3)[nH]2)C2CC2)c1 56791,S(=O)(=O)(c1cccc2nsnc12)NC(C)C(N1CCC2C(O)CC2C1)=O 56792,N1(C(C(N2CCOC2=O)C)=O)CCN(C(=O)COCC2(F)CC2)C(C)C1 56793,CCCC(C(=O)NC1CC2C(NC(c3[nH]nnc3C(F)F)=O)C2C1)OC 56794,C=C1COCCN(C(=O)C(CN(C)CC)NC(C2CC2c2ccccc2)=O)C1 56795,S(=O)(=O)(c1cc(C(F)(F)F)ccc1Cl)NC1CCN(C(c2cscn2)=O)CC1F 56796,N1(C(CC(C=C)C)=O)CCN(C)CC1CNC(c1ccn(CCF)n1)=O 56797,c1(OC)ccc(F)c(N)c1C(N1CCC(C(C)NC(C2C(C)(C)C2(C)C)=O)C1)=O 56798,N1(S(CCOCC)(=O)=O)CCC(O)C(C(=O)Nc2cnc(SC)nc2Cl)C1 56799,C1(C(=O)NC(CSCC)CO)(CSC)CCCOC1 56800,C(CCNC(C1CC1C(C)(F)F)=O)(C(=O)NCC(c1ccncc1)C)OC 56801,CCCCCCC(F)C(=O)N1CCC(CN(C(=O)COCCSC)C)CC1 56802,S(=O)(=O)(c1ccc(NCc2cccnc2F)c(F)c1)N1CCC(OC)CC1(C)C 56803,CCCCCC(O)CNC(=O)CC(CNC(c1c[nH]nc1C(C)C)=O)C1CCC1 56804,C1(NC(N(C2CN3CCC2CC3)C)=O)CN(C)C(C)(C)C1 56805,N1(OC)CCC(O)C(CC(C)C)C1.c1(C)csc(C(=O)N)c1 56806,N1(C(c2ccccc2F)=O)CCC2CCCC12C(=O)NCCCn1cnnn1 56807,C1(CC)CN(C(C2CCOC2CNC(c2cccnn2)=O)=O)CCCO1 56808,c1(C(N2C(CC)CN(C(=O)C(CC)OC)CC2)=O)cc2ccccn2c1 56809,C1(C(=O)NCCN(CCCCCC)Cc2ccccc2)(CC)CCNC1=O 56810,C1(C(=O)NCC(C(=O)Nc2csc(C)c2)N(C)C)(COC)CCOC1 56811,C1(c2c(C)n(C)nc2)C(C(=O)N(C)Cc2cnco2)CC(=O)N1C 56812,C(C)(C(C)(C)NC(C1CC=CCC1)=O)NC(CC1C(C)CC1)=O 56813,c1(C2CN(Cc3c(CNC(=O)OC(C)(C)C)scc3)C2)cccc(Br)c1 56814,c1(-c2nc(CC3(SCC)CC3)nn2-c2cnn(C)c2)ccnc2[nH]c(CC)nc12 56815,c1(CCC(N2CC(O)(CNC(CCCOCC)=O)C2)=O)cccc(C(F)F)c1 56816,C(=O)(C(CC)C(C)C)NC(C(=O)N(CCOCC#C)C)CCC1CC1 56817,C(=O)(C1=NOC(C)C1C)NCC(CCOC)NC(c1ccc(CO)c(Cl)c1)=O 56818,C1(CNC(CCCC(C)(C)C)=O)CN(C(=O)CCc2ncc[nH]2)CCC12CCC2 56819,N1(C(CCC(C)(C)C#N)=O)CCCC1C1CCCN1C(c1ccsc1)=O 56820,N1(C(C(CCC)OCC)=O)CCC(CNC(c2cc(C(C)C)on2)=O)CC1C 56821,C1C(C)(CO)NC(=O)CSc2sccc2C(=O)N1.C(CC(F)(F)F)SC 56822,C1(CNC(C2(OC)CCOC2)=O)CN(C(c2coc(C)n2)=O)C2(CCC2)C1 56823,c1(C(C(=O)N(CC(CN(C(C(C(CC)C)O)=O)C)O)C)F)ccc(Cl)c(C)c1F 56824,N1(C(C(C)=CC2CC2)=O)CCC(NC(c2ccnn2C2CCC2)=O)C(CO)C1 56825,C12(CNC(c3cc(COC)no3)=O)CCCC1N(C(C1CCOC1C)=O)CCC2 56826,C(CC1=CCN(c2ncc(I)cn2)CC1)NC(CCC(C)OC)=O 56827,c1(OC)cc(C(=O)NN2CCS(=O)(=O)CC2)ncc1-c1ccc(F)cc1SC 56828,C(=O)(CC(O)CC(C)C)N1CC(O)CC(NC(C=CCC)=O)C1 56829,c1(NC(C2CCCCN2C(c2cc(Cl)ccn2)=O)=O)cncc([N+](=O)[O-])c1 56830,C(=O)(C1CCCc2c1ncn2C)NC1CC(C)(NC(CC=C(C)C)=O)C1 56831,c1(C(=O)NCC(CNC(C2CC2C(F)F)=O)OC)cnc[nH]c1=N 56832,N1(C(c2n(C)nc([N+](=O)[O-])c2)=O)CCC2(CC1)CC(CNC(c1cocn1)=O)C2 56833,CCCCC(O)C(=O)N1CC(F)CC1CC(=O)NC1CCN(CCF)C1 56834,N1(C(C(C(C)C)CCN)=O)CCC2(CC1)CC(O)c1nn(C)cc1O2 56835,c1(C(N(CC(CC)NC(=O)Cc2n[nH]c(C)n2)C)=O)cc(C2CCOCC2)on1 56836,N1(C(c2cc(CC)[nH]n2)=O)CCC(C)(C)C(C(=O)NC(C)Cc2cc(C)[nH]n2)C1 56837,C(=O)(C1=CC(O)CCC1)NC(C)C(C)(C)NC(C1SCCCS1)=O 56838,C1(NC(CCc2ccc(N(C)C)cc2)=O)CCC2CC1CN2c1nccnc1F 56839,C1(N(C(CCC(=O)NC)=O)C)CCCN(C(c2ccc(O)nn2)=O)CC1 56840,c1(C(=O)NCC2C(NC(C(C)n3cnnn3)=O)C2)coc2cccc(O)c12 56841,Cc1c(CN2CC(C)CC2c2ccccc2F)cccc1F 56842,N(C1CCc2cc(Cl)ccc21)C1CN(C(=O)Nc2cncc(OC(C)(C)C)c2)C1 56843,N1(C(C(N2CCC(NC(Cn3c(=N)scc3)=O)C2)=O)=O)CCC(CF)(CO)C1 56844,CCCC(C)(CCC)C(=O)NC(C)C(C)C(=O)N1CCC(CC(N)=O)CC1 56845,N1(C(C2N(C(=O)OC(C)(C)C)CSC2)=O)CC(C(=O)NC2(C)CC2)CC(F)(F)C1 56846,c1(N2CCC(C#N)(F)C2)ccc(Br)c(S(=O)(=O)N2CCC2C2CCCC2)n1 56847,c1(OC)ccc(Cn2cc(C(C)N(C)C(C3CC3(Cl)Cl)=O)nn2)cc1.C1C(=O)O1 56848,CC1CC(C(=O)NC(C2CCN(C(=O)CC3CC3(Cl)Cl)CC2)C)=NO1 56849,Cc1c(CCC(=O)NCCC2(C(=O)NC3CN(C4CCC4)C3)CC2)cnn1C 56850,c1(C(=O)NCC2CC(NC(C(CCC)C#N)=O)C2)[nH]c2cc(Cl)ccc2c1C 56851,CCCC(C(O)C(=O)N1CCC(O)(CO)C1)NC(c1cc(C)c(CC)o1)=O 56852,C(=O)(C(C(C)CC1CC(F)(F)C1)N1CCC(OC(C)=O)C1)NC(CC)C 56853,c1(C(N2CC(C(C(N3CCC(CC#C)C3)=O)OC)C2)=O)cc(F)cnc1O 56854,S(=O)(=O)(CN1CCC(c2cnccn2)CC1)N(C)CC#N 56855,N1(C(CC(C)(C)O)=O)CC(NC(c2csc(Cl)c2)=O)CC(O)C1 56856,C(C1=CCN(C(C2(CF)CC2(F)F)=O)CC1)NC(C(C)Sc1cccnc1)=O 56857,N(C(=NCCC1COC(C)(C)O1)NCC1CCC1)CC(=O)Nc1ccc(OC)cc1 56858,CC1CCCN(C(c2cncc(N(C)C)c2)=O)C1CNC(=O)C(C)(C)N(C)C 56859,C1(C(N(CCC(=O)NC(CCC)C2CC2)CCO)=O)CCN(C)C(=O)C1 56860,N#Cc1ccc(S(=O)(=O)N2C3COCC2CN(C(C2CCC(=O)N2)=O)C3)cc1 56861,C(=O)(CC(C)(F)F)NC(CC)CN(C)C(c1ccnc(NC(C)=O)c1)=O 56862,C(=O)(C(F)(F)C=Cc1ccccc1)NCC1CCN(C(CCNC(N)=O)=O)C1 56863,C(=O)(CCC(C)(C)C#N)N1CC(CC=C)(C(=O)NCC2CC(C3CC3)=NO2)C1 56864,C(CN=c1[nH]c(NC2CCCc3n[nH]cc32)nc2c1CCCC2)(C(C)(C)C)OCC 56865,Fc1ccc(Cl)c(F)c1CCNCCCCc1ccc(F)cn1 56866,c1(OC)ccsc1C(=O)NCC(F)CNC(c1ccn(CC(F)(F)F)n1)=O 56867,C(=O)(CC(C)(C)C)NC1CC(C(C(=O)N(C)Cc2cnccn2)F)C1 56868,c1(OC)cccc2c1CN(C(C1C3CC(CC3F)N1Cc1ccc(C)s1)=O)C2 56869,C1(NC(c2c(C)cc(Br)o2)=O)COCCN(C(=O)C(C)O)C1 56870,c1(OC)ccc(C(=O)NCC(CNC(C2(C)SCCCS2)=O)CO)cc1N 56871,Cc1c(C(N2CCOCC2CCNC(=O)CC(C)N(C)C)=O)cccc1Cl 56872,c1(C(=O)NC2C(NC(C(C=C)C)=O)CC2)nnc2ccccc2c1O 56873,C1(C(=O)NCCCN(C(=O)C(=O)NC(C)C)CCC)CCCN(S(=O)(=O)CC)C1 56874,N1(C(C(OCC)O)=O)CC2=C(C1)CN(C(c1cc3ccccn3c1)=O)C2 56875,C(=O)(C(CCCOC)N1CCCC1COC(C)=O)NCc1ccc(CC)cc1 56876,C1(COC)(CNC(=O)NC(c2coc(C(C)(C)NC3CC3)c2)=O)CC=CC1 56877,C1(NC(C2(NC(CC(C)O)=O)CC(O)C2)=O)CCN(C)C1=O 56878,Cc1c(C(=O)NCC(C)CNC(=O)COCC2CCOC2)ccc(F)c1F 56879,CC(C)C(F)(CNC(c1ccn(C)c1)=O)C(=O)NC1C(O)C2CCOC12 56880,C=CC1(CNC(=O)C(c2cn(C)nn2)NC(C2C=C(C)CS2)=O)CCOCC1 56881,c1(N(CC(C)C)C(=O)NC2CC(SC)C2)ccc2c(c1)OCCO2 56882,N1(C(C2C(C(=O)OC)C2)=O)CC(CNC(=O)CC(C)(C)SC)OC(C)(C)C1 56883,C1(CC)C(C(=O)NC2(CF)CN(C(c3cnc(C)nc3)=O)C2)CCN1C 56884,N1(C(C2N(C(CCC)=O)CCCC2)=O)CC2(NC(C3CCC3C)=O)CCC1CC2 56885,c1(CC(=O)NC2C(C)CN(C(C3CC3(C)C)=O)C2)cc2ccccc2nc1O 56886,CCC(C)(C)C(=O)N1CCC(C(C)CNC(=O)Cc2csnc2C)CC1 56887,N#Cc1cc(Cl)cnc1N1CCCC(NC(C2CC(O)C2)=O)CC1 56888,C1(NC(C(n2c(C)ncc2)C)=O)CN(C(c2scnc2C(C)C)=O)CCC1F 56889,Cc1cc(CNC(c2coc(CNC(=O)C(O)C(C)(C)C)c2)=O)cnc1F 56890,N1(C(c2c(Cl)cc(C)s2)=O)CC(C)CCC1CNC(c1ccc(F)s1)=O 56891,CCC(C)CC(=O)NCCN(CC(CN(C(CC12CC(C(=O)OC)(C1)C2)=O)C)O)C 56892,C(Cc1cc[nH]n1)(C(=O)NCc1ccsc1C)NC(C(=O)NCC)=O.C1CC1 56893,c1(CN(CCN(CCCC)C(C2CCN(CC)C2)=O)CC)c(O)cc(F)cc1F 56894,C=CCC(C)C(=O)NC1CCN(C(c2cn(-c3ccc(C)cc3)nn2)C)CC1 56895,C(=O)(C(C)CCCC(C)=O)N1CCC(CC(N2C(C)CC(CC)C2)=O)CC1 56896,c1(NC(C2CC(NC(c3ccc(C)cc3Br)=O)C2)=O)ccc(C#N)c(Cl)c1 56897,N1(C(c2nc(C(C)C)sc2)=O)CC(NC(=O)C2=CCSC2)C2(CCC2)C1 56898,C1(C(=O)NCC(C(C)C)NC(CCCC)=O)CCCC1(C)C 56899,N1(C(CC(CC)SC)=O)CCC(C)CC1CNC(c1cnoc1-c1ccco1)=O 56900,C(CC)(CC)(CCNC(c1cccc(Cl)c1F)=O)NC(C(CC)n1ccnc1)=O 56901,N1(C(CC(=O)NCC#C)=O)CCC(C)(C)C1C(N1CCC1(C)CCO)=O 56902,c1(NC(C(C(C)C)NC(C(CC)n2ccnc2)=O)=O)cnc(Cl)nc1C 56903,C1(OC)CN(C(=O)CC2CCOCC2)C(C)(NC(c2cc(C(N)=O)[nH]n2)=O)C1 56904,C(C(C1CCCCC1)NC(=O)CCF)(C(C)C)NC(c1ccc(SC)s1)=O 56905,C=CCC(C)(CC)C(=O)N1CCC(CC(=O)Nc2cnc3ncnn3c2)C1 56906,N#Cc1ccc(CCNCc2nnco2)cc1 56907,c1(NCC(c2ncc[nH]2)C)[nH]c(=NCC2CC(CF)C2)nc2c1ncn2C 56908,n1(CC)cc(C(N2CCC2CNC(C23CC(F)(C2)C3)=O)=O)c(C(F)(F)F)n1 56909,c1(CNC(CCOC(C)C)=O)cn(CCCNC(c2ncn(C(C)C)n2)=O)nn1 56910,c1(CC)[nH]ccc1C(=O)NC(CC1CC1)C(=O)NCC1CC1(F)F 56911,c1(Nc2cc(-c3ccc(COCC)c(C)n3)ccc2F)ncnc2occc12 56912,c1(C(=O)NC2C(OC)CN(C(=O)C(CO)N(C)C)C2)cc2cc(Cl)ccc2n1C 56913,n1(CC)ccnc1C(N1CCC1CNC(C1CC(F)(F)C1)=O)=O 56914,c1(COC)ccc(NC(C2CN(C(=O)CCc3ccc(F)nc3)CCS2)=O)cc1 56915,c1(C(C)C)cnc(N2CCCC2CNC(c2ncncc2Cl)=O)c(Cl)c1 56916,N1(C(CCCOCC)=O)CCCC(CN(C(=O)C(n2cc(Cl)cn2)C)C)C1 56917,N1(C(CC(C)C)=O)CCCC(C2CN(C(C3CCc4n[nH]cc4C3)=O)C2)C1 56918,c1(N2CCCCC(NC(=O)CCCCc3cnn[nH]3)C2)nc(Cl)nc2[nH]ccc12 56919,C1(C(CC)CC)C(=O)NCCN1CC(=O)NCc1ccncn1 56920,C1(CC)(NC(=O)CC(C)(O)C2CC2)CCN(C(C2CCCN2C(=O)CSC)=O)C1 56921,N(C(=NCc1coc(C)n1)N1CCC(Cc2cccnc2)C1)C(CC)C 56922,Cc1cc(N2CCN(C(=O)CCF)C(C(C)C)C2)nc(CO)n1 56923,C12(NC(CNC(=O)OC)=O)CC(C(=O)N(C3CC3)Cc3ccco3)(C1)C2 56924,C1(CNC(C(c2nnnn2C2CC2)SC)C2CC2)CC2(CCC2O)C1 56925,c1(C(N2CCCC(O)(CNC(C3(N(C)C)CC3)=O)C2)=O)cc2ccccc2s1 56926,Cc1cc(C(=O)NCC2CC(F)(CNC(C3(C)CC3(F)Cl)=O)C2)ccn1 56927,c1(OC)ccc(C(=O)C(N2CC3CC3C2C(=O)NOCC(O)CO)=O)cc1Cl 56928,N1(C(C2(C)CC(C#N)C2)=O)CCn2nnc(C3CC3)c2C1 56929,CC1COCCN1CCNC(=O)C(=O)NCC1CC12CC(O)C2 56930,CP(C)(=O)C(O)C(=O)N1CCC(CCCCNC(C2CCC(=O)O2)=O)CC1 56931,NS(=O)(=O)CCCC(=O)NCC1CC(O)CN1C(c1ccc2cnoc2c1)=O 56932,c1(OCC)cc(Cn2nccc2NC(c2ccc(N)cc2Cl)=O)ccc1OC 56933,c1(NC(C(C)CSCC2CCN2C(=O)CC2CCCCO2)=O)c(F)cccc1F 56934,N1(C(C2(C3CC3)CN(C(C(C3CC3)SC)=O)C2)=O)CC(C2=NOCC2)C1 56935,CC12CCCC1N(C(C1C3CCN(C(C4CC5CC4CC5O)=O)CC13)=O)CCC2 56936,c1(OC)c(NC(=O)C(=O)NCC2C3Cc4ccccc4C23)nc(O)nc1O 56937,C1(=CC(=O)NC2CC(NC(Cc3ccn(C(C)C)n3)=O)C2)CN2CCC1CC2 56938,C1(C(N2C(C3CCN(C(c4ccc[n+]([O-])c4)=O)C3)CCC2)=O)OC2CCC1CC2 56939,C(=O)(C(F)(F)C(F)F)N1CCC(C(CNC(C(C)n2cccn2)=O)F)CC1 56940,c1(CC(=O)NC(C2(O)CN(C(COCCCC#C)=O)C2)C)cc(F)ccc1CC 56941,C#CCC(CCCO)NC(C1CCCC1NC(C1CC2(C1)CC21CC1)=O)=O 56942,c1(C(=O)NC2CC(NC(CCC#C)=O)C2)ncn2c1COc1ccccc1-2 56943,c1(SCC(=O)NC2CCN(C(C3CCCC3O)=O)C2)n[nH]c(O)n1 56944,C(=O)(CCC(=O)NC1C2CC1N(C(=O)CN(C1CCCCCC1)C)C2)N(C)C 56945,C1(C(=O)NCC(CNC(C2(N3CCCC3)CCC2)=O)OC)CC(C)CC(C)(C)C1 56946,c1(NC(N2CCC(NC3CCC3)C2)=O)ccc(C(F)(F)F)cc1O 56947,CCCC(C)(C)CC(=O)NCC(C1CC1)N(C)C(c1cc(CC)on1)=O 56948,c1(NC(C2(NC(CC3CC(=C)C3)=O)CC(F)C2)=O)ccc(F)cc1C 56949,C(CC(C)(C)CC(=O)N1CC(NC(c2cn(C(F)(F)CO)nn2)=O)CC1C)OC 56950,C=CCC(CNC(=O)CCC(=O)NC(C)CC)C(=O)NC(C)C 56951,c1(C(=O)NCC(CC)NC(=O)C(c2cccnc2)C)nn(C)c(Cl)c1Br 56952,N1(C(C2CCN(C)S2(=O)=O)=O)C2CCC1CN(C(C1CC(CCO)C1)=O)C2 56953,Cn1cc(Cl)c(CC(=O)NCC=CCNC(c2cnccc2-n2cccn2)=O)n1 56954,C1(C(C#C)NC(=O)NCC(O)Cc2cccc(F)c2)CCCCCC1 56955,CC(C)C1=NOC(C(=O)NCCOCCNC(=O)Cn2cc(Br)cn2)C1 56956,Cc1cc(C(=O)NC(Cn2cc(CC3CC(F)(F)C3)nn2)CC(C)C)c(C)s1 56957,CC1CCC=C1C(=O)N1CCOC(CNC(=O)Cn2ccc([N+](=O)[O-])n2)C1 56958,c1(CNC(C2C(C(C)C)CCO2)=O)cnn(C)c1C(=O)NC(C(C)C)C1CC1 56959,C1(C(=O)NCC2(C(N3CC(C(N(OC)C)=O)C3)=O)CC=CC2)CC12CCOC2 56960,N1(C(c2ncnc(C)c2C)=O)CC2CCCC1C2CNC(c1ccc(F)cn1)=O 56961,c1(C(=O)NC(CNC(c2c(C)n(C)nc2Cl)=O)C)noc2c1CC(F)(F)CC2 56962,CC1(C)CCC(C(N2CCCC(CNc3ccccn3)C2)=O)C1 56963,C(=O)(CCCCCCCC1CC1)NC1CCC(NC(C(CC=C)CC)=O)C1 56964,C(C)(C)(C(C)CC(=O)N1CC(C)CC(O)C1)NC(C(C)OCCN(C)C)=O 56965,C1(CNC(=NCCC)NCCC2CCOCC2)CCC2(CCCC2)O1 56966,CC(O)CCCNC(=O)CC1CCCC1NC(=O)Cc1ccsn1 56967,c1(OC)ccc(Br)cc1C(=O)NC1CCCN(C(=O)Cn2ncnn2)CC1 56968,N1(C(C(CC)SC)=O)CCCC2(CCN(C(C)C(=O)N(C)C)C2)C1 56969,c1(C(=O)NC(CNC(CSCC(=O)OC)=O)CO)ccc2c(c1)CCCS2 56970,C(=O)(C(O)CC(C)C)N1CCCC(CN(C(C2CN(C(C)C)C2)=O)CC)C1 56971,c1(C(N2CCN(Cc3cnc(CCCC)[nH]3)C3C2C3)=O)ccc(F)c(OC)c1F 56972,C1(c2cn(Cc3c(CC)ccs3)nn2)C(C)CCN1C(=O)C(C)N1CCC1 56973,c1(C(=O)NC(C2CCOC2)CNC(C2(CC)CC2)=O)ccnc2ccc(F)nc12 56974,N(C1CN(C(c2cc(C)c(Cl)c([N+](=O)[O-])c2)=O)Cc2ccccc21)C(C)=O 56975,c1(C(N2CCC(NC(c3ccoc3Cl)=O)C2)=O)ccc2occc2n1 56976,C1(CC(=O)NC(C2(C(=O)NCC(C)Cn3ccnc3)CC2)C)CCCCO1 56977,Cc1cc(Cc2cccnc2)ccc1C(=O)NOc1ccc(C2(C)CC2(F)F)cc1 56978,C1(NC(c2c(OC(C)C)n[nH]c2)=O)CCN(C(c2n[nH]cc2Cl)=O)C12CC2 56979,C(=O)(C(C)C(C)C(C)(C)C)N1CC(CCO)(NC(C(C)=C(C)C)=O)C1 56980,C(=O)(C(O)C(C)(C)CC)N(CCNC(C1N(CCC)CCC1)=O)C 56981,C1(COC)N(c2ncnc(N(C)C)c2Cl)CCCC1(C)C 56982,Cn1ncc2nc(Cl)nc(N3CCC(O)(CCNC(=O)CCF)CC3)c12 56983,C1(NC(c2ccon2)=O)CCN(C(C2CC(C3CC3)C2)=O)CC(O)C1 56984,C(=O)(C(C)C(C)(C)C)NCC1N(C(CCCc2c(C)ccs2)=O)CCCC1 56985,c1(C(=O)NCC2CC(NC(C3C(C)C3)=O)C(O)C2)cc([N+](=O)[O-])c(F)cc1N 56986,CC1CCN(C(=O)C(F)C(C)(C)O)CCN1C(=O)CCc1cnc2n1CCOC2 56987,c1(C(N(CCC(C)NC(C2(CO)CCOC2)=O)C)=O)cc(Cl)ccc1N 56988,C(=O)(CC1=CCCCC1)N1C(C)CCC(NC(=O)Cc2nnc(S)n2C)C1 56989,C1(NC(C2(CNC(C3CCCCC3O)=O)CC(=C)C2)=O)CCC2CCCC1O2 56990,N1(C(C2(NC(C3CC(CC)(CC)C3)=O)CC(CO)C2)=O)CC2CCCCC12C 56991,c1(C(CNC(CCCC)=O)NC(c2[nH]cnc2C)=O)ccc(Cl)cc1 56992,N1(C(=O)NC(C)(CO)C(F)(F)F)CCC2(CCOC2)C(CO)C1 56993,C(=O)(CCCCCN(C)C(C)C)NC1(CCNC(C(CC)C)=O)CCC1 56994,c1(CC(N2C3CC(N(C)C)(C3)C2)=O)cc(-c2nn[nH]n2)cc(Br)c1 56995,C#CCC(CO)NC(c1n[nH]cc1CNC(c1c[nH]cc1C(C)C)=O)=O 56996,C1(C(C)(C)NC(C=CCOC)=O)CCCN1C(=O)C(n1nccc1C)C 56997,N1(C(CCN(C)CC)=O)CCC(NC(C2(C)CC(O)CN2C)=O)C(F)C1 56998,C1(C(=O)NC2(COCC)CC2)CNC(=O)CN1C(=O)C=CC1CCCN1C 56999,C(=O)(CS(=O)(=O)CC(=O)N1CCN(C(=O)C(C)N(C)C)CC1CF)OC 57000,C(=O)(C#CC(C)(C)C)NCCOC1CCN(C(c2nn(C)c(Br)c2)=O)C1 57001,C1(CNC(=O)COC2CCC2)CC2(CO1)CN(C(C1CCC(=O)O1)=O)C2 57002,C(=O)(C(C)S(N)(=O)=O)NCC1(C(C)NC(C2CC3CC2CC3O)=O)CC1 57003,CN=c1[nH]cc(C(N2CC(O)CC2C(=O)NCC2C=CCOC2)=O)o1 57004,C1(NC(C2CCC(C(C)C)CC2)=O)CN(C(=O)C(F)F)CCC1(F)F 57005,C1(C(=O)NC2CN(C(c3ccn(C)c3)=O)CC23CC3)CCC2(CC1)CNC(=O)C2 57006,C(=O)(CCCCC(=O)N1CCC(C)(C)C(C(=O)NCc2ccc(Cl)o2)C1)OC 57007,C1(C)OCCCC1(C)C.C1(C)(C2CC2)C(=O)N2CC(C2)CC(=O)N1.CC(=O)NC 57008,N1(C(COCCCC#C)=O)CC=CCC1C(N1CCCC(COCC)C1)=O 57009,Cc1ccc(S(=O)(=O)N2CC(NC(c3c(C(F)(F)F)cccc3F)=O)C2)cc1C 57010,CCC(O)C(C)(C)C(=O)NCCCN(C)C(c1csc(-c2ccc(Cl)cc2)c1)=O 57011,C(=O)(C(C)(CO)NC(C1CC(C#N)(OC)C1)=O)NCc1n(CC)ncn1 57012,Cc1nc(C2CCCO2)sc1C(=O)NC1COCC1NC(c1ccccc1O)=O 57013,N1(C(=O)NCC=C)CCN(C(=O)NC(c2ccc(C(=O)OC)cc2)=O)CC1CC 57014,c1(C(N)=O)cc(Cl)ccc1NC(=O)CCC1CNC(=O)N1 57015,C1(CC(=O)NC(C2CCN(C(CC)=O)C2)C(C)(C)C)CCC(NC(C)(C)C)CC1 57016,C1(O)(CNC(C(C)C2CC2)=O)CC2CCC(C1)N2C(c1cnc(S)nc1)=O 57017,N1(c2ccnc(NCc3ccc(F)c(C)c3F)n2)CCCC2(CC1)CNC(=O)C2 57018,N#Cc1cc(S(=O)(=O)N2Cc3c[nH]c(=N)nc3C2)ccc1NCC1(F)CCOC1 57019,C1(C)(NC(C(C)C2CCCO2)=O)CCN(C(c2cc(N)cc(O)n2)=O)CC1 57020,C1(N(C(c2cn(-c3ccc(OC)cc3)nn2)=O)C)CN(C(=O)CCF)CC12CC2 57021,CC1OCCN(C(C2CC(=O)NC2(C)C)=O)C1C(=O)NC1CSC1 57022,N1(C(C)=O)CC2CC1CN2C(=O)CC1CC(C)(C)CN1C(C12CC(F)(C1)C2)=O 57023,C1(CC(=O)NC(CC=C)CNC(=O)Cc2sccc2C)CCCC(C)(C)CC1 57024,C1(NC(C(C)C2CC2)=O)CCC2(CC1)CN(C(=O)Cc1csc(S)n1)CCO2 57025,Cc1cccc(C)c1CC(N1CCC(CO)C(NC(c2[nH]c(O)nc2C)=O)C1)=O 57026,N1(C(C(C(CC)C)O)=O)CCN(C(=O)CCCNCc2cccs2)C2(CCC2)C1 57027,N1(C(C(C)OCCC=C)=O)CCC(NC(c2cccnc2SC(C)C)=O)CC1 57028,N1(C(C(C)C#N)=O)CCOCC1CC(=O)N(C)CC1(O)CN(C)C1 57029,C1(C2N(C(CCCC)=O)CCC2)CCCN(C(=O)CCOCC)C1 57030,C1(C)(CCCC(C2CCN(C(c3c(C)cncn3)=O)CC2)=O)NC(=O)NC1=O 57031,C12(CNC(C(C)(C)F)=O)CN(C(c3ccc(OC(F)F)cc3F)=O)CC1CCO2 57032,c1(SCC2(C(N(C3CCN(C(=O)CC4CCNC4=O)C3)C)=O)CC2)ccccc1 57033,n1(CC(=O)NC2COCCN(C(CN(C3CCCC3)C)=O)C2)ncc2cccnc12 57034,C(c1ccc(N2CCCC2=O)cc1)=CC(=O)NC1CCCNC1=O 57035,N1(C(C(=O)NC(C(=O)OC)C)C2CC2C)CCN(c2nc(C)cs2)CC1 57036,N1(C(CCCC(=C)C)=O)CCC2(CCCC2NC(c2[nH]nc3ncccc23)=O)C1 57037,CCCC(CN=c1ccc(Br)c(S(=O)(=O)NC(c2nccnc2C)C)[nH]1)OC 57038,c12ncc(cn1)[nH]c2=O.C1(CC)(NC(=O)COC(C)C)CC(F)(F)C1 57039,CC(C)C(CNC(=O)CC1CCCC1)NC(=O)C(C)n1cnnn1 57040,C1(CN(CC(CC)C)CC)CCCN1C(c1cnon1)=O 57041,c1(OC)cccnc1-c1cn(C2(C(=O)NC(C)CC3CCOC3)CCC2)nn1 57042,N1(C(CSS(C)(=O)=O)=O)CCCN(C(=O)NC2CC(N3CCCC3)C2)CCC1 57043,O=C1CCOC(C(N2CCCC2Cn2cc(Cn3ccnc3)nn2)=O)C1 57044,C1(CC(=O)NCCCn2c(C)ncc2)CCCN(Cc2ccc(C3CC3)cc2)C1 57045,C1(C(=O)OC)CNCCCN1C(C1CSCCN1C(C1CCCCC1)=O)=O 57046,N1(C(c2c(OC)scc2)=O)CC(C)(C)C1C1CCN(C(=O)C2=C(Cl)CC2)CC1 57047,N1(C(C=C(C)C)=O)CCN2CCN(C(=O)CCc3ccccn3)CC2C1 57048,CC1(C(=O)NCC2(O)CCN(C(=O)C3=CCOCC3)C2)CCC(F)(F)CC1 57049,c1(C(=O)NCC2N(C(C(COC)C)=O)CC2)nc(-c2nc[nH]n2)sc1C(C)C 57050,CC(C)C#CC(=O)NCCC(C)NC(=O)CC(C)NC(C1CCCC1)=O 57051,c1(CCC(=O)NC(C2CC=CCC2)C(=O)N(CCCO)C(C)C)nncn1C 57052,C1(C(N2CC(NC(c3cc(C)[nH]n3)=O)C3C(C2)C3)=O)CN2CCCN1CC2 57053,c1(CNC2CCN(C(CSC)=O)CC2(C)C)ccc(C#N)cc1[N+](=O)[O-] 57054,Cc1ncc(Br)c(N2CC(F)(C(N3CC(O)C(F)C3)=O)C2)n1 57055,C(=O)(CCCCC(C)C)N1C2C(NC(c3cccc(COC)c3)=O)CC(C2)C1 57056,Cc1nscc1C(N1CC=CC1CNC(c1cc(C(C)(C)C)n[nH]1)=O)=O 57057,C1(OC)CN(C(=O)CC2(C)CCOCC2)CC1C(=O)NCC1(SC)CCOCC1 57058,c1(N(CC(=O)O)C(N)=O)cccc(C2CC2)c1.CC1CCCC1N1CC(=O)O1 57059,C1(C(=O)NC2C(C(=O)OC)CCC2)CCCCN1C(=O)Cc1ccoc1 57060,C1(NC(C(C(C)OC)NC(C2CC(C)(C)O2)=O)=O)CCC12CCCC2 57061,C1(C(=O)NCCC(COC)(C)C)CCC(C)(C)N(C(=O)Cc2ccsn2)C1 57062,c1(CC(=O)NC(CCCC)CNC(C2CC(C)(O)C2)=O)cnc2ccccc2c1 57063,C1(CC)(NC(=O)CCC2CCCO2)CCCN(C(c2ncc(OC)cc2F)=O)C1 57064,CC1=C(C(=O)NC2CCN(C(=O)CC(C)F)CC2(C)C)S(=O)(=O)CCO1 57065,Cc1nnc(O)c(C(=O)NCC(O)CN(C(=O)Cc2cn3ccsc3n2)C)c1C 57066,CC1(C)CC(N=c2[nH]c(N3CCN(C(=O)CCF)CC3)nc(=N)[nH]2)CC(C)(C)C1 57067,c1(CN2CCN(C(C(CC(C)C)n3ccnc3)=O)CC2)c[nH]c2ccccc12 57068,CC1CCN(C(=O)Cc2cccc(F)c2O)CCN1C(C1CC2CCC(C1)S2)=O 57069,c1(C(C(=O)NC(C)CCNC(c2cc(=O)cc[nH]2)=O)OC)c(F)cccc1F 57070,C(=O)(CC(C)(C)C#N)NCC1C(C(=O)NC2CCN(CC)CC2)C1 57071,N1(C(c2nc(OC)c(C)s2)C(=O)NC)CCC(C)C(C)(C)C1 57072,CC(c1ccccc1F)=CC(=O)N(CC(C)CNC(=O)CCCOC(C)C)C 57073,N1(C(C(C)(C)c2ccccn2)=O)CCC2C(C1)CN2C(c1c[nH]c(C(N)=O)c1)=O 57074,c1(C(N2C(CNC(C(C)SCCCC)=O)CC2)=O)ccccc1[N+](=O)[O-] 57075,CC(C)C(O)C(C)C(=O)N1CCC(N(C(=O)CCn2cnnn2)C)C2(CC2)C1 57076,CN1CCN(C(=O)CC2(C#N)CCCCC2)CC1CNC(c1cnc(F)cn1)=O 57077,CC1(C)CCC(O)(CNC(c2ccc(CNC(=O)CC3CC3(C)C)nc2)=O)C1 57078,C(=O)(C(C)(C)C(=O)NCC(C)(O)CCO)NCC1CCC1C(=O)OC 57079,c1(N2C(C)CCN(C(CCn3c(C)csc3=O)=O)CC2)ncc2c(ncn2C)n1 57080,N1(C(=O)N)CC2C(CNC3CC(C(C(=O)C(=O)CN4CC5CC5C4)F)C3)C2C1.CO 57081,c1(C(N2C3(CCC(C(=O)NCC)C2)COC3)=O)[nH]c2cc(OC)ccc2c1C 57082,c1(C(C2CC(=C)C2)NC(C)(C)CNS(C)(=O)=O)nnnn1CCCCCC 57083,Cc1[nH]c2ccccc2c1C(=O)NC(C)CN(C(=O)CC1CC(F)C1)C 57084,C1(C)(C(N2CC(C)N(C(=O)C(=O)N(C)C)CCC2)=O)CCc2ccccc2C1 57085,C(=O)(C1CCCn2cncc21)Oc1c(OC)cccc1 57086,Cc1ccc(C(=O)NC2CCN(C(=O)Cc3ncoc3C)C(C)C2)cc1CO 57087,CC(C(C)(C)C(=O)NC12CC(F)(C1)C2)NC(=O)CCCC1CCC1 57088,Cc1cc2[nH]c(C(N3CC(O)(CNC(=O)Cc4ccc(O)nc4)C3)=O)cc2o1 57089,c1(CC=C)c(SCCS(=O)Cc2ccc(COC)cc2)nc2ccccc2c1C 57090,C(CCCCNC(c1cnn(CC(F)(F)F)c1)=O)NC(=O)Cc1cncnc1 57091,C1(C)(NC(c2ccc(C(=O)OC)cn2)c2n(C(CC)(C)C)nnn2)CC2(CC2)C1 57092,c1(C(=O)NC2CCC(NC(Cc3cc(C)ns3)=O)C2)ccc(-n2cncn2)cc1 57093,CCCC(CC)CC(=O)N(C1CCN(C(C23CCC(N=[N+]=[N-])C2C3)=O)CC1)CC 57094,c1(CNC(CC(CCC)O)=O)cccc2c1CN(C(c1sc(CO)nc1C)=O)C2 57095,c1(CCCC(=O)NCCN(C(C2C(C=C)C2)=O)C)ccccc1Br 57096,Cc1nn(C)c(Br)c1C(N1CCCC(CCNC(=O)CCOC2CC2)C1)=O 57097,C(=O)(CCCC(C)(C)CC)NCC(C(=O)NC1C2(CC(C(=O)OC)C2)C1)C(C)(C)C 57098,C1(NC(C2CC(=O)NC2)=O)C2CC1CN(C(C1CCN(CCF)CC1)=O)C2 57099,c1(C(=O)NCC2OCCN(C(c3[nH]cc(C(C)=O)c3)=O)C2)nccc(Cl)c1Cl 57100,c1(CC)cc(C(=O)N(CC(O)CNC(=O)CN2CC(=O)NC2=O)C)ccc1C 57101,C1(NC(=O)COC2CC(F)(F)C2)CCN(C(c2csc(O)n2)=O)CCC1CO 57102,N1(C(c2c(CC)scc2)=O)CCC(O)(CNC(=O)CCCN2CCCCC2)C1 57103,O=C(C1=CC2(CCOC2)C1)NCc1ccc(N2CCNCC2=O)cc1 57104,C1(NC(C2(OCC)CCSCC2)=O)CN(C(=O)CSc2cnn(C)c2)CCC1F 57105,C1(C)(C(N(CC(C)SC)C)=O)CCCN1C(c1sccc1CO)=O 57106,n1(CCC(N2CCOCC2C(C)C)=O)ncc(C(=O)OC)c1C 57107,CC(C)CCCC(C)NC(C1(NC(c2ccc(Cl)o2)=O)CC1(C)C)=O 57108,C1(CNC(C(C)OCCC(C)C)=O)(CNC(=O)C(N)=O)CC1(F)F 57109,CCCCCCCC(=O)N1C2CCC(C2)C1CNC(C1CCCS(=O)(=O)C1)=O 57110,CCCCCCCCC(C)NC(=O)NCC1CSCCO1 57111,C=C(C)CC(C(=O)N1CCC2(CC2C(=O)NCCCc2ccccn2)C1)OC 57112,C(CS(=O)(=O)CC(=O)NC1C2CC1N(C(C1CCc3nc[nH]c3C1)=O)C2C)OC 57113,c1(N(CCC(=O)NCCNC(=O)CN(C2CCC2)C)C(C)=O)ccccc1F 57114,c1(Nc2ccc(C(=O)OCCOCC(F)F)nc2)ccc(Br)nc1 57115,C1(CC(=O)NCC(CNC(c2c(C(=O)OC)csc2)=O)CO)CC=CCN1C 57116,CCC(C(=O)NCC1(C)CC(NC(=O)CCCc2cccs2)C1)C(C)C 57117,c1(OC)ccnc(F)c1C(N1CC(CNC(=O)C(C)SC(F)(F)F)(OC)C1)=O 57118,N1(C(c2c(COC)ccs2)=O)CCN(C(=O)C(F)C(C)(C)O)CC12CCC2 57119,CCC(CCCO)NC(=O)CCSc1cccc(OC)c1 57120,CCC(CC)(CO)C(=O)NCC1CCC2(CN(C(c3ccnc(C)c3O)=O)C2)O1 57121,N1(C(C(C)OCCOCC)=O)CC2(CCN(C(=O)C(C)n3cncn3)C2)C1 57122,Cc1cc(C(=O)NCC(=O)NC2CCC2CNC(=O)C(C)(C)CF)c(C)o1 57123,c1(C(=O)NC2C(CNC(C3CCC(C)O3)=O)CCC2)cnc2ccccn12 57124,c1(C(=O)NC(C(C)(C)NC(C(C)NC(C)=O)=O)C)c[nH]c2ccc(F)cc2c1=O 57125,N1(C(C=C(CCC)CCC)=O)CC2CN(C(=O)C=CCO)CCC2(CO)C1 57126,C(=O)(CC1=NNC(=O)C1)NC1CN(C(c2cc(C)nc(Cl)c2)=O)CC1C 57127,C1(NC(CN(S(CC)(=O)=O)C)=O)CCN(C(C2CC2C2(C)COC2)=O)C(C)C1 57128,N1(CC(=O)NCCOCCCN(C)C(C2C3CC(=O)CC23)=O)C(=O)CCCC1=O 57129,C(=O)(C(C)S(C)(=O)=O)NC1(CCCC(=O)Nc2cccc(C(C)C)c2)CCC1 57130,C1(C(C)(C)NC(C(C)OC)=O)CCN(C(=O)CC(C)(C)C)CC1 57131,N1(C(C(CCC)F)=O)CCC(C)CC1CNC(c1ccc(OC)nn1)=O 57132,N1(C(CCCSC(C)(C)C)=O)CCCC2(CNC(c3ccc([N+](=O)[O-])o3)=O)CC12 57133,N1(C(C(COC)O)=O)CCC12CN(C(=O)CC1(C)CCOCC1)C2 57134,c1(OCCN(C)C)c(Cl)cc(C(=O)NCC23CC(CCO2)C3)cc1Cl 57135,CS(=O)(=O)CCC(=O)NCC(C1CCOC1)NC(c1cocn1)=O 57136,C(N=c1cc(NCC2CC3CCC3C2)nc[nH]1)C1(COC)CCC1 57137,n1(CCC(N2C(C(C)NC(C(C)C(C)(C)C)=O)CCC2)=O)cnc2ccccc12 57138,CCC(C)CCC(=O)NC(Cn1cccn1)C(=O)NCc1cscc1C 57139,N(C(=NCCC(=O)NC)NCC1CC=CCO1)CC(CC)(C)OC 57140,c1(CC)cccc(C(N2CCC(C(C)(C)NC(C3SCC=C3C)=O)CC2)=O)n1 57141,C12(C(=O)NCC3CCN(C(C(CC)c4cccnc4)=O)C3)CC(CN1C1CC1)C2 57142,C(=O)(CC(C)(C)CN(C)C)N1CC(OCC)C(NC(=O)CSc2nncs2)C1 57143,C1(N(C(C(CC)C)C(=O)O)C2CC2)CCc2nc(-c3ccccc3)ncc2C1 57144,n1(CC(=O)NCCC(C)NC(=O)CC2CCC23CCC3)nc2ccccn2c1=O 57145,Cc1cc(C(=O)NCC(CC(C)C)NC(c2cc3sccc3[nH]2)=O)nc(C)n1 57146,Cc1n[nH]c(C)c1C(N)=O.C12CCCN(C1)Cc1c(con1)CNc1cn2nn1 57147,CCCCC(O)C(C)C(=O)NC(C)CN(C)C(c1ncc[nH]c1=O)=O 57148,C1(C2CN(C(COC(CC)CC)=O)C2)CN(C(=O)CCn2cccn2)CCO1 57149,n1(C(C(=O)N(C(CNC(c2c(CC)n[nH]c2)=O)C)C)C)cnc(C#N)n1 57150,C(=O)(C(C#N)CCc1ccccc1)NCCOCc1c(C)cccc1 57151,CC1CC=C(C(=O)N2CC(CC=O)CC2(C)C)CC1.N1CCN(CC(N)=O)CC1 57152,C1(CNC(CC#N)=O)CCC2(CO1)CC(NC(=O)CCC1CCCCCC1)C2 57153,Cc1[nH]nc2c1CC(C(N1CC(C(N)=O)(CNC(C3COC(=O)N3)=O)C1)=O)CC2 57154,N1(C(C(C)NC(c2ccoc2)=O)=O)CC2(CC(NC(c3cnccn3)=O)CO2)C1 57155,Cn1nc(C(=O)NCCCCCC(=O)NCCc2csnn2)cc1C#N 57156,c1(C(=O)NC2C3CC(CNC(COCCC)=O)(C3)OC2)c[nH]c2cccc(C)c12 57157,C12(CCCCC1)CC(=O)N2.N1(C(C)=O)CCCOC1CNC(=O)CC(C)C 57158,c1(C(=O)NCCCN(C(CC2(CSC)CC2)=O)C)cc(C#N)ccc1C 57159,Cc1ccc(Sc2ccccc2CNCCC2CNCCO2)c(C)c1 57160,N1(C(C2(C(C)C)COC2)=O)CCC(NC(=O)C(N2CCN(C)CC2)C)C(C)(C)C1 57161,Cc1cc(C(=O)NC2CC(CCNC(=O)COc3ccsn3)C2)c(N)c(F)c1 57162,c1(C(=O)NC(c2ccccc2)CNC(=O)CC2(O)CCC2)cnn(C2CCC2)n1 57163,N1(C(CC2CCCC(OC)C2)=O)C2CCC1CC(CNC(c1ccc(Cl)s1)=O)C2 57164,O=C(N=c1[nH]nco1)c1ccc(C(=O)NCc2cc(Cl)nc(Cl)c2)cc1 57165,CN1CCC(O)(CC(N2CCN(C(=O)Cc3nccs3)C(CCO)C2)=O)CC1 57166,C1(C)(COC)CCCN(C(C2CCN(C(c3cc(C)c(C)[nH]3)=O)CC2)=O)C1 57167,N1(C(C2C(CC)OCCC2)=O)CC2(C1)CN(C(c1csnc1OC)=O)C2 57168,Cc1cccc2c1OCC2C(=O)N(CC(C)O)CCNC(=O)C=Cc1ccco1 57169,C1(C(N2CC3C(N(C(=O)COC4CCC(C)CC4)C)C3C2)=O)(CC)CCOCC1 57170,C12(CC(N3CC4C(CNC(c5cc(COC)on5)=O)C4C3)=O)CCC(CC1)CC2 57171,Cc1cc(NC(C2COCC2NC(=O)COc2ccccc2)=O)cc(C)c1F 57172,CCC(CCOC)C(=O)N1CCCCC1CCCNC(=O)C=C1CC1 57173,C(CNC(=O)CN(C)C1CC1)(C(=O)NCC(O)CCNC(C)=O)OC 57174,N1(C(c2c(C)cns2)=O)CC(C)N(C(c2nc(N)cc3ccccc23)=O)CC1C 57175,C1(CNC(c2cccc(CO)c2)=O)C2CCC(C2)N1C(=O)CC1(O)CCC1 57176,Cc1cc(C)c(NC(=O)CNC(c2cnnn2C(C)C)=O)cc1O 57177,CCC(C)C(=O)C(=O)NCc1cc(C(N2CCCCC2C(N)=O)=O)no1 57178,C(=O)(CCCC(=O)NC(C(=O)NC1CCCCC12CC2)C1CCCO1)OC 57179,c1(C(N(C(C)CC(=O)NCCCCC2CC2C)C)=O)cc(F)ccc1F 57180,C(CCC(C(=O)OC(=O)CC1CCOCC1C)NC(=O)C(C)C)OC 57181,c1(CN(CC(C)NC(c2nc(OCC)sn2)=O)C)c(Cl)oc2ccccc12 57182,C(=O)(C#CC(C)(C)C)NCC(c1ccc(C)cc1)NC(C(CC)OC)=O 57183,c1(C(=O)NCCNC(C(C)C(C)C(C)(C)C)=O)cc([N+](=O)[O-])ccc1Cl 57184,C1(OC)CN(C(=O)C=CC2CCCN2C(=O)Cc2ncn(C)c2C)CC12CC2 57185,CC(C)C(F)C(=O)NC1CCN(C(C)C(N2CCCC(C)C2)=O)CC1 57186,c1(C(=O)NC2C(NC(CCC)=O)C2)cccc(N)n1 57187,c1(C(=O)NC(CNC(CN(CC)CC)=O)C)csc(-c2ncccc2C)n1 57188,c1(NC(C)=O)cccc(CCNC(=O)COCC)c1.N12CC(C(C)C1)OCC2=O 57189,C1(C(N2CCC(COC)(NC(=O)CCC(F)F)C2)=O)OC(C)(C)OC1(C)C 57190,CCC(C)CC(C)C(=O)N1CC2CC(C1)N(C(C1OCC1(C)C)=O)C2 57191,CC(C)C(C(=O)NCC1CC(C)(C)CO1)C(C)NC(=O)Cc1ccon1 57192,N1(Cc2ccc(CC)s2)CC2(CCN2C(=O)CCc2c(C)noc2C)C1 57193,c1(CN(C(C(CSCC)NC(C2CSC2)=O)=O)C)ccccc1O 57194,Cc1n[nH]c(C)c1CCC(=O)NC1(CNC(c2c(C(C)C)cnn2C)=O)CCC1 57195,CC1(C)COC(CC(=O)NC2CC(NC3(c4ccn(COCC#N)n4)CC3)C2)C1 57196,C1(C(=O)NC(c2c(C)nccc2)C)CCCN(C(c2cc(O)n(C)n2)=O)C1C 57197,c1(C(=O)OC)ccc(CC(=O)NC(C)CCNC(C2CC(OC)C2)C)cc1F 57198,c1(C(N2CCCC(CCCCNC(CC=C=C)=O)C2)=O)c(OC)cccc1Cl 57199,CC1=C(C(=O)NCC2CC(NC(c3ccc(Cl)c(Cl)c3)=O)C2)CCCC1 57200,c1(C(N2CCC(CCNC(c3cc(C(N)=O)no3)=O)C2)C)ccccc1Br 57201,C1(NC(C2C(=C)C2)=O)CC2(CCCCN2C(=O)CCc2ccccc2C(N)=O)C1 57202,N1(C(C2CN(C(C)C)C2)=O)CCCC(O)(CNC(c2cnc(C(F)(F)F)s2)=O)C1 57203,c1(CC(N2CCC(CN(CC(O)COC)CC)CC2)=O)cn2ccccc2n1 57204,CCCCC(C(=O)OC)NCC1CN(C(=O)OC(C)(C)C)C(C)(C)C1 57205,c1(CNC(COC)=O)oc2ccccc2c1CNC(=O)CCC(C)(C)F 57206,C12(C(=O)NCC3CC(C)N(C(c4ccnc(O)c4)=O)C3)CCCC1CCC2 57207,c1(C(c2n(C(CC)C)nnn2)NCCOc2cccc(C)c2)cc(Cl)c(Br)cn1 57208,N(C1COc2cc(Cl)ccc21)C(C(C)Nc1cc(C(C)(C)C)ncn1)=O 57209,N1(C(Cc2c(C)cco2)=O)CCC(NC(c2ccccc2CC2CCC2)=O)CC1 57210,C1(n2cc(COC)nn2)(C(=O)NC(C)COCc2ccccc2)CCOCC1 57211,C(=O)(C(C)C(=O)NC1CCCCCC1C(N1CCCC(CO)C1C)=O)OC 57212,c1(CNC(c2n(C(CC)C)nnn2)CCCc2ccccc2)ccc(F)cc1Br 57213,c1(-c2c(COC)cccc2)c(C(=O)N(C)OC)nn2c1CCCC2 57214,c1(CC)cn2cc(C(N3CCC(N(C(=O)COC(F)(F)F)C)C3)=O)cc(F)c2n1 57215,C1(C(=O)NCC(CCNC(C(C)c2ncco2)=O)O)CCCCCC1 57216,C1(C(=O)NCC(CN(C)C(c2cscc2S(C)(=O)=O)=O)O)CCCCC12CCC2 57217,C1(CC(=O)NCC(CC)(C)NC(C2CCN(C(C)=O)CC2)=O)COCCOC1 57218,C1(c2nnnn2CCCF)(N(CC2(SC)CC2)Cc2ccccc2F)CCSCC1 57219,CC1(C(=O)NCC2(NC(=O)Cc3cccc(C(F)F)c3)CCC2)CCCCCC1 57220,N1(C(c2sc(C=O)c(Br)c2Br)=O)CCC2(CC1)CC(NCc1ccncc1)CO2 57221,c1(OC)ccc(COC(C)C(=O)Nc2noc(C(C)C)n2)cc1 57222,C(C(C(=O)NCCCNC(C)=O)C(C)C)NC(C(C)=C(CC)C)=O 57223,C1(NC(c2c(CCC)occ2)=O)C2CCN(C(c3cc(O)nn3C)=O)C12 57224,c1(NC(CCN(C(=O)CCOC2COC2)C)=O)cncc(C(F)F)c1 57225,C(=O)(C(F)CC(C)(C)NC(c1ccc(C(=O)OC)o1)=O)NC(CC)C1CCC1 57226,C1(F)(CNC(C(=O)NCC)=O)CCC(NC(=O)C=C(C)Cl)C1 57227,N1(C(c2cc(CC)c(F)cc2)=O)CC(C)N(C(=O)CC(F)(F)CC)CC1C 57228,N1(C(C2CCC(c3cc[nH]n3)O2)=O)CCN(C(=O)C(O)C2CC2)C(C2CC2)C1 57229,C(=O)(C(CCc1ccccc1F)N1CCCC1CC)NCC(=C)C 57230,C=C(C)C(C)(O)C(=O)NC1CCC(NC(c2ccc(CNC(C)=O)cc2)=O)CC1 57231,C1(C(=O)NCc2c(C)ccc(C)c2)CC2CCCCC2N1C(c1cocn1)=O 57232,C1(C(N2CCCC(CNC(C(C)C3CCOC3)=O)C2)=O)CCCCC12OCCO2 57233,C1(NC(C2CC(NCC)C2)=O)(CO)CCN(C(=O)C(O)Cc2cnn(C)c2)CC1 57234,C1(OC)CC(C(N2CC(C(C)C)C2)=O)N(C(=O)Cc2ccns2)C1 57235,c1(C(=O)NCC(CC)NC(C2(C)C=CCCC2)=O)cc2n(n1)CC1(CC1)C2 57236,C(=O)(C(C)(CC)C(F)F)N(C)Cc1ccccc1CNC(c1nn(C)cc1Cl)=O 57237,N1(C(C(CCCCC)O)=O)CC2(CCCCN2C(C23CC(C)(C2)OC3(C)C)=O)C1 57238,c1(C(CC)(C)C)nnc(N2CCC(CCN3CCCCC3)CC2)n1CC 57239,C1(F)(C(=O)NC2CC(CNC(C3CC=CC3)=O)CC2O)CS(=O)(=O)CC12CCC2 57240,N1(C(C2(CNC(CC(C)n3cccc3)=O)CC2)=O)CCC(C2(C)CC2)CC1 57241,c1(C(=O)NCC2CCN(C(C3(C)C(C)C3)=O)C2)ccc2oc(O)nc2c1 57242,C=CCCC(O)CNC(c1coc(CO)c1)=O.C12(CC(C)(C)C1)C(=O)NC2 57243,Cc1cc(Br)c(C(=O)Nc2ccc(C)c(C(C)(C)C)c2)cc1Cl 57244,C1(C(=O)NCC(=O)NC(=O)C2CC2)C2CC3C(C2NC(=O)C2=CCCCO2)C13 57245,c1(NC(C23CC2CN(S(=O)(=O)CCN2CCOCC2)C3)=O)cc(F)ccn1 57246,Cc1ccc(O)cc1NC(C1CN(C)CCO1)=O.C1(Cc2cccs2)CC(=O)N1 57247,c1(CCC(=O)NC(C2CCN(C(C)=O)CC2)C)cccc(C#N)c1 57248,C(=O)(C1CCc2c[nH]nc21)N1CCC(CNC(C2N(C=O)CCOC2)=O)C1 57249,CCC(C)(CC(=O)Nc1cnn(CC2CCC2)c1)NC(=O)COCC(C)C 57250,c1(C(=O)NCC2CN(C(C#CC(C)C)=O)C(C)CC2)cccc2c1OCCC2 57251,CC1(C)CN(C(=O)NC(c2cccc(C(F)(F)F)c2)=O)Cc2c1n[nH]c2C(F)F 57252,C1(O)(C(C)CNC(=O)Cc2cnns2)CCN(Cc2cc(-c3ccoc3)[nH]n2)C1 57253,C1(S(C)(=O)=O)(C(N(CC(CC)NC(C2CCN(C)C2C)=O)C)=O)CCC1 57254,C1(C(=O)NCCCCC=C)CCC2CCC1N2C(c1cnn2c1CCC2)=O 57255,Cc1ccc(NC(=O)CNC(c2cocc2Br)c2nnnn2C)cc1O 57256,C(=O)(CCC=CC(C)C)NCC(CN(C(C1(CCOC)CCC1)=O)C)O 57257,c1(OC(C)C)ccccc1C(=O)NCCC(C)NC(C1CCCN1C(C)C)=O 57258,N1(C(=O)COc2ccc(Cl)c(Cl)c2)CCC2(CC1)CN(C(C1C=CCC1)=O)C2 57259,c1(C(=O)NCC(C)CNC(=O)CC2CC23CC3)c[nH]c(C(N)=O)c1 57260,C1(N(C(=O)C(C)n2cccn2)CC)CCCN(C(c2ccc(CO)cc2)=O)C1 57261,C1(N(C(CC(C)OC)=O)CC)CCC(NC(c2ccc(=O)oc2)=O)CC1 57262,c1(C(N(C(CNC(C(CC)C(C)C)=O)C2CC2)C)=O)cc(S(C)(=O)=O)co1 57263,C1(CN(C(=O)COC2(C)CCC2)C)CCCN(C(C2CCC(C(F)F)CC2)=O)C1 57264,C(=O)(CCCC(CC)NC(=O)CC(C)F)N(CC#C)CCOC 57265,CCC(F)(C(=O)OC)C(=O)N1CC2CC(N(C)C(c3ccccn3)=O)C1C2 57266,N1(C(Cc2c(C)n[nH]c2)=O)CCC2(CCN(C(=O)CN(C)C(=O)C3CC3)CC2)C1 57267,N1(C(C2CCC(CC)O2)=O)Cc2[nH]nc(C(N3Cc4c[nH]nc4C3)=O)c2C1 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57303,C(CC(O)CNC(c1cn(C2CCC2)nn1)=O)NC(=O)Cc1cscn1 57304,Cc1scc(C(=O)NC2CC3C(NC(=O)CC4CCCCC4O)C3C2)c1C 57305,N#CC1CCC(CC(=O)N(CCC(=O)N2CCC2CF)CCO)C1 57306,C1(C(=O)NCc2ccn(C(C)C)n2)CC12CCN(C(=O)C(C)Cn1cccn1)C2 57307,C(c1cn(C)c(=O)n(C)c1=O)=CC(N1CC(NC(c2c(C)ccs2)=O)C(C)C1)=O 57308,c1(CNC(=O)NCC2(c3ccc(Cl)cc3)CCCC2)cccc(F)c1O 57309,C(N=c1[nH]c(=NC(C)CC2CCCO2)[nH]c2c1CCC2)c1c(CCOC)c[nH]n1 57310,c1(C(=O)NC(c2nc(C3CC3)no2)C)cc2n(c1)CCS(=O)(=O)C2 57311,CC(C)(CNC(C1CCC2(CCC2)C1)=O)CC(=O)NC(C)(C)C(C)(C)C 57312,N1(C(c2ccc(CO)cc2)=O)CC2CCN(C(c3cc(Cl)c(O)cc3F)=O)C2C1 57313,CC(C(=O)N1CC(N(C)C(c2coc(C3CCC3)n2)=O)C(C)(C)C1)S(C)(=O)=O 57314,Cc1nc2sccn2c1C(=O)NCC(F)CNC(=O)COCC(C)(C)C 57315,c1(C(=O)NC2C3(CN(C(C(CCCC)CC)=O)C3)CC2)cc2c(C)cccc2o1 57316,C(=O)(C(C)S(N)(=O)=O)NCCn1ncc(C(=O)NC(COC(C)C)(C)C)c1 57317,O=C(CN=c1cc[nH]cc1)NC1(C(=O)NCCCC2CCOC2)CC(CO)C1 57318,C1(NC(=O)C(CO)c2ccccc2)CCCCCN(C(c2nccc(Cl)c2F)=O)C1 57319,C1(C(C2CC2)OC(=O)NC(c2ccc(F)cc2)COC)CCC=CCCC1 57320,CC(C)(C)C(O)CC(=O)N1CCC2(CC1)CC2NC(=O)OC(C)(C)C 57321,c1(C(N2CCC(CC)C2)=O)cccc(CN(c2cn(C)cn2)C)c1 57322,C(=O)(C1CNC(=O)c2ccccc21)N1CCCCC(CNC(C2(C#C)CC2)=O)C1 57323,c1(CN2CCC(CC(=O)NCc3cc(F)cc(I)c3)C2)cc2n(n1)CCC2 57324,c1(CC)occc1C(=O)NC1COCC1C(=O)NCC(CO)C1CC1 57325,N1(C(CCC(C)C)=O)CC2(CC(NC(=O)CC3CCOCC3(C)C)CO2)C1 57326,N1(C(COC(C)=O)=O)CCC2(CC1)CC(C)N(C(=O)C=Cc1ccccn1)C2 57327,c1(C(N2CCC(C)(NC(C3C(COC)C3)=O)C2)=O)ccc2[nH]c(=N)sc2c1 57328,C1(C)(CNC(c2cc(COC)[nH]n2)=O)CCN(C(c2snnc2C)=O)C1 57329,Cc1cc(C(=O)N(CC(O)CNC(=O)C=CC2(C)COC2)C)ns1 57330,C1(OC)CCC12CC(C(=O)NC1CCCC1(C)CN(C(=O)Cc1ccno1)C)C2 57331,N1(C(CCS(N)(=O)=O)=O)CCCCC12CC(NC(=O)C(=Cc1cccnc1)F)C2 57332,c1(CC(=O)NC(CC2CCCC2)C(=O)NCc2cnc(Cl)s2)cncnc1O 57333,N1(C(CNC(=O)OC)=O)CC(CCNC(=O)C=C2CCN(C)C2)C(C)C1 57334,c1(CCC(=O)NCC2C(CNC(c3cc(C(=O)OC)on3)=O)C2)cn(C)nc1C 57335,Cc1cc(C(=O)NCC2(F)COCCOC2)c(C)nc1C 57336,N1(C(C2COCCN(C(c3cn(CC=C)nc3)=O)C2)=O)CCCN(C)C(=O)C1 57337,C1(NC(COCc2ncc(C)o2)=O)CN(C(C2CCOCC2)=O)CCC1F 57338,C=CC1(C(=O)N(C)CCOCCCNC(=O)CCS(C)=O)CCOCC1 57339,Cc1c(C(=O)NCCN(CC(C)O)C(C2C=CCC2)=O)cnc2ccccc12 57340,CC#CCC(C(=O)N1CC(N(C)CCO)C1)NC(=O)CC(=O)OCC 57341,c1(CC(N2CCC(C)C(NC(c3ccon3)=O)C2)=O)ccc2cccnc2c1 57342,N1(C(c2cccc(C)n2)=O)CCCC2(CNC(=O)CCC3CCCC3)CC12 57343,C1(C(=O)NCCCCNCCNC(C(C)OCC#C)=O)(OC(C)(C)C)CCCC1 57344,c1(NC(c2ccc(C(=O)OC)c(Br)c2)=O)c(F)cc(OC(F)F)cc1F 57345,c1(C(N(C2C(C)CC2)C)=O)coc2c1CN(C(=O)Cc1nccn1C)C2 57346,N1(C(C2CCC(C(N)=O)O2)=O)CCCC2(CCN(C(c3cccnc3F)=O)C2)C1 57347,C(=O)(CCCC(C)(C)C)NC1CC2(CC(NC(C(C)c3ccsc3)=O)C2)C1 57348,C1(C)(N(CC(=O)N)C)CCCN(C(=O)Cn2cnc([N+](=O)[O-])c2)C1.C(C1CC1)=C(C)C 57349,c1(C(=O)NCCSCCC=C)ccnc(CNC(=O)C(C)C2CCC2)c1 57350,C1(C(N2CCC(CN(C)C)CC2)=O)C2CCC(C2)N1C(C1CC2COCC2C1)=O 57351,c1(N(C)C)cncc(C(N2CC3CC2(CC2CC2)C3)=O)c1.C1(=O)C=CC(=O)N1 57352,c1(CC)sc(=N)[nH]c1C(=O)NCCN(C)C(c1cncc(C(F)F)c1)=O 57353,CC12CN(C(=O)COC(F)F)CC1CN(C(=O)Cn1cnc3c(N)ncnc13)C2 57354,c1(C(N2CC(C(C)NC(C3(CF)CCOCC3)=O)C2)=O)cccc2c1NCCC2 57355,C1(Cn2cc(CC=C)nn2)CCCC(C(=O)N(C(=O)C(F)(F)CC)CC)C1 57356,CC(C(=O)NCCC1CN(C(=O)CCN2CCN(C)CC2)CCCO1)C(C)(F)F 57357,C=C1CC2(C1)CC(C(=O)NC1CCN(C(=O)CC3CCC(F)(F)CC3)CC1C)C2 57358,C1(CC)CNC(=O)CN1C(=O)C(C)(C1CC1)N(C)C(c1cc[nH]c(=N)n1)=O 57359,c1(NC(C2CCN2Cc2cc(O)ncc2Br)=O)ncnc2occc12 57360,CCC(C)CC(=O)N(C1CC(NC(=O)CCOc2ccccc2F)C1)C 57361,c1(N2CC(CCNC(C(CCC)C)=O)(OC)C2)ccc([N+](=O)[O-])cc1C(C)=O 57362,N1(C(c2ncc[nH]2)=O)CCCC(C2CCN(C(C3(C(F)F)CCC3)=O)C2)C1 57363,CCCCCCC(=O)N(C)CC1CCN(C(C2(C(=O)OC)CC2)=O)CC1 57364,C1(OC)COC2(CCNC2)C1.c1(C(=O)OC)cc2c(OC)c(c1)N2 57365,C(C1CCC(C)CC1)=C(C(N1CCC(N(C(C2CCN(C)C2=O)=O)CC)C1)=O)C 57366,C1(C(N2CC(N3C(=O)CC(OC)C3)C2)=O)COc2cc(OC)ccc2C1 57367,C(=O)(CS(=O)(=O)C(C)C)N1CCCC(N(C(Cc2ccc(C)cc2)=O)CCO)C1 57368,C(=O)(C(C)(CC)C(N)=O)NC1C(CNC(c2c(CC)ccc(Cl)c2)=O)C1 57369,c1(C(N(CCCCCNC(c2n(CC)ncn2)=O)C(C)C)=O)occ2c1CCC2 57370,N1(C(c2c(C)nn[nH]2)=O)C2CCC1CN(C(C1CCOC(C(F)(F)F)C1)=O)C2 57371,C1(C(=O)OC)N(C(=O)C(C2CCCC2)NC(=O)CC2CCOC2(C)C)CC1(C)C 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57391,C(=O)(CC(C)(C)c1ccccc1)NCC(Cn1cc(C(C)OCC)nn1)(F)F 57392,C1(F)(C(=O)NCC(CC)(CC)OC)CCCN(C(c2ccc(C)o2)=O)C1 57393,C1(C(=O)NCC2C(NC(c3nnn(CC)c3C)=O)CCCC2)CC2CCC(C1)C2 57394,c1(-c2cccc(CNCC(CO)OCC)c2)cccc2nc(C(=O)NCC)cn12 57395,Cc1cnn(C)c1CCNC(=O)C(=O)NCC(C)(COCc1ccccc1)CO 57396,C1(C(=O)NCC2OCC(C(=O)NCc3c(CC)n[nH]c3)C2)CC(=O)NC(=O)C1 57397,C(c1cc(Br)ccc1OCC1=CCN(Cc2ccc(CC)cc2)CC1)=C.OC 57398,n1(CCC(=O)NC2C(NC(C3ON=C(CC)C3)=O)CCC2)cc(S(N)(=O)=O)cn1 57399,C1(S(=O)(=O)N(C)C)(CN(CCOCC)Cc2sccc2C)CC1 57400,n1(CC(=O)N(CC(C)NC(c2sccc2-n2cccc2)=O)C)cc(CO)nn1 57401,c1(N2C(C)CN(C(C34CCCCC3C4)=O)CC2)ccc2nnnn2n1 57402,C1(C)(CNC(CN(CCCC)C)=O)CCCN1C(=O)C(F)COCCN(C)C.CN 57403,c1(C(=O)NC(CNC(c2ccn(CCCC)n2)=O)C)cn(CC(F)F)nc1C 57404,N1(C(C2COC(C)C2)C(=O)NC(C(=O)OC)C)CCc2ccc(Cl)cc2C1C 57405,C(=O)(CC1=NN(c2ccccc2Cl)S(=O)C1)NC(c1ccccc1)CC 57406,C1(C(=O)NCCCCNC(Cn2cc(C(C)=O)nn2)=O)CC12CCSCC2 57407,N1(C(C(C(C)C)c2ccncc2)=O)CCCCC(N(C(=O)CC(F)(F)Cl)C)C1 57408,C(CCCC(=O)NC1CCC1(C)C)NC(C1(OC)CC1)=O 57409,O(NC(=O)C(CNC(=O)CCCCCSC)C(C)(C)C)CC(CC)C 57410,N1(C(c2cnnc(Cl)c2)=O)CCN(C(C2CCCC3CCCN23)=O)CC(O)C1 57411,c1(C(N)=O)cncc(CONCCN2CC3CCC2C3)c1 57412,C=CCC(CNC(c1ccc(CCC)s1)=O)NC(c1cscc1C1CC1)=O 57413,c1(C(N2CC(C(=O)NC(c3ccccc3)CO)(SC)C2)=O)cn2ccccc2n1 57414,N1(C(C2C(CCC)CN(C(c3conc3C)=O)C2)=O)CCN(C)C(=O)C1CC 57415,c1(C(=O)NC2C(NC(CC(=C)C)=O)CCC2)cn2cc(Br)cc(C)c2n1 57416,C(N=c1nc[nH]cc1C#N)C1CC(NC(CCc2ccc(C)s2)=O)C1 57417,C1(N(C(CCC#C)=O)C)CCCN(C(c2ccc(C3CCOCC3)cc2)=O)C1 57418,CS(=O)(=NCC(=O)NCC1CCN1C(=O)Cn1ncccc1=O)c1ccccc1F 57419,N1(c2nccc(N3C4CC(C)CC3CC4)n2)CC2(CCCCN2C)C1 57420,c1(OCCNC(c2cnsn2)C)ccccc1F 57421,c1(C(=O)Nc2ccc(C(N(C(CC)C)CC)=O)cc2)cc(=N)[nH]c(F)n1 57422,CC1CC2(CO1)CN(C(=O)CC(C1CC1)NC(C1CC1C(N)=O)=O)C2 57423,C=CCC(CNC(C1CC1(C)C(F)(F)F)=O)NC(=O)C=CC(C)(C)C 57424,N1(c2cc(C)[nH]n2)CCCN(C(=O)CC23CCCC2C3)CC1 57425,N1(C(C2CCN(C(C=CCCC)=O)CC2C)=O)CC2CCC(C1)N2C(C)C 57426,c1(C(=O)NCC(C)(C)NC(CC(C)C2CC2)=O)n[nH]c(C(C)C)c1[N+](=O)[O-] 57427,c12ccc(cc1)NC(=O)C2C1CC1.c1(SC2CN(C(CC)CO)C2)ccccc1 57428,c1(C(N(CCC(=O)NCC2C(OC)CCC2)C(C)C)=O)csc(C)c1C 57429,c1(CC)cc(C(N2CC(CCNC(=O)C(C)OCC3CCCO3)C2)=O)cc(N)c1 57430,C(=O)(CC1=CCOCC1)N1C(C(=O)NC(c2nn[nH]n2)CC)CC(F)CC1 57431,CC1(C)CCCN(C(=O)CCC2CCCCCC2)C1CNC(c1n[nH]cc1F)=O 57432,c1(OC)ccc(C(=O)NCCC2(C)CCOC2)c(C)c1OC 57433,C1(CC(N2CCC(CN(C(=O)Cn3ncnn3)C)C2)=O)CCn2cncc2C1 57434,N1(C(C2C(NC(C(C)C(F)(F)F)=O)CCC2)=O)Cc2n[nH]cc2C1CO 57435,CN1CCC(CC(C(=O)O)NC(C2CCCC2CF)=O)CC1 57436,C1(NC(c2nc(COCC)sc2)=O)CC2CCC1N2C(c1cn(C)ccc1=O)=O 57437,C#CCCCCC(=O)N1CC(N(C(=O)COCCCC)C)C(C)(C)C1 57438,N1(C(c2ccc(C(=O)OC)o2)=O)CC2CCC2(CCNC(=O)C=C(C)C)C1 57439,C(=O)(CS(=O)(=O)C1CC1)N(CCCCCNC(c1ncn2c1CCC2)=O)C 57440,c1(CC(=O)NCCC(C)CCO)cc(F)c(Cl)cc1[N+](=O)[O-] 57441,CC1=C(C(=O)NC2CCCC2NC(=O)CC2CC=CCN2C)CCC1 57442,Nc1ccc(C(N2CCN(CC3(NC(C4CCCCC4F)=O)CC3)CC2)=O)cc1O 57443,C1(NC(CS(CC)=O)=O)CN(C(=O)C=Cc2ccoc2)C2(CCOCC2)C1 57444,S(=O)(=O)(c1ccc2c(c1)OCO2)N1C2CN(C(c3nn(C)c(Cl)c3)=O)CC1C2 57445,c1(C(=O)NCC(CC)NC(C2CCCCC2(C)C)=O)cccc(S(=O)(=O)CC)c1 57446,N1(c2snc(C(=O)OC)n2)C2CCC1C(CNC(=O)C(c1cscn1)N(C)C)C2 57447,c1(CC(=O)NCC(F)CNC(c2cc(F)n[nH]2)=O)nccc2ccccc12 57448,CC(C)C(C(=O)NCC1(CNC(c2cc(C#N)cs2)=O)CC12CCC2)N(C)C 57449,C1(C#CC(=O)NCc2ccc(C(=O)NC(C)CCOC)nc2)(CC)COC1 57450,c1(NC(c2ccccn2)COC)ccc(S(=O)(=O)NCCCC(F)(F)F)c(Cl)c1 57451,c1(C(=O)NC2(CO)CCN(C(CC(CC)(C)C)=O)C2)cc2cccnc2nc1O 57452,C1(CC(=O)NC2C(NC(c3c(OC)c(C)sc3)=O)C2)CCCCC12CC2 57453,Cc1[nH]c(C(C)(C)C)cc1C(=O)NCCC(C)NC(=O)CC(C)CF 57454,c1(C(CNC(C(C)CC2CC2)=O)NC(C2(C)CC2)=O)cccc(Cl)c1Cl 57455,CC1OC(C)C(C(N2CCN(C(=O)CC3(C)CC3(Cl)Cl)C(CCO)C2)=O)C1C 57456,C(CS(=O)(=O)CC(=O)NCc1cc(C(=O)N(CCC(C)(C)O)C)co1)OC 57457,c1(C(=O)NCC2(OC)CN(C(c3cc(N)ccc3Cl)=O)C2)cc2cccnc2s1 57458,N1(CCC)CCCCC1C(N1CCC(CF)(NC(c2nc(O)sc2C)=O)C1)=O 57459,c1(C(N(C(C(CC)C)C(=O)N(C2CCCOC2)C)C)=O)c[nH]c2cccnc12 57460,N1(C(c2cc(CCCCC)[nH]n2)=O)CCCC(NC(C2(C)CCOCC2)=O)C1 57461,N1(C(C2C(COC)C2)=O)CCC(C(C)(C)NC(=O)C(=CC2CCCC2)C)C1 57462,CC(F)(F)C(C)(C)CC(=O)C1=CNN=C2C(C(=O)NCCN2CC2CC2)CC1 57463,C1(CNC(CCC)=O)CC2COCC2N1C(c1cccc(C#N)c1)=O 57464,NS(=O)(=O)c1ccc(C(N2CCC(F)C(NC(=O)CCc3cscn3)C2)=O)nc1 57465,C(=O)(C(F)(F)C(F)(F)F)N(C)CC1N(C(C2(CSC)CC2)=O)CCC1 57466,C(CS(=O)(=O)CC(=O)NC1COCCC1C(=O)NCc1cc(Cl)ccn1)OC 57467,c1(C(=O)NC2CCN(Cc3nccc(C)c3)CC2O)cc2cnccc2nc1C 57468,C1(CNC(c2ccc(COC)[nH]2)=O)CCN(C(=O)COCC2CCCO2)C12CC2 57469,C1(C(=O)NCC(C(N2CCC(NC(CC)=O)C2)=O)N(C)C)CCC2(CCC2)O1 57470,c1(CC(=O)NC2C3CN(C(C(C)(C)CO)=O)CC2C3)csc2c(F)cccc12 57471,N1(C(C2(CC)CN(C(=O)CC3CC=CCC3)C2)=O)CCC(C)(O)CC1 57472,O=C1CCC(CCC(N2CCCC2C2(NC(c3ccncn3)=O)CC2)=O)CN1 57473,N1(C(c2c(C)csc2)=O)CC2CC2(CNC(=O)CC2(C)CCOC2)C1 57474,c1(C(=O)NCC2CC(NC(C3C(=C)C3)=O)C(O)C2)ccn2c(C)cc(C)nc12 57475,C1(CCNC(c2c(C)con2)=O)CN(C(C2CC2(Cl)Cl)=O)CCO1 57476,N1(C(C(C=C)(C)C)=O)CCC(NC(c2oc(C)cc2C)=O)C(F)(F)CC1 57477,N1(C(CS(CC)(=O)=O)=O)CCC2CCN(C(C3(CO)CC4CCC3C4)=O)CC12 57478,N1(C(C(C=C)OC)=O)CCOCC(NC(C2CN(CC)C(=O)N2)=O)C1 57479,CC1(C)CCCN(C(c2cccc(C(F)F)c2)=O)C1CNC(=O)C1=CSCCO1 57480,N1(C(CCN(C(Cc2cccc(C#C)c2)=O)C2CC2)=O)CCOCC2(CC2)C1 57481,C1(C(=O)NC2C(NC(c3n[nH]c(C(C)C)c3Br)=O)C2)CCCCCN1C 57482,Cc1cc2[nH]nc(CNC(=O)NC(c3ccc(C#N)cc3)C)c2o1 57483,C(C(C)(O)CC(=O)NCc1c[nH]nc1C(=O)NC1CCCCC1)OC 57484,Cc1cc(=O)c(C(N2CCC(C(=O)NCC34CC(F)(C3)C4)(CO)C2)=O)c[nH]1 57485,c1(-c2ccc(OCC#C)cc2)cccc2sc(CC(=O)N=c3nc(C)[nH]s3)cc12 57486,C(=O)(C(=O)N1CC(OCC(F)F)C1)NCCOC.C1C(C)N1 57487,C1(CC)(OC)CCOCC1.C12CN(CC1C(C)C)C(=O)C1CC(C#N)(C1)NC2=O 57488,n1(CC(=O)NC2CC3CN(C(Cc4nnc(C)o4)=O)C2C3)c(C)cc2ccccc12 57489,CC1CCN(CC(=O)NC2CCCC2NC(=O)COCCc2ccccc2)C1 57490,Cc1c(Br)noc1C(N1CCC1CNC(c1cccn1C1CCCC1)=O)=O 57491,Cn1nc(CC(C(=O)O)NC(=O)CNc2cncs2)c(Cl)n1 57492,C12(C(N3CCN(C(C4(C#C)CC4)=O)CC3)=O)CC(c3ccccc3)(C1)C2F 57493,CCC(C)CCCC(=O)NCC(CNC(C1(CC(=O)OCC)CCC1)=O)CO 57494,Cc1csc(C(N(c2cccc(Br)c2)CCCOC(C)C)=O)c1Cl 57495,CCC(CNC(C1CCN1C(=O)CN1CCOC1=O)=O)C(C)C 57496,c1(NC2CCCC(NC(=O)OC(C)(C)C)C2)ccc(Br)c(F)c1F 57497,C(CC(=O)N(CC(=O)N(C(CO)C1CC1)C)C(C)C)SC 57498,N1(C(C2(SC)CC2)=O)CCC2CC2(C(=O)NCC2CCCC3(CC3)C2)CC1 57499,C1(NC(C)=O)CN(C(c2csc(Cl)n2)=O)CC1c1cnn(C)c1 57500,c1(COC)nn(C)c(Cl)c1C(=O)NC(CCNC(C1CCC1(F)F)=O)CC(C)C 57501,N1(CC(=O)NC2CC(CNC(=O)OC(C)(C)C)C2)CCS(=O)CC1.CCCC1CO1 57502,C1(CC)(CNC(=O)CN2CCN(C)CC2)CCCN1C(=O)C(=Cc1cscn1)F 57503,C1(NC(c2cc(Cl)c[nH]2)=O)C2CN(C(C3(NC(=O)C4CC4)CCSCC3)=O)CC12 57504,C(C)(CO)(C(=O)NCCN1CCCC1)NC(c1ccc(C(C)=O)o1)=O 57505,CC1=CCC=CC1C(N1CC(C)(CC(=O)NCc2ncco2)C1)=O 57506,C1(CN)CCCCN(C(N(C(C2OCC2(C)C)=O)C)=O)C1.c1(C(C)=O)ccc(Br)cc1 57507,C1(CC(=O)N(C(C)COC)CC=C)CN(C(c2ccc(C#N)o2)=O)CCC1C 57508,N1(C(C(CCSC)OC)=O)CC2CCCN(C(c3cc4ccccn4n3)=O)C2C1 57509,C(=O)(C(C(C)C)C(C)C)N(C1CCN(C(=O)C(c2cncn2C)=O)C1)CC 57510,c1(CCC(=O)NC(C)Cc2ccccc2)ccc(OC(F)(F)F)cc1 57511,c1(CNC(c2c(C(C)C)ccs2)=O)ccnc(F)c1Cl.C12CCN(C1)C2 57512,C1(NC(c2cc(CCNC(c3ccn(C)c3)=O)on2)=O)C2CCCOC12 57513,C1(N(C(c2c(COC)ccs2)=O)C)CCCN(C(c2cc(C#N)on2)=O)C1 57514,C(=O)(C(F)(F)CCn1ccnn1)NCC(C)CN(C)C(c1cc(Cl)cn1C)=O 57515,Cc1cc(CNC(c2cnn3c2CCC3)c2nnnn2C2CCOC2)ccc1Br 57516,Cc1nc(C)c(C(C)NC(=O)C(C2CC2)NC(=O)CCC(C)N(C)C)[nH]1 57517,c1(C(N2CC3C(N(C(c4cc(COC)on4)=O)C)C3C2)=O)cc(O)cc(C#N)c1 57518,CC1(C)CN(C(=O)NCC2CCC3(C2)OCCO3)CC2(CCOC2)O1 57519,c1(NC(C2COCC2CNC(CC2(OC)CCOCC2)=O)=O)cc([N+](=O)[O-])c[nH]1 57520,c1(C(=O)NCCSCC(=O)NC2CC(C)(C)C2)ccc(C2CC2)nc1 57521,c1(CC(=O)NC2(c3cn(CCCC)nn3)CCC2)ccc(F)cc1C 57522,C#CCC(C)(CC)C(=O)NCC1(O)CN(C(c2cnn(C)c2Br)=O)C1 57523,C(=O)(C(C(CC)=Cc1cccnc1)N1CCCCC1C1(O)CC1)NCCCC 57524,C(C1=C(C)OCCS1(=O)=O)NC1(c2n(CCC)nnn2)CC(C2(C)CC=CCC2)C1 57525,N1(C(C(C(=C)Cl)(C)C)=O)CCCC(NC(=O)C2=C(C)OCC2)C(F)C1 57526,N1(C(c2c(C)nn(C)c2)=O)CCCC(O)(CN(C)C(c2ncn(C(C)C)n2)=O)C1 57527,C(=O)(CCCCCN(C)C)NC(C(C)C)C(C)NC(C1CCCCS1(=O)=O)=O 57528,c1(N2CCC(C(C)NC(=O)C(F)C(C)C)(CF)C2)ncc(S(C)(=O)=O)cc1Cl 57529,c1(C(N(C)CC2CCN(C(C(CC)SC)=O)C2)=O)cc(O)cc(F)c1 57530,CC1(CNC(C2(C)CC2(F)Cl)=O)CC(F)(F)CN1C(=O)CC#N 57531,C1(NC(Cc2c(C)ocn2)=O)CCN(C(C2(C#N)CCCCC2)=O)CC1CO 57532,c1(C(N2CCCC2C2(O)CNC2)=O)ccc(Cl)cc1Cn1ccnc1 57533,N1(C(CCOC)=O)CC2CC2(C(=O)NCc2ccccc2Oc2ccncc2)C1 57534,C(=O)(C(C)CC(=O)NCC(CO)NC(C1CN(C(C)=O)C1)=O)OC 57535,C1(C(=O)NCC(CCC)OC)CN(C)CCN1C(c1coc(C(F)F)c1)=O 57536,O=C1CCCC(C(=O)NCCCCC(=O)NC(CO)CCF)CC1 57537,N1(C2c3nc(oc3)NC2=O)CC(C)C(C)C1C.c1(N(C(C)=O)C)ccccc1 57538,CC1(CNC(C2C3COCC23)=O)COCCN(C(=O)C2=NOC(C(C)(C)C)C2)C1 57539,Cc1cnsc1C(=O)NCCC(O)CNC(C1C=CCCC1)=O 57540,C1(CCNC(C2CCOCC2)=O)CCN(C(=O)CC2CS(=O)(=O)C2)C1 57541,N1(C(COCCC)=O)CCN(C(=O)C(c2cccc([N+](=O)[O-])c2)C)CC(O)C1 57542,C1(C(=O)NC(CN(CC)CC)C)CCC2CCC1N2C(c1cncn(C)c1=O)=O 57543,C1(NC(c2nc(C(C)(C)C)oc2)=O)CC2CCCC(C1)N2C(=O)C(F)CC1CC1 57544,C1(CNC(c2ccc(CC(C)C)cc2)C)CC2(C1)CC(C#N)C2 57545,c1(OC)ccccc1CC(=O)Nc1ccsc1.C12CC1C(=O)N2 57546,C1(N(C(=O)C(C)(CO)N(C)C)CC)CCCCN(C(c2ccc(C)c(F)c2)=O)C1 57547,N1(C(CNS(N(C)C)(=O)=O)=O)CCC(C)(C)C(NC(=O)CC2CCC(F)(F)C2)C1 57548,N1(C(C(C)NC=O)=O)CCC(C(=O)NCC2CC(=O)C2)CC1 57549,c1(C(=O)NCC(=C)CCNC(=O)C=Cc2cnccn2)nncc2c1CCCC2 57550,C1(C(=O)NCC(C=C)O)(CNC(=O)CSCCOC)CCCC1 57551,C1(N(C(=O)Nc2c(C)cccc2)C)CCCN(C(C)C(N)=O)CC1 57552,C1(C(=O)NCC2(C)CCCN(C(CC3(C)CCC3)=O)C2)CNc2ccnn2C1 57553,Cc1cc(C(C)(C)C(N2CC3CC3C2CNC(=O)CC2CC2)=O)ccc1Br 57554,C(C)(CC(=O)O)(c1ccccc1)NCCS(=O)(=O)NC(C)C 57555,C(C)(Cc1cn(Cc2ccco2)nn1)(C(=O)O)NC(CCC1C(C)C1)=O.C1CCCC1 57556,N1(C(c2n(CCOC)nnc2)=O)CCC(NC(=O)NCCO)CC(C)(C)C1 57557,c1(C(=O)NC(C)CCCNC(C2CC2c2ccn(C)n2)=O)ccn2ncnc2c1 57558,n1(CCC(=O)NCC(CCOC)NC(=O)C(C)SC)ncc(=O)c2ccccc12 57559,N1(C(C(CNC(C2(OC)CC(C)C2)=O)N(C)C)=O)CCc2ccc(C#N)cc21 57560,C1(CC)CCN(C(c2coc(CNC(=O)C(C)Cn3cccn3)c2)=O)C1C 57561,C1(NC(=O)Cc2cscn2)CCC2(CCN(C(=O)C3=CC4(CCOC4)C3)C2)C1 57562,CCC(C)(C)CC(=O)N1CCC(CNC(c2cc(C)c(C(N)=O)cn2)=O)C(C)C1 57563,C1(NC(C(Cc2cn(C)nc2)O)=O)COCCN(C(=O)CN2CSCC2=O)C1 57564,c1(C(=O)NCC(CC)(C)C(=O)NCCn2ccccc2=O)cccc2ccnn12 57565,C(=O)(C(C)(C)c1ncco1)N1CC(CNC(C(C2CCC2)OC)=O)C1 57566,Cc1cc(C(C)C(=O)NC2CN(C(C3(C)COC3)=O)CC2C(F)(F)F)cc(F)c1 57567,C(CCN(C)C(C1CCCCC1C)=O)(C(C)C)NC(C1(CC=C)CCC1)=O 57568,C1(COC)(NC(=O)C(n2nccc2C)C)CCN(C(=O)CSS(C)(=O)=O)CC1 57569,C1(CC(=O)NC(c2ccco2)C)(OC)CN(C(=O)CNC(C2CCCCC2)=O)C1 57570,c1(NC2CCCN(C(c3ncncc3Cl)=O)C2)ccnc2ncnn12 57571,N1(C(C(CC)C(C)O)=O)CC2(CCCC2NC(=O)CCCn2nc(C)nc2C)C1 57572,N1(C(c2c(C)ocn2)=O)C2CCC1CC(O)(CNC(C1(C3CCC3)CC1)=O)C2 57573,N1(C(C2CCCN(C(CCCC)=O)CC2)=O)C2CCC1CC(OC)C2 57574,C12(C(=O)NC3CN(C(c4ccc(OC)cc4)=O)C(C)C3)CCCCC1C2(F)F 57575,CCCCC(C)CCC(=O)NCCCC1(NC(c2ccn(C)c(=O)c2)=O)CC1 57576,c1(CC)sc(C(=O)NC(C)(C)CN(C)C(c2ccccn2)=O)cc1C 57577,C=CC(C)(C)CCNC(C1(OC)CCN(C(=O)COCC(C)(C)C)C1)=O 57578,c1(OCCC(=O)NC(CCNC(CSCC#C)=O)C)cc(F)cc(F)c1 57579,c1(CC(=O)OCC)ccc(NCC=Cc2ccsc2)cc1 57580,N1(C(C2CN(C(CCc3cc(C)no3)=O)C2)=O)CC2(CC(CO)CO2)C1 57581,C12(NC(c3ccoc3)=O)CN(C(c3cnsn3)=O)CC1CS(=O)(=O)C2 57582,N1(C(c2cnn(C)n2)=O)CCN(C(C2CCCOCC2)=O)C(c2nccn2C)C1 57583,c1(C(=O)OC)sc(C(=O)N(C2CCN(C(C3(CCF)CC3)=O)C2)C)cc1N 57584,C1(CC(=O)N(C(CC2CC(N(C)C)C2)=O)C2CC2)CCN(C)CC1.C12(CCC1)NC2.CO 57585,C1(Nc2cc(C)n(-c3c(C)cccc3)c2C)Cc2ccc(C#N)cc2C1 57586,c1(CCC(=O)NCC(CO)C2CC2)ccnc(Br)c1 57587,CC(C(=O)N1CCCCC1CCN(C)C(C1(F)CCC1)=O)C(F)F 57588,C=CCC(C)(CC)C(=O)NCCNC(c1cccc(OC(C)C(=O)OC)c1)=O 57589,c1(C(=O)NC(CC)CN(C(=O)C(CSC)OC2CCCC2)C)cnncc1OC 57590,N1(C(C(C)OCC=C)=O)CC(COC)CC1CNC(C1CCC(C(N)=O)CC1)=O 57591,N1(C(C(C)n2cccc2)=O)CCC2(CC1)CC2NC(c1cccc2ncoc12)=O 57592,c1(C(N2C(CNC(C3N(CCCC)CCOC3)=O)CCC2)=O)c(C)nn(C)c1C 57593,c1(OC(CC)C)cccc(CN2CCNCC2C(=O)NCC)c1 57594,C(=O)(C(F)(F)C(F)F)NC(CN1CCN(C(C(C)SC(C)C)=O)CC1)(C)C 57595,c1(N2CCC(NC(C(CC)CCOC)=O)C(OC)C2)cc(C)c(C#N)cn1 57596,c1(COCCC(COC)C2CC2)cncc(C(=O)NCC2CC2)c1.C1(=O)CN1 57597,C(CC(C)C)(C(N)=O)NC(C(C1CCN(C(C2CC(CCC)C2)=O)C1)C)=O 57598,Cc1cnc(F)c(C(=O)NCC(C)N(C)C(c2ncsc2C)=O)c1 57599,C(=O)(CCCC(C)(F)F)NC1C(C)CN(C(C2CC(O)(C(F)(F)F)C2)=O)CC1 57600,C1(C)(C(=O)NCC(CN(C(c2ccc(CC)o2)=O)CC)(C)C)CC2CC2C1 57601,C1(NC(C2(COC)CC2)=O)CN(C(=O)CC2CCN(C)CC2)CCC1C(F)(F)F 57602,N1(C(CC)C(=O)N(C(C)CNC(=O)CCCCC2CC2)C)CCCCC1CO 57603,c1(C(=O)NC(C)CN(C)C(C2CCC(N(C)C)CC2)=O)ccc(F)cc1F 57604,C#CCC(O)C(=O)NCC(C)(C)CCNC(c1sccc1SC(F)F)=O 57605,C1(C(=O)OCC)CN(C(=O)NC(C)(C)C)CC12CCN(c1ncc(Cl)cn1)CC2 57606,c1(N2CCC(NC(C(C)OCCC=C)=O)C23CC3)nc(C)nc2scc(C)c12 57607,C1(CC(=O)NC2N(C(C(N3CCC(C)C3)=O)=O)CCC2)C=CS(=O)(=O)C1 57608,C1(C(N2CC(NC(C3(CC=C)CCC3)=O)C2)=O)CC(=O)N(CCC)C1 57609,n1(C(C)C)cnc2c(NCC(C)S(N)(=O)=O)[nH]c(=NCCCS(N)(=O)=O)nc12 57610,C(N=c1[nH]c2c(c(=NCc3cccc(N)c3)[nH]1)CCCC2)C1CC(C)C1 57611,C1(NC(c2cncc(C)c2Cl)=O)C2CC3CN(C(=O)C(C)CC(C)C)C1C3C2 57612,N1(C(=O)CSC(F)(F)F)CCCCC1C1CCCN1C(=O)CN1CCCNC1=O 57613,C1(C(C2CC2)NC(CN(C)C)=O)CCN(C(C2CCCC2c2cnn(C)c2)=O)CC1 57614,C1(=O)C(NC(=O)C(C)C#N)CCN1.C1(C(CC)C)CCOCC1 57615,N1(C(C(CC)CC)=O)CC2OCCN(C(C3CCC4CC34)=O)C2C1 57616,c1(NC(C23CC(NC(C(CC)(C)C)=O)(C2)C3)=O)c(OC(C)=O)cccc1C 57617,C(COC)(CC(=O)Nc1cccc(C#N)c1)NC(COCCOCC)=O 57618,CSC=CC(=O)NCC(C)(C1CC1)NC(=O)C(F)OC(F)(F)F 57619,Cc1ccc(C2CCCN(C(=O)NCCC(=O)N(C)Cc3cccs3)C2)cc1 57620,N1(C(c2c(O)cc(C)c(Br)c2)=O)CC2CCCC(C1)C2C(N1CCC1CO)=O 57621,Cc1cc(C(C)C)nc(=NCC(C(C)(C)C)NC(C2C(C)C2C)=O)[nH]1 57622,n1(CCC)cccc1C(N1C(C(=O)N(C)CCc2ncccn2)CC1C)=O 57623,CC(C)(CNC(c1occc1C1CC1)=O)CNC(C1(C)CC1F)=O 57624,N1(C(C2CC(CNC(c3c(C(C)C)nco3)=O)C2)=O)CC2CC(C)C2C1 57625,Cn1nccc1C(CO)NC(=O)NC1CC(C(=O)O)OC1 57626,N1(C(C=NOC)=O)CC2=C(C1)CN(C(C1CCCO1)=O)C2 57627,C1(CNC(c2ncc(C)nc2)=O)CC2CCC1N(C(=O)CC1CC(C)(C)CO1)C2 57628,C1(c2nnnn2C)(NC(c2ccn(C)n2)CC)CCOC2(CCCC2)C1 57629,S(=O)(=O)(c1ccc(-c2ccccc2Cl)s1)N1C(C)CC(C(=O)OC(C)(C)C)C1 57630,N1(C(=O)C=C2CCCCC2)CCCC(C2CCCN(C(C3CCCOC3)=O)C2)C1 57631,C1(CN(C(=O)CCN(CCO)CCO)C)CCCN(C(=O)C=Cc2cccnc2)C1 57632,N1(C(c2c(C)[nH]cc2)=O)CCC(O)C(NC(=O)C(C)Cc2ccco2)C1 57633,CC1CN(C(c2csc(Br)c2)=O)CCN1C(c1cc[nH]n1)=O 57634,CC(C)(C)CC(O)CC(=O)N(CC(N1CCCC(CO)CC1)=O)CC1CC1 57635,c1(N2CCCC(C)(C)CC2)nc(N2CCSC(C)(C)C2)c2ncsc2n1 57636,C1(CNC(C(C(=C)Cl)(C)C)=O)C(C2CC2)CCN1C(=O)CCc1cnc(C)s1 57637,C1(C2(O)CN(C(c3ccc(C(C)(C)C)cn3)=O)C2)(CNC(C=C(C)Cl)=O)CC1 57638,N1(C(c2ccco2)=O)CC2CCC(NC(C3(C(F)F)CCC3)=O)CC2C1 57639,C12(C(=O)OC3CCC(c4n(C)ccn4)CC3)CCC(=O)N1CC1(CC1)C2 57640,c1(OC)ccc(Br)cc1C(N(C)C(=O)On1cc(C(C)(C)O)nn1)C1CC1 57641,C1(CN(C(c2ccon2)=O)CC)CCCN(C(=O)CN2CCC(C)(O)C2)C1 57642,C1(CC(=O)NCC(CNC(C(CC)(F)F)=O)(C)O)CS(=O)(=O)CCN1C 57643,N1(c2snc(CC)n2)CCC2(CC1)OCCCC2NC(=O)CN(C)CC 57644,c1(COC)cc(C(N2CCC(C(C)(C)NC(=O)C(C)C)C2)=O)c(C)o1 57645,Cc1c(Cl)c(C(N2CC3CC3(NC(=O)CC3CC(F)C3)C2)=O)nn1C 57646,N1(CCC(=O)NCCN(C(CC2C(C)C2)=O)C)CCOC1=O 57647,C123CC(CCO1)(C2)CC3.c1(C(=O)OC)cnccc1C(=O)OC.c1(=O)c(=O)[nH]1 57648,Cc1cc(O)nc(CNC(C2CCCC2C(C)C)=O)n1 57649,S(=O)(=O)(c1ccc(-c2cccc(C(F)F)c2)cc1)NC1CCC(=O)NC1 57650,O=C(CCCC(F)(F)F)NC12CC(NC(C3CC4CCCCN4C3)=O)(C1)C2 57651,N1(C(CCNS(C)(=O)=O)=O)CCc2ccccc2C(NC(C2CCC(F)C2)=O)C1 57652,CCCC(C)CC(=O)NC12CN(C(c3cccc(OC)c3N)=O)C(COC)(C1)C2 57653,C1(C(=O)NC2C=CCN(C(C(n3cc(C)nc3)(C)C)=O)C2)CC2CCCC2C1 57654,N1(C(CS(CC)(=O)=O)=O)CCC2CN(C(=O)CC(=O)N(C)C)C(C)C12 57655,c1(C(C)(C)NC(c2ccc(-n3c(C)cc(C)n3)nc2)=O)nc2ccccc2[nH]1 57656,C1(C(C(=O)OC)OC(=O)Cc2cscc2Br)CCc2ccccc2C1 57657,c1(CSC)nc(SC(C)COC2CCOC2)n(C2CCN(C)CC2)n1 57658,CCCC(CCC)=CC(=O)N(C1CN(C(c2sc(C)cc2C)=O)C1)C 57659,C1(C(N(C)CCOCCCNC(=O)CCNC(N)=O)=O)CCS(=O)(=O)N1.C(=O)N 57660,C1(NC(CSCCC(C)C)=O)CC2(CCN(C(C3CCC(C)S3)=O)CC2)C1 57661,N1(N2C(CNC(=O)Nc3cn(C4COC4)nn3)CC2)CCc2ccncc2C1 57662,N1(C(c2csc3nccn23)=O)CCC2(CCCN2C(c2cc(O)cs2)=O)C1 57663,Cc1nnc2n1CCC2(C)C(=O)NCc1ccc2c(c1)OCC(=O)N2 57664,c1(C(c2n(CCC)nnn2)NC2CCC(OC)C2)ccccc1Br 57665,c1(C(=O)NCCN(C(C2CC(F)C(=O)N2C)=O)CC)ccnc(C)c1N 57666,Cc1ccc(Br)c(C(=O)NC2CCCCC2NC(C2CN(C)C2)=O)n1 57667,CN1CC2CC2(CNc2cccc(Oc3ccc(F)cc3F)c2)S1(=O)=O 57668,C(=O)(C(C)(F)C(C)(C)F)N1CCN(CCN(C(c2c(C)nco2)=O)C)CC1 57669,C(CCCCCCC(F)(F)F)NC(C1CC(c2ccc(C)cc2)(O)C1)=O 57670,Cc1ccnc(C(F)(F)C(=O)NCC2CCCN(C(C3CCCN(C)C3)=O)C2)c1 57671,N1(C(CN(C(=O)CCCc2ccccn2)C)=O)CCC(N2CCC2)C1 57672,N1(C(c2c(CC)n(CC)nc2)=O)CC2(CCC2)CC1CNC(C1OCC1(C)C)=O 57673,CCCC(C)(O)C(=O)N(CC(C)N(C(=O)Cc1ccco1)C)C 57674,CC#CCC(C(=O)NC1CC2CC(O)C1C2)NC(c1ccnc(C)c1)=O 57675,N12CCCC1C2=O.c1(C(C(=O)NC2CC(NC(=O)CO)C2)N(C)C)cncn1C 57676,C(=O)(C(C(=O)OC)C(C)C)N1CCCC(CC=C)(NC(=O)CCOC2CC2)C1 57677,CC1CN(C(=O)NC2CN(C(=O)CCC3CCC3)CC2C#N)CC(C)O1 57678,c1(C(=O)NC2C(C)CN(C(=O)C3=CCCO3)CC2)cnn2c1CC(C)CC2 57679,C12(C(N3CC(NC(=O)COc4nc(O)nc(O)n4)C3)=O)CCCCC1OCC2 57680,c1(C(=O)NCCCC(C)NC(C(C(C)(C)C)SC)=O)cc([N+](=O)[O-])ccc1C 57681,c1(C(N(C2CN(C(=O)Cc3ccoc3)CC2O)C)=O)cnc2ccccc2c1 57682,Cc1c(C(=O)NCC(F)CNC(=O)C(c2ccn(C)c2)C)cnn1CC(F)F 57683,N#Cc1cc(-c2cc(C(=O)Nc3ccc4c(c3)COC4)ccn2)ccc1O 57684,C1(C(=O)NCC2(NC(C3C(C)C3)=O)CC2)COC2CC1C2 57685,Cc1ccc2c(=NCC(=O)N=S(C)(C)=O)[nH]c(=NCc3cccc(Cl)c3)[nH]c2c1 57686,n1(CCC)cc(C(N2CCC(C(C)(C)NC(c3cc(C)cn3C)=O)C2)=O)c(C)n1 57687,C(=O)(CCCCCC#N)NCc1cc(C(=O)NC(CC(=O)OCC)C)ncc1 57688,N1(C(c2cccc(CSC)c2)=O)CCC(C2CCN(C(=O)C=C3CCC3)C2)CC1 57689,C1(NC(c2ncc(F)cc2F)=O)CC2CN(C(=O)C=C3CCSCC3)CC12 57690,C1(N(C(C(N2CCC(O)CC2)C)=O)C)CCN(C(C2CC(F)(CO)C2)=O)CC1 57691,C(=O)(C(F)CC(C)(C)NC(=O)CCn1ccc(C)n1)N1CC(C#C)C(OC)C1 57692,Cc1cccc2cc(C(=O)NCC3CN(C(=O)COCC(F)F)CCC3C)oc12 57693,C(CCCCCC(=O)N1CCC(NC(C2CC(OC(F)(F)F)C2)=O)C(O)C1)SC 57694,c1(COCC(=O)NC2CC(C)(NC(C3C(C)CC3)=O)C2)ccccc1 57695,n1(CC(=O)NC(CCN(C(c2cc(SC)oc2C)=O)C)C)cnc([N+](=O)[O-])c1 57696,CC1(C(=O)NCCC(O)C(=O)NCC(O)C2(Cl)CC2)C=CCCC1 57697,c1(C(N(CCNC(=O)Cc2cc(C3CC3)no2)CC)=O)cncc(C)n1 57698,CCC(C)C(C(=O)N1CCC=CC1C(=O)NC(C)CN(C)C(C)C)N(C)C 57699,N1(C(c2n[nH]c(C)c2Cl)=O)CC2CCCC(NC(C3CN4CCN3CC4)=O)C2C1 57700,CC(CS(C)=O)C(=O)N1CC(CCNC(=O)CC2=CCCC2)C1 57701,C1(CCNC(C(C)CN(C)C)=O)CCCN(C(=O)C(=C2CCCCC2)F)C1 57702,CC1(C)CCc2sc(C(c3nnnn3C3CCOCC3)NCCC3CC3)cc2C1 57703,CC(C)(CNC(C1(F)CCC1)=O)CC(=O)NC1CCNC1=O 57704,C(=O)(C1=CCCCO1)N1CCC(CCNC(C(C)Sc2ccc(Cl)cc2)=O)C1 57705,C1(NC(C2(CSC)CC2)=O)CCC(N(C(=O)CN2CCOCC2)C)C1 57706,C1(C(=O)NCC(C(C)O)C)CCOCCN1C(C1CCC(C)(C)C1)=O 57707,N1(C(CC2CCC(C)(C)C2)=O)CC(NC(C2CC2C2CC2)=O)C2CCCC12 57708,CCCCCCC(C)CC(=O)NC1(COC)CN(C(c2c[nH]nc2[N+](=O)[O-])=O)C1 57709,c1(C(=O)NC2CC(NC(C(c3cccs3)SC)=O)C2)cc(-c2cccnc2)[nH]n1 57710,C(=O)(CCCC(=O)OCc1csc(C(N2CCC(OC)C2)=O)c1)OC 57711,CC(C)CC(C(=O)NCCC(C)NC(=O)CCc1nccn1C)c1ccccc1 57712,C(C(C)(C)CNC(CCNC(=O)NC)=O)N(C(=O)C(c1ccccc1)C)CC 57713,C1(NC(C(N2C(=O)CCC2=O)C)=O)CCN(CCc2ccc(F)c(F)c2)CC1F 57714,c1(C2(C(N3CC(C)(NC(c4c(Cl)cn(C)n4)=O)C3)=O)CC2)ccccc1C#N 57715,C1(OC)CCCC1C(=O)NC(C)CCNC(c1cn(C)cn1)=O 57716,C(C(CO)CC(C)C)NC(C1(CCNC(C(C)=C2CC2)=O)CCC1)=O 57717,N1(C(c2c(CNC(c3nc(CCC)oc3)=O)c[nH]n2)=O)CC(O)CC1C1CC1 57718,c1(OC)cnc(C(=O)NC(C)(CNC(C2CCCC2O)=O)Cn2cccn2)cn1 57719,C1(NC(c2c(C)coc2)=O)CCCC(CN(C)C(c2nn(C)cc2Cl)=O)C1 57720,C(=O)(C1CCCc2cc(C#N)ccc21)NCCN(C(C(CN(CC)CC)F)=O)C 57721,C=CC(C)CN=C(NCC1CCCO1)NCC1(C(C)(F)F)CCOCC1 57722,Cc1nc(N2CC(NC(=O)CC(C)O)C(C#N)C2)c2cc(Br)ccc2n1 57723,N1(C(=O)C(c2cccc(Br)c2)O)CC2CN(C(=O)C=Cc3cnccn3)C2C1 57724,C(CCC(O)CO)N(C(=O)CC1CC1CNC(C1(CO)CCCCO1)=O)C 57725,C1(CNC(C(c2ccc(C)s2)C)=O)CN(C(=O)CCc2cncc(F)c2)CC1C 57726,c1(C(=O)NC2CN(C(c3ccc(C(=O)OC)[nH]3)=O)C3C2C3)ccccc1[N+](=O)[O-] 57727,c1(NCC2CC(O)(CNC(c3c(CC)scn3)=O)C2)cc(C)nc2ncnn12 57728,c1(OC)cc(F)c(F)cc1C(=O)N(CCNC(=O)Cc1cnn(CC)c1)C(C)C 57729,C1(OC)CN(C)C(C)(C(=O)NC2CCCCC2CNC(c2[nH]cnc2C)=O)C1 57730,C#CCC(C(=O)NCC(C(=O)OC)OC)NC(=O)C1=CCSC1 57731,CC1Oc2c(C(N3CC4(CCC4NC(=O)COCCF)C3)=O)cccc2NC1=O 57732,C1(C(N(CC(C)NC(c2cc(C(C)=O)oc2C)=O)C)=O)CCS(=O)(=O)N1C 57733,c1(SCCC(=O)N(C(C)CN(C(=O)Cc2ccoc2)C)C)ccccn1 57734,c1(CNC(C2CCN(C(=O)OC(C)(C)C)C2)C)ccc(Cl)cc1C(F)(F)F 57735,N(C1CCCOc2c(F)cccc21)C(c1ccc(SC(F)(F)F)c(F)c1)=O 57736,C(=O)(C(O)CCCNC(c1c[nH]c(=NC)s1)=O)N(CC=C)CCOC 57737,c1(OCC)ccc2ccccc2c1CN1CCC1C(=O)Nc1csc(Br)c1 57738,C1(C2CCCC2)(C(N2C3C(NC(c4ccnc(C5CC5)n4)=O)CC(C3)C2)=O)CCC1 57739,CC1(C)CC1(C(=O)NC1CC1O)NC(=O)COc1ccccc1 57740,c1(NC2C3N(C(c4cc(CCC)on4)=O)CC(CC3)C2)ncc(Cl)cc1[N+](=O)[O-] 57741,N1(CC(C)NC(=O)C(C2CCN(C(c3cc(O)cs3)=O)C2)F)CCCCC1 57742,N1(C(C2C(=C)C2)=O)CCC(C)C(NC(c2cc(C3(O)COC3)on2)=O)C1C 57743,c1(C(N2CC(NC(C=Cc3nc(C)c(C)[nH]3)=O)(CO)C2)=O)nccc2occc12 57744,N#Cc1cncc(C(=O)NCC2CCCCC2c2ccccc2C(F)(F)F)c1 57745,Cc1cc(C)c(NC(C2CC3CC3N2Cc2cnc(-c3ccccc3)[nH]2)=O)cn1 57746,C1(C(=O)NCC2CCCN(C(=O)Cn3ccnn3)CC2)CC2(CCOCC2)CO1 57747,C12(NC(CCCn3cc(C(C)(C)NC(C)C)nn3)=O)CC3CC(C1)CC(C)(C3)C2 57748,c1(CC)ccc(N)c(C(=O)NC23CCC(NC(C4CCCO4)=O)(CC2)C3)c1 57749,N1(CCC)CCCC(NC(C2CC(F)CN2C(C2CC2CC(C)C)=O)=O)C1 57750,N1(C(c2c(C)nc[nH]2)=O)CC(C)CCC1CNC(=O)COc1ccsn1 57751,N1(C(CSC)=O)CCC(CNC(=O)C=Cc2ccccc2C(F)(F)F)C12CCC2 57752,C#CCC(O)C(=O)N1CCC(C(=O)NCc2cnn(CC)c2C2CC2)C1 57753,S(=O)(=O)(c1ccc2c(c1)CCCO2)NCc1c(COC)cccc1 57754,N1(C(Cc2c(C)non2)=O)CC2C(CN(C(=O)C=CC(=O)NC3CC3)C)C2C1 57755,c1(-c2c(O)ncc(C)c2)n[nH]c2c1CN(Cc1ccc(Cl)c(Br)c1)C2 57756,c1(C(N2CCC(S(N)(=O)=O)C2)C(=O)NCC(C)C)noc2c(Cl)cccc12 57757,N1(C(c2c(C)n[nH]c2)=O)CC2CC1(C(N1CCCC1CF)=O)C2 57758,c1(C(N2CCC(NC(CCOC)=O)CC2C)=O)ccc(S(N)(=O)=O)c(C)c1 57759,CC1ON=C(C(=O)N2C3CCC2CN(C(c2cc(=O)cc(Cl)[nH]2)=O)C3)C1C 57760,c1(C(N2CCCC(NC(C(C=C=C)C)=O)C2)=O)cccc2c1CC(C)(C)C2 57761,CCCCC(C)C(=O)NC(CNC(C1(CSC)CC(F)(F)C1)=O)CC 57762,CCC(C)C(O)C(=O)NCC1CC2CN(C(c3cc(C)cs3)=O)CC12 57763,C(=O)(C(C)C(C)C(C)(C)C)N(CC)CC1CCN(C(c2ccc(C)n2C)=O)CC1 57764,C(=O)(C1CCc2ccccc21)N1CC(OC)C(NC(c2csnc2C)=O)C1 57765,C(CCC(C)C)(C(=O)N(C)Cc1cc(C)cs1)NC(C(C=C)C)=O 57766,N1(C(c2c(CC)onc2C2CCOCC2)=O)CCC(NC(=O)C=NOC)C(F)C1 57767,C(=O)(C(CC(C)C)NC(C1CC2CCC(C1)O2)=O)OC(CCCC)CNC(C)=O 57768,c1(C(N2C(C(C)NC(C=C(C)Cl)=O)CCC2)=O)cnc(C)cn1 57769,c1(-c2nn(CC)c(CC3COC(=O)C3)n2)ccc(N(C)C)cc1Cl 57770,c1(C(=O)NC(CNC(CC(C)OC)=O)C(C)C)cc2cc(Cl)sc2[nH]1 57771,C(CCC(C)(C)C(=O)NC1CCn2nnnc2C1)NC(C(COC)C)=O 57772,c1(C(=O)NCC2(OC)CN(C(=O)C3=C(C)CC3)C2)ccc(C(F)(F)F)c(N)c1 57773,C1(NC(C(c2cn(CC)nc2)(F)F)=O)CCCC1(C)CNC(=O)CN(C)C 57774,C(=O)(C(COC)CC(C)C)NCCC1CC(NC(C(CC)n2cncn2)=O)C1 57775,CC1CC(NC(c2cc3n(n2)CCC3)=O)CCN1C(C1CN(C)CC(C)O1)=O 57776,c1(OCC)ccccc1OCCSCC1COCC1(C)C 57777,N12CCCC1CN(C)C(C)C2=O.n1(CCCNC(N)=O)cc(Br)cn1 57778,C1(NC(C2(SC)CC2)=O)CN(C(=O)CNC(c2ccsc2)=O)CC1C1CC1 57779,C12(NC(c3ccc(=O)n(CCF)n3)=O)CCCC1N(c1ncc(Br)cn1)CC2 57780,c1(C(=O)Nc2cccc(NC(c3cc(C)cc(F)c3)=O)c2)cc(Br)cc(C)c1C 57781,CC(C)CCCOCC(N1CCC(C(=O)N(CC(C2CC2)OC)C)C1)=O 57782,c1(CCOCC)[nH]c(=NC2CC(N3CCC3)C2)nc2scnc12 57783,c1(C(=O)NC(CC)CN(C)C(c2cnns2)=O)ccc(-c2cnn(C)c2)o1 57784,N1(C(C2(CC)CC2)=O)CCCCC(CNC(c2nccc(Cl)c2Cl)=O)C1 57785,C1(CNC(=O)CCOCC2CCCO2)CCN(C(C2CC(=C(F)F)C2)=O)CC1 57786,C(CN=C(NCc1ccccc1)NC1CC2(C1)CC(F)(F)C2)C1NC(=O)OC1 57787,CC1(C)CC(C(=O)NC(C)(C)CCCNC(=O)CCc2nc[nH]n2)=NO1 57788,C1(CC(N2CC(N(C(C3CC(C(=O)OC)(CC)C3)=O)C)C2)=O)CC(OC)C1(C)C 57789,C12(NC(CC(=C=C)C)=O)CCCCCC1N(C(C1CC3(C1)CS(=O)(=O)C3)=O)CC2 57790,C1(CCC)CN(C(C2CC2CC)=O)CC1NC(c1cc(O)nn1C)=O 57791,c1(CC(=O)N(C(C)CNC(C2CN(C(N)=O)C2)=O)C)cc(C2CC2)no1 57792,N#CC1(CCC(=O)NCC2CCCC2NC(=O)CCN2CCOCC2)CCC1 57793,c1(OCC(=O)NCC(C)NC(c2ccc(CC)cn2)=O)ccc2c(c1)CCC2=O 57794,C1(NC(C(CO)OC)=O)CN(C(c2oncc2C)=O)C2CCCC12 57795,c1(C(N(CC(C)N(C(C(C=C=C)C)=O)C)C)=O)ccc2c(c1)NCCC2 57796,CCCCC(CC)CC(=O)NCCCN(C(=O)CC(C)c1ccco1)C1CC1 57797,N1(C(C(CC)CCOC)=O)CC2CC(C1)CN(C(C1OC(C)(C)OC1(C)C)=O)C2 57798,C(=O)(CC(C)C(=O)NCC(C)CC(=O)N(C)Cc1cncn1C)OC 57799,C1(NC(c2c(C)noc2)=O)CN(C(=O)C=C2CCCCC2)C2CCCC12 57800,c1(OC)c[nH]c(C(N2CCN(C)CC2CNC(=O)C(C)CC2CC2)=O)cc1=O 57801,Cc1[nH]c(=NC(C)c2nccn2C)sc1Br 57802,c1(CC)oc(C)cc1C(=O)NC(C1CC=CCC1)C(=O)Nc1cnsc1 57803,CC(CO)(C(F)F)NC(=O)CC1(NC(=O)C(N)=O)CC1 57804,C1(C(N(CC(C)CNC(C2(C)CCC2)=O)C)=O)OCCN(C)C1=O 57805,c1(C(N2C(C)C(C)N(C(=O)COCCN(C)C)CC2)=O)ccnc2c1nnn2C 57806,C1(NC(c2n(C)ccc2)=O)CC(NC(c2ccc(-c3ccco3)[nH]2)=O)C(O)C1 57807,N1(C(CCCCC#C)=O)CC2CC(NC(c3ccc(F)c(Cl)c3)=O)C(C2)C1 57808,Cc1ccc2[nH]c(CN(C3C4CCOC4C3(C)C)C(C)C)nc2c1 57809,C(CC(O)CO)NC(C1N(C(COCCOC)=O)CC1)=O 57810,CCC(N=c1cccc(S(=O)(=O)NC(CC2CC2)CO)[nH]1)c1cc(C)ccc1C 57811,c1(NCCC2C(C)CN(C(=O)CCC[N+](=O)[O-])C2)c([N+](=O)[O-])cnn1C 57812,CC12CC1CCN2c1nnc(-c2ccccn2)o1 57813,N1(C(C=C)=O)CCC2(CNC(c3c(F)cc(F)cc3F)=O)CCCCC12 57814,n1(CCOC)nc(C)cc1C.C1(O)(S)CC(CC(N2CCCC2C2(C(=O)N)CC2)=O)C1 57815,CCC(C)(CNC(=O)C(OC)OC)C(=O)N(C)CCOCCO 57816,C(c1ccc(OC)c(Cl)c1)=CC(=O)NCC1N(C(CS(=O)(=O)NCC)=O)CC1 57817,c1(C(N(CCCCNC(C=Cc2ncc(C)[nH]2)=O)C)=O)cnc2ccccc2c1 57818,c1(OC2(C(=O)NC(CCCNC(C3C(OC)CC3)=O)C)CC2)ccc(C)c(C)c1 57819,C#CC1(C(=O)NCC(CO)N(C)C)CCN(C(=O)C(n2cc(C)cn2)C)C1 57820,N1(C(CC(C)n2cccn2)=O)CCCC(C)(NC(c2ccc(CO)cn2)=O)C1 57821,c1(CC(=O)NC23CCCC(NC(=O)Cn4nccn4)(C2)C3)csc2ccccc12 57822,C1(CNC(CNS(NC)(=O)=O)=O)CN(C(=O)CN2CCCC2CO)CCO1 57823,N1(C(C(c2scc(C)n2)C)=O)CCCCC(NC(c2ccc(N)c(F)c2)=O)C1 57824,N1(C(c2c(C)c(N)ccc2)=O)CCC(C2CCCN(C(c3occc3Br)=O)C2)C1 57825,CC(C(C)(C)O)N(C(=O)C(C)CNC(C1CCC(C(N)=O)C1)=O)C 57826,C1(SCC)CCN(C(n2c(C(CC3CCCCC3)N)nnn2)=O)C1.C1(C)CC1 57827,c1(CCC(=O)NCCCCNC(c2ccc(CO)o2)=O)cc(F)ccc1F 57828,c1(C(c2nnnn2CCC)NCCCC=C)ccnc(-n2ccnc2C)c1 57829,N1(CCC)CCCCC1C(=O)NCC1(CCNC(=O)CC2CC(=O)NC2=O)CC1 57830,c1(C(N(C)CC2CCCN(C(COCCCC#C)=O)C2)=O)cc(F)c(F)cc1O 57831,CC(F)(F)CCCC(=O)NCCOCCNC(C1(c2ccccc2)CCC1)=O 57832,N1(C(c2ccc(=N)[nH]c2)=O)CCC(F)(CNC(=O)CC2CNC(=O)C2)CC1 57833,c1(C(=O)NCC(CNC(c2cc(C)c(C)nc2)=O)CO)ccc2cn(C)nc2c1 57834,CC1CN(CCCCNC(=O)NC2CC=CCC2)CCO1 57835,C(=O)(CN=c1cc[nH]cc1)N1C(CNC(c2ccc(F)c(C)c2C)=O)C(C)CC1 57836,C1(C(C)NC(C(C)=CC)=O)CCCN(C(C2CC(OC(C)=O)C2)=O)C1 57837,c1(NC(c2cncc(-c3cc(C)cc(F)c3)n2)=O)cc2nc[nH]c2nc1C 57838,c1(C(C)C(N2CCC(c3cn(CCCCC(=O)O)nn3)CC2)=O)cccc(C#N)c1 57839,c1(CN2CC(NC(c3ncn(-c4ccccc4)n3)=O)C(F)C2)cc(Cl)nc(Cl)c1 57840,CC1(C(=O)NC2CCCC(NC(c3cccc(C(F)(F)F)c3)=O)C2)CCCCO1 57841,Cc1nc(N2CCC3CC(C(=O)NC(C)CC(C)C)C3C2)ncc1[N+](=O)[O-] 57842,Cc1nc(=O)n(C2CCN(C(=O)CC(c3ccc(F)cc3)NC(N)=O)CC2)[nH]1 57843,C1(C(N2CCC(N(C(c3cnn(CCO)c3)=O)CC)CC2)=O)C2CC3C(C2=O)C13 57844,C1(CC=C)(C(N2CCC(C)(N(C)C)C2)=O)CCN(C(=O)CSc2nc[nH]n2)C1 57845,C1(C(N(C2CN(C(=O)C=Cc3cnn(C)c3)CC2C(F)F)C)=O)C(C#N)C1(C)C 57846,C=C=CCCC(=O)N(C)CCOCCC(N1CCCCC1C(C)(C)O)=O 57847,c1(COC)ccc(C(=O)NC(C(=O)NC2CCC2CC(=O)OC)C2CC2)s1 57848,n1(CCNC(C2CC(NC(C3(CC4CC4)CC3)=O)C2)=O)ccc(C(F)(F)F)n1 57849,c1(NC(c2ccc(CNC(C(=O)N(CC(F)F)C)CO)o2)=O)ccc(C#N)cc1 57850,C(=O)(CCCCC(F)F)NCCC(C)N(C(C(C)Cc1ccc(Cl)cc1Cl)=O)C 57851,c1(N2C(c3scc(C)c3)CCC2)ncc(C)cc1S(=O)(=O)N1CCCC(COC)CC1 57852,c1(C(=O)NCCCC(C)C)coc2c1CN(C(c1cc3n(n1)CCO3)=O)C2 57853,c1(C(CNC2CCN(C(=O)OC(C)(C)C)CC2O)=O)cc(F)c(Cl)cc1Cl 57854,N1(C(C2(NC(c3nccc(C)c3N)=O)CCCC2C)=O)CCCC2CCCCC12 57855,Cc1cc(CNC(=O)NCc2ccsc2)c(C)s1 57856,C1(CNC(C2CCC(=O)CC2)=O)CC(C(=O)NCCCCCF)=NO1 57857,c1(CN(C(C2C(NC(C(C)=C(CC)C)=O)COC2)=O)C)cccnc1O 57858,n1(CC=C)nnnc1C(C(CC)=CCC(=O)OCC)NC1CCC(C(=O)OC)C1 57859,c1(CC)onc(C(=O)NC2CCOCC2NC(=O)CC(C)n2ccnc2)c1C 57860,CCC(C)(C(=O)Nc1ccccc1CN(C(=O)C(C(=O)OC)OC)C)C(N)=O 57861,c1(CCC(=O)NCC2CC2NC(C23CCCC2C3)=O)cccc(Br)c1F 57862,Cc1nc(-c2ncc[nH]2)sc1C(=O)NCCNC(=O)Cc1ccccc1Br 57863,C(=O)(CC1=CCCC1)NC1C(C)(C)C(C(N2CCC(O)C3CC23)=O)C1 57864,N1(C(C(C)(F)F)=O)C(C(=O)NC2(CO)CC3CCC2C3)C2CC(O)C1C2 57865,N1(C(=O)OC(C)(C)C)CCCC(NC(C2CCC(=O)N(C3CC3)C2)=O)CC1 57866,Cc1cnsc1C(N1CCC1C(=O)NCCC(N1CC(c2cnccn2)C1)=O)=O 57867,N1(c2nnc(CCC)s2)CC2CCC1C1CN(C(=O)CCC(C)N(C)C)CC21 57868,N1(C(c2c(C)nn(C)c2)=O)CCN(C(c2ccncc2Br)=O)C2COCC12 57869,CP(C)(=O)CCC(=O)N1CCCCC1C1(NC(c2[nH]ncc2C#N)=O)CC1 57870,C1(CC(N2CCC(C)(CCC)C2)=O)CC(C)(C)CN1C(=O)CC(C)(C)C 57871,C(=O)(C1CC(=O)c2ccccc21)NCC1CN(C(c2ccc(C)[nH]2)=O)C(C)CC1 57872,c1(C(=O)NCC(C)N(C)C(C2C(C)C2C)=O)cc(S(=O)(=O)NCC(N)=O)c[nH]1 57873,Cc1[nH]nc2ncnc(N3CCCC(CN(C)C(c4coc(C5CC5)n4)=O)C3)c12 57874,c1(NC(C2C(NCc3cc(C)sc3C)CCCC2)=O)c(C)ccc2n[nH]cc12 57875,N1(C(CC=C=C)=O)CC(C)CN(C(C2CC(C(F)(F)F)C2)=O)C(C)C1 57876,c1(C(N(C2CCCN(C(C(C)N(C)C)=O)C2)C)=O)cc(Cl)c([N+](=O)[O-])[nH]1 57877,C1(NC(CCSCCCC)=O)CCC(CCC(=O)N(C)CCOC)C1 57878,c1(C(N2CCC(NC(CSC(C)C)=O)C(F)C2)=O)ccc(Cl)c2ccccc12 57879,CC1C(NC(c2cc(-c3ccn(C)c3)[nH]n2)=O)CCN1C(c1cc(C#N)cs1)=O 57880,c1(N2CCC(C(N3CC(S(C)=O)C3)=O)CC2)cc2ccccc2s1 57881,Cc1ccc(C(N2CCOCC2CNC(=O)CCC(C)(F)F)=O)c(C)n1 57882,c1(C(=O)NC2CCC(N(C(Cc3c(C)con3)=O)C)CC2)cnc(CO)nc1C 57883,N1(C(C(CCC)NC(=O)CCc2nc(=N)[nH][nH]2)=O)CCC2(CCOC2=O)C1 57884,c1(C(=O)NCCCNC(c2ccc(N)c(F)c2)=O)ccc2c(c1)S(=O)(=O)NC2 57885,c1(C(N2C(CC)C(NC(=O)Cc3ccc(F)cc3)CC2)=O)cnc(OC)nc1C 57886,N(C1c2ccccc2CC1NC(=O)C(C)N(C)C)C(c1n(C(CC)C)ncc1)=O 57887,N1(C(C(CC)CCOC)=O)CC2CCC1CN2C(=O)CN1CCCCC1C 57888,C=CC1(CC(N2CCC(C(C)C)(CO)C2)=O)CN(C(c2ccncc2NC)=O)C1 57889,C(CS(C)(=O)=O)(C(=O)O)NC(Cn1nc(CCC)n(C)c1=O)=O.CC#CC 57890,C1(C2CCN(C(c3cc(N)cnc3Cl)=O)C2)(NC(CC2C(C)C2)=O)CC1 57891,C1(CC(N2CC3C(NC(c4ccc(C(N)=O)[nH]4)=O)C3C2)=O)CCCC2(CC2)C1 57892,c1(C(=O)NCC2COCC2NC(C2CC2F)=O)cc2c(nc1O)CCCC2 57893,C(=O)(C(CC)C(C)C)NCC1C2CN(C(c3c(CC)ncnc3)=O)CC21 57894,C1(CC(=O)NCC=CC(=O)NCC2(OC)CCOC2)CCCCC1O 57895,C1(NC(C2(NC(C)C)CC2)=O)CCC(CNC(C2(F)CCOC2)=O)CC1 57896,Clc1cccc2c1CCC2NCc1csc(C2CCCO2)n1 57897,N1(C(C2CC3(CC(NC(C4C5CC(=O)CC45)=O)C3)C2)=O)CCC2(CCCC2)CC1 57898,c1(C(=O)NC2CC(F)(CNC(C3CC34CC4)=O)C2)nn2cccnc2c1Cl 57899,c1(C(N2CC(O)(CN(C(Cc3c(C)scc3)=O)C)C2)=O)ccc(Cl)c(O)c1 57900,N1(C(c2ccc(C)nn2)=O)CCN(C(=O)C(C(C)(C)C)n2ccnn2)CC1C 57901,c1(C(=O)NCCC(Cn2cc(CC(C)O)nn2)F)cc(F)c(F)cc1I 57902,c1(C(N2C3(CN(c4cc(C(F)(F)F)nc(C)n4)C3)C2)=O)cnn2ncccc12.COC 57903,C12(NC(=O)CO)CCCC1N(C(c1ncccc1Cl)=O)CC2 57904,c1(C(N2CCCC(C)(CNC(=O)CCCC3CC3)C2)=O)cccc2c1OCO2 57905,C(C(CC(C)C)C(=O)NCCOCCN(C)C(C1(Cl)CCC1)=O)OC 57906,c1(NC(C)=O)cccnc1C(=O)NCC1CC1CNC(=O)CCn1ccnc1C 57907,N1(C(C(CNC(C2CCC(CC)CC2)=O)O)=O)CCC2(COC(C)C2)C1 57908,c1(C(N2CC=CC(NC(c3ccc(C)c(F)c3)=O)C2)=O)cccc2c1OCCC2 57909,N1(C(C(C)NC(N)=O)=O)CC23CCCC2(C1)CN(C(=O)CC(C)(F)F)C3 57910,C#CCC(O)C(=O)N1CCCC(N2CC(NC(c3nc(C)cs3)=O)C2)C1 57911,N1(C(C(C2CCN(C(C(C)(C)C3(O)CCC3)=O)C2)F)=O)C2CSCC1C2 57912,n1(CC(=O)NC(C)CCCCNC(=O)CC2COCCO2)ccc(O)nc1=O 57913,C1(NC(CC2C(C)CC2)=O)CC2CC(NC(c3cnn(C)c3C(F)F)=O)CC12 57914,N1(C(CC2CC(CC)C2)=O)CC=C(CNC(C2CC23CCCCC3)=O)CC1 57915,c1(OC)ncc(F)cc1C(=O)N(C1CCCCN(C(C2CC(C)=NO2)=O)C1)C 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57934,C1(NC(c2cc3n(c2)CCC3)=O)CN(C(c2cscc2Br)=O)CC12CCC2 57935,n1(CCCCNC(N(CCCCc2ncc[nH]2)CC)=O)cnc2ccccc12 57936,N1(C(C(COC)(F)F)=O)CC(NC(=O)C(CO)NC(=O)C(C)C)C2(CCC2)C1 57937,c1(CC)cncc(C(N2CC=CC(C(=O)NC(C3CCC3)C3CC3)C2)=O)c1 57938,c1(NC)cccc(C(=O)NC(C(C)NC(=O)CCCc2ccccc2)C(C)C)n1 57939,C(=O)(C(O)C(F)(F)F)N(CC(=O)NC(C#C)CCC)CC(C)C 57940,CC1(C)COCCC1CNC(C12CC(NC(c3sccc3CO)=O)(C1)C2)=O 57941,c1(C(C)=O)csc(CC(=O)NCCC2CCN(C(c3scnc3C3CC3)=O)C2)c1 57942,c1(C(=O)NCCC(C)NC(C2(C(=O)OC)CC2)=O)cc(N2CCOCC2)ncn1 57943,C1(NC(Cc2ccc(OC)cc2)=O)(CO)CCN(C(C2CCCC(C)C2)=O)CC1 57944,N1(C(C2C(CC)N(C(c3cnnn3C3CC3)=O)CC2)=O)C2CCC1CC(CO)C2 57945,C#CCCCCC(=O)N(C)CC1CCCN(C(=O)C(c2cc(Cl)cc(Cl)c2)C)C1 57946,N1(C(C=CC(=O)OCC)=O)CCC(C2CC2NC(C2(Cl)CC2(F)F)=O)CC1 57947,c1(SCC(=O)N(CC(C)CNC(=O)C(C)c2ccsc2)C)ccc(F)c(F)c1 57948,C(=O)(C(CC1CCCC1)C(C)C)NCCC(CNC(CCCOCC=C)=O)O 57949,c1(C(=O)NCC2(C)CCN(C(c3cnco3)=O)C2)ccc2sc(O)nc2c1 57950,CC1CCCCC1(CNC(=O)CCc1cccs1)NC(=O)Cc1ccon1 57951,n1(CC(=O)N(CC(C)NC(C(CC)(C)C(F)F)=O)C)ncc2ccccc2c1=O 57952,CC1CC(C(N2CC(CN(C)C(C3CCN3C(C)(C)C)=O)C2)=O)CCS1 57953,C1(F)(CNC(=O)C(=O)NCC2CC2)CN(C(=O)Cc2csc(C(F)(F)F)n2)C1 57954,C1(n2cc(C(N3CCCC3)(C)C)nn2)CCCN(C(C2CC23CCCC3)=O)C1 57955,c1(C(=O)NC(CCNC(CCCC(CC)C)=O)(C)C)ccc2c(c1)OCCN2 57956,c1(OCC)cccnc1C(=O)NC1CC(C)N(C(=O)CCOC)C1 57957,N#Cc1cc(NC(C23CC2CN(Cc2ccccc2Cl)C3)=O)cc(Br)c1 57958,c1(C(N2CC(NC(=O)CCC(=O)c3ccccn3)C2)=O)ccc(F)c(C(F)(F)F)n1 57959,C(CN=c1[nH]cncc1I)(N(C(c1ccc(C#C)cc1)=O)C)C1CC1 57960,N1(C(C2N(C(C(C)(C)C)=O)CC2)=O)CCC(O)(C(=O)N(C)C)C1 57961,CCCS(=O)(=O)c1ccc(S(=O)(=O)CN(CCC#N)CCc2ccccc2)cc1 57962,O=C(C1COc2ccc(Cl)cc21)NCCCc1cn(Cc2cscn2)nn1 57963,N1(C(C2C(C=C)OCC2)=O)CCC2CCC(C1)N2C(C1(O)CC(C)(C)C1)=O 57964,C=C1CC(C(N2CCCCC2c2ccccc2F)=O)N(C(c2ccncc2)=O)C1 57965,COn1cnc(C)c1C(=O)NCC1(NC(=O)CC(C)NC(=O)NC2CC2C)CC1 57966,C=CC1(CC(=O)NCc2[nH]nnc2CC)CN(C(C2(COC)CC2)=O)C1 57967,C1(C2CCN(C(c3nnn(CC)c3CC)=O)C2)(NC(C=CC(=O)OCC)=O)CC1 57968,C(=O)(C1=CCC(C)(C)CC1)NCC(CC)(C)NC(C1CC1(COC)COC)=O 57969,c1(CCC(N2CCC3CC3(NC(=O)CSC(F)F)CC2)=O)cc2ccccc2[nH]1 57970,c1(NCC2C(C(=O)Nc3cc(OCC)ncn3)C2)c(Cl)nc(C)nc1Cl 57971,c1(C(=O)NCC(CNC(CC(CC)OC)=O)O)cc(Br)cc(C)c1C 57972,C1(NC(CC2(OC)CCC2)=O)CC2CC(NC(=O)CCSC)C1C2 57973,C(=O)(C(C(C)(C)C)OC)NCCC1CCN(C(c2c(SC)nn(C)c2)=O)C1 57974,C1(C#CC(=O)NC(c2ccccc2)C(N2CCCC(C(F)F)C2)=O)(CC)COC1 57975,C1(NC(C2CCC(C)(C)C2)=O)CC2(CCN(C(c3cc(Cl)c(N)cc3F)=O)C2)C1 57976,n1(CC(=O)NCCNC(C(c2ccc(F)cc2)(C)N(C)C)=O)ccccc1=O 57977,C1(C(N2CC(C)(CC(=O)NC(=O)CC3CCC4CC34)C2)=O)(N(C)C)CCOCC1 57978,C1(NC(c2nnnn2CC)C(C)C2CC2)CC(=O)N(CCc2cccc(F)c2)C1 57979,c1(C(=O)NCC(CNC(C(CC=CC)CC)=O)CO)c(F)ccc(C)c1F 57980,c1(OC)cccc(C(=O)NC2CN(C(C3(C(F)(F)F)CCC3)=O)CCC2C)c1F 57981,c1(C(=O)OC)cc(N2CCN(C(C(C)(C)C)c3nnnn3C)CC2)ccc1F 57982,c1(CC)nc(C(=O)NCC2CC(NC(=O)C(C)CN(C)C)C2)cs1 57983,N1(C(COC(CC)C)=O)CCC(CNC(=O)Cn2nc(C)nc2C)(COC)C1 57984,Cc1c(NC(c2cccc(CO)n2)c2nnnn2CC2CCCO2)cccc1F 57985,C1(CNC(C2CC(C)OC2)=O)CCCCN(C(c2ccnc(Cl)c2F)=O)C1 57986,C12(NC(C(CN(CC)CC)F)=O)CC1CN(C(C1CC1(C)C)=O)C2 57987,N1(C(C(=O)NC(c2c(C)nn(C)c2C)C)=O)CC2CCCOC2C1 57988,c1(C(N2CCC(C)(NC(=O)C(F)C3CCCC3)C2)=O)cnc2c(c1)OCCN2 57989,Cc1ncc(C(=O)NC2CN(C(=O)CC3CC(NC(N)=O)C3(C)C)C2)n1C 57990,N1(C(c2c(NC(C)=O)cncc2)=O)CCN(C(C2COCCO2)=O)C(C2CC2)C1 57991,c1(-n2c(C3CCC3C)nc(-c3ccc(OCC)cc3)n2)cccc2ccccc12 57992,C12(NC(Cc3cc(C)n(C4CCC4)n3)=O)CCCN(C(=O)CS(N)(=O)=O)CC1C2 57993,c1(CC(=O)NC2C(NC(C(CC)n3cccn3)=O)C2)ccc2c(c1)CCOC2 57994,N1(C(C(OC)OC)=O)CCC2(CCC(CNC(C3CC4CCCCC34)=O)O2)CC1 57995,c1(NCC2(C=C)CCC2)ccc(S(=O)(=O)N2CCC(CC)C2C)cc1F 57996,C1(OC(C2CCC3(CCC3)CC2)=O)Cc2ccccc2C1=O 57997,Cc1ccccc1COCC(=O)NC(CNC(C1CCC12CCC2)=O)C(C)C 57998,C1(N(C(C2C(=C)CC2)=O)CCOC)CCN(C(c2nccn2C)=O)CC1 57999,Cc1cc(C#N)cnc1C(=O)NC(C1CCOC1)CNC(=O)CCCCCN(C)C 58000,Cn1ncc2ncc(C(N3CCC4(CCCN4C(C4CC4(C)Br)=O)C3)=O)cc12 58001,CCS(=O)(=O)CC(=O)N1CCC(N(C(=O)CCc2ccncn2)CC2CC2)C1 58002,C(C(C)C(F)C(=O)NC(C)Cc1ccco1)NC(C(C)=CCC)=O 58003,Cc1onc(CO)c1C(=O)NCC1C(CNC(C2CCOC(C)C2)=O)C1(F)F 58004,C1(CNC(C(C(C)C)C)=O)CCN(C(c2ccc(-c3cccs3)o2)=O)CC1(F)F 58005,C1(CC(C)(C)C)CN(C(C2CC23CCOCC3)=O)CCN1C(=O)CCS(C)(=O)=O 58006,C1(N(C(=O)COCc2ccncc2)C)CC2CC1N(C(=O)C(F)=C1CCC1)C2 58007,c1(OC(C2(C)N(C(C=COCC)=O)CCC2)=O)ccc(F)cc1I 58008,CCCCCCC(C)CC(=O)NCC1CN(C(=O)CCc2ncco2)C1 58009,CN1CCCCC1CCC(=O)NCC(C)(C)C(=O)NCCC(=O)O 58010,N1(C(C(C=C)(F)F)=O)CC2CCCC(C1)N2C(=O)C=Cc1ccncc1 58011,C#CCCC(O)C(=O)NCC1(CCNC(=O)C(C)Cc2ccccc2Cl)CC1 58012,S(=O)(=O)(c1ccc(N(CC(O)CF)C)cc1Cl)N(C)Cc1c(C)ccs1 58013,C1(CC(=O)N(C)CC2CCCN(C(=O)Cc3nccn3C)C2)CS(=O)(=O)CCO1 58014,N1(C(CCCOCCOC)=O)CC2(C1)CN(C(c1cnc(C)n1C)=O)C2 58015,C1(NC(CC=C(C)C)=O)CC2(CCN(C(C3CC3Br)=O)CC2)C1 58016,C1(CNC(C2CC(N(C)C)C2)=O)CCN(C(=O)CN2CC3CC3C2)C1 58017,c1(CN2CCCC(NC(=O)NC(CC)COC)C2)nc2ccccc2n1C 58018,c1(C(=O)NCC(CC)NC(=O)C(C)(C)C(C)C)nn(C)c(Cl)c1Cl 58019,c1(CN2CCN(C(=O)CNC(c3ccccc3C3CC3)=O)CC2)ccc([N+](=O)[O-])o1 58020,C1(C)(NC(c2cc(COC)on2)=O)CCCC1NC(=O)C(C)OC(C)=O 58021,Cc1c(NC(=O)C(CC(C)C)ONC(=O)C=Cc2ccc[nH]2)cc(F)cc1CO 58022,Cc1cc(C(=O)NC(CC(=O)NCC(F)(F)Cl)C2CC2)cnc1O 58023,CCCC(CNC(c1[nH]nnc1C)=O)C(=O)NC1CC12CC(OC)C2 58024,c1(N2CC(CN(C)C(C3CC(F)C3)=O)OCC2)ccc([N+](=O)[O-])cc1[N+](=O)[O-] 58025,C1(CCC)CN(C(=O)CNC(c2cccnc2)=O)CCN1C(=O)C#CC(C)C 58026,c1(C(=O)NCC(CC)NC(C2CCCC(C#N)C2)=O)cc2c(C)cc(Cl)cc2[nH]1 58027,C1(C(=O)NCC2N(C(c3nc(C)[nH]n3)=O)CC(O)C2)CCC([N+](=O)[O-])CC1 58028,N1(CCCCCNC(C(CC)C)=O)CCC(Cc2ncc(F)cn2)CC1 58029,C(c1ccc(Cl)s1)=CC(=O)N(CC(F)(F)F)CCC(=O)C(=O)O.C1CN1C.N 58030,C1(NC(CC(C=C)(C)C)=O)CCC(O)CN(C(=O)CCOCC2CCCO2)C1 58031,c1(C(CCC(N2CCC2c2ccccc2)=O)(F)F)ccc(F)cc1F 58032,CCC(C)CC(C(=O)NC)NC(c1cnn(C)c1NC(=O)CCN1CCOC1=O)=O 58033,C1(NC(c2ccoc2)=O)CN(C(c2cccc(OCC(F)F)c2)=O)CC1O 58034,C12(C(=O)NCCCCNC(c3cnc(CC(C)C)s3)=O)CCCN1CC(O)C2 58035,c1(OCCOC)ccc(NC(=O)C=CC(C)NC(=O)Cn2ccnn2)cc1 58036,C1(N(C(c2ncc(Cl)s2)C(=O)NCC2CCCO2)C)CCN(C(C)(C)C)CC1 58037,C1(NC(CSc2nc(C)[nH]n2)=O)CCN(C(C2CC3C=CC2O3)=O)CC(C)(C)C1 58038,N1(C(CSc2cn(C)nc2)=O)CCC2CCN(C(=O)CC3CC3(C)C)CC12 58039,Cn1ccc2c(c1=O)CCN(Cc1ccc(OCc3nn[nH]n3)cc1)C2 58040,c1(N2C(C)CC(CNC(C(CCCC)N(C)C)=O)C2)cc(C)nc2c(C)cnn12 58041,N1(C(C=C(C)C)=O)CC2(C1)C(NC(c1cc3ccc(Cl)cc3[nH]1)=O)CCS2(=O)=O 58042,c1(CC(N2C(C(C)C)CN(C(C3C(F)(F)C34CC4)=O)CC2)=O)ccc(F)c(F)c1 58043,C1(NC(CCC)=O)CCCC(N(C)C(C)=O)C1.C1(=O)CCN1CC(C)(C)C 58044,C(CNC(C)=O)(C(=O)O)N(C(CCSCC)=O)C 58045,C1(C(=O)NC(C)CN(C(=O)CCCCCC#N)C)CC2(C)CCCN2S1(=O)=O 58046,C(=O)(C(CC)(CC)CC)NCc1c(C(N2CCC(OCC=C)CC2)=O)scc1 58047,c1(NC(COOCC#C)=O)ccc(S(=O)(=O)C2CC2)nc1 58048,C(CC(C)(C)C(=O)NC1CC(N(C(=O)CSc2cnn(C)c2)C)C1)OC 58049,Cc1cc(C(=O)NCC2(CNC(=O)C(F)CC3CCCC3)CCC2)nc(C)c1 58050,C1(NC(c2scc(C)c2Cl)=O)CCC2CCN(C(C3CC3(F)F)=O)C12 58051,c1(C(N2CCC(CCNC(C(C)c3cnsc3)=O)C2)=O)cc(O)cc(F)c1 58052,C12(CNC(c3n(C)ncc3)=O)CC3CC(CC(C3)C1NC(=O)CSC(F)(F)F)C2 58053,CC(CNC(=O)CN1CCCC1=O)C(F)C(=O)NCC1(CF)CC1 58054,Cc1cc(C(N2CC(CCNC(=O)Cc3ccn(C)n3)C2)=O)n(C2C(CO)C2)n1 58055,c1(NC)cccc(C(=O)NC(CCN(C)C)C(=O)NC2(C)CCCOC2)n1 58056,N1(C(CN2C(=O)CCCC2)=O)CC2OCCN(C(=O)CC3CC4(CCC4)CO3)C2C1 58057,c1(C(N2CC(NC(c3ccc(SC)cc3)=O)C(F)CC2)=O)c(F)ccc(F)c1O 58058,C=C1CCN(C(c2cn(C)cc2C)=O)C(C(=O)NC(C)CSC)C1 58059,C1(C(=O)NCc2c(C)nn(C)c2C)CC(N=[N+]=[N-])CN1C(=O)C(C)C1CCC1 58060,S(=O)(=O)(c1ccc(O)c([N+](=O)[O-])c1)N(S(CCCC(=O)OC)(=O)=O)C 58061,c1(N(C2CN(C(C3(C)CC3(F)Cl)=O)C2)C)cc(F)ncn1 58062,c1(OC)ccc2c(NC(=O)NCC(C3CC3)OC)c[nH]c2c1 58063,CC#CCCCC(=O)NC1COCC1C(N1CC(OC)CC(C)C1)=O 58064,Cc1cc(C)c(C(=O)NCC2(CNC(C3(C)CC3(C)C)=O)CC23CCC3)o1 58065,c1(NC)cccnc1C(=O)NC(C)CC(C)NC(=O)COCCCF 58066,C1(O)(CN(C(C=CC(CC)=CC)=O)C)CCN(C(=O)CC2(O)CCC2)C1 58067,N1(C(C)=O)CC2CC2(C(=O)NC2(c3cccnc3)CC2)C1.N12CC(C1)C2=O 58068,c1(C(=O)NCC(C)N(C(COCC(c2ccccc2)C)=O)C)ccc(N)cc1O 58069,c1(NC(C)CN(C(=O)C2=CCSC2)C)ncnc2c1nnn2C1CC1 58070,c1(-c2n(C3C(C)(C)OCC3)nc(Cc3ccc(F)cc3)n2)cc2c(s1)CCOC2 58071,N1(C(c2cc(C)sc2)=O)CCCOC(CNC(C2CCCN(C)C2)=O)C1 58072,O=S(=O)(c1ccc(=NCc2ccccc2Br)[nH]c1)NCC12CCCC1OCC2 58073,c1(CC)noc(C)c1C(=O)NCc1csc(C(N2CCC2(C)C(C)C)=O)c1 58074,N1(C(c2cc(N(C)C)ncc2)=O)CC2(C1)CN(C(=O)CNC(N)=O)CCO2 58075,C(CCCCC)(C1CCCCC1)(C1CC1)OC.C1CS(=O)(=O)N1 58076,c1(OCC)ncc(F)c(N2CC3CC2CN3CS(=O)(=O)CCCCl)n1 58077,c1(C(=O)NC2C(C)(C)C(O)C2)ccc(C#N)c(CC(F)(F)F)n1 58078,CC12CCC(C(=O)NC3CC3NC(=O)CCCN3CCCC3)(CC1)CO2 58079,c1(C(=O)NC(c2nnc(C)o2)C)ccc(C)c(S(=O)(=O)F)c1 58080,c1(C(N(CC(C)(C)CNC(=O)CCC2CCC(=O)N2)C)=O)ccn2cccc2c1 58081,C12CC3COCC3N1C2.c1(C(=O)OC)ccnc(N2CC3C(C(=O)OC)C3C2)n1 58082,c1(CC)[nH]c(C(=O)NC2CC(CO)N(C(=O)Cc3nonc3C)C2)nc1Cl 58083,c1(C(N2CC(NC(C(CSC)O)=O)C(C)C2)=O)coc2c(C)cccc12 58084,C1(NC(=O)NCC2C(C)CCC2)CC(=O)N(CC2CCC2)C1 58085,C(c1ccc(F)c2ccccc12)=CC(N1CC(NC(CC)=O)CC(F)(F)C1)=O 58086,c1(C(=O)OC)c(C)ccc(NC(=O)NC2CCOCC2SC(C)(C)C)c1C 58087,Cc1ccc(CC(=O)NC(C)CC2CN(C(=O)C(C)CSC(F)(F)F)C2)cc1F 58088,C(=O)(C1CCCc2nccn21)N1CC(NC(c2ncc(OC)cn2)=O)(CO)C1 58089,c1(C(N(CCCOCCNC(C(C)C(F)F)=O)C)=O)n[nH]c2cccnc12 58090,c1(CO)ccnc(N2CCCC2)c1.C123COC(C1)(C2)C(=O)NC(C)(C)CNC3=O 58091,CC1CC(C(N2CC(CC(C)(C)CNC(=O)CC3CCCCC3)C2)=O)C(=O)O1 58092,CCCC(C(=O)N1CC(NC(=O)Cn2ccnc2C(C)C)C(C)C1)OC 58093,C1(CNC(=O)C2=CCOC2)CC2CCC(C1)N2C(C1CC12CCOCC2)=O 58094,C(=O)(CS(C)(=O)=O)NC(C)C(CO)NC(=O)CCC(=O)c1cccnc1 58095,c1(NC(C2CCN(C(c3cn[nH]c3)=O)CC2O)=O)cc(C(F)(F)F)cc(Br)c1 58096,C1(CNC(c2ccncc2F)c2n(CCC)nnn2)OCCOC1(C)C 58097,N1(C(CCC#CC)=O)CCCC12CCN(C(=O)C(C(C)C)NC(C)(C)C)CC2 58098,N#Cc1cc(Cl)c(C(=O)NC2CCC2NC(c2cc(Cl)c[nH]2)=O)s1 58099,c1(C(=O)NC(CNC(c2cn(CCC=C)nn2)=O)CC)noc2ncccc12 58100,c1(C(=O)NCC2N(C(Cc3c(C)nn(C)c3)=O)CC=C2)cccc2ccccc12 58101,C=CC1(NC(C2CC23CCN(C(=O)Cn2nccn2)C3)=O)CCOCC1 58102,N1(C(C2=CC(C)(C)C2)=O)CCC(C2CC2)(CNC(C2CC2c2ccccn2)=O)C1 58103,N1(C(C(C(C)C)c2scc(C)n2)=O)CCCCC(C(=O)N(C)C)C1 58104,C(=O)(CCCCCCCCC1CC1)N1CCN(C(CC(C=C)CC)=O)C(SC)C1 58105,c1(-n2c(CC(=O)NCC(C)(O)CNC(=O)C=C3CCC3)nnc2)cccc(F)c1 58106,c1(C(=O)NC(CCOC)CNC(C2CC=CCC2C)=O)c(OC)ccc(Cl)c1F 58107,CC(C)(C)C(O)C(=O)NC1CCCCCC1C(=O)NCC1CC1c1ccoc1 58108,c1(C(=O)NCC2CCN(C(C=CCCC)=O)C2)ccc(F)c(C(C)(C)F)c1 58109,N1(c2cccc(C)c2)N=C(C(=O)NC2CC2NC(c2ccns2)=O)CCC1=O 58110,c1(N(CCC)CCNC(c2coc(C)c2)=O)ncccc1[N+](=O)[O-] 58111,C12CCCCN1C2.CCCC(CNC(=NC)NCc1ccco1)OC 58112,C(=O)(C(C)(C)CS(N)(=O)=O)N1CCC(N(C(c2coc(C3CC3)n2)=O)CC)CC1 58113,c1(C(=O)NCC(CNC(C(C)=C2CCC2)=O)(C)C)n[nH]c2ccc([N+](=O)[O-])cc12 58114,C12(CNC(c3c(SC)cccn3)=O)CCC(CC1)N2C(=O)C(c1ccccc1)O 58115,CN1CCOCC1C(=O)NCC(C(N1CCOCC1C1(C)CC1)=O)C1CC1 58116,C1(NC(CN(C(C(C)C2CCC2)=O)C2CCC2)=O)CC2(CCCO2)C1 58117,N(C(=NCCCF)NC1CC1c1ccc(F)cc1)CC1([N+](=O)[O-])CC1 58118,c1(C(=O)NC(CC)CNC(=O)CC2CCCO2)ccc(C)c2c1CCCN2 58119,C1(C(=O)NCCNC(c2c(C)nc(NC3CC3)s2)=O)CCC(F)(F)CC1(C)C 58120,C1(CNC(CCc2ccc(OC)cc2)=O)C(C)CCCN1C(C1CCCCC1)=O 58121,C(N=c1[nH]c(=NC(C)c2ncc(C)cc2F)c2c(ncn2C)[nH]1)C1(SC)CC1 58122,S(=O)(=O)(c1c(Br)cccc1[N+](=O)[O-])N1C(C)CC(C(F)(F)F)C1 58123,C1(OC)CCN(C(C2CCOCCN2C(C2CCSCC2)=O)=O)C12CCC2 58124,C12(NC(C(COC)OC)=O)CCCC1N(C(c1cc(C)cc(Br)c1O)=O)CC2 58125,c1(C(=O)NC23C(NC(c4cn(C)nc4)=O)CC(CC2)C3)ccc2c(n1)OCCO2 58126,c1(N2CCC(N(C(C(C)Cc3cnc[nH]3)=O)C)C2)ncc2c(n1)COC2 58127,C1(C(C(=O)NC(C)C)N(C2CC2)Cc2cc(F)ccc2F)CC2(C1)OCCO2 58128,c1(CC(=O)NC(CC)CNC(=O)C(C)OC)cccc(C(F)(F)F)n1 58129,c1(C(=O)NC(C)C(c2ccc(OCC(F)(F)F)cc2)=O)ccc2c(c1)N(C)C(=O)C2 58130,C1(C2(O)CN(C(C3CN(C)C(=O)N3)=O)C2)(CNC(c2ccc(C)cn2)=O)CC1 58131,c1(CC)cccc(C(CC(C)C)OC(c2ccc(C(F)(F)F)cc2)=O)c1 58132,N1(C(C=C(C)C(F)F)=O)CCC2(CC1)CN(C(C1CN(C)CC1C(F)(F)F)=O)C2 58133,c1(OC)ccncc1C(=O)NCCC1(C)CCN(C(=O)C(C)Cc2cnco2)C1 58134,C1(CN2C(=O)CN(CC3C(C(N(C)C)=O)COC3)C2=O)C2CCC3(CNCC13)O2 58135,Cc1nc(C)c(CN2CCCCC2C(=O)NCCCS(=O)(=O)N(C)C)[nH]1 58136,c1(C(=O)NCCCCNC(C2(Cl)CC23CCC3)=O)cc2c(O)ccc(F)c2[nH]1 58137,CC1(C(=O)NCC23CC(NC(=O)Cn4ncccc4=O)(C2)C3)C=CCCC1 58138,C12CCCN(C1)C2=O.c1(OCC(=O)N(C(CC)CSC)C)cccc(C)c1 58139,C1(C2C(C)(C)C2CO)CCN(c2nnc(CNC(=O)CCC3CCC3)s2)CC1 58140,c1(NC(Cc2c(C)cccc2)=O)cccc(F)c1C(=O)Nc1ccnc(OCF)c1 58141,C12(C(N3CC4C(CNC(C(CCCC)C)=O)C4C3)=O)CC3CC(CC(C3)C1)C2 58142,CC1(C)C(NC(c2cccnc2C(F)F)=O)CCN1C(=O)C(F)C(F)(F)F 58143,C1(C(N(CC(O)C(F)(F)F)C)=O)CC2CCC(C1)N2C(C1CCC=CCC1)=O 58144,CCC(C(=O)NCc1ccc(CNC(C2CC3CC(=O)C2C3)=O)cc1F)C(C)C 58145,C(=O)(C(CO)C(F)(F)F)NC(CSC)C(=O)NOCCN(C)C 58146,c1(C(=O)NC2CCN(C(CCCSC)=O)C(C)C2)ccc2c(c1)CC(=O)NC2 58147,C1(NC(CCSCCC)=O)CCN(C(c2cnc(C3CC3)o2)=O)CC(O)C1 58148,C1(C(C)(C)C)CC(C(=O)NC(C(=O)N(CCCO)CCCO)C2CCCC2)C1 58149,c1(C(C)C(N2CCC(c3cnco3)C2)=O)ccc(F)cc1 58150,n1(CC(N)=O)cc(C(=O)NC2CCCC2NC(C2CCS2(=O)=O)=O)nn1 58151,C1(F)(C(N2CC3(CCN3C(=O)Cc3c(Cl)cccc3Cl)C2)=O)CCCC=C1F 58152,CC(C)CCC(C(=O)NC1CN(C2CC2)C1)NC(c1cnn(C2CC2)c1)=O 58153,C(=O)(C(C)(C)S(C)(=O)=O)NCCC(C)N(C)C(c1coc(N(C)C)n1)=O 58154,CS(=O)C1(CNC(C2C=CCN2C(c2cc(C(N)=O)co2)=O)=O)CC1 58155,c1(SC)cccc(C(N2CCCCC2CCNC(c2coc(Cl)n2)=O)=O)c1Cl 58156,N1(C(C2CC(C(=O)OC)C2)=O)CCCCC1CC(=O)NCCN(C)C 58157,CC12CCOC(C(=O)NC3CCN(C(c4scnc4C(C)(C)C)=O)CC3O)(C1)C2 58158,CCC(CC(=O)NC1CN(C(=O)C=Cc2cc(Cl)ccc2Cl)CC1OC)C(F)F 58159,N1(C(C(CC)OC2CC2)=O)CCC(CCCCNC(=O)CCOCC(C)C)CC1 58160,c1(C(=O)NC2CC3CN(C(C#CC(C)(C)O)=O)C2C3)cccn2cncc12 58161,C1(OC)CN(C)C(C)(C(=O)NCC2CN(C(=O)CCc3cccs3)CCC2C)C1 58162,C(=O)(CCCCC(C)(C)C)N1CC2CCC(N(C(Cc3cc(C)on3)=O)C)C2C1 58163,Cc1cccc(C(C)NC(c2cccc(Br)c2Cl)C)c1C 58164,N1(C(Cc2nc(C)sc2)=O)CCC(C)(C)C1C(N1CCC(O)C(C)C1)=O 58165,CC(CS(C)(=O)=O)C(=O)NCC1CN(C(=O)Cc2cocn2)CC(C)(C)C1 58166,c1(CC(=O)NC2CN(C(CC=C(C)C)=O)CC23CC3)cnc2n1CCCC2C 58167,N1(C(C(C(=C)Cl)(C)C)=O)CCC(CNC(=O)CC2CC3CCC2C3)C(C2CC2)C1 58168,Cc1cccc2c(C(=O)NCC3CCCN(C(C4CCS4(=O)=O)=O)CC3)coc12 58169,C=C=CC(C)C(=O)N1CCCCC1CN(C)C(c1ccc(N(C)C)nn1)=O 58170,C1(O)(C(=O)NCC(CCCC)NC(=O)C(N2C(C)CCC2C)C)CCC(C)CC1 58171,N1(C(C(CCOC)C)=O)CCC(C)(C)C(C(=O)Nc2ccc(F)nc2C)C1 58172,N1(C(c2cc(CC)ncc2)C(=O)NC(C)C)CCN(C2CC2)c2ccc(C)cc21 58173,N1(c2nc(N3CCOCC3)nc(N3CCC(=C)C3)n2)CCC(O)C(C)(C)C1 58174,C1(C(N2CCC(C(=O)OC)C2)=O)(NC(C2N(CCC)CCC2)=O)CCN(C)C1 58175,c1(C(=O)NC2CCC(NC(c3scc(OC)c3)=O)C2)ccncc1N(C)C 58176,CCC(C)(C(=O)NCCCCN(C)C(C1COC2COCC2O1)=O)C(N)=O 58177,c1(C(C(=O)NCCC(C)NC(c2cn(C)cn2)=O)C)c(F)cccc1F 58178,CC1(NC2(CNc3ccc(F)cc3)CCCCC2)CCC(C(=O)O)CC1 58179,C12(CNC(=O)CCc3cnc[nH]3)CC(CO1)N(C(=O)Cn1nnc(C3CC3)n1)C2 58180,c1(CCCNCC2(CC#C)CCOCC2)cc(OC)ccc1O 58181,c1(C(=O)OC)c(Br)cc(Br)c(NC(=O)C(=O)NC2CCC(N(C)C)C2)c1C 58182,N1(C(C2CCCCO2)=O)CCC2CN(C(=O)CCc3ccccc3F)CC2C1 58183,CS(=N)(=O)C1CN(C(=O)C(CCC2CC2)NC(C2CC23CCCCC3)=O)C1 58184,c1(C(N2CC3C(CNC(C4C(C(C)C)CCC4)=O)(C3)C2)=O)n[nH]c2c1COCC2 58185,C(=O)(CCC(C)(F)F)NCC(CNC(C1(CC)CC(F)(F)C1)=O)(C)C 58186,C1(C(=O)NC2(C(=O)NC(c3cccs3)C)CC(O)C2)CCC2(CCC2)O1 58187,c1(C(=O)NC(C2CN(C(C3(n4cc(Br)cn4)CC3)=O)C2)C)cnn(C)c1 58188,Cn1ccn2ncc(C(=O)NC3CC(CNC(c4cccnc4O)=O)C3(C)C)c12 58189,CCC(CCC(=O)N1CCC(C)(C#N)C1)NC(=O)CN1CC2CC2C1 58190,N1(C(Cc2cc(C)[nH]n2)=O)CCC(CCNC(=O)CCNC(=O)C=CCl)CC1C 58191,c1(C(N2C(CN(C(CN(CCC)C)=O)C)CCC2)=O)cc(F)c(OC)c(Cl)c1 58192,CC1CN(C(c2cnn(C)c2)=O)CCC1CNC(c1cnc(N(C)C)nc1)=O 58193,C1(CCC(=O)N(C2C3CN(C(C4(C)CCCOC4)=O)CC23)C)CCCCCC1 58194,C1(F)(C(=O)NCC2(F)CC(NC(CN(S(CC)(=O)=O)C)=O)C2)CC2(CCC2)C1 58195,N1(C(c2c(C)occ2)=O)CCC2(C)CN(C(C3C4CC5C(C4)C35)=O)CC12 58196,c1(C(N2C(C)C(NC(c3ncncc3Cl)=O)CC2)=O)cc2n(n1)CCCC2O 58197,N1(C(C2(C(=O)OC)CC2)=O)CC(C2(NC(=O)Cc3ccc(Cl)cc3OC)CC2)C1 58198,CC1CCC(CNC(=O)Cc2ccc(F)nc2)CN1C(c1cncn1C)=O 58199,C1(CC(=O)NCC(CNC(CC2(C=C)CCC2)=O)(C)O)CCOC1(C)C 58200,CC1(C)CN(C(C23CCC(CC2)OC3)=O)CCC1NC(=O)CCc1cnn[nH]1 58201,CCC(C)CC(C(=O)N(C)CCN(C)CCO)NC(c1ccc(OC)nn1)=O 58202,c1(C(=O)NCC2(O)CC(NC(C(c3ccccc3)C)=O)C2)cc[n+]([O-])cc1 58203,C12CCCN1C2=O.C1(=O)C(=O)N(C)C(C)CNN1.CC(C)C(C)=O 58204,c1(C(=O)NCC2(C(C)(C)O)CN(C(CC)=O)C2)cnc2c(Cl)cccn12 58205,N1(C(C2C(C(C)C)C2)=O)CCN(C(=O)Cc2c(Br)cnn2C)C(CCO)C1 58206,c1(N(CC=C)C)nnc(-c2[nH]nc(Cl)c2C(=O)O)n1CC1CSCCS1 58207,C12(NC(Cn3c(C)ncc3)=O)CCCC1(F)CN(C(C13CCC(F)(CO1)C3)=O)C2 58208,N1(CC)CCOC(CNC(=O)C(CNC(c2cc(C)oc2CC)=O)N(C)C)C1 58209,N1(C(C(C)c2cncs2)=O)CC(NC(c2cc3ccccn3c2)=O)CC12CCC2 58210,Cc1nc(CN(C)N2CCCC2C)cn(C)c1=O 58211,c1(C(C(=O)NCCN(C2CCCCC2)C(c2cnc(C)[nH]2)=O)O)ccccc1Cl 58212,C12(C(=O)NC(C)CC3CCN(C(C4(C)CCCC4O)=O)CC3)CCC(CC1)CC2 58213,N1(C(C2CCC(=O)C2)=O)CCCOC(CNc2nccc(CO)n2)C1 58214,C1(NC(CC2(C)OCCO2)=O)C2CN(CC(F)F)CC12.C12CCCN(C1)C2=O 58215,CC(C)C(O)C(C)C(=O)NCCN(C(=O)CCC(C)CN(C)C)C 58216,C1(C(C)C)CN(C(=O)CCC(=O)C2CC2)CC1C(=O)NC(C)C 58217,C1(CC(=O)NC(CNC(C(C)n2cncn2)=O)(C)C)COCCO1 58218,c1(C(=O)NCC(CC)(C)NC(c2c[nH]nc2OC)=O)cc(C)cc(Cl)c1 58219,C1(NC(c2cc(C)sn2)=O)CCC12CCN(C(c1cc(Cl)c(F)cc1Cl)=O)CC2 58220,CC1=NN(C)C(=O)C1CC(N1C2CCC1C(NC(c1cccc(F)c1Cl)=O)C2)=O 58221,C1(CN2CC(n3cc(CCC)nn3)C2)CCCN(C(C2(C3(C)CC3)CC2)=O)C1 58222,c1(C(=O)NCCC(CCNC(C(CC)C(C)(F)F)=O)C)cc(C)cc([N+](=O)[O-])c1 58223,c1(CNC(CC2CC(CC)C2)=O)cc[nH]c1C(=O)N(CCn1cccn1)C1CC1 58224,N1(C(C(C)SCC)=O)CC(CNC(=O)C(Cl)=CCl)(OC)C1 58225,CCCCCS(=O)(=O)CC(=O)NCC1CN(C)CCN1C(=O)CC1CCC(=O)C1 58226,c1(C(N2CCCC(Br)C2)=O)ccc(NCc2ccncc2Cl)cc1 58227,C1(C(N2CC(CNC(C(COC)C)=O)CC2(C)C)=O)CN2CCCN1CC2 58228,N1(c2n(CCC#N)c(-c3ccnc(O)c3)nn2)CC(CO)OC2(CCC2)C1 58229,c1(CCC(=O)N(C2CCN(C(C3CC34CCC4)=O)CC2)C)cccnc1Cl 58230,C1(COC)CCCCN(C(=O)CC(C)CNC(=O)CC(C)O)C1 58231,c1(C(=O)NC(C(C)NC(=O)CNC(=O)NC2CCOCC2)CO)cccnc1O 58232,Cc1ccc(O)c(CC(=O)N(C2C3CN(C(C4(C)CC5(CCC5)C4)=O)CC23)C)c1 58233,C12(C(=O)NCC(C3CC3)SC)CC(C)(CN1C(=O)CCn1ccnn1)C2 58234,N1(C(C=CC)=O)CCC2(CCCC2N(C)C(c2cnn3c2OCC3)=O)CC1 58235,C1(C(=O)NC(C#C)C(C)C)CN(C(c2ccc(C(N)=O)[nH]2)=O)CC1N(C)C 58236,N1(C(CCCOCCOC)=O)CCN(C(C2CCN2C2CCCC2)=O)CC1CF 58237,N1(C(Cc2cc(C)sc2C)=O)CCC(C2CN(C(c3ccns3)=O)C2)CC1 58238,c1(C(=O)NC23CC(NC(C(CCC)C)=O)(C2)C3)ccc(O)c(O)c1 58239,CC1CCC(NC(c2ccc(CO)c(Cl)c2)=O)CN1C(=O)CCC1CCC1 58240,C(=O)(C(F)C(C)(C)O)N1C(C)(CNC(c2nn(C)c(Br)c2)=O)CCC1 58241,[N-]=[N+]=Nc1ccccc1CCC(=O)NC1CC2CC1N(C(=O)CCC(N)=O)C2 58242,c1(CC)ncoc1C(=O)NCC1CC(CNC(=O)CC2(C)CC2)CO1 58243,Cc1cccc(Cl)c1C(=O)NC1CCCC1CNC(=O)C1=C(Cl)CC1 58244,Cn1nc(O)cc1C(=O)NCc1nccn1Cc1ccccn1 58245,Cc1cnc(C(=O)NC2CCC(C(=O)NCc3ccnn3C)C2)cc1C 58246,c1(C(N2CC3C(NC(CCCN(C)C)=O)(C3)C2)=O)cc(=O)n2nccc2[nH]1 58247,N1(C(C)=O)CCN(C(CC2CC2(Cl)Cl)C(=O)NC(C2CCCOC2)C)CC1 58248,c1(C(=O)NC2CCCC2CNC(C2(CO)CCCC2)=O)ccc(F)c(Br)c1 58249,C1(NC(c2ccc(OC)s2)=O)CCCC(NC(c2ccnc(C(F)F)c2)=O)CC1 58250,C1(CC(=O)NC2C(C)N(C(=O)CCn3cncn3)CCC2)CC2(CCC2)CCO1 58251,C(=O)(C1=Cc2ccccc2C1C)NCCN1CCCN(C(C(F)OC)=O)CC1 58252,CC1CCN(C(c2c[nH]nc2C(F)F)=O)CCN1C(=O)CCc1ccccc1F 58253,Cc1nc(C=CC(=O)NCC(=O)N(c2cc(F)cc(F)c2)CS(C)(=O)=O)[nH]c1C 58254,N1(C(c2c(CC)cco2)=O)C2CCC1C(C(=O)NCCCc1nc(C)no1)C2 58255,CC1(C)CC(CNC(=O)C2=CSCS2)CN1C(=O)COc1ccccc1 58256,Cc1cncc(C(=O)NC(C2CC2C(N2CCOC(CN=[N+]=[N-])C2)=O)C)n1 58257,S(=O)(=O)(c1cnc(Cl)nc1)N1C(C(=O)Nc2c(OC)cccc2)CC(O)C1 58258,C1(NC(c2cc(C(C)=O)on2)=O)CN(C(c2ncc(Cl)cc2Cl)=O)CC1(C)C 58259,c1(C(N2CCC(N(C(C3CCCO3)=O)CC)C2)=O)cc(C)n(C)c(=O)c1 58260,O=C1NC(=O)C2(CC(C(=O)NCCNC(=O)CCc3nnc(O)nc3O)C2)N1 58261,c1(OCC)cnc(C(=O)NC(C)CC2CN(C(=O)C(O)C3CCCC3)C2)c(Cl)c1 58262,CCCCC(C(=O)NCC)N.C(=O)(C(C)(O)C1CCC1)N.C12CN(C1)C(=O)C2=O 58263,c1(NC(CCC)CC)cc(NCCc2scnc2C)nc(C)n1 58264,C1(O)(CCNC(C(C)OC)=O)CCN(C(=O)C(F)CC2CC(F)(F)C2)CC1 58265,C1(NC(CCOCC#C)=O)CC2(CCCN(C(=O)C(CC(C)C)NC(C)=O)C2)C1 58266,C(=O)(CCCCC1CC1)NC(C1(C(=O)NCc2nnc(C)o2)CC1)C 58267,Cc1cc(=NC(=O)C(=O)NC2CC3CC2N(C(c2cc(Cl)ccc2N)=O)C3)[nH]o1 58268,CCCC(C(=O)N1CCC(CO)(NC(c2ccc(F)cc2CC)=O)C1)S(N)(=O)=O 58269,C1(NC(C2N(C(C)=O)CCOC2)=O)CC12CCN(C(=O)CN(C)S(N)(=O)=O)CC2 58270,c1(OC)c(F)cc(S(=O)(=O)N(C)CC2CCCC2(C)C)cc1[N+](=O)[O-] 58271,CC1(C)CC(O)(CC(N2CCC(CNC(c3cc(O)ncn3)=O)C2)=O)CO1 58272,C(=O)(C(C)(C)CCNC(=O)CC1CCCNC1=O)N(CCC(N)=O)C 58273,C1(C(N2CCC(=CC)C2)=O)CCN(C(=O)Nc2ccccc2O)CC1 58274,CC(=O)C(C)(C)CC(=O)NCC1(CO)CCCN(C(c2sccc2C#N)=O)C1 58275,c1(OC)nc(C(=O)OCC(=O)N(C)CC2CCCCC2)sc1C 58276,C12(C(N(c3cn(CC)nc3)C)=O)CCCC1CCN2C(c1nc(C)ccc1C)=O 58277,CCC(CC(C)C)C(=O)NCC1CCN(C(C2CCSCC2)=O)C(C)C1 58278,c1(C2CC(NC(=O)CC(C)F)C2)ccc2c(c1)NC2=O.C1(CC)(NCC2CC2)CC1 58279,C1(C(N(CC)CC)=O)CC12CN(C(C13CC(C1)C3)=O)C2 58280,C12(C(=O)NCC3CN(C(c4cc(C)c(C)s4)=O)CC3(F)F)CCCCN1CCC2 58281,C(CC(C)C)(C(=O)NC(C)CC(C)O)NC(c1ccc(C)n1C)=O 58282,c1(C(=O)NCC(CN(C(CCOCC)=O)C)C)occc1F 58283,C1(C(N2CC(CC)(CC)C2)=O)CN(C(=O)C=C(C)C(F)F)CC(C)(C)C1 58284,C1(CNC(=O)CNC(C2CCCC2)=O)CCCCC1NC(C1CC=CCC1)=O 58285,n1(C(COC)C)nc(-c2ccccc2)nc1CC(C)CC(C)C 58286,C1(F)(CNC(CC2CCC(C)C2)=O)CCN(C(=O)Cc2csc(C(C)C)n2)CC1 58287,c1(C(N(C2CC3CCC(C2)N3C(C2C3CCCC23)=O)C)=O)cc(Cl)cc(Cl)c1Cl 58288,c1(C(C)C)ccc(C(=O)NC2C3CN(C(C4CCC(=O)N4C)=O)CC23)cc1 58289,C1(C(=O)NC(CNC(C(N2CCOCC2)C)=O)(C)CO)CCC(F)(F)C1 58290,c1(C(N2CC(F)CC(NC(C=C(CC)C)=O)C2)=O)cccc2nccn12 58291,C1(C(=O)NC2(CNC(CC3C(C)C3)=O)CCCCCC2)CCn2cnnc2C1 58292,N1(C(CC2N(C(c3n(C)ccc3)=O)CCC2)=O)CCC2(CNC(=O)N2)C1 58293,N1(C(c2ncc(OC)cc2F)=O)CCC2(CCC(CNC(=O)CCSC)O2)CC1 58294,C1(C)(CNC(C2(F)CN(C(c3c(C)scn3)=O)C2)=O)CCCC1O 58295,Cc1ccc(Cl)cc1NNC(=O)NCC1COc2ccccc2O1 58296,c1(-c2c(OC)ccs2)cnc2cc(C(=O)Nc3ncc(C#N)s3)ccn12 58297,C(CCCC(CO)NC(=O)C(C)n1ccnc1)NC(c1c(OCC)cccc1)=O 58298,c1(OCCCOC(c2cccc(OC)c2)=O)cc(Br)c(N)cc1[N+](=O)[O-] 58299,c1(C(=O)NCCCN(C(c2cccc(C)c2C)=O)C(C)C)ccc2nc[nH]c2n1 58300,N1(C(C(CCC=C)(F)F)=O)CCC2(CC(NC(=O)COC3CCOCC3)CO2)C1 58301,C(c1ccc2c(c1)OCCO2)=CC(=O)OC(c1ncc(C)[nH]1)C1CC1 58302,C(CC(C(C)(C)C)NC(=O)CSS(C)(=O)=O)N(C)C(C1CN(C)CCN1C)=O 58303,C1(CNC(C2CC(C)(C)C2)=O)CN(C(C2CCCC2(F)F)=O)CCCO1 58304,Cc1noc(C)c1S(=O)(=O)N(C1CC2CC1CN2)C(C)CO 58305,C(=O)(CCC(CF)CF)N(C(C)CNC(C1CCOC1)=O)C 58306,CC(CC(F)(F)F)C(=O)N1CCCCC(N(C)C(c2snnc2C2CCC2)=O)C1 58307,c1(OC)c(NC(=O)Cc2csc(NC(c3cn(C)cn3)=O)n2)cccc1F 58308,CC(C)CC(O)C(=O)N1CC(CNC(C23CC(C2)C(C)O3)=O)C1 58309,c1(NC(c2nccc(-c3cc(C)nc(C)c3)c2)=O)csc2nccnc12 58310,N1(C(C2CCCOC2)=O)CCC2C(CCCN2C(c2ncoc2Br)=O)C1 58311,C12(NC(c3c(C)noc3)=O)CCC(C(=O)N(CCF)C3CC3)(CC1)C2 58312,c1(N2CCC(CC)C2)nc(N(CCC#N)C)c2ccc(C)cc2n1 58313,c1(C(N(CC)CC)=O)cnc2ccc(-c3cccc(F)c3F)cc2c1Cl 58314,Cc1ccc([N+](=O)[O-])cc1C(=O)NCC1CN(C(=O)CCOCC(F)F)CC1O 58315,C1(NC(CC(=O)OC)=O)CCN(C2CCN(C(=O)CCNC(=O)C=CCl)C2)CC1 58316,CC1CN(C(c2ccn(CC(F)F)n2)=O)CC1NC(c1cc(N)ccn1)=O 58317,N1(C(C(CC)(C)CO)=O)CC2(CC(NC(c3ncccc3Br)=O)CO2)C1 58318,N1(C(=O)NC2(F)CC2C(F)(F)F)CCC(F)(F)C(F)C1 58319,N12CCC(F)(CC1)CNC(=O)CC2=O.N1(CC)CCCC(CC(N)=O)CC1 58320,C(C(=O)N1CC2COCC2O1)(C1CC1)CNC(CCC(=O)NCC)=O 58321,c1(C(=O)O)ccc2c(c1)C(=O)N(CCN=[N+]=[N-])C2.C1(COC(C)=O)(C)CC1 58322,N#CC1CCC(NC(=O)C(O)C2CN(C(C3(O)CC3)=O)C2)CC1 58323,Cc1c(C(=O)NC(CO)C(=O)NCC(c2cnn(C)c2)C)cccc1C#N 58324,C(C(=O)Nn1cnn(C)c1=S)C1C(NC(C2C(C)CC=CC2)=O)CCC1 58325,CC(CNC(c1n[nH]c(=N)[nH]1)=O)CC(=O)N(C(C)C(C)(C)O)C 58326,N1(C(C(F)=CCC)=O)CCC(C)C1C(=O)N(CCCc1ccco1)C 58327,C1(C)(OCC(=O)N(C)CCN(C)C(=O)Nc2conc2C2CCC2)CCOCC1 58328,c1(C(=O)NCC2CC2CNC(=O)C2CC2)cc(F)cc(F)c1Br 58329,C1(NC(CCC2CC(C)C2)=O)CC(CNC(c2nn(C)cc2N)=O)C12CCC2 58330,C1(C(N2CC(C)(c3n(CC)ccc3)OCC2)=O)CCCCN(C)C1=O 58331,N1(C(C(C=CC)O)=O)CCCCC(C(=O)N(C(C)C(C)SC)C)C1 58332,N1(C(Cc2cnc(C)s2)=O)CCC(C)C(NC(c2ccc(-c3ccco3)o2)=O)C1 58333,Cc1cc(C(=O)NC2CCN(C(C3CC3C3(C)COC3)=O)C2)cc2c1CCC2 58334,CCC(C(F)(F)F)N(CCCNC(=O)CCCSCC(F)(F)F)C 58335,C(c1cccc(Cl)c1Cl)=CC(=O)NCCC(C)NC(=O)CC1NC(=O)NC1=O 58336,CC(C)C(C)(CNC(c1nscc1Br)=O)NC(C1C=CCC1)=O 58337,c1(C(=O)NC2CCC(NC(C(CSC)OC)=O)CC2)cncc2ccsc12 58338,CC(C)(C)C#CC(=O)N1CC(C(F)(F)F)OC(CNC(c2csc(CO)n2)=O)C1 58339,c1(OC)ccc2cccnc2c1COC(C1CCC2(CC2)C1)=O 58340,N1(C(c2c(CCC)n[nH]c2)=O)CCCCC(C(=O)NCCC(CCC)C2CC2)C1 58341,c1(C2(NC(C3C(C)=CCS3)=O)CC2)ccccc1[N+](=O)[O-] 58342,c1(OC)nc(=NCCN(C(=O)C(C)(O)C2CCOC2)C)[nH]c(C)c1F 58343,Cn1cnnc1CCCC(=O)NCC1(F)CC(CNC(=O)CC2CCCO2)C1 58344,CC1(C(N2CC(NC(=O)CCC3CCOC3)C(C(F)F)C2)=O)CCCCC1 58345,C1(NC(C2C(c3n(C)cnn3)CCC2)=O)CCN(C(c2csnc2Cl)=O)CC1 58346,N1(C(C(CC)N(C)C)=O)CC2(CCC2NC(c2cc(COC)cn2C)=O)C1 58347,CC(O)CCCNC(=O)CCNC(C1(C(C)(F)F)CC1)=O 58348,CC(C)(O)C(F)(F)C(=O)N1CC(CO)(CNC(C2CCCC(C(F)(F)F)C2)=O)C1 58349,C1(C(=O)Oc2c(C(=O)OC)oc(C)n2)CCCN(C(C)=O)C1=O 58350,c1(C(=O)NC2C(SC)CN(C(C3CNC(=O)C3)=O)C2)cc(SC)cc(Cl)c1 58351,C1(NC(CCc2cc(C)no2)=O)CC2C1CCN2C(C1CC2CC(=O)C1C2)=O 58352,N1(C(C(=O)N(C(Cc2cccc(C)c2)C)C)=O)CCC2(CCOC2)CC1 58353,CCC(F)(F)C(C)(C)C(=O)N1CCN(C(c2ccc(C(C)C)o2)=O)CC1C 58354,C1(C(C)C)CCOCCN1C(=O)COC1(C)CN(C(=O)C(C)Cn2ccnc2)C1 58355,c1(OC)ccc(C(N2CC(OC)CC2CNC(C2CC2C)=O)=O)cc1S(C)(=O)=O 58356,CN1CCN(C(=O)Cc2n[nH]c(=N)s2)CC1CNC(C1CN(C)CCO1)=O 58357,NS(=O)(=O)c1nc(C(N2CCC(NC(=O)CCF)C(CO)C2)=O)n2ccccc12 58358,CN1C(=O)c2ccccc2C1C(=O)N1CCCCC1CNC(=O)CCN1CCC1 58359,CC#CCCCC(=O)NCc1csc(C(=O)NC2(C)CCC(C)C2)c1 58360,O=C1Cc2ccc(CC(N3CCCC3c3c(F)cccc3Cl)=O)cc2N1 58361,S(=O)(=O)(c1cccc(C(F)F)c1)NC(=O)CC(C1Cc2ccccc2C1)C(=O)O 58362,N1(c2cc(CC)ncn2)CCCC(CO)(NC(=O)C=Cc2ccc(C)o2)C1 58363,C1(CNC(C(C)(N(C(=O)C=C2CCC2)C)C2CC2)=O)CCOC(C)(C)C1 58364,c1(C(N(C2CN(C(C(F)OC)=O)C2)C)=O)n[nH]c(C)c1C 58365,N1(C(COCCSC)=O)CCCC1CC(=O)NCCC12CC(CO1)C2 58366,N1(C(CN(C2CC2)CC)=O)CC2C3CCC(C2C1)N(C(C1CCC(C)S1)=O)C3 58367,CN1CC=C(C(=O)N2CSCC2C(=O)NCC2CC3(CCO2)CC3)C1 58368,C12(NC(C(CSC)OC)=O)CCC(CN(C(c3cc(CO)on3)=O)C1)C2 58369,c1(-c2cc(C(=O)NCC3(O)CN(CC=CCC)C3)sn2)ccc(Cl)cc1 58370,N1(CC=C(C)C)CCCC(C(=O)NC(CC2CC2)CO)C1 58371,c1(C(N(C(c2ccccn2)C)C)=O)ccc2c(=O)n(CCC(=O)O)c(O)nc2c1 58372,c1(OC)cc(C(=O)NC2CCCCC2NC(=O)C2=CCOC2)c2c(c1)CCO2 58373,c1(N2C(=O)C2)coc2cccc(F)c12.C1(CC=C(C)C)CCOC1=O 58374,N1(C(C=CC(C)(C)SC)=O)CC=CC(C(=O)N(C)Cc2sccc2C)C1 58375,c1(OCC)cncc(C(=O)N(C2(CNC(c3cc(C#N)cs3)=O)CC2)C)c1 58376,C(C)(CCC(=O)NC1CCC1CNC(C1(CCN(C)C)CC1)=O)OC 58377,N1(C(C(C)Oc2ccccc2)=O)CCCC1(C)CNC(=O)C(C1(O)CCCC1)F 58378,n1(CCC)ncc(C(=O)NCC(C2CCC2)NC(c2sccc2C2CC2)=O)c1C 58379,N1(C(c2c(OC)nsc2OC)=O)CCC(C)C(NC(c2cc(Cl)on2)=O)C1 58380,CC(C)(CF)C(=O)NC1CCCCC1NC(=O)C=CCOC(C)(C)C 58381,CCC(CN(C)C)CC(=O)NC1CN(C(c2cc(C(C)=O)on2)=O)C(C)(C)C1 58382,c1(C(=O)NC2CC(NC(c3cnnc(O)c3)=O)C23CCC3)cccc2sccc12 58383,N1(C(C2CCC(OC)CC2)=O)CCC(NC(=O)C#CC2(C(F)(F)F)CC2)C1(C)C 58384,N1(C(C2(C)CS(=O)(=O)C2)=O)CC(CNC(c2ccc(F)s2)=O)C2(CC2)C1 58385,C1(C(=O)NCCNc2cccc(F)c2)CC(O)CN1Cc1cc[nH]c1 58386,N1(C(CC2(NC(C)=O)CC2)=O)CC2CCN(C(=O)CC3NC(=O)NC3=O)C(C2)C1 58387,c1(C(N2CC(C)NC(=O)C2)=O)cnc2[nH]cc(-c3ccnn3C3COC3)c2c1 58388,N1(C(CC(C)(C)C)=O)C2CCC1C1CC1(NC(C1CC3CCC1O3)=O)C2 58389,C1(CNC(C2C(OC)CCC2)=O)CN(C(=O)C(C)CN(C)C)CC(C)(C)C1 58390,C1(CNC(=O)Nc2ccnc(F)c2F)CC(C2CC2)=NO1 58391,C=CC(CCC)CC(=O)N1CC(CCCCNC(C2CC(n3cnnc3)C2)=O)C1 58392,C1(C(=O)OC)(NC(c2cc(C)c(OC)c(Cl)c2)=O)CC(O)C12CCC2 58393,C(=O)(C#CC1CCOCC1)NCC1(OC)CCN(C(=O)COCCOC)CC1 58394,Cc1cc(C(=O)N(CCCNC(C2CC3(CCCO3)C2)=O)CCO)c(N)c(F)c1 58395,Cc1cnc(C(N2CC(C(N)=O)(CNC(C3CSCCS3)=O)C2)=O)cn1 58396,c1(C(N2CCCC2c2nc(COCC3CC3)no2)=O)cccn2ncnc12 58397,C1(C(N2CC(CC)C2)=O)CC(NC(=O)Cn2ncnn2)CCO1 58398,C(=O)(C(C(C)C)C(C)C)N1CCC(F)(CNC(C=Cc2cncc(C)c2)=O)C1 58399,c1(C(N2C(CCNC(c3cc(C)no3)=O)CCC2)=O)ccc(C)c(Br)c1 58400,c1(-c2cccc(C)c2C)cc(C(N2CCC(CO)C(F)(F)C2)=O)cc2[nH]ncc12 58401,N1(C(C(CCC)OC)=O)CCC2(CC1)CN(C(c1cc3c(ncn3C)[nH]1)=O)C2 58402,CN=c1nc(N2CCOCC(C3CCC3)C2)[nH]c(=NC2CCCCCCC2)[nH]1 58403,c1(C(=O)NCC2CCN(Cc3sccc3Br)C2)c(F)cccc1[N+](=O)[O-] 58404,C12CC3CCC1N3C(=O)C(C(=O)OC)NC2=O.n1(CC)nnc(C)c1CC 58405,c1(C(=O)NCC2CCN(C(c3ncc(F)cc3F)=O)C2)cc(F)cc(Br)c1F 58406,c1(C(=O)NC(C)Cc2ccco2)cc(Br)c(F)cn1 58407,C(=O)(CS(=O)(=O)CC(=O)NCC1CC(O)CN1C(=O)Cc1ccc(C)s1)OC 58408,C1(CNCCC2(CS(C)(=O)=O)CC2)CCN(C(C2CC(O)C2)=O)C1 58409,C1(NC(C(N2CCCCCC2)C)=O)CCN(c2ccncc2C#N)CC1O 58410,C1(NC(=O)CN(C(=O)CC(=O)NCC(C)C)CC)CC2CC(CO)CC2C1 58411,C1(CNC(CCOC)=O)CC(C(F)(F)F)CCN1C(=O)CC1CC=CCN1C 58412,Cc1cc(O)ccc1N(C)C(c1ccnc(C2(N)CC2)n1)=O 58413,c1(CC)nn(C)c(Cl)c1C(N1CC(CNC(=O)C(C)(O)C2CCC2)C(C)(C)C1)=O 58414,CCCCCCC(CC)NC(C1CC(CCNC(=O)CC(C)n2cccc2)C1)=O 58415,Cc1cc(C(N2CCC(C3CC3)C2CNC(=O)CC(C)(C)O)=O)cc2nc[nH]c12 58416,C=CCCC1C(=O)N1C.c1(CNC(=O)CN(CC(C)(C)C)C)ccc(C)cn1 58417,N1(CC(CNC(c2cc(C)sc2)c2nnnn2CCOC)(C)C)CCN(C)CC1 58418,c1(C(=O)NCC(CNC(c2nc(CC)[nH]n2)=O)C)cc(C)ccc1[N+](=O)[O-] 58419,C1(C(N(C2CN(C(C3CCN(C)CC3)=O)C2)C)=O)CCc2nn[nH]c2C1 58420,c1(C(=O)NCCNC(c2c(C(N)=O)cccc2)=O)cnc2nccn2c1 58421,c1(C(=O)NCC(CCNC(C(CC)COC)=O)O)ccc2cn(C)nc2c1 58422,C1(N(C(=O)CN2C(=O)CNC2=O)C)CCCN(C(c2cc(=O)n(C)cn2)=O)CC1 58423,c1(C(N2CC(CNC(c3nc(CC)oc3)=O)C3C2C3)=O)cc(C)ccc1[N+](=O)[O-] 58424,c1(SC)nc2ncnc(N3CCC(NC(C4CCC(F)C4)=O)C(F)C3)c2s1 58425,N1(C(c2cocn2)=O)CCCCC1CCC1CCCN1C(C1CC=CC(O)C1)=O 58426,N1(c2c(OC)cnc(Cl)n2)CCC2(CC1)OCCC2NC(=O)C(C)OC 58427,C1(C(N(C2CC(NC(CCSC)=O)C2)C)=O)CCOCC1C 58428,c1(C(N2C(C(=O)NCC3(O)CCCC3)CC(O)C2)=O)c(F)cncc1Br 58429,N1(C(CC(C)(C)O)=O)CCN(C(=O)CCCc2ccccn2)C(CO)C1 58430,c1(CCC(N2C(CN(C(C(C)SC(F)(F)F)=O)C)CCC2)=O)ccccc1Cl 58431,n1(CC(N2CC(C)(CNC(c3c(OC)nn(C)c3)=O)C2)=O)cc(C)c(O)nc1=O 58432,c1(C(=O)NC2CC(CCNC(c3[nH]c(=N)sc3)=O)C2)n[nH]c2c1CC(F)(F)CC2 58433,c1(OC)cc(C(=O)NC2CC3(C2)CC(NC(=O)C(C)CS(C)=O)C3)ccc1C 58434,C1(C(C)NC(Cc2c(C)nc[nH]2)=O)CCN(C(c2ncc(Br)cn2)=O)CC1 58435,C1(NC(CC=C)=O)CCC(CCNC(c2cn(C(C)C)nn2)=O)C1 58436,C1(C(=O)NCC(=O)NCC)CCC(O)CN1C(c1cn(CC)nc1C)=O 58437,N1(C(CC2CC(SC)C2)=O)CCC(C(=O)N(C)Cc2ncccn2)(C(C)C)C1 58438,CC(C)CC(C(=O)N1CCC(CN(C)C(C2(C(F)F)CCC2)=O)C1)C(N)=O 58439,C1(CC=C)(NC(C2C=CCC2)=O)CCN(C(c2ccc(C(N)=O)cn2)=O)C1 58440,c1(C(=O)NCC2(C(C)(C)C)CCN(C(CNC(CC)=O)=O)C2)sc(C)c(C)c1C 58441,N1(CC2(O)CN(C(C=C(C)C)=O)C2)CCN(C(c2cn(CCO)nn2)=O)CC1 58442,C1(NC(C2C(OC)CCC2)=O)COC2(C1)CN(C(c1cc(C)c(C)o1)=O)C2 58443,N1(C(c2cn(C)nc2Br)C(=O)N(CCC(=O)OCC)CC)CC=CCC(C)(C)C1 58444,c1(CN2C(CNC(=O)NCc3scc(C)c3)CCC2)cccc2c1OCC2 58445,n1(C(C)C)ncc(Cl)c1C(=O)NCCOC(c1cc(C)ccn1)(C)C 58446,C1(N(C(CNS(NC)(=O)=O)=O)C)CCN(C(=O)CC2CCCCN2C(C)=O)CC1 58447,C1(C(=O)NCC(CNC(c2cc(O)ccc2F)=O)O)CCC2(CCC2)O1 58448,C(C(F)(F)C(=O)NCCCCCNC(=O)CN1C(C)CCC1C)OC 58449,N12CCC(C)(C1)CNC2=O.CCCC(Cc1ccccc1)NS(=O)(=O)C(F)F 58450,C1(C(N2CC(OC)C2)=O)CCC=CC1NC(C1CCCN(C)C1)=O 58451,n1(-c2c(C(=O)NCCN(C)C(C3(C)C=CCC3)=O)cccc2)ccc([N+](=O)[O-])n1 58452,c1(NC(NOCCC#C)=O)ccc(OCCc2ccccc2)cc1 58453,Cc1ccnc(C(=O)N(C2CCN(C(c3ccnc(C4CC4)n3)=O)C2)CCO)n1 58454,c1(C(C)NC(=O)CC2CSC2)nocc1C(=O)NCC1CCC(C)C1 58455,C=CCN(CC=C)N1CCC(CC(=O)N(CCCO)C)CC1 58456,CC(C)(C#Cc1cn(C2CCC2)nn1)NC(CN(CCO)CC1(CO)CCCO1)=O 58457,C#CCCC(O)C(=O)N(C)CC1CCN(C(c2cccn2C)=O)C1 58458,Cc1nc(N2C3CCCC2CC(NC(=O)C2=C(Cl)CC2)C3)c2ccsc2n1 58459,C#CC1(O)CCN(C(C2CC(C)CN(C(C3CCCSC3C)=O)C2)=O)CC1 58460,C1(C#CC(=O)NC2CCOCC2C(=O)NC(C)COC(C)C)(CC)CC1 58461,Cc1ncn2ccc(C(N3CC(CNC(=O)C=CC(C)C)C4(CC4)C3)=O)cc12 58462,c1(C(=O)NC2CCCN(C(c3cc(CC)oc3C)=O)C2)cc(C)cc(Br)c1 58463,CC(C(=O)N(C(=O)C1=C(Cl)CC1)C1CCCC1)C(C)(F)F.C1C(=O)N1C(C)C 58464,CCCN=C(NCC1(OC)CCC1)NC1CCN(Cc2ccccc2)C1=O 58465,CC(C)C(CC1CCCCC1)C(=O)N1CC2CC(C1)C2NC(c1nc(Cl)cs1)=O 58466,C(CC(C)(C)C(=O)NCC1(F)CCN(C(C2(C)CC(C#N)C2)=O)CC1)OC 58467,c1(C(=O)NC(C(=O)NOCC2CCOC2)c2cn(C)nc2)ccc(=O)n(C)c1 58468,C1(=O)CCCC(C(=O)NC)N1.c1(C(C(=O)N)C)cccnc1 58469,C(=O)(C(C)CN(C(=O)C(C1CCOCC1)O)C)NC(COC)CO 58470,C(=O)(C(C)CC(F)F)NCC(CC)(C)NC(=O)C=CCOCc1ccccc1 58471,c1(C(C)=O)cc(C(=O)NCC2CCCC2NC(=O)C#CC(=O)N(C)C)oc1C 58472,c1(C(C(=O)NCC(O)CNC(C2(O)CCC2)=O)N(C)C)c(F)cccc1Cl 58473,C1(C(N(C2CCN(CC)CC2)C)=O)CC(C)CN(C(=O)CN2CC=CC2)C1 58474,N1(C(C(C)OCCCC)=O)CC2CCC2(CNC(=O)C=Cc2cnc(C)s2)C1 58475,c1(CC(=O)NCC(CC)NC(=O)COCC2CCC2)cn(C)nc1C 58476,C1(COC)(CO)CCN(C(=O)CC(C)(C)NC(=O)C=Cc2ccnn2C)CC1 58477,c1(C(N2C(C(N(CC(F)(F)F)C)=O)CC(F)(F)C2)=O)cc2ccc(Br)cc2s1 58478,N1(C(CC=C=C)=O)CCC2(NC(c3ccc(NC(C)=O)cc3)=O)CCCC12 58479,C=CC1(C2N=N2)CCC1.C12CC(C1)NC(=O)N(C(=O)CCC1CCCC1)C2 58480,C=CCC(CC(C)C)C(=O)N(C1CCN(C(C2CC3C=CC2C3)=O)C1)CC 58481,C1(CNC(C2(C)CC(C)C2)=O)CCN(C(=O)CCc2cncs2)C1(C)C 58482,C(=O)(C(F)(F)CCC1CC1)NC1CCC(CNC(c2ccnc(OCC)n2)=O)C1 58483,C=CC1(C(=O)NCc2cccnn2)CCN(C(=O)C=CC)CC1 58484,Cc1cc(CNC(=O)COC(=O)CCc2conc2C)cc(C)c1Cl 58485,C#Cc1ccc(OCC(=O)NCCN(C(c2conc2CC)=O)C2CC2)cc1 58486,Cc1cc(C(N2CCN(C3CC3)CC2C)C(=O)NCC2(C#N)CC2)cnc1C 58487,C(=O)(C(C)CNC(c1cnc(O)o1)=O)N(CCC)C1CC1 58488,n1(CC)ncc(Cl)c1C(=O)NC1CC1CNC(C1(O)CC(F)(F)C1)=O 58489,c1(OC)cc(C(=O)NC2CCCCC2NC(=O)CCC2CC2C)cc(C)n1 58490,C1(NC(c2nccc(C)c2)=O)CC2CCC(C1)N2C(=O)C1=CCCS1 58491,N1(C(=O)CC2CCCCS2(=O)=O)CCc2nc[nH]c2C12CCN(NC(C)=O)C2 58492,c1(C(=O)NC(CC)CN(C(=O)C(C)C2=CCCC2)C)oc2ccc(C)cc2c1C 58493,c1(C(=O)NCCCN(CCCNC(C2CC(O)C2)=O)C)n[nH]c2c1CCCC2 58494,CC1CCC=C1C(=O)N1CC(O)CC1(C)C(=O)NCc1cc(F)ccc1F 58495,CC1CN(C(CC2(C#N)CC2)C(=O)OC)CC(=O)N1.C1(C)CCOC1 58496,c12ccc(cc1)CNC2=O.C(=O)(C(O)CN(C)C)NC1(CC(=O)OC)CC1 58497,C12(c3cn(CC(CC)C)nn3)COC(CN1C(=O)CCc1cnc(O)[nH]1)C2 58498,c1(C(N(C2CN(C(=O)CCCN3C(=O)CNC3=O)C2)C)=O)n[nH]c2ccccc12 58499,N1(C(CCCCCNC(C(C)CN(C)C)=O)=O)CCCC(O)(C2CC2)C1 58500,c1(C(=O)NCCOCCNC(CS(CC)(=O)=O)=O)cc2sc(=O)n(C)c2s1 58501,C1(C(N2CC(C)C(CO)C2)=O)(NC(=O)C2=CCOCC2)CCC(C)(C)C1 58502,Cc1ccc(Cl)c(O)c1C(=O)NC1CCN(C(=O)C(C)CC(C)C)CC1F 58503,C(C)(CNC(C1CC(=O)N(C(C)(C)C)C1)=O)(C(C)C)NC(c1cnc(SC)[nH]1)=O 58504,C(=O)(C(C(C)(C)C)NC(=O)OC)N1CCC(F)(CNC(c2cn(CC)nc2)=O)C1 58505,CC1(C)OCC2CC12NC(C1(NC(c2ccnn2CCF)=O)CC(F)(F)C1)=O 58506,C1(CCCCCNC(=O)CNC(=O)OCC)(CNC(CC)=O)CCCC1.CCO 58507,CC(C)(CCNC(C1CCC(F)C1)=O)NC(=O)COCCN(C)C 58508,c1(C(=O)OC)ccc(SC(C)CCNC(=O)C(=O)NC2CCCC2)c(Br)c1 58509,c1(C(N2C(CNC(CSCC=C)=O)CC2)=O)ccc(C(=O)NCCOC)nc1C 58510,Cc1ccc(O)c(C)c1C(N1CC(OCCC(=O)NCC2CCC(C)(C)C2)C1)=O 58511,c1(C(=O)NC2CCCC(NC(C(C)(C)F)=O)C2)ccc2c(Br)cncc2c1 58512,N1(Cc2c(C(=O)OC)c(C)sc2)CC2CS(=O)(=O)CC2(C#N)C1 58513,CNS(=O)(=O)NCC(=O)N(C1CN(C(=O)Cn2nnc(-c3cccs3)n2)C1)C 58514,C12(C(N3CCN(C(=O)C(F)F)CC3c3cn[nH]c3)=O)CCC(N(C)C)(CC1)CC2 58515,C1(C(=O)NC(C#C)C(C)C)CCN(C(c2ccsc2OC)=O)C12CCC2 58516,N1(C(c2sccc2SC(F)F)=O)CC(NC(C2CCCC2O)=O)C2(CC2)C1 58517,C(=O)(C(C)(CC1CCC1)OC)NC(CN(C(c1cc(CCC)[nH]n1)=O)C)C 58518,CC1(C)C2CCC1(CC(N1CC(CNC(C3SCCCS3)=O)C1)=O)CC2 58519,CC(C(=O)NCC1CCN(C(C2CCCC2F)=O)C1)C(C)(F)F 58520,CCCC(C(=O)NC(C)CC)N1CCN(C(=O)C(C2CCCCC2)N)CC1 58521,C1(NC(c2c(C)snc2)=O)CC2CCC1(NC(c1cnn(C3CC3)c1Cl)=O)C2 58522,c1(C(=O)NC(CCNC(C2N(CC)CCOC2)=O)C)ncc(Br)cc1F 58523,c1(C(=O)Nc2cncc(C3CC3)n2)ccc(=O)n2c1COCC2 58524,C1(C)(CNC(C(CN(C)C)O)=O)CN(C(=O)C(C)(C)NS(C)(=O)=O)CCO1 58525,C=C(Cl)CC(C(=O)N1CC(C(=O)OC)CC(C)C1)NC(=O)C(C)N=[N+]=[N-] 58526,N1(C(CC2(C)CCC2)=O)CCN(C(c2cc(Br)cnc2O)=O)CC2(CC2)C1 58527,C(=O)(C1=CCN(C(c2cn(C)c(=O)cn2)=O)C1)NC1CC2CC(OC)C2C1 58528,N1(C(CN(CCOC)C)=O)CCCC2CN(C(=O)C(CCSC)N(C)C)CCC12 58529,c1(C(C(=O)NCCN(C(=O)CCc2cnoc2)CC(C)O)O)ccc(Cl)cc1 58530,C1(COC)(CO)CCCN1OC.C12CC(CN1C(=O)C=CCN(C)C)CNC2=O 58531,N1(C(C=Cc2cnc(C)nc2O)=O)CC2OCCN(C(=O)C(C)N(C)C)C2C1 58532,c1(CC)nn(C2CC2)cc1C(=O)NCCNC(c1cncnc1)=O 58533,c1(OCC)ccc(C(=O)NC(CNC(c2cscc2CC)=O)CO)cc1C 58534,Cc1nc2ccccc2cc1C(=O)NC1CCCC(NC(C2CC(C#N)C2)=O)C1 58535,N1(C(c2cc(C(CC)C)no2)=O)CC2CCC2(CNC(c2ccc(OC)o2)=O)C1 58536,C=C(C)CCCC(=O)NCC(C)N(C)C(c1ccn(COC)n1)=O 58537,Cc1ccc(C(=O)NCC2(O)CCCN(C(c3nnc(O)nc3O)=O)C2)c(N)n1 58538,N1(C(CC(CCC)CC)=O)CC(CO)C2(C1)CN(C(c1ncccc1N)=O)C2 58539,C1(C(N2CCC(COC)(NC(c3cnc(C(F)F)s3)=O)C2)=O)CCC(C)=C(C)C1 58540,C(CCC(C)(C)C(=O)N1CCC(O)(C=C)C1)NC(C(C=C)CC)=O.C(=O)OC 58541,C1(c2nnnn2C2CCC2)(NC(c2ccc3c(c2)OCO3)C)CCCC(C2CC2)C1 58542,c1(C(=O)NC2CC3(C(NC(c4occ(C)c4)=O)C3)C2)ccc2c(c1)C(=O)CCC2 58543,CCC(C)(CNC(C1CC(F)CN1C)=O)C(=O)NCCCc1cn[nH]c1 58544,N1(C(c2c(C)cnnc2)=O)C(C(=O)NC2CCCCNC2=O)CCC12CC2 58545,C1(N(C2CCN(C(=O)Cn3cncn3)C2)CCO)CCCN(c2cn[nH]c2)C1=O 58546,C=CC1CN(C(C2CC(OC)C2)=O)CC1NC(=O)CC1CCCOC1 58547,CC1(C)C(NC(C2CCCCC2O)=O)CCN1c1ccnc(-c2nccs2)n1 58548,C1(NC(=NCCC)NCC(c2ccccc2)OC)CCc2cnn(C(C)C)c2C1 58549,C(C)(c1ccc2ccccc2n1)=CC(C#C)(O)CCCC 58550,C1(CNC(c2cn(CC=C)nn2)=O)CN(C(C2(C(=O)NC)CC2)=O)CCC1C 58551,C#CC1(C)CCCN1C(c1cc(=N)[nH]c(Cl)n1)=O 58552,N1(C(C2(CCCC)CC2)=O)CCC2C(CCN2C(C2C=CCS2)=O)C1 58553,C1(C(N(C2CCN(C(c3cccc(O)n3)=O)CC2)C)=O)C2CCCOC12 58554,C=C=CC(C)C(=O)NCCCC1CCCN1C(=O)CCOCCN(CCCCC)C 58555,C12(NC(C(c3ccccc3)C)=O)CC(C1)N(C(=O)C(C)N1CCCC1)C2 58556,C(=O)(C1Cc2ccc(F)cc21)NCC1CC(N)(C[Si](C)(C)C)C1 58557,C=CC(C)(O)C(=O)NCCCCC(=O)NC.C1(C)CC(=O)N1 58558,N1(C(c2c(F)ccc(OC)n2)=O)CCCCCC(NC(=O)Cc2occc2C)C1 58559,c1(C(=O)Nc2ccc(C(=O)NCc3n(C)ccc3)cn2)c(F)cc(O)cc1F 58560,c1(CC(=O)NC(C)C)nc2c(s1)CCN(Cc1ccc(C#N)c(F)c1)C2 58561,Cc1nccn1CCCNC(c1nnnn1C1(C)CC1)C1CCCCC1 58562,CC(C)CC(CNC(c1cc(CO)[nH]n1)=O)C(=O)NC1CC(CO)C1 58563,c1(C(=O)NCC(c2ccccc2)CNC(CC=C)=O)ccc2c(c1)C(=O)NC2=O 58564,N1(C(C(C)CN)=O)CCCC2(C(=O)NCc3ccccc3)CC2C1 58565,FCCCN=C(NC1CC2(CCC2)C12CCC2)N1CCC(n2cccc2)CC1 58566,C(=O)(C(C)C(C)NC(=O)CC1CN(C(=O)CCc2cncn2C)CC1C)OC 58567,C1(C(=O)NCCC(=C)CO)CC(NC(=O)CCC=C(C)C)C12CCC2 58568,c1(C(N(CC(CNC(c2c(C)coc2C2CC2)=O)C)C)=O)ccc2c(c1)CCN2 58569,C1(CC(=O)OC2(C)CCC2)CN(CC(=O)N(C2CCC2)CCNCC)C(C)(C)C1 58570,c1(CCC(=O)NCC2C(NC(c3nnn(C)n3)=O)C2)ccc(Cl)cc1Cl 58571,CC1(C(=O)NC2(C(=O)N(C)C)CCCCC2)CCCNC1 58572,Cc1nc(N(C)CC2CCCN(C(c3ccco3)=O)C2)cc2nncn12 58573,C1(OC)(CNC(=O)C=C(C)Cl)CN(C(=O)CCc2nc(C)no2)C1 58574,c1(CC(=O)N(C(CN(C(C=CCOC)=O)C)C)C)cccc(OC(F)F)c1 58575,C(=O)(CCCS(C)(=O)=O)NCCOC(C)(C)CNC(c1cc(C2CCC2)no1)=O 58576,N1(C(C(C)SCCCC)=O)CC2C(C(N3CCC(c4ncco4)C3)=O)C2C1 58577,C12(NC(C3C(CNC(CNC(C)=O)=O)C3)=O)CC1COC2(C)C 58578,c1(C(=O)NC2C(C(=O)NC(CCCCC)C)OCC2)cc(C#N)n(C)n1 58579,NS(=O)(=O)c1cncc(C(=O)NC2CCCN(C(=O)C=C3CCCC3)C2)c1 58580,CC(CCCNC(=O)CNC(=O)C(C)(C)F)NC(=O)NCc1ccccc1 58581,C1(C(=O)NC(c2ncccn2)C)CCC(NC(c2cc(Cl)ccn2)=O)CO1 58582,c1(C(=O)NCC2CCN(C(c3occ(C)c3C)=O)CC2C)ccc(Cl)c(N)c1Cl 58583,N1(C(C(C)O)=O)CCCC(CNC(=O)CC2COC(C)(C)C2)C1 58584,c1(C(=O)NC(CN(C(CS(=O)(=O)NCC)=O)C)(C)C)ccn2nccc2n1 58585,Cn1ncc2cc(C(=O)NC3CCCOC3CN)cc(O)c12 58586,c1(C(N2CC(O)CC(NC(CSCC)=O)C2)=O)c(F)ccc(OC)c1OC 58587,N1(C(c2ncn(CC)c2)=O)CCCN(C(C2(C)CC2(C)C)=O)CC1C(C)C 58588,C12(NC(=O)C3=COCCC3)CCCCCC1N(C(C1C=CCC1)=O)CC2 58589,c1(C(=O)NC2C(CNC(c3occ(C(N)=O)c3)=O)CCCC2)c(O)cccc1Cl 58590,N1(C(c2c(C)cccc2)=O)CCN(C(C2(C(F)F)CCCO2)=O)CC1C(F)F 58591,C1(F)(CNC(C(C2CCC2)OC)=O)CCCN(C(=O)C(C)(C)c2ccno2)CC1 58592,Nc1cnccc1C(=O)NC1CCC(NC(c2ccns2)=O)CC1 58593,c1(OC)ccc(CCCCNC(=O)NC2CCC(c3nc(C)no3)CC2)cc1 58594,CC(C)CCCCC(=O)N1CCC(C2CCCN2C(C2CC(C)(O)C2)=O)C1 58595,C1(C)(NC(c2cc(C)sc2C)=O)CCCN(C(C2CCCCC2(F)F)=O)C1 58596,c1(C(N2C3CC(CNC(CSCCOC)=O)C(C3)C2)=O)cc2ccccn2c1 58597,c1(C(=O)NCCN(CCC)C(C2(F)CCOC2C)=O)cn2ccnc2s1 58598,Cn1nc(C(N2CCCC2CNC(=O)CC2C=CCCC2)=O)cc1F 58599,C(=O)(CC(C)(C)C(F)F)N1CC2(CC)CC1(CNC(=O)C#CC(=O)NC)C2 58600,C1(NC(=O)Cc2sccc2Cl)CC2CC(NC(C3C4CNC(=O)C34)=O)C1C2 58601,c1(C(=O)NCC(CNC(c2c(C)cco2)=O)(C)O)noc2c(F)cccc12 58602,N1(Cc2nc(CCOCC)sc2)CC2C(=O)N(C)C(=O)C2C1 58603,Cc1[nH]nc(C(F)(F)F)c1C(=O)NCC1CN(C(=O)CC2CC2C2CC2)CCO1 58604,c1(C(N2C(CNC(c3[nH]cc(CC)c3)=O)CCCCC2)=O)cccc2c1CCC2 58605,c1(CNC(c2cscc2-c2ccccc2OCc2ccco2)=O)ccnc(F)c1 58606,C12(CC)COC(=O)N1CCN(C(C1CCN(Cc3ccc(F)cn3)CC1)=O)C2 58607,C1(NC(CC(C)(C)OC)=O)CCN(C(=O)C(C2CCOCC2)C)CC1O 58608,N1(C(Cc2c(CC)cccc2)=O)CC2CC1CCC2NC(c1cnsc1)=O 58609,C1(COC)(NC(=O)C=C(C)C2CC2)CCN(C(=O)C(C)Cc2cnco2)C1 58610,C(C1CCCCC1)=CC(=O)NC1C(NC(CCc2cc(C)[nH]n2)=O)CC1 58611,c1(Cc2onc(C(=O)NCCC(C)NC(=O)CCCF)n2)ccc(Cl)cc1 58612,N(C(=NCCC(C)(C)C#N)NCC=C)CC1CCCC(CC)C1 58613,c1(C(=O)NC(C2CCCN2C(c2cc(F)ccc2N)=O)C)ccc(S(C)(=O)=O)o1 58614,C1(N(C(C=CCN(C)CC)=O)C)CCN(C(c2c(C(F)(F)F)coc2C)=O)CC1 58615,CCCCC(F)C(=O)NC1(CCC(=O)N(C)Cc2c(C)noc2C)CCCC1 58616,S(=O)(=O)(c1ccc(NC2CCOC3(CCCC3)C2)c(F)c1)NCC(C)CO 58617,CC1CC2(CC(C(=O)NC(C3CCCN3C(=O)CC(C)(C)C3CC3)(C)C)C2)C1 58618,C1(NC(c2cc(C)sc2C)=O)CCC12CCN(C(c1ccc(O)cc1)=O)CC2 58619,C1(NC(C(C)NC(C(=Cc2ccco2)C)=O)=O)COC2(CCC2)C1 58620,CC1(C)CCCC(O)(C(N2CCC2CNC(=O)CC2CC2(C)C)=O)CC1 58621,CC1(C)C(CC(=O)OCC(=O)NCC(=O)N(C2CC2)Cc2ccco2)CC1O 58622,CC1(C)COC(C(=O)NC2CCCC(CNC(c3cc(Cl)ccc3Cl)=O)C2)CO1 58623,C1(C(N2C(CNC(c3cccc(O)c3)=O)CCC2)=O)C2CCC1(c1cscn1)C2 58624,C1(NC(c2n(C)nnc2)=O)CCCC12CCN(C(c1cc(F)c(Br)cc1F)=O)C2 58625,Cc1[nH]c(C#N)cc1C(=O)NC1COCCC1NC(c1ccc(F)c(CO)c1)=O 58626,C(CCNC(=O)Cc1cn(C)cn1)(C(C)C)NC(COCC(=C)C)=O 58627,C(=O)(CC(CN(CC(C)COC)Cc1cc(C2CCOCC2)no1)OC)OCC 58628,C(=O)(C(C)CC(F)(F)F)NCC1(C(C)NC(=O)Cc2ccn(C)c2)CC1 58629,C(CCC(O)C(=O)NCc1ncco1)NC(c1cc(CC)nn1C)=O 58630,C(=O)(CCCC(=O)N1CC(N(C)C(C2CCC(C)O2)=O)C(O)C1)N(CC)CC 58631,CN1CC(C)(C)CC1C(=O)NC1CC=C(C(=O)NCCCC(C)(C)CO)C1 58632,c1(OC)cc(OCOC)ccc1NC(C1CC(NCC(N)=O)C1N)=O 58633,N1(C(C2CC(SC)C2)=O)CCC(NC(C2CN3CCC2CC3)=O)C(O)C1 58634,N1(C(c2c(C#C)cnn2C)=O)CCC2(CCCN2C(C23CCCC2CCC3)=O)C1 58635,C1(O)(C(=O)NCC2N(C(c3cc(F)cs3)=O)CC(C)(C)OC2)CN2CCC1CC2 58636,c1(NC(C(C)NC(=O)COC(C)(C)C)=O)c(O)nn(C)c1C(F)(F)F 58637,c1(OC)cc(CNC(=O)NC(C)(C)CC=CC(=O)O)cc(I)c1OC 58638,c1(C(c2n(C(CC)C)nnn2)NCCc2nccs2)cc(Cl)ccn1 58639,C1(C(=O)NC(CC2CC2)=O)CC(=O)N(C2CN(C)C2)C1.C1(N(C)C)(COC)CC1 58640,CCCC(C#N)C(=O)NC(C(=O)NOC(C)(C)C(=O)OC)C1(C)CC1 58641,c1(N2CCCC(OCCC)C2)nc(=N)[nH]c(=NCCc2ccc(SCC)cc2)[nH]1 58642,CC1CC=C(C(=O)N2CCC(F)CC2C(=O)NOCCF)CC1 58643,C(=O)(C(CC(C)C)C(C)C)N(C(CC)CNC(c1nnn2c1CSCC2)=O)C 58644,C1(NC(c2c(CC)n(C)nn2)=O)CN(C(c2cnn(C)c2F)=O)CC12CC2 58645,C#Cc1ccc(C(=O)NC2CC3CCC(C2)N3C(=O)CC2CC2(C)C)cc1F 58646,C1(F)(C(=O)NCCN(C)C(c2cncc(-n3cncn3)n2)=O)CCOCC1 58647,Cc1ccc(C(=O)N(CCC(=O)NC(C)CCC2CCCO2)C(C)C)c(O)c1 58648,N1(C(C2C(COC)C2)=O)CC2(CO)CC1(CNC(=O)CN(c1cnccn1)C)C2 58649,C1(C)C(C)CCN1C(C1CC12CC2)=O.C1(C)(C(=O)OCC)CC1C 58650,C1(C(=O)OC)CN(C(=O)NCCCN2CC3CC3C2)C2(CCC2)C1 58651,Cc1cccc2c1CC(C(=O)NC1COCCN(C(=O)C=CSc3nc[nH]n3)C1)O2 58652,N1(CC)CCCC1CC(=O)N(CC(C)(C)CNC(=O)C=Cc1ncc[nH]1)C 58653,C(=O)(CCC(=O)NCCC1CC(NC(c2occc2Cl)=O)C1)NCC 58654,c1(OC)coc(C(=O)NCC2(C)CCCN2C(=O)COCCN(C)C)cc1=O 58655,C1(OC)CCCCC1C(=O)NC1(c2ccccc2)CN(C(C2CC(=O)N(C)C2)=O)C1 58656,C1(C(=O)NC(CO)C(N2CC3CC3(CO)C2)=O)CC2(CCCO2)C1 58657,C1(O)(CCNC(c2c(C)nsc2)=O)CCN(C(=O)C(C)Cc2cnc[nH]2)CC1 58658,C(=O)(CCCC(C)(C)C#N)N1CCN(C(C(OCC)OCC)=O)CC(CO)C1 58659,c1(OC)ccc(C(=O)NC2CCN(C(c3cnccn3)=O)C2C(C)(C)C)c(O)c1 58660,C1(C(=O)NCCN(C(CNC(c2cccc(C)c2)=O)=O)C)CCC2(CCOC2)O1 58661,C1(C(N(CCC(C)NC(c2ccc(C(C)(C)C)cn2)=O)C)=O)CC2(C1)CC21CC1 58662,N1(C(C(CSC)C)=O)CCN(C(C2CCC(=O)N2C(C)C)=O)CC1c1cn[nH]c1 58663,C12(C(N(C3CCCCCC3)CCNC(=O)CCc3ccco3)=O)CCC(CO1)C2 58664,N1(CCc2cn(NC(CC3CCC(C)(CC)O3)=O)nn2)CCC2(CC1)OCCO2 58665,c1(CNC(C2(CN(C)C)CC2)=O)ccc(CNC(=O)CC2(O)CCCC2)cc1F 58666,C1(C(=O)OC(C)(C)C)CC(OC)C12CCOCC2.c1(OC)ccc2cc1-2 58667,C1(c2ccccc2)CCCC1.c1(CC(C)N)ncn(C)n1 58668,N1(C(C2C(CC)C2)=O)CC2CCN(C(C3C(C=C(C)C)C3(C)C)=O)CCC2C1 58669,C1(CN2CCC(NC(COC(CC)C)=O)C2)CCOC(C)C1 58670,c1(C(=O)NCC2CC(NC(C3C(CCC)CCC3)=O)C2)ccc(N)cc1 58671,c1(C(=O)NC2CC(CNC(C3(C(=O)OC)CCCO3)=O)C2)nccnc1Cl 58672,c1(OCC=C)ccc(C(N2CC(CN(C)C(C3(C)CCCO3)=O)C2)=O)cc1OC 58673,CC1(CNC(C2CC2C)=O)CCN(Cc2cccnc2Cl)CC1 58674,C#Cc1ccccc1CNC(C1C2CC1N(C(=O)C(C)(C)O)C2)=O 58675,c1(N(c2ccccc2F)CCNC(C(CC)N(C)C)=O)nc(C2CC2)nc(=N)[nH]1 58676,c1(C(N2C3C(CNC(c4c(C(C)C)ncs4)=O)C(C3)C2)=O)ccn2c1CSCC2 58677,N1(C(c2c(C)cc[nH]2)=O)CCC2C(CCN2C(c2cc(F)c(F)c(Cl)c2)=O)C1 58678,C1(=CC(=O)NC2CCN(C(c3ccc(F)s3)=O)C2)CN2CCC1CC2 58679,C12(CNC(c3ccn(CCNC(C(CCC)F)=O)c3)=O)CCCN(CC1)C2 58680,Cc1nn(CC(=O)NC2CCN(C(=O)COCCCF)C2C)c(C)c1Cl 58681,CC1CC(NC(=O)C(=O)NC2CC2)CN1C(c1cnc(C(F)F)nc1)=O 58682,CC(C)C(C(F)(F)F)NC(C1COCC1NC(c1c[nH]c(=N)o1)=O)=O 58683,N1(C(CNC(=O)OC)=O)CCC(C(=O)NCC23CCCC2C3)C1(C)C 58684,c1(C(N2C(CCN(C(=O)CC(C)(C)O)C)CCCC2)=O)cc(Cl)c2c(c1)OCO2 58685,N1(CC)CCN(CC(=O)NCC(CO)NC(C2(OCC)CCOC2)=O)C(=O)C1=O 58686,N1(C(C(Cc2ccoc2)NC(c2ncc(F)cc2F)=O)=O)CC2CC1CC2O 58687,C1(F)(CNC(Cc2ccc(C)s2)=O)CCN(C(C2CCN(C)C2)=O)C1 58688,N(C1CCCn2ncnc21)C(C(CC=CC)NC(c1cnn(C(C)C)c1)=O)=O 58689,C1(N(C(Cc2c(C)non2)=O)CCO)CCCN(C(=O)C(F)CC2CC2)C1 58690,c1(C(=O)NCC2(F)CC(NC(C(C(CC)C)O)=O)C2)c(C)ccc2ncccc12 58691,Cc1nnc(CCCC(=O)N(CC(O)CNC(c2ccc(CO)cn2)=O)C)n1C 58692,Cc1nc(CC(=O)NC(CO)C(C)NC(=O)C(C)Sc2nncn2C)n[nH]1 58693,C(=O)(CC(C)C(F)F)NCCN(C(C=CCC)=O)CCOCCO 58694,CN1CCC(n2cc(NC(c3nnnn3C3CC=CCC3)C3(CF)CC3)cn2)CC1 58695,N1(C(C2CNC(=O)N2)=O)CC(NC(c2csc3cncn23)=O)C2CCCCC12 58696,C(=O)(CC(C)(C)C(C)(F)F)NCCC1(NC(C2N(CCC)CCC2)=O)CC1 58697,c1(C(N(CCOCCCNC(Cc2scc(C)c2)=O)C)=O)ccc2ncnn2c1 58698,c1(COC(C2C(C(=O)OC)CCO2)=O)cnn2cc(OC)ccc12 58699,N1(C(c2occ(C)c2)=O)CC(NC(=O)C(c2ccccc2)C)C2(CC2)C1 58700,C1(COC)CCCCN1C(=O)C(=O)NC1CC1NC(=O)OC(C)(C)C 58701,C(=O)(C#CC1CCC1)NC(C(=O)NCC(CC)C(C)C)COC 58702,C1(C(C)CNC(Cc2cc(C)[nH]n2)=O)CCN(c2nnc(C3CC3)s2)CC1 58703,c1(C(N(CC(O)CN(C)C(C2CCC2)=O)C)=O)ccc2nn[nH]c2c1 58704,CC(CC(C)NC(c1csc(Cc2ccccc2)n1)=O)NC(=O)C(F)(F)C1CC1 58705,N1(C(c2ccc(C=C)cc2)C(=O)NCCC#N)c2ccccc2C(C)C1C 58706,C(=O)(C=C1SCC(=O)N1C)NCCC1CC(NC(c2c(OC)ccc(Cl)c2)=O)C1 58707,C1(CNC(CSCCC)=O)CCCCCN1C(c1oc(CC2CC2)nc1C)=O 58708,N1(C(CCCCCN(C)C)=O)CC2CC(NC(=O)CCc3cnccn3)CC1C2 58709,c1(N2CCC(NC(C3C(=C)C3)=O)C2)nc(C(C)CC)ccc1C#N 58710,C1(C(=O)NCCCOCC#C)CCC2CCC1N2C(c1cccc(=O)o1)=O 58711,C1(C(C)NC(=O)C=CC2CCC2)CN(C(C2(C(F)F)CC2)=O)CCO1 58712,c1(C(=O)NCCN(C(=O)CC(n2ccnn2)C2CC2)CCOC)ccc(Cl)cc1 58713,c1(CN(C2CCN(C(c3c(C)cccc3)=O)C2)C)ccc(C)c(Cl)c1 58714,C(=O)(C(CNC(C1CC(N2CCCC2)C1)=O)Cc1ccc(O)cc1)OCC 58715,N1(C(C2(CCOC)CCCC2)=O)CCC(CNC(=O)CC2COCCO2)(OC)C1 58716,c1(C(N(CCN(C(c2n(CC#C)cnn2)=O)C)C)=O)cc(C(N)=O)ccc1F 58717,N1(C(C2N(CC)CCC2)=O)CCC(CC(=O)NC2CCC(=O)N(C)C2)C1(C)C 58718,CN1CC(C(=O)NCC2CN(C(c3cnn(CCF)c3)=O)C2)CC1=O 58719,N1(C(CC2N(C(C)=O)CCC2)=O)CCOC(CNC(c2cnn(CCF)c2)=O)C1 58720,CSC1=C(C(=O)NCC2CCC(NC(C3CCC(C(C)C)CC3)=O)C2)CCCC1 58721,Cc1cc(C(=O)NCC(C)(O)CNC(=O)Cc2ccn(C)n2)ccc1C(N)=O 58722,C1(C(=O)NCCc2n[nH]cc2C(=O)NC(C)C(C)SC2CC2)(CC)CCOC1 58723,C(=O)(C(C(C)NC(=O)CCc1ncnn1C)C(C)C)NCc1nccc(C)c1F 58724,N1(C(C2CC=C(C)CC2)=O)CC2(CCC2NC(c2cc(Cl)no2)=O)C1 58725,Cc1cccc(O)c1C(N1CC(N(C(=O)C(C2CCOCC2)C)C)C(C)(C)C1)=O 58726,S(=O)(=O)(c1ccc(NC2CCCC(SC)C2)c(Br)c1)NC(CC)(CC)C1CCC1 58727,C(CC(=O)NCCN(C(=O)C(C1(C)CC1)NC(=O)C(C)C)C)OCC 58728,C1(O)(CNC(c2n(C(C)C)ncc2)=O)CCN(C(=O)CN2C(=O)CCC2=O)C1 58729,N1(C(C(C(C)C)SC)=O)CCC(C2CCN(C(=O)CCCOC(C)(C)C)C2)CC1 58730,C1(NC(=O)C(F)CC2CCCC2)C2CC1N(C(=O)CC1(N3CCCC3)CC1)C2 58731,CC(CN(C)C)C(=O)NC1CCC(CNC(C2(C)CC2Br)=O)C1 58732,C1(C(=O)NCC(CCNC(c2cnc(C3CC3)[nH]2)=O)OC)C(C#N)C1(C)C 58733,Cc1c(N(CCCN2CCN(C)CC2)C)ncnc1N1CCS(=O)C(C)C1 58734,c1(C(=O)NCC(CC)(C)NC(=O)C=NOC)ccc(C(C)C(F)(F)F)cc1 58735,c1(NC(C2N(C(C3N(C(C)C)CCC3)=O)CC(C)C2)=O)ccc2sncc2c1 58736,C1(C(=O)OCC)(CC)CCN(C(c2cn(C)nn2)=O)CC1.c12cncc(n1)NC2 58737,N1(C(C(CN(C(C)C)C)C)=O)CCCC1C(=O)NC(C)Cc1cnccn1 58738,c1(C(C(=O)N(CC(C)O)CCNC(C2(OC)CC2)=O)OC)ccccc1 58739,Cc1ncccc1C=CC(=O)NCCC1CN(C(=O)COC2CC2)CC(C)O1 58740,C1(CCN(C)C(c2ccc(Cl)o2)=O)CCN(C(c2c[nH]cc2C(F)(F)F)=O)CC1 58741,C(=O)(C(F)n1ccnc1)NCCCN(C(C1CCSC1)=O)CC 58742,C#CCC(C)(CC)C(=O)NCCC1CCN(C(=O)Cn2[nH]cnc2=N)CC1 58743,CCC(CC(=O)NC1CC(CO)N(C(C2CC3(CCC3=O)C2)=O)C1)CC(C)C 58744,c1(C(=O)NCC(C)N(C(=O)CC(C(F)F)n2ccnc2)C)cc(O)ccc1OC 58745,Cc1cnc(F)c(CNC(C23CC(NC(=O)C(F)(F)CN(C)C)(C2)C3)=O)c1 58746,C1(NC(C(COCc2ccccc2)OC)=O)(CO)CCN(C(=O)CSC)C1 58747,C#CCC(C)(C)C(=O)NCC1(O)CC(C(N2CCCCCCC2)=O)C1 58748,C1(OCC)CC2(C1)CC2C(=O)NC1CC1NC(=O)CCc1ncc(C(C)(C)C)o1 58749,Cc1c(F)ccc(Cl)c1C(=O)N(CC(C)NC(=O)CCCCN1CCOCC1)C 58750,Cc1csc(CCCC(=O)NCCC2CC(NC(C3(C)CCOC3)=O)C2)n1 58751,C1(C(N2CC(OC)CC(C)C2)=O)(NC(Cn2ncc(C#C)c2)=O)CCC(C)(C)C1 58752,C1(C(=O)NC2C(C)COCC2)CCOCCN1C(=O)CC(=O)N(C)C 58753,N1(C(C(C2CCC2)OC)=O)CCC(C(C)NC(C2CCC2(C)C)=O)C1 58754,c1(CC(N2CCN(C(C(C=C)(C)C)=O)CC2)=O)cccc(C)c1Br 58755,N1(C(N(C)CCC2CC2)=O)CCC(C(=O)O)C(c2cnn(C)c2)C1 58756,C(=O)(C1=CCCOC1)N1CCC(COC)(NC(=O)CC2CCCN2C)C1 58757,c1(-c2ccn(CC)n2)cnc(NC(c2ccsc2C(C)C)=O)c(O)c1 58758,C(CCO)(C(=O)NC1CCCCC1CNC(c1cscc1F)=O)N(C)C 58759,CCC(C)C(O)C(=O)NCCC1(NC(=O)CCCN(C)C(C)C)CCOCC1 58760,c1(C(C(=O)NCC2C(NC(c3nnc(C)s3)=O)CC2)=O)cc(F)c(F)cc1F 58761,C12(CCNC(c3c(C#N)scc3)=O)CCC1CN(C(=O)C(C1CCCCC1)F)C2 58762,c1(NC(=O)C=CC(=O)OCC)ccc(C(N2CCC(CCC=C)C2)=O)cn1 58763,c1(CC)nc(=N)[nH]c(=NC2CCC3CN(C(=O)C(n4cc(Cl)cn4)C)CC23)[nH]1 58764,c1(CC(N2CC(NC(c3cc(C)sc3)=O)C3C2C3)=O)cc(F)cc(F)c1 58765,c1(NCC2C(C)CCN(C(C3CCCSC3)=O)C2)cccc(F)c1[N+](=O)[O-] 58766,CC(N=c1[nH]c(N2CCOC(C3CCCC3)C2)nc2c1SCC2)c1ccncc1 58767,C1(NC(c2ccc(CC)s2)=O)CN(C(=O)C(C)(O)CC(C)C)CC12CCOCC2 58768,C1(OCCC)CCCN(C(C2(C(C)NC(c3cnc(C)o3)=O)CC2)=O)C1 58769,c1(C(c2nnnn2CC)NCC(=C)F)ccc2ccccc2c1Br 58770,CC(CC1=CCCCC1)(c1nnnn1C1CC1)Nc1ccc(-c2ccon2)cc1 58771,CC1(C)CN(CCC2CCCC3CC23)Cc2cccc(NS(C)(=O)=O)c2O1 58772,C1(NC(=O)NC(COC)C(=O)OC)CCC2CCC1N2C(c1cnc(Cl)n1C)=O 58773,C1(CNC(c2cc(CCC)[nH]n2)=O)CN(C(=O)C(F)OC(F)(F)F)C(C)(C)C1 58774,C1(CNC(C(COC)O)=O)CCCC12CCN(C(c1cn(C)ccc1=O)=O)CC2 58775,C(C(C(=O)N(CC(=O)NC)C)C(C)C)NC(COCCCC#C)=O 58776,N1(C(C)=O)CCN(CC(=O)Nc2ccc(Cl)cc2C)CC1c1nccn1C 58777,c1(-n2cc(C3N(C(C(C)OCC)=O)CCC3)nn2)c(F)cccc1Cl 58778,Cc1nc[nH]c1C(=O)NCCCN(CCCCNC(C1CS(=O)(=O)C1)=O)C 58779,c1(C(=O)NC(CC)CNC(=O)Cc2cn(C)nn2)c(C)noc1C 58780,C1(C)(C(N(CC(C)NC(=O)C(O)CN2CCOCC2)C)=O)CCOC1 58781,N1(C(C=NOC)=O)CCC2CCN(C(=O)C(c3cc(F)ccc3F)(F)F)CC2C1 58782,C(=O)(C(C(=O)N(CC(=O)NC(COC(C)C)C(=O)SC)C)OC)OCC 58783,c1(C(N2CC(CNC(C(C3CC3)OCC)=O)C(C)C2)=O)cnn2cccc(Cl)c12 58784,C(CNC(c1nc(C)oc1C)=O)(C(C)C(C)C)NC(C=CSC)=O 58785,C1(C(N(C(CC)COC)C)=O)CC2CCC(C1)N2C(c1csc(Br)c1)=O 58786,C1(CN(CCc2c(C)c(C#N)ccc2)C)CCC2(CCCOC2)O1 58787,C1(O)(CN(C(C(C)c2cc[nH]n2)=O)C)CCN(C(=O)CCn2ncn(C)c2=O)C1 58788,N1(C(CC=CC=C)=O)CCCC2CN(C(c3cc(Br)ccn3)=O)CCCC12 58789,Cc1ccnc(C)c1C(=O)NC1CCCC(N(C(=O)CC#N)C)C1 58790,N1(C(CNC(=O)OCC)=O)CCC(N(CC(C)C)C(C2(C)CCC(C)C2)=O)CC1 58791,CC(C(=O)NC1CN(C(c2ccc([N+](=O)[O-])[nH]2)=O)CC1C(F)F)C(F)(F)C(F)F 58792,Cc1cn2cccc(C(=O)NCCC3(NC(c4cnoc4C4CC4)=O)CC3)c2n1 58793,c1(C(c2n(C(CC)(C)C)nnn2)NC2C=CCCC2)ccc2scnc2c1 58794,C1(CNC(c2c(CC)nccn2)=O)CN(C(=O)C2=COCC2)CC2(CCC2)O1 58795,CC(CC(C)(F)F)C(=O)NC1COCC1NC(c1cccc2c1COC2)=O 58796,C(=O)(CCC(C)(C)[N+](=O)[O-])N1CCC(CNC(c2c(C)con2)=O)C1(C)C 58797,Cc1cccnc1-c1cn(C(C)C(=O)NC(CCc2ccsc2)C(=O)O)nn1 58798,N1(C(c2c(C)nc[nH]2)=O)CCC(C2CCN(C(C34CSCC3C4)=O)CC2)CC1 58799,c1(C(N2CCN(C(c3occ(C(N)=O)c3)=O)C3C2C3)=O)cc2ncccn2n1 58800,c1(SC)cscc1C(=O)N(CC(C)CNC(=O)CC(C)O)C 58801,CCC(C)CC(C(=O)N1CC(C)(COC)C1)NC(=O)C1=CCCCO1 58802,N1(C(COc2cccc(C)c2C)=O)CCC(C2CC2NC(=O)CC(C)F)CC1 58803,C12(C(=O)OC(C)(C)C)CC(C(=O)NCCNC(c3csc(Cl)n3)=O)(C1)C2 58804,C1(C2CCN(C(C3CCCC(C)O3)=O)CC2)(NC(c2c[nH]c(=NC)s2)=O)CCC1 58805,C1(CNC(C=CCN(CC)CC)=O)CCC(C)N(C(=O)CN2CCOC2=O)C1 58806,N1(C(COCCN(C)C)=O)CCCC1CN(C)C(c1csc(C2CCCC2)n1)=O 58807,C1(C(=O)NC(CCC(=O)NCCCC=C)C)CC(=O)C12CCC2 58808,C1(OC)CC(C(N2CCC(CC3CC3)CC2)=O)N(C(c2ccccc2Cl)=O)C1 58809,C1(CNCC(=O)NC(c2ccccc2)CCC)CCCCC1C1CC1 58810,N1(C(C(CSC)OC)=O)CC(NC(=O)C(F)F)C(n2ccnn2)C1 58811,c1(C(N2CC(CNC(C(c3scc(C)n3)C)=O)C2)=O)cc(Br)c(C)cc1F 58812,CC1(F)CN(C(c2cnc3[nH]ccc3n2)=O)CCN(C(C2CC3CCC2O3)=O)C1 58813,CCC(C)C(O)C(=O)N1CCCC(CO)(NC(=O)CC2(C3CC3)CC2)C1 58814,C1(C(N2C(C)(CCC)CC2)=O)CSCCN1C(c1ccc(COC)o1)=O 58815,N1(C(c2cc(C)oc2C)=O)CCC(NC(=O)C(C)Oc2ccccn2)CC1C 58816,N1(C(CP(C)(C)=O)=O)CCOCC(CNC(C2CC(n3ccnn3)C2)=O)C1 58817,c1(SC)cccc(C(=O)NC2CCC(CNC(C3(C)COC3)=O)C2)c1Cl 58818,CC1(CC2CC2)CCN(N2CCOC(c3ccccc3F)C2)C1 58819,CC1CC(c2cn(-c3ccncc3)nn2)CCN1C(=O)COC1CC1 58820,C(=O)(CCC(C)CN(C)C)NCc1occ(C(N(C2(C#C)CC2)C)=O)n1 58821,CC1CN(C(C2CC(=O)N(C3CN(Cc4cc(Cl)cnc4F)C3)C2)=O)CCN1C 58822,CC1(C)CC(CNC(c2cnn(CC3CC3)c2)=O)CN1C(C1CCCC(=O)O1)=O 58823,c1(OCC(=O)NC2CCCCCC2NC(C2CC2C2CC2)=O)cc(F)ccc1F 58824,C1(NC(=O)CCOCC(F)F)CC2CCC(C1)N2C(c1cc2c([nH]1)CCC2)=O 58825,c1(NC(C2(F)CCN(Cc3nc(C)oc3)C2)=O)cncc(Br)c1C 58826,c1(C(N2C3CC(C(N(CC(C)SC)C)=O)C2CC3)=O)ccc(C#N)c(C)c1 58827,Cn1c(C(N2CCCC2C(=O)NC23CC(F)(C2)C3)=O)nnc1S 58828,N1(C(c2c(CC)cc(N)cc2)=O)CC(NC(=O)C=NOC)C(C2CC2)C1 58829,C1(NC(C2C(NC(C(C(C)O)N(C)C)=O)CC=CC2)=O)CCCC(O)C1O 58830,C12(C(N3CCC(CNC(C(C)SCC)=O)C3)=O)COCC1CS(=O)(=O)C2 58831,N1(C(c2ccn(CCC)n2)=O)CCC(NC(c2cn(C)cc2C)=O)CC1C1CC1 58832,C12(C(N3CC(C(C)NC(c4cccc(C)n4)=O)C3)=O)CCCCC1OCC2 58833,Cc1oc(C)c(C(=O)NCCOCCNC(c2nc(C3CC3)oc2C)=O)c1C 58834,C(=O)(C#CC1CCCCO1)NC1CCC(NC(c2sc(C)c(Br)c2)=O)C1 58835,c1(CC(=O)NCC(C)N(C(C(=O)NC(C)C)=O)C)ccn2cncc2c1 58836,S(=O)(=O)(c1ccc(Br)cc1F)N1C2CCN(C(c3ncccc3Cl)=O)C2CCC1 58837,CCC(F)(F)CC(=O)NCC1CN(C(c2coc(CC3CC3)n2)=O)CCCO1 58838,c1(C(N2CCCN(C(C(C(C)(C)C)O)=O)CC2)=O)cc(=O)n2nccc2[nH]1 58839,CC(CC(=O)NCC(CNC(=O)C=CC(F)(F)F)CO)c1cnn(C)c1 58840,c1(N2CC3CC(NC(C=C(C)c4ccco4)=O)C3C2)ncc2c(n1)CCCC2 58841,N1(C(C(CC(=C)C)OC)=O)CCCC(O)(CNC(=O)C(C)OCC)CC1 58842,c1(C(N2CCN(C(C3(CC)CC3(F)F)=O)CC2CO)=O)ccc2c(c1)CCC=C2 58843,C1(CNC(Cc2c(C)nc[nH]2)=O)CCCC(C(=O)NC2(C)CCCC2)C1 58844,c1(CC(=O)NC(CC(C)NC(c2nn(CC)c(C)c2)=O)C)cccc(C#N)c1 58845,C(CC1CCC1)(C(=O)N(C1CCSC1)CC(=O)N(Cc1ccccc1)CC)OC 58846,C1(CNC(c2ncn(C(C)C)n2)=O)CC(C)CCN1C(=O)CP(C)(C)=O 58847,C(=O)(CC(C(F)(F)F)NC(=O)CC(C)C1CC1)NCCN(CCOC)C 58848,Cc1cc(C(=O)NC(C)(CNC(=O)Cc2ncoc2C)CO)cn1C(C)C 58849,C1(C(N(C2CCCN(C(c3ccsc3)=O)CC2)C)=O)CC(F)(F)C12CCC2 58850,CCC(CN(C)C)CC(=O)NCC(CNC(c1ccc(N)c(F)n1)=O)S(C)(=O)=O 58851,c1(CNc2c(F)cc(C(F)(F)F)cn2)ccc2ncc(Br)cc2c1 58852,c1(C(CO)NC(C(C)C#N)=O)ccc(F)c(Cl)c1 58853,N1(C(c2c(N)cncc2)=O)C2CCC1(CNC(c1cnc(C3CC3)s1)=O)CC2 58854,C(=O)(C(C)(CO)NC(=O)C=CC1CCCCC1)N(C1CC(C)C1)C 58855,C1(CC(=O)NCC(C2(O)CN(C(C(C=CC)O)=O)C2)(C)C)CCCC12CC2 58856,C(=O)(C(O)CC(=O)OC(C)(C)C)N(CCCN(C(COCCSC)=O)C)C 58857,N1(C(C2(CC3CCC3)CC2)=O)CCCC(O)(CNC(C2(F)CCS(=O)(=O)C2)=O)C1 58858,c1(-n2c(C)cc(-c3nc(CCCC)nn3CCOC)n2)cc(F)cc(Cl)c1 58859,c1(C(N(CCN(C(C=CCCC)=O)C(C)C)C)=O)ccc(F)c(S(N)(=O)=O)c1 58860,C1(C(=O)Nc2c[nH]nc2C2CCCCN2CCO)CCCCCC1O 58861,N1(C(C2CSC2)=O)CCS(=O)(=O)C(CCNC(=O)CCc2cn[nH]c2)C1 58862,CCC(CC)(CCNC(c1nnnn1-c1ccc(Cl)cc1F)=O)NC(=O)CC1CC1 58863,n1(CC)ccc(C(=O)NCCCCCCNC(c2csc3nnsc23)=O)cc1=O 58864,C1(C(N(CCC(=O)NCC(C#C)CC2CC2)CC=C)=O)C2CCCCCC12 58865,N1(C(c2n(CCC)ccc2)=O)CC(C)OC2(CCN(C(=O)C(F)C(C)C)C2)C1 58866,CCCC(C)(C)CC(=O)N1C2CCC1CN(C(=O)NC1(n3nccn3)CC1)C2 58867,N1(C(C2(NC(C(C)OCC)=O)CCN(C)C2)=O)CCSC(C)(C)C1 58868,C1(OC)CCC12CC(C(=O)NC1CC1NC(c1c(C)noc1C(F)F)=O)C2 58869,c1(OCCCC(=O)NCC2(O)CCN(C(C3(C=C)CC3)=O)C2)ccc(C)c(C)c1 58870,c1(OC)cc(C(N2CC3CC2CCC3NC(=O)CCS(N)(=O)=O)=O)c(O)c(Cl)c1 58871,C1(C(c2ccnc(N3CCN(c4cnncc4Cl)CC3)n2)=O)CCCCCCC1 58872,c1(C(=O)NCC(CN(C(CCC(=O)NC)=O)C)O)ccc(OC)c(S(N)(=O)=O)c1 58873,C1(NC(c2c(OC)cncc2)=O)CCN(Cc2ccc(Br)[nH]2)CC1O 58874,C1(C(=O)NC(CN(C(Cc2c(C)nn(C)c2Cl)=O)C)(C)C)CN(CP(C)(C)=O)C1 58875,C#CCC(C)C(=O)NC(C)CC1CCN(C(c2ccnc(O)c2)=O)CC1 58876,c1(C(N2CCCCC(NC(C(C)(C)c3cnsc3)=O)C2)=O)cn2c(n1)COCC2 58877,c1(C(=O)NCCC2(CNC(CCC(C)OC)=O)CC2)cnn2ccncc12 58878,c1(C(=O)NC2(CCNC(C(CC#C)C3CC3)=O)CC2)ccc(C)cc1C 58879,C1(CNC(C2CC(SC)C2)=O)CCCCN(C(c2c[nH]c(=N)s2)=O)C1 58880,C1(C(C)(C)C)(CNC(C2(C)CCCS2)=O)CCN(C(c2cccn2C2CC2)=O)C1 58881,C1(CNC(=O)NCC2CC(O)(C(F)(F)F)C2)(CO)CC2CC2C1 58882,CC(=O)CC(C)(C)CC(=O)NCC(C)N(C(=O)C#CC1(C)CCCO1)C 58883,CON(CC1CC2CCC1C2)C(=O)C(CO)NC1CCC1 58884,Cc1ccc(C(=O)NCC2CCC(NC(c3csc(S)n3)=O)C2)cc1C 58885,N1(C(C(CCC)C)=O)CC(C)(C)OCC1CNC(C1CC(S(C)(=O)=O)C1)=O 58886,C1(C2CC2)(C(N(C(CNC(C(C=C)O)=O)Cc2ccccc2)C)=O)CCC1 58887,c1(OC)cccc2ccc(C(N3CCN(C(=O)C(O)P(C)(C)=O)C(C)C3)=O)nc12 58888,Oc1c(CNCCc2cc(Cl)ccc2Cl)cc(Br)cc1Cl 58889,N1(C(C(CN(C)C)NC(c2ncc(NC)nc2)=O)=O)CCC2(CCOC2)CC1 58890,C1(C(N(CCCNC(C2CC2c2cncn2C)=O)CCO)=O)CC1C1CCC1 58891,C=CCN=C(NCc1nccc(C(F)(F)F)n1)NCC(c1nc(C)cs1)(C)C 58892,c1(C(=O)NCC23CC(NC(C4CCC(C)C4)=O)(C2)C3)c(F)cc(F)c(F)c1F 58893,c1(C(C)=O)c(C)[nH]c(C(=O)NC2CC(CNC(=O)C(C)C3CCC3)C2)c1C 58894,N#CC1(C(=O)NCC2CC(NC(C3CC4(CC4)CO3)=O)CCO2)CCCOC1 58895,Cc1cc(NC(=O)C(CNC(=O)CC2CSCCO2)N(C)C)cs1 58896,C1(NC(c2nc(OCC)oc2)=O)CCN(c2nnc(C(F)(F)F)s2)CC1O 58897,c1(CN(CC(c2cn(CC)nc2)O)C=O)nc(O)c2ccc(Cl)cc2n1 58898,Cc1nocc1CC(N1CC=CC1CNC(=O)C(n1cc(Cl)cn1)C)=O 58899,C(=O)(C1(C)CCn2c(C)nnc21)N1CCC2(CCN(C(CCC)=O)C2)CC1 58900,C(C(CC1CC1)CC(=O)N1CCOC(C)(C)C1)NC(CCCOC)=O 58901,N1(C(C=CC(CC)C)=O)CC(C2CC2)(C(=O)NCc2ccc(CO)o2)C1 58902,c1(C(N(C2CCCC(NC(c3ccnc(Cl)c3F)=O)C2)C)=O)cc(F)cc(F)c1 58903,N1(C(C(CN(C)C(c2ccccc2O)=O)O)=O)CC(F)CC1C(N)=O 58904,CC(C(=O)NCC1CC1NC(=O)Cc1c(F)cccc1F)C1=CCCC1 58905,Cn1c(C(=O)NCCN2CCN(c3ncccc3[N+](=O)[O-])CC2)ccc1[N+](=O)[O-] 58906,c1(C(C(=O)C(Cc2ccsc2)NC=O)C(N2CCC(OC)C2)=O)cccc(O)c1 58907,C1(C(N(C)CC2CCN(C(=O)CCc3ccc(=N)[nH]c3)C2)=O)CCC2(CCC2)O1 58908,C(C(F)(C(=O)N1CCC(F)(C(N)=O)C1)C(C)C)NC(C1CCC(=C)CC1)=O 58909,CC(C)C(C(=O)N1CCC(CC)C1CNC(=O)CN(C)C(=O)C1CC1)NS(C)(=O)=O 58910,c1(C(=O)NCC(C)NC(C2CCC(=O)O2)=O)cn(C)cn1 58911,Cc1cccc(C(=O)N(C2CCCCC2NC(C2OCCCO2)=O)C)c1 58912,N1(C(C(C2CCC2)OC)C(=O)NC2CCOC2)C2CCC1CC(=O)NC2 58913,C1(C(C)(C)O)CCC(C(=O)NCC2CN(C(c3ncccc3C(F)F)=O)C2)CC1 58914,N1(C(=O)CSCc2cscn2)CC2(CCN(C(=O)C3=CCCOCC3)C2)C1 58915,N1(C(c2ccn(CC)c2C)=O)CCN(C(c2ccc(O)c(C)c2)=O)CC1C 58916,CN(CCCNc1ccccc1)N1CCCC2(C1)CC(F)(F)C2 58917,c1(CNc2c(C)nc(NC(N3CC(C)C(F)(F)C3)=O)s2)ccc(F)c(F)c1 58918,c1(C(=O)NCCCN(C(CCOCC#C)=O)C)c(C)nc2sc(C)nn12 58919,c1(OC(C)=O)ccc(OCCC2CCCN(C(C)C)C2)cc1C 58920,C1(OC)CC2CCC(C1)N2C(=O)CC(CC)N(C(=O)C(C)OCC(C)C)C1CC1 58921,C1(OCC)CC2(C1)CC2C(=O)NCCC(C)NC(=O)C(F)(F)COC 58922,c1(C(N2CCC(N(C(=O)CC(C)n3ccnc3)CC)C2)=O)nc(O)[nH]c(=O)n1 58923,CCCCCC(O)C(=O)N1CCC2C(NC(=O)CN(c3ccccc3)C)C2C1 58924,c1(CCC(=O)NCCCOCCCNC(C(CC#C)C)=O)cccc(F)c1F 58925,n1(C(CC)C)ccc(=NC(=O)C2C(C)OCCN2C(c2cnc(OC)s2)=O)[nH]1 58926,C1(NS(CC2(C)CNC(=O)N2)(=O)=O)C2CC3C(CO)CC1C3C2 58927,C1(CNC(C2(COC)CCOC2)=O)CCCCN(C(=O)CSc2nc[nH]n2)CC1 58928,c1(CC)ccc(F)c(C(=O)NC2CCC2NC(C2CCOC2C(C)C)=O)c1 58929,C1(OC)CC2CN(Cc3c[nH]c(=N)nc3C)CCN2C1 58930,CCCCCC(=O)NCC(COC)NC(=O)CC1CCCOC1 58931,Cc1nc(CC(=O)NCC(F)(F)CCc2ccccc2)oc1-c1ccccc1 58932,C1(C(N2CCOCC2)=O)(NC(=O)CN2CCCNC2=O)CCCCC1 58933,C1(OC)(OC)CC(C(N)=O)CN(C(C2CCN(C)C(=O)C2)=O)C1 58934,CC1CN(C(=O)CCC(C)(F)F)CCC1NC(c1ncnc(O)c1Br)=O 58935,C12(CN(C(=O)CC3CC(F)(F)C3)C1)C(=O)N2.C1(CCSC)CCSC1 58936,CC(C)C(CNC(=O)C(Cl)Cl)C(=O)NCC(O)C(C)(C)O 58937,CC1c2cccc(F)c2CCN1C(CCCCC1CC1)C(=O)NC1CC1 58938,C1(C(=O)NCC(CN(C(c2nn(CC)c(O)c2)=O)C)(C)C)CC(C(C)(C)C)=NO1 58939,CCC(CCOC)C(=O)NCC1CCN(C(=O)CCc2cnn(C)c2OCC)C1 58940,c1(CC(=O)NC2C(C)N(C(=O)C=C3CN4CCC3CC4)CC2)cc(Cl)ccc1Cl 58941,c1(CN2CC(NC(C(C)Oc3ccccc3)=O)C(C#N)C2)cccc([N+](=O)[O-])c1 58942,NC(=O)CC(C1CC1)NC(=O)CC1(NC(C2CCC(F)C2)=O)CC1 58943,N1(C(C(C)(C)CF)=O)CC(CNC(c2ccncn2)=O)C(F)(F)C1 58944,Cc1cccc(CNC(=O)CCN(C(=O)C2=COCCC2)CCO)c1C 58945,c1(C(N(C(c2cn(CCCC(=O)O)nn2)C)CC)=O)ccoc1-c1ccccc1 58946,N1(C(CCCCSC)=O)CCC2(CC1)CC2C(=O)NC1(CC2CC2)CCC1 58947,C(c1ccc(Br)c(C)c1)=CC(N1CC(COC)N(C(C2C(C)C2C)=O)CC1)=O 58948,CC#CCC(C(=O)O)NC(=O)C(c1ccc(Cl)c(F)c1)F 58949,c1(-c2ccc(N3CCCC(C=C)C3)c(N)c2)ccc(C#N)cc1F 58950,CC1CCC(C(=O)NCC2(NC(=O)CCCNC(=O)C(C)(C)C)CCC2)C1 58951,C1(C(N(C2CCN(Cc3ccccc3)C2)C)=O)CC(=O)N(Cc2ccnn2C)C1 58952,Cc1cnc2c(C(=O)N(C(C)CCNC(=O)C(O)CN(C)C)C)cnn2c1 58953,C(C(F)(C(=O)NCC(C)C=O)C(C)C)NC(C12CCC(OC)C1C2)=O.OC 58954,C1(C(N(C)CC2CCN(CC)C2)=O)CC(NC(=O)CSc2ccccc2)C1(C)C 58955,CCCC(C)(C)C(=O)NCCc1ocnc1CNC(=O)COc1ccc(Cl)c(C)c1 58956,N1(C(c2nc(CC)sc2)=O)CCCC(O)(CNC(c2ccnc(Cl)c2OC)=O)C1 58957,n1(CC(=O)N(N(C(CNC(C2C(C)C2)=O)=O)CCN)C(C)C)ncn(C)c1=O 58958,c1(C(=O)NCCC(C)NC(C(CSC)O)=O)scnc1C#N 58959,O=C(CS(=O)c1ccc(Cl)cc1)NCC1CCCN1C(=O)CC1CCCOC1 58960,c1(C(=O)NCC(C)CNC(=O)C(CC#N)c2ccccc2)csc2c1CCOC2 58961,C12(NC(c3c(CC)ocn3)=O)CCCC1CN(C(=O)CN1CC=CC1)C2 58962,c1(C(N2CCC(CC(N3CCC(=C)C3)=O)C2(C)C)=O)cc2ccccc2o1 58963,Cn1nc(C(=O)NCC2CC2NC(c2cccnc2C(F)F)=O)cc1Cl 58964,c1(C(=O)NCCN(C(c2cc(C)cc(Cl)c2)=O)CC)ccc2nccnc2n1 58965,N1(C(c2nc(CC(C)C)sc2)=O)CCC(n2cc(CNC(=O)CO)nn2)CC1 58966,C1(NC(c2cc(F)cc(F)c2)=O)CC2CN(C(=O)CC3CCSCC3)CC12 58967,N1(C(C2C(OCC)C2)=O)CC2CCCC2(Nc2nc(C(C)(C)C)ccc2C#N)C1 58968,C1(CNC(C(=Cc2cccs2)C)=O)(Nc2ncn(C(C)(C)C)n2)CCCCC1C 58969,c1(C(N(C2CCC(NC(C(C)SCCCC)=O)CC2)C)=O)cc([N+](=O)[O-])ccn1 58970,CN=c1nc(N2CCC(C)(N(C)C)C2)[nH]c(=NCCc2ccncc2C)[nH]1 58971,c1(C(N2CCCC(N(C(C(CC=CC)C)=O)CCF)C2)=O)cc(C)cc(C)c1O 58972,c1(C(=O)NCCC(=C)CNC(C2CCCC(F)C2)=O)c(OC)cccc1O 58973,c1(C(=O)NC(CNC(Cc2cn(CC)nn2)=O)C(C)(C)C)c(C)cc(C)nc1O 58974,C(=O)(C(O)CCCNC(=O)CC1(O)CCCOC1)N1CCC(C(C)OC)CC1 58975,c1(NC(c2ccc(F)c(Cl)c2)C)ccc(S(=O)(=O)N2CCOCC2CO)cc1Br 58976,C(c1cc(Cl)cc(Cl)c1)=CC(=O)NCC(CNC(C1CC(CC)C1)=O)(C)O 58977,C12(NC(C(C3CC3)SC)=O)CC(NC(=O)CN(C)S(N)(=O)=O)(C1)C2 58978,CCC(CC)C(C)C(=O)N1CCC1CNC(=O)CCc1ccsc1 58979,C(CC(C)C)(C(=O)NCC1CN(C(c2cccnc2O)=O)CCCO1)NC(C)=O 58980,C1(C(=O)NC(CCCC)C)CC2CCC1N2C(c1n[nH]c(O)n1)=O 58981,C1(C(=O)NC(C2CCS(=O)(=O)C2)C2CCCCC2)CC2(CCC2=O)C1 58982,C(=O)(CCCC(=O)OC(C)C)NC(CC1CCN(C(CCCCOC)=O)CC1)C 58983,Cc1ncc(C(N2C(C(=O)N(CCCCN(C)C)C)CCC23CC3)=O)c(C)n1 58984,C1(C(=O)NC2CC(F)(CNC(c3ncc(C)cn3)=O)C2)CC2CCC1CC2 58985,C(=O)(C1=CCN(C(C2CC2OC(C)=O)=O)C1)N1CCC(=C)CC1 58986,Cc1ncsc1C=CC(N1CCC(C(C)(C)NC(C2C(C)(C)C2(F)F)=O)CC1)=O 58987,c1(C(N2CCOCC(NC(C(=O)N(C)C)=O)C2)=O)cn2ccncc2n1 58988,C(C)(CCC(=O)NC1CCN(C(=O)C(F)(F)c2cnn(C)c2)C1)SC 58989,C(=O)(C(O)CC(F)F)NCC(C)(C)OCCNC(C(c1ccc(F)cc1)OC)=O 58990,C1(CNC(C=C=C(C)C)=O)CCN(C(=O)Cc2ccoc2)CC1C 58991,CCC(COC)(CC)C(=O)NC1CCN(C(C2Cc3nccn3C2)=O)C1 58992,C1(CCOC)(NC(=O)CCN2CCCCC2)CCN(C(C2(SC)CC2)=O)C1 58993,C1(C2CCCCC2)(NC(c2ccc(C)cc2Cl)c2n(CC=C)nnn2)CC1 58994,C1(NC(C(C)Cc2ccccc2)=O)CC12CC(NC(=O)CCCC1CC1)C2 58995,CCC(C)C(C)C(=O)N1CC(N(C(=O)CCc2c(C)nn(C(C)C)c2C)C)C1 58996,c1(C(N2CC(CC(C)NC(c3ccc(COC)[nH]3)=O)C2)=O)cc(N)c(O)c(F)c1 58997,N1(C(C2CCN(C(C)=O)CC2)=O)CC2(CCC2NC(=O)CC2CCCCCC2)C1 58998,C1(C(=O)NCC2CCN(C(C)C)C2)CCN(C(C2(F)CCCCC2)=O)CC1C 58999,C(c1cccc(F)c1F)=CC(N1CC(NC(C2CCN(C)C2)=O)C(O)CC1)=O 59000,c1(C(N2CCC(N(C(=O)C(C)CC3CC3)CC#C)CC2)=O)ccc(=O)n(CC)n1 59001,CCS(=O)CC(=O)NCC(C)(C1CC1)NC(=O)CC1CC(C)(C)C1 59002,c1(C(C(=O)N(CCCC(=O)NC)C)NC(C2CC(CF)C2)=O)c(C)cccc1Br 59003,C1(C)(NC(C(n2cc(Br)cn2)C)=O)CCCN(C(C2(O)COC2)=O)C1 59004,c1(NC(C2CCN2S(=O)(=O)c2ccc(Br)cn2)=O)ccc2c(c1)CCC(=O)N2 59005,C(=O)(C(C)CS(=O)(=O)c1ccc(F)cc1)NC1CN(C(C(C)C)=O)CC2C1C2 59006,C1(C)(C(N2CCC(CN(C)C(c3ccon3)=O)C2)=O)CCCN1C 59007,CC(C)CC(O)CNC(=O)C(Cc1ccoc1)NC(C1COC1)=O 59008,n1(CC)cc(Br)c(C(=O)NCC(O)CCNC(c2[nH]c(O)nc2C)=O)n1 59009,CC(CC(F)(F)F)C(=O)NC(CC(=O)NCCCCN(C)C1CC1)C(C)(C)C 59010,c1(C(CC)C(=O)NC(C)(C)CCNC(=O)CSc2nc[nH]n2)cccc(Cl)c1 59011,N1(C(c2ncn(C)n2)=O)CC2CC(NC(=O)C=Cc3ccco3)CC(C2)C1 59012,C1(OC2(C(N(CCCN(C)C(C3CCSC3)=O)C)=O)CC2)CCCOC1 59013,C12(C(=O)NC(C)C(=O)NC3CC3)CC(CCO1)N(C(=O)C(C)NC=O)C2 59014,C1(C(N2CC(C)(NC(c3cncc(-n4ccnc4)n3)=O)C2)=O)CCC2CC1CO2 59015,C1(CNC(C(C)OCC#C)=O)(CO)CC12CCN(C(=O)CC1CC(=O)C1)CC2 59016,Cc1nc(C(N2CCSCC2C(=O)NC(c2ccncc2)C)=O)ccc1Br 59017,N1(C(C2C(=C)CC2)=O)CCC2(CCC2CNC(=O)C2=CCOCC2)CC1 59018,C=CCC(C(=O)NC1CCCCN(C(=O)C(C)(C)C(=O)OCC)CC1)C(C)C 59019,c1(C(N2CCN(C(c3nn(C)c(O)c3)=O)CC2)=O)ccc2ncn(C)c2n1 59020,CC1CCCc2cc(C(=O)NCCCNC(C3CCC4(CCC4)OC3)=O)nn21 59021,N1(C(CC(C)N(C)C)=O)Cc2nccn2CC(NC(=O)Cc2cnccc2Cl)C1 59022,N1(C(c2ccc(C)cc2C)C(=O)NC(C(=O)OC)C)CC(C)OC2CCCCC12 59023,Cc1n[nH]c(C)c1CCCNC(=O)N(C)Cc1coc(-c2ccccc2)n1 59024,C1(CCCNC(C=CCOC)=O)CCN(C(C2COCC2(C)C)=O)CC1 59025,c1(C(=O)NCC2CCN(C(c3cn(C)nc3Cl)=O)CC2)coc2ccc(F)cc12 59026,c1(C(N2CC(CC(C)NC(=O)CN(C)C)C2)=O)cc([N+](=O)[O-])ncc1Br 59027,c1(OC)ccc(Cl)c(CN2CCCC(C(=O)Nc3ncc(F)cc3Br)C2)c1 59028,c1(C(=O)NC2CCN(C(C3(C#N)CC4CC4C3)=O)CC2)ccnc2ccccc12 59029,C1(CNC(C(n2cc(C3CCN(C)CC3)nn2)C)=O)CC2(CCC2O)C1 59030,C1(CC(=O)N(CCCOCc2ccccc2)C)CCc2ccccc2C1 59031,C(C(CO)(CO)NC(=O)C(C)Cc1cnc[nH]1)N(C(C(C)OC)=O)C 59032,CCCCCC=CCN(C1CC(C)C1)C(c1[nH]ccc1C1CC1)=O.OC 59033,N1(C(C2C(NC(c3cn(CC)nn3)=O)CCOC2)=O)CC2CCC(C1)O2 59034,N1(C(CCOCCN(C(CCC(CC)C)=O)C)=O)CC(C2CC2(F)F)C1 59035,N1(C(C2C(=C)C2C(C)=O)=O)CC=CC1(C(=O)N(CC(C)(C)O)CCC)C(=O)OC 59036,N1(CC(=O)N(CC(c2ccccc2)C)C)C(=O)C=CC1=O 59037,N1(C(C(=O)OCC)=O)CCC2(CCC(NC(=O)NCc3ccc(CC)o3)CC2)C1 59038,C1(C)(C(N(CCCO)C)=O)CC12CCN(CC1CC3CCC1O3)CC2 59039,CC1CN(C(C2CCN(C)C2=O)=O)CC(C)CN1C(c1cc(O)cs1)=O 59040,CCCC(CCC)CC(=O)NCCCN(C)C(c1sccc1CC)=O 59041,c1(NC(=O)NCC(C)Oc2ccc(OCCOC)cc2)cc(Cl)c(Cl)c(C)n1 59042,CN1CCC(CC(=O)N(C)CC2(O)CCN(C(=O)CCC3CC3(C)C)C2)CC1 59043,c1(NC(c2c(C(C)C)onc2)=O)cc(F)c(C(=O)N(C)C)c(F)c1 59044,CC1(CNC(=O)C=CC(=O)NC2CC2)CCCN(C(=O)CC(F)(F)Cl)C1 59045,C(N=c1[nH]c(=NC2CC3CC4C(C3)C24)c2ncccc2[nH]1)c1[nH]c2ccc(Cl)cc2n1 59046,O=C(C#CCNC(C1CCC(=O)O1)=O)NCC1CCOC1 59047,S(=O)(=O)(c1ccc(=NCCn2cccnc2=O)[nH]c1)NC(c1ccccc1Br)C 59048,C(=O)(C1CCc2cccnc21)N1CCC(OCCNC(=O)C2=COCCO2)C1 59049,c1(NC(C(CC)N(C2CC(OC(C)C)C2)C)=O)cn(C)cc1C 59050,c1(C(C)C)ccc(C(=O)NCC2CC(NC(c3ccc(C(C)=O)nn3)=O)C2)cc1 59051,C1(NC(c2cc3scnc3[nH]2)=O)CC2CC(C1)N(C(C1Cc3nccn3C1)=O)C2 59052,C(c1ccc(S(C)(=O)=O)o1)=CC(=O)NC1CC(CCNC(C(C(C=C)C)C)=O)C1 59053,c1(C(=O)NC2CC(NC(c3ccc(NC=O)cc3)=O)C2)ccc(Br)c(Cl)n1 59054,C(=O)(C(CC)C(C)(C)CC)NC1CCC(CNC(c2ccc(C#C)o2)=O)CC1 59055,C1(CNC(C#CC(C)(C)C)=O)C2CCC1CN(C(=O)CCN1CCCCC1=O)C2 59056,C1(C(=O)NC(CCCNC(Cc2cc(C)ns2)=O)C)CCN(C)C(=O)C1 59057,Cc1c(C(=O)NCC#CCNC(=O)CC2CCCC2(F)F)sc2ccccc12 59058,c1(CNC(c2ccc(OC)nc2OC)CC(=C)C)ncc(Cl)cc1Cl 59059,C12(NC(c3cccc(Cl)c3)=O)CCCCC1N(C(c1ccncc1)=O)CC2 59060,O=C1CC(NC(c2ccc(-c3ccncc3)cc2)=O)CCN1 59061,Cn1nc(Cl)c(C(=O)NC2CCN(C(=O)C(C3(O)CCCC3)F)C2)c1Cl 59062,C#Cc1cc(C(=O)NCC2(NC(=O)CC3OCCO3)CC2)cc(C(F)(F)F)c1 59063,c1(CNC(=O)Cn2cccc2)csc(CNC(c2cc(F)cs2)=O)n1 59064,c1(NC2(CNC(C(C3CCCOC3)OC)=O)CCOCC2)ncc(Cl)c(O)n1 59065,N1(C(COC)=O)CCC2(NC(c3cncc(C(=O)OC)c3)=O)CC2C1 59066,C1(CNC(c2csc(C)c2N)=O)C(C)CCCN1C(C1CCCN1C1CC1)=O 59067,c1(C(=O)NC2CCCC(NC(c3c(C(C)C)nn(C)c3)=O)C2)nccc(Cl)c1O 59068,C1(NC(c2ccc(C)c(C)n2)=O)Cc2ccccc2N(C(=O)C2=COCC2)C1 59069,c1(C(C)=O)ccc(C(=O)NCC(C)N(C)C(C2CCC3(CC3)C2)=O)c(F)c1 59070,N#CC1CCN(C(C2(NC(=O)Cn3ccnc3)CCOCC2)=O)C1 59071,n1(CC=C)nnnc1C(c1noc(C(C)(C)C)n1)NCC1(F)CC1 59072,C1(C#N)(C(N(CCCNC(C2(CC(F)(F)F)CC2)=O)CC)=O)CC2CCC1C2 59073,C1(CC(=O)OC)CN(C(=O)Cc2cnn(C(C)(C)C)c2)CC12CC2 59074,C1(N(C(C(=O)NCCC)C2CCCC2)C)CCS(=O)(=O)C1.c12cccc(c1)OC2 59075,N1(C(C2C(C)C2)=O)CCN(C(=O)CC(C)(C)c2cccs2)C(C(C)(C)C)C1 59076,CC1(C)CCCC(CC(=O)NCCC2CCCN2C(=O)CN=S(C)(C)=O)O1 59077,N1(C(c2ccn(C(C)C)n2)=O)CC(C)CN(C(=O)CS(=O)(=O)C(C)(C)C)C(C)C1 59078,c1(CNC(C(COC)(F)F)=O)nnc2n1CCN(C(=O)CC(C)(C)C(C)(F)F)C2 59079,C1(NC(CNC(C)=O)=O)CC(NC(c2cnc(CC3CC3)s2)=O)C12CCC2 59080,N#CC1(C(=O)NCC2CC(O)CN2C(c2cnc[nH]2)=O)CCCO1 59081,C1(NC(C(C2(OC)CCCC2)(F)F)=O)CS(=O)(=O)C2CN(C(=O)C(F)OC)CC12 59082,C#CC1(OCC(=O)N(C2CN(C(=O)CCOCCCNC(C)(C)C)C2)C)COC1 59083,c1(CC(N2C(Cn3cc(CCOC(C)=O)nn3)C=CC2)=O)cc(F)ncc1Cl 59084,C1(NC(c2c(C)[nH]cc2)=O)CCCCC1NC(=O)C(c1ccc(Cl)s1)C 59085,c1(NCC)ncc(C(=O)N(C)CCNC(=O)C(C2(O)CCCC2)F)cc1Cl 59086,n1(CC)cnc(C(=O)NC2CCC2NC(C2(F)CC2)=O)n1 59087,C12(C(=O)NCC3C(CC)C3)CC(CNC(C3(C(N)=O)CC3)=O)(C1)C2 59088,S(=O)(=O)(c1ccc(NC2CCCC3CCCCC23)c(C#N)c1)N(C)CCF 59089,c1(C(=O)NCCCC(C)(C)NC(=O)Cn2cnnc2)onc2c1CCCC2 59090,c1(C(C(=O)NC2CCOCC2)N(CCC2=CCCCC2)C)cc2cc(Cl)ncc2o1 59091,N1(C(c2c(OCC)nsc2)C(=O)Nc2ccccc2)CCN(CCC(F)F)CC1 59092,n1(CC)cnc2c(NC(CN(C)C)CC(C)C)[nH]c(=NC(C)c3cn(C)nn3)nc12 59093,c1(NC(Cc2c(C)nccc2)=O)cc(Br)c(F)cc1C#N 59094,C(C(CC(C)C)C(=O)NC(c1ccncc1F)C)NC(C(CCOC)C)=O 59095,C(=O)(C(O)CN(C)C)N(CC(CC)NC(=O)C(n1cc(C)cn1)C)C 59096,N1(C(C(CC#C)NC(C2CCN(OC)CC2)=O)=O)CCC(C)C2(CCC2)C1 59097,CCCCCCC(C)C(=O)N1C2CCC1CC(N(C)C(c1nc(C)oc1C)=O)C2 59098,c1(CCc2nc(COC)nn2-c2ccn(C)n2)ccc(Cl)c(Br)c1 59099,N1(C(CC2C(C)C2)=O)CC2CC2(NC(c2ccc(OCC3CC3)nc2)=O)C1 59100,C(C(CC1CCCC1)C(=O)NC1CCC(CCCl)CC1)NC(=O)C1CC1 59101,c1(C(N2CCC(CNC(C3C(C)OCC3)=O)C2)=O)cnn2ccn(C)c12 59102,C12(NC(CCCN(C)Cc3sc(Br)nc3Br)=O)CCC(CO)(CC1)C2.C 59103,CCS(=O)CC(=O)N(CC(C)CNC(=O)CCCSC(C)(C)C)C 59104,CC1CN(C(C2CCO2)=O)CC1NC(=O)Cc1ccnn1C1CCOCC1 59105,c1(OC)cc(C(=O)OCCCNC(C(=O)OC(C)(C)C)=O)cc(C#N)c1O 59106,C(CC(C(=O)NC1CC(OC)C1)NC(C=CCC)=O)N(C)C.C1(CO)CO1 59107,S(=O)(=O)(c1cccc(N(C)Cc2scnc2C)n1)N1CCC(OCC=C)C1 59108,c1(C(=O)NC2(C)CN(C(=O)CN3CCc4sccc4C3)C2)nnn2c1CCCC2 59109,C(N=c1[nH]c(=N)[nH]c(=NCCS(=O)(=O)CCO)[nH]1)C1(C=C)CCOCC1 59110,S(=O)(=O)(CCC(F)(F)F)N1CCC(C(C)C(=O)NCc2cnc(Cl)cc2I)CC1 59111,N1(Cc2ccc(OC)nc2Br)Cc2ccccc2C1C(=O)NC1CC1(F)F 59112,c1(C(=O)NC2CN(C(C3N(CCC)CCCC3)=O)CC2C)cc(C)c(Cl)cn1 59113,c1(CCCC)cc(C(=O)NCC2(NC(=O)C=Cc3cocn3)CCOC2)c(C)o1 59114,c1(OC)ccc2occ(C(=O)NC(c3ccccc3)CNC(=O)C(C)CF)c2c1 59115,C1(C(=O)NCC(CCOC)NC(c2cc(CF)on2)=O)(C(F)F)CCCCC1 59116,C(=O)(CCCS(C)(=O)=O)NC1CCCC(NC(CCCCOC)=O)C1 59117,c1(C(=O)NCCOC2CN(C(=O)C(F)(F)CO)C2)ccc(=O)n2c1COCC2 59118,c1(C(=O)NCCC(C)N(C(Cc2cc(C)no2)=O)C)c(C(F)F)cnn1C 59119,C(C(C(=O)NCC(C)(O)CN(C)C)NC(=O)CCNC(C)=O)OCC 59120,N1(C(CS(=O)(=O)NCC)=O)CCCC12CCN(C(=O)C(c1cccc(C)c1)O)C2 59121,C(=O)(CC(F)(F)CC(=O)N1CCN(C)CC1CNC(=O)CC(C)(C)OC)OC 59122,c1(C(N2CC(NC(C(C(C)C)(C)C)=O)C(C)C2)=O)ccc2nccn2n1 59123,C1(CSc2ccccc2)CC(C(F)(F)F)=NO1.C12(CC)CN(C1)C(=O)C(=O)NC2 59124,C12(C(=O)NCC=CCNC(c3cccc(OC)n3)=O)CCCCC(OC)(C1)C2 59125,C1(C(=O)NCC(CC)NC(=O)CCc2cncs2)CNC(=O)CC12CCC2 59126,N1(C(C(C)N(CC(=O)NCCC)C)=O)CCCC(CC)CC1 59127,C(=O)(CCC(C)=O)NC(C(=O)Nc1c(OC)nsc1)CC1CC1 59128,C1(NC(C2CC(C)=C(C)CC2)=O)CCN(c2ncc(O)cn2)CC(C)(C)C1 59129,N1(C(CN(CCOC)C)=O)C2CCC(C2)C1CNC(=O)Cn1nc(C)oc1=O 59130,C12(CNCC3(N)CCC3)CC3CC(CC(C3)C1)C2 59131,C1(NC(c2nc(COCC)sc2)=O)CN(C(=O)Cc2cnc(C)o2)CC(C)(C)C1 59132,Cc1ccc(Br)c(C(=O)NCC(C)NC(c2ccc(C3OCCO3)cc2)=O)n1 59133,C(=O)(C1=NOC2COCC12)N1CC=C(CCNC(C2CCS2(=O)=O)=O)CC1 59134,Cn1nc(C(N2CCC(C(N3CC(c4ccccc4)C3)=O)C23CC3)=O)cc1C#N 59135,C(=O)(CCCCCNC(C1CC(C)CC(=O)N1)=O)NC(C)Cc1ccco1 59136,N1(C(c2cc(CC)c(CC)o2)=O)CC(C2CN(C(=O)C(C)(O)CC)C2)C1 59137,c1(C(=O)NC(CC(C)NC(C(CC)OC)=O)C)c(C)nn(CC)c1C(F)(F)Cl 59138,C(=O)(C1=NOCC1)NCCC(CNC(C(CSC)OC)=O)O 59139,C(c1ccc(Cl)c(F)c1)=CC(N1CCC(C(=O)OCc2ccccc2)CC1)=O 59140,C(CCCCC(=O)NC(CC1CC1)CO)NC(c1cc(OC)ns1)=O 59141,Cc1cc(C(N2CC(NC(c3cn(C)cn3)=O)C(F)C2)=O)cc2c1NCCC2 59142,C1(SC)CN(C(=O)C=CC2CCCO2)CC1NC(=O)C(Cl)=CCl 59143,Cn1c(O)nc2cc(C(N3CCC(CCNC(=O)CCCC#N)C3)=O)ccc12 59144,Cc1ccc(C)n1CC(N1CC(F)CC1CC(N1CCC(CCCO)CC1)=O)=O 59145,C1(C)(CC)CCC(C(=O)NNC(=O)c2cnsc2)O1 59146,c1(N2CC=C(C)C2)nc(=NCCc2c[nH]c3ncccc23)[nH]c2cc[nH]c12 59147,c1(C(=O)NC(CNC(C=CC(C)(C)SC)=O)CCOC)cc2n(n1)CCO2.C(C)(=O)O 59148,C(=O)(C(c1ccccc1)=C(C)C)NCC1C2(N(C(C=C(COC)C)=O)C2)C1 59149,c1(N(CCCN2CCOCC2)Cc2ccc(C)o2)ccc(F)cc1C#N 59150,C1(C(=O)NCCC(=O)NC)CC(C)N1C(c1ncn(C)n1)=O 59151,CC(CC(N)=O)C(=O)NC(C)CCN(C)C(c1cc(OC(F)(F)F)ccc1F)=O 59152,Cc1ccc(Cl)cc1-c1cn(CCCNC(=O)CCNC(N)=O)nn1 59153,c1(C(N2C(C(=O)NC(C3CCCC3)C#C)CCCC2)=O)c(C)cccc1C 59154,N1(C2CCN(C(CCCOCC=C)=O)C2)CCN(C(c2ccc(Br)o2)=O)CC1 59155,C(=O)(C(F)C(C)(C)O)NCC(=O)NCCO.C(C1C(=O)N1)N(C)C 59156,C12(NC(CCNC(C(C)(C)C)=O)=O)CCCC1CN(C(C13CC1CNC3=O)=O)C2 59157,c1(CC)nccnc1C(=O)NCC(C)(C)CNC(c1cc(Cl)cnn1)=O 59158,S(=O)(=O)(c1cccc(F)c1Cl)N(C(COC)C)C 59159,c1(C(N2C(CNC(c3cc(C)sc3)=O)C(C)CCC2)=O)ccc2c(n1)CCCC2 59160,c1(CN2C(C(=O)Nc3c(C(C)=O)cccn3)CC3CC32)c(C)cc(Br)cc1C 59161,c1(C(C(C)C)C(=O)NC2CC(CF)C2)ccc(Br)cc1F 59162,c1(C(N2CC(NC(c3ccco3)=O)C(F)C2)=O)ccc(Cl)c(F)c1F 59163,c1(C(N(C(C)C)CCN(C2CCS2(=O)=O)C)=O)cn(CCCC(=O)O)nn1 59164,C(=O)(CC1CCc2ccc(O)cc21)N1CCC(=CCNC(COCC=C)=O)CC1 59165,c1(C(N2CC(O)C(C)(C)C2)C(=O)NC(C(C)C)(C)C#N)cc2cccc(Br)c2o1 59166,C(C#Cc1ncccn1)Nc1cccc(CN(C)C)c1 59167,C(CCC1CC1)(C(=O)NC(c1ncn(C)n1)C)NC(C(n1c(C)ncc1)C)=O 59168,CCC(C)CC(C(=O)OC)NC(C12CC(C)(C1)OC2c1ccccc1)=O 59169,C=C(C)CC(C(=O)N1CCC(CCCC)C1)NC(=O)C(C1CCOCC1)F 59170,c1(CC(=O)NCCN(C(=O)CN2CCCC2CO)CCOC)nonc1C 59171,N1(C(c2cc(C)no2)=O)CCCC(C(=O)NC2CN(CC(C)C)C2)C1 59172,C1(C(N(CCNC(C(c2c(OC)cccc2)(C)C)=O)C)=O)CCCCNC1=O 59173,C1(C(N2C(CC(=O)NC(C=C)(C)C)CCCC2)=O)CCC(=O)N(C)C1 59174,C(=O)(C1=NN(C)C(=O)CC1)N1CCC(C(C)NC(c2c(C)nns2)=O)C1 59175,N1(C(C(C=CC)O)=O)CCC(NC(=O)C=Cc2cccc(OC)c2)C(CO)C1 59176,c1(C(N2CCC(C(=O)OC)CC2)=O)n[nH]c2c1CN(C(=O)C(=O)c1ccco1)C2 59177,N1(C(c2coc(C3CC3)n2)C(=O)NCCC#N)CCCN(CCCO)CC1.C(N)(=O)N 59178,c1(C(=O)NC(CC)CN(C)C(C2CCOC(C)(C)C2)=O)ccc(=O)n2c1CCC2 59179,N1(Cc2c(OC)cccc2)CCC2(CC1)CC2C(N1CCCC1C(C)C)=O 59180,N1(C(C2N(CCCN=[N+]=[N-])CCCC2)=O)CC(C2CCCOC2)C1 59181,Cc1occc1CC(=O)N(CCNC(=O)C(C)n1cccc1)C(C)C 59182,C1(NC(c2c(C)sc(Br)c2)=O)CC2CCCC(C1)N2C(C1CC1(F)F)=O 59183,C12(CNC(CCC(=O)N(C)C)=O)CCC1CCN2C(=O)COC1(C)CCCC1 59184,Cc1ccc(CNC(C2CCCN(C(C3CC4CCC3C4)=O)C2)=O)c(O)c1 59185,Cc1nc(C(=O)NC2CCCC2(C)CN(C(=O)C(O)CC(C)C)C)cc(O)n1 59186,N1(CCNC(c2c(C)nc[nH]2)=O)CCC2(CCOC2)C1 59187,N1(C(C(C=C)OC)=O)CCSCC1C(=O)N(CC(C)(C)OC)C 59188,N1(C(C2(C(=O)N(CC)CC)CC2)=O)CC(C(N2CCC(C)(O)C2)=O)C2(CC2)C1 59189,c1(C(N(CC(C)O)CC)=O)cn(CCNC(C2OCCO2)=O)nn1 59190,C(C(C)(C)C(=O)NCCC1CCCN1C(=O)CC1CC2(CC2)C1)OC 59191,C(C)(CCC(C)(C)C)N.c1(-c2cn(C(C)C)nn2)nn(C)cc1C(N1CCC1C)=O 59192,C1(C(=O)OC)CCC2(CC2)N(CC2CCC3(CCC3)CN2)C1 59193,N1(C(C2N(CC)CC2)=O)CC(C)CN(C(c2cnoc2-c2cnccn2)=O)CC1C 59194,CC1=C(C(=O)NCC2CCC3(CCC3)C2NC(=O)CS(=O)(=O)N(C)C)COCC1 59195,C1(C(C)NC(c2nc(Cl)cs2)=O)CCCN(C(=O)CC23CCC(CC2)C3)C1 59196,c1(OC)cc(Br)c(NC(=O)C=Cc2ccc(C)s2)c([N+](=O)[O-])c1.C12CCCN1C2 59197,N1(C(C2C(CC)CCO2)=O)CCC(C(=O)NC(CN(C)C)C(C)(C)C)C12CCC2 59198,C(=O)(C1=CC2C=CC(C1)C2)NC(CCC=C)C(=O)OC 59199,Cc1nc(C(C)(C)C)c(C(=O)NCC2(NC(=O)CC3(O)CCCOC3)CCC2)s1 59200,C1(COC)(NC(C2CC3C(C2)C3(C)C)=O)CCCN(C(C2C=CCC2)=O)C1 59201,c1(CC2CC2)ncc(C(=O)N(C)CCSC(C)C)s1.C1(C(=O)N)(CO)CCCC1 59202,N1(C(c2ccc3ccoc3c2)=O)CCC2CN(Cc3c(OCC)nccc3)CC12 59203,c1(C(=O)NCC2(F)CC(NC(CSCC#C)=O)C2)ccc(C)c(S(C)(=O)=O)c1 59204,N1(C(CC(C)N(C)C)=O)CCCCC1CC(=O)NCC1COCCO1 59205,c1(NC(c2ccc3nc(C)oc3c2)c2n(CC)nnn2)ccc2ncnc(O)c2c1 59206,C1(NC(c2c(OC)cnnc2)=O)CN(C(C2CC(F)C2)=O)CCC1(C)C 59207,C1(NC(C=Cc2c(OC)cccc2)=O)C2CCN(C(=O)CCC3CCC3)CCC12 59208,C1(C(=O)NC2CC3(CC3)C2)CC(O)C(O)CC1CNC(C1CCCNC1=O)=O 59209,c1(NC(C2C(CNC(C3CC(O)(CC#C)C3)=O)CCC2)=O)ccc(Cl)cc1O 59210,N1(C(c2n(CC)cnn2)=O)CCC2(NC(=O)Cc3cc(Cl)sc3Cl)CC2C1 59211,N(C(=NCC1CCN(C)C1=O)NC1CCOCC1)C(C1(OC)CCOC1)Cc1ccccc1 59212,C1(NC(CC2CCC(=O)NC2)=O)CCN(C(=O)CC2C=CCCC2)C12CCC2 59213,C#CCCC(C(=O)NC(CCC)C(=O)NC)NC(=O)C(F)C(F)(F)F 59214,N1(C(C2(C)CC=CCC2)=O)CCC2(CC(C(=O)N3CC(N(C)C)C(F)C3)=NO2)C1 59215,C1(C(=O)NCC(CNC(c2cc(C)c(C)[nH]2)=O)OC)CCc2ncsc2C1 59216,c1(C(N2C(C)CC(O)C2)=O)cnc2c(-c3ccc4[nH]ncc4c3)cccc2c1 59217,C1(=CC(=O)N(C2CCN(C(c3ccc(C(C)=O)[nH]3)=O)C2)C)CC2CCC(C1)N2C 59218,C1(NC(=O)NC(c2c(C)cccc2)CN(C)C)CC2(C1)CC1(CC(O)(O)C1)C2 59219,C(=O)(C1=Cc2ccccc2C1)NCC(C(=O)N(C1C(C)OCC1)C)(F)C(C)C 59220,N1(C(C2CCCC3(CC3)C2)=O)CCC2(CC1)CN(C(=O)C(O)C1CCC1)C2 59221,c1(OC)cc(-c2ccc(F)cc2F)c(OC)cc1CN1CCCC(N(C)C)C1 59222,C1(C(=O)OCC)(NC(=O)CNC2(c3nc(C(=O)OC)sc3)CCCC2)CC1(C)C 59223,C#CCC(C)(C(=O)N(CC#CC)CC)NC(=O)C(CN(C)C)N(C)C 59224,C(=O)(C1=CCCOCC1)N1CC(CN(c2nc(C(=O)OC)c(Cl)cn2)C)OCC1 59225,CC1CCN(C(c2nonc2N)=O)CC1NC(c1cn(C)c(=O)n1C)=O 59226,N1(C(c2c(OCC)nccc2)=O)CC2(CCN(C(=O)CC(C)SC)CC2)CC1C 59227,N1(C(C)CNC(=O)NC2CC3(C2)CC(CF)C3)CCS(=O)(=O)CC1 59228,C1(OC)(CNC(C2(C)CC=CCO2)=O)CCN(C(c2nccnc2C)=O)C1 59229,c1(C(=O)NCC2(OC)CN(c3cc(C(=O)OC)ncn3)C2)cc(F)ccc1F 59230,C1(C)(C(C)NC(c2cc(C3CC3)ns2)=O)CCN(C(=O)C(C2CCOCC2)F)C1 59231,C1(C(N2CC(C)(NC(C(C)N(C)C)=O)C2)=O)CCCCN1Cc1ccccc1 59232,c1(OC)ccc(COCc2nocc2C)cc1C(=O)OC(N)=O.C(CCOC)O 59233,C1(OC)C(NC(=O)CCN(C)C(c2cc(O)n(C)n2)=O)CC1(C)C 59234,C1(C(=O)Nc2nccnc2CC)COCCN(CC2(C#C)CCCC2)C1 59235,c1(N(C)C#N)ccc(-c2ccc(-c3ccc(C(=O)N(C)C)cc3)o2)cc1 59236,C12(C(N3CC(CC)OCCC3)=O)CCC(CC1)N(C(c1ncncc1Cl)=O)C2 59237,c1(C(=O)NCC(CC)NC(C2CC(=O)N(C)C2)=O)cnc(C)cn1 59238,C1(CC(=O)Oc2ccc(OCCCC)cc2)NC(=O)CNC1=O 59239,CC(C)CC(CNC(=O)C(C(C)C)n1ccnc1)NC(=O)CCc1cc(Cl)no1 59240,O=C1CCCC(CCc2cn(CCCC(=O)NCC3CC3(F)F)nn2)C1 59241,C1(C(CNC(C2(CNC(=O)C(F)CC3CCC3)CC2)=O)O)CC(F)(F)C1 59242,N1(C2C(C)OCC2)CCN(C(c2ccc(CNc3cccnc3N)cc2)=O)CC1 59243,c1(CCC(=O)NC2CC(NC(C3(CC)CCOC3)=O)C2)ccncc1Br 59244,Cc1nc(C(=O)NCCC2CC(C(=O)N(C3CNC(=O)C34CC4)C)C2)cc(O)n1 59245,c1(C(N2CC(CNC(CC(C)C(F)F)=O)OCCC2)=O)ccc2nn[nH]c2c1 59246,c1(C(N(CCNC(c2n(C=C)ncc2)=O)CCOCC)=O)cc2cnccc2[nH]1 59247,Cc1cc(Cl)c(C(N2CCCC2CN(C(=O)C(C)CC(C)C)C)=O)cc1[N+](=O)[O-] 59248,c1(OCC(N2CC(NC(CC=C=C)=O)C3C2C3)=O)ccc2c(c1)CCC2=O 59249,N1(C(C(N2CCN(C)CC2)C)=O)CCN(C(c2ccc(N)c(N)n2)=O)C(C)C1 59250,c1(-c2cnc(NC(Cc3ccc(OC)cc3F)=O)c(C)c2)cnc(C#N)c(F)c1 59251,C1(NC(c2c(C)noc2)=O)CCN(C(c2csc(CC(C)C)n2)=O)C1(C)C 59252,C(CC(=O)N1CC2(CC(N(C)C)C2)C1)(C(F)(F)F)NC(C(C)SCC)=O 59253,C1(NC(c2n(C3(C)CC3)nnn2)c2cnc(Br)s2)CCC(C2CC2)C1 59254,C12(C(=O)NC3C(NC(c4n(C=C)ncc4)=O)CCC3)CCC(CO)(CC1)CC2 59255,N1(C(c2n(CC)nnc2)=O)CC(C)CN(C(C2CCC3(C2)CC3(F)F)=O)C(C)C1 59256,C12(CNC(C3C(C)OCC3)=O)CC(C(N)=O)(C1)C1(CN(C(=O)CCN(C)C)C1)O2 59257,C(=O)(C=C1SCC(=O)N1C)N(C)CCC1CCCCN1C(C1(CC2CC2)CC1)=O 59258,C1(C(=O)NCc2ncoc2C2CN(C(=O)COC(C)=O)C2)(OCC)CCCCC1 59259,C12(C(N3CC(O)(CCC)C3)=O)CC1CCN2C(c1ccn(C2CC2)n1)=O 59260,CC1CCc2c(C(=O)N(CC(O)CNC(c3ccc(O)cc3)=O)C)csc2C1 59261,C1(CCC)CN(C(=O)CC(C)COC)CCN1C(c1cn(C)nn1)=O 59262,c1(OC)cc(C(N2CC(NC(=O)CCc3n[nH]c(=N)s3)CC(O)C2)=O)cc(C)c1 59263,C=CCC(CC(F)F)ON.c1(C(NC)=C)ccc(F)c(C)c1 59264,N1(C(c2n(CC)cc(Cl)c2)=O)CCCC(O)(CNC(C2CN(C)CCO2)=O)CC1 59265,c1(N(C(C2C3CCC2(c2ccc(Br)cc2)C3)=O)CC)cccc2c1OCCO2 59266,N1(CC)N=C(C(=O)NCC2CCN2C(c2ncc(OC)nc2OC)=O)CCC1=O 59267,C(CCCCC(=O)N1CCC(C)(CNC(=O)CC2CS(=O)(=O)C2)CC1)=CC 59268,N1(C(C(C)P(C)(C)=O)=O)CCOC2(C1)CN(C(C1CCC1C(F)F)=O)C2 59269,C1(C(=O)NCC(C)CC2CCC2)CCN(C(=O)c2ccnc(O)c2)O1 59270,c1(CNC(c2n(CCCSCC)nnn2)c2ncc(C)s2)ccc(F)c(C)c1Cl 59271,C1(NC(CC=C=C)=O)CCN(C(c2ccc(CNC(C)=O)o2)=O)C1C(C)(C)C 59272,C(=O)(C1CCCc2sc(=N)[nH]c21)NCCC(C)NC(=O)C(F)(F)c1ncccn1 59273,C(C(=O)NCC1(CNC(=O)C(C)OCOC)CC1(F)F)(C(C)C)SCC 59274,Cc1cc(Cl)c(C(=O)NCC2CCCN(C(=O)NCc3nc(C)c(C)s3)C2)s1 59275,c1(C(N2C3CCN(C(c4c(CC)nc[nH]4)=O)CC3C2)=O)cn2ccc(F)cc2n1 59276,c1(CC(N2C(C(N3CCN(C(C)=O)CC3)=O)CC2)=O)cc(F)cc(Cl)c1 59277,c1(C(=O)NC2CCN(CC#CC)CC2C)nc[nH]c2nccc1-2 59278,C(=O)(CCC(C)CC)N1CCC(CC=C)(C(N2CC(CS(C)=O)C2)=O)C1 59279,C1(CC(N2CCN(C3CCCN(C(=O)CSCC)C3)CC2)=O)CCCC(C#N)C1 59280,O(P(C)(=O)CNC(C1CC(F)CN1C(=O)CC1CCCOCC1)=O)CC 59281,CCCCCCCCNC(=O)C(=O)NCC(C(C)C)C(c1cc(N)nc(Cl)c1)=O 59282,N1(C(CC(N(C(=O)C2CC2)CC)Sc2cccc(C)c2)=O)CCCN(CC)CC1 59283,C12(CNC(c3c(C)nsc3)=O)CCCC1N(C(=O)C(C)C1CCOC1)CCC2 59284,C1(CNC(C(CC)n2ccnc2)=O)CN(C(=O)CC(CC)C2CCC2)CCO1 59285,N1(C(C(=O)NCCOC)CCC2(C)CC2)CCCC2(CCCOC2)C1 59286,c1(C(N2CC(CCNC(C3CC(SC)C3)=O)(OC)C2)=O)cnc2cc[nH]c2c1 59287,C1(CNC(c2nc(COC)oc2)=O)CCN(C(C2CC3(CC3)C2)=O)CC1O 59288,C1(C(=O)Nc2cn(CCC)nc2)CSCCN1C(c1cc(C(C)C)[nH]n1)=O 59289,C(=O)(C(C(C)(C)C)NC(N)=O)NC1C(CNC(c2c(C)cno2)=O)C1 59290,CCC(C(=O)NCC1CC2(C1)CN(C(c1ccc(CSC(F)F)o1)=O)C2)C(C)O 59291,Cc1ccc(C(=O)NCC2CN(C(C3CCC3C(C)(C)C)=O)CCO2)c(F)c1Cl 59292,C(=O)(CCCCSC1CC1)NC(C1CC(C)(C)C1)C(C)NC(c1ccccc1)=O 59293,c1(C(=O)NC(CCCNC(C(C)NC(C)=O)=O)C)ccn2ccnc2c1 59294,C1(CN(C(C2CC(C(F)F)(OC)C2)=O)C)CCN(C(C2CC(O)C2)=O)CC1 59295,C(N=c1nc(OC)c2ccccc2[nH]1)C1(CNC(CS(CC)=O)=O)CCC1 59296,C1(C(=O)NC2C(NC(c3cnc(C4CC4)s3)=O)CCCC2)CS(=O)(=O)CCO1 59297,N1(C(C=CCOC)=O)CC(O)CC1C(N1CCCC1C1(C)CC1)=O 59298,c1(C(=O)NC2CC(CNC(C3C(C)C3)=O)C2)ccccc1C(C1CCCCO1)=O 59299,N1(C(c2cnc(CC)[nH]2)=O)CCC(CC)C1CNC(=O)C(CC)SC 59300,C1(Br)(C(=O)NCCOCCN(C(C2(C)C(C)C2)=O)C)CC1(F)F 59301,N1(C(c2cn(C)nc2Cl)=O)CC2CC(C1)C(CO)C2NC(c1cccc[n+]1[O-])=O 59302,N1(C(=O)OC(COC(CC)C)C(C)C)CCC(C)(C(=O)OC)CC1=O 59303,c1(C(CC)CN(C2CC2)C(c2nc[nH]n2)C)ccccc1 59304,CCCC(C)CC(=O)N1CC(CCO)(NC(C2COCCN2CC)=O)C1 59305,CC1(NC(C2CCCN(S(C)(=O)=O)C2)=O)CCN(C(=O)COC(F)F)C1 59306,N1(C(C(CC)F)=O)CCC(N(C)C(c2ccn(C3CCC3)n2)=O)C2(CC2)C1 59307,CC(C)CC(O)C(=O)NC1CN(C(c2cccc(CC(F)(F)F)c2)=O)CC1C 59308,CC1CC(N=c2c(Br)c[nH]cc2[N+](=O)[O-])CN1C(c1nc[nH]c2nccc1-2)=O 59309,C(CC(C)CCNC(c1cc(C(C)CC)no1)=O)NC(CCCOCC)=O 59310,c1(OC)ccc(C(=O)NC2CN(C(c3coc(O)n3)=O)CCC2O)c(OC)c1 59311,C(=O)(C(CCOCC)NC(=O)C(C)C1CCCC1)N(CC=C)CCOC 59312,CC1(CNC(=O)CN(C(C2OC3CCC2C3)=O)CC2CC2)CC=CCC1 59313,c1(C(=O)NCC(C)(C2CC2)NC(CC(C)OC)=O)c(Cl)c2ccccc2n1C 59314,C1(NC(C2CC(CCC)C2)=O)CCN(C(c2cnn(CCC#N)c2C)=O)CC1 59315,C(=O)(C(C)CC(F)F)NC1C(NC(CCc2cccc(C)c2)=O)CCCC1 59316,c1(C(=O)OCC)cccc(S(=O)(=O)NC(c2cnsc2)C)c1 59317,C(=O)(C#CC(C)(C)C)NCc1c(C(=O)NCC2(O)CCN(C)C2)nco1 59318,C(=O)(C(C)(C)CC#N)N1C(C)CC(CNC(=O)C=CCOCc2ccccc2)C1 59319,N1(C(C(=O)N(C(C)C)CC2CC=CCC2)=O)CCOC2(CCS(=N)(=O)CC2)C1 59320,C1(C2(O)CCOC2)(C(N(CC)CC2CCCN(C(c3scnc3C)=O)C2)=O)CC1 59321,n1(CC(=O)NCC2CC(NC(=O)C(O)C3CC3)C2)cc(Br)cn1 59322,c1(OC)cc(OC(F)F)[nH]c(=NCc2ccc(CN3CCC(CO)CC3)cc2)n1 59323,Cc1nc(C2CCCO2)sc1C(=O)N(C)CC1CCN(C(=O)CC2(O)CCC2)C1 59324,C1(CC)(Nc2nnc(SC)s2)CCN(c2nnnn2-c2cccc(C)c2)CC1 59325,n1(CC2(C)CC2)nc(SC#N)nc1CCC1CSC1 59326,C1(NC(=O)NCc2nc(C(C)C)oc2)CCCC(O)CC1 59327,C1(C(N2CC(CC(=O)OCC)C2)=O)C(C)OCCN1C(c1c[nH]c(=NC)o1)=O 59328,C1(NC(C(CC)N(C)C)=O)CCCN(C2CCc3ccc(Cl)cc32)C1 59329,CC1(CO)CCCN1C(c1ccoc1CNC(c1cnn(C2CC2)c1)=O)=O 59330,C1(OCCNC(CC2C(C)CC2)=O)CCN(C(c2cnn(CCO)c2)=O)CC1 59331,C1(NC(c2sc(N(C)C)nc2C)c2n(CCCC)nnn2)CC(O)CC(C)(C)C1 59332,C(=O)(CC(C)(C)CN(C)C)N1CC(OC)C(NC(c2sccc2Br)=O)C1 59333,C1(c2ncc(C(=O)OC)s2)CCN(C(=O)N(C)C)CC1.C1CCNS1 59334,C(=O)(C(C)C(C)COC)NCC#CC(=O)NC(CC#C)C 59335,N1(C(=O)CCc2cscn2)CC(NC(C23CC(c4ccccc4)C2C3)=O)C(O)C1 59336,c1(C(=O)NCC2(CCNC(CC(CN(C)C)O)=O)CC2)cc(C)cc(Cl)n1 59337,C(CCCCC(=O)N1CCCC(CC(=O)NC(C)(C)CCCO)CC1)=CC 59338,C1(NC(C(CC)(C)OC)=O)CC=C(C(=O)NCC(C)(C)CO)C1 59339,N1(C(C2(CC=C)CCCC2)=O)CCN(CC(C)NC(=O)C(C)CC=CC)CC1 59340,C1(C(=O)NCC(C)N(C(c2sc(C)c(Br)n2)=O)C)CNC(=O)C(C)(C)C1 59341,c1(C(=O)NCC(CC)NC(=O)CCc2ccnn2C)cn(CCC(C)C)nn1 59342,N1(C(C(C)CC(C)(C)C)=O)CCC2CCN(C(=O)Cc3cc[nH]n3)C2C1 59343,C1(C(N2C(C)(C)C(CO)CC2)=O)N(C(c2cc[n+]([O-])cc2)=O)CC12CCCC2 59344,c1(-c2cn(C)nc2)cccc(C(=O)NCC2CC(NC(=O)CC=CC(=O)O)C2)c1 59345,C(C)(CNC(=O)CC1CCOCC1)(C(C)C)NC(C(c1ccccc1F)C)=O 59346,c1(C(N(CCC2N(C(CS(=O)(=O)NC)=O)CCCC2)C)=O)ccc2ncnn2n1 59347,c1(C(N2C3CC(NC(C(CC)(C)O)=O)CC2CC3)=O)cccc2oc(C)nc12 59348,CC1(C)CCN(C(C23CC2COC3(C)C)=O)CC1CNC(=O)C=CBr 59349,C1(C(=O)NC(C(C)C)CO)(CO)CCN(C(c2ccc(C(F)F)o2)=O)C1 59350,c1(C(=O)OC)ncc(N2CCC(OCC)C2)nc1C.C(=O)CC(C)(O)C1CC1 59351,C(=O)(C1=CCCN(C(=O)CC2(C)CC2)C1)NC(C)CN1CCC1 59352,Cc1[nH]c(C#N)cc1C(=O)NC1CCCCN(C(=O)CC2CC3CC3C2)C1 59353,CCCCC(C)C(=O)NCCOC1CN(C(=O)C(c2ccn(C)c2)C)C1 59354,CCCCC(C(=O)NCCN1CC(CF)C1)NC(C1CCOC(C)(C)C1)=O 59355,C12(NC(c3cnc(C4CC4)o3)=O)CCCC1N(C(c1ncccn1)=O)CCC2 59356,C1(C(N(C)Cc2cncs2)=O)CCCCC1(C)NC(C1(c2nccs2)CC1)=O 59357,N1(C(C(C=C)(C)C)=O)CC2CC(NC(=O)CC(C)n3cccn3)C2C1 59358,C1(C(N(CCN(C(=O)CCCc2nncn2C)C(C)C)C)=O)CCC(C)(C)CC1 59359,c1(C(N2CC3C(CNc4nc(OC)nc(OC)n4)(C3)C2)=O)ccc(C#N)cc1Cl 59360,Cc1ccc2c(c1)N(C(=O)C(CNC(=O)Cc1ccc(O)cn1)C(C)C)CC2 59361,CC(C)CCCC(=O)N1CCC(C=CC(=O)NC(CO)CC(C)C)CC1 59362,C1(C(=O)NCc2nc(C(C)C)on2)CN(C(=O)CCc2ccccn2)CCN1 59363,c1(OC)cc(Cl)ncc1C(N1CCN(C(c2oncc2C)=O)CC1CC#N)=O 59364,Cc1ncn(C)c1C(=O)N(C(C)CNC(c1cnn(CCO)c1)=O)C 59365,n1(CCC)nccc1C(=O)NCC(c1ccccc1)NC(C12CSCC1C2)=O 59366,C1(NC(=O)CCc2ccccn2)CCN(C(c2coc(O)n2)=O)C12CCCC2 59367,c1(OC)cnc(C(N2CCC(N(C(=O)C(c3ccc(F)cc3)F)C)C2)=O)c(F)c1 59368,c1(C(N2C(CC(C)O)CC(C)CC2)=O)cnc2c(Br)c[nH]c2c1 59369,N1(C(C=CC2N(C)CCC2)=O)CCC(NC(=O)Cn2ccnn2)C2(CCC2)C1 59370,C1(C(=O)NCC2C(C)OCC2)C2CC3C(C2NC(C2CN(C(N)=O)C2)=O)C13 59371,c1(OC)cc(NC(C2CCCC(NC(c3cnnc(O)c3)=O)CC2)=O)ccc1O 59372,C(=O)(C(CCC(C)C)Nc1nonc1C)NC(C1CN(C(C)=O)C1)=O 59373,C(CN(C(C(=O)NCC1CC1)c1cncs1)C)(CO)(CO)OC(C)C 59374,Cc1cc(-c2cn(C3CC(C(=O)Nc4ncccc4F)C3)nn2)cc(F)c1 59375,Cc1nc(Cl)[nH]c(=NC2CN(C(=O)CCN3CCCC3=O)CC23CCC3)c1C#N 59376,C(=O)(C(=O)C(C)(C)C)NC1(CNC(c2n[nH]c(C)c2C)=O)CC1 59377,N1(C(c2n(C)cc(N)c2)=O)CCCN(c2ccnc(NCc3ccoc3)n2)CC1 59378,c1(C(=O)NC2CC(NC(c3sc(C)c(Br)c3)=O)C2)cccc(F)c1N 59379,CN=c1[nH]c(=NC2C=CCCCC2)[nH]c(=NC2COCC2OC)[nH]1 59380,N1(C(CC2(C(=O)OCC)CC2)=O)CCCC(C(C)NC(=O)C(F)=C(C)C)C1 59381,C1(NC(C=CCCC)=O)CCC(C)(CNC(c2cnc(O)o2)=O)C1 59382,N1(C)CCN(C)CC1.c1(OC)nscc1C(=O)OC.n12cc(nn1)CN(C1CC1)C(C)C2 59383,c1(CC(CNC(COC2CN(C(C)=O)C2)=O)NC(c2cnco2)=O)ccccc1 59384,c1(NC(C)Cc2ccco2)[nH]c(=NCc2cccc(F)c2Cl)nc2c1cnn2C 59385,c1(C(N2CC(NC(CC(CN(C)C)(C)C)=O)C2)=O)ccc2c(c1)OCCC2 59386,Cc1cc(C(=O)NC(CNC(c2c(C3CCC3)cnn2C)=O)CO)cc(F)c1 59387,C1(C(=O)NCCCNC(c2cnn3ccn(C)c32)=O)C2CCN(CC2)S1(=O)=O 59388,C1(S(=O)(=O)CCN2CCCC(C(N)CO)C2)(CC=C)CC1 59389,CCC(C)(C)C(O)C(=O)NC1(CNC(=O)C(C)(C)c2cscc2Cl)CCCCC1 59390,C(CN=C(NC1CC2(CC2)C1)NC1Cc2ccccc21)c1ccc(N(C)C)cc1 59391,CC1(F)CC(C(=O)NCC(CNC(=O)CNC=O)CO)C1 59392,N1(C(c2nccc(CC)c2)=O)CC2(CCN(C(=O)CCN(CC(F)(F)F)C)C2)C1 59393,C1(CC(=O)NC2C(CC)CN(C(=O)COCP(C)(C)=O)C2)CC(C)(C)CCO1 59394,c1(C(N2CCC(N(C(CN(C)CC)=O)CCO)C2)=O)ccc(C(C)(C)C)cc1C 59395,N1(C(CC(C)(C)C)=O)CCC2C(C1)OCCN2C(c1cc(Cl)ccn1)=O 59396,C(=O)(CCCOC1CC(NC(=O)CNC(C2CC2C)=O)C1)OC 59397,C(=O)(C(C)C(F)(F)C(F)F)N(CCNC(c1coc(C2CC2)n1)=O)CC 59398,C1(C(N2C(CCNC(C(C)(C)CO)=O)CCC2)=O)Cc2ccc(Cl)cc2C(=O)O1 59399,c1(NC(c2nnnn2C2CCC2)C2(C(=O)OCC)CC2)ccc(Br)c(Cl)c1 59400,CC1(C(=O)NCC2(O)CC(NC(=O)CSC3CC3)C2)CCC(O)CC1 59401,Cn1cnc2c1CCN(C(=O)C(F)C(F)(F)F)C21CCN(C(=O)CC2(C)CC2)C1 59402,c1(C(=O)NC2(C3CCCN3C(=O)C(F)=C3CCCC3)CC2)cc(C(F)F)c[nH]1 59403,C1(C(=O)NCC2(CNC(=O)OC(C)(C)C)C(C=C)C2)CCOC2(CCCCC2)C1 59404,Cc1[nH]nc2cc(NC(=O)Cc3cccc4c3OCCC4)ccc12 59405,C12(C(N(C3CCCN(C(C(CCOC)C)=O)CC3)C)=O)CCC(CC1)C2(C)C 59406,C1(C(=O)NCC2(C(F)F)CCN(C(Cc3c(C)ccs3)=O)C2)CCC2(CCC2)C1 59407,C1(N(C)CC)CCN(C(=O)CC(=O)OC(C)C)CC1.c12cnc(s1)C(=O)OC2 59408,c1(C(N2CC(O)(CNC(C(CC)(C)C#N)=O)C2)=O)cn2ccc(C)cc2n1 59409,c1(C(N2CCC(CN(C(CCC=CC)=O)C)C2)=O)csc(Br)c1C 59410,c1(C(=O)NC(C(C)NC(C(CC)(C)CC)=O)C)cccc(F)c1C#N 59411,C=CCCCC(C(=O)N(CCCC(CC)CC)C)NC(=O)C(OC)OC 59412,c1(SCC)ccc(C(=O)NC2CCCC(C(N3CCSCC3)=O)C2)cc1 59413,C1(C)(C(N2CC(CN(C(C(CC)(C)C)=O)C)OCC2)=O)CC(=O)N(C)C1 59414,CN1CCC(C(=O)N(C2CC2)CC2CC(NC(=O)CC3CN(C)C3)C2)C1=O 59415,C1(CC)CN(C(C2(n3cc(CS(C)(=O)=O)nn3)CC2)=O)CC(C)(C)O1 59416,N1(C(c2ccc(C)o2)=O)CCC(CNC(c2nc(Cl)cs2)=O)C(O)C1 59417,CC1(C)CCCC(O)(CNC(=O)Cn2cc(C3(C)CCCO3)nn2)CC1 59418,C(=O)(C(COC)CC)N(CC(C(N1CCC(OCC=C)C1)=O)O)C 59419,C=CC(C)(C)CC(=O)NC1CC(F)(F)CC1NC(=O)Cc1cccc(F)c1F 59420,C1(CC(N2CCC(c3cnco3)CC2)=O)CNCCS1(=O)=O 59421,C1(C(=O)NC2CCN(C(c3cc(C(C)=O)[nH]n3)=O)C2)CC12CC(C)(C)C2 59422,C(C(CNC(c1cncc(N)n1)=O)C(F)(F)F)NC(c1c(C)ccs1)=O 59423,c1(C(N2CC(NC(c3ccc(C)cc3Cl)=O)C2)=O)cc(Br)cc2c1OCC2 59424,c1(CC(=O)NC(C2CCN(C(C3CCC3(C)C)=O)C2)C)coc2ccccc12 59425,Cc1nn2cc1C(=O)OCC2.C1(COc2ccccn2)CCCCCC1 59426,CCC(C)C(C)C(=O)N(C(C)CNC(=O)Cc1csc(C(=O)OC)c1)C 59427,CC1CN(C(C2CC2c2ccnn2C)=O)CC1NC(c1cnsn1)=O 59428,Cc1cc(CCC(=O)NCCC2CN(C(=O)CN3C(C)CCC3C)C2)cc(C)n1 59429,N1(C(CN(CCC)C)=O)CCC2(NC(C3CC3CF)=O)CCCC12 59430,CC1CN2CCN1C(C(N1CC(CNC(=O)CCc3ccc(N)cc3)C1)=O)C2 59431,O=C1NCC2(CCN(C(C3CSCCN3C(=O)C(O)CC(F)(F)F)=O)C2)O1 59432,C1(C(=O)NC(COC(C)=O)CO)(COC)C=CCN1C(=O)C(n1ccnc1C)C 59433,CC1(C)CN(C(=O)CC(CNC(C2(C)CC3CC3C2)=O)C2CCC2)CCCO1 59434,C1(C(=O)NCC(C)N(C(c2c(OC)nn(C)c2)=O)C)CCc2ccc(F)cc2O1 59435,C1(C(=O)OC)COCC1NC(=O)CNC(=O)C=CCN1CCC1 59436,Cc1cc(S(N)(=O)=O)cc(-c2cc(N)c(C#N)c(F)c2)c1C 59437,C(=O)(CCC(F)(F)F)N(C)CC1CCCN1C(C1CC(CC(F)(F)F)C1)=O 59438,C12(C(N3CCCC(C)C3CNC(=O)Cn3cc[n+](C)c3)=O)CC=CCN1CCC2 59439,N1(CC(=O)NC(=O)NCC)CCCN(C(C2CCCC(OC)C2)=O)CC1 59440,Cn1nc([N+](=O)[O-])cc1C(=O)NC1CCC(NC(c2ccc(F)c(F)c2N)=O)C1 59441,c1(C(=O)NCCC(=O)NCc2cnc(CC)o2)cc(CC)oc1C 59442,C(C)(CCC(=O)Nc1ccc(C(=O)NOCC=CCl)o1)OCC 59443,c1(NC(c2c(CCCN)ccs2)=O)nccc(CCCN2CCCC2)n1 59444,c1(C(=O)NC2CCCCCN(C(C(CC)(C)CO)=O)C2)cc(F)c(Cl)c(N)c1Cl 59445,CCC(C)CC(C)C(=O)NC1CCCC1CNC(c1ccccc1Cl)=O 59446,C1(NC(c2cncc(C#N)c2)=O)CC2CCC1C(NC(C1CCCC1(F)F)=O)C2 59447,C12(C(=O)NC3C(NC(c4cc(C)n(C(F)F)n4)=O)C3)CCC(C)(C(=O)O1)C2(C)C 59448,C1(C(N2CC(C=C)(CC(N3CC(N(C)C)CC3C)=O)C2)=O)CC2(CCC2O)C1 59449,c1(C(=O)NCCCN(C(=O)CCC2CCCO2)C)ccc2c(Cl)nccc2c1 59450,C=CC(C)(C)C(=O)NCC1CCCN1C(=O)CCc1ccoc1.CC1CCC1 59451,N1(C(C2CC(F)CN(Cc3nc(Cl)ccc3F)C2)=O)Cc2cccc(F)c2C1 59452,c1(CC)ccc(C(N2CCOCC2CC2CN(C(=O)C(C)C(F)F)C2)=O)cc1F 59453,C(=O)(CCCCC(F)(F)F)NCC(C(C)C)NC(CC(CC)C)=O 59454,c1(C(N2CCC(NC(CC(CC)O)=O)CC2C)=O)c(C)nn2cccnc12 59455,N1(C(c2cnsn2)=O)CCC2CCC(C1)N2c1cnc(F)cn1 59456,c1(C(C)OC)nc(C)c(C(=O)NC(C)(CNC(=O)C2CC2)CO)s1 59457,C1(C)(c2cn(CC(=O)NCC)nn2)COCCN1C(C1CCCCC1(C)C)=O 59458,N1(C(c2ccon2)=O)CCC2(CCCN2C(c2ccn(C3CCCC3)n2)=O)CC1 59459,N1(C(c2cc(OC)cc(F)c2)C(=O)NCC(F)F)CC2CCCCCC2(C#N)C1 59460,c1(C(N(C(CNC(c2cnsn2)=O)C2CC2)C)=O)ccc(=O)n2c1COCC2 59461,C(CCS(C)(=O)=O)(C(=O)N=S1(=O)CCCCCC1F)OC 59462,Cc1c(C(=O)NC2CCC(CNC(c3n[nH]cc3C(C)C)=O)C2)sc2nccn12 59463,Cc1cn2cc(CC(N3CCC(O)(C(C)NC(=O)C(C)C)CC3)=O)nc2s1 59464,N1(C(C2CCN(C)C2)=O)Cc2ccc(C(N3CC4CC3CO4)=O)cc2C1 59465,N1(C(COC)=O)CCCC(C)C1CNC(c1ccnc(I)c1)=O 59466,N1(C(C(N)c2ccco2)=O)CC2COCC2(C(N2CC(O)C(F)C2)=O)C1 59467,C(CCN=C(NCC(=C1CCCC1)F)NCC1(C)CCS(=O)(=O)N1C)OCC 59468,N1(C(C(C(C)C)NC(=O)OCC)=O)CCCN(CCNC(=O)CC(C)CF)CC1 59469,c1(CC)cc(C(=O)N(C2CCN(C(C3(CF)CCOCC3)=O)C2)CCO)ncn1 59470,c1(C(N2CCCC(O)(CNC(c3c(C)oc(Cl)n3)=O)C2)=O)ccc2nncn2c1 59471,C1(NC(c2ccc(C(F)F)nc2)=O)CC2CC1CN2C(=O)C1=CCC1 59472,N1(Cc2cccc(C(=O)OC)c2)CC2CCC(C1)N2C(c1cccc(CO)c1)=O 59473,C1(CNC(C2N(C(C(c3cnn(C)c3)C)=O)CC2)=O)CC2(CC2)CO1 59474,c1(CN(C(Cn2c(C)ncc2)C)C=O)cccc(Cl)n1 59475,c1(C(N2CC3C(CNC(c4[nH]cc(C)c4)=O)(C3)C2)=O)ccsc1S(N)(=O)=O 59476,c1(C(=O)NC(C)CNC(=O)C(=O)Nc2cc(F)ccc2F)occ2c1CCCC2 59477,N1(C(C2CC(=O)NC(=O)N2)=O)CC2(NC(=O)C3CC3)CCCC2(F)C1 59478,N1(C(COCCSC)=O)CCCN(C(c2cccc(F)c2N)=O)C(C)C1 59479,Cc1nc2ncnn2cc1C(=O)N(CC(O)CN(C(=O)CO)C)C 59480,c1(OC)cc(OC)c(NC(C2CC2NC(=O)Cc2ccncc2)=O)cc1Cl 59481,c1(C(=O)NCc2ccc(-c3cccc(CC(=O)OC)n3)cc2)cc(O)cc(Cl)c1 59482,c1(OC)cncc(C=CC(=O)NCCCCNC(=O)C(C(=O)C(F)(F)F)=O)c1 59483,c1(C(N2CC(C(C)NC(C3CC(C)OC3)=O)C2)=O)ccc2nn(C)cc2c1 59484,N1(C(C(C)(C)OC)=O)CCC(C)(CCNC(C2CC2C2CC2)=O)C1 59485,C(=O)(CCCCCc1ccccc1)NC1C(CNC(c2ccc(SC)s2)=O)C1 59486,CC1CC(=O)NC1C(=O)NC(c1ccnn1C)C(N1CCC(OCC2CC2)C1)=O 59487,c1(SCCNC2(CS(N)(=O)=O)CCC2)ccc(Br)cc1 59488,c1(N2CCC3(C(C(=O)Nc4cc(OC)cc(F)c4)C3)C2)ncnc2occc12 59489,Cc1nc(C)n(CC(=O)NCc2occc2C(=O)NC(c2cncs2)C)n1 59490,c1(N(C(C2C(C(=O)OC)C2)=O)CC#N)ccccc1NC(c1cccc(Cl)c1)=O 59491,c1(C(=O)NC2CCN(CCC3N(CC)CCC3)C2)cc2ccccn2n1 59492,c1(CC)cc(C(=O)NCCCCC(C)NC(=O)CCCc2ccccn2)ccn1 59493,N1(C(C(CNC(CC(CC)(C)C)=O)O)=O)CCN2CC(C)CC2C1 59494,N1(C(C2C(C)(Br)C2)=O)CCC(NC(c2nccs2)=O)C(F)C1 59495,CCCCC(C(=O)N1CC(C)C1C(=O)N(C)CCOCC1CC1)N(C)C 59496,c1(C(N2CCC(NC(=O)OC)CC2)C(=O)NCC(=C)C)cc(C(C)C)oc1C 59497,CC1=NOC(CCNC(c2nnnn2C(C)(C)C)COc2ccccc2)C1 59498,C(=O)(CCCN=[N+]=[N-])NC1CCC(C(=O)OC(C)(C)C)C1.C12CCC1CC(=O)N2 59499,Cc1ccc(C)c(C(N2CC(O)CCC2C(=O)NCCCN(C)C)=O)n1 59500,c1(CC(=O)NCC2CCN(C(C(C(CC)C)O)=O)C2)ccc(OC)c([N+](=O)[O-])c1 59501,C(=O)(CCCCC1CC1)N(C1CCN(C(=O)CC2C(=O)NN=C2C)CC1)CC 59502,C1(CC(=O)N(C(C)CNC(C2CCCN2c2cnccn2)=O)C)CCCC12CC2 59503,c1(C(N2CCC(OC)(CNC(=O)C(C)c3ccco3)C2)=O)ccc(F)c(F)c1N 59504,C(=O)(C#CC1CCCC1)NC(CC)CN(C(=O)C(C1CCOCC1)OC)C 59505,c1(OCC=C)ccc(CC(=O)NC2CC(F)(CNC(C3CCC(F)C3)=O)C2)cc1 59506,CC1(C)CCCC(C(=O)NC2CCN(CCCNC(=O)Cc3ccon3)C2)C1 59507,c1(CC(=O)NC2C(NC(c3c(CC)con3)=O)CC2)ccc(C)cc1F 59508,C(=O)(C1OCCn2ccnc21)NC(CNC(c1c(NC)ccc(F)c1)=O)CO 59509,C=C(Cl)CN=C(NC1CCC1)NC1CCC(=O)N(C)C1 59510,CC1ON=C(C(=O)N2CCN(C(=O)CS(=O)(=O)N(C)C)CC2CO)C1C 59511,CCCCCC(C)CC(=O)NC(C)(C)C(C)NC(=O)CC(C)(C)CN(C)C 59512,CC1CN(C)CCC1NC(C1(C)CC(O)CN1C(=O)C=Cc1cscn1)=O 59513,CCC(CC(=O)N1C2CCC1CC(CNC(C1CCOC1)=O)C2)C(C)C 59514,N1(C(C)C)N=C(C(=O)NCC2CC(O)(CNC(=O)Cn3cccn3)C2)CCC1=O 59515,Cc1ccc(C(=O)NCC2C(C)CCN2C(=O)CCc2ccnc(Cl)c2)n1C 59516,c1(C(=O)NCC2CC(NC(Cn3c(CCC)ncc3)=O)C2)cc(C)nc(O)c1 59517,c1(CN(CCN(C(C(=O)OCC)=O)CCC(C)C)CC)c(F)ccc(OC)c1F 59518,Cc1ccc(O)cc1C(N1CC(C(O)C(=O)Nc2ccc(O)c(Cl)c2)C1)=O 59519,Cc1nc2ccccn2c1C(N1CCC1CNC(=O)CCC1CCCOC1)=O 59520,C1(NC(CC)=O)CC=CCC1C(N1CCC(C(N)=O)CC1)=O 59521,c1(CNC(COCC(=C)C)=O)occc1C(=O)NC1CC=CCC1 59522,C(=O)(C1OCCc2ccccc21)NC(C)CCNC(=O)Cn1cc(Br)cn1 59523,C1(CNC(c2c(NC)cccc2)=O)CN(C(c2ccc([N+](=O)[O-])o2)=O)CC1(C)C 59524,CCCC(C(=O)NCc1cccc(CNC(C2(C)C=CCC2)=O)c1)OCC 59525,c1(C(CC)C)ccc(C(=O)NC(C)(CNC(=O)C(O)C(C)C)C2CCC2)cc1 59526,Cc1cc(Cl)ccc1CC(=O)NC(C)C(C)NC(=O)C(C)(C)C 59527,C(C)(C(CC(=O)N(CCN(C)C)C(C)C)NC(C1CC2COCC2C1)=O)OC 59528,C1(C)(C(=O)NC(c2ccccc2)C2C(NC(C3CN(C)C3)=O)C2)CS(=O)(=O)C1 59529,N1(C(CN2CC(CC)C2)=O)CCCC2(CCN(C(c3cc(C(N)=O)cs3)=O)C2)C1 59530,c1(OC)ncc(NC(c2ccc(OC)c(C3CC3)c2)=O)c(C)n1 59531,c1(CNC2CC(CC(=O)NC3CCC(O)(C(=O)O)CC3)C2)cc2ccccc2o1 59532,C1(CNC(c2c(CC)con2)=O)(COC)CCN(C(C2CC(C)(C)O2)=O)CC1 59533,CCCC(F)(F)C(=O)NCC(CCOC)NC(=O)C(O)CN(C)C 59534,c1(CC)cnccc1C(=O)NC1CC(NC(=O)C(=O)Nc2ccc(C)cc2)C1 59535,C(CCCCCN=C(NCC(c1ccccc1Cl)OCC(C)C)NCCF)SC 59536,CC1CC(C(=O)NCC2(C)CCOCC2)CN(C(=O)COCCCN(C)C)C1 59537,C(=O)(C1=CC2C=CC(C1)C2)NC(CC(C)NC(c1c(OC)c(C)sc1)=O)C 59538,N1(C(Cc2n(C)c(S)nn2)=O)CCCC2(C1)CN(C(c1cnc(S)[nH]1)=O)C2 59539,CCCC(C)CC(=O)N(C(C)C(=O)NOCC1CCC1)C 59540,c1(N2CCCC(NC(C(C)CF)=O)C2)cc(C(F)(F)F)nc2ncnn12 59541,C=CC1CN(C(C2CN(C(c3cnncc3OC)=O)CC23CC3)=O)CCO1 59542,C(C)(C(C)COC)(c1nnnn1C)NCCCc1cc(CC)no1 59543,c1(C(N2CCOCC2CC2CCC2)C(=O)NC(C)C)ccc(C(F)(F)F)nc1 59544,c1(C(=O)Nc2c(C(N(C)Cc3ccc(Cl)s3)=O)n[nH]c2)ccc(Cl)c2[nH]ccc12 59545,C=CC(C)CC(=O)N1CC(CO)(NC(=O)CSCc2c(C)noc2C)C1 59546,N1(C(C(=O)NCC(CNC(c2ncn(C(C)C)c2)=O)(C)C)(C)C)CCN(C)CC1 59547,c1(OC(C)C)ccc(C(=O)NC2(C)CN(C(=O)CC3CC(C(F)F)C3)C2)cn1 59548,C=CCC(C(=O)OC)NC(C1C=CCN(C(c2ccc(OCC)o2)=O)C1)=O 59549,c1(C(=O)NC(CNC(C(C)(C)OCC)=O)CCOC)cc(C)c(CC)o1 59550,c1(C(N(C(CNC(c2cc(OC(CC)C)ncc2)=O)C)C)=O)nc(C)ccc1O 59551,c1(C(=O)NC2CC3CN(C(C4CCC(C)(CC)O4)=O)CC32)cccc2c1COC2 59552,Nc1ccc(C(=O)NC2CCCC2NC(c2ncoc2C(F)(F)F)=O)cc1Cl 59553,N1(C(c2cccc(C(C)C)c2)=O)CC2(CC(NC(C3(C)CCC(=O)N3)=O)CO2)C1 59554,c1(C(=O)NC2CC(CC)(CC)N(C(=O)C3=NOC(C)C3)C2)c(C)ccc(C)c1O 59555,N12CCOC(C1)CNC2=O.C1(N(C)C)CCC(N2CCOCC2)C1 59556,c1(NC(c2cccc(C)c2)CN(C)C)ncnc2cc(F)c(Br)cc12 59557,Cc1cnc(CC(=O)NCC(C)CN(C(=O)CCNC(=O)NC2CCCO2)C)o1 59558,C1(C(=O)NCCC(C)N(C(=O)CC2CC3(CCC3)C2)C)CCCCC12CCC2 59559,N1(C(C(CCC)N(C)C)=O)CCC2(C1)CN(C(C1CC1(C)C)=O)C2 59560,N1(C(C2(C)CN(C(C3(COC)COC3)=O)C2)=O)CC2CC(O)CC1C2 59561,C1(C(N2CC(O)CC(OC)C2)=O)CN(C(c2cc(C)cc(F)c2)=O)CCC1(C)C 59562,O=C1NCc2c1ccnc2C(N1CC(NC(c2cccc(F)c2)=O)CC1CO)=O 59563,C1(C(N2C(C)(C(=O)NCCC3CCN(C)C3)C=CC2)=O)CCCC(C#N)C1 59564,C(C(C)(C)CC(C)O)NC(CN(C(c1c(C)ccnc1)=O)CC1CC1)=O 59565,c1(CC(=O)N(C2CCC2)C(C2CCCC2C)C)cccc(Br)c1.C(=O)N 59566,Cc1cccc(NC(C2CCN(C(=O)Cc3cc(F)ccc3Br)C2)=O)c1[N+](=O)[O-] 59567,N1(C(c2cncc(C#C)c2)=O)CCC(NC(=O)C#CC2CC2)C12CCC2 59568,N1(C(c2cccc(O)c2)=O)CC2CCN(CC)CC2C1.c12cccc(n1)C(=O)N2 59569,c1(CC(N2CC(CCCCNC(CCCCC=C)=O)C2)=O)nc2ncccn2n1 59570,C1(C(=O)NCC2CCCS2)(COC)C=CCN1C(=O)CC1CC2CCC1O2 59571,c1(C(=O)NC)cccc(C(N2CCC(C)(NC(=O)C(C)CO)C2)=O)n1 59572,Cc1sc2ncc(C(N3C4CCC3(CNC(=O)C(C)O)CC4)=O)c(=O)n2c1C 59573,Cc1cc(C(=O)NC2CC(NC(=O)CC3CCC4(CCC4)O3)C2)cc2c[nH]nc12 59574,c1(COCC(=O)NCC(CNC(CCNS(CC)(=O)=O)=O)O)ncc(C)o1 59575,n1(C(C)C)cc(C(=O)NCC(CO)NC(C2(F)CC2)=O)c(Br)n1 59576,C=CCC(C)(C)CC(=O)NCc1cncc(C(=O)NC2CN(C(N)=O)C2)c1 59577,C1(CC(=O)NC(CC(=O)NCCC(C)(C)O)C2CC2)CC2(CC2)CO1 59578,Cc1ccc(F)c(O)c1C(=O)NCCN(C(C1OCCC1C(F)(F)F)=O)C(C)C 59579,C1(C(N2CCOC(CC)C2)=O)(CNC(C(COCC)C)=O)CC12CCC2 59580,c1(C(N2CCN(CC(=O)NCC3N(CC)CCC3)CC2)=O)cc(F)cnc1O 59581,c1(C(=O)OC(CSCCN(CC(C)C#N)CC)=O)cn(C)nc1SC 59582,CCCCC(=O)N(C1CC(NC(=O)CN(C(=O)C(C)C)C)C1)C 59583,c1(C(=O)NCC2(NC(C3CCC(CC)CC3)=O)CC2)ccc(N)cc1[N+](=O)[O-] 59584,c1(C(N2CCN(C(C(C(CC)O)C)=O)C(C(C)C)C2)=O)cccc2sncc12 59585,c1(C(=O)NC2C(NC(CCC3C(C)C3)=O)COC2)cnn(C)c1Cl 59586,C1(C(N(CCNC(CC(=C)I)=O)C)=O)CCC(C(F)(F)F)CC1 59587,C(=O)(N=c1nc2ccccn2[nH]1)c1n[nH]c2c1CN(C(CCN=[N+]=[N-])=O)CC2 59588,C1(COC)C=CCCN1C(=O)CC(O)CNC(c1ccncc1N)=O 59589,c1(NC(C2(OC)CCOCC2)C)cc([N+](=O)[O-])c(C#N)cc1F 59590,C1(NC(COC(C)C)=O)(CF)CCN(C(=O)CCC2CCCCN2C)C1 59591,c1(C(=O)NC(CC=C)CNC(=O)CC2(C)CCCO2)cc(C)nc2[nH]nc(C)c12 59592,CC1CC(CNC(C2CC3CC3C2)=O)CCN1C(=O)COC1(C)CCC1 59593,C1(C)(C(=O)NCC(CC(C)C)NC(CCC(=C)Cl)=O)CCCC1(F)F 59594,c1(C(=O)NC2CCCC2NC(C2CC2F)=O)cnc2scc(Br)n12 59595,c1(OC)cc(C(=O)Nc2cc(C)cc(C)c2Br)c(N)cc1Cl 59596,c1(C(=O)NCC(C)CNC(=O)C(N2CCCCC2=O)C)cccc(F)c1N 59597,C(CC(=O)N1CC(C)(C)C1C(=O)OC)(CC(C)C)NC(C1N(CC)CCC1)=O 59598,C1(C(=O)NCCCN(C)C(c2ccc(Cl)c(O)c2)=O)COc2ccccc2C1 59599,N1(C(C2CC(=O)CN2C(c2cnn[nH]2)=O)=O)CC2(CCNC2=O)C1 59600,c1(C(N(C2CCC(NC(C3C=CC=CC=C3)=O)C2)C)=O)cnn(CCO)c1O 59601,C=CC(C)CC(=O)NC(C1CN(C(=O)CCc2cncnc2)C1)C 59602,C1(NC(=O)NCC2(CCO)CN(C(=O)OC(C)(C)C)C2)CCc2ccnn2C1 59603,c1(C2(C)CCO2)ccccc1CNC(C1CCC1)C1CC1 59604,N1(C(c2cc(SC)nn2C)=O)CCC(N)c2ccc(F)cc2C1 59605,c1(C(N2CCC(C)(NC(c3ccc(O)cn3)=O)CC2)=O)cncc(P(C)(C)=O)c1 59606,c1(C(CC)C)ccc(NC(C2CCN(CC3(SC)CC3)CC2)=O)cc1 59607,Cc1ccc(C(=O)NC2CC2C(=O)N(CCO)C2CC2)cc1[N+](=O)[O-] 59608,c1(C(C(=O)NCCCCCC)N(CCC(=O)OC)C2CC2)ccc(CC)cc1Cl 59609,C(CC(=O)NCc1cc(C(N)=O)no1)(C(F)F)NC(CNC(C1C(C)C1)=O)=O 59610,N1(C(CCC2(C)CCCN2C(=O)C(O)C2CC2)=O)CCCCCCCC1 59611,Cc1nc2ccc(NC(=O)C(N3CCCC3C(c3cccc(Cl)c3)O)=O)cc2o1 59612,Cc1n[nH]c(C)c1CC(C)C(=O)NC(C)CC(C)NC(=O)C(C1CCCCC1)O 59613,C(=O)(C(CNC(=O)CC(C)(F)F)CC1CC1)NCc1ccc(CC)o1 59614,C1(C(C)NC(C23CC2C3)=O)CCCCN1C(c1ccc(C2CC2)s1)=O 59615,c1(C(N(CCNC(c2cc(C)oc2)=O)CCOCC2CC2)=O)c[nH]ccc1=O 59616,CCCC(F)C(=O)NC1(CCCNC(=O)CCCNC(=O)OC)CC1 59617,CC(C)(C)C(=O)C(=O)N1CCN(C(c2sccc2F)=O)CC1CC1CC1 59618,CON1CCC(CC(=O)NC2CC(F)(CNC(C3CCN3S(C)(=O)=O)=O)C2)CC1 59619,C1(NC(c2nccc(OC)c2O)=O)CCCC12CN(c1nccc(CC#N)n1)C2 59620,C1(CC=C)(NC(C2CC2c2ccccc2Cl)=O)CCN(C(=O)C(F)(F)COC)C1 59621,C1(C(N2CCN(C(=O)C3CC3)CC2)=O)CCCCCN1C(C12CCC(CC1)CC2)=O 59622,C1(C(N2C(CN(C(=O)CCS(N)(=O)=O)C)CCCC2)=O)CCC(N=[N+]=[N-])C1 59623,CC(C)(C)C#CC(=O)N1CCN(C(=O)CC2CCCCC2)C(CS(C)(=O)=O)C1 59624,C1(OC)CN(C(c2ccccc2CSC2CC2)=O)CC1OC.c12nc(no1)CS2 59625,C(CCC(=O)NC(CSC1CCN(C(C)=O)C1)C(=O)NC)OCC 59626,Nc1ccc(C=CC(=O)NCC2CCCN(C(C3CCCOCC3)=O)C2)cc1N 59627,CCC(C)C(O)C(=O)N(C)CC1(NC(c2cc(-n3ccnc3C)ccn2)=O)CC1 59628,C(CC(C(C)(C)C)NC(=O)Cn1cnnc1)N(C(c1c(C)nccc1)=O)C 59629,CCC(CC)(CCNC(=O)C(C)Cn1ccnc1)NC(c1cc(F)n(C)n1)=O 59630,Cc1c(Cl)c(C(N2CCC(C)(NC(C3CC34CCCC4)=O)C2)=O)nn1C 59631,N1(C(C(=O)NC(C(=O)N(C(=O)C2CC2)CC)C)=O)CCCC2(C=CCO2)C1 59632,C12(NC(C(C)NC(C)=O)=O)CC1CN(C(c1ccc(N(C)C)nn1)=O)C2 59633,C1(C(N2CC(O)(C(C)NC(=O)Cc3csc(C(C)C)n3)C2)=O)(COC)CC1(F)F 59634,CC(C)(C)CC(O)CC(=O)NCCCC1(NC(=O)Cc2nn(C)cc2Cl)CC1 59635,N1(C(CCN(CCCCC)C(C)C)=O)CCCC1CNC(=O)C=C(C)C(F)F 59636,c1(C(N2CC(CN=c3c(C(=O)OC)cc(Cl)n[nH]3)C2)=O)nc2nccc(C)n2n1 59637,c1(C(N(C2CCCOC2)CCC)=O)cnc(CNC(=O)NC)s1 59638,c1(OC)nccc(C(N2CC=CCC2C(=O)NCC2C(C)C2(F)F)=O)n1 59639,C(=O)(C(F)(F)CCCn1cc(C(c2ccccc2)=O)nn1)NCC1(C)CCCN1 59640,CC(C)CC(C(=O)N1CC2CC(CNC(C3CCCS3)=O)CC1C2)C(N)=O 59641,c1(CCC(N2CCC(c3c(OC)cccn3)CC2)=O)c(OC)cccc1Br 59642,N1(C(C(CC(C)C)O)=O)CCC2(CC(NC(c3cc(C4CC4)ccc3F)=O)C2)C1 59643,C1(C(=O)NCCCN(C(C(C(=O)OCC)OC)=O)C2CC2)CN2CCCN1CC2 59644,c1(C(N2C(C(=O)Nc3onc(C)c3C)CCC2)=O)ccc2c(Br)nn(C)c2c1 59645,C1(NC)CCCN(C(=O)CC(c2ccccc2)NC(=O)OC(C)(C)C)CC1(F)F 59646,C1(C)(CNC(c2ccc(CCC)s2)=O)CCC(NC(C2(CF)CC2)=O)CC1 59647,C(=O)(C(F)C(F)(F)C(F)(F)F)N1CCC(NC(C2CC(C)(C)C(=O)NC2)=O)CC1 59648,C(C(N=c1[nH]c(Cl)ncc1[N+](=O)[O-])C1CCCCC1)NC(C(CCC)OC)=O 59649,n1(CCN2CCC(CNC(=O)Cc3cn[nH]c3)CC2)cnc2ccc(F)cc2c1=O 59650,C(C)(C)(C(=O)NC1CCC1CNC(C1(F)CCOC1)=O)NC(=O)NCCC 59651,C1(Cl)(C(=O)NCC2(NC(c3nc(CC(C)C)sc3)=O)CCOC2)CC12CCC2 59652,c1(C(=O)NCC(CC)N(C(=O)COCC2CCCC2)C)cc(C(F)(F)F)n[nH]1 59653,c1(C(=O)NCCC2(CNC(C(C)=C3CC3)=O)CC2)ccc2nc(S)oc2c1 59654,C(CNC(=O)CC1(N(C)C)CC1)(C(C)(C)C)NC(C(C=C)C)=O 59655,c1(C(C(=O)NC)N(CC(C)OC(C)(C)C)CCOC)cc(C)c(C)c([N+](=O)[O-])c1C 59656,[N-]=[N+]=Nc1ccc(C(=O)NC2CCC3CN(C(=O)Cc4cccnc4)CC23)cc1 59657,C1(C(N(C2CC=CC2)C)=O)CC1C1CN(C(c2cc(Cl)cs2)=O)C1 59658,C1(CNC(c2n(C)ncc2)=O)CN(C(c2cc(F)n(C)n2)=O)CCN1C 59659,C1(CC(=O)NCC=C=C)CN(C(C2(O)CC(CF)C2)=O)CCO1 59660,c1(COCC)cn(CC2CCN2Cc2ccc(-c3cccs3)[nH]2)nn1 59661,N1(CC=C)CCCN(C(=O)C(C)SC)CC1.C12CC(OC)(C1)OC2=O 59662,C12(C(=O)NC(CNC(CCC=C(C)C)=O)CO)CCC(C)(C1)OC2 59663,n12nc(c3c1CCOC3)NCC2.c1(C(C(=O)OC)=O)cnn(C)c1 59664,N1(C(c2c(CCCC)occ2)C(=O)Nc2ccccc2C)CCC(O)CC1(C)C 59665,O=C(CC(F)(F)F)NC(CCC1CC1)C(=O)NCC(c1ccccc1)O 59666,C1(C(=O)N(CCNC(C)=O)Cc2ccncc2)(OC)CCOC1 59667,c1(CC(=O)NC)ccc(C(=O)NCC2C=CCN2C(C2CC2(C)C)=O)cc1 59668,N1(C(c2c(CC)cns2)=O)CCN(C(=O)CCc2cncc(F)c2)CC1CCO 59669,C1(C)(CC)CC(NC(=O)CN(C(=O)C=Cc2cscn2)CC2CC2)CCO1 59670,C1(NC(C2(C)C=CCN2)=O)CCCC12CCCC2 59671,N1(C(C(CSCC)NC(c2ccsc2)=O)=O)CCC2(CCC(OC)C2)C1 59672,C1(c2c(OC)nccn2)NC(=S)N(CC(C)C)C2=C1C(=O)NC(c1nccn1C)C2 59673,C1(C)(C(=O)NCC(C)N(C(=O)COCC2CCCOC2)CC)CCC(C)=C(C)C1 59674,C1(N(C)CC)CC(C(=O)N(C(C)C)Cc2cn(-c3sc(C)nc3C)nn2)C1(C)C 59675,c1(C(=O)NC2C(C(=O)NCC3OC4CCC3C4)CC=CC2)ccnc(CO)c1 59676,CCC(CC(=O)NC(c1cccnc1)C(N1CC(C)(C#N)C1)=O)C(F)F 59677,N1(C(CCN(CCC)C)=O)C2CCC(C2)C1CC(=O)NC(c1cc[nH]n1)CC 59678,C#CCC(C)(C)C(=O)N1CC2(NC(=O)C(O)Cc3ccccc3)CC1C2 59679,N1(C(Cc2c(OC)ccc(C)c2)=O)CC(C2CN(C(C3CC(C)CCO3)=O)C2)C1 59680,CC1CCN(C(c2cnn(C)n2)=O)C1CNC(=O)CCCN1CCCCC1 59681,C1(C(=O)NCC(CNC(C(C)O)=O)C)CC(S(C)(=O)=O)C1 59682,Cc1ccc(OCC(=O)NC2CC3CCC2(NC(c2cncnc2)=O)C3)cc1C 59683,C=CC1CN(C(c2cccc(COC)n2)=O)CC1NC(C12CC(F)(C1)C2)=O 59684,N1(C(C(CCC)CNC(C2C3CCC(F)C23)=O)=O)CCC(O)C12CCC2 59685,C1(C(=O)NC2C3CN(C(c4nn(CC)c(O)c4)=O)C2C3)CCc2c[nH]nc2C1 59686,C(=O)(CCS(C)(=O)=O)NC(C)C(CO)NC(C1COC(=O)C1)=O 59687,c1(CC)nccnc1C(=O)NC1CCCC(NC(C2(SCC)CC2)=O)C1 59688,c1(-c2cc(C)ncc2)cccc2c1CCN(C(=O)C(C)C)C2 59689,C(=O)(CS(C)(=O)=O)NCCC(CNC(C)=O)O 59690,c1(C(N(C2CCN(C(CC(c3c(C)noc3C)C)=O)C2)C)=O)cn2c(n1)CCC2 59691,N1(C(C2(NC(C)=O)CCCCC2)=O)CCC(C)N(C(=O)C(C)OCCC(C)C)CC1 59692,CC(C)(CC(=O)N1CCN(C(c2ccc(N)c(F)n2)=O)CC1)C(F)F 59693,C1(CCNC(c2c(C)cnn2C)=O)CCCN(C(=O)C(F)(F)C(F)F)CC1 59694,c1(C(=O)NC2CN(C(c3c(C)n(C)cc3)=O)C(C)C2)c(F)cccc1Br 59695,C#CCCN=C(NCC1(C)CCS(=O)(=O)N1C)NC(CF)CF 59696,c1(C(=O)NCCC2CCN(C(c3c(CC)csc3)=O)C2)ncc(N(C)C)cn1 59697,c1(C(=O)NC2C(CNC(C(C)(C)N3CCCC3)=O)CCC2)cnc2n1CCCC2 59698,CC(C)C(O)C(=O)NC1CCC(NC(C2(Cc3ccccc3)CCC2)=O)C1 59699,c1(C(C)C(=O)OCCC(C)O)ccc(Cl)cc1Cl.n12cc(nn1)CC1CN(C1)C2=O 59700,C(CC(F)F)(C(=O)NCC1(C)CC(C)(C)C1)NC(c1cn(C)nn1)=O 59701,C12CC1C2(F)F.C1(CNC(C2(C(=O)OCC)CC2)=O)(CNC(=O)CC)CCC1 59702,c1(C(=O)Nc2cccc(C3(C(=O)OC)CC3)c2)cc2cccc(Cl)c2nn1 59703,c1(C(N2CC(NC(C(C)(C)OC(C)C)=O)C(C)C2)=O)cnc(OC(F)F)c(F)c1 59704,N1(C(C(COC)C)=O)CC2(C)CN(C(c3ccn(CC4CC4)c3C)=O)CC2(C)C1 59705,CCCCCC(O)C(=O)N1CCC(C(C)(C)NC(c2ccc(CC)c(C)c2)=O)C1 59706,c1(C(=O)NCCCCc2cn(-c3ccc(Br)cc3Cl)nn2)ccc2ncsc2c1 59707,C12(C(=O)NCC3(NC(CCC=C=C)=O)CCCC3)CCCCC1C2(F)F 59708,Cn1cc2cccc(C(=O)N(C)C)c2n1.C12(C)CN(C1)C(=O)C1(CC1)NC(=O)CC2 59709,N1(C(c2cc(N)cc(F)c2)=O)CCCC2CN(Cc3ccc(F)cn3)CCC12 59710,n1(CCS(=O)(=O)N(C(CCC)C(=O)O)C)nc2ccccn2c1=O 59711,C=CCC(C)(C)CC(c1nnnn1C1(C)CC1)NCc1cccc2c1OCC2 59712,Cn1ncc2nc(O)c(C(N3CC(CNC(=O)Cc4cccs4)C3)=O)cc12 59713,C1(CC)CN(C(C2CC(C#N)(OC)C2)=O)CCN1C(=O)CCc1cccc(C)n1 59714,Cc1nc2nccc(C(=O)NCC3CC(O)(CNC(=O)C(O)C(C)(C)C)C3)n2n1 59715,C(CNC(c1nn(C)cc1Cl)=O)(C(C)C(C)C)NC(C1CCC(CC)CC1)=O 59716,c1(CC(=O)NC2CCN(C(c3cc[nH]c3)=O)CC2F)cccc2sccc12 59717,N1(C(C(C)=C2CC2)=O)CCC(NC(=O)COC2CCOCC2)C2(CCC2)C1 59718,C(=O)(C(C)C(CC)CC)NCC(CC)NC(=O)CCCC1CCOCC1 59719,c1(CC)cc(C(=O)NC(C)(CSC)C(=O)NCC2CC2Cl)n(C)n1 59720,CC(O)C(C)C(=O)NCc1ncc(C(=O)NCCC2CCSC2)cn1 59721,CCC(C)C(C(=O)NC1(CO)CC2CCCC12)NC(=O)C=CC(F)(F)F 59722,c1(C(C)=O)ccc(=NCCNC(c2ccc(-c3cccs3)cc2)=O)[nH]c1 59723,Cc1cnc2c(cnn2CC(=O)N(CC(C)NC(=O)CC2CCOC2)C)c1 59724,C12(NC(CCCN(C)C)=O)CCC1CN(C(=O)CCN1CCCS1(=O)=O)C2 59725,N#CC1CN(Cc2ccc(Br)cc2F)CC1NC(=O)COc1cccc(Cl)c1 59726,C(=O)(C1=Cc2cc(Cl)ccc2OC1)NC1(CO)CN(C(C(CC(=C)C)C)=O)C1 59727,C1(C(=O)NCC(C)NC(c2ccc(N(CC)CC)cc2)=O)CN2CCCN1CC2 59728,C1(CC(=O)NC2CN(C(C(C=CC)O)=O)CC(F)C2)C2CC3CC(C2)CC1C3 59729,CN1CCC(O)C(NC(N2CCN(CC3CCCCC3)CC2)=O)C1 59730,N1(C(c2c(C)nc(COC)s2)=O)CC2CCN(C(=O)CCC3CC3(Cl)Cl)C2C1 59731,CC1(C)CC(C)(C(=O)NN(C2CC(CO)C2)C)CN1C(c1ncoc1C1CC1)=O 59732,CC1(CC(N2CC(N=[N+]=[N-])C2)=O)CCN(C(C2(C#N)CCCO2)=O)CC1 59733,c1(C(N2C(CNC(Cc3cc(C)on3)=O)CC2)=O)ccc(C(F)(F)F)c(F)c1 59734,C(=O)(C1=NNC(=O)C1)NC1CCCC(NC(C(N2CCCC(C)C2)=O)=O)C1 59735,c1(C(N2CCCC(N(C(C(C)CO)=O)C)CC2)=O)cc([N+](=O)[O-])cn1C 59736,c1(CCC(=O)NC(C)CNC(=O)C2CC2)ccc(Br)cc1 59737,C(=O)(C(C)(C)C1CCOC1)NCCC(C)N(C(C=C(COC)C)=O)C 59738,CCCCCCCC(F)C(=O)N1CC(C)(C)CC1CNC(=O)C=C(C)CCC 59739,N1(C(CNC(CCC2C(C)(C)C2)=O)=O)CCN(C(=O)CC2CCCC23CC3)CC1 59740,N1(C(C23CC(C)C2C3)=O)CCN(C(=O)C=C(Cl)Cl)C2COCC12 59741,C1(CCn2cc(-c3c(C)cn(C)n3)nn2)CCN(CCn2c([N+](=O)[O-])cnc2C)CC1(F)F 59742,N1(CCCC(CC)=O)CCN(Cc2ccncc2)C2CC12 59743,N1(C(C2N(C)CCC2)=O)CC2CC1C2NC(=O)CC1CCN(CC(F)(F)F)C1 59744,c1(C(=O)NCC2C(NC(CCC(=O)NC)=O)CCC2)ccnc(F)c1OC 59745,C1(NC(C2(C)CCN2C(C2(F)CC2)=O)=O)CCCC(O)C1 59746,C1(CN(C)C(C2CC2F)=O)CN(C(=O)CCOC2CC2)CC12CC2 59747,c1(C(N(C(CNC(C2CC(C(F)F)C2)=O)C2CC2)C)=O)cccc2nccn12 59748,C1(NC(c2c(NCC)scn2)=O)CCCC12CN(C(c1cc(C#N)[nH]c1C)=O)C2 59749,C1(CC(=O)O)CC2(CCN(C(C3CC3c3ccc(-c4cccs4)cc3F)=O)C2)C1 59750,C1(CC(=O)NCCN(CCCN(C)C)C(=O)C=C(C2CC2)C2CC2)NC(=O)NC1=O 59751,N1(C(CCC#C)=O)CC(CNC(C2CCCC23CC3)=O)C2CCCCC12 59752,c1(C(C(=O)NCC(C)(C)NC(c2c(N(C)C)nccc2)=O)=O)ccc(Cl)cc1O 59753,C(=O)(C#CC(C)(C)C)NCCN(C(c1snnc1C(C)C)=O)CC 59754,Cc1ccc(Cl)cc1C(=O)NCCC1(O)CN(C(C2COCC(C)O2)=O)C1 59755,N1(C(CCOCCN(C)C)=O)CCCCCC(NC(c2cncc(OC)n2)=O)C1 59756,S(=O)(=O)(c1cnc(NCCc2cc(Br)no2)c(Cl)c1)N1CCn2c(C)ncc2C1 59757,CCC(C)C(O)C(=O)N1C2CCC1(CNC(C1(C)CCC1)=O)CC2 59758,c1(C(=O)NC2C3CC2CN(C(C2CC=CC2)=O)C3)cc2scc(Br)c2[nH]1 59759,C1(C(=O)NCC(COC)(C)C)(C(=O)O)CCN(C(=O)OC(C)(C)C)CC1O 59760,C(CNC(c1cnnn1C)=O)(CC(F)(F)F)NC(C(C)SC)=O 59761,C1(CNC(CCc2cn(C)nc2)=O)CCCCN(C(C2CCCC23CCC3)=O)C1 59762,c1(OCC(=O)NC(CN(C(C(C=C=C)C)=O)C)C)ccc(F)cc1O 59763,Cc1nc2cc(C(=O)NCC3CC(O)(NC(c4cnc(C5CC5)[nH]4)=O)C3)[nH]c2s1 59764,c1(NCC23C(CN(c4nccc(CC(=O)OC)n4)C2)C3)nc(OC)ncc1F 59765,N1(C(C(C)OCC#C)=O)CCN(C(c2c(C)csc2Cl)=O)CC1c1ccccc1 59766,N1(CC)CC(NC(=O)C(CC2CCCC2)NC(=O)C(C2CCOCC2)=O)C(C)C1 59767,N1(C(C2(C(=O)NC)CCCC2)=O)CCCC(C)(NC(C2CC(OC)C2)=O)C1 59768,CCC(C)C(O)CC(=O)NC1(C)CC(NC(c2n[nH]c3c2CCSC3)=O)C1 59769,N1(C(COCC(=O)NC)=O)CC2C(NC(C3CN(C(C)C)CCO3)=O)C2C1 59770,N1(C(C2(C#C)CC(NCN3C(=O)CCCC3=O)C2)=O)CC2(CC2)CC1CO 59771,C(=O)(CS(=O)(=O)C1CC1)NCC(C(C)C)NC(C1(CC(=O)OC)CCCC1)=O 59772,C1(=O)C(CCC(C)(C)C)N2CC(C(C(C)C)C2)C(=O)N1.c1(OC)ccccc1SC 59773,C(c1ccccc1Cl)=CC(=O)NC1CCCN(C(=O)CC2COCCO2)CC1 59774,C(c1ccncn1)=CC(=O)NC(C(C)NC(c1cscc1F)=O)C 59775,C1(C(N2CC(C)N(C(=O)CCc3cccs3)CC2)=O)COC2COCC2O1 59776,C1(CC)CC1N=c1[nH]c(N(C)Cc2nn(C)c3ccccc23)nc2ccsc12 59777,c1(C2(C(=O)NC(CC)C(C)(C)O)CC2)ccc(C)c(Cl)c1 59778,c1(N2CCC(C)SCC2)ccncc1S(=O)(=O)N1CC(C)(C)OCC1CO 59779,c1(C(=O)NC2CC(C)(NC(C(C=C=C)C)=O)C2)cc(O)nc(C)n1 59780,c1(C(=O)NCC2C(NC(C3(COC)C=CCC3)=O)COC2)[nH]c(O)nc1C 59781,CCCC(C(=O)NC(C)CNC(=O)CCc1cc(C)on1)C(C)C 59782,N1(C(c2noc(C)n2)=O)CCC(NC(C(C2CN(C(CC)=O)C2)OC)=O)C1 59783,C1(C(=O)NCCC(C)CCO)(OC)CCN(C(=O)OC(C)(C)C)C1 59784,c1(-n2cc(C3CN(CC(c4cccnc4)OC)C3)nn2)ccc(Cl)cn1 59785,N#Cc1cc(C(N2CCC(CC(=O)Nc3ccc(F)c(F)c3Cl)C2)=O)ccc1F 59786,C1(C(=O)NCCCNC(CC=C=C)=O)CCOC1C=C 59787,N1(C(=O)Nc2c(C(C)(C)C)nccn2)CCC2CCC12c1cccs1 59788,N1(C(Cc2c(C)cco2)=O)CCCC(CCNC(c2ccc(F)cc2)=O)CC1 59789,C1(C)(C(=O)NCC(C(=O)OC)(C)C)CCCN(Cc2cccc(O)n2)C1 59790,CC(C)CC(C)ONC(ONC(c1coc(C2CCCC2)c1)=O)=O 59791,C(=O)(C(F)C(C)CNC(c1cc(C)c(N)cn1)=O)N1CCC(C(=O)OCC)C1 59792,C(=O)(CC1C(=O)Nc2ccc(C)cc21)NC(CC)CNC(=O)C(OC)OC 59793,C(CCN=c1cc(C)[nH]c(=NCC2CCN(C)C2C)[nH]1)S(CC)(=O)=O 59794,C(=O)(C1CNc2ccccc21)NCC1C(C)(C)CCN(C(C23CC(CO2)C3)=O)C1 59795,C12(NC(C3CCCCN3C(C3CCC3)=O)=O)CC(C1)N(C(=O)CCCCO)C2 59796,c1(C(=O)NC(C2CC(NC(C3(Cl)CC3(C)C)=O)C2)C)cc(-c2cnn(C)c2)[nH]n1 59797,CC1CN(C(=O)C(=O)C2CCCC2)CC(C)CN1C(c1cc(C(N)=O)co1)=O 59798,c1(C(c2ncc(-c3cn[nH]c3)cc2O)=O)cc(Cl)cc(Cl)c1F 59799,Cn1cc(C(=O)NCC2CCCC2NC(c2ccccc2Cl)=O)nc1O 59800,c1(CC(=O)NC(CN(C(=O)C(CC)OC)CC)C)ccnn1C(C)CC 59801,C1(C(N2CCCCC2C2CC2)=O)C2CC(O)C(C2)N1C(=O)C(O)CC(F)(F)F 59802,CC1=NN(C)C(=O)C1CC(N1CCC(NC(c2ccnn2C(C)C)=O)C1)=O 59803,C1(O)(C(=O)NCC(N(C(c2ncn(CC)n2)=O)C)C2CC2)CCC(C)CC1 59804,c1(CC(=O)Nc2ccc(O)c(F)c2)ccc(F)cc1Cl 59805,c1(C(=O)NC(C(C)NC(=O)CCN2CCCC2)C)coc(C(N)=O)c1 59806,N1(CC(=O)N(C(C)CNC(=O)CNS(=O)(=O)N(C)C)CC)CCCCCCC1=O 59807,C(=O)(CC(C(F)(F)F)NC(=O)COCCF)NC1(CC#C)CC1 59808,N1(C(C2CCC(CC)O2)=O)CC=CC(NC(c2csc(CO)n2)=O)C1 59809,c1(C(=O)NC2C(CNC(c3ccnnc3O)=O)CCC2)cccc2[nH]nc(O)c12 59810,C#Cc1cncc(C(N2CCCC2C2CCN(CCN3CCNC3=O)CC2)=O)c1 59811,C1(C(N(C2C3CN(C(c4cncc(O)c4)=O)CC23)C)=O)CC2CCC1O2 59812,c1(OCC(N2CCC(C(=O)OC)(CN)CC2)=O)ccccc1[N+](=O)[O-] 59813,C(=O)(CC(C(N)=O)NC(C)=O)NCC(CNC(CCNS(CC)(=O)=O)=O)O 59814,c1(N(C)C)ccccc1C(N1CC(C)(NC(C2C3CC4C(C3)C24)=O)C1)=O 59815,c1(CC(C(=O)OCC)OCc2cn(CCOCCO)nn2)ccc(I)cc1 59816,C1(C(=O)NCCOCCCN(C(C2(OCC)CCC2)=O)C)CC12CCOC2 59817,c1(CCN2CCC(C(C)NCCO)CC2)ccccc1F.c1(OC(=O)C)ncccn1 59818,C12(CN(CC(c3nn[nH]n3)C)Cc3ccc(C)cc3)CC=CCN1CCC2 59819,c1(NCCCOCC)ncc(S(=O)(=O)N2CCS(=O)(=O)CC2C)cc1Cl 59820,Cc1cccc(Cl)c1C(N1CCC(OCCNC(=O)Cc2ccsc2)CC1)=O 59821,C(CC(=O)NCc1cnns1)(C(F)(F)F)NC(CC(C=C)(C)O)=O 59822,c1(CNC(Cc2c(C)nn(C)c2C)C)ccc2c(c1)sc(=O)n2C 59823,CC(C)CC(C)(CN=c1[nH]c(Cl)ncc1Br)NC(=O)Cc1cn2c(n1)CCCC2 59824,C1(CS(=O)(=O)NC2(CC3CCC3)CC2)CCC2(CCOCC2)CO1 59825,c1(C(=O)NC2CN(C(CCN3CCC(C)CC3)=O)CC2O)cc(F)c(Cl)cc1O 59826,Cn1cnc2c(NC3CCN(Cc4ccc(Br)c(Cl)c4Cl)C3)ncnc12 59827,C1(NC(C)=O)CCC(C(=O)NCCC2CCCN(C(=O)CC3CCCO3)C2)CC1 59828,C1(N(C(=O)CC2(NC(c3cc(F)n[nH]3)=O)CCCC2)CC)CCCN(C(C)=O)C1 59829,C1(CN(C(=O)C=Cc2ccoc2)C)CCCN(C(C2CCC(=O)N2C2CC2)=O)C1 59830,c1(C(=O)OCC2(N(CC(C)C)C(c3ccco3)=O)CC2)ccn(CC(C)C)n1 59831,S(=O)(=O)(CC(=O)NCC1CN(C(c2cnc(Cl)n2C)=O)CC1O)NC(C)(C)C 59832,C1(C)(CNC(C=C(C)C(F)F)=O)CN(C(=O)CN(C)CCO)CCO1 59833,C1(COC)(CNC(=O)CC(C)F)CCCN1C(c1cccc[n+]1[O-])=O 59834,CCCC(CCC)C(=O)N1CCCN(C(=O)Cn2cccc(N)c2=O)C(C)C1 59835,C1(c2onc(C)n2)C(C)OCCN1C(=O)Nc1cc(O)cc(Br)c1 59836,S(=O)(=O)(C1CCCN(OC2CC(=O)NC2)C1)Nc1c(SC)cccc1 59837,N1(C(c2cn(CCNC(c3c(COC)noc3)=O)nc2)=O)CCC(CO)C(O)C1 59838,N1(C(CC2CCC(C)C2)=O)CC2(C1)CN(C(c1cn(C)cc1C(=O)C)=O)C2.C(N)=O 59839,C1(C(=O)NCCOC)CC12CCN(C(c1ccsn1)=O)C2 59840,C1(c2n(C(C)C)nnn2)(NCc2ccncn2)CC2CC1CC2(F)F 59841,c1(CC(=O)NCC2(C)N(C(Cc3c(C)n(C)nc3)=O)CCC2)cc(F)ccc1Cl 59842,C(CNC(C1CC=CC1)=O)(C(C)C(C)C)NC(c1c(NCC)cccn1)=O 59843,N1(C(C(N2CCNC2=O)C)=O)CCCC(N2C(=O)C2)C1.c1(CC2CC2)n[nH]c(=N)s1 59844,c1(-c2c(C)ncs2)nnc(N2CCOC(Cn3cccn3)C2)n1CC1CCOC1 59845,c1(C(=O)NC2CCCC2C(N2CCC(O)CC2)=O)ccc2occc2c1 59846,C12(CCCN(C3CN(C(C4CCOC4)=O)C3)C)CCC(CC1)C2 59847,c1(NC(C2CCN2C2CCC(=O)N2)=O)nc(Cl)cc(Cl)n1 59848,CCC1=C(C(=O)N2CCCCC2CCNC(=O)CC(O)CN(C)C)CCCO1 59849,N1(C(C(c2ccn(C)c2)C)=O)CCCC1CC(N1CC(F)C1)=O 59850,C(=O)(C(C(C)(C)C)NC(c1ccccn1)=O)N1CCN(C(CC)=O)CC1 59851,C1(C(=O)NC(CNC(c2c(C)ocn2)=O)(C)C2CC2)CCn2ccnc2C1 59852,c1(OC)ccc(N=c2ncnc(N3CCC3)[nH]2)cn1.C12CCC(CC1)NC2=O 59853,C1(CNC(CC=C)=O)CC2(CC2)CN1C(=O)Cc1cn(C(C)C)nn1 59854,C1(C(=O)NC2C3CN(C(c4cscc4Br)=O)C2C3)CC2C=CC1CCC2 59855,C(=O)(C(F)(F)c1cncs1)NCC(C)NC(=O)C(c1ccc(Cl)s1)C 59856,N1(CC(N2C(c3ccc(C)cc3)CCC2)=O)C(=O)CN(C)C1=O 59857,Cc1nc(N2CCC(c3cccc([N+](=O)[O-])c3)C2)nc2ccccc12 59858,C1(O)(C(=O)NC(C(C)NC(C(C)(C)NC(=O)OC)=O)CO)CN2CCC1CC2 59859,C#CCCN=C(NCCc1ccccc1C#N)NCCc1ccn(C)c1 59860,CC1C(C)N(C(c2ccc(CO)o2)=O)CCN1C(c1ccc(C#N)cc1O)=O 59861,N1(C(COC(C)=O)=O)CC(NC(C2(C)CC=CC2)=O)CC12CCC2 59862,C(CC(C(=O)N1CCCCC1CNC(=O)CCCc1ccsc1)OC)OC 59863,c1(C(N2CC3CN(Cc4ccc(Br)nc4Br)C3C2)=O)nc2ccccn2n1 59864,c1(CNC(C2CCCN(C(c3ccc(Br)cn3)=O)C2)=O)ccc(F)c(F)c1 59865,N1(C(c2ccc(OC)o2)=O)CC(C(=O)Nc2cc(C)sc2C)CC(C)C1 59866,C(=O)(C1=CCCCO1)NCCCCCCNC(CCC1CCCN(C)C1)=O 59867,c1(C(=O)NCC(C)(C)CNC(C23CC4CC2C3C4O)=O)ccc2c(n1)CCCN2 59868,C(C1C(C(=O)NCC(C2CCCC2)NC(=O)CC(C)O)C1(C)C)=C(C)C 59869,CC1(C)CNC(=O)C1NC(=O)CN(C(c1ccc(F)cn1)=O)C1CC1 59870,c1(C2(C(=O)NCC=CCNC(CCC(C)OC)=O)CC2)ccccc1C#N 59871,C1(C(=O)NC(CNC(C(C)=C(C)C)=O)(C)CO)C2COC(C)(C)OCC12 59872,c1(C(N2CC(CNC(C(c3ccccc3)NC(N)=O)=O)C2)=O)cc[n+]([O-])cc1 59873,C1(O)(CNC(C2CC(SC)C2)=O)CCCN(C(=O)C(N2CCCCC2)C)CC1 59874,C1(NC(C(CNC(c2c(NC)scn2)=O)(C)C)=O)CN(C)C(C)(C)C1 59875,Cc1ccc(C)c(CCCC(=O)NCC#CCNC(=O)CNC(C2CC2C)=O)c1 59876,C#CC1(C(N2CCC(OC)C2C)=O)CCN(C(C2C(C)(C)C2(F)F)=O)CC1 59877,c1(COCC(=O)NC2CCC(CNC(C3(N(C)C)CC3)=O)C2)ccc(Cl)cc1 59878,C(C(=O)NC(CCC1CCC1)C(=O)Nc1cnc(F)nc1)(C(C)C)SC 59879,C(=O)(C(C)(C)C)NCC(C)(C)O.C(C(=O)NCCN(C)C1CC1)N 59880,c1(C(N(CC2(O)CCN(C(CCC)=O)C2)CC)=O)coc2ccc(OC)cc12 59881,C(=O)(C1=C(Cl)CCOC1)N1CCC(CC)CC1C(N1CCC1(C)C)=O 59882,C12(C(=O)NC3(CCCC)CC3)CCCC1CCN2Cc1cncc(C)c1 59883,CC1(C)CCCN(C(c2cscn2)=O)C1CNC(=O)CSCc1ccccc1 59884,C1(C(=O)NCCCOC2CC(NC(C3(Cl)CC3)=O)C2)CCCC(F)C1 59885,C=C=CC(C)C(=O)NCC12COC(CNC(C3CCC(CCC)CC3)=O)(C1)C2 59886,CC1(C)Cc2cc(Br)ccc2C1NC(=O)C(N1CCC(SC(F)(F)F)CC1)=O 59887,N1(C(CCNC(C)C)=O)CCCN(C(=O)CC2COC(=O)C2)CC1 59888,C1(F)(C(=O)NC(C)CCCNC(=O)Cn2cc(C3CC3)cn2)CCCN(C)C1 59889,C(C(O)CC(=O)NC(C)Cc1ccnn1C)NC(CC1CC(=C)C1)=O 59890,c1(CCN(CCc2ccc(C=C)cc2)C2CC2)ccc2c(c1)CCO2 59891,C1(OC)(CNC(=O)Cc2cnc(C)[nH]2)CCN(C(C2(OC)CCSC2)=O)C1 59892,c1(C(=O)NC(CCc2ccc(C)o2)C)cc(Br)c(=O)n(C)c1 59893,c1(C(=O)NCCC(=C)CNC(=O)CCN(C)CC)ccc(O)c(N)n1 59894,c1(OC)ccc(CN2CC3CC3(C(=O)Nc3cc(Cl)ncc3Cl)C2)cc1Br 59895,C1(CC(=O)NC2(C(N(C(C)C(N)=O)C)=O)CC2(C)C)C(C)(C)C1(C)C 59896,Cc1nc(C)c(CC(=O)N(CC(C)(C)CNC(C2(CCN(C)C)CC2)=O)C)s1 59897,C1(NC(CC=C)=O)CCN(C(c2ccnc(OCC)c2)=O)C(C)C1 59898,N1(C(CC=C(C)C)=O)CC2CC(NC(=O)C(C(C)C)n3ccnc3)C1C2 59899,N1(C(c2scc(OC)c2)=O)CCCC(F)(C(N2CCC(C#N)C2)=O)C1 59900,Cc1c(F)ccc(N)c1C(=O)NCC1CCN1C(c1ccn(C2CC2(F)F)n1)=O 59901,c1(C(N(CCNC(=O)C(C)(O)COC)CC)=O)cc(F)c(F)c(Cl)c1F 59902,c1(C(N2CC(C(=O)Nc3nnc(C)o3)C(O)CC2)=O)cc2cccc(O)c2[nH]1 59903,Cc1cc(F)ccc1Cn1nnnc1N(C1(CC(F)(F)F)CCCOC1)C 59904,CC1=C(C(=O)NCCCN2CCC(NC(C3CC3(F)F)=O)C2)COCC1 59905,c1(CC(=O)NC2CCN(C(CCCOC)=O)C2)c[nH]c2cc(OC)ccc12 59906,CC1(C(=O)NCCC(N)=O)CCN(Cc2ccncc2Cl)C1 59907,C1(CN(C)C(C2CCN(C(c3cc(C(C)=O)oc3)=O)C2)=O)COCCOC1 59908,N1(C(CC)=O)CC2=C(C1)CN(C(=O)Cc1cnc(C3CC3)[nH]1)C2 59909,C(=O)(C(F)(F)C(F)F)N(CC(C)(C)CNC(C1CCCC1)=O)CC 59910,C(C(CNC(C1(Cc2cnn[nH]2)CCCC1)=O)CO)NC(c1cscn1)=O 59911,N1(C(C2C(COC)C2)=O)CCC(CCNC(c2cnn(C)n2)=O)C(F)(F)CC1 59912,c1(N2CCC(C3N(C(CCCC(C)=O)=O)CCC3)C2)nc2cccnc2s1 59913,Cc1sc(Br)c(C(=O)NC2CC(F)CN(C(=O)Cc3cn[nH]c3)C2)c1C 59914,CC1CN(C(C2(C#N)CC2)=O)CCN1C(=O)C(C)C(F)(F)F 59915,Cc1cccc2cc(C(=O)NCCNC(=O)C(C)Cc3ccc(C#N)cc3)nn12 59916,C1(C)(C(=O)NC(CNC(c2nn(CC)c(O)c2)=O)CO)CC(C(F)(F)F)=NO1 59917,N1(C(Cc2ncc(CC)[nH]2)=O)CCCC(NC(c2c(C)nc(C)n2O)=O)CC1 59918,Cc1ccc(C=CCC(=O)NC2(CCNC(C3CC3F)=O)CC2)cc1 59919,Cc1c(C(N2CC(NC(=O)C3=CCCCO3)C(C)C2)=O)sc2cncn12 59920,N1(C(c2c(C)coc2C)=O)CCC(NC(c2cnn(C)c2C(F)(F)F)=O)C(F)C1 59921,c1(C(=O)NC(C2CCCN(C(c3cc(C(C)=O)on3)=O)C2)C)cccc(Cl)c1F 59922,c1(CC(=O)N(CC(CC)NC(C2CC2(C)C)=O)CC)cc(=O)n(-c2ccccn2)[nH]1 59923,C1(NC(C2CC(C)(O)C2)=O)CN(C(=O)C=CC(=O)N(C)C)CC1C(F)(F)F 59924,N1(C(C2C(C=C)C2)=O)C(CNC(c2c[nH]nc2C(F)F)=O)CC2CCCC12 59925,CCC(C(=O)NC1(C2CCN(C(c3cccc(COC)n3)=O)C2)CC1)C(C)(F)F 59926,n1(CC(N2C(CN(C(c3n(C(CC)C)ncc3)=O)C)CCC2)=O)cccnc1=O 59927,c1(-c2c(C(=O)Nc3ccc(C(CC)C)cc3)n[nH]c2)ccc(O)c(C)c1 59928,O=C1CC(C2(C(N3CCCC(N4CCOCC4)C3)=O)CC2)C(=O)N1 59929,C=C1CCCN(C(=O)CCNC(=O)CCC(N)C(C)C)C1 59930,N1(C(=O)NCC2CCCS2)CC2(CC(N)C(O)C2)C1 59931,CCC(C)(COC)C(=O)N(CCCN(C(=O)C(C)c1ccon1)C)C 59932,C1(F)(CNC(CCCOC)=O)CCCN(C(=O)COc2ccccc2Br)C1 59933,N1(C(C=CC(C)NC(C(C)OCCOCC)=O)=O)CC(F)(C(N)=O)C1 59934,Cc1cc(NC(=O)C(N2CCCC2CC(c2ccccc2)O)=O)c(C)s1 59935,N(C(=NCCc1ccc(F)cc1C)NN1CC2C(CO)C3CCC2C13)CCOC 59936,C(CCC(CO)NC(=O)CC(C)(C)C)NC(C1CCN(C)C1)=O 59937,N1(C(c2cccc(OC)n2)=O)C2CCC1C(CNC(c1cc(C)cc(Cl)n1)=O)C2 59938,c1(CCCC(=O)NCCC2CN(C(C3C(=C)C3)=O)C2)cc(F)ccc1F 59939,O=C(CCN=c1[nH]ccs1)NC1CC(NC(c2ccn(C3CCCCC3)n2)=O)C1 59940,N1(C(C23CCC(N=[N+]=[N-])C2C3)=O)C2CCCC1CN(C(=O)C=C1CCC1)C2 59941,C1(CNC(c2csc3nnsc23)=O)CC2CCC(C1)N2C(c1cscn1)=O 59942,c1(NCC(F)=C(C)C)cc(Br)ccc1S(=O)(=O)N1CCCC1C 59943,c1(C(N2CCC3C(C2)CN3C(c2n[nH]c(C3CC3)n2)=O)=O)ncc2[nH]ncc2n1 59944,O=CN1CCCC1C(N1CCC(CNC(=O)Cc2cnco2)C1)=O 59945,c1(NC(c2ccc(-n3cncn3)cc2)C)nc2c(F)cccc2n1C 59946,Cc1ccc2ncnc(N(Cc3ncccn3)CC3CNCCOC3)c2c1 59947,c1(C(N2CC(CC)(NC(=O)Cn3ccnc3C)C2)=O)cnc2[nH]cncc1-2 59948,C1(NC(C2(F)C(C)C2)=O)(CNC(=O)CCCOC(C)=O)CCCC1 59949,N1(C(C2C(C3(C)COC3)C2)=O)C2CCC(C(N3CCCC(F)(CO)C3)=O)C1CC2 59950,C(=O)(C(O)CC(F)(F)F)N1C(CC)C(C(=O)NCC(C)Cc2cn[nH]c2)CC1 59951,c1(CNC(CC2=CCN(C)CC2)=O)cccc2c1CCN(C(c1cnns1)=O)C2 59952,Cc1nc(-c2ccccn2)sc1C(=O)NCC1C=CCN1C(C1(O)CCCC1)=O 59953,c1(C(N2CCC(Cn3cc(C(C)(C)C)nn3)C2)=O)ccc2c(c1)C(=O)C(=O)N2 59954,CC12CCCC1N(C(C1CN(C(=O)CN3CC=CC3)CCO1)=O)CCC2 59955,c1(CC)ccccc1C(C(=O)NC1CCCC1)N(n1ccnc1C)CCOC 59956,c1(OCC)cc(C(=O)NCC(CNC(C2(CC)CC2(F)F)=O)CO)ccn1 59957,c1(C(N2CCC(N(C(=O)C(C)NS(C)(=O)=O)CCC)C2)=O)c(C)ccc(C)c1O 59958,C(CNC(C1CC1c1ccn(C)n1)=O)(CC(C)C)NC(c1nc(OCC)sn1)=O 59959,CC(C(=O)NCCC1(NC(c2ccc(C(C)(C)C)cn2)=O)CCC1)S(N)(=O)=O 59960,c1(C(=O)NC2CC(CNC(C3(COC)COC3)=O)C2)sc(C)c(C)c1C 59961,C(=O)(CCC(C)(C)NC(C12CC1CNC2=O)=O)N(C)CC1CCOC1 59962,C1(CC(N2CC3C(N(C(Cc4cc(C)on4)=O)C)C3C2)=O)COC2(CCC2)CO1 59963,C1(NC(=O)CCC2CCCO2)CC2CCC(C1)N2C(C1CCC2C(C1)C2(F)F)=O 59964,CC1CN(C(c2ncc(F)cc2F)=O)CC(C)C1NC(c1cnc(Cl)s1)=O 59965,N1(C(=O)COCC2CC2)CC2CCC1(CO)C2 59966,N1(C(CN(C)CC)=O)CCC2CC1CN(C(=O)CCc1cnc3n1CCOC3)C2 59967,CC1(C)OCCN(CC(O)Cc2ccn(C(F)F)n2)C1CO 59968,Cc1cc(=NCC2C(C)CCCN2C(c2cccc(O)n2)=O)[nH]c(CO)n1 59969,Cc1nc(C(=O)NCC(CNC(=O)C(C)C(F)(F)F)CO)ccc1[N+](=O)[O-] 59970,N1(C(c2ccc(CC)[nH]2)=O)CCOCCC1C(=O)NC(c1cc(C)on1)C 59971,c1(-c2nc(C)c(NC(=O)NCc3ccccc3I)s2)cc(F)cc(F)c1 59972,c1(CC)ccccc1CC(=O)NCC12CC1CN(C(C1CC(SC)C1)=O)C2 59973,C12(CNC(=O)C3=CCCCCC3)CCCC1N(C(c1cccc(O)n1)=O)CCC2 59974,c1(C(N2CCC(C(C)NC(C(C(CC)C)O)=O)C2)=O)cnc2c(c1)c(C)nn2C 59975,c1(OC)cncc(C(=O)NC(CNC(c2ccc(O)cn2)=O)CC(C)C)c1 59976,C1(CNC(=O)CC2CC2CNC(c2sccc2CO)=O)C(C)(C)C1(F)F 59977,CN1CC2CC1CN2C(C1C=CCN1C(C1CNC(=O)O1)=O)=O 59978,C1(CC(=O)N(CC(C)C#N)CCOC)CC2(CCC2)CO1 59979,C1(C(=O)NCC2C(CO)C2(C)C)(CC)CN(C(=O)C=CCN2CCC2)C1 59980,C12(NC(c3nc(CC)sc3N)=O)CCC(CNC(=O)C(O)C(C)OC)(CC1)OC2 59981,C(=O)(C1(C)CCn2ccnc21)NCCN(C(CCCCC=C)=O)CCC 59982,C(=O)(CC(C)C(F)(F)F)NC1(CNC(C2(CCOC)CCC2)=O)CCOC1 59983,C(CC)(CC(=O)C(C(C)NC(CC)(C)C)=O)N.C(C(C)(C)C)NC 59984,C1(F)(CNC(c2ccon2)=O)COCCN(C(c2ccc(Cl)s2)=O)C1 59985,N1(C(C(C)CC(F)F)=O)CC2(CCCC2NC(c2cc3c[nH]nc3s2)=O)C1 59986,c1(C(C)C)scnc1C(=O)NCC(O)CNC(c1ncc(C(F)F)s1)=O 59987,C=C(C)CC(C(=O)NC1C2CCC1CC2)NC(C1CCN1CC)=O 59988,c1(C(=O)NCC(CO)NC(C(C)OC(CC)=O)=O)ccc(OC)cc1F 59989,n1(CC(C)C(N2CC3C(CNC(=O)C(F)(F)CO)C3C2)=O)cc(P(C)(C)=O)cn1 59990,Cc1ccc(C(N2CC(F)CC2C(N2CC3C(CN(C)C)C3C2)=O)=O)nc1C 59991,c1(CC(=O)NCCC2(CNC(C(C)S(N)(=O)=O)=O)CC2)cccc2c1OCC2 59992,CC1CCCCC1(CNC(C1CC2CCC1O2)=O)NC(C1CCCC2(CC2)C1)=O 59993,c1(C(=O)NCCC(=C)CNC(=O)C(O)C2CCC2)cc(OC)c(OC)cc1N 59994,S(=O)(=O)(c1cnn(C2CCCC2)c1)N(CC=C)CCN(C)C 59995,N1(S(Cc2cccc(C)c2)(=O)=O)Cc2ccc(C(=O)Nc3cncc(Cl)n3)cc2C1 59996,C1(C(=O)NC2(CC=C)CN(C(C3CC4CCC3CC4)=O)C2)CC2CCC1CC2 59997,c1(C(=O)NCC2CC(C)N(C(=O)C3CC3)C2)nc(O)nc(O)c1F 59998,C12=NC=CC(=NC(=O)Cc3csc(n3)C(=O)NC1)N2.c1ccccc1.CC(C)C 59999,N1(C(C2CCN(Cc3cncc(N(C)C)c3)CC2)=O)CCc2ccc(O)cc2C1 60000,C(=O)(C(CCF)NC(C1CC(C)CCO1)=O)NCCCNC(C)=O 60001,N1(C(C2C=CC(=O)N=N2)=O)CC(NC(c2cc(Br)ncc2F)=O)C(F)(F)C1 60002,CC1(C)CCCC1(C)NC(=O)Nc1cnc(SCC2COC3CC2C3)nc1 60003,c1(C(C)(C)C)nc[nH]c1S(=O)(=O)NC1CNCC12CCC2 60004,c1(OCC(=O)NC2CCCC(C)C2)cc(Cl)c(Br)cc1F 60005,c1(CCSC)nc(CCn2ccnn2)n(-c2cccnc2)n1 60006,C1(C(=O)NCC(CNC(=O)OC(C)(C)C)(C)F)(C2CC2)CCCS1(=O)=O 60007,c1(N2CC(CCC)OCC2)nc(=NC(C)C(F)F)[nH]c2c1cnn2C 60008,N1(C(C2(C(N(C)C)=O)CC2)=O)CCC2C(C1)CN2C(=O)C(O)C(F)F 60009,C(=O)(C(F)C(F)(F)C(F)(F)F)N1CCCC(NC(c2ccc(COC)o2)=O)CC1 60010,C(=O)(C(CCC(C)C)N=C1NS(=O)(=O)c2ccccc21)NCCNC(=O)NC 60011,c1(OC)cc(C(=O)NC2CCC(NC(c3ccn(C)c3)=O)CC2)c2c(c1)CCO2 60012,c1(C(N(CC(CC)NC(C2(C)CCC(=O)NC2)=O)C)=O)cn2c(C)cccc2n1 60013,N1(C(CC(C)N(C)C)=O)CC2(C1)OC1(C)CC2(NC(=O)COc2ccccn2)C1 60014,C1(NC(C2(OC(C)C)CCC2)=O)CCC(C)N(c2nccc(CO)n2)C1 60015,N1(C(CC(COC)C)=O)CCC(C)(C)CC1C(N1CCC12CC(C)(OC)C2)=O 60016,CC1(C)CCN(C(c2ncncc2Cl)=O)C1C(=O)NCCC1(O)CCCCC1 60017,C(=O)(C(CC)CCCCC)N1CCCC(O)(CNC(CCC#CC)=O)C1 60018,C1(C(=O)NC(C2CCN(C(c3conc3C(C)(C)C)=O)C2)C)CCS(=O)(=O)C1 60019,c1(OC)ccc2c(=NC(C)CCF)[nH]c(=NCc3ncn(C)n3)[nH]c2c1 60020,Cc1cc(OCCC(=O)NCC2(F)CCCN(C(=O)CCC(F)F)C2)cc(C)c1 60021,C#CCC(C)(CNC(=O)CCCN(C)C(C1CC2CC2C1)=O)CO 60022,N1(C(CC(CC(=O)OC)C)=O)CCCCC2(C1)CN(C(c1cscn1)=O)C2 60023,C=CC(CCC)CC(=O)NCC(C)=CC(=O)NC(C)C(N1CCOCC1)=O 60024,c1(OC)c(C)ccnc1NC(N1CCC(N2CCC(F)CC2)C1)=O 60025,C(=O)(CC(=O)NC1C=CC(CNC(=O)C(F)CC2CCC2)C1)OC 60026,N1(C(C2(CC=C)CCOCC2)=O)CCCN(C(=O)Cn2cnnc2O)CCC1 60027,c1(C(=O)NCc2ccns2)cc(O)nc2c1CN(C(C1CC1C1CC1)=O)CC2 60028,C1(N(C)C(=O)OCCCC)CCCN(N2CCC(OC)C2)C1 60029,C1(C(=O)NC(C(=O)N(CCOCC)C)c2ccoc2)CCS(=O)CC1 60030,C=C1CC2CCCC(C1)N2C(=O)C(CC)NC(C1CCC2(CC2)C1)=O 60031,C=CC1(O)CN(C(C2CCN(C(=O)C(C)(COC(C)=O)OC)CC2)=O)C1 60032,Cc1nc2ccc(C(=O)NC(C)CNC(c3cc4ncc(C)cn4n3)=O)cn2n1 60033,C1(CNC(c2c(OC)nc(C)s2)=O)CCN(C(=O)Cc2cnsc2)C1(C)C 60034,C(CCC(N)=O)(C(=O)NCCn1ccnn1)n1cc(CC(C(=O)OC)(C)C)nn1 60035,C1(F)(CNC(C=CCCC)=O)CCCN(C(=O)CCn2c(C)c(C)sc2=O)C1 60036,Cc1cncc(F)c1C(=O)NCC(=O)NC1CCC(C(N)=O)C1 60037,C1(CC#C)(C(=O)NC(C2CCCC2)CNC(=O)CCn2ccnc2C)CCCO1 60038,C(=O)(CC(C)(C)C(F)(F)F)NCC1N(C(CCOC)=O)CCC1C1CC1 60039,c1(CC(=O)NC)ccc(C(=O)NCC2CCN2C(=O)CC2COC(=O)N2)cc1 60040,CC(C)(C)CC(C)(C)C(=O)N1CCC(O)(CNC(C2(N(C)C)CCCC2)=O)C1 60041,Cc1cc(C(=O)NCCNC(=O)C2=NOCC2)c2[nH]cnc2c1 60042,N1(C(C2=CC(C)(CC)C2)=O)CC2CCC(C1)N2C(C1CC2(C1)CC(C)(C)C2)=O 60043,CCC(CC)C(F)C(=O)NCC1(C)CN(C(C2CCCN2CC(C)C)=O)CCO1 60044,Cc1cc(C)c(C)c(C(N2CC(F)(CNC(=O)Cn3nccn3)C2)=O)c1C 60045,C1(c2onc(C(C)OCC3CCC3)n2)CC2CC1(c1ccc(F)cc1)C2 60046,C1(CC(N2CCC(C(C)OC)CC2)=O)CC(C)(C)CN1C(=O)CC1COC(=O)C1 60047,c1(C(C(=O)NCCC2CC2)C2CCCC2)cccc(OC2CC2)c1 60048,C1(C)(C(N(C(c2ccco2)C)C)=O)CCCN(C(=O)CCc2cncn2C)C1 60049,c1(OC)nc(OC)nc(N2CC3CC3(C(N3CC4CCCC4C3)=O)C2)n1 60050,c1(C(N2CCC(NC(C(C)F)=O)C(F)C2)=O)ccc(Br)c2cccnc12 60051,C(CCC=O)(C(N)=O)NC(C(C)N(CCC)C(c1ccc(Cl)cc1)=O)=O.NC 60052,C1(C(=O)NC(CC=C)(C)C)CN(C)CCN1C(=O)C(=Cc1ccco1)C 60053,c1(C(=O)NCC2N(C(C(C)(C)C3CCC3)=O)CCOC2)cccc(C(N)=O)c1N 60054,C1(C(N(C)CCN2CCCC2=O)=O)CCCCC1NC(=O)CCC1(C)N=N1 60055,CCC(CC(=O)NCC1CCOC1C(=O)NCC(C)(C)N(C)C)SC 60056,c1(CN(S(=O)(=O)c2cn[nH]c2)C)cc2c(O)cccc2s1 60057,C(CC(C)CCO)NC(c1cncc(C(C)(C)C)c1)c1n(CC(=C)C)nnn1 60058,N1(C(c2c(SC)scc2)=O)CCN(C(=O)CS(N)(=O)=O)CC12CC2 60059,c1(COCC)nc(C)c(C(N2CC3CC3(NC(=O)CCCOCC)C2)=O)s1 60060,C=C(C)CCC(=O)NC(C1CCN(C(=O)C(C)N(CC(F)(F)F)C)CC1)C 60061,N1(C(C(C)OCOC)=O)CCC2CN(C(C3(C(N)=O)CC3)=O)CC2C1 60062,c1(C2(C(=O)NCC(C)(CO)NC(c3cnc(OC)s3)=O)CCC2)cccc(Cl)c1 60063,C1(C(N(C(CNC(c2n(CC)cnn2)=O)C2CC2)C)=O)CCC(F)CC1 60064,C1(N(C(c2n(CC)ncc2)=O)C)CN(C(c2cn(C)nc2COC)=O)CCC1O 60065,C12CCN(CC1C#N)CCO2.c1(OC)cc(C)ccc1C1CC1 60066,c1(CC)cc(C(=O)NCC2C=CC(NC(c3ccn(COC)n3)=O)C2)c(C)o1 60067,CC12CSCC1CN(c1ncncc1Br)C2 60068,c1(C(=O)NCC2CCCN(C(C=CC3(C)COC3)=O)C2)ccc2ccsc2c1 60069,c1(C(C(=O)OCC)(C)C)nnc2n1CCN(C(C(=O)NCCC#N)C(C)CC)C2 60070,C1(C)(C(c2n(CC=C)nnn2)NC(c2ccc(Cl)c(Cl)c2)C)CCS(=O)(=O)CC1 60071,c1(C(N(C(C2CCCC2)C)C)=O)ncccc1NC(=O)NC(c1ccco1)=O.C(C[SH](CC)C)NC 60072,c1(OC(C)C)cccc(C(=O)NC(C)C(C)NC(c2ccsc2Cl)=O)c1 60073,C1(C(=O)NC(C2CC(NC(C3N(CC)CCC3)=O)C2)C)CCCCCC1 60074,C(CN=c1[nH]c2c(Cl)c(Cl)ccc2s1)N1CCC(C(C)(C)C)CC1 60075,C1(CNC(CSC(=N)N)=O)C2CN(C(=O)CCc3ncc[nH]3)CC12 60076,C(C(C)(CO)Nc1csc(CCP(C)(C)=O)n1)NC(C=CC(=O)N(C)C)=O 60077,C(=O)(C(C)(C)CN1CCCC1)N(C)CC1CCN(C(C2C(C)C2C)=O)C1 60078,C12(NC(C3CC(N(C)C)C3)=O)CC1CN(C(=O)C(C)(C)c1ccccn1)C2 60079,N1(C(C(COC)C)=O)CCN(C(=O)Cc2ccc(Br)s2)C(CO)C1 60080,C(=O)(C(F)C(C)CNC(=O)CCC(C)(C)OC)N1CCC(OC)C1C(C)C 60081,C1(C)(C(=O)NC(C)CCNC(=O)Cc2cnoc2)CC1(F)Cl 60082,c1(C(N(C(C2CCNC2)C)CC2CC2(F)F)=O)ncnc(Cl)c1C#N 60083,c1(C(=O)NC(CC)CNC(c2cc(Cl)n(C)n2)=O)c(O)nnc2c1CCC2 60084,c1(C(=O)NC2C(NC(c3ccc(C(N)=O)cc3)=O)C2)cccn2ccnc12 60085,Cc1cc(O)ccc1C(N1CCC(NC(=O)C(c2ccccc2)C2CC2)CC1)=O 60086,C1(N(C)C)CN(C(=O)NCc2ccc(Br)s2)C(C)(C)CO1 60087,C(=O)(CCCn1cc(CCC(N)=O)nn1)NCC(=O)NC(C)(C)C 60088,C(CC(=O)N1CCOC(CCC)C1)(C(C)C)NC(CCC=C)=O 60089,C1(NC(C)=O)CCC2CN(c3ncc(C)c(Sc4ccncc4)n3)CC2C1 60090,C(C(CC(C)C)C(=O)NC1(CNC(C23CCC(CC2)C3(C)C)=O)CCC1)OC 60091,CC(CC(=O)NCC1C=CCN1C(=O)C=C1CCN(C)CC1)CC(C)(C)C 60092,N1(C(C2CC(C)C2)=O)CCC(N=c2cc(Cl)nc(-c3cccnc3)[nH]2)C1 60093,c1(C(=O)NC2(C)CN(C(Cc3cc(C)ns3)=O)C2)cc2n(n1)CCCC2O 60094,CCCCC(C(=O)NC(C)C(C)n1cccn1)NC(=O)Cc1cncnc1O 60095,CCC(C)(COC)C(=O)N1CCN(CC(C)(C)NC(=O)C=CS(C)=O)CC1 60096,N1(C(CCC#C)=O)CC=C(C(C)(C)C(=O)N(C(C)COC)C)C1 60097,C(CNC(=O)C(O)CC(C)(C)C)(CC(=O)N=c1ccn(CCO)[nH]1)OCC 60098,C1(CNC(c2c(CN(C)C)ccs2)=O)COCCN1C(=O)CC1CCC(C)(C)C1 60099,c1(C(N(CCCCNC(C2CCC(C)O2)=O)C)=O)cnc2c(Br)cccn12 60100,C(CN(C)C)(C(=O)N=c1cc2n([nH]1)CCCC2)NC(C(C1CC1)SC)=O 60101,C(C(=O)NCCN(C)C(C1(C(O)C(C)C)CC1)=O)(C1CCCC1)OCC 60102,CC(C)CC(CNC(C1CCCC(=O)N1)=O)NC(=O)C(c1ccccn1)O 60103,CC1(C)OC(=O)CC1C(N1CC(C(O)C(=O)NCCC2NC(=O)NC2=O)C1)=O 60104,C1(C(C)C)CN(C(c2cc(Cl)ns2)=O)CCN1C(c1c[nH]c(=S)cn1)=O 60105,N1(C(c2cnn(CC)n2)=O)CCC(C2CC2NC(=O)C(C(C)C)OC)CC1 60106,C(C(C)(C)C(=O)NC1CCC(CNC(=O)CC2CC2(C)C)C1)N(C)C 60107,C1(C2CC2)(C(=O)NC2C(NC(c3ccc(COC)o3)=O)CC2)CC=CC1 60108,c1(CC(N2CCC(NC(C(COC)C)=O)C23CC3)=O)cnc2n1CCOC2 60109,CC1C(C(=O)NC2CC23CCC3)CCN1C(N1CCC(O)CC1)=O 60110,C(=O)(CCCC(C)(C)C#N)N1C(C(=O)NCc2c(CC)onc2C)C(CC)CC1 60111,c1(C2C(C(=O)NCCC3(CNC(CSC(C)C)=O)CC3)C2)ccccc1Cl 60112,C1(CCC(=O)NCC(=C2CN(c3nc(C(F)(F)F)ns3)C2)F)CCCC(=O)N1 60113,c1(C(=O)NC2(CNC(c3cncc4nc[nH]c34)=O)CCC2)n[nH]c2c1NCCC2 60114,N1(C(CCC(C)C#N)=O)CC2(C1)OC1(C)CC2(NC(c2c(Cl)cnn2C)=O)C1 60115,CC1(C(=O)NCCCN(C(=O)Cn2ccnn2)CCO)CCCS1(=O)=O 60116,Cc1cnc2nc(C(=O)N(CC(C)(C)CNC(=O)C=CC3CCCO3)C)nn2c1 60117,N12CC3CC3(C1)C2=O.c1(C(=O)NCC=CCN(C)C)cn(CC(=O)N(C)C)cn1 60118,C1(C)(CC)C=C(C(=O)NCC(C)CC(=O)N2CC(N(C)C)C(C)C2)C1 60119,CC1NC(=O)OC12CN(C(=O)CCOCCCNC(=O)CCc1ccccn1)C2 60120,N1(C(C(CC#C)C)=O)CCC2(CCCCN(C(=O)C(C)(C)CS(C)(=O)=O)C2)C1 60121,c1(C(N(CC(=O)Nc2c(C)c(F)ccc2)C)=O)cc2cc(C3CC3)cnc2[nH]1 60122,c1(OC)cc(C(=O)NC(C)(C)CN(C(=O)Cn2cnc(Br)c2)C)ccn1 60123,C1(C(N2CC(CC)C(C(=O)Nc3cncc(F)c3)C2)=O)CC12CCOCC2 60124,c1(OC)ccnc(F)c1C(N1CCC(O)(C(=O)NCc2nccnc2Cl)C1)=O 60125,CCC(CC)(CO)C(=O)NCCC1CN(C(C2CCCCC2F)=O)C1 60126,CCCC(CC)C(=O)NC1CCCN(C(=O)CC2CCN(CCF)CC2)CC1 60127,N1(C(CCc2c[nH]c(=N)[nH]2)=O)CCCC(NC(C2CCNC2=O)=O)CCC1 60128,O=C1CCC2(CCCN(C(=O)Nc3cccc(CCO)c3)C2)CN1 60129,O=C(CCCCCCNC(C1CCCC1)=O)NCC1CCC2(CC2)CO1 60130,N1(C(C2(OC)CCC2)=O)CC(NC(=O)C=CC(C)C)C(O)C1 60131,CC1CN(C(c2c(CCC(N)=O)c[nH]c2C)=O)CCCN1C(C1CNC(=O)O1)=O 60132,C1(CC(=O)NC2CCCN(C(=O)C(c3ccc(Br)cc3)O)C2)CCC(O)CC1 60133,N1(C(c2c(O)nc(=N)[nH]c2)=O)CCCC(C2(NC(=O)COCCN(C)C)CC2)C1 60134,C(C(C)C(=O)N(C1CCC1)C1CC1)N(C(C(C)C)=O)C 60135,C1(C(=O)NCCCC(=O)NC(C)(C)C)CCN2CCCCC12 60136,c1(OCCO)nc2ccccc2cc1C=O.N1(CCC)CCC2(C1)CN(C)C(=O)N2 60137,c1(CC)cc(C(=O)N(C)CCN(C(C2CCOC(CC)C2)=O)C(C)C)ncn1 60138,CC1CN(C(c2cc(Cl)no2)=O)CCC1NC(C1(Nc2ncccn2)CC1)=O 60139,C1(C)(C(=O)NCCCC(C)NC(C2CCCCC2O)=O)CCC(=O)N1 60140,c1(C(=O)NC2CCC(NC(=O)CC3CCCCC3)C2)ccn2nccc2n1 60141,c1(CC)c(C(=O)NC(CNC(=O)C2CC2)(CC)CC)cnn1CC(C)C 60142,C1(F)(C(N(CCN(C(C(C)SCC)=O)C(C)C)C)=O)CCOC1 60143,N1(C(C(C2N(C(CC=CC)=O)CCC2)(C)C)=O)CC2(CCC(=O)N2)C1 60144,c1(CC(C)C(=O)NCCCCNC(C2CCOC2C(F)(F)F)=O)cccc(Cl)c1 60145,C1(NCc2cccnc2)OCCOC1(C)C.C12CCN(C1)C(=O)C=CCN(C)C2 60146,C1(CNC(C(c2n(C)ccc2)=O)=O)CC2(CC2)CN1C(c1cnccc1Br)=O 60147,c1(NS(CCC2C(C(N3CC(C)NC(=O)C3)=O)C2)(=O)=O)ccc(S(C)(=O)=O)cc1F 60148,C(=O)(C1=CS(=O)CCC1)NC1C(OC)CN(C(c2ccc3ccnn3c2)=O)C1 60149,C12CN(CC13CCC3)C2=O.C1(O)(C(=O)NCC2(C(C)(F)F)CC2)CC(CF)C1 60150,C1(CNC(=O)CCCF)CCCCN(C(c2cc(Cl)cc(C(F)(F)F)n2)=O)C1 60151,C1(CNC(CN(C2CC2)CC)=O)CN(C(=O)CCC#N)CC(C(F)(F)F)O1 60152,c1(C(=O)NC2CC(C(C(=O)NCCCCSC)F)C2)nocc1Cl 60153,c1(C(=O)NC(C)CN(C)C)n[nH]cc1-c1ccccc1 60154,c1(C(N2CCC2c2cn(CC(c3ccccc3)O)nn2)=O)csc(I)c1 60155,c1(C(=O)NCC2(F)CC(CNC(C(C)SC(F)(F)F)=O)C2)ccc(C2CC2)nc1 60156,C1(C(N(CC(C2CC2)OC)C)=O)CN(C(=O)CCCn2ccnc2)C2(CCC2)C1 60157,N1(C(c2ccc(C)s2)=O)CC=C(C(=O)NC2CN(C(N)=O)C2)CC1 60158,C(=O)(C(C)CCCCCC)NCc1occ(C(N2C(C)(CCC)CC2)=O)c1 60159,C1(CNC(c2c(C(C)O)cccc2)=O)CCCN(C(=O)Cn2nnc(=N)[nH]2)CC1 60160,c1(C(N(CC(C)O)CCNC(C2C(OC)CC2)=O)=O)cocc1C 60161,C1(N(CCCN(S(C)(=O)=O)C2CC2)C)CCc2ccccc2NC1=O 60162,N#Cc1c[nH]c(=NC(=O)C2C=CCN2Cc2ccc3c(c2)C(=O)NC3=O)cc1F 60163,N1(CC(N2CC(N(C(CC(C=C)C)=O)C)C2)=O)CCCCC(O)C1=O 60164,C(=O)(CC(C)(C)CC(F)(F)F)NC1(CO)CN(C(Cc2ccc(C)s2)=O)C1 60165,c1(OC)ccc(C(=O)NC2CC(NC(c3cnc(O)s3)=O)C(O)C2)c(N)c1 60166,C#CCC(C)(C(=O)NC(CO)CCC=C)NC(=O)C(C)C#N 60167,c1(C(N2CCC(NC(C3CCS3(=O)=O)=O)(CF)C2)=O)c[nH]c2cc(F)c(F)cc12 60168,c1(C(N2C(CNC(c3cc(CC)[nH]n3)=O)COCC2)=O)cnn2ccnc(N)c12 60169,S(=O)(=O)(c1ccccc1Cl)N1CC(NC(=O)CSCC(N2CCCCC2)=O)C1 60170,CC(C)C(C(=O)N1CCCC(CN(C)C(c2nnn(C(C)(C)C)n2)=O)C1)NC=O 60171,n1(CCOC)ncc2c1C(NCC1CC(F)CN1)CCC2 60172,c12ccc(c(I)c1)[nH]c2=O.C1(C)(C(=O)OC)C=CCN1C(C)=O 60173,C(=O)(CC1=CCOCC1)NC1C(CNC(CCOc2cc(C)cc(C)c2)=O)CC1 60174,c1(OC)ccc2c(=NC3CCCN(C)C3C)[nH]c(=NCCCCC(N)=O)[nH]c2c1 60175,C1(C(N2CCC(N(C(=O)CC3CC=CC3)C)C2)=O)CCC(=O)N(C2CC2)C1 60176,Cc1cccc(C(N2CC(CC(=O)NC3(CC4CCC4)CC3)CC2C)=O)c1 60177,CC(C)(CC#N)C(=O)NC1COCCN(C(c2c[nH]nc2Br)=O)C1 60178,c1(C(=O)NC2(CCO)CN(C(C(=O)NCC)=O)C2)ccc(C2CCC2)nc1 60179,C1(NC(C2(CCNC(C(C)Cn3ccnc3)=O)CC2)=O)CC2(C1)CC2(F)F 60180,CCCCCCC(F)C(=O)N(C)CC1CCCCN1C(=O)Cc1ccn(CC)n1 60181,CC(C(=O)NCC12CCC(CC1)N2C(=O)CN1CCCCC1)C(C)S(C)(=O)=O 60182,S(=O)(=O)(c1ccc(C(=O)O)cc1F)NC1(CC(N2CC(C)C(=O)C2)=O)CCC1 60183,C1(CC=C)(C(=O)NC2(CNC(=O)Cc3cncnc3)CCCCC2)CCCCC1 60184,C1(CNC(C(=O)NCCNS(C)(=O)=O)=O)CC2(CCNC2)CO1 60185,C1(F)(CNC(C2CC(N(C)C)C2)=O)CCCN(C(C2CC23CCC3)=O)C1 60186,Cc1cc(N2CC3CC2CN3C(=O)C(O)CC(F)(F)F)nc(C)c1C#N 60187,C12(NC(CN3CC(C)(C)C3)=O)CCC(CC1NC(=O)C=CSc1ccccc1)C2 60188,C1(C(=O)NCCC(CC)C)CCCN(C(C2(OC)CCC2)=O)C1 60189,c1(-c2cc(NC(=O)CCc3cc(Br)ccc3F)sc2)c(F)ccc([N+](=O)[O-])c1F 60190,C(CCCOC)(C(=O)NCC(C)(C)COC)NC(C(=O)OCC)=O 60191,CCCC(C)(C)CNC(=O)CC1CC1CNC(=O)CCc1ccc[nH]1 60192,C(CCCN(C(=O)C(C)c1ccon1)C)NC(C1(CC=C)CC1)=O 60193,c1(C(=O)NC2C(C)N(C(c3n[nH]c4c3CSCC4)=O)CC2)ccc(S(C)=O)cc1 60194,c1(CN2C(C)(C(N3CCOCC3)=O)CCC2)c(OCC2CC2)cc(Cl)cc1F 60195,c1(C(=O)NCC(N2C(C)C(C)(C)CC2)=O)n[nH]c2cc(Br)ccc12 60196,n1(-c2cn(CCOCC(CC(=O)O)C3CCCCC3)nc2)cc(CNC)ccc1=O 60197,CC1(C)CC(C(=O)NC(C)(CNC(C2CCS(=O)CC2)=O)CO)CNC1=O 60198,S(=O)(=O)(c1cn(C2CC2)nc1C)N(CC)CC.c12cccc(c1)C2 60199,N#Cc1ccc2c(c1)CC(NC(C1CNCC1CC(F)(F)F)=O)C2 60200,C#CCC(C)C(=O)N(C1CCN(C(c2n[nH]c(C)c2C(F)(F)F)=O)C1)C 60201,c1(C(N2CCC(N(C(=O)CS(=O)CC)CCC)CC2)=O)cnc2snc(C)c2c1 60202,N1(C(C2CCC(C(N)=O)O2)=O)CCCCC1CCNC(=O)CCOCC1(F)CC1 60203,N1(C(C2C(C(C)C)OCC2)=O)CCCC2(C1)CN(C(c1ccnc(Cl)c1N)=O)C2 60204,C(CCCCC(=O)N1CCCC1CNC(c1oc(C)nc1C)=O)(OC)OC 60205,c1(OCC)ccnc(O)c1C(=O)NC1(Cc2ccc(C3CC3)cc2)CC1 60206,CCCC(F)C(=O)NCC1CCCC1C(=O)NCCN(CC(F)F)C 60207,c1(CCC(=O)NCCN(C(C)C(=O)NC(C)CC)CCC)nccn1C 60208,O=C1CC2OCCC2(C(N2CCCN(C(C3(CO)CCCO3)=O)CC2)=O)CN1 60209,c1(C(C(=O)NC(C(CO)NC(CC(=C=C)C)=O)C)(C)C)ccc(Br)c(C)c1 60210,C1(CC(=O)NCCCSC)CCN(C(C23CSCC2C3)=O)C1(C)C 60211,c1(OC)noc(C)c1C(=O)NCC1CC(F)CN1C(=O)C(c1ccccc1)OC 60212,N1(C(CC(=O)NCC)=O)CCC2(CC1)CC2NC(C1C=CCS1)=O 60213,C(=O)(C1CCCn2cncc21)N(C)CC1(CNC(C(CCCC)O)=O)CC1 60214,C1(C)(C(=O)NCC2N(C(CC(C=C)(C)C)=O)CCC(C)C2)CC(C(C)C)=NO1 60215,C(C)(CCCCNC(C1CCOC1(C)C)=O)NC(C1CC(CCCCCC)C1)=O 60216,N1(C(C)C(=O)OCCOc2ccc(Cl)cc2)Cc2ccccc2C1=O 60217,CN1CCC(O)(CC(N2CC3CC2CC3CNC(=O)Cc2cnsc2)=O)CC1 60218,CC1(C)COC(CC(N2CCCCC2C2(NC(=O)CNC(N)=O)CC2)=O)C1 60219,N1(C(C2OCCN(C(C(CC=C)C(C)C)=O)CC2)=O)CCC2(CNC(=O)C2)C1 60220,C1(C(=O)NCC2C3N(C(c4c(C)nsc4C)=O)C(CC3)C2)CCc2ccnn2C1 60221,C1(NC(c2cc(OC)n[nH]2)=O)C2CC1CN(C(=O)C=CI)C2 60222,C12(CNC(C=CCCC)=O)CC(NC(=O)C(C)C(F)(F)F)(C1)C1(CCOCC1)O2 60223,c1(CC)cc(C(=O)NCC2(NC(=O)COc3cc(C)on3)CC2)cs1 60224,C(=O)(C(CNC(c1ccc2ccoc2c1)=O)CC(C)C)NC(CCCC)C 60225,CCC(CNC(=O)CCP(C)(C)=O)(CC)C(=O)NC1CCOC1(C)C 60226,C1(N(C)C(c2ccc(C(F)(F)F)o2)=O)CN(C(=O)Cc2ccsc2)CC12CC2 60227,N1(C(CNC(C(C)(C)C)=O)=O)CCC(C2CN(C(=O)CCCS(C)(=O)=O)C2)CC1 60228,N1(CCCNC(C(CC)O)=O)CCN(C(C2CCSCC2)=O)CC1=O 60229,N1(C(CC2OCCN(C(C3CCN(CC)C3)=O)C2)=O)CCOC(C2CC2)(CC)C1 60230,C(=O)(C(CC)CCCCCC)N1CCC(CNC(CCCCC)=O)(OC)CC1 60231,c1(C(=O)NCCC2C(C)CN(C(C3CCCC3)=O)C2)c(F)ccc2cnn(C)c12 60232,N1(C(c2cc(C(=O)OCC)c(C)cc2)=O)CC2CC(C)N(C(=O)C3CC3)C2C1 60233,C(C(CNC(=O)COCC(F)F)C(F)(F)F)NC(C=CC1C(C)C1(Cl)Cl)=O 60234,C1(NC(CC(CNC(c2c(C)nsc2)=O)O)=O)CC2(C1)CC(C#N)C2 60235,c1(NC(C(CN(C)CC)NC(C2CCC(=O)NC2)=O)=O)cc(C)cc(C)c1C 60236,N1(C(C2CC(NC(C(CCC)CCC)=O)C2)=O)CCc2nnnn2CC1 60237,C1(C(N2C(CNC(C(CC(C)C)(C)C)=O)C=CC2)=O)CCc2ccccc2CC1 60238,c1(OC)cc(Cl)c(CN2CCN(c3ncccn3)C3CC23)cc1OC 60239,N1(C(C(CC)(C)C)=O)CCC2(CC1)CC(NC(c1cc(SC(F)(F)F)c[nH]1)=O)C2 60240,C(C(O)C(=O)NC1CC(F)(CNC(=O)CCC#N)C1)N(C)C 60241,c1(C(=O)NC(C(C)(C)NC(C(C)OCCOCC)=O)C)cc(C#N)ccc1O 60242,c1(NC(C2CC(F)CN(Cc3cc(Br)ccc3I)C2)=O)cnc2ccc(F)cn12 60243,CCC(C(=O)N1CCC(CNC(c2csc(CC(F)F)n2)=O)C12CC2)C(F)(F)F 60244,c1(CC)ccc(C(=O)NCC(c2ccccc2)NC(=O)CCCNC(N)=O)[nH]1 60245,c1(C(=O)Nc2ccc(C)c(C(F)F)c2)cc2c(nc1N)CCC2 60246,C1(C(N(C(C)CCNC(=O)CCSC(F)(F)F)C)=O)C2CC3C(C2=O)C13 60247,C1(CNC(COc2cc(C)on2)=O)CN(C)CCN1C(C1CCCN1C1CC1)=O 60248,N1(C(CNC(=O)CC2CCS(=O)(=O)CC2)=O)CC2CC1CN2C(C1CC1(F)F)=O 60249,C(C(C)(O)C(C)CC)OC.C(Cc1cnc[nH]1)(C(=O)NC1CC(NC)C1)OC=O 60250,C1(OC)C2CC3CC1CC(C(N1C4CCC1C1CC1(NC(=O)COC)C4)=O)(C3)C2 60251,c1(OCC)c(CC(N2CC(OC)C(NC(=O)C(C)CC(N)=O)C2)=O)cccc1Cl 60252,C#CC1(C(=O)NCC2CC(C(=O)N3CCC(O)C(C)C3)=NO2)CCCCC1 60253,C1(N(C(=O)C(O)CC2CCCO2)C)CCN(C(=O)C(C)(C)c2ccccn2)CC1 60254,c1(OC)cnnc(C(=O)NCC=CCCC(C)C=O)c1.OC 60255,c1(C(=O)NC(CCC)CNC(=O)C(N2CCCC2)C2CC2)cn(CC)nc1C 60256,C1(OC)NC(C(=O)NCCn2cc(CN3CCNC3=O)nn2)CCC1Br 60257,N1(Cc2c(OC)ccs2)Cc2[nH][nH]c(=NC(=O)c3ccc(F)c(C#N)c3)c2C1 60258,N1(C(C(C=C)(C)C)=O)CCC2(CC1)OCCC2NC(C1CCCN(C(C)=O)C1)=O 60259,N1(C(CCOC)=O)CC2CC1CN(C(=O)CCc1cc(C)[nH]n1)C2 60260,N1(C(C(C)CSc2ccccc2)=O)CCC2CCC(C1)N2C(=O)CCC(F)F 60261,N1(C(CC2CN(C(c3cc(CC)[nH]n3)=O)C(C)C2)=O)CCC(C)(C2CC2)C1 60262,CCC(C)CCC(=O)NCC=CCNC(C12CCC(CC(C)(C)C)(CO1)C2)=O 60263,N1(C(C(CCCC)NC(N)=O)=O)CCN(C(=O)C=Cc2ccsc2)CCC1C 60264,Cc1cc(Cl)cc(C(=O)N(C)CCNC(c2ncc(Cl)cc2Cl)=O)c1N 60265,C(=O)(C(C)C(C)S(C)(=O)=O)NCC1(CNC(CCOCCC)=O)CCCC1 60266,c1(C(N2CCCC(NC(CCC#CC)=O)C2)=O)ccc(C#N)c(C)n1 60267,C(C)(C(O)C(=O)NCC#CCNC(=O)C(C)(C)Oc1ccccc1)SC 60268,c1(C(c2n(CC)nnn2)Nc2cccc(CO)c2)cc(Cl)c(Br)cc1F 60269,c1(OC)ncc(Br)cc1CN1CCCN(C(c2ccnn2C(C)C)=O)CC1 60270,N1(C(c2ncc(C)nc2)=O)CCC2(CC1)CC2(CO)CNC(c1cocn1)=O 60271,C1(C(=O)NCC(CNC(c2c(CC)scc2)=O)(C)C)CCC(N(C)C)CC1 60272,C1(NC(C(OC)OC)=O)CS(=O)(=O)N(C)C12CCN(C(=O)CC1(C)CCC1)CC2 60273,c1(OCCC)cccc(C(=O)NCc2cnsn2)c1 60274,C1(NC(C(C)SC(C)C)=O)CCCN1CCNC(=O)Nc1ccccc1 60275,c1(C(=O)NC(C(C)NC(c2csc(CO)n2)=O)C)ccccc1Br 60276,C(CN(C(=O)CC1CN(C(C)=O)C1)C)(CO)(CO)NC(c1cc(COC)sc1)=O 60277,C(C)(CCC(=O)NCc1nc(CO)n[nH]1)NC(CCC=CCC=C)=O 60278,N1(C(C2CC(CC)C2)=O)CC(C)(C)OC2(C1)CN(c1cc(OC)nc(OC)n1)C2 60279,C1(CCCNC(c2c(C)occ2)=O)CN(C(=O)CN2CCOC2=O)CCO1 60280,c1(CN(c2ccc(Br)cn2)C(C2CC2C2CCCN2)=O)cc(C(F)(F)F)ccc1Cl 60281,Cc1ncc(C(N2CCC(NC(C3C4CNC(=O)C34)=O)C2)=O)cc1C#N 60282,C1(CN2CC(NC)C(O)C2)CC2(CCCO2)C1 60283,N1(c2nccc(OCCC)n2)CC2(CCC(NC(c3ccc(O)cc3)=O)CC2)C1 60284,N1(C(CS(=O)(=O)NC)=O)CC2CCCC(NC(=O)C(O)C3CCCC3)C2C1 60285,N1(C(c2c(C)ccs2)=O)CC2CCN(C(=O)C(c3ccc(Cl)cc3)O)CCC2C1 60286,CS(=O)(=O)c1cccc(SCC(N2CCCC(N3CCCC3)CC2)=O)c1 60287,C1(CNC(c2n(C)cnc2)=O)C2CC2CN1C(c1cncc(O)c1)=O 60288,c1(C(=O)Nc2ccc(NCC3C(N)CC=CC3)cc2)ccc(O)c(C(=O)O)c1 60289,C1(CC)C(NC(=O)COCCOCCO)CCN1C(=O)CCc1cccnc1C 60290,c1(OC)cc(F)c(Br)cc1C(=O)NCC(O)CNC(=O)C=Cc1cnc[nH]1 60291,Cc1c(C(N2CC(O)(CC(N3CC(N(CC(C)C)C)C3)=O)C2)=O)ccn1C 60292,N1(C(C(C)C(C)(C)C)=O)CC(NC(c2occc2Cl)=O)C(C2CC2)C1 60293,CC1CCN(CCC(=O)NC(C)(C)C2(C3CCCN3C(CC(C)(C)C)=O)CC2)CC1 60294,C1(C)(C(N2CC(CC(=O)NC(COC)C3(C)CC3)(OC)C2)=O)CCC(O)CC1 60295,C=CCN=C(NCC(=C)CC)NCc1csc(COCC)n1 60296,CC1CCN(C(c2c(C#N)ncn2C)=O)CC1CC(=O)N(C)CCF 60297,C(=O)(C1=C(C2CC2)N(CC(F)F)C(=S)NC1c1cn2ccsc2n1)OC 60298,c1(C(N(CCNC(C(C(CC)O)C)=O)CC)=O)cc2ccc(Cl)cc2[nH]1 60299,c1(C(N2CC(CNC(c3nc(C)oc3)=O)C(C)C2)=O)cccc2occc12 60300,N1(C(c2c(CC)cno2)=O)CC2CCC(NC(=O)CCc3ccon3)CC2C1 60301,C=CC1(CC(N2CC(CC3CC3)C2)=O)CN(C(S(C)(=O)=O)=O)C1.C1(C)(N)CCOC1 60302,C(N=c1nc2sccc2c(N2CC=C(Cl)C2)[nH]1)c1ccc(-c2ccn(C)n2)o1 60303,C1(NC(C(CC)F)=O)CN(C(=O)COCC(F)F)C2(CCOCC2)C1 60304,C1(NC(CC2CC(=C)C2)=O)CCC(C(=O)NC2(COC)CC(F)C2)CC1 60305,Cc1c(C=CC(N2CCC(C)C(NC(=O)C(C)(C)N3CCCC3)C2)=O)cnn1C 60306,c1(C(=O)NCCC(C(C)C)NC(C(C=CC)O)=O)ccc(Cl)c(F)c1 60307,c1(CC)[nH]nc(C(=O)NC2CCCCCC2NC(=O)CC(C)C)c1[N+](=O)[O-] 60308,C(CCN(C)OC)NC(C1N(C(C(CC2CC2)OC)=O)CCC1)=O 60309,CN1CCN(C(c2cnc[nH]c2=N)=O)CC1C(=O)NC1(C)CCCC1O 60310,c1(C(N2CCC(N(C(CNC(CC(C)C)=O)=O)C)C2)=O)ccc(C(C)C)cc1 60311,c1(CNC(CCCC#CC)=O)ccc2c(c1)CN(C(c1cccc(Cl)c1C)=O)C2 60312,C1(C)(C(N(CC)Cc2ccoc2)=O)CC(O)CN1C(=O)CC1CCCC2CC12 60313,CCC(Cc1ccccc1)CC(=O)NC(CNC(=O)CC1(O)CCOCC1)CC 60314,C1(C(N(CCC)CCNC(C2CC2c2cccs2)=O)=O)SCCCS1 60315,c1(C2CC(c3n(C)nnn3)(NCC3CC(F)(F)CO3)C2)cc(Br)ccc1Cl 60316,c1(C(=O)NCCOCCNC=O)cc(Cl)ccc1C.C1(C(C)C)CC1C(=O)OCC 60317,c1(C(=O)NC2C(CNC(CC3(NC(C)=O)CC3)=O)C2)coc(C#N)c1 60318,N1(C(C2OCC3CCCCC23)=O)CCC2(CCN(C(c3cnccc3Cl)=O)C2)C1 60319,C(=O)(C1CCCc2ncccc21)NCC(CNC(c1cn(CC(N)=O)nn1)=O)F 60320,c1(C(C)OC)ccc(CN(CCO)CC)cc1.C(COC)S 60321,C1(C(N2CCC(OC)(CNC(c3cscc3Cl)=O)C2)=O)CCC2(CCC2)CC1 60322,C1(NC(C(CC=C)(C)N(C)C)=O)CC2(CCN(C(=O)C(n3cc(C)cn3)C)C2)C1 60323,C=CCCCC(C)NC(C1(NC(C2CCCCC2)=O)CC(F)(F)C1)=O 60324,CC(C(C)(C)C(=O)NC1CCC2(CCC2)C1)NC(=O)CCC(=O)NC1CC1 60325,N1(C(c2cc(C)sn2)=O)CC(C(=O)NCC2(C)CC=CCC2)C2(CC2)C1 60326,C12(NC(=O)Cc3cccnc3)CCCC1CN(C(c1cccc3c[nH]nc13)=O)C2 60327,c1(COC(N(CCCC(=O)NCC(CCC)C)C)=O)ccc(F)cc1 60328,N1(C(C(c2ccc(CC)[nH]2)=O)=O)CC(NC(=O)Cn2nc(C)cc2C)CC(O)C1 60329,c1(C(N(CC(C)N(C(=O)CC(C)C(F)F)C)C)=O)ccc2c(c1)CCC2 60330,N1(C(C=NOC)=O)CCC2(CC1)OCCC2NC(C1CC1c1ccccc1)=O 60331,c1(C(N2C3C(NC(CCc4scc(C)n4)=O)CC(C3)C2)=O)cccc2c1CCO2 60332,c1(C(=O)NCCCC(C)NC(CC2(C=C)CCCCC2)=O)coc(S(N)(=O)=O)c1 60333,C1(CC)CCCCCCN1C(C1CC(CCNC(C2OCCC2(C)C)=O)C1)=O 60334,c1(C(=O)NCCC(C)N(C(C(CC(=C)C)C)=O)C)nn(C)c2ccccc2c1=O 60335,c1(CC(=O)NC2CCCCN(C(=O)C(=O)NC3CC3)C2)cccc(F)c1Cl 60336,C(C(=O)N1CCCC(C(=O)NCCOCCN(C)C)C1)(C(C)C)OC 60337,CC(C)CCC(=O)NCC(=O)NC1CCC(NC(c2nc(C3CC3)cs2)=O)C1 60338,CC1(CNC(=O)CCC(N)=O)CCN(C(=O)C(c2ccccc2)O)C1 60339,c1(C(N2CCCC(NC(C(C)OCCC=C)=O)C2CC)=O)cnc2n1CCCC2 60340,c1(C(N2C3CN(S(CC(=O)OCC)(=O)=O)CC32)=O)ccc2nc[nH]c2c1 60341,N1(C(c2c(C)n(CCO)cc2)=O)CC(C)CCC1C(=O)NC1CC(OC(C)C)C1 60342,C(=O)(CS(C)(=O)=O)NC(C)(C)C.C12CCCC1NC(=O)C(C)NC2=O 60343,N1(C(C(C)(C2CCC2)NC(=O)Cc2ccsc2)=O)CC2CC(O)CC2C1 60344,CN1N=C(CC(=O)NC2(C)CCN(Cc3ccncc3Cl)C2)CC1=O 60345,c1(C(C)(C)C)ccc(C(=O)NC2(CNC(c3ccoc3)=O)CCOC2)s1 60346,C1(C(=O)NC2(C)CN(C(C(COC)(F)F)=O)C2)CC2(CCC2OC)C1 60347,C1(NC(c2[nH]cc(CC)n2)=O)CCCN(C(c2cc[nH]c2C2CCC2)=O)C1C 60348,CCCC(C)C(C)NCC1CC1C(=O)OC(C)(C)C 60349,C1(NC(C(CCC)CNC(=O)CCCNC(N)=O)=O)C2CCCCCCC12 60350,Nc1cnc(C(=O)NC2CCC2NC(c2cccn2C2CCCC2)=O)cn1 60351,c1(C(N(CCC(N2CC3(C2)CC3(F)F)=O)C)=O)ccc2[nH]nc(Cl)c2c1 60352,c1(C(N2CC(OCCNC(c3cc(CCC)n(C)n3)=O)C2)=O)cnc(N)c(Cl)c1 60353,C1(CNC(c2c(C)snn2)=O)(OCCNC(C2CCC3(CC3)C2)=O)CCOCC1 60354,c1(C(C(=O)NCCC(=C)CNC(c2ccnc(OC)c2)=O)O)ccc(Cl)c(Cl)c1 60355,N1(C(c2cnc(C(C)C)s2)=O)CCC(NC(=O)CSCc2cccs2)CC1C 60356,N1(C(C)=O)CC(NC(C2CC2c2cccc(C(C)C)c2)=O)CC1(C)C 60357,C(=O)(CC(C(F)(F)F)n1ccnc1)NCCC(C)NC(c1ncc(F)cc1F)=O 60358,C=CCC(CNC(c1ccnn1C1CC1)=O)C(=O)N1CC=CC1 60359,c1(CC)ncc(C(=O)NC(C2CC(NC(=O)C(N3CCNC3=O)C)C2)C)c(C)n1 60360,Cc1cn2ccc(C(=O)NC(CNC(=O)C(C)(C)N(C)C)C(C)C)cc2n1 60361,c1(C(=O)NCC(=C)CCNC(c2ccnn2C)=O)nccnc1C 60362,c1(NCCOCCNC(C(C)NS(C)(=O)=O)=O)cnn2ccncc12 60363,c1ccc2c(c1)CCCC2CCc1noc(-c2cc[nH]c2C2CCCN2)n1 60364,C(c1ccsc1)=CC(=O)NCC=CCNC(C1CC(=C2CCC2)C1)=O 60365,CC=C=CCCN=c1nc(N2CCOC(CF)C2)c2ncccc2[nH]1 60366,c1(CC)cc2c(NC3(CO)CCCN(C(=O)CC4CC4(Cl)Cl)C3)nc(C)nc2s1 60367,c1(COC(c2c(C)nc(-c3ccccc3F)s2)=O)nc2ccsc2s1 60368,N1(C(c2c(CC)[nH]cc2)=O)CCCC(O)(CNC(C2(CO)CCOCC2)=O)CC1 60369,c1(C(=O)Nc2ncc(CCNC(=O)CCC3CC3)s2)ccc2ccccc2c1O 60370,c1(C(N2CC(NC(C=CC)=O)C(C(F)F)C2)=O)nc(OC(C)C)ccc1Cl 60371,c1(C(=O)NC(C2CCCN2C(=O)C#CC2CCOC2)C)ccc2c(n1)CCCC2 60372,c1(C(=O)NC2CC(NC(Cn3c(C)c(Cl)cn3)=O)C2)cc(O)cc(Cl)c1Cl 60373,N#CC1(C(=O)NCC23CC(CNC(C4CCNC4=O)=O)(CO2)C3)CCC(=O)CC1 60374,c1(N(C)C(c2cccc(Br)c2)C2CC2)ccc(S(N)(=O)=O)c(F)c1 60375,CS(=O)(=O)CCCNC(C1CC(NC(c2cccc(CN3CCCC3)c2)=O)C1)=O 60376,N12CC(F)(F)CC1C(=O)N1CC(CCC=C)(C1)C2=O.C1(CO)CC(C=C)C1 60377,C1(CC(=O)NC2C3CCN(C(c4cocn4)=O)C23)CCC=CCC1 60378,c1(N2CCC(C=C)CC2)nc(=NC2COCC2C2CC2)[nH]c2ncn(C)c12 60379,c1(C(=O)NCC(C)NC(Cc2cc(CC)no2)=O)cc(-c2ccccc2)ncn1 60380,N1(C(C2CC(C)(O)C2)=O)CCC2(CC1)CN(C(=O)CCC1CCC1)C1COCC21 60381,C1(NC(c2ccc(OC)c(I)c2)=O)CC2CCC(C1)N2C(=O)Cc1cc[nH]n1 60382,c1(C(=O)NC2CN(C(C(C(C)C)OC)=O)CC2C)cn2cc(Br)sc2n1 60383,N1(C(Cc2cc(C)on2)=O)CCC(NC(=O)Cc2c(C)n[nH]c2C)C(CO)CC1 60384,S1(=O)(=O)c2ccc(Br)cc2N1.Cc1cc(C(=O)NOCC(C)C)nc(C)c1 60385,CC(C)(C)C(=O)C(=O)NC1CCC(NC(=O)CSCCC(F)(F)F)CC1 60386,C1(C(=O)OC)(NC(=O)NC2CCOC2c2ncnn2C)CC(O)C1(C)C 60387,C1(CCNC(C2(C)CC(F)C2)=O)CCCN(CC(=O)N)C1.c1(CN)ccccc1 60388,c1(C(N(CC(CN(C(C(C)NC(=O)OC)=O)C)O)C)=O)ccc2nc(C)nn2c1 60389,C1(CC(=O)NC(CC2CCCO2)C(F)(F)F)CNC2(CC2)CO1 60390,c1(CC)ncc(C(=O)NC(C)CCNC(c2sc(=N)[nH]c2CC)=O)cn1 60391,N1(C(C(C)O)=O)CCc2[nH]nc(CNC(=O)CCC3CCOC3)c2C1 60392,S(=O)(=O)(c1csc2ccccc12)N1CCC(NC(c2nc(Br)ccc2Cl)=O)C1 60393,C(=O)(CCC(C)C)NCC(CCOC)NC(C1CCCCS1)=O 60394,CC(C)C(CCC(=O)N1CC2CC3CC2C1C3)NC(C1OCCC1(C)C)=O 60395,C(CS(=O)(=O)CC(=O)NCC1CC(C)N(C(=O)CCCC(C)O)C1)OC 60396,CC1(CCc2ccccc2)CCCN1N1CCCC2(CC1)NC(=O)NC2=O 60397,N1(C(c2ccc(OC(CC)C)cc2)=O)CCC(NC(=O)C(C)=CC2CC2)C(O)C1 60398,C12(C(=O)OCC)CCC(CC1)N(C(c1ccn3c1CCC3)=O)C2 60399,C(CC(=O)NCCc1nccs1)N(C(C)C)C(C1CC(=C2CC2)C1)=O 60400,CC(C(=O)NCCOCCNC(=O)COC1CC=CC1)c1ccsc1 60401,N1(C(C(C=C)(C)C)=O)CC(C2CCCN(C(=O)CC3CC4CCC3O4)C2)C1 60402,C1(NC(C2(C#C)CCC2)=O)CCC(C)(C)CC1CNC(c1coc(C(F)F)c1)=O 60403,c1(CC)cc(C(N2CCC(NC(=O)CCc3nc(O)n[nH]3)CC2C)=O)cc(C)c1 60404,C1(CN(C)C(c2cccc(O)c2)=O)CCCN(C(=O)CN2CCCC2CO)C1 60405,N1(C(C(C)N(C(c2ccon2)=O)C2CC2)=O)CC2(C1)CC(C)(C)C2 60406,c1(OC)cc2nn[nH]c2cc1C(=O)NC1CC(NC(=O)C(C)(C)CC#N)C1 60407,n1(CC(=O)Nc2cccc(NC(C3CCC(=O)NC3=O)=O)c2)ncc2ccccc12 60408,CC1(C(=O)NCC2C=CCN2C(=O)CCc2ccco2)CC(F)C1 60409,N1(C(C2C(C)(CC)C2)=O)CCOC(CNC(=O)CCCCN2CCOCC2)C1 60410,C1(=O)NN2CCN(CC2)C(C)(C)c2cn1nn2.Cc1n[nH]cc1-c1nn[nH]n1 60411,N1(CC)CCC(NC(=O)CN(C(=O)CCc2ccc(C)cc2)CC)C(C)C1 60412,c1(OC)csc(C(=O)NC(C)CC(C)NC(C23CC2C3)=O)c1 60413,c1(C(N2CCC(C)C2CNC(=O)CC2(C)CCOC2)=O)cc[nH]c2nccc1-2 60414,C1(C(N2CCC(NC(c3c(C)nc[nH]3)=O)C2)=O)CCCC(=O)N1C.C1(O)CC(C(=O)O)C1 60415,c1(C(N(CC(C)NC(c2cccc(OC)n2)=O)C)=O)ccc2c[nH]nc2n1 60416,N1(C(C2(N(C)C)CC2)=O)CCOC2(CCN(C(C3CCCC(F)C3)=O)C2)C1 60417,Cc1c(C(c2cccs2)N(C(C)CCC(C)C)C)cccc1F.C1C(=O)N1 60418,c1(C(N(C)CC2N(C(CC(C(C)C)O)=O)CCC2)=O)ccn2ccnc2c1 60419,C1(C(=O)NCCC2(CNC(C(CSC)O)=O)CC2)CC(=O)N(c2nccs2)C1 60420,c1(C(=O)NCCCN(C(c2cn(C)nc2C2CC2)=O)CC)ccccc1F 60421,c1(C(=O)NCCC(C)NC(C(C(C)C)C#N)=O)c(C)oc2ncnc(O)c12 60422,C1(CC)CN(C(C2CCN(C3CC3)C2=O)=O)CCN1C(=O)Cn1nccn1 60423,c1(C(=O)NC(CCC)CNC(=O)C(C)=C(C)C)cc(Cl)nn1C 60424,C(=O)(C1CC(=O)Nc2ncccc21)NC(C)(C)CCCNC(=O)C(O)C1CC1 60425,c1(C(=O)NCC(C)(C)NC(=O)CSc2ccccn2)cccnc1O 60426,c1(C(N(CCCCCC)CCNC(=O)C(C)CC2CC2)=O)ncc(N)cc1Cl 60427,c1(CCC(N2CCC(N(C)CC3CC(F)(F)C3)C2)=O)cc(F)ccc1F 60428,C1(CNC(C2CCC(C)(C)C2)=O)CC(F)(F)CN1C(C1C2CCC(=O)C12)=O 60429,C(=O)(C(C(C)CC)NC(=O)C(CC1CC1)OC)N(CC(CCC)C)C 60430,C(=O)(C(CC(C)C)OC)NCC(CC)N(C)C(C1COCCN1C)=O 60431,C1(C(=O)Nc2cccc(C)c2C#N)C2CCCC1CN(C(c1c(C)cc[nH]1)=O)C2 60432,Cc1cc(=O)oc(C)c1C(=O)NC1CCCCN(C(=O)CCC2(C)CC2(F)F)C1 60433,c1(C(F)(F)F)cccc(C#CCNCCSc2cc(Cl)sc2Cl)c1 60434,C1(C(=O)NC2(C(N(C)C(C3CN(C4COC4)C3)=O)=O)CCC2)CCN(C2CC2)C1 60435,C1(C(N(C)CC2(NC(C=CCCC=C(C)C)=O)CC2)=O)Cc2cccnc2C1 60436,CCC(CNC(c1conc1CNC(C1CNC(=O)N1)=O)=O)CC(C)C 60437,C1(C(=O)NCCN(C(CC2(C=C)CC2)=O)CCc2ccccc2)CN(C)CCO1 60438,CCCC(C(=O)N1CCC(CCC(=O)N(C)CCOCC2CC2)C1)NC(C)=O 60439,CC(=O)CCCC(=O)NCC1CC(NC(C2(c3cc(C)no3)CC2)=O)C1 60440,c1(C(=O)NC2CC(C)(CNC(C(CC=CC)C)=O)C2)ccc(F)c(C(=O)CC)c1 60441,N1(CC(=O)N(C)C)CCCC(C(=O)NCc2cccc(CN)c2)C1 60442,c1(NC(C2CN(C(C(CCC)(C)C)=O)CC(F)C2)=O)ccc(F)c(Cl)c1F 60443,c1(CC)cccnc1C(=O)NC1CCCC1NC(C1COC(=O)O1)=O 60444,c1(CNCC23CC(C(=O)Nc4ccc(Br)cc4I)(C2)C3)c[nH]c2cccc(F)c12 60445,c1(C(N2C(CC(=O)OC)CC2)=O)cc(Br)ccc1C 60446,C1(CCCC)CN(C(c2n[nH]c(C)c2Br)=O)CCN1C(=O)CC(C)F 60447,C=C(F)C1(CC(=O)NCC2(NC(C3CC4(CCC4)CO3)=O)CCC2)CCOCC1 60448,S(=O)(=O)(c1ccc(F)cc1F)N(C1CC2CNC1C2)C(=O)CC1CCCC1 60449,c1(C(C)OCC)noc(CN(C)C(C2(C)CCCS2)=O)n1 60450,c1(C(=O)NC2CC(NC(Cc3nc(C)sc3)=O)C2)ncnc2sccc12 60451,C1(CNC2CCC(NC(c3cnn(-c4ccccc4)n3)=O)C2)CCC2(CCC2)C1 60452,CCC(C)C(C)(O)COC(c1cncc(C=CC(=O)N(C(C)C)C(C)C)c1)=O 60453,CC(C)CCCC(=O)N1CC(O)(CN(C)C(C2CCCCN2CC(F)F)=O)C1 60454,N1(C(C(CC(C)(C)NC(c2cn(CCC)nn2)=O)F)=O)CCC2(CC=CCO2)C1 60455,c1(NC(CN2CCN(C(C3=CCCCC3C)=O)CC2)=O)cnc2ncnn2n1 60456,C(CN=c1c(C#N)c[nH]c2ccc(C)cc12)N(C(C1CCC(C)C1)=O)CC 60457,O=S(=O)(c1cnc(N2CCCC(OCCF)C2)c(Cl)c1)NCC1(CCCO)CC1 60458,c1(C(=O)NC2CCC(NC(CC(CC)OC)=O)CC2)ccc2c(c1)CCN(C)C2 60459,c1(C(=O)NCC2CCN(C(c3c(N(C)C)cccn3)=O)C2)ccc(P(C)(C)=O)s1 60460,C1(CC)CN(Cc2ccccc2N(C)C)CCN1C(=O)Cc1ccsc1 60461,C1(NC(n2nnc(C)c2CC)=O)CC2CN(C(=O)COCC3CCCO3)CC2C1 60462,c1(OC(C)C)ccc(C(=O)NCC(CO)NC(c2ccccc2)=O)cc1 60463,CCCC(C)(C)CC(=O)NC(CCC(=O)N1CCC1C(N)=O)C(C)C 60464,C1(COC)(CNC(C2(NC(c3ccn(C)n3)=O)CC(O)C2)=O)CCOC1 60465,c1(CC)cc(C)nc(N2CCCC2CCCNC(C2(C3CC3)CCCO2)=O)n1 60466,Cc1ccc(C(=O)NC2(CS(N)(=O)=O)CC2)nc1C 60467,C(=O)(C(C)(CSC)NC(=O)C=Cc1ccoc1)NC(C#C)C 60468,C1(NC(C(=O)N(C2CN(S(C)(=O)=O)C2)C)=O)CC(C)(C)C(C)(C)C1 60469,C(C(C)(C)CNC(c1ncoc1C1CCC1)=O)N(C)C(c1coc(Br)n1)=O 60470,CC1C2CCCCC2CN1C(=O)C(CC1CC1)NC(C1CCC(=O)O1)=O 60471,c1(CSCCC(=O)NCCC2CCN(C(CC(=O)OCC)=O)C2)ccc(F)cc1 60472,N1(C(c2ccc(C#C)cc2OC)=O)CCC2C(CCCN2C(=O)CC(C)(C)C)C1 60473,C=CC1(C(=O)NCCCc2ncn(C)n2)CCN(C(=O)CCc2cccs2)C1 60474,CC1(C#CC(=O)NC2CC3CCC2N3C(c2cc(Cl)c(Cl)s2)=O)CC1 60475,C1(CNC(=O)Cn2ccccc2=O)CCC2(CN(C3CCCNC3=O)C2)O1 60476,C1(NC(Cc2c(C)non2)=O)CN(C(C23CC2COC3(C)C)=O)C2(CCC2)C1 60477,c1(C(=O)NC(C2CN(C(=O)C(C)(C)C(=O)N(C)C)C2)C)nccc(Cl)c1C 60478,CCC(C)CC(C)C(=O)NCC(C)=CC(=O)Nc1cc(CO)cc(C)c1 60479,CC(CC(=O)N1CCC1C1CCOCC1)NC(=O)COCc1ccnn1C 60480,C=CCC(CC(=O)N1CCC(COC)CC1)NC(=O)C(C)(C)COC 60481,C1(F)(CNC(=O)CC(F)F)CCCN(C(c2ccoc2Cl)=O)CC1 60482,CC(CC(=O)NCCSCC(=O)N(C)CC1(CO)CCC1)C(F)(F)F 60483,C(CCCCC(=O)NCc1nccn1C)N(C)C(C1(F)CCOCC1)=O 60484,c1(C(=O)NCC2CC(F)CN2c2ccnc(Br)n2)nc(C(F)(F)F)ccc1Cl 60485,C1(NC(C=C)=O)CCCC2CN(C(C3Cc4cccc(C)c4O3)=O)CC12 60486,CC1(C)CCCN(C(=O)CCCC2CCCO2)C1C(=O)NC1CC=CCC1 60487,C1(NC(C(C=C=C)C)=O)CCCCN(C(c2cnc(OC)s2)=O)C1 60488,CC1(NC(=O)CC2CCCC23CC3)CCN(C(=O)Cn2nnc(=N)[nH]2)CC1 60489,CC#CCCCC(C(=O)O)NS(=O)(=O)c1ccccc1C1CC1(F)F 60490,c1(OC)ccc(F)c(C(=O)N(CC(C)(C)CNC(C2CCCC2(C)C)=O)C)c1N 60491,C(C(C)C(C)C(=O)N1CCCC1CN(C(=O)CCNC(c1ccco1)=O)C)OC 60492,CC1CC(OCCSC(C)(C)C)CCO1.C1(=O)C(C)(C)O1 60493,C12(CNC(c3ccoc3)=O)CCCC1N(C(c1ncnc3sccc13)=O)CCC2 60494,C1(NC(C2CCC(=O)NC2)=O)CCCCN(C(=O)C(c2cccc(Br)c2)O)C1 60495,C1(C(=O)NC2(CC=C)CCCCC2)CC(C)CN(C(=O)Cc2ccc(O)cn2)C1 60496,C1(CCC)(NC(=O)CCc2cnoc2)CCN(C(c2ccc([N+](=O)[O-])s2)=O)CC1 60497,C1(C(=O)NCCC2CCN(C(C(c3n(C)ccn3)(F)F)=O)C2)CCC(F)(F)CC1 60498,N1(C(c2cn(C(C)(C)C)nn2)=O)CCN(CCCNC(c2n[nH]cc2Cl)=O)CC1 60499,CCC(C)(CNC(=O)CN1CC2CC2C1)C(=O)N1OC2CCC1CC2.C(=O)(CSCC)N 60500,C#CC1CCN(C(C2COCCN2C(=O)C(C)=C2CCCC2)=O)CC1 60501,CC1(C(=O)NC2CN(C(c3cccc[n+]3[O-])=O)CC2C(F)F)CCC(O)CC1 60502,c1(C(=O)NCC2CCCCN2C(=O)C2=NOCC2)n[nH]c2cc(Br)ccc12 60503,c1(C(=O)NC2CC3CN(c4ncc(C#N)nc4)CC32)nnn2c1COCC2 60504,C12(NC(CC(COC)NC(=O)Cn3nc(C)nc3C)=O)CCC(C1)OC2C 60505,C1(C(N2CCC(C)C2)=O)(CF)CCN(C(C2CC3CCC2O3)=O)C1 60506,C=Cc1cccc(CN2CCCC(NC(=O)CCc3ccccc3)C2)c1 60507,C1(NC(C=CC)=O)CN(C(c2cc(C)cc(Br)c2OC)=O)CC1N=[N+]=[N-] 60508,c1(C(C(=O)NC(C(=O)OC)C)N(C(C)C(F)F)C)ccc(OC)c(Br)c1 60509,CCCCC(O)C(=O)N(CC(N1CCC(O)(CCC)CC1)=O)C 60510,c1(C(=O)NCCN(C(C(c2cnn(C)c2)OC)=O)C)nc(C)n2ccccc12 60511,CC(CC(C)(C)C)C(=O)NCC(C)(CO)NC(=O)CCc1nnc(C(F)F)o1 60512,c1(C(N2CC(F)(F)CC2CCNC(=O)C(F)(F)CC2CC2)=O)cccc(=S)n1O 60513,c1(OC)ccccc1C(CF)NC(=O)NCC(C)(O)CCO 60514,Nc1cccnc1S(=O)(=O)NC1CC(=O)NC1c1ccccc1 60515,c1(C(N(C2C3CN(C(C(C(C)(C)C)OC)=O)CC32)C)=O)cccc2c1OCCC2 60516,c1(C(=O)NCC(C)N(C(c2c(C)c(F)ccc2)=O)C)cc(N)c(Br)c(F)c1 60517,N1(C(C2C(SC)CCC2)=O)CC2CCC(CNC(C3CCCN(C)C3)=O)(C2)C1 60518,C=C(C)C1OCCCC1C(N1CCC2(C1)CN(C(c1cc(O)ncn1)=O)C2)=O 60519,C1(NC(C=C(C)c2ccsc2)=O)CCC2(CC1)CN(C(=O)C(C)S(C)(=O)=O)C2 60520,CN1CCNC(=O)C12CCCN(C(c1cnc3ccc(Cl)nn13)=O)C2 60521,C1(C(=O)NCC2(CO)CCCC2)CC2(CCC2)CN1C(c1ccnc(O)c1F)=O 60522,C(c1ccc(C)cc1)=CCC(N1CC2C(CNC(C(CCC)OC)=O)(C2)C1)=O 60523,C1(NC(=O)CC2CC3C=CC2C3)CC2CC1N(C(C1CCCCC1)=O)C2 60524,c1(C(N2C(C(N3CC(C(CC)C)C3)=O)CNC(=O)C2)=O)ccc2[nH]ccc2n1 60525,C1(OC)CCC2(C(=O)N(CC(C)C(=O)N(C)Cc3cnco3)C)CC12 60526,Cc1cc(Br)cnc1C(N1CCC(NC(=O)CCN2CCC2)C1C1CC1)=O 60527,C(CN=c1nc2c(ncn2C)c(NC2CCN(C)C(C)C2)[nH]1)OCCOCCC 60528,c1(C(=O)NCC(CC(F)(F)F)NC(=O)C(O)C2CCC2)cc2ccc(F)cc2[nH]1 60529,C1(NC(c2c(CC)nc[nH]2)=O)CC2(CCN(C(=O)C(C)CCCOC)C2)C1 60530,C(CCC(O)C(=O)NC1CCOC(C)(C)C1)NC(C1(OC)CC(C)C1)=O 60531,N1(C(CCCc2onc(C)n2)=O)CCC2(NC(c3ccncc3)=O)CC2C1 60532,N1(C(CCCCN(C)C)=O)CC2CCN(C(c3snc(Cl)c3Cl)=O)CC2C1 60533,Cc1cnc(C)c(C(=O)NC(C)C(C)(C)NC(=O)CSc2ccc(F)cc2F)c1 60534,c1(C(=O)NC2C(NC(C(CC)(C)C#N)=O)CC2)cc2c(cc1F)OCC(=O)N2 60535,N1(C(C)=O)CCCC(CC(=O)NC(C)(CNC(=O)C2=COCC2)C(C)C)C1 60536,c1(SC)cc(C)c(C(N2CCC(C(C)(C)C)(CNC(=O)C(=O)NC3CC3)C2)=O)s1 60537,C(=O)(C(C)C(C)(C)C)NCc1cc(C(=O)NCC(C#C)C(C)C)sc1 60538,c1(C(N(C)CCN(C)C(C2(O)CCOC2)=O)=O)ncc(C(C)(C)O)cn1 60539,c1(NC(=O)NC2C(CCCC)CCC2)cnc(O)n(C)c1=O 60540,C1(NC(CC2(CC)CCOCC2)=O)COC2(CCCN(C(=O)C(F)=C(C)C)C2)C1 60541,c1(-c2cc(CCN(C)C)on2)nc(C2CCCCC2)nn1CCS(C)(=O)=O 60542,c1(OC)ccc(CCCNC(=O)Cn2cc(CC3CCCC3)nn2)cc1.C1CC1 60543,Cc1ncnc(C)c1C(=O)N(CCCNC(=O)C1=NOC(C)C1)C 60544,C1(C(N2CCC(N(C(C3(C4CC4)CC=CC3)=O)CC)C2)=O)(OC)CCS(=O)(=O)C1 60545,c1(NC(CC2OCCN(Cc3c(NC)cccc3)C2)=O)cc(OC)nc(C#N)c1 60546,N1(C(CC2(SC)CC2)=O)CCC(C(=O)N(C(C)C)C(C)C)C1C(C)C 60547,N1(C(C(CO)N(C)C)=O)CCC(C2CCN(C(=O)Cc3cnns3)CC2)C1 60548,N1(C(C=CC(C)(C)SC)=O)CCCC2C1CCCN2C(c1ccoc1C1CC1)=O 60549,C1(C(=O)NCc2c(C(C)C)nco2)CCC2(CCN(C(=O)OC(C)(C)C)C2)O1 60550,C(C(C(=O)NCc1c(C)nnn1CC)NC(C1C=C(C)CS1)=O)OCC 60551,c1(OCC)cncc(C(=O)NC2CCCC2NC(=O)C(C)NC(=O)C(C)(C)C)c1 60552,C1(N(CC2C(=O)N2)C)CC2CN(C(C)=O)CC12.N1(CCC=CC)CCNC(=O)C1 60553,c1(OC)ccc(C=CC(=O)NCCCCCNC(=O)C(C)(C)C2CC2)cc1 60554,C(CC)(CC)(CCNC(=O)CCCCC#N)NC(c1ncc(CC)nc1)=O 60555,c1(CC(N2CC3C(NC(C4C(=C)C4)=O)(CCC3)C2)=O)c[nH]c2ccc(OC)cc12 60556,C12(NC(C(Cc3c(C)n[nH]c3C)C)=O)CCCC(CN(C(=O)C#CC3CC3)C1)C2 60557,CCC(C)(F)C(=O)NCCC1CCC(NC(c2ccccc2NC(N)=O)=O)C1 60558,C#CCC(CC(F)F)C(=O)NC1CC=C(C(=O)NC2(CO)CC(F)(F)C2)C1 60559,C1(CC(=O)NCC2OCC(=O)NC2)C2CCCC2N1C(c1ccco1)=O 60560,c1(-c2cccc(SC)c2)ncc(F)c(C(=O)Nc2cc(C(F)(F)F)cc(Br)c2)n1 60561,Cc1ccc2[nH]c(C)c(CC(N3CCC(NCCO)CC3C)=O)c2c1 60562,N1(C(c2ccc(CCC)s2)=O)CCC(C)(CNC(=O)CC2COCC2O)C1 60563,c1(C(=O)NC2CN(C(C(CC=C)C(C)C)=O)C2)[nH]c2c(F)cc(F)cc2c1C 60564,CCC(C)C(O)C(C)C(=O)N1CCOC(C(N2CCC3(CCCCC3)C2)=O)CC1 60565,C1(N(C(CCN(CCC)C)=O)CC)CN(C(c2snc(C)c2N)=O)CC1O 60566,C1(C(=O)NCCCOCCNC(C(n2ccc(C)n2)C)=O)CCC(=O)N(CO)C1 60567,C1(NC(C(C=C)CC)=O)CN(C(=O)CCC(C)OCC)CC1C1CC1 60568,Cc1c(C(=O)NCC2CCCCC2NC(=O)COc2cnn(C)c2)cccc1O 60569,c1(CC(=O)NCCOCCn2cc(-c3ccc(C(F)(F)F)s3)nn2)cncnc1 60570,N1(C(C2CCC(OC)CC2)=O)CCN(C(c2ncn3c2CCC3)=O)C2CCCC12 60571,N1(C(C2CC(OC)C2)=O)CCOCC(CNC(=O)COC2CCC(F)(F)CC2)C1 60572,N1(C(C(C)OCC)=O)CCC2CN(C(=O)C(O)C(C)c3ccccc3)CC2CC1 60573,c1(NCCC)ccc(C(=O)NCC(C)NC(=O)C(=O)N(C)C)cc1[N+](=O)[O-] 60574,C(C(O)CN=c1[nH]nco1)NC(N)=O.CCCCC1C(=O)N1 60575,C=CCC(C)(C)CNC(=O)CCCCN(C(=O)CC1CCCC(C)O1)C 60576,N1(C(C2CN(C(C)=O)C2)=O)CC(NC(c2cc([N+](=O)[O-])c[nH]2)=O)C2(CCCC2)C1 60577,C(c1ccc(Cl)cc1F)=CC(=O)N(CCOCCN(C(C1CC(C)OC1)=O)C)C 60578,N1(C(CC2(C)CCCC2)=O)CC(CNC(c2cccc(F)c2Cl)=O)CC12CCC2 60579,N1(C(c2ncn(CC)n2)=O)CCCC1C=CC(=O)NC(C1CC1)C1CC1 60580,c1(C(=O)NC2C(NC(CC3CCC(C)(C)C3)=O)CC2)ccc2nc(O)[nH]c2n1 60581,c1(C(=O)NCCC2COCCN2C(=O)CCOCC2CC2)nccc2n[nH]cc12 60582,c1(CC(=O)NCCC2CC(NC(c3cnc(OC)s3)=O)C2)cc(C)ccc1OC 60583,N1(C(C(CCC)C)=O)CC2(C1)CN(C(C1CCC(F)(F)C1)=O)CC2C(=O)O 60584,C1(NC(CCNC(=O)NC)=O)CCC(O)CN(C(c2cn(C)c(O)n2)=O)C1 60585,N1(C(CC2CC(=C)C2)=O)CCN(C(c2ccc(N)cc2OCC)=O)CC(C)(C)C1 60586,Cc1nc(O)c2c(n1)CCN(C(c1ccsc1S(C)(=O)=O)=O)C2 60587,N1(C(C(N2CCCCC2)C)=O)CCOC(C(C)(C)CNC(=O)CP(C)(C)=O)C1 60588,C(=O)(C(=O)N=S(C)(C)=O)NC1C(C)CN(C(c2ccc([N+](=O)[O-])s2)=O)CC1 60589,C1(O)(C(N(CCC)C)=O)CCN(C(c2nnc(C)s2)=O)CC1 60590,c1(C(N2C(CCCNC(CSC)=O)CCC2)=O)ccc(F)cc1N 60591,CN1CC=C(CC(=O)NC2CCCC2NC(C2CC23CCCCC3)=O)CC1 60592,c1(C(=O)NC2CC(NC(=O)COc3ccsn3)C2)cn2c(Br)cccc2n1 60593,N1(C(C2C(NC(c3c(OC)ccc(Cl)c3)=O)CCC2)=O)CCCCC1C#N 60594,C1(CCC)CCCN(C(C2(C(C)C)CCN(Cc3cc(C)c[nH]3)C2)=O)CC1 60595,C(N=c1nc(C)[nH]s1)C1(C)CCN(C(c2c(CC)ccs2)=O)C1 60596,N1(C(c2ccc(Cl)cc2)=O)CCC(C(=O)NCC2(CC3(O)CC3)CC2)C12CC2 60597,c1(C(=O)NC(CC)CNC(=O)CC2CCC(=O)O2)ccc(C)c(C(C)(C)C)c1 60598,c1(C(C)=O)cc(C(=O)NCCCN(C)C(c2cn[nH]c2)=O)ccc1C 60599,N1(C(c2n[nH]c(CC)c2C)=O)CC(C)N(C(c2cccs2)=O)CC1C 60600,C1(C(=O)NCC23OCC(CNC(CCNS(C)(=O)=O)=O)(C2)C3)CC(S(C)(=O)=O)C1 60601,C1(NC(c2cc(C3CC3)oc2C2CC2)=O)CCC(NC(C2CCCSC2)=O)CC1 60602,c1(CC)c(C(N2CCCC(N(C(=O)CN(C)C(C)=O)C)C2)=O)oc2ccccc12 60603,c1(C(=O)NCC2(O)CCCN(C(C3C(C=C)C3)=O)C2)cc2ccccn2c1 60604,c1(CC)[nH]nc(C(N2CCCC2CCC2CCCCN2C(=O)CSC)=O)c1C 60605,C(CN=c1[nH]c(=NCc2nnc(C)o2)c2c(F)cccc2[nH]1)C1C(C)C1 60606,C1(CC)CN(C(c2cc(C)c(C)s2)=O)CC1C(=O)NC(c1ccco1)CO 60607,CC(CC(F)F)C(=O)N1CC(C(C)NC(=O)CC2CC2)(Cc2ccccc2)C1 60608,N1(C(C2C(C=C)C2)=O)C(CNC(=O)Cc2ccc(OC)c(F)c2)CC2CCCC12 60609,CON1CCC(C(=O)NC(C(C)NC(c2ccc(N(C)C)cc2)=O)C(C)C)CC1 60610,Cc1ccnc(O)c1C(N1CCN(C2CN(C(c3c[nH]c(=N)s3)=O)C2)CC1)=O 60611,C1(NC(C2(C)CCN(C)C2)=O)CN(C(c2cn3c(n2)SCC3)=O)C(C)(C)C1 60612,n1(C(C)C(=O)NC2CCSC23CN(C(c2ccsc2)=O)C3)cnc2ccccc12 60613,C1(CNc2cc(NC(c3nc(C(F)(F)F)n[nH]3)C)ncn2)CC2CCC1CC2 60614,C1(CNC(CCC=C=C)=O)CN(C(c2cnc(C)[nH]c2=N)=O)C2(CCC2)C1 60615,Cc1nn(CC(N2CCC(NC(C3C=CCC3)=O)C(C)C2)=O)c2ncccc12 60616,c1(C(=O)NC2(C)CC(NC(C=CSC)=O)C2)coc2c(F)cc(F)cc12 60617,c1(C(=O)NCC2(C)CCCN2C(C2C3CCC23)=O)ccc(F)c2cccnc12 60618,c1(CNC(C2(CC#C)CCCCC2)=O)cnn2c1CN(CC#CC)CC2 60619,C1(CNC(CN(C(c2c(CC)n[nH]c2)=O)C(C)C)=O)CCCC(C)O1 60620,n1(CCC(=O)NC(CC)CN(C)C(C2CC2C(N)=O)=O)ncc2c1CCCC2 60621,N1(C(CCNC(COC)=O)=O)CCN(C)CC1CNC(c1scnc1C)=O 60622,Cc1ccc(F)cc1C1(C(=O)NCC23CC2CN(C(C2CCCSC2)=O)C3)CC1 60623,C1(C(=O)NC2(CCC)CCC2)CCN(C(C2C3CCC(C3)C2C)=O)C12CC2 60624,C(=O)(C(C#N)C(C)(C)C)NCCOCC(=O)NCC(CC(C)(C)O)=O 60625,CS(=O)CCC(O)C(=O)NCCCNC(c1cc(O)cc(Cl)c1Cl)=O 60626,N1(C(CCC(C)(C)OC)=O)CCC2CCCC12CNC(C1(C)CC(F)(F)C1)=O 60627,C1(C(N2CCN(C(CN(C(C3CC(OC)C3)=O)C)=O)CC2)=O)CC(F)C(=O)N1C 60628,Cc1cnc(C)c(C(=O)NC2(C)CCN(C(=O)CCC3CCCN(C)C3)C2)c1 60629,c1(CC(=O)NC(C2CCN(C(C(CCC)(C)C)=O)C2)(C)C)cn2cc(C)sc2n1 60630,N1(CCC(N2CCC(NS(CCC)(=O)=O)C2)=O)CCN(C)CC1.C1CO1 60631,C(=O)(CN=S(C)(C)=O)N(C1CCCN(C(=O)Cc2coc(C)n2)CC1)CC 60632,CCC(COC)C(=O)N1CC(OCCC(=O)NC(C)CCOC)C1 60633,c1(OC)ccc(S(=O)(=O)N2Cc3ccc(C(=O)N=c4cnc(I)c[nH]4)cc3C2)cc1 60634,N1(CC(c2ccc(OC)c(C#N)c2)=O)CC(C(C)(C)C)Cc2cc(OC)ccc21 60635,c1(C(N2CCCC(CNC(C3CCC4CC34)=O)C2)=O)cc(Cl)cc2c1CCC2 60636,N1(C(Cc2ccn(C)n2)=O)CCC(C)(CC(=O)Nc2cnc(F)nc2)C1 60637,c1(C(=O)NC2C(C)CN(C(=O)C#CC3CC3)C2)cc(=NS(C)(=O)=O)cc[nH]1 60638,Cc1nc(C2CCC2)ccc1-c1nc(C2CC2)nn1CC(C)C 60639,N1(C(c2c(SC)cnn2C)=O)CCCCC(CNC(c2cncn(C)c2=O)=O)C1 60640,N1(C(C2ON=C(C)C2)=O)CCC(C)C1CNC(c1ccnn1C(C)C)=O 60641,c1(C(=O)NCC(C)(C2CCC2)NC(C(CC#C)O)=O)cc([N+](=O)[O-])n[nH]1 60642,C1(NC(C2CCCN(C(C)C)C2)=O)CCN(C(C2(CCF)CC2)=O)C12CCCC2 60643,N1(C(CCC)=O)CC(NC(c2cc(F)cc3nccnc23)=O)C2CCCCC12 60644,C12(CNC(CN(C)CCO)=O)CCCC1CN(C(C13CCC(CC1)CC3)=O)C2 60645,N1(C(c2cc(C)c(C)[nH]2)=O)CCC(CNC(c2coc(Br)c2)=O)C12CC2 60646,Cc1nnc(C(=O)N(CC(O)CN(C(=O)C(C)C)C)C)s1 60647,C1(OC)(CNC(=O)C(CC2CCC2)NC(C2(O)CCOC2)=O)CCCC1 60648,C1(SC)CN(C(c2ccc(F)cn2)=O)CC1n1cc(CCCC(C)=O)nn1 60649,N1(C(C(C)NC=O)=O)CCC(C(F)(F)F)CC1C(=O)NCC1CCOC1 60650,c1(CC(c2cnccn2)=O)c(Cl)n[nH]c1-c1ccccc1 60651,CCC(CC(=O)NC1CCCCCC1C(=O)NC1CCCC1O)C(C)C 60652,C1(S(C)(=O)=O)(C(=O)NC2CCN(C(C3CC(SC)C3)=O)C2C2CC2)CCOCC1 60653,c1(C(CNC(=O)CCCCN(C)C)NC(CCOC)=O)ccc(F)cc1 60654,C12(C(=O)NC(CCC)CCCNC(=O)C=CSC)CC1COC21CCC1 60655,C1(C)(C(N2C(CNC(CC3ON=C(C)C3)=O)CCC2)=O)CS(=O)(=O)C1 60656,N1(C(c2cncc(CC)c2)=O)CC(CO)C2(C1)CN(C(c1coc(Cl)n1)=O)C2 60657,O=C(C1=CCSC1)NCC1CCN1C(=O)C(c1ccc(Cl)cc1)CO 60658,C1(CC=C)(NC(c2nnc(C)s2)=O)CCN(C(c2cccc(OC)c2F)=O)CC1 60659,n1(C(C)C)cnc2c(NCC3CC4C=CC3O4)[nH]c(=NC3CC(C)(CO)C3)nc12 60660,C1(C2(O)CCCOC2)(CNCc2cc(C)c(F)c(C)c2)CC1 60661,C(=O)(C(CC1CCC1)N(C)C)NC1CC(CNC)C1.C1(NC(=O)CO)CCCOC1 60662,C1(C(=O)NC2CC23CC(NC(C2(CCO)CC2)=O)C3)CCCCCCC1 60663,CC1CCS(=N)(=O)CCN1C(=O)C(C(C)(C)C)n1cc(C2CCC2)nn1 60664,C(C)(CNC(c1ncccc1Cl)=O)(CC(C)C)NC(C(CC)OC)=O 60665,C1(C(=O)NCC2N(c3c(CC)c(Cl)ncn3)CCC2C)COC2COCC2O1 60666,N1(C(C2CC(CCC)C2)=O)CCC(C(=O)NC(C2CCOC2)CO)C1C 60667,N1(C(C(n2c(C)ccn2)C)=O)CC(F)(F)CC1C(=O)N(C)CC1COCCO1 60668,C1(CN(C(=O)CCc2ccnc(Cl)c2)CC)CCN(C(=O)C(C)C2CCC2)CC1 60669,c1(SCC(=O)NC2C(CNC(C3(CCC)CC3)=O)C2)ccccc1F 60670,N1(CC(C)C(C)N2CCOCC2)CC(=O)N(Cc2ncccc2C(F)F)C1=O 60671,C1(C(N2CCN(C(CC)=O)CC2C)=O)CN2CCCN1CC2 60672,N1(C(C=CSC)=O)CC(NC(c2ccc(F)c(F)c2N)=O)C(C2CC2)C1 60673,N1(C(c2ccn(CC)n2)=O)CCCC(N(C)C(c2cc(CO)[nH]n2)=O)CC1 60674,n1(CC(F)F)nnnc1C(c1ccc(Br)s1)NCC(C)(C)SCl 60675,CC(CCC(C)(C)C)NC(C1CCCC1CNC(c1cc(F)cnc1O)=O)=O 60676,c1(C(=O)NC2CN(C(c3cccc(OC)c3)=O)C2)ccc(C#N)cc1F 60677,c1(N(CCOCC=C)C)nc(=NC(C)c2ccc(F)c(C)c2)[nH]c2c1CSC2 60678,C1(C(=O)NC23C(CN(C(C(C)(C)OC(C)C)=O)C2)C3)CCOC(=O)CC1 60679,O=S1CCC(N=c2ccnc(N3CCC4(CCOC4)C3)[nH]2)CC1 60680,c1(C(N(C)CC2CN(C(=O)CC(C)(O)C3CC3)CCO2)=O)cc(O)nc(O)n1 60681,C1(CCCNC(c2ocnc2C2CC2)=O)CCCCN1C(C1CCOC1)=O 60682,Cc1ccc(C=CC(=O)NCCC(C)CCNC(c2occ3c2CCC3)=O)cn1 60683,N1(C(C2C(C#N)C2)=O)CCCC2(NC(=O)Cc3cnn4c3CCCC4)CC2C1 60684,Cc1ccc(C2CCN2C(=O)NC(C(N)=O)C(N)=O)cc1 60685,c1(C(=O)NCCN(C(=O)CCC(C)OCC)CCC)c[nH]c2c(CC)cccc12 60686,c1(OCCC(=O)NC2CCC(CCNC(C=NOC)=O)C2)ccc(OC)cc1 60687,CC1(C)CC=C(C(=O)NC2CN(CC(=O)N3CCCC3)NC(=O)C2)CC1 60688,N1(CC(=O)NCC(CCCC)NC(=O)Cc2occc2C)C(=O)CN(C)C1=O 60689,CCCCCCN(C(=O)Cn1cccn1)CCN(C(C1CCCC1C)=O)CC 60690,Cc1cc(NC(c2ccc(S(C)(=O)=O)o2)c2nnnn2C(C)(C)C)cc(C)c1F 60691,c1(C(C)C)sc(Cl)nc1C(=O)NCC(C1CCCCC1)NC(=O)CC(C)F 60692,C1(C(N2C(CNC(CCNS(C)(=O)=O)=O)CCCC2)=O)CC12CCSCC2 60693,c1(C(=O)NC2CC3CC(NC(C(F)=CCC)=O)C3C2)c[nH]c2ccc(Cl)cc12 60694,c1(C(N2C(CO)CC(NC(CC3C(C)(C)C(O)C3)=O)C2)=O)cc(Cl)ccc1Cl 60695,c1(C(=O)NCC2CCN2C(c2cnco2)=O)cnn(CC2CCCCO2)c1 60696,C(CCC(=O)NC1(C(=O)NCC(c2cccs2)C)CCC1)NC(C)=O 60697,C(=O)(C#CC1(C)CC1)N1C(C(C)NC(c2cn(C)nc2O)=O)CCC1 60698,CCCCCC(C)CC(=O)N1CCC(C)C(CNC(c2sccc2C(C)C)=O)C1 60699,Cc1cc(C(N2CCCCC2C2(NC(=O)CCc3ccccn3)CC2)=O)sc1C 60700,c1(CC(=O)NC2(CNC(CC(C)C3CC3)=O)CC2)ccc(Br)cn1 60701,c1(C(C(N2CC(OC)C(NC(C3(F)CCOC3)=O)C2)=O)(F)F)ccc(F)c(F)c1 60702,c1(C(N2CC(NC(=O)CC(C)F)CC(C)C2)=O)ccc2nc3n(c2c1)CCC3 60703,c1(CNC(c2n(CC)nc(C)c2)=O)ccc(CNC(=O)C(C)NC(C)=O)cc1F 60704,CC1=C(C)CC(C(N2CC(O)(C(F)C(N3CCCC(C)C3C(N)=O)=O)C2)=O)CC1 60705,C1(CC(N2CCC(C(C(=O)N(CCC(=O)NC)C)F)C2)=O)CCC(=O)N1C 60706,C1(C)(C(N2C(C)(C(=O)O)C=CC2)=O)CC(O)c2ccccc2O1 60707,CCC(F)(F)CC(=O)N1CCCC(C2CCCCN2C(C23CSCC2C3)=O)C1 60708,C1(NC(c2ncn(CC)c2)=O)CCCC2CN(C(c3c(Cl)cccc3Cl)=O)CC12 60709,N1(C(c2cccc(C)c2)=O)CCC(NC(=O)CC2(CO)CC2)C(F)C1 60710,CC1(C)C(CC(N2CCOC3CC23)=O)CCN1C(c1ccoc1)=O 60711,C1(CC)CN(C(c2cnc(Cl)cc2I)=O)CCN1Cc1ccnc(OC)c1F 60712,c1(C(N(C)CC2CCCN(C(C3CCC3(F)F)=O)C2)=O)cc2nc[nH]c2cc1F 60713,CC1(C(=O)NC2CC3CC2CN3C(=O)CNC(N)=O)CC2CCC1CC21OCCO1 60714,N1(C(CCc2nc(C)sc2)=O)CCc2c(CNC(=O)C=CC(C)C)cccc2C1 60715,c1(C(C)(F)F)cccc(C(=O)NC2CC2NC(=O)CC2C=CS(=O)(=O)C2)c1 60716,c1(OC)cc(CCC(N2CC(O)(CCNC(C3(Cl)CC3)=O)C2)=O)ccc1F 60717,N1(C(C(C)Sc2cccc(F)c2)=O)CCN(C(c2cccc[n+]2[O-])=O)C2(CC2)C1 60718,c1(CC(=O)NC2CCN(C(C=C(C)C3CC3)=O)C2C)cc(C(F)(F)F)c(O)nn1 60719,CN1CCC(C)(C(=O)N(C)CC2CCN(C(C3(CCF)CCC3)=O)C2)CC1 60720,N1(Cc2nnc(OCC)s2)CCC(C)C(NC(c2cnn(C)c2C)=O)C1C 60721,N1(C(=O)C=C2CC2)CCOC2(C1)CN(C(=O)Cc1ccc(Cl)cc1O)C2 60722,Cn1cc2c(n1)CCCC2C(=O)N1CCCCC1CNC(=O)CC#N 60723,C(N=c1[nH]c2c(c(=NC(C)c3cnc[nH]3)[nH]1)CCC2)C1(C(=O)NC)CCOCC1 60724,C1(CN(C)C(c2ccnc(C3CC3)c2)=O)CCCCN1C(c1cccn1C)=O 60725,C1(NC(C(C)Cc2ccccn2)=O)CC2CC1N(C(=O)Cc1csnn1)C2 60726,N1(C(c2c(C)ncnc2)=O)CC2CCCCC2(NC(=O)CC(C)CC(C)C)C1 60727,CCCC(C(=O)NC1(CCNC(c2nc(Br)c(C)s2)=O)CCC1)N(C)C 60728,c1(C(C)Cc2nc(-c3cccc(F)n3)no2)ccc(S(C)(=O)=O)cc1 60729,C(C1c2ccccc2CN1C(C1C2(CC2)C12CC2)=O)NC(C(C)OCCCC)=O 60730,N(C1CCCn2ncnc21)C(C(C)N(C(=O)CC(C)C(F)(F)F)CCC)=O 60731,Cc1nc(C(=O)NC2CC(NC(C3CCCN3C3CCCCC3)=O)C2)cc(O)n1 60732,C=CCCCC(C(=O)N1CC(=CC)C1)NC(C1C2CCCCC12)=O 60733,C1(NC(c2cc[n+]([O-])cc2)=O)CCCC12CN(c1nc(Cl)ncc1Br)C2 60734,C1(C)(CNC(c2cc(Br)ccn2)c2n(CCCSCC)nnn2)C=CCCC1 60735,N1(C(C(=O)NCC)=O)CCC2(CCN(C(c3cccnc3NCC)=O)C2)C1 60736,c1(C(=O)Nc2ncc(Br)cc2I)cc2c(s1)CCN(Cc1cc(Cl)cc(I)c1)C2 60737,CON1CCC(C(=O)NCc2scc(C(=O)NC3CC(C)N(C4CC4)C3)c2)CC1 60738,C1(N(C(C(C)=C2CC2)=O)C)CC2CCC(C1)N2C(=O)COc1ccsn1 60739,C1(CC(C)NC(=O)Cc2cncs2)CCN(C(=O)Cc2ccc(N)cn2)CC1 60740,CC(C)(C)C(=O)C(=O)N1CCCOC(CNC(=O)CC2CCNC(=O)C2)C1 60741,c1(C(N2CC3(Cn4cccn4)CCCC23)=O)cnn2c1CCCC2 60742,c1(C(=O)NCC=CC(=O)NCC(C(=O)OCC)C)ccccc1NC 60743,c1(OC)cccc(COC(c2c[nH]nc2I)=O)c1CC1CCCO1 60744,c1(CC(N2CC3C(C(N4CCC(CC)C4)=O)(C3)C2)=O)cccc(C#N)c1 60745,N1(C(c2c(NC)cncc2)=O)CCCCC(NC(=O)C(C)(C)C(C)O)C1 60746,N1(C(C2CCC(OCC)CC2)=O)CCCN(C(c2cnn[nH]2)=O)CCC1 60747,CC(C)CCCC(=O)NCCNC(c1scnc1C(C)C)=O 60748,C1(CN(CCC)CCNC(C2CC3CCC2C3)=O)CCC(F)(F)C1 60749,N(C(=NCCCF)N1CCC2C(C1)NC(=O)N2C)C(c1c(C)nn(C)c1)C 60750,C1(COC)(NC(c2cscc2C)=O)CN(C(=O)C(N2CCSCC2)C)C1 60751,c1(C(C)C)ccc(C(CNC(=O)CSC2CCOC2=O)NC(=O)C(N)=O)cc1 60752,CC1CN(C(C2CC(C)(F)C2)=O)CCC1NC(c1cc(N(C)C)cs1)=O 60753,C=C(C)CC(C)C(=O)NCC(C)(C)NC(c1ccsc1C)=O 60754,c1(CC)ccc(C(=O)N(C2CN(C(=O)CC3CC(SC)C3)CC2(C)C)C)c(O)c1 60755,N1(CC(=O)NC(CNC(c2cc(O)ccc2F)=O)CO)Cc2ccccc2C1 60756,N1(C(Cc2ccc(C)cc2)=O)CCC(O)C(NC(=O)C(O)C2CC2)C1 60757,N1(CC)CC2CCC(NC(=O)CCc3cc[nH]n3)(C2)C1.c12ccc(o1)CNC2=O 60758,N1(C(CC2CN(C(C)=O)C2)=O)CC2CC(NC(=O)CC3CCC3)CC(C2)C1 60759,Cc1nn(CCN(C)C)c(C)c1S(=O)(=O)N1CCCCC12CCN(C)C2 60760,C1(C2(NC(c3cnnc(O)c3)=O)CC2)CCCCN1C(=O)Cc1c[nH]nc1O 60761,c1(C(=O)Nc2cc(C)c(C(=O)NCCC(CO)C(C)C)s2)ncc(C)cc1F 60762,CC1C(NC(c2c[nH]cc(F)c2=O)=O)CCCN1C(c1ccccc1O)=O 60763,C1(CCC)(NC(=O)CS(=O)CC)CCCN(C(=O)C2=CCCCC2)C1 60764,c1(C(N2CCC(O)(C(=O)NCC3(F)COC3)C2)=O)cn2cc(F)ccc2n1 60765,C(=O)(CCCS(N)(=O)=O)NC1(CO)CCCN(C(C(CCCOC)C)=O)C1 60766,N1(C(CS(CC)(=O)=O)=O)CCC2C1CCCN2C(=O)C(O)C(C)CC 60767,C(=O)(CC1OCCc2ccccc21)N1C2CC(NC(C3CC3F)=O)CC1CCC2 60768,C1(CC(=O)NC(CC)CN(C)C(C2(CCOC)CC2)=O)SC(=N)NC1=O 60769,c1(C(=O)NCC(C)(CO)NC(C2CC(C)C2)=O)ccc2cccc([N+](=O)[O-])c2n1 60770,c1(NC(C2CC2C(=O)Nc2cccc(F)c2Br)=O)ccc2ccccc2c1Cl 60771,CC(C(O)CC(=O)OCCC=Cc1ccc(Br)cc1)Sc1ccccc1 60772,c1(C(=O)NC2(CO)CCN(C(CCC(=O)NCC)=O)C2)cnn2c1NCCC2 60773,N1(C(c2cc(C)[nH]n2)=O)CC2CS(=O)(=O)CC2(CNC(=O)CCC(C)(C)C#N)C1 60774,C1(NC(C=CC(=O)NC2CC2)=O)CN(C(c2sccc2F)=O)C2(CCCOC2)C1 60775,N1(C(CC2C(C)=NNC2=O)=O)CC(CNC(c2[nH]cnc2C#N)=O)C(C)(C)C1 60776,N1(C(CC2ON=C(CC)C2)=O)CCC(C(=O)NC(CC(=O)NC)C2CC2)C(C)C1 60777,c1(C(C2CCC(C)C2)C)cnccc1SC(C)(C)C.C12(O)CN(C1)C(=O)NC2 60778,C(C(COC)C(=O)N1CCCC1CCC1CCCCN1C(=O)C1CC1)OC 60779,CC1CCCc2cc(C(=O)NC3(CNC(=O)COCCCF)CCOC3)nn21 60780,CC1(C2CCN(C(=O)CCC3CCCCN(C(=O)C4=NOCC4)C3)C2)CC1 60781,c1(NC2C(OC)C(C)(C)C2)nc2cccnc2c(=NCc2ccncn2)[nH]1 60782,S(=O)(=O)(c1cc(Cl)c(Cl)cc1Cl)NC(C1C(C(C)C)(CC)C1)=O 60783,c1(C(=O)NC2CC(C)(NC(C3C(C)OC(=O)N3)=O)C2)cnc(S(C)(=O)=O)s1 60784,c1(C(=O)NC(C2CCCCN2C(c2cnnc(Cl)c2)=O)C)nc(=O)n(C)[nH]1 60785,C123CCC(CC1)N(C2)c1nc(cc(C)n1)NC3=O.C1(CC)(CN(CC)CC)CC1 60786,C1(C(N2C(C(=O)Nc3c(C)[nH]nc3Cl)CCCC2)=O)CCc2ccccc2O1 60787,C1(NC(C(COC(C)C)NC(C=C(CCC)C)=O)=O)CC2CC1CC21CC1 60788,c1(C(=O)NC2CCN(C(c3c(C)csc3)=O)CC2C)cnn2c1CC(F)(F)C2 60789,c1(C(N(CCC)CCNC(=O)C(C2CCOCC2)F)=O)ccc(C)cc1O 60790,C(N=c1[nH]c2cnccc2s1)c1ccc(CNC(=O)Cn2cncn2)cc1 60791,C(=O)(CC(C)C(C)C)NCC1(CNC(C2N(CC)CCC2)=O)CCC1 60792,N1(C(CC2N(C(CCCC3C(C)C3)=O)CC(O)C2)=O)CCC(F)(C#N)C1 60793,c1(C(=O)NCC(CC2CN(C(C(C)c3cc[nH]n3)=O)C2)(C)C)cccc(=O)n1C 60794,C(CC(C)(C)CC(=O)NC(C1(O)CN(C(=O)CC(C)c2cccnc2)C1)C)OC 60795,C1(C(=O)NCC2C(NC(c3c(Cl)ccc(OC)n3)=O)C2)(OC)CCCCCCC1 60796,N1(C(CC(CNC(C(CCCC#C)C)=O)C)=O)CCC2CCCC2CC1 60797,C1(SC)CN(C(=O)CC2CCC(=O)N2C)CC1NC(C1CC=CC(O)C1)=O 60798,C=C(C)CC(C(=O)NCC1(C)CCCS1)NC(=O)CCOCCOC 60799,c1(CN2C(C(N3CCCC(C)(O)C3)=O)CC2)n[nH]c2ccc(F)cc12 60800,CCC(C)(C(=O)NCC(CNC(C1(Cc2cccc(Cl)c2)CC1)=O)CO)OC 60801,N1(C(c2ccn(CCNC(C3C(=C)C3)=O)c2)=O)CCN(C)C(=O)C1CC 60802,CC1CN(C(=O)C(F)(F)Cl)CC1C(N1CCC(Cc2ccc(F)cc2)C1)=O 60803,c12ccc([N+](=O)[O-])cc1C(=O)N1CC(C(C)(C)O)(C1)CNC(=O)C2.CCSC 60804,Cc1cc(C(N2CC3CC(C2)N3C(C2CCOCC2)=O)=O)ccc1C#N 60805,C(CC1CCCC1)(C(=O)N(C)CCn1cncn1)NC(C(c1cnn(C)c1)C)=O 60806,c1(C(N2CCC(NC(CNC(CNC(C)=O)=O)=O)(CF)C2)=O)cc(O)ccc1C 60807,c1(CC)nc2n(n1)CC(NC(=NCCCF)NCC1(CSC)CCN(C)CC1)CC2 60808,c1(CC)cc(C(=O)N(CC(C)N(C(=O)C=Cc2nc(C)co2)C)C)ccc1OC 60809,CC1CCN(C(=O)CCNC(=O)CO)CC1CNC(c1cc(F)cc(F)c1)=O 60810,CC(C)C(O)C(=O)NCC(C)(C)CNC(c1cn(C)cn1)=O 60811,c1(CC)n[nH]c(=NC2CCN(C(c3cnn(-c4ccncc4)c3)=O)C(C)C2)s1 60812,N1(C(C2CN(CC)C2)=O)CCN(c2cc(NC(=O)OCC(=C)Cl)ncn2)CC1 60813,C=CCCCC(C(=O)NCc1cc(Br)c(F)cc1OC)OC 60814,c1(CCCC(=O)N(C)CC2(NC(c3cnn(CC)n3)=O)CC2)ccccc1OC 60815,C1(C(=O)NCC2CC(C(=O)NCCC(O)C3CC3)C2)CCCN1C=O 60816,Cn1nnc2cc(C(N3CC4CCC4(NC(c4csc([N+](=O)[O-])c4)=O)C3)=O)sc12 60817,C1(C(=O)NC(CN(C(c2cnc(O)n2CC)=O)CC)C)CCCCC1(C)C 60818,C(C1c2ccsc2CCN1C(C1CCC1)=O)NC(C(C)NC(=O)C(C)(C)C)=O 60819,Cc1cc(C(N2CCCCC2CS(C)(=O)=O)=O)ccc1Br 60820,S(=O)(=O)(c1cc(C)cnc1Cl)N1CCC(N(C)Cc2cccc(SC)c2)C1 60821,C(=O)(C(=O)CCC(C)C)NCCCC(CCC)NC(c1cc2c([nH]1)CCC2)=O 60822,C#Cc1ccnc(C(=O)NCC2C(CNC(=O)CC(CN(C)C)CC)C2(F)F)c1 60823,Cc1cc(C(N2CCC(F)(CNC(c3ccc4c(c3)CC4)=O)C2)=O)ccc1C#N 60824,c1(OC)cccc(-c2cn(CC3C(CNC(=O)C(C)(C)OC)C3(F)F)nn2)c1F 60825,c1(-c2onc(CN3CCC(O)(CO)C3)n2)cc2ccccc2c(O)n1 60826,C=CC1(C(=O)NCCCN2CC=CC2)CCN(C(=O)C(C2CCCCC2)C)CC1 60827,c1(C(=O)NC(CNC(c2c(NCC)scn2)=O)C2CC2)cnc2c(c1)CCCO2 60828,c1(C(C)=O)cnn(C)c1C(=O)N(C)CCNC(=O)C(N1CCNC1=O)C 60829,c1(OC)c(C)csc1C(=O)NCC(CNC(c1cc(-c2ccoc2)[nH]n1)=O)OC 60830,c1(-c2cc(OC)c(C#N)cc2)cnc2[nH]cc(C(=O)NC(C)CF)c2c1 60831,c1(C(=O)NC(C)Cc2ccc(CNC(C3CC3C)=O)cc2)ccc(N)cc1F 60832,C1(CNC(C(n2cc(Cl)cn2)C)=O)CC2(CCC2)CN1C(C1CCCC12CC2)=O 60833,Cc1ccc(O)c(NC(c2nn(C)nc2Br)=O)c1 60834,CC1CN(C(=O)CNC(N)=O)CC1NC(c1cncc(C(C)(F)F)c1)=O 60835,CC(c1ccsc1)=CC(=O)NC1(C2CCCCN2C(c2ccc(O)cn2)=O)CC1 60836,C(c1ccc(Br)cc1)=CCC(=O)NCCCCNC(C1CCC(F)C1)=O 60837,c1(C(=O)NC2(CCNC(=O)Cn3cc(Cl)cn3)CC2)cc(O)nc(O)n1 60838,Cc1cc(C(=O)NC2CCC2NC(c2[nH]nnc2C)=O)cc(C)c1Cl 60839,C1(C(=O)Nc2c(COC)ncs2)CC(=O)N(C2CN(Cc3cnc(C)s3)C2)C1 60840,C1(CNC(C(CC=C)C)=O)COCCN(C(c2ccncc2OCC)=O)C1 60841,C1(CNC(C2C(COC)C2)=O)CCCN1C(C1CCCN1C)=O 60842,C1(C(=O)NC(C2CCOC2)CC)(CNC(c2ccns2)=O)CCCC1 60843,c1(C(N2CCC(F)(CNC(C(C)CC3CCC3)=O)C2)=O)ccc2c(n1)COCC2 60844,c1(NC(C)=O)cnccc1C(=O)N(CCNC(C1CC1(C)C(C)C)=O)C1CC1 60845,C#Cc1ccc(CC(=O)NCC=CC(=O)NCC(C)C)cc1 60846,c1(C(N2CCC(O)(CCNC(CSSC)=O)CC2)=O)ncnc2c(C)csc12 60847,Cc1nn(C)c(N)c1C(=O)NCC(C)=CC(=O)NCc1cnccc1Cl 60848,c1(NC(C2N(C(CSCC)=O)CC=C2)=O)cccc(-n2cccn2)n1 60849,C1(C(=O)NC(CC=C)CO)CC2(CCN1C(C1CCCC(C#N)C1)=O)CC2 60850,C(c1cccc(Cl)c1)=CC(=O)N(C1CCN(C(c2c(C)coc2)=O)C1)CCO 60851,C1(CC(=O)NCCNC(C(C)c2ccsn2)=O)CCN(CCF)CC1 60852,C1(C(=O)NCCOCCN(C(C(C(C)C)O)=O)C)CN2CCN1C(C)C2 60853,C(N=c1[nH]cc(-c2ccc(Br)nc2)s1)c1cn(-c2cnc(CC3CC3)[nH]2)nn1.C1CC1 60854,N1(C(COc2cccc(C)c2F)=O)CCC2(NC(=O)COC3COC3)CCCCC12 60855,Cc1nc(Cl)[nH]c(=NCC2C3CN(C(=O)CCCc4cc(Cl)sc4Cl)CC23)c1F 60856,C(=O)(C(O)C(CCC)NC(=O)C(C#N)C(C)C)NCC1(C=C)CCC1 60857,C12(CNC(C(CC=C)(F)F)=O)CCC(CNC(C3CCCC(F)C3)=O)(CC1)CO2 60858,c1(CNC2CCC(C(=O)NCc3ccc(C=C)cc3)C2)cccn2ccnc12 60859,CC(CC(F)F)C(=O)N1CCCC(O)(CCNC(=O)CC2CCSCC2)C1 60860,C1(CS(=O)(=O)NCC(CCOC)O)CN2CCCCC2CO1 60861,C12(C(N(C(C)CNC(=O)Cc3ccnn3C)CC)=O)CC3CC(CC(C3)O1)C2 60862,N1(C(Cn2c(C)ccn2)=O)CC(C)CN(C(=O)C2=CSCCO2)C(C)C1 60863,[N-]=[N+]=NC1CC2(C(N3CC(O)(CCNC(C4(Cl)CC45CCC5)=O)C3)=O)CC12 60864,N1(C(CC(=O)NC(C)CS(C)=O)=O)CCC(C(=O)Nc2ccccn2)CC1 60865,C(=O)(C(C)(C)CC(C)C)NC1(CNC(C(C)SC)=O)CCC1 60866,C=Cc1ccc(C(=O)OCC)cc1.N12CC3CCC13C2 60867,C(=O)(C1CCCn2nccc21)NCC1CCC2(CN(C(C3CC(=O)NC3)=O)C2)O1 60868,O=CN1CCCC1C(N1CC(O)CC1CNC(=O)C(O)c1ccco1)=O 60869,Cc1nc(CC(N2CCC(CNC(=O)CCC3CSCCS3)C2)=O)cs1 60870,c1(OCC)ccc(S(=O)(=O)NC2CC(S(C)(=O)=O)C2)cc1-c1cccc(C)c1 60871,Cc1cnc(C)c(NC(C2CC(F)CN(C(=O)Cc3cccs3)C2)=O)n1 60872,C1(NC(c2cnc(C)o2)=O)CCN(C(C2CC23CCSCC3)=O)C1(C)C 60873,S(=O)(=O)(c1ccc(Br)cc1NCC(c1ncccn1)(C)C)N(CCCOC=C)C 60874,N1(C(C2OCC(C)(C)C2)=O)CC(NC(c2cc(N)nc(Cl)c2)=O)CC(C)(C)C1 60875,c1(OC)ccc(CNCC2(C(=O)Nc3ncoc3C)CC2)nc1Br 60876,C1(C(N(CC(C)NC(CC(C)n2ccnc2)=O)C)=O)CC2(C1)CC2F 60877,C=CC(C)(O)C(=O)NCCNC(C1C2COCC12)=O 60878,N1(C(c2nc(CCC)oc2)=O)CC2CC1C2CNC(C12CCCC1C2)=O 60879,CN1CC2CCN(C(=O)CCN(C(C3CCC(=O)N(C)C3)=O)CC3CC3)CC2C1 60880,CN1CCCC(C(N2CC(NC(c3ocnc3-c3ccccc3)=O)C(O)C2)=O)C1 60881,c1(CC(=O)N(C2CCCCN(C(c3cnc(O)o3)=O)C2)C)cn2ccsc2n1 60882,c1(C(=O)NC(CC=C)CNC(=O)C(O)CC(N)=O)cc2cc(Cl)sc2[nH]1 60883,C1(C(N(C2CCN(C(c3cnc(O)s3)=O)C2)C)=O)CCC2(CC1)CC2(F)F 60884,N1(C(COCCCC)=O)CC(C(N2CCCC(C(C)(C)C)C2)=O)CC1(C)C 60885,CCCCS(=O)(=O)NC(C)C(=O)N(CCCNC(=O)CC1(CO)CC1)C(C)C 60886,c1(C(N(C)Cc2ccccc2CNC(=O)CSC(F)(F)F)=O)cnc(Cl)cc1Cl 60887,c1(CC(=O)NCCCN(C(c2ccnnc2)=O)CC)cc(Br)cnc1OC 60888,CN1CCC2C1CCCN2CC1CC2(C1)OCCO2 60889,C1(CNC(CCNC(C)=O)=O)CC(C(=O)NCCN2CCCCC2)CO1 60890,c1(N2C(C)CCN(C(=O)CCC(=O)OC(C)(C)C)CC2)ncnc2ccccc12 60891,CCC(C(=O)NC1CC(CN(C(=O)C(C)N(C)C)C)C1)C(C)(C)CC 60892,C(CC(C(=O)NCC1(CC2CC2)CC1)NC(c1cc(CO)on1)=O)=CC 60893,O=C(C1=CCCOCC1)NC(CNC(C1(F)CC1c1ccccc1)=O)CO 60894,CC1CCC(CNC(=O)Cc2cncnc2O)CN1C(c1cc(=O)n(C)cn1)=O 60895,CCC(C)C(O)C(C)C(=O)N1CC2CCC1CN2C(=O)CN1C(=O)CNC1=O 60896,Cc1nc2cccc(C(=O)NCC(CO)NC(C3(C)CCN(C)C3=O)=O)c2[nH]1 60897,N1(C(C(C)(Cl)CCl)=O)CC2CC1CC2NC(c1cccs1)=O 60898,C(=O)(C(=O)N=S(C)(C)=O)NCCC1CN(C(=O)C=Cc2ccsc2)CC(C)O1 60899,c1(CN2C(CC(N3C4CCCC3COC4)=O)CCC2)cc(Br)cc(Cl)c1F 60900,C1(NC(c2n[nH]c(C3CC3)c2Br)=O)CCCCN(C(=O)CC2CCCC2)C1 60901,c1(OC)ccc(Br)c(C(N2CC3CN(C(=O)CC4OCCO4)CC3C2)=O)c1C 60902,N1(C(C(CC=C)(C)C)=O)CCCC2C1CCN2C(=O)CCCc1cccc(C)c1 60903,C1(NC(c2c(C)cns2)=O)CCS(=O)(=O)C12CN(C(=O)Cc1ccccc1N)C2 60904,CCC(CC(=O)NC1COCC1NC(c1ccnc(C2CC2)c1)=O)C(C)(C)C 60905,N1(C(C2(CC=C)CCCC2)=O)CCCC1(C)C(=O)OCC.C12CC(C1)NC(=O)C2 60906,c1(CCC(=O)N(C)CC2CN(C(C(COC)N(C)C)=O)C2)cccc(F)c1 60907,CCCCCC(O)CNC(c1ccc(OC(C)C)nc1)=O 60908,N1(C(C=C(CCC)C)=O)CC2CC(NC(=O)C=Cc3cccs3)CC(C2)C1 60909,C(C(=O)NNC(=O)C(F)(F)F)n1c(C(C)=O)c(C)cc1C 60910,Cc1nc(C)n(CC(=O)NC2COCCC2C(=O)NCC2CCOC2)n1 60911,N#Cc1ccc(C(F)(F)C(N2CCOCC2CC2CC2)=O)cc1 60912,C(=O)(C(C)(C)C(=O)NCC(C)NC(c1ccc(SC(F)(F)F)s1)=O)OCC 60913,c1(C(N2CC3N(C(CCCCCCC)=O)C(CC3)C2)=O)cncc2c1CCCC2 60914,N1(C(c2sccc2Br)=O)CC2(C1)CN(C(c1ccc(O)cc1F)=O)C2 60915,Cc1cc(CCC(=O)NCC(C)(C)CN(C)C(C2CCN(C)C2)=O)nn1C 60916,C(=O)(C(F)CC(C)(C)NC(=O)C(c1ccccc1)=O)N1C(C)(CC)CC1 60917,C(CC(C)(C)NC(c1cnoc1-c1cnn(C)c1)=O)N(C(=O)C=CC(F)(F)F)C 60918,C1(NC(c2n(C)nc(Br)c2)=O)CCN(Cc2cccc(C(F)(F)F)c2O)CC1F 60919,C1(NC(=O)COCCCF)CN(C(c2cnc3ncccn23)=O)C2(CCCC2)C1 60920,C(=O)(C(C)(C)C)NC(C)C(=O)N(C)CCNC(C1(CC2CC2)CCCO1)=O 60921,Cn1c(O)ncc(C(=O)NCC2CCC(NC(=O)CC3CC4CC4C3)CC2)c1=O 60922,c1(C(N2CCN(Cc3ccc(C)o3)C(CC3CC3)C2)=O)ccc(Br)cc1Br 60923,n1(C(C(C)O)C)cc(C2(O)CN(C(=O)C(c3ccccc3)F)C2)nn1 60924,C1(NC(CS(=O)(=O)NC)=O)CCN(C(=O)C(n2cc(Cl)cn2)C)CC1O 60925,c1(CC(=O)NCC(CNC(Cn2c(C)c(Cl)cn2)=O)C)cc(C(F)(F)F)cc(F)c1 60926,C1(NC(COCc2ncc(C)o2)=O)CCC(C)(CNC(=O)C(C)(C)N(C)C)C1 60927,c1(C(=O)NCCCC(C)NC(c2cn(CCC)nc2)=O)cccc2c1CCCC2 60928,N1(C(=O)Nc2ccccc2)CCN(CC(c2ccccc2)F)CC1 60929,C(=O)(C(C)(CC)OC)NCC(CN(C(c1n(C(CC)CC)ncc1)=O)C)O 60930,C1(C2CCN(C(=O)Cc3cc(Cl)ccc3Cl)CC2)(NC(C2CNC(=O)N2)=O)CC1 60931,C1(C(=O)NCCC2CCCCN2C(=O)COCCCF)CC2CC1CC2(F)F 60932,c12ccccc1CN2.N1(C(C)=O)CC(N(C(=O)Cc2cscn2)C)C(F)C1 60933,O=C(CC1COc2ccccc21)NC1CC(NC(=O)C(F)(F)c2cncs2)C1 60934,C(=O)(CC(CC)C(F)F)N1CCC(N(CC#C)C(c2csc(C3CC3)n2)=O)C1 60935,c1(C(N2CCC(N(C(C(C)OCC=C)=O)CCO)CC2)=O)ccc(F)cc1C 60936,N1(C(CCCC)=O)CC(OC)C(OC)C1CNC(=O)Cc1sccc1C 60937,C(=O)(C(O)C(F)(F)F)NCCSCC(=O)NC(c1ccccc1O)C 60938,CCC(CC(=O)N(CC(C)NC(C1(c2cc[nH]n2)CC1)=O)C)SC 60939,C1(C(N2CCC(COC)C2)=O)CCN(C(c2cc(C(C)C)no2)=O)CC1 60940,N1(C(CNC(=O)NC)=O)CCC(CO)C(NC(=O)CN2CCC(C)(C)C2)C1 60941,Cc1cc(=NC(C)C(c2ccccc2)NC(=O)C(C)(C)F)[nH]c(C)c1C#N 60942,c1(OC)cc(C(=O)NC2CC(NC(=O)CC(C)(C)SC)C(O)C2)cc(C)c1 60943,c1(NC(C2CCN(C(C3(OCC)CC3)=O)C2)=O)cc(C)ccc1C1CC1 60944,C1(CNC(CC2(C(C)(C)OC)CC2)=O)CC(NC(=O)C(=O)NC2CC2)CC1O 60945,C(CC(C)C)(C(=O)N1CCC(CNC(c2nnn(C(C)(C)C)n2)=O)C1(C)C)OC 60946,CC(C)CCCS(=O)(=O)NNC(=O)CC(O)Cc1ccccc1 60947,CC1(CC(=O)NCc2ocnc2C(=O)NCC(c2ccsc2)O)CCCCC1 60948,c1(C(=O)NCCCC2(NC(C(C)C3CCCC3)=O)CC2)csc(Br)n1 60949,C1(CC)CN(C(C2CN(C)C2)=O)CCN1Cc1cc[n+]([O-])cc1 60950,C1(CNC(C=C(C)C)=O)(CNC(=O)Cn2cnc([N+](=O)[O-])n2)CC2CCCC2C1 60951,c1(OCC(=O)NCC(Cn2cc(CCC(C)(C)O)nn2)OC)cccc(C)c1 60952,C1(C(=O)NCC(CC)N(C(CSCC=C)=O)CC)CCc2ncc(C)n2C1 60953,c1(OC)csc(C(=O)N(C2CCC(NC(C3(n4cccn4)CCC3)=O)C2)C)c1 60954,C12(NC(=O)NCCC(C)(O)C3CC3)CC1CS(=O)(=O)C2 60955,N#Cc1sc(=NCC(CNC(c2cnc(Cl)cn2)=O)C(F)(F)F)[nH]c1Cl 60956,C1(NC(C2C(C)C2)=O)CC2(CCN(C(c3ccc4c(c3)OCC4)=O)C2)C1 60957,c1(OC)cc(C(=O)NC2COCC2NC(C2C3CC4C(C3=O)C24)=O)ccc1Cl 60958,C(=O)(C(CCC(N)=O)N=[N+]=[N-])NCC(CNC(c1c(C(C)C)ncnc1)=O)O 60959,c1(C(N(C)CCNC(C2CCCN(C(=O)CNC=O)C2)=O)=O)ccccc1[N+](=O)[O-] 60960,CCCCC(CC)CCC(=O)N(CC(C)NC(c1ccn(CC)c1C)=O)C 60961,c1(C(N2CCC(CNC(C(CCC)O)=O)C2(C)C)=O)nccc2cccnc12 60962,Cc1noc(-c2cn(CC(=O)NCC(C3CC3)N(C)C(c3ccon3)=O)cn2)n1 60963,C1(CCNC(CSSC)=O)CSCCN1c1ncncc1Cl 60964,CS(C)(=O)=Nc1ccc(C(N2CC3CCCC3(CNC(C3(F)CC3)=O)C2)=O)cc1 60965,Cn1cnc(NC(=O)NCC2(c3cccc(C(F)(F)F)c3)CCC2)cc1=O 60966,N1(C(c2ccc(C)o2)C(=O)NCC2(CC3CC3)CC2)CCn2c(C)nnc2C1C 60967,C=CCC(C)C(=O)NC(C)CCN(C(=O)COCc1c(C)noc1C)C 60968,C(=O)(CCC(C)C#N)NC1(C2N(C(c3c(C)cc(C(F)F)o3)=O)CCC2)CC1 60969,c1(C(N2CCC(CNC(C(F)=CC)=O)(OC)C2)=O)cc(C)c(C)cn1 60970,C(=O)(CC(C)(C)C(C)(F)F)NC(CCNC(CCCCOC(C)=O)=O)C(C)(C)C 60971,Cc1[nH]nc2c(C(N3CCC(C)(NC(c4ncccn4)=O)C3)=O)cccc12 60972,N1(C(C2CN(C(CNC(N(C)C)=O)=O)CC(F)(F)C2)=O)CCC2(CCOC2)CC1 60973,C(N=c1[nH]c(=NCC(C)(F)c2ccccc2)c2[nH]ccc2[nH]1)C1C(C)(C)C1 60974,C(C)(c1ccccc1C)=CC(=O)N(CC(CNC(CC(C)SC)=O)O)C 60975,c1(OCC)ccc(CC(N2CCC(NC(=O)C=CSc3ccccc3)C2)=O)cc1 60976,N1(C(C(CC(CC)C)OC)=O)CC2CCCN(C(C3CC3(C)C)=O)C2C1 60977,C1(C(N(CCC(=O)N(CC(F)(F)CO)C)CC#C)=O)CCCCCCC1 60978,C1(NC(C2CN(CC)C(=O)C2)=O)CCC12CN(C(c1cn(CC(N)=O)nn1)=O)C2 60979,CC1(C)C(CN(C(=O)Cn2ncnn2)C2CC2)CCN1C(C1CC1c1ccco1)=O 60980,C12(NC(CCc3cnc(C)o3)=O)CCN(C(c3ccn(C)c3)=O)CC1C2 60981,c1(CNC(COCCCC)=O)cc[nH]c1C(=O)NC1C=CC(C(=O)NC)C1 60982,c1(C(=O)NCC(C)NC(=O)C(F)CC2CC2)ccc(Br)cc1 60983,c1(CC)nn(C)c(Cl)c1C(=O)NC1C2CN(C(C3C4CCN3CC4)=O)CC12 60984,Cc1nn(CC(F)F)c(C)c1C(N1CCC(c2ccnnc2)CC1)=O 60985,CC1CN(C(=O)C(=O)NC(c2ccccc2)=O)CCN1C(=O)C(CO)SC1CC1 60986,c1(C(=O)NCC(C(=O)Nc2c(CC)nn(C)c2)(C)CC)ccc2nccn2c1 60987,C1(NC(CC2N(C(c3nn(C)c(C(N)=O)c3)=O)CC2)=O)CC2CC1CC21CC1 60988,C1(NC(C2N(C)CCCC2)=O)CN(C(c2ccnc(F)c2Cl)=O)CC1C#N 60989,N12CCCCC1C1(CC1)NC2=O.C#CCOCCN(C)CCOC 60990,N1(CCCNC(C2C3CCC(F)C23)=O)CCN(C(=O)CC2CC=CCC2)CC1 60991,C(=O)(CS(=O)(=O)C(C)C)NCCC(C(C)C)NC(C1CCCOC1)=O 60992,CC1CC(C)N(C(c2cn3c(Br)cccc3n2)=O)CCN1C(=O)COCCF 60993,N1(C(C2C(C=C)C2)=O)CCN(C(c2c(C(C)C)nn(C)c2Cl)=O)CC1C1CC1 60994,C1(NC(CCCCC)=O)CCC2CN(C(c3ccncc3N(C)C)=O)CCC2C1 60995,c1(CC(N2CC(C(N)=O)(CNC(C3C(C)C3C)=O)C2)=O)cccc(Br)c1 60996,N1(C2CCC(NC(COCCCCC)=O)C2)CCN(C(=O)C(Cl)=CCl)CC1 60997,CC(C)=C=CC(=O)N(CCC(C(C)C)NC(c1ncoc1C1CCC1)=O)C 60998,C1(C)(C(=O)NC2CN(C(Cc3cc(C)[nH]n3)=O)C2)CCCS1(=O)=O 60999,N1(C(c2c(OC)n[nH]c2)=O)CC(C(=O)N(C)Cc2cnn(C)c2C)CC12CCC2 61000,C(=O)(C(C)S(C)(=O)=O)NC1C(CC)N(C(=O)CCn2ccnc2)CC1 61001,N(C1CCCc2cc(C#N)ccc21)c1nccc(N2CCN(CC)CC2)n1 61002,C(C(C)C(F)C(=O)NC(C)C(C)N(C)C)NC(C)=O.C1(=O)CC2(CC2)C(=O)N1 61003,C(=O)(C1=CC2CCCC12)N1CCCC(C)(NC(C(c2c(C)noc2C)C)=O)C1 61004,Cc1onc(C(F)(F)F)c1C(=O)NC1CCC1CNC(C1(O)CCSC1)=O 61005,Cc1ccc(=O)n(CC(=O)NCCCCNC(=O)C(c2ccc(F)cc2)(C)F)n1 61006,CCC(C)(C)C(C)Cc1nc(-c2cccs2)nn1-c1nccn1C 61007,C1(C(C)C)C(C(=O)NC2CC2)CCN1C(=O)Cc1cccnc1C.C1(C)CC(O)C1 61008,CC(CCN=c1[nH]c(=NCC2CC23CCOC3)c2[nH]ccc2[nH]1)P(C)(C)=O 61009,CCCC(C)(O)C(=O)N(C)CCN(C(=O)C(Cc1ccccc1)CC)C 61010,C1(Cl)(C(=O)NCC(C)NC(c2cnc(C(C)(C)C)s2)=O)CC12CCOCC2 61011,C12(CNC(C3(CC)CC3)=O)CCCCC1CN(C(c1ccc(CSC)cc1)=O)C2 61012,Cc1nc(N2CCCC2CNC(=O)CCCCCN(C)C)c2cc[nH]c2n1 61013,c1(C(=O)NCC(C)CNC(c2cnn(CC(F)F)c2)=O)cc(C(N)=O)c[nH]1 61014,c1(C(N2C(C)CN(C(c3ccc(SC)s3)=O)C(C)C2)=O)ccc2c(c1)N(C)CC2 61015,CCC(C)C(C(=O)NC1CCN1C(=O)CCS(=O)(=O)Cc1ccncc1)OC 61016,C(=O)(N=c1[nH][nH]c2c1CNC2)NCCN(C(c1ccc(NC)cc1)=O)CC 61017,CCC(C)C1C(=O)NC(C)C2CCN1CC2.C1(NC(C)=O)CCCC1 61018,C1(C(=O)NCC2CCN(C(c3ccccc3O)=O)C2)CCC2C(CC1)C2(F)F 61019,C1(NC(Cc2c(C)ccs2)=O)CCCC(NC(=O)CC(=O)N(C)C)CC1 61020,N1(C(c2c(C)sc(Br)n2)=O)CCN(C(=O)Cc2csc(=N)[nH]2)C(CCO)C1 61021,c1(C(N(CCOC)CCNC(=O)C(O)C2CCC2)=O)cc(P(C)(C)=O)cs1 61022,c1(CC(=O)NC2CC(CNC(c3snc(O)c3Cl)=O)C2)c[nH]c2ccc(F)cc12 61023,c1(C(N2CC(CNC(CC(CCC)O)=O)CC2(C)C)=O)ccc(N)cc1[N+](=O)[O-] 61024,C1(NC(C(C(C)C)O)=O)CCC(C)(CNC(c2nn(C)cc2Br)=O)CC1 61025,CC(C(=O)N1CCCN1C(=O)C(=O)NC1CC1)C(F)(F)F 61026,Cc1ccc(C(=O)NCC(c2ccccc2)CNC(=O)CC#N)c(F)c1 61027,n1(CCC)cc(Cl)c(C(=O)NC2CCC(C)(CNC(C3CN(C(C)=O)C3)=O)C2)n1 61028,C1(CC(C(=O)NCCCF)N(C)CCn2cncn2)CCC(C)(C)O1 61029,Cc1ccccc1C=CC(N1CCC(OCC(N2CC3(CC3CO)C2)=O)C1)=O 61030,c1(C(N(C2CC(NC(C3CCC(C)O3)=O)C2)C)=O)cc2sc(Cl)cc2s1 61031,N1(C(C(CC)NC(N)=O)=O)CC(NC(=O)C#CC(C)C)C(C)C1 61032,C(c1ccncc1)=CC(=O)NC1(CCCC(=O)N(N2CCC(OC)C2)C)CCC1 61033,Cc1cccc2c1OCC2C(=O)NCC(C)NC(=O)COCC1CCOC1 61034,CC(O)(C(=O)N1CC(C(=O)NCCN2CCC(O)C2)C2(CCC2)C1)C(F)(F)F 61035,C#CCC(C(=O)N(c1ccccc1O)C)NC(=O)C(C)OCC 61036,C1(CC)CCN(C(c2cscc2Cl)=O)C1C(=O)NC1(CC(C)C)CC1 61037,c1(SCC(=O)NCC2C(CNC(c3c(C)cccn3)=O)C2)ccc2c(c1)CCC2 61038,CC1(C)OC2(CN3C(CNC(c4cncc(C(N)=O)c4)=O)CC3)CCC1C2 61039,C(=O)(C(CCC)C(C)C)N1CC(NC(CCC=CC)=O)C2(C1)CC2 61040,N1(C(C(C(C)(C)C)OC)=O)CC2(CC(NC(=O)CSCc3ccccc3)CO2)C1 61041,C(C)(CSC)(C(=O)NCCCC1CC(C)C1)NC(CC1CC(=C)C1)=O 61042,c1(OC)cccc(C=CC(=O)NCC2(NC(=O)CCC3CCC3)CCOCC2)c1 61043,CCCC(C)(CC)C(=O)N1CCC(C(C)NC(=O)C(C)=CC(C)(C)C)CC1 61044,CC1(C)CN(C(c2sc(F)cc2Cl)=O)CC(CNC(C2(C)CC2(F)F)=O)O1 61045,Cc1c(C(=O)NCC2(NC(=O)C(=O)NC3CC3)CCOCC2)cncc1Cl 61046,C(CC(=O)N1CCC(CC(N)=O)C1)(C(C)(C)C)NC(Cc1ccc(C#C)cc1)=O 61047,N1(C(c2c(C)c[nH]n2)=O)CCOC(C)(CNC(C2CN(C(N)=O)C2)=O)C1 61048,Cc1cc2c(C(=O)NC(C)CCN(C)C(C3CCNC(=O)C3)=O)cccc2o1 61049,c1(C(=O)NCC2C(CNC(=O)CCc3cocn3)C2)cc2occc2s1 61050,c1(C(=O)NC2CCN(C(C(C)(C)NC(=O)OC)=O)C2)cc(C)nc2cc(C)nn12 61051,C1(CCNC(C2C(CNC(C(CC#C)O)=O)C2)=O)CCC2(CC2)CO1 61052,c1(C(=O)NC2C(NC(C(C(=O)OC)C)=O)CC2)cnc2cc[nH]c2c1 61053,c1(OC)ccc(CN2CCC(C(=O)NCc3ccncn3)C(O)C2)c(Cl)c1 61054,c1(C(N(C)CC2CCCN(C(CC(COC)C)=O)C2)=O)c(OC)cccc1F 61055,C#Cc1ccc(OC)c(C(N2CC(CNC(=O)C=CSC)CC23CCC3)=O)c1 61056,Cc1cc(C(N2CC(NC(=O)CNC=O)C3(CC3)C2)=O)cc2ccoc12 61057,C1(CC(N2CC(O)(C(C(=O)NCC(C=C)C)F)C2)=O)CC2(CCC2)C1 61058,C1(NC(c2ccc(N(C)C)cc2)=O)CC2CC1CN(C(c1cc(Cl)no1)=O)C2 61059,c1(C(=O)NCC2N(C(c3n(C)cnn3)=O)CCC2)ncsc1S(N)(=O)=O 61060,CCS(=O)CC(=O)NCC1CCCC(CNC(C2(n3cccc3)CC2)=O)C1 61061,C(=O)(C1CCc2cccnc21)NCC(CCNC(c1ncn(C)n1)=O)O 61062,C=C(Cl)CCC(=O)N1CCCC(N(C(=O)CC(=O)NCC2CC2)CC)C1 61063,N1(C(c2cc(C)n(C)c2)=O)CC2(CCN(C(c3ccc4occc4n3)=O)CC2)C1 61064,C#CCCCC(=O)N1CCN(c2ccccc2NC(C2CC=C(C)CC2)=O)CC1 61065,Cc1ccc([N+](=O)[O-])cc1C(N1CC=CC1C(=O)Nc1c(O)cccc1C#N)=O 61066,c1(C(=O)N(C2CC3(CNC3)C2)Cc2ccncc2)c(F)cc(F)cc1Br 61067,C(C)(CCC(=O)NC(CCC1CCC1)C(=O)NCCc1ncccc1F)OCC 61068,CC1(C)CC(NC(=O)C=CC2CCCN2C(=O)C(=O)C(C)(C)C)C(=O)O1 61069,c1(CC)ccc(C(N2CCCC(C)C2C(=O)OC)C(=O)NC(C)C)cc1CC 61070,c1(CS(C)(=O)=O)oc2ccccc2c1NC(c1csc2ccc(Cl)cc12)=O 61071,N1(C(CN2CCC(C)C2)=O)CCC2(CC2)CC1C(=O)Nc1cnc(Cl)nc1 61072,c1(C(=O)NC(CNC(C(CCCC#C)C)=O)C)cnc2[nH]c(C)nc2c1 61073,c1(-c2ccc3[nH]nc(C(N(CCSC)CC)=O)c3c2)nc2cc(C)cc(C)c2[nH]1 61074,CCCCCCC(C)(CC)C(=O)NCCCC(C)NC(c1csc(Cl)c1OC)=O 61075,C=CC(C)(CC)C(=O)NCC1=CCN(C(=O)C(C)c2cncs2)CC1 61076,CCCCC(C(=O)NCC1(O)CC(CNC(C2CC(C)(C)C2)=O)C1)N(C)C 61077,C1(NC(C(CCC)NC(N)=O)=O)CC2CC1CN(C(=O)CCCCC(C)C)C2 61078,CC1(C)C(c2cccc(F)c2)CCN1C(=O)NC(c1cccnc1)CC1CC1.O 61079,C=CCC(C(=O)NC(CO)CCCCNC(=O)CN(C)C(=O)OC)C(C)C 61080,CC(C)(CC1CCOCC1)C(=O)NCC(C1CCCC1)NC(C1CC(CF)C1)=O 61081,CCCS(=O)(=O)c1ccccc1C(=O)NC(CN(C(=O)C(F)(F)CC)CC)CC 61082,C1(C(=O)NC(c2ccc(F)cc2)c2n(C)ccn2)CCCN(CP(C)(C)=O)C1 61083,CC1CN(C(C2(C)COC2)=O)CCC1NC(=O)CC1(C)CCCCC1 61084,C(=O)(C#CC(C)(C)CNC(=O)C(COC)CC)NC(CCCC=C)C1CC1 61085,C1(O)(C(C)NC(CCC(=O)c2ccc(C)s2)=O)CCN(C(C2CCCS2)=O)CC1 61086,N1(CCNC(=O)CC2CCCC23CC3)CCN(C(=O)CN2CCCNC2=O)CC1 61087,c1(C(N(C2CCCN(C(=O)CCc3ncc[nH]3)C2)C)=O)cnc2c(Cl)cccn12 61088,S(=O)(=O)(CCC(=O)NC1CCN(C(=O)Cn2cnc(Br)c2)C1)N(C)C 61089,c1(C(=O)NCC2N(C(COCC)=O)CCC2C)ccc2c(c1)N(C)CCO2 61090,N1(C(Cc2c(C)ncs2)=O)CCCC2(CCN(C(C3CN(C4CCC4)C3)=O)CC2)C1 61091,c1(C(=O)NCCC(C)NC(C2C(C)C2C)=O)cccc2c1OCCCO2 61092,N1(C(CCC(C)OCC)=O)CCCC2(C1)CN(C(C1(C#N)CCC1)=O)C2 61093,Cc1nc2ccccc2c(C(=O)NCC2CCCN2C(c2ccc[nH]2)=O)c1O 61094,N1(C(c2c(CN)c3n(n2)cccc3)=O)CCC2(CC1)CC(O)(C(F)(F)F)C2 61095,CCC(CC(=O)NF)N(C(=O)C(C)CS)C.C1(C(=O)O)CC(C(F)F)C1 61096,Cc1oc(C)c(C(=O)NCC(O)CN(C(=O)Cn2cc(F)ccc2=O)C)c1C 61097,Cc1cc(C(=O)NCc2ccc(NCCC3(C)CCCN3)[nH]2)ccc1[N+](=O)[O-] 61098,C(C)(CCC(=O)NC(C)(CNC(=O)C(N1CCC(C)C1)=O)CO)OCC 61099,CCCCC(C)(F)C(=O)NC1CCN(C(c2ccc(CN(C)C)o2)=O)CC1CO 61100,C1(CC)CCC(N(C(=O)CCOCCCNC(=O)C(CC)NC(C)=O)C)CC1 61101,c1(C(=O)NC2CN(C(CN(C(COC)=O)C)=O)C(C)C2)cc(F)ccc1Br 61102,C(=O)(C1COc2ccccc21)NC(c1ccc(N(C)C)cc1)CNC(=O)CO 61103,C(=O)(C1=CCCCC1C)NC1(CNC(C2CCN(CCC)C2)=O)CC(F)(F)C1 61104,C1(COC)CN(C(c2ccc([N+](=O)[O-])[nH]2)=O)CCN1C(C12CCC(F)(CC1)C2)=O 61105,CC(C)CC(CNC=O)CC(=O)NCC(C)N(C)C(c1cccc2nonc12)=O 61106,N1(C(CNC(=O)NC)=O)CCCC2(NC(=O)CC3CN(C)C3)CC2C1 61107,Cc1nc(C(C)C)sc1C(=O)NC1CC(CCNC(C2CCC(C)(C)C2)=O)C1 61108,C1(CNC(c2c(CC)cno2)=O)CC2(CC2)CN1C(c1ccc(Cl)c(OC)c1)=O 61109,C1(CC(=O)NC(C2CCOC2)CN(C(=O)C=Cc2cocn2)CC)(OC)CCCCC1 61110,C12(NC(c3nccc(C)c3F)=O)CCCC1N(C(C1CC13CCCCC3)=O)CC2 61111,C1(NC(C(C)OCC)=O)CCCCN(C(=O)Cn2cc(C)c(O)nc2=O)CC1 61112,CCCCC(C(=O)NC1(C2CCCCO2)CC1)NC(=O)C1=CCOCC1 61113,c1(OC)ccc(C(N2CC(NC(C3CC(CN(C)C)C3)=O)CC2C)=O)nc1Cl 61114,Cc1ncc(Cl)cc1C(=O)NC1(CNC(C2(F)CCOC2)=O)CCCC1 61115,N1(S(CC2(N(C)C)CC2)(=O)=O)CCCC(C(N2CCCCCC2=O)=O)(C(=O)O)C1 61116,N1(C(CCN(C(c2cn(CC)nn2)=O)CC)=O)CC(CO)CC(C)(C)C1 61117,Cc1ccnnc1C(N1CCC(Cn2cc(-c3cccnc3)nn2)C1)=O 61118,C(CC(=O)NCC(C)S(N)(=O)=O)(CC(C)C)NC(C1N(C(C)=O)CCC1)=O 61119,C(=O)(CC(C(F)(F)F)NC(=O)CC1CCC(=O)C1C)NCCC1CC(C)OCC1 61120,CCC(C)CCC(=O)NCC1(OCC)CN(C(c2cc(=O)cc[nH]2)=O)C1 61121,N1(C(c2ncn(CCNC(C3C(C(C)C)CCC3)=O)c2)=O)CC2(CCC(=O)N2)C1 61122,c1(C(=O)NCC2(COC)CN(C(CCC=C=C)=O)C2)cc(C(F)(F)F)ccc1Cl 61123,c1(C(=O)NCC2(NC(C(C)NS(C)(=O)=O)=O)CC2)ccc(C2CCC2)nc1 61124,C12(NC(c3nn(C)c(O)c3)=O)CCCC(NC(=O)CSCC(N)=O)(C1)C2 61125,C1(NC(CS(CC)=O)=O)C2COCC1CN(C(c1nnc(O)nc1O)=O)C2 61126,N1(C(c2c(C)nc(Cl)cc2)=O)CCOC2(CCN(C(c3ccon3)=O)C2)C1 61127,CC(C)C(CNC(=O)CC1CCOC1)C(=O)N1CC(S(C)(=O)=O)C1 61128,CCCCC(=O)C(=O)N(C(C)CNC(C1(c2cccc(Cl)c2)CCC1)=O)C 61129,CC1=C(C(=O)N2CCCCC(CNC(C3CCC3)=O)C2)CCC1 61130,C(=O)(C(N)CCCCC#N)N1CCCC(N(C)C)CC1 61131,C1(C(=O)NC2(CO)CN(C(c3c(OC)cc(C)s3)=O)C2)CCc2nnnn2C1 61132,n1(C(CC)C)ccc(=NC(=O)C23CC(CN2C(=O)C(C)(C)C(C)(C)C)C3)[nH]1 61133,Cc1noc(C)c1CCNC(c1cn(C)nc1O)c1nnnn1CC1CCCO1 61134,Cc1conc1C1CN(C(=O)CCCC2CN(C(=O)C(O)C3CCC3)C2)C1 61135,C1(CNC(Cc2cncc(C)c2)=O)CCN(C(c2cc(Cl)nc(=N)[nH]2)=O)CC1C 61136,C1(NC(C2CCN(Cc3c(C)ccs3)CC2)=O)CCC2(CCC(=O)N2)CC1 61137,C1(C(N2CC3C(NC(c4n(C)ncc4)=O)(CC3)C2)=O)CC(C)(C)SC(C)(C)C1 61138,c1(OC)cc(OC)c(-c2nnc3n2CC2N3CCC2)c(OC)c1.C1(SC)CCCO1 61139,c1(NS(CCC)(=O)=O)cccc(C(=O)N(CCCNC(=O)CCN(C)CC)C)c1 61140,CC1(C)CCN(C(C2(NC(=O)C(O)C3CC3)CC(O)C2)=O)C1 61141,c1(C(=O)NCCOC2CN(C(C(N3CCC(C)C3)=O)=O)C2)c(F)cccc1F 61142,c1(C(N2CCCC(CN(C(COC)COC)C)C2)=O)cnc2cc(C)ccn12 61143,C(C(C(=O)NC(CC)C1CC1)NC(c1cc(CC)[nH]n1)=O)OCC 61144,C1(NC(CSCCCC)=O)C=CCC(C(=O)NCCOc2nccs2)C1 61145,N1(C(C2C(C(=O)OCC)C2)=O)CCOC(C(=O)OC(C)(C)C)C1.C1(=O)CS(=O)(=O)N1 61146,C=CC1(C(=O)NC(C(C)(C)O)C2CC2)CCN(C(c2ccncc2O)=O)C1 61147,C(=O)(C(CCC1(C)CC1)N(C(C)CN(C)C)Cc1ccccc1)NC(C)C1CC1 61148,N1(C(c2n(CCC)ccc2)=O)CC(NC(=O)Cc2cnn(CC)c2)C(C)C1 61149,c1(C(N(CC(C)NC(c2nocc2Br)=O)C)=O)cccc(Cl)n1 61150,c1(CC)nc(C)n(C)c1C(=O)NC1C2CN(C(c3csnn3)=O)CC12 61151,C(=O)(CCC(=O)c1cccnc1)N1CC(CCCC(=O)O)(OC)C1 61152,c1(C(CNC(C(c2cn(C)nc2)O)=O)CN(C)C)c[nH]c2cccc(Br)c12 61153,C1(O)(CN(C)C(c2cc(Cl)cc(Cl)c2)=O)CCN(C(c2cn(C)nn2)=O)CC1 61154,c1(CC)cc(Cl)ccc1C(=O)N(C(CNC(C1CCO1)=O)C1CC1)C 61155,Cc1cc(C(N2CCCC3(NC(=O)Cn4ccnc4C)CC23)=O)cnc1C(F)F 61156,C1(C#N)(C(=O)NCC(CC=C)NC(=O)Cc2[nH]cnc2C)CCCC(=O)C1 61157,N1(C(c2c(C)nsc2N2CCOCC2)=O)CCN(C(=O)C(F)F)CC(C)(C)C1 61158,C1(O)(CCNC(C(c2ccnn2C)C)=O)CCCN(C(C2CN(C(C)C)C2)=O)C1 61159,C#CC1(C(N2CC3CC2CS3)=O)CN(C(=O)Cc2ccc(C)nc2)C1 61160,c1(NC(C(CC)NC(=O)Nc2ncc(C(F)(F)F)s2)=O)cccc(C(C)C)c1 61161,C1(CC)(OC(=O)CCc2cnc(O)[nH]2)CCN(C(=O)OC(C)(C)C)C1 61162,C1(NC(c2c(CC)onc2C(F)(F)F)=O)COC2(C1)CN(C(=O)C=NOC)C2 61163,C(=O)(CC(C)P(C)(C)=O)N1CC(CN(C(c2cc(OC)c(C)cc2)=O)C)OCC1 61164,c1(C(=O)NC2CCCC(CNC(CC(C)(C)N(C)C)=O)C2)ccc2c[nH]nc2c1 61165,CC1CC2(CCO1)CCN(C(=O)COc1ccc([N+](=O)[O-])c(C(F)(F)F)c1)C2 61166,C1(O)(C(C)CNC(=O)C=CC(F)(F)F)CCN(C(c2cnc(S)n2C2CC2)=O)C1 61167,N1(C(N2CCC3(CC2)CC3(F)Br)=O)CC(=O)Nc2ncccc21 61168,CCC(CC)CC(F)C(=O)NC1(C(N2CCC(NC(C)=O)C2)=O)CC(CO)C1 61169,C1(C2CCCCC2)(C(=O)NC(CNC(C(COCC)(C)C)=O)(CC)CC)CC1 61170,c1(C(=O)NCCCN(C(CC(C)C2CCCC2)=O)C2CC2)nccc(C(F)F)n1 61171,C1(CCCNC(c2c(C)scn2)=O)CCCCN1C(=O)CCc1ccncc1 61172,C1(CN(C)C)CCc2nn[nH]c2C1.C12CCN(C1)CCN(CCC)C2=O 61173,c1(C(N2CCC(N(C(CC=CCC)=O)C)C2)=O)cc(Cl)c(C)cn1 61174,c1(C(=O)NCC2(CO)CCN(C(CC=CC=C)=O)CC2)cc(F)cc2cc[nH]c12 61175,N1(C(C2CC2COCC)=O)CC2CC(NC(c3ccnn3C3CC3)=O)CC(C2)C1 61176,CC(C)C(C(C)NC(=O)Cc1ccccc1CC(N)=O)NC(=O)CS(C)(=O)=O 61177,c1(N(C2CCCN(C(=O)C(C)(F)F)C2)C)cc(S(=O)(=O)Nc2nccs2)c[nH]1 61178,C1(CC)CN(C(C2CCCC(OC)C2)=O)CC1NC(c1ccc(C)n1C)=O 61179,C(c1ccccc1)=CC(c1ccccc1)NCC1N(C(CC)=O)CCC1 61180,C(CN=c1nc(N2CC3CC(C)(C)C3C2)c2c([nH]1)CCCCC2)N(C(C)=O)CC 61181,C1(C(=O)N(C2CCCC2O)C2CC2)CCCC(NC(C2CC3C=CC2O3)=O)C1 61182,c1(C(N2CCC(NC(C(C)NC(COC)=O)=O)C2CO)=O)cc(O)cc(N)c1Cl 61183,C(=O)(C(C)(C)C(F)c1ccccc1)N1CCC(C)(NC(c2c(Cl)cn(C)n2)=O)C1 61184,c1(C(=O)NC2CC(C)(C(F)(F)F)C2)cnc(O)n(C2CC2)c1=O 61185,c1(C(N(CC(=O)OC)Cc2cn(CCCO)nn2)=O)cc(Br)cc2nc(O)[nH]c12 61186,CCC(O)CCc1cn(CC2CC(NC(c3cnn(CC4CCOC4)c3)=O)C2)nn1 61187,c1(C(=O)NC(C(C)NC(C(C)NC(COC)=O)=O)CO)ccc(CC2CC2)cc1 61188,CC(C)(C)CC(F)C(=O)N1CCC1C(=O)NCCC(O)CO 61189,N1(C(C(CCC)O)=O)CCN(C(C2CCC2CF)=O)C(c2ccncc2)C1 61190,c1(C(=O)NCC2N(C(C3CN(CC)C(=O)C3)=O)CC2)cc(OC)c(OC)cc1F 61191,C1(C(N(C)CCn2ccnc2)=O)CC(O)CN1C(=O)Cc1cccnc1 61192,C1(NC(Cc2c(CC)con2)=O)CCC(NC(=O)COCC(F)(F)F)CC1 61193,c1(OC)nscc1CNC(c1ccoc1CNC(=O)CCCC1CCC1)=O 61194,Cc1ccc(C(F)F)c(C(N2CC(O)(CCNC(=O)Cc3cocn3)C2)=O)c1 61195,N1(C(CC2(COC)CC2)=O)CCC2(CCN(C(=O)Cc3ccsc3)CC2)C(C)C1 61196,N1(C(C(C)N=[N+]=[N-])=O)Cc2[nH]nc(C(=O)N(C3CCN(C(C)C)C3)C)c2C1 61197,CCC(C#N)(CC)C(=O)N1CCC(OC2CCN(C(C34COCC3C4)=O)CC2)C1 61198,CC(C)(CN=c1cc(OCC2CCOC2)cn[nH]1)OC(F)F 61199,C(CC(C(=O)NCCC(C)(C)N(C)C)NC(=O)CCS)SC.C(N)(=O)N 61200,C1(C(N2CCC(N(C(c3cnc(S)nc3)=O)CC)C2)=O)NC(=O)OC1(C)C 61201,c1(C(C)(C)C)cc(C(=O)NC2CCC(CNC(=O)Cn3cnnc3O)C2)on1 61202,N1(C(C(c2cccc(C)c2)=O)=O)CC2CC1CCN2C(c1nncn1C1CC1)=O 61203,C(=O)(C(CC(C)C)ONC(C1CN(C(c2ncsc2NC)=O)CC1OC)=O)OC 61204,c1(C(=O)NCC(C)N(C)C(c2c[nH]cc2-c2cnn(C)c2)=O)ccc(N)c(O)c1 61205,N1(C(CC(CCC)O)=O)CC2CCC1CN2C(=O)C(C)Cc1cccc(F)c1 61206,N1(C(C2CCC(CC)O2)=O)CCC(C(=O)NOCc2ccc(F)cc2)C(O)C1 61207,N1(C(c2nc(CC)oc2)=O)CC(CNC(=O)CCC=CBr)C(O)C1 61208,N1(C(c2cc(COC)on2)C(=O)NCCCC)c2ccccc2CC1C 61209,c1(NC(=O)NC)ccc(C(=O)N(CCC2CC2)O)cc1.C1(CC)C(OC)C1(F)F 61210,c1(C(N(CCCNC(=O)CCc2cc(C)no2)CC)=O)c(F)cccc1[N+](=O)[O-] 61211,CCCCCCC(CC)NC(C1CC=CCC1NC(=O)CC1CCCN1CC)=O 61212,CC1(NC(c2n[nH]c3c2COC3)=O)CCC(NC(C2(C)CCCCO2)=O)CC1 61213,C(C(C)(O)CC(C)C)NC(CC1C2CN(C(C(C3CCC3)OC)=O)CC21)=O 61214,CC12COCC1CN(C(=O)CCc1nnc(C3CC3)o1)C2 61215,c12cc(S(N)(=O)=O)cc(c1F)-c1ccc(s1)N(C)C(N)C2.N1(OC(C)(C)C)CCOC(C)(C)C1 61216,C(=O)(C1=NN(C)C(=O)CC1)NC1CCC(N(C(c2c(C)c(N)cnc2)=O)C)C1 61217,n1(CC)cnc2c(N3CCCCCCCC3)[nH]c(=NCc3cccc(Cl)n3)nc12 61218,C1(C(=O)NC(CCOC)CNC(c2ccc(Cl)s2)=O)CC2(C1)NC(=O)NC2=O 61219,c1(NC(c2ccc(F)cc2F)=O)ccc2c(-c3cncs3)n[nH]c2c1 61220,C1(NC(C=CCN(C(C2CN(C(C)C)C2)=O)C)=O)(CO)CC2CCCC12 61221,C1(F)(CNC(C2C(NC(C)=O)C2)=O)CC(NC(=O)OC(C)(C)C)C1 61222,C(C)(CCN=c1[nH]c(=NCC(C)(C)N(C)C)[nH]c2cc[nH]c12)OC 61223,N1(C(c2c(Cl)ccnc2Cl)=O)CCC2C(CCN2C(=O)Cc2cccc(Cl)c2)C1 61224,C1(C)(C(=O)OCC)CN(C(C2CC3CCCCC3O2)=O)C(C)(C)C1 61225,N1(C(c2cc(COC)on2)=O)CCC(C)(C)C1C(=O)NOCCC1CC1 61226,N1(C(C(C)OC)=O)CC=C(CNC(c2ncccc2Cl)=O)CC1 61227,c1(CC(=O)NC2CCC(CNC(=O)C=CCN3CCC3)C2)cnccc1Cl 61228,N1(C(C2CC(C)SCC2)=O)C2CCC1CC(C(=O)NCCOCF)C2 61229,Cc1cccc(C(=O)N(CCCNC(=O)C(c2cnccn2)C)C2CC2)c1Cl 61230,c1(CC(=O)NC2CC(NC(Cc3c(C)n[nH]c3C)=O)C2)c(F)cccc1Br 61231,C(CC(C)C)(C(=O)N(C)CCOCCCN(C)C(c1ncc(C)cc1F)=O)OC 61232,N1(CCNC(CC2C(C)CCC2)=O)CCN(C(=O)C(C)(C)N(C)CCO)CC1 61233,c1(C(=O)NCCCNC(N(C(C)C)C)=O)cccc(Br)c1 61234,C(=O)(CC(C(C)C)NC(c1cnncc1C)=O)N1CCC(CC)(CC)C1 61235,c1(CCCC)ccc(NC(=O)NC2(C(=O)NC)CC2(C)C)c(C#N)c1 61236,N(C1CCc2cc(CNC(=O)Cc3cncs3)ccc21)C(c1cnc(C)[nH]1)=O 61237,c1(C(=O)NC(CNC(c2cnc(OC)s2)=O)C)sc(F)cc1Cl 61238,C12CC(OC)CN(C1)C(C)C(=O)N2.c1(SCC)ccccc1.C1COC1 61239,N1(C(Cc2cc(N)cc(F)c2)=O)CCC(S(=O)(=O)N2CCOCC2)CC1 61240,N1(C(c2cnn(CC)c2Cl)=O)CCN(C(=O)CCc2ccoc2)CC1CO 61241,c1(C(N(CC(C)NC(C(C2CCOCC2)OCC)=O)C)=O)[nH]cnc1C#N 61242,N1(C(c2c(C)nc(O)[nH]2)=O)C2CCC1C(C)C(NC(C1CC(C)(C)CN1C)=O)C2 61243,CC(C)C(C)(C)CNC(=O)CC(c1ccccc1)N1CCCC1 61244,C1(C(N2C(CN(C(=O)CCc3nnc(C)n3C)CC)CCC2)=O)CC2CCC1C2 61245,c1(C2CCCN(C(C(=O)NC3CCOC34CCOC4)=O)C2)c[nH]c2cccnc12 61246,c1(C(C(=O)N2C(c3cccnc3)CC2)OC)cccc([N+](=O)[O-])c1 61247,N1(C(C(CC#C)CC#C)=O)CC2CCCC(C1)N2C(=O)CC1(C(F)F)CC1 61248,Cc1cc(=NC(=O)N2CC(C)(C)c3ccccc32)[nH]n1C1CCCO1 61249,C1(OC(C)C(N2CC(O)(CCNC(C3(C#N)CCC3)=O)C2)=O)CCOCC1 61250,CC(C)CC(C)C(=O)N1CC(OCCNC(=O)CCC2CCCN(C)C2)C1 61251,C1(NC(c2nn(CC)nc2C)=O)CCN(C(=O)CCc2cscn2)C12CCC2 61252,n1(CC(N2C(CNC(c3nc(C)oc3)=O)C3CCC2C3)=O)cc(C)c(O)nc1=O 61253,c1(OCCCC(N2CC(NCCCOC)OCC2)=O)cc(C)ccc1C 61254,c1(C(N2CC3CCN(C(CC(C)SC)=O)C3C2)=O)ccnc2ncccc12 61255,C1(NC(c2ccc(CCF)cc2)=O)CCC2CN(C(C3CCCO3)=O)CC2C1 61256,c1(OC)cc(C(N2CCCC2C=CC(=O)NCCC2CCN(C)C2)=O)ncn1 61257,C(N=c1[nH]nc(C(N)=O)s1)C1C2CN(C(c3nc(CC(C)C)sc3)=O)CC21 61258,CCC(CCC(=O)Nc1ccc(CO)nc1)NC(=O)CCc1ccncc1 61259,C1(C(=O)NC(C)CNC(C23CC2CCC3(F)F)=O)(OC)CCC(C)CC1 61260,c1(C(=O)NC2CC(NC(C3CCC(CN(C)C)O3)=O)C2)n[nH]c2c1CN(C)CC2 61261,CCCC(C)(O)C(=O)N1CCOCC(NC(=O)C(C(C)C)c2ccccc2)C1 61262,C1(NC(c2cnn(C3CC3)c2)=O)CC2CCC1N(C(c1ccsc1)=O)C2 61263,CC(C)C(CC(=O)NC1(C)CCN(C(c2cc(C#N)on2)=O)C1)c1ccccc1 61264,c1(C(N2CC(C)C(NC(c3nc(Br)cs3)=O)C2)=O)ccc2c(c1)C(=O)NCC2 61265,C1(C(N2CC(CNC(C=C(c3ccn(C)n3)F)=O)C2)=O)CCc2ccnn2C1 61266,C1(CC=C)(C(=O)NCc2nnc(C)o2)CCN(C(=O)COC2CCCCC2)C1 61267,C1(CNC(C(CO)NC(C)=O)=O)CCN(C(C2(CC(C)C)CCC2)=O)CC1(F)F 61268,CC1CC(C(=O)NCCN2CCN(CC(F)(F)F)CC2)CCS1 61269,C1(C(N(CC(=O)O)Cc2cn(C3C(C)(O)CCC3)nn2)=O)CC2(CC(=O)C2)C1 61270,C(C(C)(C)C(=O)NC1CCC(CNC(c2cc(Br)oc2C)=O)C1)OC 61271,N1(C(COCCC=C)=O)CCC2CN(C(c3ccnc4c3CCC4)=O)CCC12 61272,Cc1cc(NC(C2(C)CN(C(=O)CCc3ccccn3)C2)=O)cnc1F 61273,c1(CNC(=O)Cc2cccc(O)c2)cccc(F)c1F.C123CC1CN(C2)C3=O 61274,C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CN(C(=O)C=Cc1ccccc1Cl)C)(C)C 61275,C(=O)(C1CN(C(=O)CN2c3ccccc3CS2(=O)=O)c2c(C)cccc21)OC 61276,N(C(=NCC1CC1(F)F)NCC1CCCO1)CCOCC(=O)OCC 61277,C1(CNC(C2(OCC)CC2)=O)(NC(=O)C2=COCCC2)CCCCC1C 61278,C1(NC(C2(C(N)=O)CC2)=O)CC(CNC(=O)C=CC2CCCO2)C(O)C1 61279,N1(C(c2ncc(NC)nc2)=O)CC(O)CCC1C(=O)Nc1c[nH]ccc1=O 61280,Cc1oc(C(N2CCCCC2CNC(c2ccc(C(F)(F)F)[nH]2)=O)=O)cc1Br 61281,Cc1cnc(C(N2CC3CC2C3NC(=O)Cc2cc(Cl)cs2)=O)nc1 61282,N1(C(C(F)=CCC)=O)CCN(C(C2CCCCC2(C)C)=O)CC1CS(C)(=O)=O 61283,c1(C2(C(=O)NCC(CC)(C)NC(c3conc3C)=O)CC2)ccnc(Cl)c1 61284,C(=O)(C1=C(Cl)CCC(C)C1)NCCC(=C)CNC(c1[nH]nnc1C)=O 61285,c1(CNC(c2c(C)coc2C)=O)cc(O)nc(CNC(=O)CC(O)C(C)C)n1 61286,c1(N(C)C)ccc(-c2ccc(F)c(CN3CCC(CCCO)CC3)c2)cc1CO 61287,C(C(F)(F)C(=O)NCC1(NC(=O)C(n2cc(C)cn2)C)CCCCC1)OC 61288,CC(C)CC(CNC(=O)C(C)C(F)(F)F)C(=O)Nc1ccc2nc[nH]c2c1 61289,CCC(C)(C(=O)NCC1(F)CC(NC(=O)Cc2cccnc2)C1)C(F)F 61290,c1(OC)cc[n+]([O-])c(C(=O)NCC(O)CCNC(=O)C2=NNC(=O)C2)c1 61291,N1(CC(c2ccc(C)cc2)C)CC(OCC(O)CN(C)C)CCC1(C)C 61292,C(=O)(CC1=Cc2ccccc2C1)N1CC(CCC)N(C(C2CCNC2=O)=O)CC1 61293,C=C(C)CCCC(=O)N(CC(C)(C)CNC(c1ccc(OCCC)c(N)c1)=O)C 61294,C#Cc1ccc(C(N2CC(C3(NC(=O)C(F)CC4CCC4)CC3)C2)=O)cn1 61295,N1(C(C2CC(C)OC2C)=O)CC(NC(C2CC2(Cl)Cl)=O)CC2(CCC2)C1 61296,Cc1cn2cc(C(=O)N(C)CC3(O)CN(C(C4(O)CCOCC4)=O)C3)sc2n1 61297,N1(C(C2CCN(CC)C2)=O)CC2CCC(C1)N2C(=O)C=Cc1cccc(Br)c1 61298,N1(C(C(C=C)O)=O)CCC(CC)(NC(=O)CC(C(N)=O)NC(C)=O)CC1 61299,N1(C(C2C(C(C)C)C2)=O)CCC2CN(C(c3cn(CC4CCOC4)nn3)=O)C2C1 61300,C#Cc1nc(C(N2CC3CC3(CNC(=O)COCC(C)(C)C)C2)=O)cs1 61301,C(=O)(C1=CCC(C)(C)CC1)NCC1CCN(C(COC(CC)C)=O)C1(C)C 61302,C1(NC(C(C(C)C)C#N)=O)CN(C(=O)CC2CC3(CCC3)C2)CC2(CCC2)C1 61303,c1(C(=O)NC(c2ccc(F)cc2)CO)ncc(-c2cc[nH]c2)cn1 61304,C(C)(C(O)C(=O)NCC1(CC(=O)NCC2CCC2N(C)C)CC1)SC 61305,C(CCCCCNC(=O)C=CCOCCOC)N(C(c1c(CC)cco1)=O)C 61306,C(=O)(C(Cc1ccccc1)NC(C)COc1ccccc1)OC 61307,C1(CNC(c2c(COC)cco2)=O)CC2CCC1N2C(c1cc(OC)ns1)=O 61308,N1(C(CCNC(=O)NC)=O)CCN(CCN(C)C(C2CC2C(C)C)=O)CC1 61309,N1(C(C(C)SC(C)C)=O)CCC(C(O)CNC(=O)C(C)n2cncn2)CC1 61310,c1(C(=O)NC2CC3N(C(C(=O)N(C)C)=O)C(CC3)C2)cnc2ccc(F)cc2c1 61311,CC(C)CC(O)C(=O)N(CC(Cc1ccccc1)NC(C1CC1(Cl)Cl)=O)C 61312,C1(C(N2CCC(O)C2)=O)CC2CC2N1Cc1ccccc1COc1ccccc1 61313,N1(C(C(CO)NC(=O)CC2CCC2)=O)CCCCC1C1(N)CC1.O=CC=C1CCC1 61314,c1(OC)ccnc(F)c1C(=O)NCC12CC(CN1C(=O)C(C(C)C)OC)C2 61315,C1(C(C)NC(C2(CC(C)C)CCC2)=O)CCCN(C(c2cnccc2Cl)=O)C1 61316,CC1(CCC(=O)NC(CNC(c2ccsc2)=O)C2CC2)CCC(=O)N1 61317,Cc1ccc(C(N2CCCC(N(C)C(C3CC34CC4)=O)C2)=O)c(F)c1C 61318,c1(N2CC(C)CC(C)C2)ccc(S(=O)(=O)N2CCC(OCCCO)CC2)cc1F 61319,Cc1cc2c(C(=O)NCCCCCCN(C)C(C3CCCC3O)=O)cccc2o1 61320,C(CN=c1[nH]c(=NCCN2CC3CCC2C3)[nH]c2c1COC2)SCC 61321,CCC(C)(C)C(=O)N1CCC(C(=O)NCCN=[N+]=[N-])O1 61322,C#CCCC(O)CCN(C(C(O)CCOC)c1ccccc1)C 61323,CC(C)C(C(=O)NCC1CCC(=O)N1)n1cc(CCCNS(N)(=O)=O)nn1 61324,Cc1ccc(SCC(N2CCCC(c3nn[nH]n3)C2C)=O)cc1C 61325,C1(NC(CC(=O)NCC)=O)CC2CN(C(c3cnc(C)cc3Cl)=O)CC2C1 61326,CCC(C)(C(=O)NCCC1CC(NC(C2CC2c2cccnc2)=O)C1)C(F)F 61327,CC(C)CC(F)(F)C(=O)NC1CCCCC1CNC(=O)CCC1CCCCN1C 61328,n1(CCC)nnnc1C(c1nc(C)co1)NC(c1nnc(C)s1)C 61329,c1(C(=O)NC2CCCC(NC(C(COC)(F)F)=O)C2)cccc2c1NC(=O)CC2 61330,C1(NCCC2CC(OCC)C2)CCS(=O)C1 61331,c1(C(=O)NC(C(C)(C)NC(C(COCC)C)=O)C)cc(C)n(C(C)C)n1 61332,Cc1c(C(=O)NCC(C)CN(C(=O)C=C2CCC(C)C2)C)ncn1C 61333,C(=O)(CCC(=O)NC1CCCCC1CNC(=O)CN1CSCC1=O)NC 61334,C1(Nc2c(C)cn(C(C)C)c2)CC2CC1CN2C(=O)OC(C)(C)C 61335,c1(CC)ncncc1C(=O)NC1CN(C(=O)Cc2ccc(Cl)s2)CC1O 61336,Cc1nc(C)c(S(=O)(=O)N(C2C(C)C2)C)o1.c1ccccc1 61337,C1(C(=O)NCC2N(C)CCCC2)CCN(C(c2ccc(CO)o2)=O)C(C)(C)C1 61338,N1(C(c2cc3sccc3[nH]2)=O)CC2CCN(C(=O)CC34CCC(CC3)C4)C2C1 61339,c1(C(=O)NCC(C)(C)CNC(c2n[nH]c3c2COC3)=O)cc(Cl)c(Cl)cc1N 61340,C1(CC)CCCC(NC(=O)CC(C)NC(c2cn(C(C)C)nn2)=O)C1 61341,C(CCCCCNC(=O)C(F)n1ccnc1)NC(=O)CCCn1ccnc1 61342,C12(CNC(CCCCCC)=O)CCCC1N(C(=O)C=CC(F)F)CCC2 61343,Cc1nc(C#N)c(NNC(=O)N2CC(CSc3ccccc3)OC(C)C2)o1 61344,C1(C(N2CC(O)(CNC(C3(C)COC3)=O)C2)=O)CCC(=O)N(C2CC2)C1 61345,c1(C(=O)NC(C2CCCN2C(C2CN(C(N)=O)C2)=O)C)ccc2cccc(F)c2n1 61346,C1(C(=O)NC(CCC)CNC(c2cc(C3CC3)ccn2)=O)CC2(CCO1)CC2 61347,CC(C(=O)N1CC(O)CC1CNC(c1ccc(SCCCO)cc1)=O)C(C)(C)C 61348,c1(C(=O)NCCC(C)CCNC(C2CCCOC2)=O)ccc2c(c1)C(=O)NC2 61349,Cc1ncc(C(=O)NC(C2(CNC(=O)CCN3CCCCC3C)CC2)C)c(=N)[nH]1 61350,CCC(CC)CCC(=O)N1CC2CC2(NC(C2(C)C=CCC2)=O)C1 61351,C1(C(N(C)Cc2cccnc2)=O)CC12CCN(C(C1COCCO1)=O)CC2 61352,c1(OC)nc(C(=O)NCC2CC3CC3N2C(=O)C=CC(C)C)cc(O)n1 61353,C(=O)(C1=C(Cl)CCOC1)N1CCC(C(C(=O)N(CC)Cc2ccccc2)C)CC1 61354,C1(NC(=O)C2CC2)CCN(C(c2ccccc2Sc2ccccc2)=O)CC1F 61355,N1(C(c2cnc(C)[nH]2)=O)CC(NC(c2cc(C(C)(C)C)nn2C)=O)C(C)C1 61356,C(=O)(N1Cc2ccccc2CO1)C1N(C(=O)C=CC2CCOC2)CCC(=C)C1 61357,N1(OC(=O)OC(C)(C)C)CCN(c2ccc3nc(C)nn3n2)CC2(CC2)C1 61358,C1(C(=O)NCc2cscn2)CC12CCN(C(c1cnc(Cl)cc1Cl)=O)C2 61359,C1(CNC(CC(C)N(C)C)=O)CN(C(=O)C(c2cccnc2)O)CCC1(C)C 61360,N1(C(C2(CC#C)CCC2)=O)CC2CC1CN2C(=O)CCC(C)n1ccnc1 61361,C(CCC(CC)CC)NC(=NCC=C)NCC(C)(C)C(=O)OC 61362,N1C(NCCF)=NCC(F)(F)COC2CCC1CC2.S(C)(=O)(=O)NCCC 61363,C1(N(C(C(C=C)O)=O)C)CCC2(CC1)CCN(C(=O)COc1ccsc1)C2 61364,c1(C(=O)NCC2CCN(C(c3c(OC)ccs3)=O)CC2C)cnc2ccoc2c1 61365,N1(CC)CCC(CNC(C2C(C)CCN2C(C2CC(F)CN2C)=O)=O)CC1 61366,c1(C(=O)NC2(C)CN(C(C3COCCOC3)=O)C2)ccccc1OCC1CC1 61367,N1(C(=O)Cc2cc(C3CC3)on2)CC2CN(C(C3(F)CC3(Cl)Cl)=O)CCC12 61368,c1(C(N2CCC(NC(CN(c3ccncc3)C)=O)C2)=O)ccnc(Cl)c1O 61369,c1(Oc2ccc(OC)c(-n3cnnn3)c2)c[nH]c2c(C)c(Cl)ccc2c1=O 61370,c1(CC(=O)N(CC(C)N(C)C(CC(F)(F)F)=O)C)csc(-c2nc[nH]n2)n1 61371,C1(C(N2CCC(N(C(c3c(C(C)C)con3)=O)C)C2)=O)CC2(C1)CC(F)C2 61372,C1(CC(N2CCC(CC)C2)=O)CCCN(C(c2ccc(C(C)C)o2)=O)C1 61373,n1(CC(=O)NCC2=CCN(C(=O)C=C(Cl)Cl)CC2)nc2n(c1=O)CCCC2 61374,CC1CCCCCN1C(=O)NCCSCCC(F)(F)F 61375,C=CCC(C(=O)OCC)NC(=O)CC1C=CC(NC(=O)C(C)C=C)C1 61376,c1(C(=O)NC(C2CN(C(CCNC(C)=O)=O)C2)C)ccnc(S)c1 61377,C1(CCC)CN2CC1C(=O)N1CC(C1)CC2=O.C(C(C)(O)COC)NC(C)=O 61378,CCC(C(=O)NC1(C)CCCN(C(c2ncoc2C2CC2)=O)C1)C(C)(C)CC 61379,N1(C(CCCC(N)=O)=O)C2CCCC1CN(C(=O)CCOC1CC1)CC2 61380,Cc1cc(CNC(N2CCC(C)CC2C(C)O)=O)cnc1C 61381,C(=O)(C(C)(O)CC(C)C)N1CC(N(C(c2[nH]cc(C)c2)=O)C)C(C)(C)C1 61382,N1(C(C2CCC(NC(c3ccccc3)=O)C2)=O)CCCCCC1C(=O)O 61383,c1(C(N(CCN(C(=O)Cn2cnnc2O)C(C)C)C)=O)ccc(C(F)(F)F)cc1 61384,C1(C2CCOCC2)(C(N2CCN(C(c3c(C)[nH][nH]c3=N)=O)CC2C)=O)CC1(F)F 61385,n1(CC(=O)N(C(C)C(=O)NC(CC)C(C)O)CCC)ccc(C)n1 61386,Cc1nsc(C)c1NC(C1(NC(=O)CC(=O)N(C)C)CC(F)C1)=O 61387,N1(C(C2CC(C)(F)C2)=O)CCC2C(C1)NC(=O)CN2C(c1ccc(O)c(Cl)n1)=O 61388,c1(C(=O)NCC(CO)NC(c2c(C)nco2)=O)cnc(S)n1C 61389,C1(CC(N2CC(NC(c3ccc(OC)s3)=O)C(C(F)F)C2)=O)C(=O)N(C)N=C1C 61390,C1(C(=O)NC(CCNC(c2c(CC=C)cccc2)=O)(C)C)CS(=O)(=O)CCO1 61391,N1(C(CC2(COC)CC2)=O)C(C)CN(C(=O)C#CC(C)(C)O)CC1C 61392,N1(C(c2c(NCC)ccc(Cl)c2)=O)CCC(C)(C)C(NC(=O)CCC2CC2C)C1 61393,N1(C(CCC)=O)CC2CCC(NC(=O)CCC(C)c3ccccc3)CC2C1 61394,C1(NC(C(C2CCCC2)OC)=O)CCN(C(C23CC(CCO2)C3)=O)CCC1CO 61395,N1(C(Cc2c(C)ccs2)=O)CCC(NC(C2CCOC2C)=O)C(F)C1 61396,c1(C(=O)NCCC2(O)CN(C(C(C)=O)=O)C2)ccc2c(c1)CCC=C2 61397,C(=O)(C1CCCc2nc[nH]c21)OCc1cc(-n2c(C)c(N(C)C)cn2)ncn1 61398,N12CC3CC(C1)CN(C3)CCSCC2=O.C1(NC2CCOCC2)CC(F)(F)C1 61399,CC(C)(C)CCCCNC(C1C(CNC(=O)CCc2ccccn2)C1(C)C)=O 61400,C(=O)(C(O)P(C)(C)=O)N1CC(c2cn(CC(C3CCCC3)OCOC)nn2)C1 61401,Cc1c(C(N2CC(CNC(=O)C(F)(F)C3CC3)CC(C)C2)=O)[nH]ccc1=O 61402,c1(CS(=O)(=O)NC(C2CCC3(CCNCC3)O2)=O)ccc2ccccc2c1Br 61403,c1(-c2n(CCC#C)c(N3CCOC(C(F)F)C3)nn2)c(F)cc(Br)c(F)c1F 61404,N1(CC(=O)OC)C(=O)CC1S(=O)(=O)NC1CCCSCC1 61405,NS(=O)(=O)C1(C(=O)NCCN(C2CCCCC2)C(C2CC(F)(F)CS2)=O)CC1 61406,C(=O)(C(F)C(C)(C)O)NC(CC=C)CNC(c1cnn(-c2ccc(F)cc2)c1)=O 61407,CC(CCCCNC(C1CCC(=O)N1C)=O)NC(c1ccn(CCF)n1)=O 61408,c1(C(N2CCOC(c3ccco3)C2)C(=O)NCC=C)ccc2cc(Br)ccc2c1 61409,C(=O)(C(C1CCOC1)NC(C1CC1CSC(C)C)=O)NCC1(OC)CC1 61410,Cc1cccn(CC(=O)NC2CC(F)CN(C(=O)Cc3ccc(Cl)nc3)C2)c1=O 61411,N1(C(=O)CC23CCC2CN(C(c2cccc(O)c2F)=O)C3)CC2(CCOC2)C1 61412,C(=O)(CCCCC(C)C)N1CCC(C(=O)NC(COC)C2(C)CC2)(CF)C1 61413,C12(C(N(CCOCCN(C(CC(C(C)C)O)=O)C)C)=O)CCCC(C)(C1)OC2 61414,Cc1ccnc2c(-c3nnc(N4CC5CCN(C)CC5C4)n3CC3CC3)cnn12 61415,c1(NC(c2n(CCCSC)nnn2)(C)CSC)ccc2cnn(C)c2c1 61416,c1(C(N2CC(CNC(C3(CC=C)CC3)=O)C2)=O)nc(C)ccc1C 61417,CC1(C)COC(CS(=O)(=O)Nc2ccc(C3(C)CC3(F)F)cc2)CO1 61418,c1(COCC)nc(C(N2CCC2CNC(C2CC3CC3C2)=O)=O)cs1 61419,N1(C(CCNS(CC)(=O)=O)=O)CCC(NC(=O)C(=O)NCCNC(C)=O)C(F)C1 61420,N1(C(C2C(C=C)CC2)=O)CCc2nc(CNC(C3(C)CC(C)=NO3)=O)sc2C1 61421,C(=O)(C(C)(C)CS(C)(=O)=O)NCC1C(CNC(c2c(C)ncn2O)=O)OCC1 61422,N1(C(C(CCC)C#N)=O)CCC(C2CC2)C1C(N1CC(C(N)=O)C1)=O 61423,C1(CN(C(C)C)CCc2cccc(-c3nn[nH]n3)c2)CC2CCC1O2 61424,C1(NC(CS(C)(=O)=O)=O)CC2CN(C(=O)Cn3cccnc3=O)CCN2C1=O 61425,C1(C(=O)OC)CN(C(C2CC(C)N(C(=O)OC(C)(C)C)C2)=O)C(C)(C)C1 61426,N1(C(CCC=CCC=C)=O)CCC(C(=O)N(C(C)CCN(C)C)C)C1C(C)C 61427,N1(C(Cc2c(C)noc2)=O)CCOCC1CCNC(C12CC(C(C)C)(CO1)C2)=O 61428,C1(CNC(c2cnn(CC)n2)=O)CC(C)N(C(=O)CCCN(C)C(C)=O)C1 61429,C1(CCOC)(C(=O)NCC(=C2CN(c3nnc(C(=O)OC)s3)C2)F)CCCC1 61430,c1(CNC(C(C)Oc2ccccc2F)=O)ccc2c(c1)S(=O)(=O)C=C2 61431,N1(C(C(CC)(CC)CO)=O)CCC2(CCC2NC(c2cnc[nH]2)=O)CC1 61432,c1(Cc2cccc(-c3cn(CCC(=O)N(C)CC)nn3)c2)cccc([N+](=O)[O-])c1 61433,C12(C(NOC(C)C)=O)CCC(CC1)N(C(c1cccc3[nH]ncc13)=O)C2 61434,C1(C(=O)NC(CC)C(=O)N(C2CNC(=O)C23CC3)C)CC(C)(C)CCO1 61435,C(=O)(C(C)(C)S(C)(=O)=O)NC1C(c2n(C)ncc2)CN(C(C2(C#N)CCC2)=O)C1 61436,CC(C)(C)C(O)C(=O)NC1CC2(C1)CC(CNC(=O)C(c1ccccc1)O)C2 61437,C(=O)(C1=CCCC1C)NCC1(C(=O)NCc2cn(CC)nn2)CCCO1 61438,c1(C(=O)NCc2cnc(CC)[nH]2)cc(Cl)cc(Cl)c1F 61439,C1(=O)CCCCNC(=O)C(=O)NC(CCO)C2=CC=CCC12.CC(C)O 61440,N1(C(CSC)=O)CCCN(C=O)CC1.C12(CCC(C)(C)C1)C(=O)NO2 61441,Cc1cc(F)c([N+](=O)[O-])cc1NC(C12CC(Nc3ncncc3F)(C1)C2)=O 61442,N1(C(C2(C#C)CN(C(c3cnc(NC)cn3)=O)C2)=O)CCC(C2CC2)C1 61443,c1(OC)cccc(F)c1CNC(C1CCN1C(c1ccc(Br)s1)=O)=O 61444,c1(OCOC)ccccc1C(C)NC(=O)CNc1ncnc(C(C)(C)C)n1 61445,N(C1c2ccccc2OCC1(C)C)Cc1ccc(OC(F)F)nc1 61446,C#CCCCC(=O)NCCCC(C)NC(=O)C(O)Cc1[nH]cnc1C 61447,N1(C(c2ccc(CC)c(N)c2)=O)CC2CCN(C(c3ccc(O)nc3)=O)CC12 61448,N1(C(c2c(CC)c(C)ccc2)=O)CC2(CCCC2NC(=O)CS(=O)(=O)C2CC2)C1 61449,C(N=c1nc(N2CCC(CCO)C2)cc(C)[nH]1)C1(CCC=C)CCCC1 61450,C1(CNC(c2c(C)n[nH]c2C)=O)CC2(CC2)CN1C(=O)C=CCF 61451,CCCCCC(F)C(=O)N1CCC=CC1C(=O)N(Cc1cn(CCO)nn1)OC 61452,C1(NC(c2cccc(CC)c2)=O)CS(=O)(=O)CC1NC(=O)C(C)=C1CC1 61453,C12(C(=O)OCC)CNCC1(C(=O)NC(C)C(N)=O)C2 61454,c1(C(C)C)c(N2CC3C(CNC(c4ccc(C#N)cc4)=O)C3C2)ncnc1Cl 61455,c1(N(CCN(C(=O)C(C(=O)OC(C)(C)C)OC)C)C)cc2occ(Br)c2[nH]1 61456,C1(NC(c2ncc(C)cc2F)=O)CCC2(CC1)CN(C(C1C(CF)C1(C)C)=O)C2 61457,c1(C(N(CC(O)CN(C)C(c2cc(O)ncn2)=O)C)=O)cc2c(=O)cc[nH]c2s1 61458,n1(CC(=O)N(C)CC2CCN(C(C3COC3)=O)C2)cc(Br)c(O)nc1=O 61459,C1(c2n(CCCSCC)nnn2)(NCc2nnn(C(C)(C)C)n2)CC2CCCC12 61460,C(=O)(C1=NOCC1)NC(C1CCN(C(C2(C)COCCO2)=O)CC1)C(C)C 61461,C(=O)(CCCCC(N)=O)NC(C1CCCN1C(=O)CNc1ccccc1)C 61462,N1(C(C(C)(C)N(C)C)=O)CCC(NC(C2CN3CCN2CC3)=O)C(O)C1 61463,N1(C(C(C)O)=O)CCN(C(=O)CCc2n[nH]c(=N)s2)C(C(F)F)C1 61464,CC(C)CC(F)C(=O)NCC(C)(C)NC(=O)C(C)Cc1ccc(Br)cc1 61465,C1(C(C)NC(C(N2CCOC2=O)C)=O)CCN(C(=O)CSc2cnn(C)c2)CC1 61466,C(C)(CNC(=O)C(c1ccc(C)cn1)=O)(CC(C)C)NC(C(C)OCC=C)=O 61467,Cc1c(C(=O)NC2(C)CN(C(=O)CC3CC4CCC3C4)C2)cncc1Cl 61468,c1(C(C2CCCCC2)NC(C2C=CC(=O)N=N2)=O)ncc(Br)cc1OC(F)(F)F 61469,C(CN=c1[nH]c(C)cc(=NCCCCO)[nH]1)C(c1ccc(OC(C)(C)C)cc1)CC 61470,C1(NC(CCc2c(OC)cccc2)=O)CCN(C(=O)Cc2ncoc2C)C12CC2 61471,C=CCC(CNC(=O)CCCF)C(=O)NCC(n1cccn1)C 61472,Cc1cc(C(=O)NC2CN(C(c3cccc4c3OCO4)=O)C2)c2c(C)noc2n1 61473,N1(C(CC(C)C2CC2)=O)CCCCC1CCC(C)(C)NC(=O)CC1(O)CCC1 61474,N1(C(C2(C)CCN(C)C2=O)=O)CC2CCC1C(CNC(=O)C=Cc1ccoc1)C2 61475,c1(C(=O)NC2C3CN(C(C=C(CCC)C)=O)C2C3)cc(Cl)c(Cl)c(Cl)c1 61476,C1(CC)CN(C(=O)C2=CCC2)CCC1NC(c1nc(C)ccc1C)=O 61477,c1(C(NOCC(=O)NCC2(CC3CC3)CC2)=O)ccncc1F 61478,C(C(C(=O)N1CCN(C)C(CO)C1)C(C)(C)C)NC(C1(SC)CC1)=O 61479,N1(C(CCC)=O)CCCN(C(c2cccc(N3CC=CC3)c2)=O)CC1CO 61480,n1(C(C2CCN(C(C3CCC(C(N)=O)C3)=O)C2)C(=O)NC)c(C)ccc1C 61481,c1(C(N2CCN(CCNC(CCC(=C)Cl)=O)CC2)=O)coc2ccc(Cl)cc12 61482,N1(C(c2nc(OC)c(Br)cc2)=O)CC2CN(C(=O)C(O)C3CC3)CC2C1 61483,C(=O)(C(O)CC(F)(F)F)NC1CC(C(=O)NC(C2CCCCC2)C#C)C1(C)C 61484,C(C1=CCN(C)C1)NC(C(C1CCN(C(C2(F)CC2)=O)CC1)C)=O 61485,n1(CCOC)ncc(C)c1C(N1CCSC(C(F)(F)F)C1)C(=O)Nc1ccccc1 61486,n1(CCC(=O)OC)c(S)nc2cc(C(=O)OC(CSC)C3CC3)ccc2c1=O 61487,C1(CNC(C(CCC)C)=O)CC2(CC2)CN1C(c1cc2c(s1)CCC2)=O 61488,C1(C(=O)NC(C2CC(NC(c3cnn(CCO)c3)=O)C2)C)C2CC3C(C2)C13 61489,c1(CC(N2CC(OC)C(NC(C3(C)CCSCC3)=O)C2)=O)ccc(S(C)=O)cc1 61490,c1(CN2C(CC(=O)Nc3ncc(C)c(F)c3)CCC2)ccc(Br)c2nsnc12 61491,c1(CNC(=NC)NC(C)C(C#N)CC)ccc(C(F)(F)F)cc1SC 61492,c1(C(=O)NCC(CNC(C2(CC#C)CCOC2)=O)O)cc(O)cc(F)c1F 61493,c1(C(N2CC(NC(c3ncc(C)cn3)=O)C(C)CC2)=O)cccc2scnc12 61494,C1(CC)CN(C(=O)CC2COCC2(C)C)CCC1NC(C1CCCC(=O)C1)=O 61495,Cc1nc2c(NCC3CC(CNC(=O)Cn4ccnn4)CO3)ncnc2s1 61496,Cc1c(C(N2CC(CNC(c3c(F)ccc(F)c3O)=O)C2)=O)nn2c1OCCC2 61497,C(=O)(CCCC(C)(C)CC)NC1CN(C(c2c(CC)noc2)=O)CC1C(F)(F)F 61498,c1(OC)cc(F)c(CNC2CC2C(=O)Nc2cc(Br)c(F)cc2Br)cc1F 61499,N1(C(C=CC(C)(C)C)=O)CCC(O)C(F)(F)C1.C1C(=O)NOC1=O 61500,c1(C(=O)NC2(C(=O)NC(C#C)C)CSC2)cc(C)nnc1C 61501,C1(CNC(c2n(C(C)C)ncc2)=O)CN(C(=O)C2=CCCC2)CCC1C 61502,n1(CC(=O)NCC(C2CCC2)NC(C(CC=C)(F)F)=O)cc([N+](=O)[O-])nc1C 61503,Cc1nnccc1C(N1CC2CC1(C(=O)NCCn1ccnn1)C2)=O 61504,c1(SC)cc(C(F)(F)F)ccc1C(=O)N(C)CCN(C(=O)CC1CCC(=O)N1)C 61505,c1(C(N2CC(CNC(C3(CC)CC3(F)F)=O)C(F)(F)C2)=O)noc2c1CCCC2 61506,N1(C(C2(C3CC3)CNC2)=O)CCCC12CCC2 61507,C1(NC(C2C(C)(C)C(NC(c3ccc(Cl)cc3)=O)C2)=O)CC(F)(F)C1(C)C 61508,c1(CN(C)C(C2(CC(F)F)CCC2)=O)cnn2c1CN(C(c1ncc[nH]1)=O)CC2 61509,c1(C(=O)NC2CCCN(C(c3c(C)cccc3O)=O)CC2)ccc2ccsc2c1 61510,CC(C)C(C)CC(=O)NC1CCCC(NC(c2ccoc2C(F)(F)F)=O)C1 61511,c1(OC)cccc(C(N2CCN(C(=O)Cc3cccc(C)c3)C3CC23)=O)c1C 61512,C1(N(C2CCCCC2(F)F)C(C2CCC2)=O)COC2(CCNCC2)C1 61513,c1(OCC)ccc2[nH]cc(CN3CC(F)CN(c4nc(OC)c(Br)cn4)C3)c2c1 61514,c1(N2C3CN(C(CS(C(C)C)(=O)=O)=O)C(C3)C2)nc(Cl)nc2nc(Cl)n(C)c12 61515,CON=Cc1ccc(C(=O)N(CCC(C)NC(C2(C(F)F)CC2)=O)C)cc1 61516,C#CCC(CC#C)C(=O)N1CCC2(C1)CN(C(C1CC(O)(C#C)C1)=O)C2 61517,N1(C(C(C=C)(F)F)=O)CCC2(CC1)OC1(CO)CC2(NC(c2cncn2C)=O)C1 61518,c1(C2(C(N(CC(CNC(Cn3ccc(C)n3)=O)O)C)=O)CC2)ccccc1Cl 61519,C(=O)(C1CCc2snnc21)NC(c1ccccc1Br)C(N)=O 61520,c1(OC)cnnc(OC)c1C(=O)NC1CN(C(=O)C=C2CCC(C)C2)C1 61521,CC1CN(C(C2CCS(=O)CC2)=O)CCC1C(N1CCC(F)(CF)C1)=O 61522,C(C)(C)(CC(=O)NCC1(C)CNC(=O)O1)N(C)C(C1CC2CC2C1)=O 61523,N1(C(C(c2ccccc2)OC)=O)CC(CNC(=O)CC(C)(O)C2CC2)C(C)(C)C1 61524,c1(OCC)ccccc1C(=O)NC(CNC(C1CCCO1)=O)C(C)C 61525,Cc1nnc2c(C(N3CC(NC(=O)C(C4CC4)C4CC4)CC(C)C3)=O)cccn12 61526,C1(CC(=O)NC(CNC(CC(C)C)=O)C(C)C)CCCCCO1 61527,CCC(C)CC(=O)NC(C1CCN(CC(=O)Nc2cnn(C)c2C)CC1)C 61528,c1(C(=O)NCC2(NC(CNC=O)=O)CCCC2)cc(Cl)sc1S(N)(=O)=O 61529,C1(CNC(C(=C(C)C2CC2)F)=O)CN(C)CCN1C(C1CCCO1)=O 61530,[N-]=[N+]=NCC(F)CCNC(=O)C(O)CCCNC(C1CC2(CCCO2)C1)=O 61531,Cc1oc(C(=O)NCC2(F)CC(CNC(C3CCOCC3)=O)C2)cc1Br 61532,c1(CNC2C(C(N(CC)Cc3cccc(Br)c3)=O)C2)c[nH]c2ccc(Br)cc12 61533,O(NC(=O)C(F)C1CCOC1)CC(ONC(=O)Cn1[nH]cnc1=N)(C)C 61534,CC1CN(C(c2ncc(F)cc2F)=O)CCC1N(C)C(c1ccccc1F)=O 61535,C1(C(=O)NCC(CC)NC(c2cc(CCO)on2)=O)CCC(O)CN1C 61536,Cc1ccc(C(N2CCN(c3ncncc3I)C(C(F)(F)F)C2)=O)c(O)n1 61537,N1(C(C2N(C(CC)=O)CSC2)=O)C2CCC1CC(NC(=O)C(C)(C)OC)C2 61538,C1(C(N2CC3(NC(C(CC)C)=O)CC2(COC)C3)=O)CCc2nc[nH]c2C1 61539,Cc1nccnc1C(C(=O)NC1CN(C(=O)OC(C)(C)C)C1)N(C)C1CC1 61540,C1(N(C(CCCc2ncc(C)o2)=O)C)CCC(NC(C2CC2C2CC2)=O)CC1 61541,C1(NC(=O)CCNC(=O)NCC(F)F)CC12CCc1ccccc12 61542,C(=O)(C1=CCC(C)CC1)NC(CNC(c1c(CC)nn[nH]1)=O)(C)CO 61543,CC1CC(NC(c2ccoc2C(C)C)=O)CN(C(C2(CO)COC2)=O)C1 61544,C1(N(C(C2CCOC2C(C)C)=O)CC)CCCN(C(C2CC=CC2)=O)C1 61545,c1(C(=O)NCC2CN(C(C3CC4COCC4C3)=O)CC2O)n[nH]cc1[N+](=O)[O-] 61546,CC(CSc1ccc(Cl)s1)C(=O)NC1CC1 61547,c1(N(CC(=O)NCC(C)NC(=O)C(C)(O)c2ccccc2)C)ccccc1 61548,C#Cc1cncc(C(=O)NC2CC(NC(=O)C(c3ccccc3)OC(C)=O)C2)c1 61549,CCC(C)C(CC(=O)NC1CC(C2CC2)C1)NC(=O)COCC(=O)NC 61550,c1(C(CC(=O)O)NC(C2(CSC)CCC2)=O)ccccc1C 61551,CC(Cc1ccccc1)C(=O)NCC(O)CNC(C1CC(=O)N1)=O 61552,N1(C(C(C)(C2CC2)OC)=O)CCC(C2CCC(NC(=O)C(C)CC3CC3)O2)CC1 61553,c1(OC)nc(=N)nc(N(C)CC2CN(C(c3cc(C)cc(C)c3)=O)CCO2)[nH]1 61554,C(CC(C(=O)N1CCCC(OCC)C1)NC(=O)CCCSC)OCC 61555,N1(C(C=C(CCC)C)=O)CC2CCCC(CNC(=O)CC3CC(C)=NO3)C2C1 61556,C1(C(=O)NCCCC(C)C)CC(NC(=O)CCC2(C)CC2)CCO1 61557,C1(C(=O)NCC2CC(C(N3C(CC(=O)OC)CCC3)=O)C2)CC(N=[N+]=[N-])C1 61558,C1(NC(C(C)c2ccco2)=O)CC(NC(C2CCC(=O)N(C)C2)=O)CC1O 61559,C#CCC(C(=O)OC(C)=O)NC(=O)C(O)CNC(=O)C(C)(C)N(C)C 61560,C#CC1CN(C(C2CCC2(F)F)=O)CCN1C(=O)CCOC1CCCC1 61561,c1(C(=O)NC2(C)CN(c3c(OC)c(C)ncn3)C2)noc2ccc(Cl)cc12 61562,Cc1ccc(F)c(C(=O)NCC(C(=O)N2CCC(C(C)C)CC2)C(C)C)c1 61563,N1(C(C2C(CCOC)C2)=O)CCC(F)C(NC(c2cscc2C)=O)C1 61564,C1(CC)(NC(c2ccc(F)c(CO)c2)=O)CCN(C(C2CCCOC2)=O)CC1 61565,C(=O)(CC(=O)NCCn1cc(CC(C)O)nn1)OC 61566,C1(C)(CNC(CC2CCC(NC(Cn3c(C)csc3=O)=O)C2)=O)NC(=O)NC1=O 61567,Cc1cc(NCCCSCc2ccccc2)ncc1S(=O)(=O)NC1CCC(F)C1 61568,CC1(C)CCC(C)(C(=O)NCCOCCNC(=O)Cc2ccccc2O)CC1 61569,CCCCCC(O)C(=O)NCCN(C(=O)CC1CC(=O)NC1=O)C 61570,C(=O)(CCCC(=O)NCCC1CCCN(C(C2CC3C=CC2C3)=O)C1)N(C)C 61571,c1(C(=O)NC(CN(C(C(COC)(C)O)=O)C)C)coc2c(F)cccc12 61572,c1(C(N2CCCC(F)(CNC(C(C)=C3CC3)=O)C2)=O)cccn2nccc12 61573,N1(CCC(=O)NCC2(NC(C(CC)C)=O)CC2)CCSC(C)(C)C1 61574,c1(CC(=O)NC)ccc(C(=O)NCC2CCN2C(=O)CCn2cncn2)cc1 61575,C12(C(N3CC(NC(C(C)(C)OC(C)=O)=O)C(C)C3)=O)CC=CCN1CCC2 61576,c1(C(N2CC(OCCNC(C(C)S(N)(=O)=O)=O)C2)=O)cc2cc[nH]c2cn1 61577,c1(C(=O)NCC2CC(NC(c3ncn(CC)c3)=O)C2)c[nH]c2ccccc2c1=N 61578,N1(C(C2(CCC)CC2)=O)CCC2CCCN(C(c3ccsc3)=O)C2C1 61579,c1(SC)nc(C)cc(=NCC2CN(C(c3cnc(C(C)(C)C)o3)=O)CC2C)[nH]1 61580,c1(NC(CCN(C(=O)CC(C)SC)CC#C)=O)cccc(F)c1 61581,CC1C(CO)CCCN1CC(=O)Nc1cccc(OC(F)(F)C(F)F)c1 61582,C(=O)(C1=CC(O)C(NC(c2ccc(C)c(F)c2)=O)C1)NCC1CC(OCC)C1 61583,C(=O)(C1=CCCCCC1)N1CCCN(CCNC(C(n2cc(Cl)cn2)C)=O)CC1 61584,C1(C(N2CC(C3N(C(C(OC)OC)=O)CCC3)(O)C2)=O)CC(C)CCO1 61585,N1(C(CN(C)C)=O)CC2CC1CN2C(c1ccc(NCc2cc[nH]n2)cc1)=O 61586,N1(C(C(C)O)=O)CCCC(NC(C2CC3C=CC2C3)=O)CC1 61587,c1(OC)ccc2c(ccn2CC(=O)NCC(CNC(=O)Cc2ccsn2)OC)c1 61588,Cc1cc(C(=O)NCC2(O)CN(C(=O)C(F)CC3CCCCC3)C2)n(C)n1 61589,c12ccc(cc1Br)CN2C=CCO.C1(C(F)F)(OC)CCCC(C)C1 61590,c1(OCC)cnc(C(=O)N(C2CCCC(NC(c3cc(C)cs3)=O)C2)C)c(Cl)c1 61591,Cc1cc(C(CO)NC(c2oc(C3CCCNC3)nc2C)=O)ccc1Br 61592,C1(NC(C2C(C(=O)OC)C2)=O)CCCCCCC1NC(=O)CC(C)C(F)F 61593,C1(CNC(C2(CC#C)CCCO2)=O)CN(C(c2ncc(C(F)F)s2)=O)CC1C 61594,N1(Cc2ccc(-c3ccc(CC)cc3)o2)C(=O)C2C(O)CCCN2C1=O 61595,C1(NC(=O)Nc2n(Cc3ccc(C)o3)ncc2)CC(S(C)(=O)=O)C1 61596,c1(NCCN(C(C)C)C)cccc(S(=O)(=O)N(C2CC2C)C)n1 61597,C(=O)(C(F)CC(C)(C)NC(=O)CCC(C)(C)N(C)C)N1CCN(CCCC)CC1 61598,c1(C(C)C(=O)NCCCNC(=O)CN(C2CCSC2)C)c(F)cccc1F 61599,N1(C(CC(C=C)CC)=O)CC2=C(C1)CN(C(C1CC(OC)C1)=O)C2 61600,C(C)(CC(C(=O)NC1(CF)CCC1)N(CC(=O)NC1CCCCC1)C)SC 61601,C1(C(=O)NC2C(NC(C3CSCCS3)=O)CCCC2)CC2COCC(C1)C2 61602,c1(C(CC(=O)NCCCOCCNC(C(CC=CC)C)=O)O)cc(Cl)cc(Cl)c1 61603,C#Cc1cccc(CC(=O)Nc2nc(SC)ns2)c1 61604,CC(C)CC(C(=O)NCC1CC(C(=O)NCCc2ccncn2)C1)C(C)C 61605,CC(C)C(C)C(=O)N(C)CC1CCN(C(c2ccnc(-c3ccsc3)c2)=O)C1 61606,N1(C(C(CCCNC(c2c(F)ccc(C)n2)=O)(C)C)=O)CCC2CCC(O)C1C2 61607,C1(NC(COCCOC)=O)CC2(CCCN(C(=O)CC3CCC(F)(F)CO3)C2)C1 61608,CCC(O)C(C)C(=O)NCC=CCNC(=O)Cc1ccccc1OC(F)(F)F 61609,c1(C(=O)NC(CNC(C(CC)Cc2ccccc2)=O)CO)nc(OC)ccc1C 61610,C=CCCC(C(=O)NCC(C)(C)C=C)NC(=O)CCCCNC(N)=O 61611,n1(C(CC)C)nccc1C(=O)NCC1(F)CN(C(=O)C(O)CN2CCOCC2)C1 61612,C1(C(=O)OC)CCC(C(=O)NCC2CCN(C(=O)CNS(=O)(=O)C3CC3)C2)C1 61613,C1(CNC(c2c(CC)non2)=O)CCN(C(c2occ(C)c2C)=O)C12CC2 61614,c1(C(=O)NC(CN(C)C(C2COC(=O)C2)=O)Cc2ccccc2)ccc(F)cn1 61615,N1(C(C23OCC(C(=O)OC)(C2)C3)=O)CCC2(C1)CN(C(=O)C(C)O)C2 61616,Cn1cnc([N+](=O)[O-])c1NC(=O)C(N1CCC(CCN2CCOCC2)CC1)=O 61617,CC1CC(CO)CN(C(c2ccn(C3CC3(F)F)n2)C(=O)NCC(F)F)C1 61618,C1(C(=O)NC2CN(C(CCC=C)=O)C2)CCCC2(C1)NC(=O)NC2=O 61619,Cc1noc(C)c1C(=O)NCC1(F)CCC(NC(C2(CO)CCC2)=O)C1 61620,c1(C(N2CCCC(C)(CNC(C(C(C)C)F)=O)C2)=O)cc2cc(Cl)c(Cl)cc2[nH]1 61621,N1(C(CC2N(C)C(=O)CC2)=O)CCC(F)(CNC(C2C(F)(F)C23CC3)=O)CC1 61622,C1(CCNC(C=C(C)Cl)=O)CN(C(=O)CCCc2ccsc2)CCS1(=O)=O 61623,c1(C(N2CC(N(C(C3CC(C)OC3C)=O)C)C2)=O)cccc(S(C)=O)c1 61624,c1(C(C(=O)NC2(CC(=O)NC(CSC)C)CCC2)F)ccccc1 61625,N1(C2CCN(C(C3(OC(C)=O)CC3)=O)C2)CCN(C(C2CC(C)(C)CO2)=O)CC1 61626,c1(C(=O)OCC(N2CCS(=O)CC2)=O)cccc2snnc12 61627,CC1CCCC(C)N(C(=O)CCC2CCN(C(C3CS(=O)(=O)C3)=O)C2)C1 61628,c1(C(=O)NC(C(C)NC(C2CCCS(=O)(=O)C2)=O)CO)ccc2ncccc2c1 61629,CN1CCN(C)C(C(=O)NC2CCC2NC(c2ccc(N)c(F)n2)=O)C1 61630,CC(C)C(Cc1ccccc1)C(=O)N1CC(CCNC(C2CCNC2=O)=O)C1 61631,C1(C(N2C(CC)CC(F)(F)C2)=O)CN(C(=O)CC2OCCO2)CCC1(C)C 61632,Cc1ccc(C(=O)NCC2(CNC(=O)C(C)(C)c3ccsc3)CC2(F)F)c(O)c1 61633,Cc1nn(C)cc1C(N1CC(C(C)NC(=O)C=C(Cl)Cl)C1)=O 61634,n1(C(C)C)nccc1-c1cn(CC2CCN(C(=O)CSc3nnnn3C)C2)nn1 61635,CC(=O)C(C)CC(C)C(=O)N1CCCCCC(NC(=O)CCCN(C)C(C)C)C1 61636,Cc1nn(C)c(C)c1CC(=O)NCC1CCC(C)CN1C(=O)CCc1cnc[nH]1 61637,CCC(C(=O)NC(CCCNC(=O)Cc1cnns1)c1ccccc1)SC 61638,c1(CC)ncc(C(=O)NC2CCC(CCNC(=O)CC3CC(F)(F)C3)C2)[nH]1 61639,Cc1nc(C)c(CC(=O)NC2CN(C(=O)C(C(C)C)NC(C)C)CC2C)c(O)n1 61640,c1(C(N2CC(NC(C3(O)CCSCC3)=O)CC(OC)C2)=O)c(C)ncn(C)c1=O 61641,C(=O)(CCCC(=O)NCC(C1CC1)N(C(c1coc(C2CC2)n1)=O)C1CC1)OC 61642,C(=O)(C1Cc2ccccc21)NC1(CCCNC(c2nccc3nn[nH]c23)=O)CC1 61643,c1(CCNC(=O)Nc2n(Cc3ccc(C)cc3)ccn2)cc(Cl)ccc1O 61644,C(=O)(CN=c1cc[nH]cc1)N1C(CCNC(C2C(C)SCCC2)=O)CCCC1 61645,C1(CNC(CCCNC(c2c(C)ccnc2)=O)c2ccccc2)CCC(C)(C)CO1 61646,C(CC(C)N=c1nc(CNC(C(CC)CCOC)=O)[nH]s1)OC 61647,N1(C(C2(C)CCCN(C(=O)CC(F)(F)F)C2)=O)CC2CCNCC2C1 61648,C=CCC(CC)C(=O)NC1CCN(C2CCN(C(=O)CC(C)C(F)F)CC2)CC1 61649,CC1CC(Nc2ncncc2Cl)CCN1C(=O)C(O)C1CC1 61650,N1(CC)CC(C(=O)N(C)Cc2nccn2C)c2ccccc21 61651,CC#CCCCC(=O)N1CCC(N(C(C2(OC)CC2)=O)CCC)C1 61652,C(CN=c1cc(C)[nH]c(=NCCN(C(C)C)C(C)C)[nH]1)(C1CCOC1)OCC 61653,C1(CNC(C2(N(C)C)CCCC2)=O)CN(C(=O)CCC2CC(C)(C)CO2)CCO1 61654,N1(C(COC(C)=O)=O)CCCC1C1CCCCN1C(c1cncc(Cl)c1)=O 61655,S(=O)(=O)(c1cccc(F)c1)N1C(C(=O)Nc2cccc(C)n2)CC2CC21 61656,C(=O)(CP(C)(C)=O)NCC(C)CN(C(=O)C(C)(C)Oc1ccc(Cl)cc1)C 61657,CCCC(O)C(=O)NC(CCN(C)C)C(=O)N(C)CCc1cnn(C)c1 61658,C(=O)(N=c1[nH]nc(C(c2ccco2)=O)s1)N(C)CC1(OC)CCSCC1 61659,n1(C(c2ccccc2)C(=O)N(C(CCC)CO)C(C)=O)cnc(C)c1C 61660,c12ccncc1C(F)(F)CC(OC)CC(C)CC(=O)NNC2=O 61661,c1(C(=O)NCC(C)(CO)NC(c2ccc(COC)cc2)=O)cncc2c1CCC2 61662,C1(NC(C=CC(CC)C)=O)CCC2CCN(C(=O)Cc3cc(C)cs3)C12 61663,CC1(C)CCN(c2nc(Cl)ncc2Cl)CC1CNC(c1nc(F)ccc1Cl)=O 61664,c1(CN(C2CCNCC23CC3)C(c2scc(C)c2)=O)ccc(O)c(Cl)c1 61665,c1(CC)ncnc(N2CC=C(CNC(C3(C)CCC(F)(F)C3)=O)CC2)c1F 61666,C1(F)(CNC(C2(C)CCC2)=O)CCCN(C(=O)CC2(C)CCOCC2)C1 61667,C1(CC(=O)OC)CC2CC1CN(C(=O)NCc1ncccc1Br)C2 61668,C1(CC)(CC)CC(NC(=O)CSc2cccs2)CN1C(=O)C(O)C(C)C 61669,c1(C(N2C(CC)CN(C(=O)COC3(C)CCC3)CC2)=O)cc(C)c(C)nc1C 61670,C1(O)(C(N(c2[nH]c(C)nc2C(F)(F)F)C(C)=O)=O)CCN(c2ccccc2)C1 61671,c1(C(N2C(C(N3CC(OC)C(F)C3)=O)C(O)CC2)=O)cnn2ccncc12 61672,C(=O)(C(CCCC(=O)OCC)N1CCC2C(O)C(C)(C)C12)NCCCC 61673,C1(F)(C(=O)NC(c2c(C)nccc2)C)CCN(C(=O)C(C)CC(N)=O)CC1 61674,S(=O)(=O)(c1nc(Br)cs1)N(CC)C.c12c(cccc1F)N2 61675,CC(C)(CC1CCCC1)C(=O)N1CC(NC(c2cncs2)=O)C(CCO)C1 61676,N1(C(C2(CNC(=O)Cc3cnn(C4CC4)c3)CC(=C)C2)=O)CCN(C)C(CC)C1 61677,c1(C(=O)NC2C(CNC(c3cnc(OCC)s3)=O)C2)ccccc1C(C)=O 61678,c1(OC)noc(C)c1C(=O)N(C)CC1(O)CCN(C(=O)C(c2nc(C)cs2)C)C1 61679,Cc1ccc(N(C(=O)C(C(C)C)NC(=O)Cn2ccccc2=O)C)cn1 61680,C1(C(N2CCC(C(C)=O)CC2)=O)CC(=O)OC1(C)C 61681,c1(NC(=O)NC(C(c2ccccc2)OC)C)n[nH]c(COC(C)(C)C)n1 61682,C1(COC)CN(C(c2cnn(C)c2N)=O)CCN1C(c1ncccc1Br)=O 61683,c1(OC)cc(CNCc2ccncc2C(F)(F)F)cc2cc(C)oc12 61684,c1(C(C)C)nc(C(=O)NC2CCCC2C(N2CCCC2)=O)co1 61685,N1(C(CCSCC=C)=O)CCCC(COC)C1.C1(=O)CCN1CC 61686,C1(CNC(C2(CNC(c3cncn3C)=O)CC(=C)C2)=O)COCC(C)O1 61687,C(=O)(C(C)CC(C)C)N1CC(C(=O)N(C)Cc2cnccn2)(COC)C1 61688,C(C(=O)N1CC(C(=O)NCC2(CC3CC3)CC2)(C(N)=O)C1)(C(C)(C)C)OC 61689,C12(C(=O)NCCCCCNC(C3=CC(C)(C)C3)=O)CCCC1CS(=O)(=O)C2 61690,C(=O)(CCC(C)(C)C(=O)OC)N1C(C)(COC)CC(NC(=O)C=CCCC(C)C)C1 61691,C(=O)(C(F)C(CC)CC)N1CCC(CCC=C)(C(=O)NCC(=O)NC2CCC2)C1 61692,N1(C(C(N2CCCS2(=O)=O)C)=O)CCCCC1CNC(c1ccncc1F)=O 61693,c1(SCC(=O)N(C)CCNC(=O)COCc2ccncc2)ccccc1O 61694,CN1CCN(C(=O)C(C(C)(C)C)NC(=O)Cc2cscn2)CC1(C)C 61695,c1(OC)cc(C(N2CC(NC(C3CCOC3(C)C)=O)C(O)C2)=O)cc(N)c1O 61696,Cc1ccncc1-c1ccc(C(N2CCC(C)CC2)=O)nc1 61697,c1(SCC(=O)NCCN(C(C2C(C)(COC)C2)=O)CCSC)cc(F)cc(Cl)c1 61698,N1(C(c2c(C)n(CCO)nc2)=O)CC2CCC1CC2NC(=O)C(C)C1CCCO1 61699,c1(-c2cccc(C3(C(=O)Nc4cncnc4I)CC3)c2)cccc(F)c1F 61700,N1(C(C(C)C(C)(C)C)=O)CCC2(CCCN(C(C3CCS(=O)(=O)C3)=O)C2)C1 61701,c1(C(=O)NCCCN(C(CC)=O)C2CC2)cc2c(OC)c(F)ccc2[nH]1 61702,S(=O)(=O)(c1ccn(C2CC2(F)F)n1)NCC1(C)CNCCC1O 61703,C1(CCC)CCCN(C(C2(NC(=O)CCC(C)C)CCCC2)=O)C1 61704,N1(C(C(C)NC(=O)C(O)CN2CCCC2)=O)CCC(O)C12CCCC2 61705,n1(CC)nnc(C)c1CNC(C1(CCCO)CCCC1)=O 61706,C12(C(=O)NCC(CN(C)C(C3(CCF)CCC3)=O)O)COCC1C2(F)F 61707,c1(NC(=O)NC)cccc(C(=O)N(C(C)CNC(=O)CSC2CCOCC2)C)c1 61708,c1(NC(C(C)C)=O)ccccc1C(=O)NC1CCC(NC(c2ncccn2)=O)C1 61709,C1(C(=O)NCC2(CNC(C(C)O)=O)CCC2)(N(C)C)CCOCC1 61710,N1(C(C2(CC)CCCN2C(C2CCC(C)(C)C2)=O)=O)CC2CC1CN2C 61711,c1(C(=O)NCC(=O)N(CCCN(C(C2C(C)(C(C)C)C2)=O)C)C)ncccc1O 61712,C(=O)(C(F)C(CC)CC)NCCC(C(=O)N1CCC(CCO)CC1)OC 61713,N1(C(C(C2CCC(=O)N2)C)=O)CCC(C)(NC(c2ncccc2N)=O)CC1 61714,C1(C(=O)NCC2CN(C(CC(C=C)C)=O)C(C)(C)C2)CC2CCC1C21CC1 61715,Cc1ncc(C(N2CCCCC(CNC(C3CC3C3CCCO3)=O)C2)=O)cc1N 61716,C1(CC(=O)NC2CCC(CNC(C3(C=C)CCC3)=O)C2)(C(F)(F)F)CNC(=O)C1 61717,C1(NC(C=CCOC)=O)CCC12CN(C(=O)CSc1ccc(NC(C)=O)cc1)C2 61718,c1(CCn2c(C)ncc2)cc(NC(=O)NC(CO)CC(C)C)ccn1 61719,C1(NC(CCNC(COC)=O)=O)CCCCCN(C(C2CCC(F)(F)CC2)=O)C1 61720,C1(OC)CC2CC(C(=O)NC(C)CCNC(=O)C(C)(C)CN(C)C(C)=O)CC12 61721,C1(CCNC(C=COCC)=O)CN(C(=O)CCc2scnc2C)CCCO1 61722,c1(OC)cc(C(C)NC(c2ccnc(O)c2)=O)ccc1CN1CCCC1 61723,N1(C(CCCC)=O)CCC(C(F)(F)F)C(NC(C2(S(C)(=O)=O)CC2)=O)C1 61724,CCC(F)(F)CC(=O)N1CC(C)(NC(=O)C2=C(Cl)CC2)C1 61725,c1(C(=O)NCC(C2(O)CCN(C(CC3(C=C)CC3)=O)C2)C)cc(OC)cc(Cl)c1 61726,c1(C(=O)NC2CCCN(C(CN3CCC(C)CC3)=O)C2)cc2c(s1)CCC(C)C2 61727,C1(C(=O)NC(CNC(C(CCC)(C)C)=O)CCOC)CCc2cnnn2C1 61728,c1(C(N(C(C(=O)OC)C)C)=O)ccc(CNC(=O)CC2C=CCCC2)s1 61729,c1(OCC)ccc(C(=O)NCCCN(C(=O)CCn2ncn(C)c2=O)CC)cc1 61730,C1(N(C)C(C2CCCN2S(C)(=O)=O)=O)CC2CC1N(Cc1ccc(Cl)c(F)c1)C2 61731,CC1(C)CC1(Cl)C(=O)NCCC1CCCN1C(c1cnn(C2CCCCC2)c1)=O 61732,C(C(C)C(=O)NCC(C)N(C(=O)Cc1[nH]cnc1C)C)OCC 61733,c1(C(N2C3C(NC(c4nc(C)n(C)n4)=O)CC(C3)C2)=O)coc2c1C(O)CCC2 61734,S(=O)(=O)(c1c[nH]c(C(N2CCN(C(C3(C#N)CCCO3)=O)CCC2C)=O)c1)NC 61735,N1(C(C(N2CCSCC2)C)=O)CCN(C(=O)Cn2ncccc2=O)CC1CO 61736,c1(C(=O)NCCCNC(C2(C(C)(C)C)N=N2)=O)cccc(Br)n1 61737,n1(CCC(=O)N(C)CCN(C(=O)CCOCC(C)C)C(C)C)ccnn1.CO 61738,C1(C(C)NC(=O)COCc2nc[nH]n2)CCN(C(c2c[nH]c(=S)cn2)=O)CC1 61739,C(C)(C)(CCC(=O)NC1CCC(N(C)C(C2CC3CCCC3C2)=O)CC1)OC 61740,c1(-c2nnc(C)o2)ccc(C(=O)NCC(C)NC(C2CCCC23CC3)=O)cc1 61741,C(=O)(C(C)CCCC(C)=O)NC(C(=O)NCC1(OC)CCOC1)c1ccco1 61742,C1(C(=O)NC(c2nn[nH]n2)CC)CCCN1C(=O)COC1CC1 61743,c1(C(C(C)C)NC(=O)NC2COCC2F)ccc(C(C)(C)C)cc1 61744,Cc1cc(NC(=O)CCNC(=O)C(C)O)cc(Cl)c1 61745,C1(NC(CC(=C)Br)=O)CC2(C1)CN(C(=O)C=Cc1ccccc1F)C2 61746,CC1CCCn2ncc(C(=O)NC3C4CN(C(C5CC6(C5)CC6(F)F)=O)CC34)c21 61747,c1(C(=O)NCC2CC(NC(=O)Cc3ccc(Cl)cc3)C2)csc2c1CCCC2 61748,C1(CNC(C(C)=CC)=O)CCCCN1C(=O)Cc1ccccc1Cl 61749,c1(CCC(=O)NCCC(N2CCN(C(C=C(C)Cl)=O)CC2)=O)nnc(S)nc1O 61750,C(=O)(C1=NOC(C)(C)C1)NC1N(C(C23CCCC2(C(N)=O)C3)=O)CCC(C)C1 61751,C1(C(N2CCC(NC(C=C(C)C)=O)C(O)C2)=O)CCc2nnc(C)n2C1 61752,C1(CCC(=O)Nc2cn(CC)nc2)CCCN(C(=O)CCC(=O)C2CC2)C1 61753,N1(C(CC(C(C)C)C)=O)C2CCC1C(C)C(NC(C13CC(CC(F)F)(C1)C3)=O)C2 61754,C1(CN(C(C(C2CC2)OCC)=O)C)C2CN(C(c3cc(CC)[nH]n3)=O)CC12 61755,c1(OC)cc(C(=O)NC(C)C(C)NC(c2cnc(C(C)C)o2)=O)cc(F)c1F 61756,c1(OCCC)cc[nH]c(=NCCC(C)NC(=O)C=Cc2cncs2)n1 61757,C(=O)(CS(=O)(=O)CCO)NC(C(CO)NC(c1c(OC)cccn1)=O)C 61758,c1(CNC(c2csc(S)n2)=O)ccc(CNC(C2CC3CC2CO3)=O)c(F)c1 61759,C1(CCC(=O)NC(CC)CC2CC2)CCCCC1 61760,c1(OC)cc(N)c(F)cc1C(N1CC2CCC1CN2C(=O)CC1CCOC1)=O 61761,c1(CC(N2CCC(N(C(=O)C(c3cncnc3)C)CC)C2)=O)ccc(O)cc1C 61762,C1(C(=O)NC2CN(C(c3ncccc3Br)=O)CC2O)CC2(CCCC2)CO1 61763,C1(C)(C(=O)NCC(CNC(C=CC)=O)C)COCCO1 61764,C1(=CC(=O)NCC23CC(C(=O)NC4C(C)CCCC4)(C2)C3)CCC(C)(C)CC1 61765,C(C(CC(C)C)C(=O)NCC(C)(O)CC(C)C)NC(c1n[nH]c(CC)c1C)=O 61766,C1(NC(c2nc(C)oc2)=O)CC2(CCN(C(=O)C(=O)C(C)(C)C)CC2)C1 61767,N1(C(c2cc(OCC)ns2)C(=O)NC(C)(C)C)Cc2cccc(F)c2C1 61768,c1(C(=O)NC2CC(NC(c3c(C)c(C#N)ccc3)=O)C2)cncc(P(C)(C)=O)c1 61769,Cc1cnc(C(=O)NCC(C)(O)CNC(c2c[nH]c(=N)s2)=O)cc1Br 61770,C12(F)CCN(CC1)C2=O.n1(C2(C(=O)NC3C(CCC)C3)CC2)cccn1 61771,C(C(CC1CC1)C(=O)N1CCCCC1CSC)NC(CCOCC#C)=O 61772,c1(SC)ccc(C(N2CC(N(C)CC3CC3)CC(F)C2)=O)cc1[N+](=O)[O-] 61773,CCN=c1cc(-c2nc(C(C)C(=O)OC)n(-c3cc(C)c(F)c(F)c3)n2)cc[nH]1 61774,C(C(CC(=O)N1CCCC1CO)NC(c1ccc(CSC)o1)=O)SC 61775,n1(CC(=O)NCC(C2CCOC2)NC(=O)Cc2cccs2)cc(Cl)cn1 61776,c1(OCCCC(=O)NCCN(CCC)C(C2(C)CC2C)=O)ccc(Cl)cc1C 61777,c1(C(=O)OC)ccc(C(N2CCC(C(C#N)C#N)CC2)C(=O)NCCSC)cc1 61778,c1(N2CCC(N3CCCC3)(CC)CC2)[nH]c(=NCCS(C)=O)c(C)cc1N 61779,C1(CN(C)C)CCCC1NC(C1(N(C(=O)C=CCF)C)CC1)=O 61780,C(=O)(CCC(F)(F)C(F)F)NCCCCC(C)NC(CC(C)OC)=O 61781,C(=O)(C1=CC2CCCC12)NCCOCCCN(C)C(c1cnn(C)c1Cl)=O 61782,N1(CC)CCC(COC(C2CC2C(=O)NOCCC(F)F)=O)CC1 61783,C1(NC(CC(C)C)=O)CN(C(C2CCCC3(CCC3)O2)=O)C2(CCCCC2)C1 61784,c1(C(=O)NC(CC)(C)CNC(=O)Cc2cncs2)cnc(C)c(C#N)c1 61785,C12(CCNC(c3c(C)nn(C)c3)=O)CCC(C1)N(C(C1CCC3CC1CO3)=O)C2 61786,c1(C(=O)NCC(C)N(C)C(c2c[nH]c(=O)cn2)=O)cnc(C(F)F)cn1 61787,C1(NC(c2c(CC)csc2)=O)CC=C(C(=O)NCCc2ccon2)C1 61788,n1(CC)cnc2c(N3CCCCC(C)C3)[nH]c(=NCC(COC)OC)nc12 61789,C12(NC(C(C=C)CC)=O)CCCC1N(C(c1oc(C3CC3)nc1C)=O)CCC2 61790,CC12CCN(C1)C2=O.C1(C(=O)N)CCCC2CC12.c1(-c2ccccc2)ccccc1F 61791,C12(C(=O)NCCn3cc(C(N(C(C=C)C)C)=O)nc3)CCCC1CCC2 61792,N1(C(c2noc(CC)c2C)=O)CCC2CCN(C(c3c(Br)n[nH]c3C)=O)CC12 61793,C1(C(N2C(C(N3CCCC(OC)C3)=O)CCC2)=O)CC2CC(=O)C1O2 61794,C#CC1CN(C(=O)C(c2ccnn2C)NC(=O)C(C)S(N)(=O)=O)CC1O 61795,n1(CCC(N2C(CC)CCC2)=O)nc(O)c2c1CCCC2 61796,c1(C(=O)NC(CCCC)CNC(=O)CC2CCC(C)CC2)cc(F)ccc1C 61797,c1(OC)nc2ccccc2cc1CN1CC(CC(=O)Nc2ccc(I)c(Cl)n2)C1 61798,C1(C(N2C(CC)CC2)=O)CCN(C(=O)Cc2nccn2C)C1(C)C 61799,c1(NC(N2CC(=CC(=O)OC(C)(C)C)C2)=O)cccc2c1OCO2 61800,Cn1c(O)nc2cc(C(N3C4CCC3CC(NC(C3CC3CF)=O)C4)=O)ccc12 61801,CN(CCCC(=O)NCC1(F)CCN(C(=O)CCNc2ncccn2)C1)N=O 61802,c1(NCC(C)C)[nH]c(=NCc2nc(Br)n[nH]2)nc2c1cnn2C 61803,N1(C(CCCOCCC)=O)CCN(C(=O)C(C)c2ccco2)CC1C1CC1 61804,C(c1cccnc1)=CC(=O)NC1(CNC(COCc2onc(C)n2)=O)CCCC1 61805,N1(C(C2CC3CCCC23)=O)CC2CCCN(C(=O)COC(F)F)C2C1 61806,C(CS(=O)(=O)CC(=O)N1CCC(C2CC2)C1CNC(c1c[nH][nH]c1=N)=O)OC 61807,C1(C(=O)NC2(CC#C)CCCOC2)CCCN(c2ccnc(C(F)(F)F)n2)CC1 61808,C1(NCC2CC(C(=O)OCC)C2)CCCn2cncc2C1 61809,C(=O)(N1CC(C)(O)CO1)C1N(C(CC2(COC)CC2)=O)CC(=O)NC1 61810,C(CC(O)CNC(=O)C(C)N(C(=O)CN1CCNC1=O)C1CC1)OC 61811,c1(CN2CCC(C(=O)NCc3ccc(Cl)s3)C(O)C2)cc(Cl)c(O)c(Cl)c1 61812,N(C1CCc2c(Br)cccc21)CCC(C(CC)C)C 61813,C1(C(=O)NC(CNC(CC=CC=C)=O)CC(C)C)CCCCC(=O)N1 61814,CC1(C)C(NC(=O)C(C2CCCCC2)F)CCN1C(=O)CC(F)(F)Cl 61815,N1(C(C)=O)CC(NCC(C2CCCC2)NC(=O)CCNS(=O)(=O)CC)C(C)(C)C1 61816,C1(CCC=C)(C(=O)NCC2(OC(C)=O)CC2)CN(C(=O)C(C)CC2CC2)C1 61817,c1(C(=O)NCC(C2CC2)OC)n[nH]c2c1CN(C(=O)C(C)CC1CCCC1)C2 61818,C1(C(=O)NC2CCN(C)C2)COC2(C1)CN(C(C1OCCC1(C)C)=O)C2 61819,c1(C(N2CC(C)C(CCNC(C3(CF)CC3(F)F)=O)C2)=O)cccc(Cl)c1N 61820,c1(C(=O)OC)ccc(CN2CCN(S(=O)(=O)Cc3ccccn3)CC2)cc1F 61821,CC(CN=c1nc(-c2ccccc2)[nH]s1)NC(C1CC2(CCOCC2)C1)=O 61822,C1(CNC(C2CCCC3CC23)=O)CCN(C(c2nnc(O)nc2O)=O)C12CCC2 61823,c1(NC(CCC(C)(C)NC(=O)CC2=CCCC2)=O)cncc2ccccc12 61824,c1(NCCC)ccc(CNC(=O)C(=O)NC2CCCN2)cc1 61825,c1(C(=O)NC(CNC(C=CC2C(C)CCC2)=O)(C)C2CC2)nc(F)ccc1Cl 61826,C1(C(N(CC(C)(C)NC(=O)C=CC2CCCO2)C)=O)CCCC(=O)N1 61827,c1(CC)nc2ccccc2c(C(=O)NCC2(N(C)C)CCOC2)c1C 61828,C(=O)(C(C)(C)CN=c1[nH]c(=NCC#CC2CC2)c2cccc(F)c2[nH]1)NC 61829,C1(C(N(CC(=O)NCC2CCOC2)Cc2ccncc2)=O)C2CN(CCO)CC12 61830,C1(C(=O)NCc2cnccc2Cl)CC(C2CCC2)CN1 61831,Cc1c(CC(=O)NC2CC2CNC(=O)C2=CC(C)(C)C2)c(O)nc2[nH]nc(O)c12 61832,CON(C)S(=O)(=O)c1cccc(C(N2CC3CC2C3NC(C2CC(F)C2)=O)=O)c1 61833,Cc1cc(C(=O)NCc2cccc(C(=O)NC(C)C(F)(F)Cl)n2)c(C)s1 61834,CC1(C)CCN(C(C2CSCCS2)=O)CC1NC(c1coc(Cl)n1)=O 61835,CC(C)(O)C(C1CC1)NC(=O)COC1CCOC1 61836,C(N=c1ccc(C#N)c[nH]1)C1OCC(CNC(c2c(Cl)cn(CC)n2)=O)C1 61837,Fc1ccc2c(c1)C(Nc1ncc(NC3CC34CCOCC4)s1)CCCO2 61838,Cc1ccc(-c2nc(C)c(C(=O)NC3CCC(CNC(=O)C(C)O)C3)s2)c(F)c1 61839,c1(CC(=O)NCC(CCNC(CCC=CC)=O)(C)C)coc2c(F)c(F)ccc12 61840,C(C(C)C(C)C(=O)Nc1ccc(NC(C2CCC=CCC2)=O)cc1C)OC 61841,c1(C(N(CC(=O)NC(C2CCOC2)CC)C)=O)cnsc1C 61842,CCN=C(NCc1cnc(-c2ccccc2)o1)N1CCC2(CCCC2)C1 61843,CCC(C)C(C(=O)NC1CN(C(=O)Cc2ccnc(OC)c2)CC1C)N(C)C 61844,CN1CCN(C(C2CCOCC2(C)C)=O)C(C(=O)NCC(O)C(C)(C)O)C1 61845,Cc1oc(S(N)(=O)=O)cc1C(N1CCN(C(C2CCC3(CCC3)O2)=O)C(C)C1)=O 61846,CCS(=O)(=O)c1cnc(O)c(C(=O)N(CCC(C)NC(C2CC2CF)=O)C)c1 61847,C(=O)(C(O)CC(C)(C)C)NCCN(CCC)C(C1CNC(=O)C1)=O 61848,C#CC1(NC(=O)CC2(CNC(=O)C(C)=CC(C)(C)C)CC2)CCC(C)(C)C1 61849,c1(C(=O)NC2CC3CC(NC(C(C(=C)Cl)(C)C)=O)CC32)cc(F)c(F)c(C#N)c1 61850,c1(C(=O)NC2C(NC(C3CC(=O)NCC3)=O)COCC2)cc2n(n1)CCOC2 61851,S(=O)(=O)(C1CCCC1(F)F)N1CCC(C)CC1 61852,c1(N(C2CC(c3ccccc3)(NC(=O)CP(C)(C)=O)C2)C(C)=O)ccc(F)c(F)c1 61853,c1(OC)cccc(CNC(=O)CSCCNC(C2CC=CCO2)=O)n1 61854,c1(OC)ncc(NC(c2ccc(OC(c3ccc(F)cc3)=O)cn2)=O)cn1 61855,C1(C(C)O)CCN(CC(N2CCCC2CCC(=O)NCC2(O)CN(C)C2)=O)CC1 61856,c1(C(=O)NC2CCCN(C(C(C(C)C)NC(C)=O)=O)C2)ccc2c(c1)COC2 61857,CCC(CC(=O)NC1CCC(CNC(c2cc[nH]c2C2CCC2)=O)C1)C(C)C 61858,c1(C(N2CC(C)C2C(N2CCOC(CF)C2)=O)=O)cc2ncccc2[nH]1 61859,C1(C(=O)NC(CN(C)C(c2cc(-c3ccccn3)[nH]n2)=O)(C)C)CC(F)CN1C 61860,CCCCC(C(=O)N(CC)CC1CCCCN1C(=O)CSCC)C(C)C 61861,c1(C(=O)NCC(O)CNC(=O)C(F)CC2CCC2)nc(Br)n2ccccc12 61862,N1(C(CCN(CC)CC)=O)CC2CCC2(CNC(c2c(C)ccn2C)=O)C1 61863,C1(CCC)(NC(=O)COCC)CCCN(C(c2cccc(OC)c2O)=O)C1 61864,C1(OC)CC(CNC(=O)C(F)Cc2ccccc2)N(C(=O)CCC2OCCO2)C1 61865,n1(CCC(=O)NC(CC=C)CNC(=O)C(F)(F)C(C)O)nc(O)c2ccccc12 61866,N1(C(c2cc(C(C)(C)O)on2)C(=O)NC2CC2)CCCC(O)(C(=O)OC(N)=O)C1 61867,N#Cc1cc(C(N2CC(NC(C3CCCOC3)=O)CC(F)C2)=O)ccc1F 61868,n1(CC(=O)NC(C2CN(C(=O)C(O)CC3CCOCC3)CCO2)C)ncccc1=O 61869,CC1(C)CCOC1C(=O)NCC1(C(=O)Nc2cncc(Cl)c2)CC1 61870,C(CCCC(=O)N1CCC(N(C(=O)C(C2CC2)C2CC2)CC)CC1)OCCC=C 61871,N1(CC(N2CCC(CN(C(C=C(C)C(C)(C)C)=O)C)C2)=O)CCc2ccccc21 61872,c1(C(CNC(=O)NC2CC(C(=O)OC(C)(C)C)C2)O)ccc(F)cc1Cl 61873,N1(C(=O)NCC(c2cccc(N(C)C)c2)F)CC(=O)Nc2ccc(C#N)cc21 61874,c1(C(=O)NC(C(C)C)CNC(=O)CCc2cncnc2)cccnc1O 61875,C(=O)(C(O)C1=CCCCC1)NC(C(=O)NCC(C#C)OC)CC(=C)Cl 61876,c1(CCC)ncoc1C(=O)N(C)CCNC(c1cnn(C(F)(F)F)c1)=O 61877,CC(CC(C)NC(=O)Cc1cnn2ccccc12)N=c1[nH]c(Cl)nc2c1SCC2 61878,CC(C)C(C)CC(=O)NC1(C2CCCN2C(=O)CN2C(=O)CCCC2=O)CC1 61879,c1(C2C(CC(=O)NCCn3cc(CC)nn3)C2)nc(C)nc2sc(C)c(C)c12 61880,C(C(C)(C)CCCNC(=O)CN1CCCC1CSC)SC.C1C(=O)N1 61881,C1(OCC)CCC(C(N2CCCC2c2csc(NC(=O)C(C)C3CC3)n2)=O)CC1 61882,c1(C(N2CC(CC(C)NC(C(CC)=CC)=O)C2)=O)cc(OC)ncc1Cl 61883,C12(NC(c3c(CC)csc3)=O)CCCC1CN(C(=O)CC(C1CC1)C1CC1)C2 61884,N1(C(C(C(CC)C)N)=O)CCC2CN(C(=O)Cc3cccc([N+](=O)[O-])c3)CC12 61885,C1(NC(c2c(Cl)cnc(C)n2)=O)COC2(CCCN(C(C3CCS3(=O)=O)=O)C2)C1 61886,C=C(Cl)CC(C(=O)NCC1CCC(C)(C)CO1)NC(c1cc(C#N)c[nH]1)=O 61887,N1(C(CC2CC(NC(=O)C(=O)C(C)C)C2)=O)CCCC(O)(C(N)=O)C1.CO 61888,c1(OC)ccc(C(C(=O)NC2(C)CC2)N(C)C(c2ccccc2OC)C)nn1 61889,CCC(C(=O)OC)C(=O)NC1CC1NC(c1cn(C(C)(C)C)nn1)=O 61890,c1(C2CN(C(C(C3CC(C#N)C3)NC(C=CC(C)(C)SC)=O)=O)C2)cc(O)n[nH]1 61891,O(NC(=O)CCCN(C(C1CC1C(F)F)=O)C(C)C)CCCC 61892,N1(C(c2c(N)ccc(C)c2)=O)CCC2(CCN(C(C3(C(N)=O)CC3)=O)C2)C1 61893,C1(C(=O)NCC(C(=O)NC)C)CC1C1CN(C(=O)Cc2ncn(C)c2C)C1 61894,CC1(CNC(c2cc(N)ccn2)=O)CCCN(C(C23CCCC2CCC3)=O)C1 61895,c1(CC(=O)Nc2occ(COC)n2)c(C)nc(-c2ncccn2)nc1O 61896,C1(C)(NC(C2CC(=C)C2)=O)CCN(C(=O)CCn2c(-c3cccs3)nnc2S)CC1 61897,n1(C(COC)C)nc(-c2ccoc2)nc1Cc1noc(CCC(C)C)n1 61898,CC(C)CC(C(=O)N1CCC(N(C(=O)CCc2ccccc2)CCO)CC1)N(C)C 61899,CC1N(C(c2ccc(CNC(c3cc(C#N)cs3)=O)o2)=O)CCCC1(C)C 61900,C=C(C)C(CC(=O)N1CCC(NC(=O)CN2CCC(CC)C2C)CC1C)OCC 61901,c1(C(N2CCC(CCN(C)C(C3(C4CC4)CC3)=O)CC2)=O)cccc2sccc12 61902,C1(C)(NC(CCSCCCC)=O)CN(C(c2scnc2COC)=O)C1 61903,N1(C(=O)Cc2cc[nH]c2)CC(C2CCCN(C(=O)CCn3cccn3)C2)C1 61904,Cc1cc2ncnc(NC3CC4CN(C(c5c(Cl)cnn5C)=O)CC34)c2[nH]1 61905,C(C(COCC(F)F)CC(=O)OC1CCS(=O)(=O)C1)OC 61906,c1(CC)ccc(O)c(C(=O)NCCC(C)NC(=O)C(c2ccc(F)cc2)(C)C)c1 61907,N1(c2c(C)c(SCc3cc4ccccc4nn3)ncn2)CCNC(=O)C(F)(F)C1 61908,C1(CC)(CC)CC(NC(c2ocnc2C(F)F)=O)CN1C(=O)CC1CC1C1CC1 61909,c1(C(=O)NCC(CNC(=O)C=Cc2cn[nH]c2)O)cccc(F)c1[N+](=O)[O-] 61910,C1(C(N(C2CCCC2)CCNC(C2CC2C2CCC2)=O)=O)Cc2nncn2C1 61911,C1(C(=O)NCC(N(C)O)=O)CCCN1NC(=O)CC1=CCCC1 61912,c1(CNC(NC(C=C)C)=NCc2cc(C)nn2C)cc2cc(OC)ccc2s1 61913,C1(O)(C(C)NC(C(CSC)C)=O)CCN(C(c2cc(Cl)cnc2C)=O)CC1 61914,C1(C(N2CCC(C(=O)NC)CC2)=O)CN(C(c2nccs2)=O)Cc2cccn2C1 61915,O=C(C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)Cl)Nc1cccnc1 61916,c1(C)ccc(CNC(=O)CCc2cnc[nH]2)cc1.C1(C(C)NC(N)=O)CCCCO1 61917,CCS(=O)(=O)CC(=O)N1CC=CC(C(=O)NCc2cncnc2)C1 61918,c1(CC(=O)NCC2CN(C(C3CCC4CC4CC3)=O)C2)c[nH]c2cccc(F)c12 61919,c1(CCC)nc(-c2cnn(C3CCC3)c2C)n(C(c2cnn(C)c2)C)n1 61920,c1(C(=O)NCC=CCNC(c2nncc(CCC)c2)=O)cc(F)ncc1NCC 61921,C12(NC(C(Cc3cn(CCOC)nn3)NCCSC)=O)CCCC1OCC2 61922,c1(N(CCOC)CCNC(C2CC(C)(F)C2)=O)ncnn2cccc12 61923,c12c[nH]c(c1)C(=O)NCCC1(CC1)NC(=O)CC2.C1(CC)(N)CC1.C(N)=O 61924,c1(C(N2CC(NC(=O)Cc3ccoc3)(CO)C2)=O)c(Cl)cc(F)cc1Br 61925,Cc1nsc(N(C)CCOCCNC(C2CCC(C)O2)=O)c1C#N 61926,N1(C(=O)Cc2cn[nH]c2)CCC(OCCNC(=O)CCCC2CC2)C1 61927,c1(SCC)ccc(C(N2CCC(F)(C(=O)N(C)C)C2)=O)cc1 61928,CC1CC(=O)NCC1C(N1CCC(CC(=O)Nc2cncc(C(F)F)c2)CC1)=O 61929,C1(C(=O)NCCCCCC)CCN(C(C2CCN(C)C(=O)C2)=O)CCO1 61930,N1(C(CCSC(C)C)=O)CC2(C1)CN(C(c1cccc(C(C)C)n1)=O)CC2CO 61931,c1(OC)ccc2cc(C(=O)NC3CCN(C(=O)CC=C(C)C)C3)n(C)c2c1 61932,N1(C(C(C)SC)=O)CCCC(C)(C)C1C(=O)NCC1CCCN1C 61933,CN1C(=O)CN(C(C2CC2c2cn[nH]c2)=O)CC1=O 61934,c1(CNC(=O)C(=O)NCC2CCCCO2)c(F)ccc(F)c1O 61935,CCCCCCC(=O)NC1CCC1NC(c1cc(Cl)cnc1O)=O 61936,Cc1cc(C(N2CCC(NC(C3CC4(C3)CC(C)(C)C4)=O)C2)=O)c(N)cc1F 61937,CC1CN(C(c2cnnc(O)c2)=O)CC(C(=O)NC(c2nc[nH]n2)CO)O1 61938,C(=O)(C1=CCCC1)NCCN(C1CCCCC1)C(C=C(CC)CC)=O 61939,c1(C(=O)NCC2C(NC(C(C(C)C)(C)O)=O)CCC2)cccc2cc[nH]c12 61940,C1(C(N2C(C3(NC(Cc4n(C)cnc4)=O)CC3)CCC2)=O)OCCOC12CCC2 61941,C1(CC(N2CCCC(CNC(=O)C3CC3)C2)=O)Oc2ccccc2NC1=O 61942,N1(C(c2cc(C(C)=O)on2)=O)CC2CC1CN2C(c1cnc(C(F)(F)F)s1)=O 61943,c1(OC)cc(C(=O)NCC(C(C)C)NC(C23CCC(F)(CO2)C3)=O)cnc1OC 61944,c1(CC)c(C(N2CCCCC2Cc2cn(Cc3ncc(Br)cn3)nn2)=O)csc1C 61945,c1(CNC(c2c(F)cccc2F)CCOC)ccc(OC)c(F)c1 61946,C1(C)(CCNC(CC(=O)N(C)C)=O)CCN(C(=O)CC23CCCC2C3)C1 61947,N1(C(C2CCC(Nc3ncnc4ccccc34)CCCC2)=O)CCC2(CCCOC2)C1 61948,CN1CCN(C(C(=O)NCC2CCCO2)C2CC2Cl)C(CN(C)C)C1 61949,C(=O)(CCCCC(C)(C)C)N1C2C(C(N(OC)CC3CCCCC3)=O)C(CC2O)C1 61950,C1(C)(C(=O)NCC(CC(C)C)NC(=O)Cc2cn[nH]c2)CCOC(C)C1 61951,Cn1cnc2[nH]c(C(=O)NC(C)(CNC(=O)C(C)(C)S(C)(=O)=O)C3CCC3)cc12 61952,c1(C(N2CC(CCNC(c3c(CC)nc[nH]3)=O)OC(C)C2)=O)cccc2cncn12 61953,N1(C(c2ncc(C(F)F)s2)=O)CCC2CCN(C(C3CC=CC3)=O)C2C1 61954,C(=O)(C#CC1(C)CC1)N1CCC(C)(CCNC(C2CN(C)C2)=O)C1 61955,c1(CCC(=O)NCC2CC2NC(=O)CC2CNC(=O)C2)cccnc1Br 61956,CCCCCCCCC(=O)Nc1cccc(S(=O)(=O)NCC(=O)NC2CC2)c1 61957,C(=O)(CC(C(F)(F)F)NC(=O)Cc1cccnc1O)NCCSCC#C 61958,C#CCC(CC(=O)NC(c1cscn1)CO)NC(c1ccc(=N)[nH]c1)=O 61959,C1(C(=O)NCC(CN(C(C(C#C)(C)C)=O)C)(C)C)CC(c2cccc(F)c2)=NO1 61960,c1(C(=O)NCCCN(c2nnc(CC)o2)C2CCCC2)ccc(C)c(F)c1F 61961,Cc1cccc2c(C(=O)NCC3(C)CCCN(C(c4ccnnc4)=O)C3)coc12 61962,C(C(C)(O)C(=O)N1CC(C)(O)C1)OC.C1C(F)C(=O)N2CC1C2 61963,C1(NC(C=CCC)=O)CC(C(=O)NC2CCN(OC)CC2)C12CCC2 61964,N1(C(C(=C(C)C2CC2)F)=O)CC2(COC(CNC(=O)C(F)C(F)(F)F)C2)C1 61965,C1(C(C)C)CCc2sc(C(=O)OCCC3CN(C(=O)OC(C)(C)C)C3)cc2C1 61966,n1(C(C=C)C)nc(-c2ccc(Cl)cc2)nc1C(O)C(C)(C)CC 61967,C1(NC(Nc2cc(C)c(F)cc2)=S)CC(F)(F)CCC1(C)C 61968,C(c1ncc[nH]1)=CC(=O)NCC(CN(C(=O)C=CC1CCCC1)C)O 61969,CC1CNC(=O)CN1C(=O)C=CC1CCN(C(C2CC2Cl)=O)CC1 61970,Cc1cc(C)c2[nH]cc(C(C=CC(N3CC(C)C3)=O)=O)c(=O)c2c1 61971,N1(c2nccc(-n3c(C)cc(C)n3)n2)CCC(NC(c2cccnc2)=O)C(O)C1 61972,C(CCC(CCC)NC(=O)C=Cc1cncc(F)c1)NC(C(C=C)OC)=O 61973,CC1(C)COC(CC(=O)NC2CC(NC(=O)C=C3CCC3)C2)CO1 61974,C(=O)(C1=C(C#N)CCC1)N1C(CN(C(c2cccc(C)c2F)=O)C)COCC1 61975,CCC(C)(C)C(O)C(=O)NCC1(C(C)NC(=O)COc2ccc(F)c(Cl)c2)CC1 61976,N1(C(c2c(OCC=C)cccn2)=O)CCC2(CC1)CN(C(C1CCC3CC13)=O)C2 61977,C1(CNCc2ccc(C)s2)COCCN1C(=O)Cc1ccc(C(=O)N(C)C)cc1 61978,C1(C(N2CCC(O)(CO)C2)=O)(CNC(=O)C(O)CC2CCCC2)CC(F)(F)C1 61979,CC1(C)CC(NC(C2CCCN(CC(F)(F)F)C2=O)=O)CCS1(=O)=O 61980,c1(CC)ncc(C(=O)NC(C)CCN(C(=O)Cc2cccc(O)c2F)C)c(C)n1 61981,N1(C(CN(C(=O)C=C2CCCCC2)C)(C)C)CCN(Cc2cccc(I)c2)CC1 61982,CCCCC(C(=O)N1CCCCCC1C(N1CCCCC1CCCO)=O)C(C)C 61983,c1(C(=O)OC)ccc(O)nc1N1CCC(C(C)NC(=O)C(=O)NCC2CC2)C1 61984,C1(CNC(CC(=O)N(C)C)=O)CN(C(c2cc(O)ncc2F)=O)CCCO1 61985,N1(C(c2ccc(CN(CC)CC)o2)=O)CCC(NC(C2SC3C=CC2C3)=O)CC1 61986,C1(NC(COC(CC)(C)C)=O)CN(C(=O)C=Cc2ccccc2C)C2CCCC12 61987,N1(C(C=COCC)=O)CCC2(CC1)CCN2C(c1cccc2[nH]ncc12)=O 61988,C1(C(=O)NC(C)C(CO)NC(c2nnn(C)c2N)=O)CC(=O)NC(=O)N1 61989,c1(C(=O)NC(C2CCN(C(=O)CSCc3cccs3)C2)C)ncc(Cl)s1 61990,c1(C(=O)Nc2nc(C(=O)NCCC#C)n(C)c2)c(C)cc(OC)cc1C 61991,C(CC(CNC(C1(C)CCC1)=O)NC(c1cnnn1-c1ccccc1)=O)OC 61992,Cc1cnc2nccc(C(=O)NC(CNC(C3(O)CCSC3)=O)C(C)(C)C)c2c1 61993,Cc1nn(-c2ccccc2)cc1C(=O)NCC(F)CNC(=O)C=CS(C)=O 61994,O=C1NC(C(=O)NS(=O)(=O)CCC2CCCC2)Cc2n[nH]cc21 61995,CC(C(=O)NC1CCC(CNC(=O)CC2CCCC(F)(F)C2)CC1)S(C)(=O)=O 61996,Cc1csc2c(C(N3CCCC3C(C)(C)NC(=O)Cc3ccoc3)=O)cccc12 61997,c1(OC)cccc(OC)c1C(=O)NC(C)CCNc1ncnc(Cl)c1CO 61998,Cc1cc(C)c(NC(C2CCC(NC(c3cc(O)ccc3Br)=O)C2)=O)c(Br)n1 61999,Cc1cccc(N)c1C(=O)NCC1CCCN(C(c2csc(Cl)c2Cl)=O)C1 62000,C1(CC=C)(NC(c2cccc(C(F)F)c2)=O)CCN(C(C2OCCO2)=O)C1 62001,Cc1cccc(C)c1CCN=C(NCCF)NCC(C)Oc1ncccn1 62002,c1(C(=O)NC23CC(NC(c4csc(C5CC5)n4)=O)(C2)C3)cc(Cl)c2n[nH]cc2c1 62003,c1(N(C)C)ccc(-c2nc(CCc3nccn3C)n(CC(C)(C)C)n2)cn1 62004,c1(C(=O)OCC)nc(=NC(C)CNC(=O)C2=CCCS2)cc(C(C)(C)C)[nH]1 62005,c1(OC)cc(C(=O)NC2CC2CNC(c2cn(C)c(O)n2)=O)cc2cccnc12 62006,N1(C(C(F)(F)C2(OC)CCC2)=O)CC(N(C)C(C2CC3(CC3)CO2)=O)C(F)C1 62007,c1(C(=O)OC)ccc(C(=O)NC2CC2NC(C23CCCC2C3(F)F)=O)c(C#N)c1 62008,CC1CN(C(c2cc(CC3CC3)on2)=O)CC(C)N(C(=O)CC(=O)N(C)C)C1 62009,c1(C(=O)NC2C(C)CN(C(C3CCCC3(C)C)=O)C2)cn2c(n1)SCC2 62010,C#CCCCC(C)C(=O)NCC(CC=C)C(=O)N1CCC(CN=[N+]=[N-])C1 62011,C12(C(=O)NC(C#C)C)CC1CN(C(=O)C=CCOCCOC)C2 62012,N#Cc1cccc(NC(c2ccc(NS(=O)(=O)c3cn[nH]c3)nc2)=O)c1[N+](=O)[O-] 62013,N1(C(C(c2ccc(F)cc2)NCCC#C)=O)CCCCC1C1(CN)CC1 62014,Cn1cc(C(N2CCC(C(F)CNC(=O)CCS(C)=O)CC2)=O)c(Cl)n1 62015,c1(CC(N2CC3(CN(C(c4c(C)ccnn4)=O)C3)C2)=O)cccc2cnccc12 62016,C(=O)(CCCCCC#N)NC(C)C(=O)NC(CCO)C(C)(C)C 62017,CC(C)(C)C(Br)C(=O)N1CCCCC1c1cccc(Cl)c1 62018,Cc1ncc(Cl)cc1CC(=O)NCC(n1cc(COCc2ccccc2)nn1)C 62019,C1(C(=O)NC2C(NC(C3(C(=O)OCC)CC3)=O)C2)CC(=O)N(C)C(=O)N1 62020,Cc1cc(C(N2CCOC(C(N3CC(C)C(O)C3)=O)C2)=O)cnc1Cl 62021,Cc1cc(C)c(C(=O)NC(CNC(C2(C)CC2C(F)(F)F)=O)C2CC2)[nH]1 62022,C1(C(=O)NCC2(C(N)=O)CN(C(C3CC(CF)C3)=O)C2)C2CC3C(C2)C13 62023,c1(-c2nc(C3CCN(c4nccc(=N)[nH]4)CC3)on2)ccc(F)c(Cl)c1 62024,C(=O)(C(C)(C)CC(C)(C)C)NCCC(=C)CNC(c1onc2ccccc12)=O 62025,C(=O)(CCCC(=O)N1CCOCC1CC(=O)NC1CN(C)CC1(C)C)N(C)C 62026,c1(C(=O)OC)cc(C(=O)N(C(C)CC(C)C)C)cc(COC)c1 62027,c1(C(=O)NC(C(C)C)CCNC(c2cccc(Cl)c2Cl)=O)nccc(C#N)c1F 62028,N1(C(COCCC=C)=O)CCC2CCN(C(=O)C(c3ncccc3C)(F)F)CC12 62029,CC(C)(C(=O)NCCC1CCCN(C(C2(O)CCOC2)=O)C1)S(C)(=O)=O 62030,CCCCC(CNC(c1cncc(N)n1)=O)NC(=O)C(C(C)C)c1ccccc1 62031,C1(NC(C(C=C)O)=O)C2CC1N(C(C1(S(C)(=O)=O)CC1)=O)C2 62032,c1(C(=O)CC(F)F)cc(CO)cc(F)c1.C12CCCN(C1)C1(c3cn2nn3)CC1 62033,N1(C(C(CC2CCC2)OC)=O)CCOC(C)(CNC(c2ccncc2F)=O)C1 62034,c1(CCC(=O)NCC(CC)N(C)C(C2CCOC(C)C2)=O)ccc(SC)cc1 62035,c1(C(=O)NC(CCN(C(c2c(C)[nH]nc2Cl)=O)C)C)ccc(S(C)=O)cc1 62036,C1(CNC(c2nn(C)c(Br)c2)=O)CC2(CCC2)CN1C(=O)C(F)=C1CCC1 62037,C1(CC#C)(C(=O)NCCC(C)CCNC(c2c[nH]cc2C)=O)CCOCC1 62038,c1(C(=O)NC(C2OCCN(C(C3CC(N(CC)CC)C3)=O)C2)C)cncc(Cl)c1C 62039,C(=O)(C(C)(O)C(F)(F)F)N1CCCC(CC(=O)NC(C(=O)OCC)(C)C)C1 62040,Cc1cc(C)c(C(=O)N(C)CC2CCCN2C(C2CC2C(F)F)=O)cc1N 62041,N1(C(CC(C)OC)=O)CCC(NC(=O)CSc2nnnn2C2CCCC2)C12CC2 62042,Cc1ccc(N)c(C(N2CC(O)(CCNC(C3CC(C)CC(=O)N3)=O)C2)=O)c1 62043,CCCC(C)(CCC)C(=O)NCCOC1CCN(C(C2CCCCS2)=O)C1 62044,C#Cc1cc(C(=O)NC2CCN(C(c3cnc(N(C)C)cn3)=O)C2)cc(F)c1 62045,C#CC12CC(CN1C(C1CCC(CNC(=O)C(C)CC(C)C)CC1)=O)C2 62046,C(C(=O)Nn1cccn1)N(CC(C)C)C(c1cccc(C)c1N)=O 62047,C1(C(N(CCNC(=O)C=C2CCN(C)CC2)CC)=O)CCOC2(CCC2)C1 62048,c1(CC(=O)NCC2CCN(S(=O)(=O)CCCN3CCOCC3)C2)ccnc(F)c1 62049,c1(OC)cc(C=CC(N2CC(=CC(=O)O)C2)=O)sn1 62050,c1(C(N2C(C(=O)NC(CC)CC)CC(C)C2)=O)cc(OC)cc(C(F)(F)F)c1 62051,c1(OC)cc(C(=O)NC(c2ccc3c(c2)CCC3)C)nc2ccccc12 62052,C1(C(=O)OCC(C)(C)C)CCN(C(=O)CCOC(CCSCCOC)=O)CC1C 62053,C1(NC(c2c(CNC(Cn3c(C)ncc3)=O)c[nH]n2)=O)CCSC(C)C1 62054,C1(NC(C2CN(C)C2)=O)CCN(C(c2cn(C)c(=O)cn2)=O)CC1O 62055,C1(C(=O)NCC(CC(C)C)NC(=O)C(C)n2cccn2)CC(S(C)(=O)=O)C1 62056,C1(F)(C(=O)OC)CCN(C(c2nc(CS(C)(=O)=O)cs2)=O)C1 62057,N1(CCNC(c2c(CC)nccn2)=O)CCCN(C(c2cccs2)=O)CC1 62058,c1(COC)ccc(C(=O)NC(C)CN(C(=O)COCCCC(C)C)C)cc1 62059,C#CC1CCCN(Cc2ccc(C(=O)OC)cc2)C1.N12CC(C(F)C1)CC2 62060,c1(C(=O)OC(C(=O)N(C(C)C)C)C)cc(F)c(Cl)c(N)c1Cl 62061,N1(C(C(=Cc2cccs2)C)=O)CC(NC(=O)C(N2CCOCC2)C)C(C2CC2)C1 62062,c1(CNC(c2ccccc2F)(C(=O)OC)C)cc(Cl)c2c(c1)OCCO2 62063,c1(C(C(=O)NC(C)CC)N(CC=C)CC#N)ccc(CCCOC)o1 62064,N1(C(CC2(OC)CC2)=O)CC(CNC(c2ccc(C3CCC3)cc2)=O)C(C)C1 62065,c1(C(N(C)CC2CCCO2)=O)cccnc1CNC(=O)COCCC(F)(F)F 62066,C1(C(NOCC=CC)=O)COC2(C1)CN(C(C1CC3CCC(C1)O3)=O)C2 62067,C(N=c1[nH]cnc(Cl)c1C)c1ccc(CNC(c2c(N)ncc(C)c2)=O)c(F)c1 62068,c1(C(=O)NC2(CNC(c3c(C(C)C)cco3)=O)CCCC2)ccnn(C)c1=O 62069,CCCC(CNC(C1CC1(F)F)=O)NC(c1cn(C2CC2)cn1)=O 62070,c1(NC(CC(=O)OC)Cc2cccc(Br)c2)ncc(C#N)c(OC)n1 62071,Cc1cc(S(=O)(=O)OCC(O)CN2CCC(C(C)(C)C)C2)ccc1OC 62072,N1(C(c2cccc(-c3ccncc3)n2)=O)CC2CC1CN2Cc1cccs1 62073,C1(NC(C2CC(C)CN2C(c2ccc(C#N)o2)=O)=O)CC(C)N(C)CC1C 62074,CC(CCN=c1[nH]cnc2cccnc12)NC(=O)CCC1CCCOC1 62075,CC1CCN(C(=O)CCC2CC2)C(C)C1NC(c1cncc(C2CC2)c1)=O 62076,N1(CC=C)CCC(C(N2CCCC(C(C(=O)O)NCC(C)C)C2)=O)CC1 62077,C(CC(C(C)(C)C)NC(C1CCC(C)(C)C1)=O)N(C(C1(CCCC)CC1)=O)C 62078,c1(NC(c2ccc(C(N(CC)CC)=O)cc2)=O)cc(C)c2c[nH]nc2c1.C(COC)S 62079,C(=O)(C(F)C(F)(F)F)NCC1C(NC(=O)Cc2csc(C3CC3)n2)C1 62080,N1(C(C(C(C)C)C)=O)CCN(C(c2ccc(Br)c(F)c2F)=O)CC(CO)C1 62081,C#CCCN=C(NC1CC(SC(C)C)C1)N1CC=C(c2ccc(OCC)cc2)CC1 62082,CC1CN(C)C(C)CC1NC(C1C(NC(=O)COCCCF)C1(C)C)=O 62083,c1(OC)cc(C(=O)N)sc1Cl.c1(C)cn(C2CCN(C(C3CCOC3)=O)C2)nn1 62084,Cc1[nH]nc(C(N2CCOCC2CN(C(=O)C(F)(F)c2nccn2C)C)=O)c1N 62085,C12(C(=O)NCC3(C(N4CCC(C(=O)OCC)C4)=O)CCCO3)CCN(CC1)CC2 62086,c1(N2CCC(CC)CC2)ccc(S(=O)(=O)NCCN)cc1F.C(C(C)C)N(CC)CC 62087,c1(C(N2CC(CC=C)(NC(=O)C=NOC)C2)=O)sc(Cl)cc1Cl 62088,c1(C(=O)NC(CN(C(c2cnc(N(C)C)s2)=O)CC)C)cc2n(c1)CCSC2 62089,c1(C(=O)NCC2(CN(C(c3ccc(C)s3)=O)C)CC2)ccc(Cl)nc1N 62090,c1(NC2C(CCOC(C)(C)C)CCC2)nc2ccccc2o1 62091,C1(N(CC(c2nc(C)sc2)=O)C)CCC(NC(C2CCN2S(C)(=O)=O)=O)CC1 62092,C1(C(=O)NC(C#C)C)(NC(=O)C(COC)N(C)C)CC1(C)C 62093,C1(CNC(C(CC)NC(C)=O)=O)CC2CCC1N2C(=O)CCCCN(C)C 62094,C1(NC(=O)C(F)CC2CC2)CC(Nc2cc(O)ncn2)C12CCC2 62095,C1(NCc2cn(-c3cccc(OC)c3)nn2)COC2(CCC2)C1N 62096,C1(c2nnnn2Cc2ccco2)(NCc2nc(C)c(C)[nH]2)CCCCCC1F 62097,N1(CC)CC(c2nnnn2CCCC2CC2)(NCCn2ccnc2)CCC1=O 62098,C1(C(N(CCNC(=O)C(N2CCCC2)C2CC2)CC)=O)CNC(=O)CC1(C)C 62099,C1(CNC(C(F)=CCC)=O)CCCC1NC(c1cc(C(=O)OC)[nH]n1)=O 62100,C1(CNC(C(C)CO)=O)CCN(C(C2(C#N)CC3(CC3)C2)=O)CCC1(F)F 62101,C(=O)(C(O)C(C)(C)C)NCC(C)(C(C)C)NC(C1(C(=O)OCC)CCC1)=O 62102,C(=O)(CCCC(C)C)NCC1CCN(C(C=C(C)C(C)C)=O)CC1O 62103,c1(SC)ccc(C(=O)NC2CC(NC(=O)CN(C)C(C)=O)C23CCC3)c(Cl)c1 62104,CC(C)(C)CC(=O)NCCOCCC(N1CCC(CCCF)CC1)=O 62105,C1(CCCOC)C(=O)N1.c12cc(F)ccc1N2.c1(COC)ccc(C(N)=O)o1 62106,N1(C(CCn2c(C)ncc2)=O)CCC2(CCCC2NC(=O)Cc2n[nH]c(=N)s2)C1 62107,CN1CCCC(n2cc(C3(O)CN(C(c4cncc(C(F)(F)F)n4)=O)C3)nn2)C1 62108,C(=O)(CCCC(C)(C)C#N)NCC(C)(C)NC(Cc1cc(OC)cc(OC)c1)=O 62109,N1(C(COCC)=O)CC2COCCC2(NC(=O)CC(n2nc(C)cc2C)C)C1 62110,n1(CC(=O)NCC2C3N(C(C(COC)O)=O)C(CC3)C2)nc2ccccn2c1=O 62111,C1(C(=O)NC(C)(C)C=CC(=O)NCCCC2(O)CCC2)C2CCC(C2)C1(C)C 62112,N1(C(=O)Cc2cnsc2)CCC2(CCCN2C(C2CCCCS2(=O)=O)=O)CC1 62113,c1(C(N2CCC(NC(CCC#CC)=O)CC2)=O)cc(OCC)ncc1Cl 62114,c1(CC)cc(C(=O)NC2C3CC2N(C(c2oc(C)nc2C)=O)C3)ccc1C 62115,CCC(CN(C)C)(CC)NC(=O)CC(C)Cc1ccc(Cl)cc1 62116,C1(COC)(CNC(N2CC(CC(=O)O)C(C)C2)=O)CCCCC1 62117,N1(C(C(C)CF)=O)CCCC(N2CCN(C(c3n[nH]c(=N)s3)=O)CC2)C1 62118,c1(C(N2CC(O)CCC(NC(C(C)N3CCC3)=O)C2)=O)nc2n(c1Cl)CCCC2 62119,c1(C(=O)NC(CNC(C(C)C2CCCC2)=O)(C)CO)cc2c(s1)CC(C)(C)C2 62120,n1(CC)nc(C(=O)NC(C2CCN(C(C3CCCCS3)=O)CC2)C(C)C)cc1C 62121,c1(N(C)C)nc(NC(C2CC(C)(NC(C3CC4CC4C3)=O)C2)=O)ccn1 62122,C1(NC(C=CC=CC)=O)CCN(C(c2ccccc2-c2ncn(C)n2)=O)CC1C 62123,N1(C(C=C(C)C2CC2)=O)CCC(CNC(=O)C(C)(C)c2cnsc2)C(C)C1 62124,c1(C(N2CC(CC)C(C(=O)NCC=CCl)C2)=O)cc(C)nc(C)n1 62125,c1(SCCCN(C(=O)NN2C(C)CCC2)C)ccccc1OC(F)F 62126,C(=O)(CCCC(=O)NCCCCNC(=O)Cc1ccccc1NC(N)=O)OC 62127,C1(N(C(C(CC=C)(F)F)=O)C)CCCC2CN(C(=O)CC(C)(C)CC)CC12 62128,CCN=C(NCc1csc(C2CC2)n1)N1CCC2(CCC2)C1 62129,C1(O)(C(C)NC(=O)CC(C)c2ccco2)CCN(C(c2ccc[nH]2)=O)CC1 62130,c1(C(N(CC(C)CO)C)=O)coc(CNC(C2(O)CCOC2)=O)n1 62131,c1(NC)c(C(=O)NC(C2CCN(C(C3CC4CCCC34)=O)C2)C)cccc1N 62132,C(=O)(C(C)CCCc1ccccc1)N1CCC(C(C)NC(=O)CC2CC2(C)C)C1 62133,C1(C)(CNC(c2n(CC#C)cnn2)=O)CC(OC)CN1C(=O)CCCCCOC 62134,C1(NC(=O)C(O)Cc2ccccc2)CC2CC1CN(C(C1CCC3(CC3)C1)=O)C2 62135,C12(C(=O)NCCC(C)N(C(c3ccc(C(=O)OC)[nH]3)=O)C)CCCN(CCC1)C2 62136,N1(C(c2cccc(C(F)(F)F)n2)C(=O)NCC=C)CCCN(C)CC1C 62137,CN1CC(CNC(C2(NC(c3ccncc3O)=O)CC2)=O)OCC1=O 62138,C1(NC(CSC(C)=O)=O)COC2(CCN(C(=O)Cn3ccc(C)n3)C2)C1 62139,c1(OCC)ccccc1OC(C)C(=O)NC(C)C(C)F 62140,N1(C(CN(CCC#C)C)=O)CCCC(F)(C(N2CCS(=O)C(C)C2)=O)C1 62141,c1(C(N(C2CC(NC(C(C)NC(N)=O)=O)C2)C)=O)cccc2c1CCOC2 62142,c1(NC(N(CC(CC)N2CCCC2)CC)=O)ccc(Cc2nc[nH]n2)cc1 62143,Cc1cc(N)cnc1C(N1CC(CC(F)C(=O)NCC(CC)C(C)(F)F)C1)=O 62144,c1(C(=O)NC2CC(NS(=O)(=O)c3cccnc3)C2)cc(Cl)nc(Cl)c1F 62145,n1(CC(=O)NCc2onc(-c3cccc(C)c3)n2)c(C(C)C)nc2ccccc12 62146,C1(OC)CC(C)CN(C(C2(C)CCCN2C(=O)COCc2nc[nH]n2)=O)C1 62147,C1(C(=O)NC(C2CN(c3cnc(F)cn3)C2)C)CCC(N(C)C)CC1 62148,n1(CCC(=O)NCCCC2(NC(C(C)C#N)=O)CC2)cnc2sccc2c1=O 62149,c1(NC(=O)CC2CN(C(C3CN(CCCO)CCO3)=O)C2)ncc(Cl)nc1Cl 62150,C1(NC(=O)CC2(c3ccccc3)CC2)COC2(C1)CN(C(=O)C1=CCCOCC1)C2 62151,N1(C(CC(C)n2ccnc2)=O)CC2CC(NC(C3CCCC(C)(C)C3)=O)CC1C2 62152,C1(NC(C=CC(C)NC(c2n(CCC)ncc2)=O)=O)CCN(C)CC1C 62153,N1(C(CSC2C(=O)OCC2)=O)C2CCCC1CN(C(c1csc(S)n1)=O)C2 62154,c1(C(=O)NCCOCCNC(c2c(C)nc(N)cn2)=O)cccc2scnc12 62155,c1(C(=O)NCC2N(C(c3cc(SC)oc3)=O)CCCC2C)n[nH]c2c1CSCC2 62156,CC1CCCC(C(N2CC3C(CNC(=O)C=Cc4cnn(C)c4)C3C2)=O)C1 62157,Cc1ccc([N+](=O)[O-])c(C(=O)NCC2CC3CCC2N(C(C2CCOC2)=O)C3)c1 62158,CC1CC(=O)NC(C(=O)NCc2cccc(NC(=O)C(F)(F)c3cncs3)c2)C1 62159,N1(C(COCCCCC)=O)CCCCC2(CCN(C(=O)C3=C(C)CCCC3)C2)C1 62160,CC(O)CCN=c1ccc(Br)c(S(=O)(=O)N2CCC(N(C)C)(C(N)=O)CC2)[nH]1 62161,c1(NC(C2(F)CN(C(=O)C(Cl)(Cl)Cl)C2)=O)ccccc1N1CCCC1 62162,c1(CC)cc(F)c(F)cc1Nc1cc(OC)cc(C)c1O 62163,C12(C(=O)N(c3ccc(C#N)cn3)c3ccc(NC(C)=O)cc3)CCC(CC1)C2(C)C 62164,c1(C(C(C(=O)NC(c2ccc(F)cc2)CC(=O)OCC)C)C)c(C)noc1C 62165,C1(C(N2CC(CN(C(CCCC=C)=O)C)OCC2)=O)C(C)(C)CCCC1(C)C 62166,Cc1nc(C(=O)NC2(C(N3CCC(CCF)CC3)=O)CCCC2C)c(C)o1 62167,c1(N)cccn1CC.C1(OC(NOCC(=O)NC2C(N(C(C)=O)C)CC2)=O)CCCCC1 62168,C(C(O)C(F)(F)F)NC(c1cncc(OCCN2CCCCC2)c1)=O 62169,N1(CCc2cn(C(C)CNC(=O)CCc3cn[nH]c3)nn2)CCN(C)C(=O)C1 62170,C1(C(N2CC(OCCNC(C(C)N(C)C)=O)C2)=O)COCCOC1 62171,c1(C(c2nnnn2C)NC2(CO)CC(OC)C2)ccc(NC(C)=O)cc1 62172,N1(C(CC2C(C)(C)C2)=O)CC(NC(=O)Cc2csc(-c3ccco3)n2)C(O)C1 62173,C1(CNC(Cn2c(C(C)C)ncc2)=O)CN(C(=O)CCn2ccnn2)CCCO1 62174,CC1CC2(CCN(C(=O)CCC3CC3)CC2)CN1C(c1ccc(S(C)=O)cc1)=O 62175,C=CC(C)(CCOC)C(=O)NC1CCN(C(=O)CCCSC)CC1C(N)=O 62176,c1(C(N2CCCCC(N(C)C(C3COCC3(C)C)=O)C2)=O)cc2n(n1)CCCN2 62177,c1(C(=O)OCC)sc2ccncc2c1OC(c1ccc(C(F)F)o1)=O.C1C(=O)O1 62178,Cc1ccc(C(=O)NC(C)CCN(C(=O)CCc2cnn(C)c2)C)nc1 62179,N1(C(CC(C=C)CC)=O)CCC2C(CCC2)C(CNC(c2cncnc2C)=O)C1 62180,C1(NC(CC)=O)(CNC(=O)CNc2nc(C)cs2)CCCCC1C 62181,c1(C2C(c3ccccc3)CCN(C(CC(C=C)(C)C)=O)C2)cccc([N+](=O)[O-])c1 62182,C1(C(=O)NCCN(C(=O)C=CCO)CC)CCCC1N(C)C 62183,OCC(CN=c1nc2sccc2c(N2CCOCC2C2CC2)[nH]1)C1CCCCC1 62184,Cc1cc(Cl)ncc1NC(=O)C(C)C(C)NC(c1ccn(CO)c1C)=O 62185,C1(C(N(CCOCCNC(C(C)=CC2CC2)=O)C)=O)CC(C2CC2)C1 62186,Cc1cc(=O)oc(C)c1C(=O)NCCC1CN(C(c2cnc3n2CCCC3)=O)C1 62187,C=CC(CCC)CC(=O)N1CCCC1CCCNC(c1cc2n(n1)CC(F)C2)=O 62188,Cc1nc(NC(C2CC2(C)C)=O)sc1C(=O)NC(c1cccc(C(F)(F)F)c1)C 62189,CCCCN=C(NCC(c1cccc(F)c1F)(C)C)NC1CN(C2CCCC2)C1 62190,C1(CNC(C2(CC#C)CCOC2)=O)CC2CCC1N2C(=O)C(C)(CC)CC 62191,C1(CC(=O)NCC=CCNC(C(C)OCCC(C)C)=O)CCNC(=O)C1 62192,CCCC(C(=O)OC)C(=O)NCC1(C2(O)CN(C(=O)C=Cc3cnc[nH]3)C2)CC1 62193,c1(N(CC)CC2CC(=O)N(C)C2)nnc(-c2cccnc2)n1CC(C)C 62194,Cc1nc(C=CC(=O)NCC2(C)CC(NC(C3CCC3)=O)C2)[nH]c1C 62195,c1(CC)cc2c(NC34CCCCC3CN(C(=O)CSC(C)C)C4)nc(C)nc2s1 62196,C#Cc1ccc(F)cc1C(=O)NC1CN(C(c2ccc(F)cc2C#N)=O)CC1C 62197,N1(C(C(CCC2CC2)NC(C(CC(C)(C)C)O)=O)=O)CCC(C2(O)CC2)CC1 62198,N1(C(=O)NCC(c2cc(F)ccc2OC)C)CC(C)(C)C(O)C1(C)C 62199,C1(C)(C(=O)NCC(C)(C(C)C)NC(C(CCC)=CCC)=O)CCCCC1(F)F 62200,c1(C(=O)NC2CN(C(C(CC=CC)C)=O)CC23CC3)cc(C)c(C#N)cn1 62201,N1(C(CCC)=O)CCC(C(C)(C)OC(C2CCOCC2)C(=O)NCC)C1 62202,C1(NC(c2c(O)ncc(C(C)C)c2)=O)CCC2CCN(C(=O)C=CCO)C1C2 62203,CCC(CC)C(=O)NCCC1CC(C(=O)OCC(=O)NCCn2cccn2)C1 62204,N1(C(C=Cc2occ(C)n2)=O)CC2CN(C(=O)COC(F)F)CCC2(CO)C1 62205,C(C1CCCN1C)=CC(=O)N(C(C)C(=O)N1CC(F)C1)C1CC1 62206,C(c1ccc(OC)c(Cl)c1)=CC(=O)NCC1CCC(NC(C(CC)COC)=O)C1 62207,c1(C(N2C(C(=O)Nc3ccc(N(C)C)nc3)CCC2)=O)ccc(C#N)cc1O 62208,C(=O)(N=c1cccn[nH]1)C1(c2ccccc2)CCN(C(c2ccsc2Cl)=O)CC1 62209,c1(NC(=O)NCCOc2ncccc2Cl)ccc2c(c1)CCCO2 62210,C1(NC(C(C)OC2CCCC2)=O)CN(CCOCc2ccn(C)n2)CCC1(F)F 62211,N1(CC)C(=O)NC(c2ccc(Br)c(OC)c2)C(C(=O)N2CC(C)CC(C)C2)=C1C 62212,N1(C(CCC)=O)CC2CCC1C(CNC(=O)CCN1CCC(O)CC1)C2 62213,N1(C(=O)Cn2cc(Cl)cn2)CCCC1C(C)(C)CNC(=O)COCCN(C)C 62214,S(=O)(=O)(c1ccc2onc(Cl)c2c1)C(=O)NCCC1CCCC(C)(C)O1 62215,N1(C(C(C)=CC)=O)CCC2(NC(c3sc(N4CCCCC4)nc3Cl)=O)CC2C1 62216,CC1CCCN(c2ccc(Cl)cc2)N1C(C1CC(OCCF)C1)=O 62217,c1(C(=O)OCC)cc(Br)ccc1NC(C1CN(Cc2cc(C)[nH]n2)CCC1O)=O 62218,c1(C(N2C(CN(C(c3c(CC)nc[nH]3)=O)C)CCC2)=O)cnc(CN(C)C)nc1 62219,C1(CNC(C(C(C)C)OC)=O)CC2CCC1N(C(C13CCCCC1C3)=O)C2 62220,c1(CC(=O)N(CCCNC(=O)CCN(C)CCO)CC)csc2ccc(Cl)cc12 62221,C(CC(C(=O)N1CCCC1NC(=O)CNC(C)=O)NC(=O)OC(C)(C)C)SC 62222,c1(C(=O)NCC(C)NC(C(C(CC)C)OC)=O)c(Cl)cc(CO)cc1Cl 62223,C(=O)(CCCCC(F)(F)F)NCC12CCC(NC(CC3(C)CCC3)=O)(C1)CO2 62224,CCCC(C(O)C(=O)Nc1ccc(O)nc1)NC(=O)COCC1CC1 62225,n1(CC)c(C)nn(CC(=O)NCCCNC(c2ccc(C(N)=O)cc2)=O)c1=O 62226,C(=O)(C(F)(F)C(F)F)NCCCC1CCN(C(C=CC(C)(C)SC)=O)CC1 62227,CCC(CN1CC(=O)N(CC(C(C)(C)C)N(C)C)C1=O)(CC)C(=O)OC 62228,N#Cc1c(CCNC(N2CCC3CCCC23C(=O)OC(C)(C)C)=O)cccc1F 62229,Cc1nc2c(n1C)CCCC2C(=O)N(C(C)C)C(C)C1CC1 62230,C1(O)(c2cn(CCN3CC(O)(C(C=O)F)C3)nn2)CCSCC1.CNS(N)(=O)=O 62231,C1(NC(=O)CCC2CC2(F)F)CCN(C(c2ccnnc2O)=O)CC12CCC2 62232,CC(C)CC(CC(=O)NC1(CO)CCC(C)C1)NC(C1CC2(CCC2)C1)=O 62233,c1(C(C)(C)C(=O)NC(CNC(=O)CC2CC=CCC2)CO)ccc2c(c1)OCO2 62234,CC1CCC(OCCNC(=O)C(O)C(C)c2ccccc2F)CC1 62235,c1(OC)ccc(C(=O)N(C)CCNC(C2(C)CCCC2(F)F)=O)c(N)c1F 62236,C1(CNC(C2CC(C)C(C)CC2)=O)C(C2CC2)CCN1C(c1cnc(N)cn1)=O 62237,c1(C(=O)NC2(CC#C)CC2)cc(Cl)cn1C.C12(CC(CO)C1)C(=O)N2 62238,N1(C(=O)CCOC2CC2)CCCN(C(C2(C(F)(F)F)CC3CC3C2)=O)CC1 62239,c1(CC(C)N(C(c2ncccc2C)C(=O)NCC)C2CC2)ccc(C)cc1 62240,N1(C(CSc2n(C)ccn2)=O)CCC2(NC(=O)Cc3ccnnc3O)CC2C1 62241,c1(N(CCCC)C)nc2ccccc2c(=NC2CCc3ncccc3C2)[nH]1 62242,N1(C(=O)CNc2ccc(C3CCCCC3)cn2)CC2CCC1CO2 62243,C1(C(=O)OC)C(C)CCCN1Cc1c(-c2cccc(O)c2F)cnn1C 62244,C1(CNC(CNC(CNC(=O)NC)=O)=O)C2CCCCC12 62245,CC(C)S(=O)(=O)C(C)C(=O)NC1(CNC(c2cc3c(nc2O)CCC3)=O)CC1 62246,c1(C(=O)NC(CNC(CNC(=O)NC)=O)C)cc2oc(Cl)cc2[nH]1 62247,C1(C)(CC(=O)NCC(C(=O)NC(C)Cc2cnn(C)c2)O)CCCCC1 62248,c1(CC)cc(F)ccc1C(=O)NCC(C)(C)CNC(=O)C=CCCCN=[N+]=[N-] 62249,C1(CNC(c2ccc(CSC)o2)=O)CN(C(=O)C(C)C2CC2)C2(CCC2)C1 62250,c1(OC)cncc(C(=O)NC2CCCC(CC(=O)N(CC(C)(F)F)C)C2)c1 62251,C1(CC(=O)NCC(CNC(C2N(C(=O)NC)CCC2)=O)O)C(C)(C)C1(C)C 62252,c1(OCCN(CC(=O)N)CCOCC(F)(F)F)ccc(Cl)cc1.C1(C(=O)N)CNC1 62253,C1(C2CCC2)(CNC(COC2CN(C(C(C)(C)OCCC)=O)C2)=O)CC1 62254,n1(CC(=O)NC2(COC)CN(C(=O)C(C)(C)F)C2)ccc(C)cc1=O 62255,c1(C(=O)NC2(CNC(C3(C)COC3)=O)C(C)CCCC2)cc2c(nn1)OCCS2 62256,c1(C(N(CCCCN(C(C(C)C2CCOC2)=O)C)C)=O)ncccc1N 62257,c1(-c2cn(C(Cc3ccc(F)cc3)NC)nn2)cc(F)c(F)c(F)c1 62258,Cc1cc(F)c(C(=O)N(CCCCCCNC(C2COCCN2C)=O)C)cc1F 62259,c1(CC(=O)NCC2(OC)CN(C(C=NOC)=O)C2)sc(C)cc1C 62260,c1(NC(c2ccccc2-c2nn[nH]n2)=O)cc([N+](=O)[O-])ccc1SCCCOC 62261,C1(CCOC)CN(C(=O)CCCC(=O)OC)CCN1C(C1CC(=O)N(C(C)C)C1)=O 62262,c1(N(CC=C)C(C2CCCC2)=O)ccnc(N2CCN(C)CC2)c1 62263,CCC(CC(=O)NCCn1cc(C(=O)Nc2ccc(C)c(O)c2)nn1)C(C)C 62264,N(C1CS(=O)(=O)N(C)c2ccccc21)C(=O)NC(c1cccnc1)CC 62265,Cc1[nH]c2ccccc2c1NC(=O)Cc1ccc(CCC(=O)O)cc1C 62266,CC1(C)CC(C(N2CC=CC2CNC(=O)C=C2CCCCC2)=O)CCO1 62267,N1(C(CCOCC)=O)CC(NC(c2ccnnc2NC2CCCC2)=O)C2CC12 62268,Cc1c(Cl)ccc(C(N2CCCC2C2CCN(C34CC(C3)C4)CC2)=O)c1F 62269,c1(C(=O)NC(C)CNC(=O)C(C)n2cncn2)cccc2c1OCCN2 62270,c1(C(=O)NC(CC)CNC(c2cc(C(C)=O)cs2)=O)ccc2nccc(C)c2c1 62271,C1(OC(C)C)CCC(C)CC1OC(c1ccccc1Cl)CO 62272,C1(C(N2CC(NC(c3c(C)cn(C)n3)=O)C(C)C2)=O)CC2CCC(C1)C2 62273,C(C1c2ccccc2CN1C(=O)OC(C)(C)C)N(C)C.C12(CN(C)C1)C(=O)N2 62274,N1(C(C(F)=CCC)=O)CC(NC(c2c(OC)noc2C2CC2)=O)C(F)C1 62275,N1(C(C(=O)NCCC(F)F)=O)CCc2nc(S)[nH]c2C1 62276,c1(CC)ncc(C(N2CCN(C(c3cnc(=N)[nH]c3)=O)C(C(C)C)C2)=O)c(O)n1 62277,N1(C(C#CC(C)C)=O)CC2COCCC2(NC(c2nccnc2N)=O)C1 62278,C1(C(=O)NC2CC(NC(c3cnn4ncccc34)=O)C2)CC2CCC(C1)C2(F)F 62279,CC(C)C(O)C(=O)N1CC(NC(=O)C=CC2CC2)C(c2ccccc2F)C1 62280,Cc1cc(C(=O)NCC(C)(C)CNC(=O)C(O)Cc2ccc(F)cc2)cc(C)c1 62281,C(=O)(C(C)(C)CCCF)NCCC1CC(NC(C(c2n(C)ncc2)O)=O)C1 62282,C1(CCNC(C(C)SC)=O)CCN(C(=O)CSCC(C)C)C1 62283,c1(C(N2CCN(C(Cc3c(C)non3)=O)C(CF)C2)=O)cn2c(n1)CCC(C)C2 62284,C1(NC(CNS(CC)(=O)=O)=O)CN(C(=O)C(CC)NC(C)=O)Cc2nccn2C1 62285,CC1(C(=O)NC2CCC(NC(=O)CCc3nc(=N)[nH][nH]3)CC2)CCC(=O)NC1 62286,c1(NS(C)(=O)=O)ccc(C(=O)NCC23CC2CN(Cc2cscc2C)C3)c(Cl)c1 62287,Cc1ccc(C(=O)NCCC(C)NC(c2cnc(C(N)=O)s2)=O)c(N)c1F 62288,CC(CCCCNC(C1CCC(N(C)C)C1)=O)NC(C1CC1c1cnc[nH]1)=O 62289,CCCCS(=O)(=O)CC(=O)N1CCC(NC(c2n[nH]c(CC)c2F)=O)C1(C)C 62290,CC1(C(=O)NCc2ccc(C(F)(F)F)nc2)CCN(S(=O)(=O)CCCl)C1 62291,C(=O)(C(C)CCC(C)(C)C)NC(CC)(CNC(c1sc(OC)nc1C)=O)CC 62292,N1(C(C2CCCN(C(C)C)C2)=O)CC(CNC(C2CC(O)C2)=O)C(C)(C)C1 62293,c1(NC(C23CC(C2)C(C(F)(F)F)O3)=O)ccccc1-n1ccccc1=O 62294,CN=c1nc(N(CC(C)C#N)C)[nH]c(=NC(CCO)C2CC2)[nH]1 62295,c1(OC)cc(C(F)(F)F)ccc1C(=O)NC1(C)CC(NC(=O)Cc2ccon2)C1 62296,Cc1nn(CCO)cc1C(N1CC(CNC(C2(C3CCCO3)CCCCC2)=O)C1)=O 62297,C1(C(=O)Nc2ncc(N(C)C)nc2)CC12CCN(C(=O)CCNC(=O)CO)C2 62298,Cc1nc(=NC(=O)CC2CN(C(=O)Nc3ccccc3C#N)CCO2)s[nH]1 62299,Cn1ccnc1C(F)(F)C(=O)NCC1(NC(=O)C(O)C2CCCC2)CC1 62300,c1(C(N(C2CN(C(C3C(C)(CC)C3)=O)C2)C)=O)cc(C2CC2)n(C)c1C 62301,C1(C(=O)NC(C)Cn2cccn2)COCC1NC(=O)Cn1ncnn1 62302,N1(C(c2ccc(C)c(C)c2)=O)CC(C2CN(C(c3csc(Br)c3)=O)C2)C1 62303,C1(C2CCN(C(C3CC3C(N)=O)=O)C2)(NC(Cc2c(C)cc(Cl)nc2)=O)CC1 62304,C1(C(N(C)Cc2cccnn2)=O)CSCCN1C(c1ccn(C)n1)=O 62305,c1(CNC(C2(OC)CCN(C(c3cc(CC)[nH]n3)=O)C2)=O)ccc2c(c1)CC2 62306,C1(CC(=O)NCC(C)(C2CC2)NC(=O)CCCC2CCCO2)CNC(=O)O1 62307,C1(C(=O)NC(CCC)CCC)N(C(c2cccc(F)c2F)=O)CC12CCCC2 62308,CCC(C)(C)CCCC(=O)N(CCCC(=O)NCC1CCCC(C)CC1)C 62309,CN(C)NC(=O)CCC(=O)NCC12CC(NC(C3CC4C=CC3CC4)=O)(CO1)C2 62310,Cc1cnc(C(=O)NC(CNC(c2cncc(N(C)C)c2)=O)CC(C)C)c(F)c1 62311,Cc1cc(C(N2CCC(NC(=O)Cc3ccco3)C23CC3)=O)cc([N+](=O)[O-])c1Cl 62312,CC1CCC(CC(=O)NCC(C)(C)N(C(=O)Cn2cc(C3CC3)cn2)C)O1 62313,c1(C(N2CC(S(C)(=O)=O)C2)=O)cccc2ccc(Br)cc12 62314,Cc1ccc(C(F)(F)F)cc1C(N1CC2CC1CC2CNC(=O)CCC#N)=O 62315,C1(NC(c2c(CC)ccs2)=O)CCC2CCN(c3ncnc4sccc34)C1C2 62316,O=NN1CCCCC1C(=O)NCc1cccnc1CNC(c1ccnc(O)c1)=O 62317,N1(C(C2N(C(CC(C)C(F)(F)F)=O)CC(O)CC2)=O)CCC12CCCOCC2 62318,C1(CC=C)(C(=O)NC2CCC2NC(=O)CCC)CC=CC1.C1CO1 62319,C1(C(N(CCCn2cc(-c3c(C)nccc3)nn2)C)=O)CCn2cncc2C1 62320,C1(OC)CC(C)CN(C(C2CN(C(=O)CC3NC(=O)NC3=O)CCO2)=O)C1 62321,Cc1[nH]c2ccc(Cl)cc2c1C(N1CC(NC(C2CC=CC2)=O)CC(O)C1)=O 62322,N1(C(c2c(OC)nccc2)=O)CCC2CN(C(C3CCCCO3)=O)CC2C1 62323,CCCCC(CC)C(C(=O)Nc1ccc(F)cc1)N1CCCC1C1(C)CC1 62324,Cc1nc(Br)sc1C(=O)NC1CC(CNC(C2CCOC2)=O)C1 62325,C1(O)(CNC(C(C)(CO)OC)=O)CCCN(C(=O)CCC2(C)CC2)CC1 62326,N1(C(C2C(C)(NC(CCC(=O)N(C)C)=O)CCCC2)=O)CCOC2(CCCC2)C1 62327,S(=O)(=O)(c1cc(NCC(C(F)(F)F)OC2CCCC2)ccc1F)NC 62328,C1(C(=O)NC(C(C)(C)C)CNC(=O)C=CSc2ccccc2)CCC2CC1CO2 62329,Cc1nsc(N2CCN(CCCNC(=O)C(C)(C)C3CCOCC3)CC2)c1C#N 62330,N1(C(C=CC(C)C)=O)CCC2(CCC2CNC(=O)CCNC(=O)C=CCl)CC1 62331,C1(NC(c2cnn(C(C)C)n2)=O)CCCN(C(=O)CCOC2COC2)CC1 62332,C1(CNC(c2ccc(CC)nc2C)=O)CC2COCC2N1C(C1(F)CC1)=O 62333,C1(N(C(=O)C(C)c2ncco2)CCNC2CC(CC(=O)OC)C2)CCCCC1 62334,C1(C(=O)NCCC(=C)C)CC(F)(F)CN1C(c1ncsc1C)=O 62335,c1(C(=O)NC2(CNC(c3ccn(C4CC4(F)F)n3)=O)CCC2)ccc(CO)o1 62336,C(=O)(C1=CS(=O)CCC1)N(CCC(C(C)C)NC(=O)COc1ccc(F)cc1)C 62337,N1(C(CCCOCC=C)=O)CC2CC1CN2C(c1ncccc1C(=O)OC)=O 62338,c1(CNC(CC)Cc2nnnn2C2CCCC2)cc(=O)oc2cc(C)ccc12 62339,C=C=CCCC(=O)NCC(C1CCC1)NC(c1ccoc1-c1ccc(Cl)cc1)=O 62340,C1(C(N2CC(CCC)C(Cc3ccccc3)C2)=O)NCCOC1(C)C 62341,c1(C(=O)NC(CC(C)NC(CCCC(C)=O)=O)C)ncn2cccnc12 62342,CC1(CCC(=O)NCCOc2ccncc2)CN(C(c2cnco2)=O)C1 62343,c1(OC)c(C(=O)NCC(C)(C2CC2)NC(c2ccc(CO)s2)=O)csc1C 62344,C1(CC(=O)NCCC2(C(N(CC(CC)O)C)=O)CCC2)CC2(CC2)CO1 62345,C=CCC(C)(C(=O)NC1(CNC(c2ccc(F)cn2)=O)CCCC1)N(C)C 62346,Cn1nc(C(=O)NC(CNC(C23CC(C)(C2)C3)=O)C2CC2)cc1C#N 62347,C1(c2cn(Cc3c(C)cn(C)n3)nn2)CCN(C(=O)CCC(N)=O)C12CC2 62348,C1(C(=O)NC(C)Cn2cccn2)C=CCN(C(C2CCCC(=O)C2)=O)C1 62349,Cc1[nH]nc(CO)c1C(N1CCCC1Cn1cc(COCCN(C)C)nn1)=O 62350,N1(C(C2(C)COC2)=O)CCN(C(C2CCCC2C(F)F)=O)C(CO)C1 62351,c1(CC(=O)N(C)CCN(C)C(c2cocn2)=O)cccc2nonc12 62352,C(=O)(C1CCCc2nn[nH]c21)N1CCC(F)(CNC(c2nc(C)nc(O)c2)=O)C1 62353,N1(CC(C)C)CCN(C(=O)CC(C)(C)C)CC1=O.N12CCCC1C2=O 62354,C1(CNC(C(C2CN(C(C3(C)C=CCCC3)=O)C2)OC)=O)CCCC(=O)C1 62355,N1(C(C(CC)CCO)C(=O)NC)CC2(C1)CN(CC1CCOCC1)CC(C)(C)O2 62356,CCCC(O)CC(=O)N1CCN(C(C2(c3ccccc3)CC2(F)F)=O)CC1 62357,CC(C(F)(F)C(F)(F)F)=CC(=O)N(C)CC1C2CN(C(=O)COC(F)(F)F)CC12 62358,C1(CCNC(CCC#CC)=O)CN(C(=O)CCS(C)(=O)=O)CC(C)O1 62359,C1(C)(C(N2CC(CCCC)N(C(c3n[nH]cc3F)=O)CC2)=O)CCCNS1(=O)=O 62360,c1(C(N2CCN(c3cc(SC)ncn3)C(CO)C2)=O)cc(F)cc([N+](=O)[O-])c1Br 62361,C1(C(N2CC(C)(C)C(c3cc[nH]n3)C2)=O)Cc2ccccc2C(=O)O1 62362,c1(C(=O)NCCN(C(CC2(C)OCCO2)=O)C2CC2)ccc(Br)cc1F 62363,c1(CN(CCCCC)C2CCCC2)cc(C(F)F)cc(Cl)n1 62364,c1(C(=O)NCC(CO)NC(c2ccc3c(c2)CC3)=O)cc2n(n1)CCC2 62365,N1(C(=O)C=C(Cl)Cl)CCCC2(CCN(C(C3(CC(F)F)CCC3)=O)C2)C1 62366,Cc1cc(Cl)c(C(N2CC(NC(=O)CC3CCCN3C(C)C)CC2C)=O)cc1C 62367,C(c1ccccc1)=CC(C(N1CCC(NC(C2(OC(C)=O)CC2)=O)C1)=O)C 62368,C1(COC)(NC(c2sccc2F)=O)CCN(C(=O)CC2(O)CCOCC2)C1 62369,N1(C(C(C)S(N)(=O)=O)=O)CCC2CC(NC(c3cc(O)cc(O)n3)=O)CCC2C1 62370,N1(C(C2(CF)CCC2)=O)CCCN(C(=O)CS(=O)(=O)Cc2cccs2)CCC1 62371,C1(C(N2CC(C#C)(C(=O)NCc3ccc(C)c(O)c3)C2)=O)CCC(C)=C(C)C1 62372,CC1CCCC(N(C(=O)CN2CCN(C(C3C4CCC(F)C34)=O)CC2)C)C1 62373,Cc1cc(C(=O)NCC(F)CNC(C2CC(C)(C)O2)=O)nc(C)n1 62374,c1(C(=O)NCCN(C(C2CCCCNC2=O)=O)CC)cc2ccncc2cc1F 62375,c1(C(=O)NC(C)CN(C(=O)C(C)(C)N(C)C)C)nn(C)c(Cl)c1Br 62376,c1(COC)cnc(NC(C2C=CCN2C(C)=O)=O)nc1.c12ccc(cc1)[nH]c2=O 62377,CC1(C)C(NC(c2cccc(OC3CC3)c2)=O)CCN1C(=O)C1CC1 62378,CC1C(NC(=O)CSCc2cccc(Cl)c2)CC2CCC1N2C(=O)CCCC1CC1 62379,CC1(CNC(=O)Cc2sc(S)nc2C)CCCN1C(C1CC12CC(O)C2)=O 62380,C1(CN)CC2CCCC2N1S(=O)(=O)CC1(CCO)CCOC1 62381,C1(C(=O)NC2C(C(=O)NCCn3c(C)nnn3)OCC2)CCOCC1(C)C 62382,c1(CC)ccc(C(N2CCC(O)CC2C(=O)NCC(=O)N(C)C)=O)cc1Br 62383,CC(C)(F)CCC(=O)NCCCNC(c1cc(-c2ccc(Cl)cc2)ns1)=O 62384,C(=O)(C(O)C(C(C)C)OC)NCC(COC)NC(c1cc(C)nn1C(F)F)=O 62385,c1(OC)ccc2[nH]c(C(N3CCSC(C(=O)NCC(C)O)C3)=O)cc2c1 62386,N1(C(C2CC(CNC(c3cc(C)c(C)[nH]3)=O)C2)=O)CC2CC(C1)N(C)C2 62387,C1(CNC(c2ccco2)=O)(CNC(c2nc(C3CC3)cs2)=O)CC1(F)F 62388,N1(C(C(CCC)C(C)C)=O)CC(NC(=O)C(C)(C)CS(C)(=O)=O)CC12CCCC2 62389,C1(NC(CNC(C(C)(C)C)=O)=O)CCN(C(=O)CN2CCCC2)CC1(C)C 62390,C(=O)(CCC(F)(F)CN=[N+]=[N-])N1CC(O)(C(C)NC(c2ccc(C(N)=O)o2)=O)C1 62391,O=C(CCCC(F)(F)F)N1CCC2CN(C(C3Cc4nccn4C3)=O)C2C1 62392,c1(C(=O)NC2C(C)CN(C(=O)C(F)F)CC2)nc2ccc(Br)cn2n1 62393,C1(C(=O)NCC(C)(F)CNC(=O)C(C2CCCCCC2)O)CCc2nncn2C1 62394,c1(C(=O)NCC(C(C)O)O)nn(C)c2ccc(Br)cc12 62395,CCCCC(C(=O)N1CCC(F)C(NC(c2cocc2C)=O)C1)ON=C(C)C 62396,C(=O)(CCCNC(c1cnn(CC2CC2)c1)=O)N1C(CN=[N+]=[N-])CC1 62397,N1(C(CNC(C2CCCN2C(=O)C2CC2)=O)=O)CC2C3CCC(C3)C12 62398,Nc1sc2c(c1C(=O)NC1CCCC1NC(=O)C(=C1CCCCC1)F)CCC2 62399,C(=O)(C(C)(CC)OC)N(CCNC(CC(=O)NCC#C)=O)C.C1C(=O)N1 62400,N1(C(C2(c3cccnc3Br)CC2)=O)CCCCC1c1cn(C2CCCC=C2Br)nn1 62401,Cc1cccc(C)c1C(=O)NCC1CC1C(=O)NCC1CC1c1ccoc1 62402,C1(C(C)C)(C(=O)NCCN(CCc2ccccc2)C(C2C=CCC2)=O)CCCO1 62403,c1(C(=O)NCCCN(CCO)C(C2CCC3CC23)=O)ccc(=NCC2CC2)[nH]c1 62404,Cc1cc(N)ccc1C(=O)NCCNC(C1CC2(C1)CC2F)=O 62405,N1(C(c2c(SC)cn(C)n2)=O)CCC(C)(C)C(CNC(=O)C(C)=CC2CC2)C1 62406,c1(CC)ccc(C(=O)NC(CNC(=O)C(CSC)OC)C(C)C)o1 62407,N1(C(C(CCF)NC(c2n(CC)ccn2)=O)=O)CCSC(C)(C)C1 62408,C1(NC(C2C(CNC(c3cc(-c4ccccc4)no3)=O)C2)=O)CCC(CO)CC1 62409,c1(C(N(C2CN(C(=O)C3=CCC3)CC2(C)C)C)=O)csc(N=S(C)(=O)CCO)n1 62410,c1(C(N(CC(CNC(C2CN(C(C)=O)C2)=O)C)C)=O)cc(-c2cccn2C)[nH]n1 62411,c1(C(N2C(CNC(C(CC=C)N(C)C)=O)CC3(CC3)C2)=O)cc(C)c(N)cc1Cl 62412,c1(N(C)C)cccc(I)c1NC(=O)CNS(=O)(=O)C(F)(F)F 62413,c1(N(C)CC2CCN(C)C2)nc(N(C)Cc2ccsc2)nc2c1SCC2 62414,C(CCCCCC(=O)N1CC(COC)CC1C)NC(C1C(CC)OCC1)=O 62415,Cc1cc(C)n(CCCC(=O)N(C2CN(C(C3CSCC(=O)N3)=O)C2)C)n1 62416,c1(SC(C)C(N2CCN(C(C3(O)COC3)=O)CC2CF)=O)ccc([N+](=O)[O-])cc1 62417,C(CC(C)C)(C(=O)OC(C)=O)ONC(CC1(NC(C2N(CC)CCCC2)=O)CC1)=O 62418,C1(NC(C2CC(C)SCC2)=O)CC2CCC1CN2C(c1sccc1CC#N)=O 62419,N12CC3COCC3(C1)C2.c1(C(=O)O)ncc(C(=O)N(C2CCCCC2)CCO)[nH]1 62420,C1(c2c(C(=O)NCC(=O)NCC)c[nH]n2)CCCCN1C(=O)C(C)C1CCC1 62421,C1(CNC(c2cccc(SCC3CCC3)c2)=O)CCC(N)CCC1 62422,C12CC(F)(F)CN1C(=O)CS2.C1(CC)(CNC(c2cccs2)=O)CCCCC1 62423,c1(C(=O)NCCOC(C)(C)CNC(=O)Cc2ccon2)ccc2nccn2n1 62424,CC(C)(C)C(O)C(=O)N1CC(F)(F)CC1CCNC(C1CCNC1=O)=O 62425,CCCCC(F)C(=O)NC(CN(C)C(c1cnc(C)[nH]1)=O)CC 62426,C1(NC(C(=O)NCC2C(C(N)=O)C2)=O)CC2(O)C1OCCO2 62427,c1(C(N2CCC(C)(NC(C3C(C(=O)OC)CC3)=O)C2)=O)cc(C)nc2ncnn12 62428,N1(C(c2c(C)nco2)=O)CCOC(C)(CNC(c2cccnc2S)=O)C1 62429,c1(CNc2c(C(CC)OC)cccc2)cn(C)nc1OC(F)F 62430,C(C(CC1CC1)C(=O)NCCCC1CCCCO1)NC(c1c(C)occ1)=O 62431,C1(C(N(C(C#C)C2CCC2)C)=O)(CC)CCN(C(C2COCCN2C)=O)CC1 62432,C1(C(N2CC(C3(C)CC3)OCC2)=O)C2CCC(C2)N1C(C12CC(C#N)(C1)C2)=O 62433,Cc1cc(CC(=O)NCCNC(c2c[nH]nc2C(F)(F)F)=O)no1 62434,N1(CCCNC(c2c[nH]c(=N)o2)=O)CCN(C(c2ccc(C(N)=O)o2)=O)CC1 62435,C1(C(C)NC(CSCC(C)C)=O)CN(C(C2CCN2C)=O)CCO1 62436,C(C)(C(C(=O)NCCCCCN=[N+]=[N-])C(C)C)NC(CCCOC)=O 62437,c1(C(N2CCC(C(C)NC(=O)CC3(C#N)CC3)C2)=O)ccc2c(c1)CC2 62438,C1(C(N2CCC(C(CNC(C(CO)N(C)C)=O)O)CC2)=O)CCCCN(C)C1=O 62439,C12(N(C)C)CCC(C(=O)NC3C4CN(C(C5(C#N)CCCO5)=O)CC34)(CC1)CC2 62440,N1(C(C(C)Cn2cccn2)=O)C2CCC1CC(NC(c1cnn(C)c1F)=O)C2 62441,Cc1ccc(Br)c(CN2CC(NC(c3cnc(O)nc3O)=O)C3(CC3)C2)c1F 62442,C1(OCC(=O)NCCN2CCN(C(C3CC3(F)Cl)=O)CC2)CCC(F)(F)CC1 62443,C1(C(=O)NCC2(C)CCC2)CCN(C(=O)Cc2ccncc2F)CC1(C)C 62444,Cc1cccc(CSCCC(C)CCO)c1C 62445,CCC(C)CC(C)C(=O)NC1CCN(C(=O)C=CCN(C)C)CCC1CO 62446,N(C1c2ccccc2CC12CC2)C(c1ccc([N+](=O)[O-])c(C)c1)C(=O)NC 62447,C1(NC(c2cc(CCC)oc2C)=O)CCCN(C(c2nc(CC)no2)=O)C1C 62448,c1ccc2c(c1)OCCO2.Cc1ccc(Br)c(C)c1.C12CC(C1)NC(=O)NO2 62449,N1(CC(=O)N(CCCNC(=O)CSc2n[nH]c(=N)s2)C)CCS(=O)(=O)CC1 62450,Cc1ccc(-c2cnc(NC(=O)NC(C3CCOCC3)CF)s2)cc1Cl 62451,c1(-c2ccc(CN(C3CCOC3)C)s2)ncccc1OCCO 62452,C1(CNC(C2CC(C)SCC2)=O)CN(C)CCN1C(c1cccnc1O)=O 62453,C1(C)(C(N(C2CSC2)C)=O)CCCN(C(=O)CC2NC(=O)NC2=O)C1 62454,c1(C(=O)NC(C(=O)NCCCC=C)CC2CC2)cc(O)ncn1 62455,CC1CN(C(=O)C(O)CC(N)=O)CCC1C(=O)NCCC1CCCC1O 62456,C(=O)(C(C)C(F)(F)F)N1CC(c2cn(OC3(c4ccc(C)o4)CCCCC3)nn2)C1 62457,C(=O)(C1=CCC(C)CC1)N1CCC(CNC(C2CCCC(OC)C2)=O)CC1 62458,c1(CC)nc(C(=O)N(C)CC2CN(C(=O)Cn3cnnn3)C2)n[nH]1 62459,C1(NC(C(c2c(C)noc2C)C)=O)CCC2CN(C(c3ns[nH]c3=O)=O)CC2C1 62460,c1(NC(C(c2ccc(OC)cc2)N2CCCC2CCO)=O)cccc([N+](=O)[O-])c1 62461,n1(CCCOC)cc(CCC2CN(C(=O)CC(C)C3CCCO3)C2)nn1 62462,c1(CC(=O)NCC2(NC(C(C)n3cccn3)=O)CCCC2)cccc(C(F)F)c1 62463,Cc1[nH]c(C(=O)NCC2CCCCC2NC(C2CN(C)C(=O)N2)=O)c(C)c1C 62464,Cc1csc(=NCC(=O)NCC2CC(C)N(C(c3cscc3F)=O)C2)[nH]1 62465,C1(NC(C(C)(C(C)C)OC)=O)CCC2(CCCN2C(=O)CS(=O)(=O)C2CC2)CC1 62466,C(=O)(C(=O)NOC)NCCOCCCNC(C1N(CCC)CCC1)=O 62467,C#CCC(C)(CNC(=O)C(CNC(=O)C(CC1CCCCC1)OC)CC=C)CO 62468,N1(C(C(CC=C)C)=O)C2CCC(C2)C1CNC(c1cccnc1C)=O 62469,c1(N(C(=O)NCCC(N2C(Cc3cnc(C)s3)CCC2)=O)C)ccccc1Cl 62470,c1(OC)ccc(C(=O)NCC2CCCCC2NC(c2n[nH]c(C)c2O)=O)cc1F 62471,Cc1[nH]nc(C(N2CC(C(N)=O)(CNC(=O)C(C)C(C)(F)F)C2)=O)c1[N+](=O)[O-] 62472,N1(C(C(=O)NCCS(=O)(=O)N(C)C)=O)CC(C)(C)CC1c1ccccc1 62473,Cc1noc(Cl)c1CC(=O)NC1CCN(C(=O)CC2C=CS(=O)(=O)C2)C1C 62474,N#Cc1ccc(CN2CCC(CC(=O)NCC=Cc3cccnc3)C2)c(Cl)c1 62475,N1(C(C(C)N2CCCC2)=O)CC=C(CC(=O)NC2CCCC2C(N)=O)CC1 62476,O=C1CC2(C1)CC(C(=O)NCC(CC1CC1)C(=O)NCC(F)CO)C2 62477,CC1(C)CCC(O)(CNC(=NCCN2CCOCC2)NC2C=CCCCC2)CC1 62478,C1(C(N(CC(C)N(C)C(C23CC(CO)(C2)C3)=O)C)=O)CCCCS1 62479,c1(C(=O)NCC(CC=C)NC(C2CC(C)(C)CN2C)=O)ccnc2c1cnn2C 62480,N1(C(c2c(OCC)oc(C)n2)=O)CCC(NC(C2CCS(=O)(=O)N2)=O)C(C)C1 62481,C12(NC(c3c(F)ccc(C)c3)=O)CC(C)(C1)OC21CN(C(=O)CCCCC#N)C1 62482,c1(C(N2C(CNC(c3cc(OC)c(Cl)cc3)=O)CC2)=O)cc2sc(F)cc2[nH]1 62483,N1(CCCNC(=O)Nc2c(C)nn[nH]2)CC(C)OCC1C 62484,N12CCC3(CCN1CC3)C2.Cc1nn(C(C)C)c(C)c1C(=O)NCc1ncc[nH]1 62485,C(=O)(CC1=CCCC1)NCC1(NC(C(Cc2c(C)noc2C)C)=O)CCOCC1 62486,C1(OC)CC(NC(=O)C(F)OC)CN(C(c2csc(=N)[nH]2)=O)C1 62487,c1(OC)ccc(O)c(C(=O)NCC(O)CNC(=O)CCn2ccc(C)n2)c1 62488,c1(C(=O)NCC23CC2CN(C(=O)CCCc2nccs2)C3)ncc2ccccn12 62489,N1(C(C(COC)C)=O)CC(NC(c2[nH]nc(C(F)(F)F)c2C)=O)C(O)C1 62490,c1(OCC2CC2)nn(C)cc1[N+](=O)[O-].C12CCN(C1)C(=O)COCC(=O)N2CCC 62491,c1(C(=O)NCC(C2CC2)NC(c2cccc3[nH]ncc23)=O)coc2c1COC2 62492,CCC(C)(CC(=O)N(CCCNC(c1ccc(O)nc1C)=O)C)C(=O)OC 62493,N1(C(c2c(CNC(COCC(=O)NC)=O)occ2)=O)CCC2CN(C)CC2C1 62494,Cc1[nH]nc2ncnc(N3CCC(NC(=O)CCC(N)=O)C3C)c12 62495,c1(C(=O)NCC2CC(CNC(c3cnc(Cl)s3)=O)CO2)ccc2n[nH]cc2c1 62496,C(CC(N)=O)(C(=O)NCc1cc(C(C)C)n[nH]1)NC(C(CN(C)C)O)=O 62497,N1(CC(=O)NCC=CCN)CCN(CC2CC2)CC1.CCC1C(=O)C(=O)S1 62498,C1(CN(C)C(C2CCCCC2)=O)CCCN1C(=O)CCCc1nccs1 62499,c1(CC)cc(F)ccc1CC(=O)NC1(C)CC(NC(C2CCCN2C)=O)C1 62500,N1(C(CCC(C)SC)=O)CCC2(CC1)CCN(C(C1(S(N)(=O)=O)CCCC1)=O)C2 62501,C1(=O)C(F)CC(C)(C)N1.CC(C)C(C)(O)CN1CC(N2CCNC2=O)C1 62502,Cc1ccc(C(=O)NCC(C)(C)OCCNC(=O)CC2CC(=O)NC2=O)cc1F 62503,C1(CNCCC2(CS(=O)(=O)N(C)C)CCC2)CC(=O)N(C2CC2)C1.C1(N)CC1 62504,n1(CC(N2CCC(F)(c3cn(C4CCOCC4)nn3)C2)=O)ncc2c1CCCC2 62505,C1(NC(=O)CCOCCNC(C2CC=CCC2)=O)CCCCC12CCC2 62506,CCCCC(O)CC(=O)NCC1CCN(C(=O)CCc2ccc(=N)[nH]c2)C1 62507,c1(C(=O)NCc2occ(C(=O)NCC3C(C)OCC3)n2)ccc(O)nn1 62508,O=[N+]([O-])c1ccc(Br)cc1-n1cc(CNCC2CCCCC2)nn1 62509,c1(C(N2CCC(CN(C(C(CC#C)O)=O)C)CC2)=O)cccn2nnnc12 62510,CC(c1ccsc1)=CC(=O)NC(C)(C)C(C)NC(=O)CC(C)n1ccnc1 62511,c1(COC)nc2cccc(C(N3CCSCC3C(=O)O)=O)c2[nH]1 62512,c1(N2CCC(C(C)NC(Cc3scc(C)n3)=O)CC2)nn(C(C)C)cc1[N+](=O)[O-] 62513,Cc1cc(F)ccc1NC(=O)C(=O)NC(c1ccccc1F)C 62514,c1(C(=O)Nc2ccc(OC(C)C(=O)N(C)C)cc2)cc(Br)c2occc2c1 62515,N1(C(c2n(CCC)ncc2)=O)CC2CC2(CNC(c2nn(C)cc2C)=O)C1 62516,c1(C(=O)NC2CC(CNC(CC3C(C)=NOC3=O)=O)C2)cc(N(C)C)ccc1F 62517,c1(C(=O)NC(CC)CN(C)C(C2(CC(=O)OC)CC2)=O)cnc(O)c(F)c1 62518,CC1CN(C(=O)NC23COC(C2)C(C(c2ccccc2)C)C3)CC1(C)C 62519,c12ccc(cc1)s2.C=C=CCC(=O)NCCN(C)C(c1coc(C(=O)OC)n1)=O 62520,C1(NC(c2c(C)nccn2)=O)CCC2(CC1)CN(C(C1CC3(C)CC1CO3)=O)C2 62521,Cn1cc(C(=O)NCC2CCCC2NC(=O)Cc2cn(C)nn2)n(C)c1=O 62522,c1(C(N2C(CNC(C3N(CC)CCC3)=O)(CO)CCC2)=O)n[nH]c2c1COCC2 62523,N1(C(C(C)OCC)=O)CCn2cccc2C12CCCCC2 62524,C12CC(O)CN1C2=O.c1(NC)scc(CC(C)C)c1C=O.C(=O)(N)NC 62525,Cc1ccccc1OCCC(N1CCCC(NC(=O)C(C)(O)C2CC2)C1)=O 62526,Cc1c(NC(C2CCC(C(C)C)N2C(c2c[nH]ccc2=O)=O)=O)cccc1CO 62527,c1(OC)cc(C)ccc1C1CN(C(=O)C(C)CN(C(=O)C2=CCCC2)COC)C1 62528,Cc1ccc([N+](=O)[O-])c(N(CC(=O)NC=O)C)c1.C(=O)CC1CCC1 62529,C1(COCC(=O)NCC(CNC(C2(CC=C)CCC2)=O)O)CCCOC1 62530,c1(CN(C)C)ccc(C(=O)NC2(C)CCN(C(C3CC34CC4)=O)C2)nc1 62531,N1(C(C2N=C(C)SC2)=O)CCN(C)C(CNC(=O)CC=Cc2ccccc2F)C1 62532,C1(C(=O)NC(CC=C)CNC(=O)Cc2cncn2C)CCCCC1O 62533,C1(C(=O)NCC(C)CNC(=O)C(C)SC(F)(F)F)CN(C)CCN(C)C1 62534,O=S(=O)(c1ccccc1)C1CC(NCc2cccc(N3CCCC3=O)c2)C1 62535,c1(C(=O)NCC2CC(NC(c3nc(C(C)=O)sc3)=O)C2)ccc2cncn2c1C 62536,N1(C(c2cccc(C)c2)C(=O)NCCCC)CC(O)CC2(CCCC2)C1 62537,C1(NC(C=CC(C)(C)NC(C(CSC)O)=O)=O)CCCCC12CC2 62538,c1(OC)cc(OC)nc(C(N2C3CCC2C(CNC(=O)CC2=CCCC2)C3)=O)n1 62539,c1(C(=O)NC(C(C)NC(CSc2ccc(OC)cc2)=O)C)cccc2nncn12 62540,c1(C(N(CCCN(C(c2c(CC)[nH]c(=N)s2)=O)C)C)=O)cc2occc2[nH]1 62541,C1(C(=O)NCc2c(C)cccc2)CCC(C)(C)N(C(C2(C)CCCCCC2)=O)C1 62542,C1(NC(c2c(N)nccn2)=O)CC12CCN(C(c1ncccc1Cl)=O)CC2 62543,CCC(CC(F)F)C(=O)N(CCCOCCN(C)C(c1cc(C)cc(C)n1)=O)C 62544,CCCC(C)C(=O)N(CC(N1CC(CC)(CO)C1)=O)CCC 62545,C1(OCC(=O)NCC2(F)CCN(C(CNC=O)=O)C2)CCC(F)(F)CC1 62546,c1(CC)cc(C)c(C(N2CCC(CN(C(=O)Cc3csc(Cl)n3)C)C2)=O)o1 62547,Cn1nc(Br)c2ncnc(NC3CC(NC(=O)CC45COC(C)(C4)C5)C34CCC4)c12 62548,c1(C(CC(=O)NCCCOC)NC(c2nccn2C)=O)ccc(C#N)cc1 62549,CC1CN(C(c2cnn(CC(F)(F)F)n2)C(=O)NC2COC2)CC2(CCC2)O1 62550,c1(NC(C2CC(NC(C3(C)CCC3)=O)C(O)C2)=O)ccc(O)c(Cl)c1 62551,C(N=c1nc(OC)[nH]c(N2CC3CC2CS3=O)n1)C1(CC)CCC1 62552,C1(CC(C)C)CCN(C(C2(C(C)C)CCCN2C(=O)CC2CCC(=O)N2)=O)CC1 62553,C(=O)(CCC(=O)NN(C)C)NCCC(C)NC(c1nccc(COC)c1)=O 62554,C1(O)(CCNC(C=CC)=O)CCCN(C(=O)C(C)(C(C)C)OC)C1 62555,c1(C(N2CC(O)(CN(C(CC3C(C)C3)=O)C3CC3)C2)=O)snc(Cl)c1Cl 62556,C1(C(N(CCCCCCNC(c2c(C)noc2C)=O)C)=O)CCN(C)S1(=O)=O 62557,C1(OC)CC(CNC(C2(C(F)F)CC(O)C2)=O)N(C(c2cc[nH]c2)=O)C1 62558,c1(C(=O)NC(CC(C)C)CNC(C2(C#N)CCC2)=O)cc(Cl)cc2ccncc12 62559,N1(C(CCc2cnc(C)s2)=O)CCC2C(C1)CN2C(=O)COCc1ccnn1C 62560,C=C1CC2CCC(C1)N2C(C1CCC(C)CN1C(=O)CC1CC(OCC)C1)=O 62561,N1(C(c2c(C)nc3ccccn32)=O)CCC(C2CCN(CC(C)O)C2)CC1 62562,C1(C(C)C)CCC(NC(=O)C(=O)NC(c2cccc(Cl)c2)C)C(=O)N1 62563,n1(CC)nncc1S(=O)(=O)N1CCOC(c2ccccc2)C1c1ccccc1 62564,C=CCS(=O)(=O)CCNC(=O)CSCc1nnc(-c2ccccc2Br)o1 62565,CC(CC(N)=O)C(=O)NCC(=C1CN(C(C2CC2C(F)(F)F)=O)C1)F 62566,C1(C(NOCCCC)=O)C(C)OCCN1C(=O)CCCN(C)C(C)=O 62567,C1(SC)CN(C(=O)CCCN2CCCCC2)CC1NC(C1CCS(=O)CC1)=O 62568,CC(C)(C)C(CNC(=O)CC1CC2CC2C1)NC(c1cccc(C(F)(F)F)c1)=O 62569,c1(C(=O)NCC(C)(CO)NC(COC(C)=O)=O)cnn2cccc2c1 62570,N1(C(C2(COC)N(C(c3ccc(CC)[nH]3)=O)CC=C2)=O)CC(C)(C2CCC2)C1 62571,c1(C(=O)NC(CCCC)CNC(=O)C(C)(C)n2cnnn2)nc(OC)ccc1C 62572,C1(C(=O)NCC2(NC(C(C)O)=O)CC3CCC2CC3)COc2ccc(F)cc2C1 62573,c1(CNC(=O)NCCCCCl)cc(O)nc(O)n1 62574,c1(C(N2CCC(N(C)C(c3ccc[nH]3)=O)C2)=O)cnc(C2CC2)nc1O 62575,c1(C(=O)NCCOC2CCN(C(c3c(C)nn[nH]3)=O)C2)cnc(O)n(C)c1=O 62576,C1(CC(N2CCC(C)(CNC(C3C(=C)C3)=O)CC2)=O)CCC2(CCC2)CO1 62577,Cc1cc(NC(C)C)cc(-c2cncc(C(=O)Nc3ncc(C)cc3I)n2)c1 62578,Cc1nc[nH]c1-c1cc[nH]n1.C1(C(=O)N(C2CC2)C)(C)CCOC1.C1C(=O)NC(=O)N1 62579,N1(C(C(CC)(C)CO)=O)CCC2C(C1)NC(=O)CN2C(=O)C(CO)OC 62580,c1(C(N(C)CC2N(C(CC(C)C(F)F)=O)CC(F)C2)=O)ccc2c(c1)CCCC2 62581,CN1CCC(O)(C2(C(=O)NC3CCCC3CNC(=O)CS(C)(=O)=O)CC2)CC1 62582,Cc1nc(CNC(c2ccc(CNC(c3csc(F)c3)=O)nc2)=O)sc1C 62583,CC1CN(C(c2cc3ccccc3o2)=O)CCCN1C(c1cnc(N(C)C)o1)=O 62584,N1(C(c2cncc(Cl)c2Cl)C)CCCC2C(C(c3n(C)ncc3)(n3cncn3)CC)CC12 62585,C1(N(C(CSCC#C)=O)C)CCCCN(C(=O)CSCCC)C1 62586,C(=O)(C(F)C(C)(F)F)OCCn1cc(C(=O)NCC(C)(C)N(C)C)nc1 62587,N1(C(c2cn(CC3CC3)nn2)C(N2C(CC)CC2)=O)CCOCC1Cl 62588,N1(C(c2c(CC)non2)=O)CCC12CN(C(c1c(C(F)F)cccc1N)=O)C2 62589,c1(OCC)ccc(C(=O)NC2(COC)CCN(C(=O)C(C(C)C)OC)C2)cn1 62590,N1(C(C2CC(=O)OC2)=O)CCOC2CCN(C(c3cc(Cl)ccc3Cl)=O)CC12 62591,C1(O)(CNC(C(CC)OCC)=O)CCN(C(C2(c3ccnc(Cl)c3)CCC2)=O)C1 62592,C12CN(C(=O)NC(C)(C)C)CCN1Cc1cccnc12.S(=O)(=O)(CCCC#N)NC 62593,c1(C(=O)NC(C)(C)CCNC(C2CCS2(=O)=O)=O)ccc(C(O)CF)cc1 62594,N1(C(CN2CCN(C(C3(COC)CCC3)=O)CC2)=O)CCN(CCO)C(=O)C1 62595,S(=O)(=O)(c1cc(Br)cnc1N)N1CCN(C(C)C2CC2)CC1 62596,Cc1cc(F)cnc1C(N1CCCC(CNC(c2cn(C)ccc2=O)=O)CC1)=O 62597,CC1CC(CNC(=O)C(C)(C)c2ccccc2)CN1C(=O)CCNC(N)=O 62598,c1(OC)cc(F)c(C(=O)NC2CC(O)CN(C(=O)COCCF)C2)cc1N 62599,C(CCCC(=O)N1C(CNC(C2CC2CC)=O)CC2CC12)OCCC=C 62600,C1(NC(c2ccccc2)=O)CCCCC12CCCN(C(=O)COCC(F)F)C2 62601,c1(C(=O)NCC2N(C(CCCOCCOC)=O)CC2)ccc(C)c(OC(F)F)c1 62602,C#Cc1ccccc1C(=O)NC1CC1.C(C(=O)N(CCNC(C1CC1)=O)CC)S 62603,N1(C(C(C)OC(=O)Nc2ccccc2)=O)CC2C(C(c3cc(C#N)cs3)=O)C2C1 62604,O=C1CCc2c(C(N3CCC(CCNC(C4CCCO4)=O)C3)=O)cccc2N1 62605,C(=O)(C(C)(O)CC(C)C)NC(C1CCCN(CC=C)C1)C 62606,Cc1cc(C(=O)NC(C(C)NC(=O)Cc2c[nH]nc2O)C(C)C)c(O)nc1C 62607,C1(CCOC)(C(=O)NCc2cccs2)CCN(C(C2CC2C(F)F)=O)C1 62608,Cc1ccoc1CC(=O)N(CC)C.c12ccnn1CCN(C)CC(CC)C1CCN1C2=O 62609,C(=O)(C(C)(C)CC(C)(C)C)NCC1(C)N(C(C2ON=C(C)C2)=O)CCC1 62610,c1(C(=O)NC2C(CNC(c3cnn(CC)n3)=O)CC2)ccc(Cl)cn1 62611,c1(OC)ccc(CC(C)C(=O)NCC(C)(C)CNC(C2(C)CC2(C)C)=O)cc1 62612,C(=O)(CCCS(C)(=O)=O)N1CCC(C)(CN2CC(NC(CC(CC)SC)=O)C2)C1 62613,N1(C(c2ccncc2)=O)CCC2C(CCN2C(c2cccc3scnc23)=O)C1 62614,C1(CNC(C2CCC(N(C)C)C2)=O)(NC(=O)C2=CCCSC2)CCCCCC1 62615,C1(C(C(=O)NCCOCCNC(C(n2ccc(C)n2)C)=O)=O)CCCCCCC1 62616,c1(CC(=O)N(CCN(C(C)C)C(C2CCCCC2C)=O)C)ccc(O)cc1 62617,c1(NC(C2CC(=C)CN2C(=O)CCc2ccc[nH]2)=O)ccc(OC)nc1Br 62618,n1(CCC)cc(C(=O)NCCCCCNC(=O)C(C2CCC2)OC)nn1 62619,c1(CC)c(NC(c2ccn(CCN(C)C)n2)=O)ncnc1Cl.C12CCN(C1)C2 62620,N1(C(CC(CCC)O)=O)CC2CC1CCC2NC(=O)C(F)(F)C(C)O 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62656,C(=O)(C(F)C(C)C)NCC(c1ccccc1)CNC(c1nc(NC(C)=O)sc1)=O 62657,CC1CCc2onc(C(=O)NCC(C)(C(=O)O)c3ccccc3)c2C1 62658,c1(CC(=O)NC2CC(N(C)C(c3cnc(O)n3C)=O)C2)cnn2c1OCCC2 62659,CCC(CC)(CCNC(C1CC2(CCO1)CC2)=O)NC(C1C(C)(C)C1(F)F)=O 62660,S(=O)(=O)(c1ccncc1)NC1CCC(NC(c2ccccc2Cl)=O)C1 62661,C1(C#N)(NC(c2ccnn2C)=O)CCN(Cc2c(SC)cccc2)C1 62662,C1(C(=O)NCCN(C)C(c2ccnn2-c2ccncc2)=O)(CC)CCOC1 62663,N1(C(C(=O)N(C)C)=O)CCCCC1C1(C(=O)N(CC(F)F)CCO)CC1 62664,c1(C(N(C)CC2OCCN(C(C(CCC)C)=O)C2)=O)c(C)nn(C)c1C(F)F 62665,N1(C(c2ccn(CC)n2)=O)CCC(C(F)CNC(c2nn(C)cc2Cl)=O)CC1 62666,C1(NC(c2cccc(C(N)=O)n2)=O)CC(F)CN(C(c2scnc2C(F)F)=O)C1 62667,c1(C(=O)NCCSCC(=O)N(C(CC)C2CC2)C)ccncc1Cl 62668,C(CCN(C)C)(C=O)N.C(C)(C)(CCCO)NC(CC(=O)N(C)C)=O 62669,N1(C(CC(C)OC)=O)CCC2(CC1)CC(NC(=O)C=C(C)C(C)C)C2 62670,N1(C(Cc2c(C)occ2)=O)CC(O)CCC1C(=O)NCCSCC(C)C 62671,C(=O)(C1CCCc2nc[nH]c21)NCCCNC(c1c(C)n(C2CC2)cc1)=O 62672,c1(OCC)cnc(C(=O)NCCC2CN(C(=O)C(C)COC)CCO2)cn1 62673,CC1CCCCN1CC(=O)NCCCCN(C)C(c1cccc(CC2CC2)c1)=O 62674,N1(C(C(CC=CC)C)=O)CCN(C(=O)COc2ccc(SC)cc2)CC1C(C)C 62675,Cc1nc(C=CC(=O)NCCCN(C(C2CCC2(F)F)=O)C2CC2)cs1 62676,c1(C(N(CCNC(C(C)NC(CC)(C)C)=O)C(C)C)=O)sccc1Br 62677,c1(OC)ncc(C(=O)NCCCn2cc(-c3cccnc3O)nn2)c(C)c1Br 62678,c1(C(N(CC(=O)NCC(=O)NC)CC)=O)ccc(C#N)n1C 62679,N1(C(c2cnn(C)c2Cl)=O)C2CCC(C2)C1CNC(C1(C#N)CCCCC1)=O 62680,CC(C(=O)NN1CCCC1C(=O)N(CCN=[N+]=[N-])C(C)C)=CC1CC1 62681,Cc1cc(C)n(CC(=O)N2CCC2N2CCC(N)CC2)c(=O)n1 62682,CCCC(CCC(C)(C)O)(c1nnnn1CC(F)F)NCCC(C)C(F)(F)F 62683,CCCCCCC(=O)N1CCCCC1CNC(c1c(Cl)cncc1Cl)=O 62684,N1(Cc2c(OC)cccc2)CCC2C1CCCN2C(=O)CCc1cnc[nH]1 62685,c1(NC2CCCN(C(c3n(CCOC)ncc3)=O)C2)ccc(C(C)=O)c(C)n1 62686,CC(C)C(O)C(=O)NCC(C)CC(=O)NCC1CC1(C)C 62687,C1(CC(=O)NC2C(C(=O)Nc3cncc(OC)c3)CCC2)Cc2ccccc2C1 62688,CC(C)(C)CC(O)CC(=O)NC1CCC(NC(=O)Cn2ccnn2)C1 62689,N1(C(Cc2cccc(C)c2)=O)CCN(C(=O)C(C)C2CCC2)C(CCO)C1 62690,N1(C(C(F)OC)=O)CCCC(C2CCN(C(=O)C(C3CCC(=O)N3)C)C2)C1 62691,c1(C(=O)NC2CCCC(C(N3C(C)CC3CO)=O)C2)cn2c(n1)CCC2 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62709,C(CN=C(NCc1cnco1)NCC1CCCCC1(C)C)OC(C)CC 62710,C#CCC(C(=O)NCc1nc(C)cs1)NC(c1sncc1C)=O 62711,C(=O)(C(O)CC(C)C)N1C2CC(NC(c3n[nH]c(C)c3Cl)=O)(C2)C1 62712,c1(NC(c2n(-c3c(CC)cccc3)nnn2)c2ccc(Cl)s2)cc(C)cc(Br)c1 62713,C(=O)(C1CCc2c[nH]nc21)NC1(C2CCN(C(CN(C3CCC3)C)=O)C2)CC1 62714,CCCCC(=O)C(=O)N1CC(CNC(C2(CO)CCOCC2)=O)C(C)(C)C1 62715,N1(C(C2CC(=C)C2)=O)CCN(C2COCC2NC(=O)CC23CCCC2C3)CC1 62716,C1(CNC(c2c(OC)scc2)=O)C(CN=c2[nH]cncc2I)CCC12CCC2 62717,N1(C(C2(C)CCC(C)C2)=O)CC2CCC1CN2C(C1C=CCC1)=O 62718,N1(C(c2c(C)onc2)=O)C2CCC1CC(N(C)C(C1CC(=O)N(C3CC3)C1)=O)C2 62719,C1(OC)CN(C(c2cccn3ncnc23)=O)C2(CCCC2)C1 62720,C1C(=O)N2CCC(O2)C1=O.N1(C(C=C(C)C)=O)C2CCC1CC2 62721,c1(N(CC(=C)Br)C)ccnc(N2CCN(Cc3nc(O)n[nH]3)CC2)n1 62722,c1(C(N2CCC(CCC(=O)NCC3(CCC=C)CC3)C2)=O)cc(C)c(O)nn1 62723,c1(C(N2CC(C)CC(C(N(CCC)CC)=O)C2)=O)c[nH]c2ccccc12 62724,c1(-c2nc(C(CN)OC3CCNC3)on2)cccc(-c2cscn2)c1 62725,N1(C(C(C)CN2CCOCC2)=O)C(C)C2CC1C2NC(=O)C(C)(C)N(C)C 62726,CC(CC(=O)N1CCC(C2CCCN2C(c2ccc(CO)cn2)=O)C1)C(F)F 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63024,c1(C(N2CC(NC(C(C)(O)C(F)(F)F)=O)C(C#N)C2)=O)ccc2nc(Cl)sc2c1 63025,C=CCC(C)(C#N)C(=O)N1CC(C(O)C(=O)NC2(c3nc[nH]n3)CC2)C1 63026,n12cc(nn1)NC(=O)C2C.C(=O)(COCCC1CC1)OC 63027,c1(C(=O)NCCCCCNC(C2CC(C)(C)O2)=O)ccn2ccccc12 63028,N1(C(C(C=C)O)=O)CCCC(C2CCN(C(C3(C)CCCC3C)=O)C2)C1 63029,c1(C(C)(F)F)ccccc1C(=O)NC1CN(C(c2cccnc2O)=O)CC1O 63030,N=S1(=O)CCC2(CCCN(S(=O)(=O)c3nncs3)C2)C1 63031,N1(C(CSCC(C)=O)=O)CCC(N(C(=O)CN2CC=CC2)CC)C1 63032,CCCC(CCC)C(=O)NCC(C)NC(=O)CN(C)C(c1cc2c(s1)CCC2)=O 63033,C=CCC(CN=c1[nH]c(=NC)[nH]c(=NCC(C)n2ccnn2)[nH]1)c1ccccc1 63034,C1(CNC(c2c(C)con2)=O)CC2(CN1C(=O)CNC(=O)C(F)(F)F)CC2(F)F 63035,c1(CC(C)C)cc(C(=O)NC2CCCC2NC(c2ccc(Cl)o2)=O)n(C)n1 63036,C#CC1(N(C)C)CCN(C(C(=O)NCC(F)F)C2CC(CC(C)(C)C)C2)CC1 63037,c1(C(N2CC3C(NC(c4cn(CC)nc4C)=O)C3C2)=O)c(F)cc(N)cc1F 63038,c1(C(N2C(c3cn(C)nc3)C(C)(C)C2)C(=O)NC2CC2)cc2ccc(Cl)cc2o1 63039,c1(C(=O)NCC23N(C(c4c(C)nccn4)=O)CCC2CC3)cc(F)c(Cl)cc1Cl 63040,C1(C(N2CCC(C(C)(C)NC(c3c(C)noc3C)=O)C2)=O)CC2(COCCO2)C1 63041,C1(CNC(=NCC=C)NC(C)CC)CS(=O)(=O)c2ccccc2O1 63042,c1(C(=O)NC(CCCNC(c2c(CC)con2)=O)C)cc(O)c2ccccc2c1 63043,N1(C(CCCCSC)=O)CCCCC2(C1)CN(C(c1[nH]c(C)nc1CC)=O)C2 63044,c1(C(=O)NCC2(F)CC(NC(CC3N(CC)CCC3)=O)C2)ccc(OC)cc1 63045,c1(C(N2CCN(C(C=CCC)=O)C(C(F)F)C2)=O)cn2cc(Cl)cc(Cl)c2n1 63046,c1(C(=O)OC)nn(C)c(SC)c1N=c1cc[nH]c(C2CCC2)n1 63047,CCCCCCC(C)CC(=O)NC(CNC(=O)C(=O)NC(C)C)C1CCC1 63048,c1(C(=O)NCC(C)N(C(CCc2c(C)cccc2)=O)C)cc2c(C)sc(C)c2s1 63049,C1(CCC)(NC(=O)C(F)C(F)(F)F)CCN(C(c2ccc(C(F)F)nc2)=O)CC1 63050,C(=O)(C(CC(C)(C)C)NC(c1ccc(C#N)n1C)=O)N1C(C(=O)OC)C(C)CC1 63051,C1(CNC(c2c(C)sc(Cl)n2)=O)CN(C(c2n[nH]cc2C2CCC2)=O)CCN1C 63052,N12CCC(C(F)(F)CC1)CNC(=O)c1c(OC)ccnc1C2=O.C(C)(C)(C)O 63053,c1(CC)cc(C(=O)OCC2CCC(C(=O)OC(C)(C)C)C(=O)N2)cc(Cl)c1 63054,C1(C(=O)Nc2cn(CCC#C)nc2)CCCN(C(=O)C(C)=C2CCCC2)C1 63055,C(CNC(=O)C(C)SC(F)(F)F)(CCCC)NC(C1(C#C)CCC1)=O 63056,N=c1nc(N2CCCC(n3nccn3)C2)[nH]c(=NCc2cccc(CO)n2)[nH]1 63057,N1(C(CCC(C)(C)F)=O)CC(CNC(C2(S(N)(=O)=O)CC2)=O)N2CCC1C2 63058,c1(N2CCC(CCOC)(NC(C3COC(C)C3)=O)C2)ncccc1[N+](=O)[O-] 63059,c1(OC(C)C(N2CCN(C)CC2NC(=O)CC(C)(C)O)=O)c(F)cccc1F 63060,C1(C(N(CCC)CC2CC2)=O)CCCC1NC(=O)CC1(OC)CCC1 63061,c1(CNC(C2C(NC(CNc3ccc(C)cc3)=O)COC2)=O)cc(F)ccc1F 63062,c1(C(=O)NCC2CC(NC(C(C3CCCC3)OCC)=O)C2)ccn2nncc2c1 63063,c1(C(=O)NC2(C)CN(C(=O)C(F)(F)c3ncccn3)C2)scc(Cl)c1Cl 63064,c1(C(=O)NC2C(C)CN(C(=O)CCCF)C2)n[nH]c2c1CC(C(C)(C)C)CC2 63065,C(=O)(C(C)C(C)(C)c1ccccc1)NCC(CC(C)C)NC(CC(COC)C)=O 63066,C1(NC(C=CSC)=O)CC(OC)CN(C(c2nc(-c3cnn(C)c3)oc2C)=O)C1 63067,C1(NC(C2C=C(C)CS2)=O)COC2(C1)CN(C(c1coc(C3CC3)n1)=O)C2 63068,c1(OCC=C)ccccc1-c1cc(C(=O)N(c2cccc(C)c2)C)n[nH]1 63069,C1(CNC(CC2(C=C)CC2)=O)C2CCC(C2)N1C(=O)Nc1cccc(NCC)c1 63070,c1(-c2c(C(=O)Nc3cccc(NC(=O)OC)c3)nccc2)cc(Cl)c(C)cc1O 63071,C(=O)(CC1COc2cc(O)ccc21)NC1C(n2cc(CCC#N)nn2)CCC1 63072,c1(C(=O)NCC(=C)CCNC(=O)C(CC)NC(C)=O)cc2sccc2s1 63073,C1(C(=O)NC(C(=O)NC(CC)COC)CC2CC2)CCCC(O)C1 63074,c1(C(N2CCC(N(C(=O)COCC3CCOCC3)C)C2)=O)c(Cl)nsc1Cl 63075,C#CCCCCCC(=O)NC1CCC(NC(=O)CC2CCN(C)C2=O)CC1 63076,c1(NC(C(CC)C)CN(C)C)nc(N2CC3CC2C3)nc2c1ncn2C 63077,N1(C(CC(CC)SC)=O)CC(NC(c2conc2C)=O)CC12CCOCC2 63078,N1(C(c2n[nH]c(=N)[nH]2)=O)CCC2(C1)CN(C(C1CN(CC(F)(F)F)C1)=O)CCO2 63079,N#Cc1c[nH]c(C(=O)NC2CN(C(=O)CC3CCC(C4CC4)O3)CC2C(F)F)c1 63080,Cc1ccc(C=CC(=O)NCCN(C)C(C2CN(c3nnnn3C)C2)=O)o1 63081,N1(C(C(C(C)C)OC)=O)CC(C(=O)NCCc2ncccc2F)C(C2CC2)C1 63082,N1(C(CC(CC)(F)F)=O)CC2CCCCC2(CNC(=O)CCc2cnc[nH]2)C1 63083,C#CC(CC(C)C)NC(=O)C(C)(C)NC(C1CCC1COC)=O 63084,C1(C(=O)OC)C2CCC(C2)N1C(=O)Cn1cnc(Br)n1 63085,Cc1ccc(C=CC(N2CCCCC2CCCNC(=O)CN(C)C(N)=O)=O)o1 63086,C(CCCC(=O)NCC1=CCCC1)N(C(=O)C(F)CC1CCOC1)C 63087,CCCC(C)(C)CC(=O)N1CCC(C)(CNC(c2ccnn2COC)=O)C1 63088,CC(C)CCC(F)C(=O)NCCC1CCC(NC(=O)CC2CN(C)C2)C1 63089,C(C)(C(=O)N(O)Cc1cn(C2CCCC2O)nn1)Oc1ccc(C)cc1 63090,c1(CNC(CCC2CC(NC(CCN(C)CC)=O)C2)=O)nc(C)sc1C 63091,N1(C(c2c(C)nc(Br)cc2)=O)CC2(CCN(Cc3cccc4[nH]ccc34)CC2)C1 63092,c1(OC)cccc2c1C(C(=O)NCC1(OC)CN(C(C3CC4CCC3O4)=O)C1)CC2 63093,N1(C(C(C)Sc2nccn2C)=O)CCCC(O)(CN(C)C(c2cnn(C)n2)=O)C1 63094,c1(OC)ccc(F)cc1C(=O)NC1CC(OC)CN(C(=O)CN2CCCC2C)C1 63095,c1(OC)cnc(NC(C2C3CC2N(Cc2cccc(CO)c2)C3)=O)cn1 63096,CCC(C)(C)C(O)C(=O)N1CC(CNC(=O)Cn2ncc(C#N)c2N)C(C)(C)C1 63097,c1(OCC)cc(C(=O)NCC(C2CC2)N(C)C(c2ccsc2C)=O)ccc1C 63098,N1(C(C2(COC)CC=CCC2)=O)CCCC(NC(=O)CSC)CC1 63099,c1(N2CCCC(N(C(c3c(C)snc3)=O)C)CC2)ccc2c(n1)CCCC2=O 63100,C12(C(=O)NCCN(C)C(c3sc(N(C)C)nc3Cl)=O)CCC(F)(CC1)CC2 63101,c1(OCC)ncccc1C(=O)NCCOCCNC(=O)CC1CCC1(C)C 63102,c1(OC)ccc(C(N2CC(C)CC2C(N2CC(NS(C)(=O)=O)C2)=O)=O)cn1 63103,C1(C(C)C)CN(C)CCN1C(C1CC(O)CN1C(=O)CCC1CCCC1)=O 63104,c1(OC(C)C)ccccc1CNCCC(=O)NO 63105,c1(NC(C)CCNC(C2CC3CCCC23)=O)ncccc1C#N 63106,N1(C(CC(=O)NCC)=O)CC2ON=C(CNC(c3cncc(F)c3)=O)C2C1 63107,C1(NC(c2cc(C(N)=O)oc2)=O)CC2CC(C1)N(C(C1CC=CCC1)=O)C2 63108,O=C(C(F)C(F)(F)F)NC1CC2(C1)CN(C(=O)CCc1ccc(F)cc1)C2 63109,N12CC3CCCC3(C1)C2=O.Cc1ccc(NC(=O)C(F)C(F)(F)F)c(C)c1 63110,N1(C(C(C)(C2(C)CC2)OC)=O)CC2C(CNC(C3CCC=CCC3)=O)C2C1 63111,CC1N(C(=O)C(C2CCNCC2)F)CCCC1(C)C 63112,c1(SC)ncc(Br)c(=NC2CC2C(=O)NCCCn2nc(C)nc2C)[nH]1 63113,N1(C(C(C=C)O)=O)CCC2(CC2NC(=O)CC(C)C(F)F)C1 63114,Cc1cnc(C(=O)NC2(C)CCCN(C(C3CCOC(=O)CC3)=O)C2)c(Br)c1 63115,C1(OC)CC(NC(=O)CSCC(N)=O)C12CCN(C(c1cccc(N)c1)=O)CC2 63116,C1(OCC)(CNC(c2coc(C(F)F)n2)c2nnnn2C2CCCC2)CCCC1 63117,N#Cc1cccc(C(O)C(=O)NCc2ccnc(OC3CCCCC3)c2)c1 63118,O=C(C1=CC2C=CC(C1)C2)NCCCC(O)C(=O)N1CCC1CF 63119,Cc1cncc(C)c1C(=O)NCC(c1ccccc1)CNC(=O)C(N)=O 63120,C12(CNC(C)=O)CC(CCO1)N(C(=O)C1=C(Cl)CC1)C2.C12CCCN1C2=O 63121,C(CNC(c1cnc(Br)s1)=O)(CC(C)C)NC(CCNC(=O)NC)=O 63122,C1(C)(C(N2CCC(C(=O)NCC(=O)N(C)CC)CC2)=O)CCC2CC2C1 63123,C(CCC)(C(=O)NC(C)(CNC(c1c(C)n[nH]c1C)=O)C1CC1)=CCC 63124,c1(C(C)NCC(=O)NC(C2(CC(C)(C)C)CCC2)=O)nnc2ccccn12 63125,c1(CC)c(C(N2CC3CC3C2C(N2CCOC(C)C2)=O)=O)ccn1C 63126,c1(OCC(=O)NCC2(CN(C(c3cc(OC)no3)=O)C)CC2)ccccc1F 63127,N1(C(CN(C(C)C)C)=O)CCN(C2CN(C(C3CC34CCC4)=O)C2)CC1 63128,N1(C(C(C(CC)C)O)=O)CC2CCC(N(C)C(c3ccncc3N)=O)C2C1 63129,CCN1C(=O)C(NC(c2ccccc2)CNC2CC2)c2cc(C)ccc21 63130,N1(C(c2nc(CC)sc2)C(=O)NCCCSC)CCc2nnnn2CC1 63131,C1(C(N(C)Cc2ncc[nH]2)=O)CN(C(C2CC(F)(CF)C2)=O)CC1F 63132,C1(OC)CC2(C1)CC2C(=O)OC(C)(C)C.C1CCN(C(N)=O)C1 63133,C(=O)(C(F)C(C)CC(C)(C)C)NCC1CC(CNC(CC(C)SC)=O)C1 63134,Cc1ccc(C(C)NC(N2CCN(Cc3nc(-c4ccsc4)n[nH]3)CC2)=O)cc1 63135,C(=O)(CC(C)(C)C#N)NCC1(OC)CN(C(c2ccc(SCCC)cc2)=O)C1 63136,c1(C(=O)NCc2c(CNC(C3CCC(C)(C)C3)=O)cccn2)cnc(N)c(N)c1 63137,CC1CS(=O)CCN1C(=O)C(Cc1cnc[nH]1)NC(C1CCC(C)(O)CC1)=O 63138,N1(C(C(C)C)=O)CCCC1(C)CNC(=O)Cc1cncs1 63139,C1(C(=O)NC(CN(C(c2sc(CO)nc2C)=O)CC)C)CCC2(CCOCC2)O1 63140,C1(NC(C2(CF)CC2)=O)CC2CC(NC(C3CC(O)C3)=O)CC12 63141,Cc1nccc(C(=O)NC2CC(CNC(c3cc(C(C)C)on3)=O)C2)c1C 63142,c1(C(=O)NC2CN(C(CC(=C=C)C)=O)CC(C)C2)c[nH]c2cc([N+](=O)[O-])ccc12 63143,Cc1nc2ccccc2cc1C(=O)N(C)CC1(NC(=O)C(O)CC[S+](C)C)CC1 63144,CC1(C(=O)O)CC(F)(F)CN1C(c1nc(C2CC2)n(-c2ccccc2)n1)=O 63145,C1(C2(NC(Cc3cc(C)sc3)=O)CC2)CCCCN1C(C1COCCN1C)=O 63146,C(=O)(C1CCCn2cc(C(C)(C)C)nc21)OCCSC(c1nc(C)cc(C)n1)C 63147,Cc1cc(CNC(c2sc(C)cc2Br)c2nnnn2C2COC2)n(C)n1 63148,C1(OC)CC(N(C(=O)C(N2CCN(C(C)=O)C(C)(C)C2)=O)C)C12CCOCC2 63149,CC1CCC(C(N2CC(S(C)(=N)=O)C2)=O)CN1C(c1ccc(C(N)=O)o1)=O 63150,c1(C(=O)NC2CC(NC(c3ccc(I)cc3O)=O)C2)ccc2nc(O)oc2c1 63151,C1(C(=O)NC2C=C(C)CCC2)C(C)OCCN1C(=O)Cc1cccnc1C 63152,c1(C(N2CCC(C(CNC(CCCC#C)=O)(C)O)CC2)=O)ccc2c(c1)CC2 63153,c1(C(=O)NCC2C(NC(C(C)C#N)=O)CCC2)cc(Cl)cc2c1CCC2 63154,N1(C(C(C2CN(C(CC3C(C)OCC3)=O)C2)O)=O)CC2OC(=O)N(C)C2C1 63155,C1(C(=O)NCCCS(C)=O)CCN(C(=O)CCn2ccnc2)C12CC2 63156,C1(NC(C(CC)O)=O)CC(F)CN(C(c2ccccc2C2CCCC2)=O)C1 63157,CC(C)CC(O)C(=O)N(CCCNC(c1ncncc1N)=O)CC1CCCC1 63158,c1(CC)n[nH]c(CC)c1CC(=O)NC1CN(C(=O)COC2CCC2)CC1C(F)F 63159,C1(C(C)NC(c2cnn(CC3CCCC3)c2)=O)CN(c2cnc(F)cn2)CCO1 63160,N1(C(c2c(C)con2)=O)CC(CNC(=O)C=CCCc2ccccc2)CCC1C 63161,C1(C(N(C(C)CNC(C2CC2C(C)(C)C)=O)C)=O)CCC2(CCC2)CC1 63162,c1cccc(OCC)c1.C(C(=O)NCCC1(C(=O)NCC(=O)NC)CC1)OCCC 63163,N1(C(CC(C)(C)OC)=O)Cc2nccn2CC(NC(C2(F)CCCOC2)=O)C1 63164,O=C1CC(C(=O)N2CCCC2CCNC(C2CSC2)=O)c2ccccc2N1 63165,c1(NCC)ccnc(C)n1.C1(C(=O)OC)(NC(C2C(=C)C2)=O)CCOC1 63166,N1(C(CC(C2CC2)NC(c2c(OC)cccc2)=O)=O)CCCOC(C)C1 63167,CC1(C)C(C(=O)NC(CNC(C2CCOC2)=O)C2CCC2)C1C#N 63168,Cn1c(-n2cc(C3CCCN3CC(F)(F)C(C)(C)O)nn2)nc2ccccc12 63169,c1(CC(=O)NCC2(OC)CN(C(c3sc(N(C)C)nc3C)=O)C2)ccc(Cl)nc1 63170,C(=O)(CCCCC(F)F)N(CC(C)(C)NC(C1C(C2CC2)C1(F)F)=O)C 63171,C1(NC(C(c2ccc(C)s2)C)=O)C=CCN(C(=O)Cc2cnnn2C)C1 63172,C(=O)(C1=CC2(CCOCC2)C1)NCC#CCNC(C(C)NC(CC)(C)C)=O 63173,CC1(C)C(NC(=O)CC2CCC=CCC2)CCN1C(=O)C(c1cc(F)ccc1F)=O 63174,c1(CCNC(=O)NC2CCOCC2O)cncnc1O 63175,c1(C(N2CCC(C(C)NC(=O)CC3(O)CCC3)C2)=O)ncc(F)cc1N 63176,c1(C(N2CCC(CC=C)(NC(C3CC(=O)N3)=O)C2)=O)c(Cl)ccnc1C.C(=O)CC 63177,C1(NC(COc2ccc(C)c(C)c2)=O)CC2(CCN(C(C3CC3C#N)=O)CC2)C1 63178,c1(CC)nc(-n2cccc2)sc1C(=O)NCC(O)CNC(c1cnccc1C)=O 63179,N1(CC)CCC(C)C(CNC(=O)C(C)SC(F)(F)F)C1.c12c[nH]cc1CNC2=O 63180,c1(OC)cc(C(=O)NCC2CCN2C(C2CC(CF)C2)=O)cc([N+](=O)[O-])c1Cl 63181,Cc1c(N)ccc(C(=O)NCC(C)CNC(=O)CN2OC(C)(C)CC2=O)c1C 63182,c1(C(C)C)nc(NCC2CC2)cc(=NC(C)C2CCN(C)C2)[nH]1.c1(C)ccccc1C 63183,N1(C(c2n(CC)ncn2)C)CC(c2ccccc2F)CC1C 63184,c1(C(N2CCC(CCNC(c3c(CCC)occ3)=O)C2)=O)cccc(F)c1Br 63185,CCC(C)(C(=O)Nc1cccc(NC(C2CCN(C)C2)=O)c1)OC 63186,C1(NC(C=CCOC)=O)CC2CC1N(C(=O)C(F)C(C)(C)O)C2 63187,N(C1CN(C(c2nccn2CC)=O)CCc2ccccc21)C(C1(C=C)CCC1)=O 63188,C#CC(C)(C)C(=O)NC(CO)CCCNC(=O)C(CC)C1CCC(=O)N1 63189,c1(OC)cc2cc(COc3ncnc(C)c3F)[nH]c2cc1C(=O)OC 63190,C(CC(F)F)(C(=O)Nc1cncc(CO)c1)N(C)C(C1CCC(C2CC2)C1)=O 63191,N1(CCC)CC(C(N2CCC(CN(C(=O)CCc3nccs3)C)CC2)=O)CC1=O 63192,C(CC(F)(F)C(=O)N(C1CCC(=O)NC1)C)n1cc(CC(C)C2CC2)nn1 63193,N1(C(C2C(C)(C)OCC2)=O)CC2(CCCC2)C1C(=O)NCC1CN(C(N)=O)C1 63194,n1(CC)ncnc1C(=O)NC(CC(N)=O)c1ccccc1 63195,c1(C(=O)OC)ncccc1C(N1CCC(F)(C(=O)Nc2ccc(CO)nc2)C1)=O 63196,c1(OCC)ccc(Br)c(C(=O)NCCc2nn[nH]n2)c1 63197,CCCC(C)(CC)C(=O)N1CC(CNC(=O)C(C)C(C)O)C(C)C1 63198,C1(NC(C=CCC)=O)CC2CCC1N2C(c1c(C)nn(C)c1-n1cc(C)cn1)=O 63199,C(CC(C(=O)N1CCCCC1CNC(c1cc(C(C)=O)cs1)=O)N(C)C)SC 63200,N1(C(c2cc(OC)ncc2Cl)=O)CC2CN(C(c3ccc(C#N)o3)=O)CC2C1 63201,N1(C(c2c(C)scn2)=O)CCC2(C1)CN(C(c1csc(O)n1)=O)CC(C)O2 63202,C#Cc1ccc(C(=O)N(C(C)C(N2CCCC(F)CC2)=O)CCC)cc1C 63203,CN(C)S(=O)(=O)NCC(=O)NC1CN(C(=O)CSC2CCCCO2)CC1CO 63204,CN1CCC(C(=O)NCC2CC2NC(c2cc(C#N)no2)=O)CC1 63205,N1(C(c2cc(C3CC3)on2)=O)CC2CCN(C(C3CC3C3CCOCC3)=O)C2C1 63206,N1(C(CC(=O)NCC#C)=O)CCC(NC(=O)C(=O)NCC)CC1 63207,Cc1cccc2cc(C(=O)NCCCN(C)C(C3(O)CCOCC3)=O)nnc12 63208,CCCCCC(CC)C(=O)N1CC(C)CCC1C(=O)NCCF 63209,C1(CC)(NC(=O)C2=NOC(C)C2)CCCN(C(=O)COC(C)C)C1 63210,C1(CNC(Cn2nnc(=N)[nH]2)=O)CC2CC2N1C(=O)COCC1CCCCO1 63211,C1(C(C(=O)N(CCCC)C)NC(=O)CC2CCCC2)CC=CCC1 63212,c1(C(N2CC(CC(=O)NC3CC34CC(O)C4)C3(C2)CC3)=O)cc2ncccc2[nH]1 63213,CN(CCc1ccccc1)N1CCCC(CN2CCN(c3cccnn3)CC2)C1 63214,CN1CCCCC(C(=O)NC23CCCC2N(C(c2c[nH]cc2Br)=O)CC3)C1=O 63215,c1(CCN2C3CC(CC(=O)NC4(c5cscn5)CC4)C2CC3)cc(F)ccc1O 63216,CCCCCS(=O)(=O)CC(=O)NCC(CNC(=O)CC(F)F)C(F)(F)F 63217,c1(CC(C)NC(C2CC(c3ncc[nH]3)C2)=O)ccc2c(c1)CCCO2 63218,c1(C(=O)NC2C(NC(C=CC=CC)=O)CCCC2)c(C)nc(C)n1O 63219,N1(C(=O)CCCOc2ccccc2)CC2CC(C1)N(C(=O)Cn1ncnn1)C2 63220,c1(C(=O)NC(CNC(c2c(C)nsc2NC2CC2)=O)C)nc2c(s1)COCC2 63221,Cn1c(C(N2CC(NC(c3ccc(C(C)(F)F)cn3)=O)C2)=O)cnc1S 63222,N1(C(C(CN(C)C)(C)C)=O)C2CCCC1CC(NC(c1cc(N)c(F)cn1)=O)C2 63223,C(=O)(C(=O)NOCC(=O)N(CC)Cc1cccnc1F)OCC 63224,C(=O)(CCCCCCn1cc(CC2(CO)CCC2)nn1)NC(CC)CC(C)O 63225,CC(C)CC(CC(=O)NC1CCC1CNC(=O)CCC(F)(F)F)CC(N)=O 63226,c1(C(N(CCCNC(C23CCC2C3)=O)C)=O)cc2c(s1)CCCCC2 63227,C(C)(C(=O)N(C)OC)NC(=O)CCC=CCCC1CC(OC)C1 63228,N1(C(c2ccc(NC(C)=O)s2)=O)CCC2CN(C(C3OCCO3)=O)CC2C1 63229,O(NC(=O)C(c1ccoc1)NC(=O)CC1CC2CC2C1)CCCOC 63230,N1(C(=O)NC2CNC(=O)O2)CCCC2(CCc3ccccc3O2)C1 63231,c1(C(N2CC=CC(NC(CC3ON=C(C)C3)=O)C2)=O)n[nH]c2c1CCC(C)(C)C2 63232,N1(C(C2CCC3N(C(c4c(C)ccnn4)=O)C2CC3)=O)CCc2ccncc2C1 63233,c1(C(=O)OCC)nn(C)c(C)c1CNC1CC2CNCC12 63234,C1(CNC(CC=C(C)C)=O)CC(C)CCN1C(=O)CC1CCC(F)(F)CC1 63235,N1(C(c2c(C(C)=O)cn(C)n2)=O)CC(CNC(=O)C(O)C(F)F)OC2(CCC2)C1 63236,C1(CN(C)C)COCCC1(c1nnnn1-c1ccc(Cl)cc1F)NC1(CC)CC1 63237,C1(NC(C2CC(OC)C2)=O)(CO)CCN(C(c2cn(C(C)C)nc2Br)=O)C1 63238,Cc1[nH]nc(C(F)F)c1C(=O)N(CC(O)CN(C)C(C1CCS1(=O)=O)=O)C 63239,Cc1ccc(F)cc1C(N1CC(CNC(=O)Cc2cn(C)nc2C)CCC1C)=O 63240,N1(C(C2CC23CN(Cc2ccc(O)c(Cl)c2)C3)=O)CCN2CCOCC2C1 63241,Cn1ncc([N+](=O)[O-])c1C(=O)NC1C2CN(C(=O)COC(C)(C)C)CC12 63242,N1(C(C2CCC(=O)N2)=O)CC2CCCC(NC(=O)C(=O)C(F)(F)F)C2C1 63243,N1(C(c2nc(C)oc2)=O)CCCC2(CNC(c3ccoc3C)=O)CC12 63244,C1(N(C)C(c2csc(Br)c2)=O)CCCC(O)C1 63245,N1(C(C2C(CC)C2)=O)CCC2(CCC(CNC(=O)COCC(=O)NC)O2)CC1 63246,C12(C(=O)NC3CCN(C(=O)CCC=CBr)CC3)CCCC1CCC2 63247,CCCCCCCc1cn(CC(C)NC(c2cc(C)co2)=O)nn1 63248,N1(C(=O)CC2CC23CC3)CC(C2CCCN(C(C3(F)CC4(CCC4)C3)=O)C2)C1 63249,C1(CNC(COCc2onc(C)n2)=O)CN(C(=O)Cc2cccs2)CC(C)(C)O1 63250,c1(C2(C(N3C4CC(NC(CN(C)C(N)=O)=O)(C4)C3)=O)CC2)c(F)cccc1Br 63251,Cc1ccc2c(c1)CC(C(=O)NCC(O)CNC(C1(C(F)F)CCC1)=O)O2 63252,C1(NC(CCOCC#C)=O)CC2CC(NC(=O)C=Cc3cccc(C)c3)CC2C1 63253,c1(OC)ccc(O)c(C(N2CCOC(CNC(=O)C(O)CC(N)=O)C2)=O)c1 63254,C(CN=c1cc(C)nc(-c2cc(F)ccc2F)[nH]1)N(CC(OC)OC)C(C)=O 63255,c1(CC(N2CC(NC(c3n(C)ncc3Cl)=O)C(C)(C)C2)=O)c[nH]c2ncccc12 63256,C1(C(N(C2CCCCCC2)C)=O)(NC(c2ccncc2N)=O)CCOCC1 63257,c1(C(C)NC(CCOCC)C)cc(C(=O)O)cc(C(F)(F)F)c1 63258,N(C1CCOc2c(Cl)cccc21)C(c1cc(C(=O)OC)no1)=O 63259,N1(C(C2N(C(CCC(=O)NCCC)=O)CCC2)=O)CCC(CO)C(C)(C)C1 63260,C1(C)(NC(C=CC(C)NC(=O)Cn2cnnn2)=O)CC2(CCC2)C1 63261,C(C(CC(C)C)C(=O)N1CCC(CCNC(c2cnc3[nH]ccnc2-3)=O)C1)OC 63262,c1(C(=O)NCC(CN(C)C(C2(C)CC=CCC2)=O)O)ccc(N)cc1Cl 63263,Cc1oc(Cl)nc1C(=O)NC1(C(=O)N(C)Cc2cnn(C)c2)CCSC1 63264,c1(C(=O)NC(C)CNC(=O)C(O)(C2CC2)C2CC2)ccc2c(c1)C(=O)CCC2(C)C 63265,N1(C(C(=O)NCC(F)F)=O)CCC(NC(=O)C(O)Cn2cncn2)C1C1CC1 63266,N1(C(COC2(C)CCOCC2)=O)CC2COCC2(C(=O)NCC2CCCS2)C1 63267,N1(C(c2c(CC)[nH]nc2Cl)=O)CCCC2C1CCCN2C(=O)CSc1nc[nH]n1 63268,N1(C(c2ccc(NC)c(F)c2)=O)CC2CCC1CN2C(=O)CC(C)CN(C)C 63269,c1(CC(=O)NCCC2CCC(NC(CSC)=O)C2)ccccc1[N+](=O)[O-] 63270,c1(C(=O)NC(C2CN(C(C3(C#N)CCCO3)=O)C2)C)cc2nccnc2cc1F 63271,c1(CCC(N2C(CNC(C3CC3C(F)(F)F)=O)CC2)=O)ccc2c(c1)OCO2 63272,C1(c2ccccc2)(NC(C(F)=CC)=O)CCN(C(c2ocnc2CCC)=O)C1 63273,c1(CC(N2CC(CNC(C3COCCO3)=O)C(O)C2)=O)nc2ncccn2n1 63274,c1(C(N2C(C)(C(=O)Nc3c(Cl)ccc(C(C)=O)c3)CC2)=O)cccc2c1CCC2 63275,C(=O)(C1=C(C)C(C)(C)OC1=O)NC1CCC(N(C(=O)Cn2cnnc2)CC)CC1 63276,c1(NCC2N(CC)CCC2)nc(=NC2CC2CF)[nH]c2c(C)nn(C)c12 63277,c1(C(=O)NCC2CC(NC(=O)C=Cc3ccco3)C2)cc2ccc(Cl)c(F)c2[nH]1 63278,c1(NC(=O)NCCC2C(C)CCC2)ccc(N2CCOCC2)cc1Cl 63279,C(C(CC(C)C)C(=O)N1CCC(NC(c2nc3ncccn3n2)=O)C1(C)C)OC 63280,N1(C(c2n(CCC)ncc2)=O)CC2CC1C2NC(c1ncccc1OC)=O 63281,C1(CNC(C=CCCC)=O)CC(OC)CN1C(c1cnc(O)o1)=O 63282,c1(N2CCC(CC)(CC)C2)nc(=NC(C)c2ccc(OC)cc2)[nH]c2cc[nH]c12 63283,N1(c2nc(C)nc(O)c2C)CC(CNC(C23CC(CO2)C3)=O)OC2(CCC2)C1 63284,Cc1cnc(N(C)Cc2cc(C)no2)c(S(=O)(=O)NCc2ccno2)c1 63285,CCCC(C)(O)C(=O)N1CC(CCNC(=O)C(c2ccccc2F)C)(OC)C1 63286,C#Cc1cc(C(=O)NC2CCC(NC(=O)C(C)O)CC2)cc(N)c1 63287,c1(C(=O)NC2CN(C(c3c(C(C)C)ccs3)=O)CC2O)c(Cl)nc2ccccn12 63288,C1(CC)CCN(C(=O)Cc2ccccc2C)C1C(=O)NC1CC(=O)N(O)C1 63289,c1(CN2C(CC(=O)NC3(C#N)CCOCC3)CCC2)c[nH]c2nc(Cl)ccc12 63290,C(C(C(=O)NC1CCC1NC(c1cccc2nsnc12)=O)C(C)(C)C)OCC=C 63291,Cc1cccc2[nH]c(=NCC(C)N(C(=O)CC3CC3C)C)oc12 63292,N1(C(COCC)=O)CCC(NC(=O)C(C)(C)CCCOC)C(CO)CC1 63293,Cc1ccc(CNC(N2CC=CC2C(=O)NCC2(O)CCCC2)=O)cc1 63294,c1(C(=O)NCCC2N(C(C(C=C)O)=O)CCOC2)cc(F)c(Cl)cc1Cl 63295,c1(C(=O)NCC2N(C)CCN(C(c3ccoc3CO)=O)C2)c2c(nn1C)CCC2 63296,C1(C(=O)NCc2nc(CC)sc2)CCCCCCN1C(=O)CCc1cc(C)no1 63297,C(=O)(C(F)CCC(C)C)N1CC(NC(c2[nH]cc(C)c2)=O)C(O)C1 63298,c1(NC(C)=O)ccc(N2CC(SC(C)C(=O)N(C)CC3(N(C)C)CC3)C2)nc1 63299,N1(C(c2c(C)n[nH]c2)=O)CCCC(C(C)NC(=O)Cc2csc(S)n2)C1 63300,C(=O)(C1CCOc2ccccc21)NC(C)CN(C)C(c1c(Br)cnn1C)=O 63301,N1(C(C(CC)SC)=O)CCOCC(CNC(=O)CC2(N(C)C)CC2)C1 63302,CCC(C)C(O)CN(Cc1ccc(OCC)cc1)Cc1ccccc1 63303,N1(C(CC(C(F)(F)F)NC(C2CCCC23CCC3)=O)=O)CCCC2CNC(=O)C12 63304,C1(O)(CCNC(C2(CC#C)CCCC2)=O)CCN(C(c2ccnn2C(C)C)=O)C1 63305,C1(C#N)(C(=O)NCCC(C)NC(C(C)N2CCCC2)=O)CCSCC1 63306,N1(C(C2(C)N(C(C(N3CCCCC3)C)=O)CCC2)=O)CCOCC2(CC2)C1 63307,Cc1cc2ccc(C(=O)NCC3=CCN(C(C4NC(=O)OC4C)=O)CC3)cn2c1 63308,C1(C(C(=O)NC(CCOC)CNC(c2cnccn2)=O)C)CCN(CCF)CC1 63309,Cn1cnc(NC2CCC(NC(=O)CCc3ccncc3)CC2)cc1=O 63310,C1(CCc2csc(COC)n2)CCN(NC(C(CCC)NC(N)=O)=O)CC1C 63311,N1(C(C)=O)CCCCC1C(N1CCC(CNC(=O)CCCc2csc(=N)[nH]2)C1)=O 63312,C(C1CCOC1)=CC(=O)NCCC(O)CNC(=O)C(F)(F)C1CCCC1 63313,CC(C)(CCCC(=O)NCC1CCCC1O)NC(=O)C(N)=O 63314,C(=O)(C(CC)CC=CC)NCCC1CCCN(C(C(C=C)(C)O)=O)C1 63315,C(CN=C(NCC1CC=CCC1)N(C)Cc1ccnc(F)c1)OCCC 63316,C1(C(=O)NCC(C)(C)NC(c2nc(OCC)sn2)=O)NC(=O)CC1C(F)(F)F 63317,c1(C(c2n(C)nnn2)NC(C2CCCC2)CO)cc(S(C)(=O)=O)cs1 63318,CC1OC2(C(=O)NC3CC(NC(C4(C)CCC(F)(F)C4)=O)C3)CCC1C2 63319,CCC1=C(C(=O)N2CC3CC2CCC3NC(c2ccnc(F)c2)=O)CCCO1 63320,C1(C2CCC2)(C(=O)NC(CC)CNC(=O)CC(C)(C)SC)CC1(F)F 63321,C1(C(N(CCNC(CC)=O)CC)=O)C2Cc3c(Br)cccc3C12 63322,c1(C(=O)NC(CC)CN(C(c2ccco2)=O)CC)ccccc1N=NN(C)C 63323,n1(CCC(=O)NCCCN(C)C(C2CC2F)=O)c(-c2cccs2)nnc1S 63324,C1(CNC(C=CC(C)=O)=O)CN(C(c2sccc2F)=O)CCC12CCOC2 63325,C12(C(=O)NC3CN(C(Cn4c(C)ccn4)=O)CC3C(F)F)CC1COC2(C)C 63326,c1(C(N2C(C3CCN(C(=O)C(F)C4CCOC4)C3)CCC2)=O)cccc(F)c1O 63327,c1(C(=O)NC2CC(NC(c3ccccc3-n3ccnc3)=O)C2)cc(F)ccc1Cl 63328,c1(CCC(=O)N(CCC(C)NC(=O)C#CC2CCC2)CC)cc(F)c(F)c(F)c1 63329,Cc1cccc(C(N2CC3(NC(c4ccsn4)=O)CCC2C3)=O)c1Cl 63330,c1(CC(=O)NCC(C)NC(C2C(C(=O)OC)CC2)=O)coc2c(C)c(Cl)ccc12 63331,c1(C(=O)NCC(C)NC(C2N(CCC)C(=O)CC2)=O)cccc2cccc(O)c12 63332,N1(C(CN(C(COC)=O)C)=O)CC(NC(=O)C(C)(C)C2CCC2)C(O)C1 63333,N1(C(CC(C)O)=O)CC(F)(F)CC1C(N1CCC(CO)C(O)C1)=O 63334,N(C(=NCc1ccc(C(N)=O)cc1)NS(=O)(=O)CC1CC1)C1C(C)(C)CC1 63335,C(CC(C)(C)C)(C(=O)N1CC(C2CC2C(N2CCCC23CC3)=O)C1)OC 63336,c1(OCC)nc2ncc1[nH]2.C(=O)(C1=CCCNC1)N1CCOC(CCO)C1 63337,C(=O)(C1=CCC(F)(F)CC1)N1CCC(CCNC(CCC(C)OC)=O)C(F)(F)C1 63338,N1(C(CC(CC)C)=O)C(CC(=O)NC2CCCCCC2C)C2CCCC12 63339,C1(CC)CCN(C(=O)CCc2cn(C)cn2)C1C(=O)NCC#CCOC 63340,C(=O)(CCC(C)CN(C)C)NC1CN(C(COCc2onc(C)n2)=O)C(C)C1 63341,C1(C(CNC(CCC)=O)Cc2ccccc2)CCN(C(c2ccoc2Cl)=O)CC1 63342,c12cccc(C)c1OC2.c1(NCC2C(CC)CCO2)cccc(C(F)(F)F)c1 63343,C=CC(CC)C(=O)N1C(C(=O)Nc2ccsc2C(C)C)CC1C 63344,N1(C(c2n(C(C)C)ncn2)=O)CC2(CC(NC(=O)CSC3CC3)CO2)C1 63345,CC1=C(C)CC(C(=O)NCC(C(=O)N(CC(C)C#N)C2CC2)C(C)C)CC1 63346,N1(C(CCC2CCCN(C)C2)=O)CCN(C)CC1CNC(=O)CCNC(N)=O 63347,Cc1cc(CNC(C2COC(CNC(c3sccc3C)=O)C2)=O)cc(C)c1 63348,c1(-c2c(C(=O)NCC3CN(C(C(COCC)C)=O)C3)snn2)ccccc1F 63349,Cc1cccc(C(CNC(=O)CSc2nc[nH]n2)NC(=O)C(O)C(F)F)c1 63350,N1(C(C(CCC2CC2)NC(c2c(OC)ccs2)=O)=O)CC2COC(=O)C2C1 63351,C1(C(=O)NCC(=O)N(CC)CC)CC(F)(F)CN1C(=O)CC1COCCOC1 63352,C1(NC(C2N(C(=O)OC)CCC2)=O)CCC(C)N(C(C2(C3CCC3)CC2)=O)C1 63353,c1(-c2cn(C(C3C(C)CN3C(=O)CN3CCCC3)=O)nn2)ccc2ccn(C)c2c1 63354,c1(CC)ccc(C)c(C(N2CCC(NC(=O)C(c3cccnc3)O)C2)=O)c1 63355,CC(CCCC(=O)NC(C)(C)CC1CCOC1)NC(c1cc(Cl)no1)=O 63356,c1(C(=O)NCC2CN(C(=O)CC3CC(C(F)F)C3)C2)ccc[n+]([O-])c1 63357,C1(C(=O)NC(C)CCCCNC(=O)C=C2CCC2)CC2CC1CC2(F)F 63358,Cc1nc(C(=O)NC2CN(C(C3CCC3c3nc[nH]n3)=O)C2)cn(C)c1=O 63359,c1(C(=O)OCC)cc2c(c(Cl)c1)OC2=O.c1(COC)cncc(Br)c1O 63360,c1(CC(=O)NCC(CNC(C2CC(C(F)F)C2)=O)OC)ccc2c(c1)OCCO2 63361,c1(CNC(c2ccc(CC)o2)=O)c(C)nn2c1CN(C(C1(C)CC1F)=O)CC2 63362,N1(C(CC2N(C(c3cc(C)on3)=O)CC2)=O)CCc2ncc(Br)cc2C1 63363,c1(C(=O)NC2(CCNC(CCCOCC)=O)CCC2)ccc(N)c(Cl)n1 63364,C=CCC(F)(F)C(=O)NC1CCC(NC(c2ncccc2CSC)=O)C1 63365,c1(C(=O)NC2(C)CC(C(=O)NC3CCCCCCC3O)C2)cc2ncccc2[nH]1 63366,c1(C(=O)NC2CN(C(c3c(C)ocn3)=O)CC3C2C3)ccnc2ncccc12 63367,c1(OCC(N2C(CNC(=O)CCCF)CCC(C)C2)=O)cccc(S(C)(=O)=O)c1 63368,c1(C(=O)NC(C(C)NC(c2c(OC)ccc(F)c2)=O)C)cccn2ccnc12 63369,C1(N(C(C(C)NS(CC)(=O)=O)=O)C)CCCCC1N(C)C(c1cccc(C)c1)=O 63370,N1(CC(C)NC(c2cc(C(C)=O)on2)=O)CCN(C(=O)Cn2nnc(C)n2)CC1 63371,C12(C(=O)NCC3N(C(C4CCC(F)(F)C4)=O)CCN(C)C3)C3CC(CC13)C2(F)F 63372,C(=O)(C(C)CC)NC(C(=O)N(CC(CSCC)O)C)c1ccoc1 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63425,C(CC)(CC(F)(F)F)NC(C1(CCC=C)CN(C(=O)C(CC)SC)C1)=O 63426,C1(NC(c2c(CC)cno2)=O)CC2CC1CN(C(c1ccsc1C)=O)C2 63427,CC(CC(=O)NC1CCC1NC(=O)CC(=O)N(C)C)P(C)(C)=O 63428,Cc1ccc(CN2CC3C(C2)N3c2ncncc2C#N)c(F)c1 63429,C1(CNC(C2CC(=O)N(CCOCCO)C2)=O)CC(C2CC2)=NO1 63430,c1(C(N2C(C(=O)NCCC#C)CC3(CC3)C2)=O)cccc2c1CCC2 63431,C1(NC(=O)OC(C)(C)C)COC2(CCC2)CN1N1C2CCCC1C2 63432,CCCCCC(O)C(C)C(=O)N1CCCC(CCNC(C2CCN2CC)=O)CC1 63433,C(C1CCC(C)CC1)=C(C)C(=O)Nc1ccc(NC(=O)C(C)(C)C2CC2)c(C)c1 63434,CC1(C(=O)NC(C)(CNC(=O)Cn2ccc(C3CCC3)n2)C2CC2)CCCCO1 63435,C1(CC(=O)NCC(C)CNC(=O)C(F)(F)c2csc(=N)[nH]2)CC(=O)NC1=O 63436,N1(C(c2c(C)csc2)=O)CCC(C)(C)C1C(=O)NCC1CCCCC1(C)C 63437,C1(C(=O)NCC2(F)CC(NC(CCNC(C)=O)=O)C2)CCCC(O)C1 63438,CC1CN(C(c2cnc(Cc3ccccc3)s2)=O)CC1NC(=O)CCS(C)=O 63439,C1(C)(C(=O)NC(CCCNC(C2(CC(C)=O)CCC2)=O)C)CCCCO1 63440,c1(CN2CC(C(=O)Nc3ncc(F)cc3Br)OCC2)ccc2ncnn2c1 63441,C1(NC(c2ccnc(OC)n2)=O)CCCCCC1NC(=O)CN1CCN(C)CC1 63442,CC1CC(C(=O)N(C)CC2(CN(C(=O)CCCCC3CC3)CC)CC2)CCS1(=O)=O 63443,c1(CC)ccc(N)c(F)c1.c1(C2c3nnnn3CC2)cnn(CC(F)F)c1 63444,C1(NC(CCc2cn(C)nn2)=O)CN(C(C2(O)CCOC2)=O)CC(C)(C)C1 63445,N1(C(CNC(CN(C)C)=O)=O)CCN(C(=O)CCc2cncn2C)CC1C1CC1 63446,C1(CNC(C2C(C)CCCC2)=O)CC(C)CN(C(C2CN(C3CCC3)C2)=O)C1 63447,N1(C(C=CC(CC)=CC)=O)CCC(C)(C)C(CNC(C2CCCC3(CC3)C2)=O)C1 63448,N1(C(CCN(CC)CC)=O)CC(NC(c2cnn(C)c2C(C)(F)F)=O)CC1C 63449,CN1CCc2cc(C(=O)NCC(C3CCC3)NC(=O)C(O)CC(N)=O)ccc2C1 63450,C#CCCC(C(=O)NCCCC(O)CO)NC(=O)CCC=CCC=C 63451,C(CN=C(NCc1nc(C(F)(F)F)cs1)N1CC2CCOCC2C1)c1ccsc1 63452,N1(C(COCCCCC)=O)CC(C)(CNC(c2cc(SC)c(C)o2)=O)CC1(C)C 63453,c1(C(=O)NC(CC)(C)CNC(=O)C(C)n2cncn2)cc2c(ccn2C)s1 63454,C(=O)(CC1=CCN(C(=O)CC2(C)CC2)CC1)NCC(c1cn(C)nc1)O 63455,C(N=c1[nH]c(Cl)nc2cccc([N+](=O)[O-])c12)C1N(CC2ON=C(CC)C2)CCC1 63456,Cc1ccc(CNC(C2C3CN(Cc4ccc(O)c(O)c4)CC23)=O)cc1C 63457,C1(CC)=NC2=CC(=NCC(c3cccs3)N2)N1.N(C)(C(=O)OC)CC 63458,N1(C(c2c(C)noc2C)=O)CCC2(CCN(C(=O)Cc3cc(Br)ccc3Cl)C2)C1 63459,Cc1cc(=NCC2(C)CCC(C)(C)CC2)[nH]c(=NCCCC(C)O)[nH]1 63460,N1(C(CCN2CCN(CC)CC2)=O)CCN(C(C2(F)CC=CC2)=O)CC1C1CC1 63461,C1(C)(CC)CCC(C(=O)NCC(C)N(C)C(c2csnc2C)=O)O1 63462,C12(NC(C(CC(C)C)C)=O)CCCN(C(=O)COC3(C)CCCC3)CC1C2 63463,N1(C(C(CCSC)O)=O)CC(C2(NC(C3CCN(C(C)=O)CC3)=O)CC2)C1 63464,O=C1CCC(=O)N(CCSSc2cncs2)C1.C12CCN(CC1)C2=O 63465,N1(C(CN2CC(C(C)=O)C2)=O)CCN(C(C2CC2C2CC2)=O)CC1 63466,C12(C(=O)OC(C)(C)C)CC(CC(N3CCCC3CNC(=O)C(F)Br)=O)(C1)C2 63467,N1(C(C2(N(C)C)CC2)=O)CC(NC(=O)Cc2cc(Br)cs2)CC(F)(F)C1 63468,C1(O)(C(=O)NCC2CCCN(C(C(C)C3CCOC3)=O)CC2)CCC(C)(C)CC1 63469,C1(C2(O)CN(C(C3CCc4nn[nH]c4C3)=O)C2)(CNC(CCNC(N)=O)=O)CC1 63470,c1(CC)[nH]nc(C(=O)NC2CC2CN(C(C)=O)C2CC2)c1Br 63471,C#CCCCCCC(=O)N1CC(NC(=O)Cc2cnccc2Cl)C(N=[N+]=[N-])C1 63472,N1(C(COC(C)C)=O)CCCC(C)(C)C1C(=O)NC(CC1CCCC1)CO 63473,N1(C(C2(CNC(C(COCC)C)=O)CC=CC2)=O)CCCSCC1C 63474,c1(C(=O)OC)cnn2c1CC(NC(c1cccc3ccc(O)nc13)=O)CC2 63475,C1(N(C(C2CC2CF)=O)CC)CCN(C(=O)C(F)(F)C2(OC)CCCC2)C1 63476,C12(C(=O)NC3CCN(C(C(CC)c4ccccc4)=O)CC3)CC3CC(CC1C3)C2 63477,c1(C(N2CC(C)C(O)(C(F)(F)F)CC2)=O)nnc(C2CC2)n2cccc12 63478,C1(CC=C)(C(=O)O)CCCCN1C(=O)C(F)CC 63479,CC(CC(F)(F)F)C(=O)N(C1CN(C(C2CCCC3(CC3)C2)=O)CCC1O)C 63480,Cc1csc(C(=O)NCCC2COCCN2C(=O)CC2(C)CCC2)c1Br 63481,c1(-n2cc(C(=O)OC)nn2)cccc(NC(c2ccoc2)C)c1 63482,CCC(CC#N)N=c1ccc(Br)c(S(=O)(=O)NCC(O)CN(C)C)[nH]1 63483,C(C(=O)N(CC(C)C(=O)NCc1c(CC)noc1C)C)(C(C)C)OCC 63484,N1(C(Cc2ccc(OC)c(Cl)c2)=O)CCN(C(=O)C(C#N)C2CC2)CC(C)(F)C1 63485,N1(C(c2n[nH]c(O)n2)=O)CCC2CCN(c3c(Cl)cccc3[N+](=O)[O-])CC2C1 63486,c1(C(=O)NC(CN(C(C2(CCC=C)CCCC2)=O)C)C)nccc(Cl)c1O 63487,c1(C(=O)OCC)cc(Cl)c(F)cc1S(=O)(=O)N(c1cc(Cl)nc(OC)n1)C 63488,CCCCC(CC)C(=O)NCC1CCCN(C(=O)CC2CCOC(C)(C)C2)C1 63489,N1(CC(=O)NC2CCOCC2NC(C2CC(=C3CC3)C2)=O)C(=O)CCC1=O 63490,Cc1cc(CNC(c2cc(C)oc2C)C)nc(N2CCOCC2)n1 63491,c1(CC(N2CCN(C(c3c(C)nn(CCO)c3)=O)CC2)=O)ccc(F)cc1F 63492,C(=O)(CC(C)(C)C(F)F)N1CCCCC(NC(CCC=C=C)=O)C1 63493,C1(NC(CCC(=C)Cl)=O)CN(C(=O)COc2cc(Cl)ccc2C)CC12CCC2 63494,CC1CC(C2CN(C(=O)C=CC(C)NC(=O)Cc3cncn3C)C2)=NO1 63495,C1(NC(=O)OC(C)(C)C)CN(C(=O)CCCCc2cn[nH]c2)NC1=O 63496,N1(C(CCC(C)OC)=O)CCCC2(NC(=O)C(N3C(C)CCC3C)C)CCCC12 63497,c1(C(=O)Nc2ccc(NC(C(CCC)CC)=O)cc2)cnc2c(c1)NCC(=O)N2 63498,N1(C(CNS(NC)(=O)=O)=O)CCCN(C(C2CC(O)C2)=O)C(C(C)C)C1 63499,C1(NC(CCN(C(CSC)=O)CCCO)=O)CCCCN(C)C1 63500,c1(N2CC(CN(C)C(C3CC(=O)N3)=O)OCC2)nc(Cl)nc2c1COCC2 63501,C12(NC(c3nc(CC)sc3)=O)COCCC1CN(C(=O)CCc1ccc(C)s1)C2 63502,C1(C(=O)NC(C)CNC(=O)C(C)(C)n2cc(Cl)cn2)CCC(=O)NC1 63503,C1(C(=O)NCCCC(=O)N(C)C)CCC2(CC2)N1C(C1CCCN1C)=O 63504,Cn1c(C(=O)NC(c2ccncc2)C2CC2)ccc1C12CCC(CO1)C2 63505,c1(OC)c(C(C(=O)NCCCF)N(C2CCOC(C)C2)C)ccnc1F 63506,Cn1nccc1CCC(=O)NC1(CCC(=O)NCCc2cn[nH]c2)CCCC1 63507,c1(C(N2C(C(=O)Nc3cc(C)nc(F)c3)CC(F)C2)=O)ccc2c(c1)C(=O)CC2 63508,N1(CCn2c(C(C)C)nnn2)CCC(NC(c2csc(C3CC3)n2)=O)CC1C 63509,N1(Cc2c(C)nc(Cl)cc2)CCC2(CC1)CC2NC(c1ccc(C#N)cn1)=O 63510,N1(C(C=C=C(C)C)=O)CCN(C(=O)CC(C)n2cccn2)C(CC(C)(C)C)C1 63511,C(=O)(C(CC(C)C)N(C)C(c1cnsc1C)=O)NCc1nc(CSC)sc1 63512,CC1CCN(C(C2(C(F)(F)F)CC(F)(F)C2)=O)CCN1C(=O)Cc1cnns1 63513,Cc1nccn1CCCC(=O)NC1CCC(C(N2CCC(O)C2)=O)C1 63514,C(=O)(CC(C)(O)C(F)(F)F)N1CCCC(CCNC(C2(SC)CC2)=O)CC1 63515,c1(CC(C(=O)NCCC)NC(=O)Cc2cccnc2Br)cccc(OC(C)C)c1 63516,C1(NC(C=Cc2n(C)ncc2)=O)CN(C(=O)Cc2n[nH]c(=N)s2)CC1S(C)(=O)=O 63517,c1(C(N2CC3C(NC(CCCC#C)=O)C3C2)=O)cc(C)nc(N(C)C)n1 63518,CC1(C)CN(C(C2CN(C(c3csnn3)CCl)C(C)(C)C2)=O)CCC1NC(N)=O 63519,C(=O)(CCC(C)(C)C)N(C(CCNC(C(CN(CC)CC)F)=O)C)C 63520,c1(C(N2CCC(N(CCC)C(C3CCCC3C)=O)C2)=O)cnn2cccc2c1 63521,C1(NC(CCOCC)CO)CC2CCC1O2 63522,C(=O)(C(CCC(=O)NC1(C)CCSC1)OC)N1CC(CCC#C)C1 63523,N1(C(C(C)(C)OC)=O)CCN(C(c2ccc(C#N)c(F)c2)=O)CC(C)C1 63524,C(=O)(C(C)(O)C(C)(C)C)NC1CC(NC(c2ccc(CC)nc2C)=O)C1 63525,C12(NC(c3ccc(Cl)cc3F)=O)COCCC1CN(C(c1ccns1)=O)C2 63526,c1(C(C(=O)NCc2cccs2)N(C2(C#N)CC2)C)cc(-c2ccccc2)nn1C 63527,c1ccc(N2CCCC2)cc1.C1(CN2CCC2)CCCN1 63528,Cc1cncc(CCNC(=O)C(C2CCN(C(c3cnncc3O)=O)CC2)C)n1 63529,N1(CC)CCN(C(F)(F)F)C(=O)C1.c12cnc(nc1)CCNC(=O)C(=O)N2 63530,c1(NC(=O)NC2CCN(C(C3CC4CC3CC4O)=O)CC2)c(Cl)cccc1Cl 63531,c1(OC)ccc(CNc2cc(C)cc(SC)n2)cc1S(=O)(=O)N1CCOCC1 63532,C12(OC)CCC(CN(C3CCOC3)CCO)(CC1)C2 63533,c1(OC)ccc(CC(N2CCCC(CCCCOC(=O)C(C)=C(C)C)C2)=O)nc1 63534,c1(C(=O)NC2C(CNC(C3CCC(C)CC3)=O)CCC2)cccc2cncn12 63535,N1(C(Cc2c(C)scc2)=O)CCC(NC(=O)C=Cc2ccoc2)C(C)C1 63536,c1(OC)cc(C)c(C(=O)NC(C)CN(C)C(c2nonc2N)=O)cc1Cl 63537,C(=O)(C(F)C(C)(F)F)NC(C(=O)NC(c1nc(CC)on1)C)(C)CSC.C(C)(=O)O 63538,c1(C(=O)NCCCC)c(Cl)cc(Cl)nc1N.N12CCC(CC1)C(=O)NC1CN2C1 63539,C(=O)(C(C)(C)CCCO)N(C)CC1CCCN1C(c1ccc(C(F)F)cc1)=O 63540,N1(CC(=O)Nn2cc(CC(N3CCOCC3CC3CC3)=O)nn2)C(=O)CCC1=O 63541,c1(C(N(CCC(C(C)C)NC(C(CC(=O)OC)C)=O)C)=O)cc2cn[nH]c2cn1 63542,O=C(CC(CNC(C1(F)CCCC1)=O)C1CCC1)NCC(CO)C1CCC1 63543,C1(CC(=O)NCC2C(C(N(C(c3cc(C)on3)C)C)=O)C2(C)C)CCCNC1=O 63544,C1(CN(C(=O)COCP(C)(C)=O)C)CN(C(=O)CC2(O)CCOC2)CC12CC2 63545,C12(C(=O)NC3C(NC(CSC(C)(C)C)=O)COC3)C3C4C1C1C2C3C41CO 63546,C1(NC(C2N(CC)CCOC2)=O)CCN(C(=O)Cc2cccs2)CC1C 63547,N1(C(C(C)(C)SC)=O)CCCCC(NC(=O)CCn2ccnc2C(C)C)CC1 63548,Cc1c(C(N2CCCN(C(C3CCC(=O)N3)=O)C(C)C2)=O)[nH]c2cc(F)ccc12 63549,C(=O)(CCC(=O)NC1CCCO1)NCCN(CCC)CCOC 63550,C1(C(=O)NCCOCCCC#C)CC(C)CN(C(c2occc2C2CC2)=O)C1 63551,C1(NC(C2C(=C)CC2)=O)CN(C(c2ccc(C)c(C)c2)=O)C(CC)(CC)C1 63552,c1(C(N(CCCNC(c2c(C)nc(CC)o2)=O)C2CC2)=O)ccc2c(n1)NCC2 63553,N1(C(c2c(C)coc2)=O)CCC(N(C(=O)CCc2c(C)noc2C)C)C2(CC2)C1 63554,C1(CC(=O)NC2CCC2)(NC(C2CC=CC2)=O)CCCC1 63555,C1(NC(C2(CC(C)C)COC2)=O)CCC(NC(=O)C(c2cccn2C)=O)C1 63556,c1(CC)c(C(=O)NCCNC(=O)CCCc2nc(C)no2)cccc1Br 63557,c1(C(N2C(CNC(c3c(C)coc3)=O)CC2)=O)c(C)nn(CC(F)(F)F)c1Cl 63558,Cc1nsc(C(=O)NCCc2csc(-c3cccs3)n2)c1NC(=O)OC(C)(C)C 63559,N1(C(c2[nH]cc(C)c2)=O)CC(N)C2(CCOCC2)C1 63560,C1(NC(C2C=CCC2)=O)CC2CC(NC(c3sc4sccc4c3Cl)=O)CC2C1 63561,S(=O)(=O)(c1ccc(=NCC2CCCCN2C2CC2)[nH]c1)N1CCC(C(CC)=O)C1 63562,Cc1cc(C(=O)NCC2COC(CNC(=O)CCc3n[nH]c(=N)s3)C2)nc(O)n1 63563,CC1N(Cc2cnn(C)c2C(=O)O)CCC1(C)C 63564,C=C(Cl)CCC(=O)NC(C1CC=CCC1)C(=O)NCCF 63565,N1(C(C(N2CCCCC2=O)C)=O)CCC(F)(CNC(c2cn(CCO)nn2)=O)C1 63566,c1(CNC(=O)NC(CC)CCOC)cc(Br)c(C)s1 63567,N1(C(C=CC)=O)CC(CNC(c2cc(NC3CC3)nc(C(F)F)c2)=O)C(C)(C)C1 63568,c1(CS(=O)(=O)NCC2CC2Cl)ccc2c(c1)CCCC2 63569,CC1(C)CCC(CNC(=O)C(CCF)NC(c2ccc(C(F)F)o2)=O)O1 63570,CC(C)C(O)C(=O)NC(C)(CNC(c1ccc(CS(C)(=O)=O)cc1)=O)C(C)C 63571,Cc1conc1C(=O)NC(C)C(c1ccccc1)NC(C1CSC1)=O 63572,CC(=O)CCCCC(=O)N(CC(=O)NCC(O)C(F)(F)F)CC1CC1 63573,C1(C)(C(N2CCC(O)(C(C)CNC(c3ccc(CO)o3)=O)C2)=O)CCC2CC2C1 63574,c1(CC(=O)NC2C(CNC(C3(C)CCCCO3)=O)CC2)ccc(S(N)(=O)=O)cc1 63575,C1(OCC)CC(N2C(=O)CN(Cc3ccncc3)C2=O)C12CCC2 63576,C12(C(=O)NCC(C)(C)CNC(C3(C)CCOC3)=O)CCC(CC1)C2(C)C 63577,CC1CCC(O)CN1Cc1nc(Cc2cccc(Cl)c2)no1 63578,N1(C(C(CCSC)O)=O)CC(C(=O)NC2CCCC2N=[N+]=[N-])CC(C)(C)C1 63579,c1(C(N2C(C(=O)Nc3cc(OC)n[nH]3)CC3CC32)=O)cnc(Cl)cc1OC 63580,c1(C(N(C2CCCC(NC(CCC=CC(C)C)=O)C2)C)=O)cc(Cl)cc(F)c1F 63581,c1(CNC(C(=O)NC(c2nc(C3CCCCC3)no2)C)=O)cccc(F)c1 63582,N1(C(c2cnc(C(C)C)s2)=O)CCC2(CC1)CN(C(=O)C(O)P(C)(C)=O)C2 63583,C(C(C)(C)CC(=O)N1CCC(C)C(C)C1)NC(CCCOCCOC)=O 63584,N1(c2ncc(C)c(C)n2)CCC(NC(=O)C(C)S)C(C)(C)C1 63585,CCCCCCCCC(C)CC(=O)N1CC(NC(=O)CCNC(=O)OC)C(C)C1 63586,CN1CCN(C(c2ccccc2)=O)CCC1=O.C1(=O)CCCn2cc(nn2)CN1 63587,C1(=CC(=O)NCC2CCC(NC(C(C=C)O)=O)C2)CCC(C)CC1 63588,C(CCCCCC(=O)N1CCC2C(C(=O)Nc3cnn4c3CCCC4)C2C1)OC 63589,N1(CC)CCCC(C(=O)NCC2CN(C(=O)COCP(C)(C)=O)CC2O)C1 63590,Cc1noc(C(F)F)c1C(=O)NCC(C)(C)CCNC(C1(N(C)C)CCC1)=O 63591,c1(OC)ccc(I)cc1C(N1CCSC(C(=O)Nc2ncc(Cl)cc2F)C1)=O 63592,c1(CNC(=O)CC2CN(C(C3(CO)CC3)=O)CCO2)ccc(Cl)c(C(F)(F)F)c1 63593,C1(NC(=O)CCC2CC2(Cl)Cl)CC2CCCC(C1)N2C(=O)CCOC1CC1 63594,N1(C(C(C(CC)O)C)=O)C(CNC(=O)CC(C)(C)C)CC2CCCCC12 63595,C1(CNC(c2occ(C)c2C)=O)CN(C(=O)COC2CCCOC2)CCC1(F)F 63596,Cc1cc(CC(=O)N(C(C)CNC(=O)CC2CCC(=O)CC2)C)n(C)n1 63597,N1(C(c2c(SC)scc2)=O)CC2CC(CNC(C3CC4(CC4)CO3)=O)C2C1 63598,C1(CNC(N2C(C(=O)OC)CCC2c2ccccc2)=O)CCC(OC)CC1 63599,Cc1nc(=N)[nH]c(=NCCCC(C)NC(C2CC3CCC2CC3)=O)[nH]1 63600,c1(COCC)nc(N2CCC(NC(=O)Cn3nc(C)cc3C)C(F)C2)cc(Cl)n1 63601,c1(C(C)=O)cc(C(=O)NC(C)C(C)NC(=O)CCn2cccnc2=O)ccc1F 63602,N1(C(C2C(C)(C)C2)=O)CC(C2CCCN(C(c3ncn4cc(Cl)ccc34)=O)C2)C1 63603,c1(C(=O)NC(C2CCN(C(c3csc(CN(C)C)n3)=O)C2)C)cnc2[nH]cncc1-2 63604,C(=O)(C1=CS(=O)(=O)CCC1)N1CCCC(CCNC(=O)Cn2cncn2)C1 63605,CCCCCC(O)C(=O)NCC1CC(F)(F)CN1C(=O)CC(C)CCC=C(C)C 63606,c1(CC)cnc(C(=O)N(C2CCN(C(C3COCC3(C)C)=O)C2)C)nc1 63607,c1(C(c2n(CCCCCC)nnn2)Nc2cn(C)cn2)cccc(OC)c1Cl 63608,C1(CNC(c2cncs2)=O)CN(C(=O)CN2C(=O)CCC2=O)CCC12CCOC2 63609,CCC(CCOC)C(=O)NCC(CNC(=O)CCn1ccnc1C)OC 63610,c1(N2CCCC(C(F)F)C2)nc(N2CC=CC(C(F)(F)F)C2)nc2c1COCC2 63611,C(=O)(C(F)(F)C(C)O)NCCC1(OC)CN(C(=O)C(C2CCOCC2)C)C1 63612,c1(C(N2CCC(CC)C2CNC(=O)COC2(C)CCCC2)=O)ccc(F)c(C)c1 63613,c1(OC)cccc2c1OC(C(=O)NC1C3CCC1N(C(C1(CF)CCC1)=O)C3)C2 63614,CCCC(CNC(C1CCCSC1)=O)NC(c1cnc(C(C)C)[nH]1)=O 63615,C(=O)(C(C)C(C)(C)C)N1CC(CC(C(=O)NCc2n(CC)ccn2)F)C1 63616,Cc1noc(-c2ccco2)n1.C1(C(N(CC(C)N)C)=O)(C(N(C(C)=O)C)=O)CC1C 63617,c1(C(CCO)NC(c2n(CCC)nnn2)C(C)(C)SCC)ccc(C(C)C)cc1 63618,C1(NC(CCC(C)NC(c2c(C)scc2)=O)=O)C2C3CCC(C3)C12 63619,S(=O)(=O)(c1cccc(N2CC3CC2CS3=O)n1)NCC(c1ncc(C)s1)C 63620,C1(NC(=O)Cc2ccsc2)CC(F)(F)CC1NC(C1(O)CCC1)=O 63621,CC(C)C(CN(C)C)C(=O)N1CCCCC1C1C(CCNC(=O)CNC=O)C1 63622,c1(NC(C2CN(C(C)(C)C)C(=O)C2)=O)scc(Cl)c1C#N 63623,C1(C(=O)NCC2(OC)CN(C(C(CC=C)(C)C)=O)C2)CC2COCC(C1)C2 63624,c1(OC)ccc(C(=O)NCC2(CNC(C3CCC(C(C)C)CC3)=O)CCC2)cc1 63625,c1(NC)ccc(C(=O)N(CCCCN(C(=O)CC(C)F)C)C)cc1[N+](=O)[O-] 63626,N1(C(CCC#C)=O)CCC2(CC1)C(NC(=O)CN1CCC(C)C1)CS2(=O)=O 63627,C1(C(N2CCC(O)(C(F)F)C2)c2nnnn2C(C2CC2)NC)(SC)CC(F)(F)C1 63628,C1(CC)(NC(=O)CC(F)F)CCN(C(=O)CCC(=O)Nc2nccs2)C1 63629,C1(C)(C(CNC(C(C)C2CCCC2)=O)=O)CCCN(C(=O)C=CC=C(Cl)Cl)C1 63630,C(c1cccc(F)c1)=CC(=O)N(CC(C)O)CCNC(CN(C)CC)=O 63631,C1(NC(c2ncn(C(C)C)n2)=O)COCCN(C(=O)CN2CCCCCC2)C1 63632,Cc1cc(=O)c2cc(NC(=O)NC3(c4ccc(F)cc4F)CC3)ccc2[nH]1 63633,CC1(C#CC(=O)N2CC3CN(C(=O)C=Cc4cccs4)CCC23)CCCO1 63634,C1(C)(C(N2CCC(C)C2CNC(c2ccn(C3CC3)n2)=O)=O)CCC(C)(C)CC1 63635,C1(CC)CCN(C(C2COCCN2C)=O)C1CNC(c1nnn(C)c1C)=O 63636,C1(C(N(CC(C)NC(c2ccc(Br)o2)=O)C)=O)CS(=O)(=O)CC12CC2 63637,C1(CNC(CC2N(C)CCC2)=O)(CO)CCN(C(C23CCCC(CO2)C3)=O)CC1 63638,O=C(N=c1cc(Cl)nc(C(F)(F)F)[nH]1)C1C2CCC(C2)N1Cc1ccccc1Br 63639,Cc1cc(N)c(C(=O)NC2CCC2NC(=O)C(C)C(F)F)c(F)c1 63640,C1(NC(CNC(C2CC(=O)C2)=O)=O)CCCC2(CC2)C1 63641,N1(C(C(c2ccccc2)C)=O)CC2(CCCCN2C(c2cnc(S)n2C)=O)C1 63642,C(CC(C)C(=O)C(CCc1ccc(C(=O)NCC(CN)C)o1)=O)=CC.OC 63643,c1(CC(N2CCCC(CN(C(C(CC(=C)C)C)=O)C)C2)=O)nc2ncccn2n1 63644,C1(CNC(c2cc(C)no2)=O)CCN(C(C2CC(C)CCC2C(C)C)=O)C12CC2 63645,C1(NC(C2CCN(C3CC3)C2=O)=O)CC2CCC1N2C(=O)COCC(F)(F)F 63646,C(=O)(CC(C)C(=O)N1CC=C(CNC(=O)C(C)NS(C)(=O)=O)CC1)OC 63647,CC1(C)CN(C(=O)CCN(C(=O)C(C2CCCCC2)O)CCO)CCC1O 63648,C(C(CC)(CC)C(N)=O)NC(CN(C(c1cccnc1S)=O)CC)=O 63649,C1(NC(C2CCCCC2)=O)CC2CCC1N(C(c1ccn(C3CC3)n1)=O)C2 63650,C(=O)(C(F)C(C)C(F)(F)F)NCC1(C)CCN(C(CCSCCCC)=O)C1 63651,N#Cc1ccc(F)cc1NC(c1cncc(-c2c[nH]c3cnccc23)n1)=O 63652,c12cc(ccc1O)C(=O)NC2C.c1(COC)cn(CCCN(C)CCO)nn1 63653,CON=C1CN(C(=O)C(C)(C)Oc2ccc(Br)cc2)C1 63654,C1(CC(C)C)CCCCN1C(=O)C(C)CN(C(=O)CSC(F)(F)F)C 63655,C1(NC(c2scnc2Cl)=O)CN(C(=O)CC2OCCCO2)Cc2nccn2C1 63656,C(=O)(C(C)CNC(=O)C(CSC)NC(c1nc[nH]n1)=O)NC 63657,CC1C(C(=O)NCCC2CC(F)(F)C2)CCN1C(=O)CCC1CCCC1 63658,C1(NC(C2CC(N3CCN(C)CC3)C2)=O)CCN(C(C2(C)CC2)=O)CC1F 63659,c1(CC(F)F)nc(CNC2CC(N3CCCC3)C2)c(Cl)n1-c1ccccc1 63660,C1(NC(c2c(C)cc(CO)o2)=O)CN(C(=O)C=Cc2cccs2)CC2CC12 63661,C1(NC(C(C)C)=O)CCN(C(c2ccc(CN(C)C3CC3)o2)=O)CC1 63662,C1(N(C(CS(=O)(=O)NC)=O)C)CCCCN(C(c2nnc(S)n2C)=O)C1 63663,CCC(CCCC(=O)NCCCC1CCOC1)NC(c1ncncc1C)=O 63664,C(CCCCC(=O)N1CC(Cn2ccnn2)C1)N(C(C1OCCN(C)C1)=O)C 63665,c1(CC)cc(C)ccc1C(N1CCCC1CCNC(c1c(C)ncn1OC)=O)=O 63666,C1(NC(c2cc(N)nc(Br)c2)=O)CCN(Cc2ccccc2)CCC1(F)F 63667,N1(C(c2ncn(C)n2)=O)CCN(C(=O)Cn2ncc(C#N)c2N)C(CC(F)F)C1 63668,N1(C(c2nc(C(C)NC(c3cnc[nH]c3=N)=O)oc2)=O)CC2(CNC(=O)N2C)C1 63669,CC(CC(=O)NCC(C1CC1)NC(c1cnn(C)c1Cl)=O)C(F)F 63670,CCCCC(CNC(c1cncc(F)n1)=O)NC(=O)Cn1ccnn1 63671,CC(Cc1c(F)cccc1Cl)N=c1[nH]c(N2CCOC3COCC3C2)nc(=N)[nH]1 63672,C12(C(=O)NC3(CC)CCOC3)CC(CO)(CN1C(=O)C=NOC)C2 63673,c1(CC(=O)NCCN(C(=O)C(C(C)O)N(C)C)CCOC)ccc2c(c1)CC2 63674,N#CC1CN(C(C2(C3CCCN3C(c3cnn(C4CC4)c3)=O)CC2)=O)CC12CCC2 63675,C(=O)(CC(C)CCC=C(C)C)NC1CC(N(C(c2c(O)ccc(OC)c2)=O)C)C1 63676,c1(C(=O)NCCN(C)C(c2cc(C(F)F)n[nH]2)=O)ccc(F)cc1C(C)(F)F 63677,C1(C(N2C(C)CC(CNC(=O)C(F)C(F)(F)F)C2)=O)CCCC2(CCC2)C1 63678,CC1(C)CN(C2CN(C(=O)Nc3cc(F)ccc3C3CC3)C2)C(=O)O1 63679,CCCS(=O)(=O)CC(=O)NCCC(O)CNC(c1cc(OC)cs1)=O 63680,c1(CC)cccc(OCc2nc(-c3ccncc3)nn2-c2ccnc(O)c2)c1 63681,N1(C(C(CCC)NC(N)=O)=O)CCC(NC(c2ccc(C)cc2F)=O)C12CC2 63682,N1(C(CC(C(C)C)C)=O)CCCCC(C2CN(C(C3(C(C)(C)O)CC3)=O)C2)C1 63683,c1(C(N2CC(C)N(C(c3ccno3)=O)CC2)=O)cc2c(F)ccc(F)c2[nH]1 63684,c1(C(C(=O)NC2CC(CF)C2)N(C2C(OC)COC2)C)cc(C)c(C)cc1C 63685,CC(C(=O)NC1(CCC(=O)N(C)Cc2cocn2)CCC1)n1ccnn1 63686,C(C(C)(O)C(=O)N1CCC(F)(C(=O)NCC2=CCCOC2)C1)OC 63687,c1(CC(N2CC(F)(CNC(c3c(C)n[nH]c3)=O)C2)=O)ccn2cncc2c1 63688,c1(C(=O)NCC(C)CN(C)C(c2cccc3sccc23)=O)cccc([N+](=O)[O-])c1 63689,c1(NCC(CSC)OC)ncnc(N2CCOC(C)(c3ccccc3)C2)c1C 63690,c1(C(C(N2CCC(NC(CN3CC(C)C3)=O)CC2)=O)(C)C)c(F)cccc1Cl 63691,c1(C(=O)NCC2CN(C(C(C)O)=O)C(C)(C)C2)cccc2c1OCCCO2 63692,O=C(CCC1CC1C(=O)O)NCC1CC(NC(=O)CC2OCCO2)C1 63693,c1(C(=O)OC)cc(OC)cc(C(N2CC(CC3(CC(C)C)CC3(F)F)C2)=O)n1 63694,C1(N(CCOCCN(C(CCOCCN(C)C)=O)C)C)CCN(C)CC1 63695,N1(C(c2c(Cl)ccc(NC)c2)=O)CC(C)CN(C(C2(SC)CC2)=O)CC1C 63696,C1(=O)C(CCC(N)=O)N1.c1(OC)ccc(-c2cn(CC3CCC3)nn2)c(F)n1 63697,CC(C(=O)NC1CCCCC1CNC(c1cnccc1C(F)F)=O)C(F)(F)F 63698,c1(CC(N2CC(CC(C)NC(C3(OCC)CCC3)=O)C2)=O)coc2ccccc12 63699,CCCCC(O)C(=O)NCC1(O)CCCN(C(=O)CCCNS(C)(=O)=O)C1 63700,N1(C(CC2(OC)CC2)=O)CC(NC(=O)Cn2nc(C)c(C)c2C)CC(F)C1 63701,C(=O)(C(=O)N=c1nc(C2(C)CC2)[nH]s1)Nc1c(C(C)C)noc1 63702,N1(C(C(CC)CC)=O)CC(CNC(c2ccnc(C)c2C)=O)OC2(CCC2)C1 63703,N(C1c2ccccc2CC1O)c1c(OCC)ccc(CC2CCS(=O)(=O)C2)c1 63704,CCC(C(=O)N1CC2CCC(CNC(C34CCCC3CCC4)=O)C2C1)C(F)(F)F 63705,C1(NC(C(C)OCC#C)=O)CC2CCC(C1)N2C(c1cccnc1OCCO)=O 63706,n1(CC)cncc1C(=O)N(CCNC(C1(CN(C)C)CCC1)=O)C1CC1 63707,c1(CNC(N(C)C)=O)csc(=NC(CCO)C2CC2)[nH]1 63708,N1(C(c2ccc(OC)c(I)c2)=O)CC(NC(c2cnsn2)=O)CC(F)(F)C1 63709,CC(CC(=O)NC1(C)CC(NC(c2cc(C(N)=O)cs2)=O)C1)C(F)F 63710,c1(OC)ncc(C(N2CC3CCC3(CCNC(=O)C(C)(C)C(C)C)C2)=O)cc1C 63711,Cc1ccc2c(=NCCc3cscn3)[nH]c(=NC(C)c3cnn(C)c3C)[nH]c2c1 63712,C1(OC)CN(C(=O)C(C)=C(C)C)CCC1NC(=O)CN1CCCCC1C 63713,c1(C(CNC(C=CSC)=O)NC(c2coc(O)n2)=O)ccccc1C(F)(F)F 63714,Cc1cc(C(N2CC(C(N3CC=CCC3)=O)CC(C)C2)=O)nnc1C 63715,c1(C(N(CCC)CCNC(=O)CN2CCCCC2=O)=O)nnc(S)nc1C 63716,N1(C(c2c(OC)oc(C)n2)=O)CC(NC(c2ccc(C#N)s2)=O)C2(CC2)C1 63717,N1(C(c2n(C)ncn2)=O)CCCC(C2CN(C(=O)CCC3CCC3)C2)C1 63718,CC(C)(O)C(F)C(=O)NCC1CC(F)(F)CN1C(=O)CCCn1ccnc1 63719,c1(C(N2CCC(C)(NC(CN3CCC(C)CC3)=O)C2)=O)cccc2c1COCC2 63720,c1(CCC(F)F)nc(-c2ccccc2Br)nn1CCc1ccncc1 63721,N1(C(c2ccc(CC)[nH]2)=O)CCC2(COC(CNC(=O)CSc3nc[nH]n3)C2)C1 63722,C1(NC(CC2N(C(C)=O)CCC2)=O)CCC(CNC(c2cnnn2C)=O)CC1 63723,C1(CC=C)(NC(c2ccc(F)c(CC)c2)=O)CCCN(C(=O)C(C)(CC)OC)C1 63724,C1(C(N(CCC(=O)OC)C)=O)CCC(NC(c2ccn(C3CC3)n2)=O)C1 63725,c1(NC(C2CCN(Cc3ccncc3O)CC2O)=O)cnc(Cl)cc1[N+](=O)[O-] 63726,C(CNC(c1n[nH]c2c1COC2)=O)(CC(F)(F)F)NC(CC(C)N(C)C)=O 63727,c1(C(=O)NCC2N(C(C(C)SC)=O)CC2)ccc(S(=O)(=O)N2CCCCC2)cc1 63728,c1(NC(C(c2ccccc2)NC(=O)C(c2ccccc2)O)=O)csc(CO)n1 63729,Cc1cc(C)n(C(C)CN(CCC2(C)CCC2)C2CC2)n1 63730,CCC(C(=O)N1CC(CC(F)C(=O)NC(C)Cc2ccco2)C1)N(C)C 63731,C(=O)(CCCCCC#N)N1CC(CNC(C(C)(C)SC)=O)OCCC1 63732,C1(F)(C(=O)NC2CC(C)N(C(C3CN(C)C(=O)N3)=O)CC2)CCC(F)(F)CC1 63733,C(=O)(CC1CCOc2ccccc21)N1CC(C)C(NC(=O)C=CBr)C1 63734,Cc1cccc(NCC(N2CCC(CO)(NC(=O)CC(C)(F)F)CC2)=O)c1F 63735,N1(C(CCOCC)=O)CCCC2CN(C(c3ccc(CC(C)(C)O)s3)=O)CC12 63736,Cc1ccc(C(=O)N(C2CC(NC(=O)Cc3ccc(F)cc3F)C2)C)cc1CO 63737,c1(C(N2CCC(c3cn(-c4ncc(Br)cn4)nn3)C2)=O)cccc2oc(O)nc12 63738,c1(CC(=O)NC(C2(O)CN(C(=O)C=Cc3ccncc3)C2)C)ccc(N(C)C)cn1 63739,N1(C(c2c(C(C)C)scn2)=O)CC(CNC(C2CCCN(C)C2)=O)C2(CCC2)C1 63740,S(=O)(=O)(CCC(=O)NC1(C)CC(NC(c2sc(C)cc2OC(F)F)=O)C1)NCC 63741,c1(C(C)N(C(CSCCOC)=O)C(C2CC(C)=NO2)=O)cccc(Cl)c1.N 63742,C1(CC)OCCC1NC(=O)CCCNC(=O)CNC=O 63743,C1(CC(=O)NCC(O)CNC(c2c(Cl)n[nH]c2C2CC2)=O)CCCCC(=O)N1 63744,C1(C(N)=O)CN(C(=O)C(CCF)NC(=O)CC2CC(=O)NC2=O)CC12CC2 63745,C(CC(C)C(=O)NC(CNC(C1(c2cc[nH]n2)CCC1)=O)C(C)C)=CC 63746,CCCCCC(F)C(=O)N1CC(CNC(=O)CCN2CCOC2=O)CC(C)C1 63747,C1(NC(C(C)N(C(=O)CC2(O)CCOCC2)C)=O)CCOC(C2CC2)C1 63748,c1(CNC(C(c2ccc(F)c(Cl)c2)N)=O)cc(C(F)(F)F)ccc1Cl 63749,C1(NC(=O)NCc2c(C)cc(C#N)cc2)CCC2(CC1)OCCO2 63750,C12(NC(c3c(C)con3)=O)CCC(CC1)N(C(=O)CN1C(=O)CN(C)C1=O)C2 63751,Cc1nn(C)cc1C(=O)NC1CCCC1C(=O)NCC(O)C1(Cl)CC1 63752,C1(C(N(C2CCCN(C(=O)Cc3cscn3)C2)C)=O)CCCCCCC1 63753,C1(OC)CCC(C(N2CCCC(NC(c3cnn(C)c3C)=O)C2)=O)CC1 63754,CC1CCC(C(=O)NC(C2CN(c3ncc(I)cn3)CCO2)C)CC1C 63755,C(C)(C(=O)OC(C)Cc1cccnc1)(C1CC1)OC 63756,Cc1cccn2c(CC(=O)NC(C)CCNC(=O)C(C3CC3)C3CC3)cnc12 63757,Cc1nc(N(CC(C)CNC(=O)NC(=O)CCCN=[N+]=[N-])C)cc(Cl)n1 63758,c1(C(=O)NC(CNC(COCC=C)=O)C(C)C(C)C)cc(Cl)cc(Cl)c1Cl 63759,Cc1cnc(C)c(NC(C2(F)CCC(=O)CC2)=O)c1 63760,C1(C(=O)NC(CC)C)CC2CCC1N2C(=O)C=C=C(C)C 63761,N1(C(C(COC)C)=O)CC2CCCC(CNC(C3CCC(=O)N(C)C3)=O)C2C1 63762,CCN=c1[nH]c(C)c(C(=O)NC2CCC(N(C)C(C3CN(C(=O)NC)C3)=O)C2)s1 63763,c1(OC)ccc(Br)c(C(C)CC2CCCN2C(=O)COCC(F)F)c1 63764,Cc1scc(C(=O)N(C2CN(C(=O)CC3CCC34CCC4)CC2O)CCO)c1C 63765,CC(C)C(C(=O)NCC1C2CCCOC12)C(C)NC(c1cc(C#N)ccc1N)=O 63766,N1(C(c2cc(C)sn2)=O)CC(CNC(C2(O)CCOC2)=O)C(O)C1 63767,C(=O)(C1=Cc2cc(F)ccc2OC1)N1CC(NC(C2C3CCCCCCC23)=O)C1 63768,c1(OCC)cccc(CC(=O)NC2CC2CNC(=O)Cc2ccnc(OC)c2)c1 63769,N1(C(CSCC(N)=O)=O)CC2CCCCC2(CNC(=O)C=C2CCCCC2)C1 63770,c1(OC)cc(Cl)ccc1Cn1c(N2CCC(O)C(F)C2)nnc1C1CCCCC1 63771,Cc1nccnc1C(N1CCC(CC(=O)N(C(C)C)CC2CCC2)C1)=O 63772,C1(CC(NOCC#C)=O)CC(NC(C2CCN2CC)=O)C1(C)C 63773,C1(C(C(=O)NCCCOC=C)NC(=O)CCn2cccc2)CC=CCC1 63774,c1(CC(=O)NCC(CNC(COCC=C)=O)(C)C)cc(Cl)cc(Cl)c1 63775,C1(C(N2CC(CN(C(c3c(C)cc[nH]3)=O)C)OCC2)=O)CSc2ccccc2O1 63776,N1(C(=O)Nc2c(C)cc(N3CCOCC3)cc2)CCN2CCOCC2C1 63777,Cc1ccsc1CC(=O)NCCC1CC(NC(c2nocc2C(C)C)=O)C1 63778,C1(C(N2C(COC)CCCC2)=O)CCC(O)CN1C 63779,N1(C(c2n(CC)ncc2)=O)CC(C(=O)NCC(C)OCCO)CC12CCC2 63780,C1(CNC(C(C2CCCC2)OC)=O)(NC(=O)CCc2cccn2C)CCCCC1 63781,c1(C(N2CCC3(CN(C(c4cc(C)ns4)=O)C3)C2)=O)cn2cccc(F)c2n1 63782,O=C(C1=CC2(CCOC2)C1)NC1CCCCN(C(C2(C3CC3)CC2)=O)C1 63783,C(=O)(CC1CCOc2ccccc21)N1CC2(CC(NC(C3N(C)CCC3)=O)C2)C1 63784,C12(CS(=O)(=O)C1)C(=O)N2.c1(C(=O)OC)ccc(C(C)(CO)OC)o1 63785,C(c1ccc(F)c(Cl)c1)=CC(=O)NC1C(C)CN(C(=O)CN2CSCC2=O)C1 63786,C(CCCC(=O)N1CCSCC1C(=O)NCCC(O)CCO)OCC 63787,CC1CC(C(N2CC(O)(CCNC(=O)CCc3nc(O)n[nH]3)C2)=O)CCS1(=O)=O 63788,CN1CC(NC(C2CC(CNC(=O)CCC3CC3(F)F)C2)=O)CC1=O 63789,CCC(C(=O)NC1CC(NC(=O)COC2CCCOC2)C1)C(C)(C)CC 63790,c1(C(=O)OCC)cc(=NCCC2CC3(CCS(=O)(=O)CC3)CO2)[nH]cc1C#N 63791,c1(OC)cc(C(O)CNC(=O)NCCCCc2ccc(C(C)(C)C)o2)ccc1O 63792,c1(CC(=O)NC(C)(C)C)ccc(C2CC2)cc1.C1CC(O)CNC(=O)C(C)N1C 63793,S(=O)(=O)(C1CCNC(C)C1)Nc1cc(C)cc(C(=O)O)c1 63794,N1(C(C=C(CC)CC)=O)CCC2CCCC12C(N1CCCC1CSC)=O 63795,C1(CC)CN(C(c2c(Cl)cccc2Cl)=O)CCN1Cc1cccc(I)c1 63796,C(=O)(CCCCCNC(C1CC(C)(F)C1)=O)NCCCOCCCC 63797,c1(C(=O)OC)ncccc1S(C)(=O)=NC(=O)C1CC1(C)C(C)C 63798,C1(C)(C(=O)NC(c2n[nH]c(=N)s2)C)CC12CCN(c1cccc(C3CC3)n1)CC2 63799,Cc1c(C(N2CCC(NC(c3cc(Cl)ccc3O)=O)C2)=O)ccc2c1CCC2 63800,c1(C(N2CC(NC(CCCNC(C)=O)=O)C(O)C2)=O)ccc(N(C)C)nc1Cl 63801,CC1CN(C(C2CC23CCSCC3)=O)CCN1C(=O)CCCC1CCCCC1 63802,C=CC(CC(=O)NC(C)CCCCNC(c1cc(OC)no1)=O)c1ccccc1 63803,c1(C(=O)NCCC2CCCN(C(C(CCC)O)=O)C2)cc(=O)c2c(cnn2C)[nH]1 63804,C1(N(C(=O)COOC(F)(F)F)C)CCN(C(C2CC2c2ccn(C)n2)=O)CC1 63805,N1(C(c2c(OC)csc2)=O)CC(NC(C2(c3ccccc3Cl)CCC2)=O)C(C)C1 63806,C=CCCC(CC(C)C)C(=O)NCCOCCNC(=O)C(C(C)C)n1cnnn1 63807,C1(C(C)NC(=O)C(C)N(CC(F)(F)F)C)CCN(C(C2(F)CCC2)=O)CC1 63808,C1(NC(C2CCCCCCC2)=O)CCN(C(C2CCS(=O)(=O)C2)=O)C12CCC2 63809,Cc1n[nH]c(C)c1C(C)NC(=O)C(C1CCCC1)NC(c1cc(C(N)=O)[nH]n1)=O 63810,C1(CC)CN(C(c2cc(C3CC3)cnc2Cl)=O)CCN1C(=O)C(C)n1cccn1 63811,c1(N(CCCCC=C)C)cc(=NCC(Cc2ccccc2OC)CO)[nH]c(C)n1 63812,CC1CC(C)CN(C(=O)CNC(=O)C(F)CN(C(C)(C)C)C)C1 63813,C1(C(=O)NCC(CC=C)NC(C2(CCOC)CCCC2)=O)CCCC2(CC2)C1 63814,n1(CC(=O)NC2C(C)CN(C(=O)CN3CC=CC3)C2)ccc([N+](=O)[O-])n1 63815,Cc1ccc(C(=O)NCCC(C)NC(c2cnn(CC(C)C)c2)=O)cc1F 63816,CN1CCC2(CCN2C(C23CC(C(=O)Nc4ccc(Cl)cn4)(C2)C3)=O)C1 63817,N1(S(CC)(=O)=O)Cc2ccccc2CC1C(=O)NCc1cc2c(cc1Cl)OCO2 63818,Cc1cnc(C(=O)NC2CCN(Cc3cc(Cl)ccc3Cl)CC2C)c(C)c1 63819,CN1CCC(NC(=O)CC(C)(C)C)C12CCCN(C(C1(O)CCCCCC1)=O)C2 63820,C1(NC(CCNC(N)=O)=O)CCOC12CCN(C(=O)CCC1CCC(=O)C1)CC2 63821,c1(N2CC3(C(NC(C4C(C)(Br)C4)=O)CCS3)C2)nc2cc(F)c(F)cc2s1 63822,N1(C(c2nc(CC)sc2)=O)CC2(CCC2NC(c2cc(C(N)=O)cc(C)c2)=O)C1 63823,c1(NC(C(=O)NC2COCC2CO)=O)ccc(F)cc1OC(F)F 63824,c1(C(N(C2(COC)CC2)CCO)=O)cnn2ccncc12.C1(CC(=O)O)CCCO1 63825,CCC(C)(C)C(=O)NCC(C)(C)NC(c1cnc(C2CC2)[nH]1)=O 63826,N1(C(CC2(OC)CC2)=O)CC(CNC(C2CC2C(F)(F)F)=O)C2(CC2)C1 63827,c1(OC)ccc2c(CC(N3CCC(CCNC(=O)CCCSC)C3)=O)coc2c1 63828,N1(C(c2cncnc2)=O)CC2CC1(CN(C(C1(C3CCCCO3)CC1)=O)CC)C2 63829,c1(NCC2C(NC(c3cnn(C)c3C3CC3)=O)CCC2)ncc(Br)cc1[N+](=O)[O-] 63830,c1(CC(=O)NC2CN(C(C3CCCC4CC34)=O)C2)ccc2c(c1)OCCO2 63831,C1(C(=O)OCC)CCN(C(c2ccc(-c3ccc(F)c(C#N)c3)o2)=O)C12COC2 63832,C(=O)(CC(C)(C)SC)NCCC1N(C(C(C)OCCOCC)=O)CCC1 63833,C=Cc1ccc(C(N2CCC(NC(c3ccccc3CC(C)C)=O)CC2)=O)cc1 63834,c1(-c2nn[nH]n2)ccc(Cl)cc1.C12(C(=O)OC)CN(C1)C(=O)C1(CC1C)N2 63835,N1(C(c2c(CNC(c3cc(C)ncn3)=O)ocn2)=O)CC2CCC(O)C2C1 63836,C1(C)(CNC(CCOC(C)C)=O)CCCN1C(=O)Cc1cn(C)nn1 63837,c1(C(N2C(CNC(c3c(OC)c[nH]n3)=O)CC2)=O)[nH]c(-c2cccc(C)c2)nc1C 63838,C(c1ccc(F)c(F)c1)=C(C(N1C2CN(C(C3(COC)CC3)=O)C(C2)C1)=O)C 63839,N1(C(C2CN(C(N)=O)C2)=O)CC2CCCC2C1C(N1CCC(n2cnnn2)C1)=O 63840,N1(C(C(CCSC)OC)=O)CCC2(CC1)CCN(C(C1(CO)CCCC1)=O)CC2 63841,S(=O)(=O)(c1c[nH]c2ncccc12)NCC(N1CCC(NC(C)=O)C(C)C1)=O 63842,N1(C(CS(CC)=O)=O)Cc2ccccc2C1CNC(=O)CNc1cccnc1 63843,N1(C(C2N(C)CC2)=O)CCCC(c2cc(OCC(F)(F)F)n[nH]2)C1 63844,C1(N(c2ccc(F)cc2)C(=O)C(O)C2CN(CC)C2)C2CCC(C2)C1C 63845,c1(CC(CO)NCCCCC2CCOCC2)ccc2c(c1)OCCO2 63846,C1(CC(=O)Nc2cccc(CNC(c3c(C)snn3)=O)c2)CS(=O)(=O)CCN1C 63847,c1(C(=O)OC)cnc2n1CCN(C(=O)C(C1CC1)Nc1ccc(O)c(CO)c1)C2 63848,c1(NC(C2C(C)C2)=O)cnc(F)cc1C(N1CC2CC2C1C#N)=O 63849,C1(NC(C(C=C)(F)F)=O)CC2(CCCCN2C(c2coc(CC)n2)=O)C1 63850,C1(C(=O)NCCC2(O)CN(C(CCSC)=O)C2)CC2CC(C1)CC(F)(F)C2 63851,C1(C(=O)NCCOC2CCN(C(c3n(C)ncc3)=O)C2)CC2(C1)CC2F 63852,N1(C(c2ncccc2C)=O)CCC2(CC(C(=O)N(CC(C)C)CCO)=NO2)C1.CO 63853,CN1CCC(C(N2CC(O)(c3cnn[nH]3)C2)=O)(NC(C2CC=CCO2)=O)C1 63854,CCC(CC(=O)N(CC)CC1CCCN1C(c1cn(C)c(C)n1)=O)OC 63855,c1(CN(C(=O)NC2CN(C(C)=O)C2)C)ccc(-c2ccccc2)[nH]1 63856,N1(C(c2scc(OC)c2)=O)CC2(CCC2)CC1CNC(=O)C(C(C)(C)C)N(C)C 63857,c1(C(=O)NCCC2(CNC(c3n(CC)ccn3)=O)CC2)cc2n(n1)CC(F)C2 63858,n1(CCC(=O)N(C2CN(C(c3c(C)nns3)=O)CC2F)C)cnc([N+](=O)[O-])c1 63859,C=C1CCC(C(=O)N(CCC(=O)N(C)CC2(OCC)CCCC2)CC)CC1 63860,c1(C(C(=O)NCCOC)N(CCCc2ccccn2)C)cnc(C2CC2)[nH]1 63861,CCCCC(F)C(=O)NC(C)CC(=O)NC(C(=O)OC)C1CCC1 63862,c1(C(N2CCC(NC(C(CC)O)=O)C3(C2)CCC3)=O)cc2cccnc2cc1F 63863,N1(C(CCNS(C)(=O)=O)=O)CCCC12CN(CC(N)=O)C2 63864,c1(C(=O)NC2CC(C)N(C(=O)CCCCO)CC2)ccc2c(c1)CCC=C2 63865,Cc1ncc(C(N2CC3CC(NC(c4nccc(Cl)c4F)=O)C3C2)=O)c(O)n1 63866,c1(C(=O)NCCCN(C(=O)C(O)c2ccco2)C)c[nH]nc1S(N)(=O)=O 63867,N1(C(CNC(c2c(C)occ2)=O)=O)CCC2CN(C(=O)CCCN(C)C)C2C1 63868,c1(CC(N2C(C)CC(NC(C(c3cccc(C)c3)O)=O)C2)=O)cc(C)ccc1O 63869,CC1(C)CN(C(=O)CC2(C#N)CC2)C(CNC(=O)Cc2c(Cl)cccc2Cl)CO1 63870,C1(CNC(c2ccc(SC)s2)=O)CC(NC(c2nncn2CC2CC2)=O)C1(C)C 63871,N1(Cc2nnc(C)o2)CC(NC(=O)Nc2ccc(CO)cc2)CC1=O 63872,c1(C(N2C(CNC(c3nc(C)sc3C)=O)C3CCC2C3)=O)ccc2snnc2c1 63873,C1(C(=O)NC(C)(C)CCCNC(=O)C=Cc2ccccc2)CCC2(CCOC2)O1 63874,C12(NC(C3SCCS3)=O)CC(CO)(C1)OC21CN(C(C2(n3cnnn3)CC2)=O)C1 63875,C(=O)(CC(C)C(F)F)N1CCC(OCCNC(C(CC#C)C)=O)CC1 63876,c1(CC(=O)NC(C(C)(C)NC(C(CC)C#N)=O)C)ccc(Br)c(OC)c1 63877,N1(C(C2C(C(N)=O)COC2)=O)CC2CCCC2(NC(=O)CCNC(=O)C=CCl)C1 63878,c1(C(C)N(CCO)C=O)ccccc1Cl.c1(C(CCCC(=O)N)O)ccccc1 63879,C=CC1(CNC(=O)C(O)CNC(=O)CCC2CCC2)CCCCC1 63880,C1(C(=O)NC(C(C)C)(C)CNC(=O)CC(=O)N(C)C)CC2C(C1)C2(F)F 63881,C1(N(C(C2C(C)CC(C)O2)=O)C)CCCCN(C(C2C3CC4C(C3=O)C24)=O)C1 63882,C1(NC(CNC(N)=O)=O)C=CCC(C(=O)NCCOc2cccnc2)C1 63883,Cc1cn2cc(C(=O)NCC3CCN(C(=O)COCCN(C)C)C3(C)C)sc2n1 63884,c1(C(N2CCN(C(C3(O)C(C)(C)C3)=O)CC2)=O)ccnc2[nH]c(O)nc12 63885,c1(-c2nc(CC(C)(C)CO)nn2CCCCO)cc2ccc(Cl)nc2s1 63886,N1(C(CCNC(=O)OC)=O)CCC(CO)(NC(c2ccc(OC)cc2)=O)C1 63887,C(C)(CC(=O)NCC1(NC(c2ccc(Br)o2)=O)CCC1)(C(F)F)N(C)C 63888,C(=O)(CC(C)CC(C)(C)C)N1CCC(NC(c2c(N)sc(C)c2C)=O)C1 63889,c1(NCC(=O)NC2(C=O)CCOC2)cc(NC(C)C)nc(C(C)C)n1.CCO 63890,N1(C(CS(CC)(=O)=O)=O)CCC(C)N(C(=O)C(N2CCCCC2=O)C)CC1 63891,C1(NC(c2cc(-c3nc(C)sc3)sc2)=O)CCC(NC(c2cnn(C)c2)=O)CC1 63892,C1(NC(COCC#C)=O)CN(C(C2CCCC(O)C2)=O)CC2(CCC2)C1 63893,c1(NC(C(=O)NC(COCC)CO)=O)ccc(C)c(O)c1 63894,C#Cc1cccc(C(=O)NC(c2cccc(Br)c2Cl)C(=O)OC)c1Cl 63895,C(=O)(C#CC1CCOCC1)NC(C1CN(C(C2CCc3nnnn3CC2)=O)C1)C 63896,c1(C(N2CC3(C(NC(c4cn5ccnc5s4)=O)CC3)C2)=O)c(F)ccc(F)c1Cl 63897,C1(NC(C2(NC(c3cc(C)on3)=O)CC(F)(F)C2)=O)CC2(CCC2)C1O 63898,C(C(C(=O)NC1CC2CCC1C2)N1CCC(OC)CC1)(C1CCOCC1)OC 63899,c1(NCCOC)nc(OC2(C)CCOCC2)cc(=NCCN2CCCC2=O)[nH]1 63900,c1(CC(=O)N)ccc2[nH]ccc2c1.N1(C(C(CC)=CC)=O)CC(OCC)C(SC)C1 63901,C#CCC(CC(=O)OC)NC(C1CCC(CNC(=O)Cn2cccc2)O1)=O 63902,N1(C(C(CC)C)C(=O)Nc2ccccc2Cl)CCc2ncn(C)c2CC1 63903,C1(CNC(Cc2c(C)nc(S)s2)=O)COCCN(C(C23CCC2C3)=O)C1 63904,C1(CC(=O)NCCC(CNc2nccc(C3(C)CC3)n2)(F)F)CCCNC(=O)C1 63905,c1(C(=O)NC2C(NC(c3c(C)c[nH]n3)=O)CCC2)ccc(OC(C)C)nn1 63906,C1(CC=C)(C(N2CCN(C)CC2)=O)CCN(C(=O)C(=Cc2cnn(C)c2)C)C1 63907,N1(C(CN2CCN(C)CC2)=O)CC(CC(=O)NC2CCCC2N=[N+]=[N-])CC1(C)C 63908,C1(OCCCNC(CC2(C#N)CC2)=O)CCN(C(C23CCCCC2C3)=O)CC1 63909,c1(C(=O)NCC(C)CNc2cnc(C#N)cn2)ccc(C2CC2)cc1F 63910,N1(C(C=C(CC)C)=O)CCC2CCC12CNC(c1ccnn1C)=O 63911,C1(NC(C(CC)O)=O)CC=C(C(=O)NCCc2cncn2C)C1 63912,c1(-c2cc(C(N3CC(NC(C4CC=CC4)=O)C(F)C3)=O)on2)cccc(Cl)c1Cl 63913,c1(-c2nc(CCCCC)nn2CCCO)cccc2occ(Br)c12 63914,CCC(F)(F)CC(=O)NC1CS(=O)(=O)CC1NC(c1ccc(N)c(Cl)c1)=O 63915,N1(C(C(CCC)CNC(c2cc(CO)on2)=O)=O)CCOCC(F)(F)C1 63916,C=CC(CC)CC(=O)N1C2CCC1C(NC(=O)CS(C)(=O)=O)C2 63917,C1(CCOC)(NC(c2nc(C)c(C)s2)=O)CCN(C(=O)CCNC(C)=O)CC1 63918,N#CC1CN(C(C2(C3CC3)CC2)=O)CC1NC(c1c(F)cccc1Cl)=O 63919,Cc1ccc(F)cc1C(=O)C(=O)N(C1CCN(C(C2(C#N)CC23CCC3)=O)C1)C 63920,CC1CCN(C(=O)CCNS(C)(=O)=O)CC1CNC(c1ccc(F)c(Cl)n1)=O 63921,c1(C(=O)NC(CN(C(CN(CC)CC)=O)C)C)cc2c(s1)CC(C)(C)C2 63922,C1(C(=O)NCC(C)N(C(=O)CC2CC(=O)NC2=O)C)CCCOC1c1ncc[nH]1 63923,c1(C(=O)NC23CCN(C(CS(CC)(=O)=O)=O)CC2C3)ccn2cc(C)nc2c1 63924,c1(N(C)CC)ccc(CCCCNC(c2ccccc2SCCOC)=O)cc1 63925,c1(C(=O)NCCC2CC(NC(Cn3c(C)nc(C)n3)=O)C2)c(C)cccc1F 63926,N1(C(c2c(OC)ccc(F)c2)=O)CC2(NC(C3OCC3(C)C)=O)CCCC2(F)C1 63927,c1(C(N2CC(SC)C(NC(c3cccn3C)=O)C2)=O)n[nH]c2ccc(Cl)cc12 63928,C(=O)(C1=CCS(=O)(=O)C1)N1CCCC(NC(C2C3(CC(C)(C)C3)C2)=O)(CO)C1 63929,c1(COC)nc2n(n1)CC(NC(c1cccc(C(F)F)n1)=O)CC2 63930,C(=O)(CC(C(C)C)c1ccon1)N1C(C2(NC(c3c(C)c[nH]n3)=O)CC2)CCC1 63931,N1(C(C(=O)NCCOCCC#C)=O)CC(=O)N2CCOCC2C1 63932,C1(C2(O)CCN(c3nc4cccc(C)c4o3)CC2)(NC(COC(CC)C)=O)CC1 63933,C12(C(=O)NCC3N(C(=O)CC4CC4)CC=C3)CC3CC(C1)CC(O)(C3)C2 63934,c1(CC(=O)NC(C2(O)CCN(C(=O)C3=CSCS3)C2)C)cn2cc(F)ccc2n1 63935,Cc1nc(-c2ccccc2)[nH]c1C(=O)N(CCCNC(c1ccsc1)=O)CCO 63936,c1(C(N(CCOC)CCNC(=O)C(C)SC(F)(F)F)=O)ccoc1Cl 63937,C(=O)(C1CCCc2nccn21)N1CCC(CCNC(c2c(CC)non2)=O)C1 63938,C(=O)(CC1COc2cc(O)ccc21)N(CC(C)NC(=O)CCC(=O)NN(C)C)C 63939,N1(C(c2ncccc2Br)=O)CCC2(CCC2N2CCC23CCCCC3)CC1 63940,N1(C(C2(C(=O)OC)CC2)=O)CCC2C(C1)CN2C(C1CNC(=O)N1C)=O 63941,c1(CNC(=O)NC2C(COC)C2)ccn2cncc2c1 63942,N#CC1(C(=O)NCC2CCN(C(=O)CCC3CCCCO3)CC2)CC2C=CC1C2 63943,c1(C(N=S(C)(=O)C2CNC2)=O)ccc(O)c2c1CCCC2 63944,N1(C(C(Cc2ccoc2)NC(c2c[nH]c(=N)o2)=O)=O)CCN2C(=O)NCC2C1 63945,C1(CC(=O)NCC(CC)(C)NC(c2csc(Br)n2)=O)CC2CCC1O2 63946,C=CC(CC)CC(=O)NCCN(C(=O)CCOc1cccc(C(N)=O)c1)C 63947,N1(C(c2nc(-c3c(C)snc3)sc2C)=O)CCC(O)(C2(c3nn[nH]n3)CC2)CC1 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64107,N1(C(C(CC)NC(C)=O)=O)CCC12CN(C(C1CCC(C(F)(F)F)O1)=O)C2 64108,C1(CC(=O)OC)Cc2ccccc2CN1C(c1cnc2c(Cl)cccn12)=O 64109,C1(C(=O)Nc2cccc(Cn3ccnc3)c2)Cc2cc(C(F)(F)F)ccc2O1 64110,c1(C(=O)NCC2(NC(C(F)=C(C)C)=O)CCCCC2)cccc(S(N)(=O)=O)c1 64111,c1(C(N2C(CN(C(c3c(CC)n(C)cc3)=O)C)CCC2)=O)cnc2cc[nH]c2c1 64112,c1(C(N2CCC(NC(C3CCCC3(F)F)=O)(CO)C2)=O)ccn2c(O)nnc2c1 64113,C1(N(C(c2csc(CO)n2)=O)CC)CCN(C(=O)COC(C)=O)CC1 64114,C(CNC(=O)CCCSC)(CC(F)(F)F)NC(c1ccc(OCC=C)cc1)=O 64115,C1(C(=O)NC(CCNC(=O)CCc2cc(Cl)cs2)CO)CN2CCCCC2CO1 64116,Cc1cccc(C(=O)NC2(C)CCN(C(C3CC(=O)N3)=O)C2)c1N 64117,C=C(Cl)CC(C(=O)NCC(C)C(=O)OC)NC(c1ccn(COC)n1)=O 64118,c1(NC)scnc1C(=O)NC(CO)C(C)NC(=O)C(CC)OC 64119,C1(CCNC(c2c(C)snc2)=O)CCCCN1C(=O)C(C)Oc1ccccc1Cl 64120,C(=O)(C(CC(C)C)NC(=O)C(C)CCOC)N(CC(CCC=C)O)C 64121,C1(NC(c2ccc(C3CC3)nc2)=O)CC2(C1)CC2NC(c1ccc2c(c1)CC2)=O 64122,C12(CNC(CSC)=O)CN(C(=O)C=Cc3ccc(C)c(C)c3)CC(F)(C1)C2 64123,C1(S(N)(=O)=O)(C(=O)NC2CCC(NC(c3cnn(C)c3C(F)F)=O)C2)CCCC1 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64141,C1(C(=O)NCc2cccnc2O)CSCCN1C(c1ccnc(Br)c1)=O 64142,C1(CNC(C2N(C(C)=O)CSC2)=O)CCCCN1C(=O)CC1CCC(C)(C)C1 64143,c1(SCC)ccc(C(=O)NCCCn2cc(C3(F)COC3)nn2)c(Br)c1 64144,N1(C(c2ccc(OC)o2)=O)CCCC(C2CCCCN2C(C2CCCOC2)=O)C1 64145,CC1(C)C(NC(=O)CCOc2cccc(F)c2)CC1NC(=O)CCC1CCCO1 64146,c1(-c2scc(C(N3CC(C)(NC(C4C5CCCC45)=O)C3)=O)n2)ccc(F)c(F)c1 64147,C(=O)(C(CCS(C)=O)N(C)C)NCCC(C)CCNC(c1cnnn1C)=O 64148,N1(C(C)COCC(=O)NCCCN(C(=O)C=CC(F)(F)F)CCO)CCOCC1 64149,Cc1nn(C)cc1S(=O)(=O)NC(c1cc(N(C)C)nc(Cl)c1)=O 64150,C12(NC(c3cc(O)ncn3)=O)COC(C1)C(NC(c1scnc1Cl)=O)C2 64151,N1(C(c2cnc(OC)nc2C)=O)CC2CC(NC(C3CN(C(C)=O)C3)=O)CC1C2 64152,C1(C)(CC)CCC(C(=O)NC2C=CCN(C(C3CC=C(C)CC3)=O)C2)O1 64153,C(=O)(C(C(F)(F)F)C(F)(F)F)NC1CCN(C(CC2CCN(C)C2=O)=O)C1 64154,C1(C(=O)NCCCC2N(C(CSCC)=O)CCC2)CC2CCC1CC2(F)F 64155,C#CCCCCCNC(=O)C(F)C1CC(NC(c2ccc(C=C)cc2)=O)C1 64156,c1(C(=O)NCC(CO)NC(c2n(CC)ccc2)=O)cnc(N)cn1 64157,c1(C(=O)NCC(C)N(C(c2n(CCC)ncc2)=O)C)ccc2c(c1)C(=O)CCN2 64158,N1(C(C)C)CC(NC(c2cc(CNC(C3CC3(F)Cl)=O)[nH]n2)=O)CC1=O 64159,C(CC(CC)CC)(c1n(CCCC)nnn1)Nc1cc(CC)ccc1C 64160,c1(C(=O)NCC2C(NC(C(CC)NC(C)=O)=O)CCCC2)ncc2[nH]ncc2n1 64161,N1(C(Cc2cc(C(C)C)no2)=O)CCC(C(C(C)C)NC(c2csnn2)=O)CC1 64162,C12(C(N3CCC(C(C)NC(C=C(C)Cl)=O)C3)=O)CC3CCC(CC(C3)C1)C2 64163,Cc1cccc2c(CN3CCC(NC(c4cnn(C)c4)=O)C(O)C3)c[nH]c12 64164,C(c1nc(C)c(C)[nH]1)=CC(=O)NC1C(CC)N(C(c2ncc(C)cc2O)=O)CC1 64165,C1(CNC(c2ncncc2Cl)=O)C2CCC(C2)N1C(C12CC3CC1C2C3O)=O 64166,Cc1cc(=NCCC2CCC(=O)N2)[nH]c(N2CCN(CC(C)C)CC2)n1 64167,CCCC(CCC)C(=O)NC1CCCC(NC(c2cc(C(F)(F)F)on2)=O)C1 64168,CC1CCCCC1(C)C(=O)NCCOCCN(C(=O)COc1cncc(Cl)n1)C 64169,c1(C(=O)NCCN(C(C(CCC)(C)O)=O)CC)ncnc2c1CCC2 64170,C1(CNC(C(CC)CC)=O)CN(C(c2ccnc(C3CC3)n2)=O)CC1(C)C 64171,N#Cc1cc(C(=O)NCC2(NC(=O)C=CBr)CCC2)c2c(c1)OCCO2 64172,c1(N2CC3CN(C(c4cc(C)nc(C)c4)=O)C3C2)ncnc2n[nH]cc12 64173,c1(CC)cccc(C(=O)NCC2(CNCc3cc(CC)no3)CCOCC2)c1C 64174,Nc1cc(C(=O)NCCNC(=O)CC2C=CCC2)cc([N+](=O)[O-])c1 64175,c1(C(=O)OC)ncc(Cl)nc1NC(c1scnc1NC(c1[nH]cnc1C)=O)=O 64176,C1(NC(c2n[nH]c(C)c2C)=O)CCN(C(c2ccc(C(C)C)c(F)c2)=O)C(C)C1 64177,c1(CN2C(C(N(CC)CC)=O)CCCC2)c(F)cc(F)cc1Br 64178,c1(C(=O)Nc2c(C)nccc2)c[nH]c2cc(-c3ccsc3C#N)cnc12 64179,c1(C(=O)NC(CC=C)CNC(C2(OC)CCSC2)=O)cn2ccsc2n1 64180,c1(C(N2CCC(N(C(CN(CC)CC)=O)C)C2)=O)nnc(O)c(Br)c1O 64181,C(=O)(C1=CCC(C)(C)CC1)NC1C(C)N(C(=O)CCNC(=O)CO)CCC1 64182,C1(C(=O)NC2(C)CN(C(C(c3cscn3)N(C)C)=O)C2)CC2CCC(C1)C2(F)F 64183,c1(C(=O)NCC(CC=C)NC(=O)CC(C)n2cccn2)cnc2cccc(C)n12 64184,n1(CC)ccc(CC(=O)NCC(CNC(C2CC=CCC2)=O)OC)n1 64185,N1(C(C(C=C)C)=O)CCN(C(c2cn(C)nn2)(C)CNC(=O)CO)CC1 64186,Cc1cnn(C)c1CC(=O)NCC1(C)CC(NC(c2ccc(N(C)C)nn2)=O)C1 64187,c1(C(N2CCC(NC(C(C(C)(C)C)OCC)=O)(CF)C2)=O)cc(C)c(N)cc1Cl 64188,c1(NCC(CNC(C(C(CC)C)O)=O)O)ncnc2sc3c(c12)CCCC3 64189,N1(C(C2CCN(C(C3CCC(CC)CC3)=O)C2)=O)CCCNC(=O)C12CC2 64190,c1(C(=O)NCC2N(C(c3nccc(CC)c3)=O)CCCC2)cc(Cl)c(Cl)cc1O 64191,c1(C(=O)NC2(C)CN(C(C34CCCC3CCC4)=O)C2)cc(C#N)ccc1F 64192,C(=O)(C(COC)COC)NC1C(NC(c2cc(OCC)no2)=O)CCC1 64193,C1(CCN(C(C2CCN(C(=O)NC)C2)=O)C)CCCCN1C(c1ccc(F)s1)=O 64194,C1(CCCNC(C2C(CC)CCO2)=O)CCCCN1C(C1CC(N(C)C)C1)=O 64195,N1(C(C(OC)OC)=O)CCC2(CCC(NC(c3[nH]c(O)nc3C)=O)C2)CC1 64196,C(CCCC(C)(C)C)NC(CC(CNC(C1CC1(C)C)=O)OC)=O 64197,Cc1nn(C)c(C)c1C(=O)NC12CC1CN(C(=O)CC1CCC(C)(C)CO1)C2 64198,c1(COC)nc(NCc2cnn(CCF)c2)cc(=NC(C)C2CCCO2)[nH]1 64199,C(=O)(CC1=CCCCC1)NCCNC(C1(CCC)CCC1)=O 64200,C1(NC(c2cc3c([nH]2)CCCC3)=O)CCN(C(C2(O)COC2)=O)CC12CCC2 64201,C1(NC(COCCCC)=O)CC2CCC(C1C)N2C(c1cnn(CCF)c1)=O 64202,C(N=c1ccc(NC(c2cncc(Cl)c2)C)c[nH]1)c1c(SC)cccc1 64203,CCC(CC(=O)NCC1C=CCN1C(c1cc(OC)cs1)=O)C(C)C 64204,Cc1nc(C(=O)N(C)CC2CCCCN2C(=O)Cn2ncccc2=O)c(C)s1 64205,C1(C(N2CCC(NC(C3CCOCC3)=O)C2)=O)(OCC)CCOCC1 64206,CCC(F)(F)CN(C(C1C=CCC1)=O)C(c1cc(C2CC2)[nH]n1)=O.CCC 64207,c1(C(=O)NC2CCN(C(C3NC(=O)OCC3)=O)C2)ccc2nc(O)[nH]c2c1F 64208,Cc1cccc(Br)c1C(C(=O)N(C)CCN(C)C)NC(=O)CC1(O)CCCOC1 64209,c1(C(=O)NCCC(C)(C)NC(C2C(C)OCC2)=O)ccc(C(F)(F)F)cn1 64210,CC1(C)CCN(C(C2CC3C2CCN3Cc2ccccc2)=O)CC1C(=O)O 64211,CCC(CN(C)C)CC(=O)NC1(CO)CN(C(C2CC(OC3CC3)C2)=O)C1 64212,c1(C(=O)NC2CCCC(NC(c3ccc(CC)o3)=O)C2)ccc2ccccc2c1 64213,C1(NC(CC2CN(C(C)=O)C2)=O)CCC2CCN(C(c3csnc3C)=O)C1C2 64214,N1(C(C(C)CN(C(=O)CSCCC(F)(F)F)C)=O)CCCCC(CO)C1 64215,N1(C(C(C)SC)=O)CC2(CCCC2)C1C(=O)NCCc1ccccc1 64216,C(c1ccc(OC)cc1OC)=CC(N1CCCC(NC(C(CC)OC)=O)C1)=O 64217,C(=O)(C(C)(C)COCC)N(CC(=O)NC(C=C)CO)CCOC 64218,C1(N(C(CCOCCOC)=O)C)CCN(C(c2cnn(C)c2N)=O)CC1C 64219,N1(C(=O)COCC2CCOC2)CC2(C1)CN(C(=O)C(F)C1CCC1)C2 64220,C1(NC(Cc2n(C)ncc2)=O)CC2CN(C(c3ccn(C(C)(C)C)n3)=O)CC12 64221,N1(C(Cc2nnc(C)o2)=O)CC2(CO)CC1(C(=O)NCCOCC(C)C#N)C2 64222,C1(F)(CNC(C2N(C)CCC2)=O)CCN(C(c2cnc(-c3ccccc3)s2)=O)C1 64223,C1(CNC(C(C=CC)O)=O)CC2COCC2N1C(=O)CC1CCC2CC2C1 64224,c1(C(N2CC(C(C)NC(=O)CC(O)C3CC3)OCC2)=O)ccc2nc(O)[nH]c2c1 64225,N1(C(C)C)CCCCC1C(=O)NCCCN(C(=O)C(C1CCOCC1)C)C 64226,C(=O)(C(F)C(C)(F)F)N1CC(C)(C(N2C(C)(COC)CC2)=O)C1 64227,N1(C(c2cc(C)oc2C)=O)CCCOC(CNC(=O)Cc2cocn2)C1 64228,C(=O)(CC1=CCOCC1)N1C(CCNC(CCC(=O)OCC)=O)CSCC1 64229,CCC(CC)C(F)C(=O)NCCCC(O)C(=O)N(C1CC1)C(C)C1CC1 64230,C12(NC(CC3CC(=O)NC3)=O)CCCC1CN(C(c1c(O)cc(Cl)cc1F)=O)C2 64231,Cc1cc(C=CC(=O)NCC(O)CN(C(=O)C(C)c2ccsc2)C)c[nH]c1=N 64232,C(=O)(C(O)CCNC(c1cc(C2CC2)on1)=O)N1C(C=C)CC1 64233,c1(C(N(C(CN(C(C2(OC)CCC2)=O)C)C)C)=O)ccccc1CC(C)(C)C 64234,CCC(CC(=O)NCCC(C)(C)NC(C1(C)CCNC1=O)=O)C(=O)OC(C)(C)C 64235,N1(C(Cc2scc(C)n2)=O)CCCC(C)C1CNC(=O)Cc1cnoc1 64236,c1(NC(=O)NCCN(C(C(=O)NCCOCCC=C)C)C)cc(Cl)ccn1 64237,c1(C(=O)Nc2ccc(CNC(CC(=C)C)=O)cc2)cc(N)cc(F)c1 64238,C(=O)(CC(CC)C(C)C)N1CCN(C(c2c(OC)cncn2)=O)C(C2CC2)C1 64239,N(C1CC(C)n2ncnc21)CCC(=O)NC(C)Cc1ccccc1 64240,C(CCCC(=O)NC1CCCC1NC(=O)Cc1ccc(C)o1)OC 64241,c1(SC)nc(N(C(C)CCNC(=O)C(CO)NC(N)=O)C)cc(Cl)n1 64242,CN1C(=O)OCC1C(=O)NCC12CC1CN(C(=O)CC1CC1C(F)(F)F)C2 64243,C(C(C(=O)NC1CC(N(C(=O)CCF)C)C1)C(F)(F)F)OC 64244,C(c1cocn1)=CC(=O)N(CCOC)CCNC(=O)CC1(OC)CCC1 64245,c1(CC)cc(C(=O)NC(C)CNc2cnncc2C(=O)OC)c2c(c1)CCO2 64246,c1(N(CC(N2CC(N(C)C(C3CC3F)=O)C2)=O)C)ccccc1 64247,c1(C(=O)NC2C(C(C)(C)C)N(C(=O)C(=O)N(C)C)CC2)nnn2c1CCCC2 64248,C(N=c1[nH]c2ccc(N)cc2s1)C1CCCCN(C(c2nn(CC)c(C)c2)=O)C1 64249,c1(OC(C(=O)NCC)(C)c2ccccc2)cc(C)c(NC(=O)NCCSC)cn1 64250,c1(OC)c(Br)cc(CN2C(C(=O)NC(c3ccc(I)cc3)C)CC3CC23)cc1Br 64251,C(C(C(C)C)NC(=O)C(C#N)=C1CCCC1)NC(C(C)OCCOC)=O 64252,CC(C)(C(=O)NCC1CCC(NC(=O)CN2CCCC2=O)C1)c1cc[nH]n1 64253,c1(N2CCCN(Cc3c(C)c(F)ccc3F)CC2C)ncnc2c(F)cccc12 64254,c1(C(N2CCCC(C(C)NC(c3cc(C)sn3)=O)C2)=O)n[nH]c2cc(Cl)ccc12 64255,Cc1cnn(CC(N2C(C(=O)NCC(=O)OC(C)(C)C)CC2C)=O)c1 64256,C1(NC(CCc2cc(C)[nH]n2)=O)CC(C(=O)NC(c2cnn(C)c2C)C)=CC1O 64257,C1(CNC(C2CCCCS2)=O)CN(C(c2ccc(Cl)cn2)=O)CC12CC2 64258,CC1(C)CCN(C(c2csnc2Cl)=O)C1CNC(c1cc(C2CCCC2)no1)=O 64259,c1(CC(C(=O)N(C2CC(NC(C3(C)CCCO3)=O)C2)C)O)cccc(C(F)(F)F)c1 64260,C1(NC(c2nc(C)oc2C)=O)CCN(C(=O)C(C)Cc2cnn(C)c2)CC1F 64261,CCC(CC(=O)NCC1CN(C(c2ccncc2)=O)C2COCC2O1)C(C)(C)C 64262,C(CO)(C(=O)N1CC=CC1C(N1C(CO)CC1CO)=O)OC 64263,c1(C(=O)Nc2ccc(O)c(F)c2)cn2c(n1)CN(Cc1cc(I)cnc1Cl)CC2 64264,Cn1cc(C#CCN=C(NCc2ccnn2C2CC2)NC2CCS(=O)(=O)C2)cn1 64265,C1(CC(=O)OC(C#C)(C)C2CC2)CN(C(=O)OC(C)(C)C)CC1C 64266,C12(NC(=O)CCC3CCCCO3)CCOC(CNC(c3cc(Br)no3)=O)(C1)C2 64267,c1(Cn2cc(C(C)NC(c3ccc(Cl)nc3O)=O)nn2)cc(F)c(F)cc1F 64268,C1(CC(=O)NC2CCN(C(=O)CC34CCCC3C4)C2)(CC=C)CCCC1 64269,C1(NC(CCC2(C)CC2)=O)CCCCC1CNC(c1cnnc(O)c1)=O 64270,C(=O)(CCC(C(=O)N1CC(C)N(C(=O)C=CSC)CC1C)N(C)C)OC 64271,N1(C(Cc2c[nH]cc2C(=O)NC2(CC)CCOCC2)=O)CC(OC)C2(CC2)C1 64272,O=C1NCC2(CCN(C(=O)C(=O)NCC(F)Cl)CC2)CCN1 64273,C1(NC(CC2C(C)OCC2)=O)CCN(C(c2cccc(O)c2)=O)CC1C(N)=O 64274,c1(C(N(C)CC2CCN(C(=O)Cc3cc(Cl)cs3)CC2)=O)ccc(O)c(O)c1Cl 64275,C1(C(=O)NCC2CCCCN(C(Cc3c(C)noc3)=O)C2)Cc2ccncc2C1 64276,C1(C(C)(C)C)CCC(C(O)C(=O)NCCNC(c2ccccc2C2CC2)=O)CC1 64277,Cc1[nH]c(C(=O)NCC2CN(C(=O)C(N)=O)CC2(C)C)c(C)c1C(=O)OC(C)C 64278,CC#CCCCC(=O)NC(COC)CC(=O)NC(c1nncn1C)CO 64279,C12(C(=O)NCC3(OC)CN(C(=O)C(F)C(C)C)C3)CC(C)(C1)OC21CCOCC1 64280,c12nc(OC)cc(n1)N2.C1(CNC(CCOCC)=O)CCCSCC1 64281,C(N=c1[nH]c(=NC(CCO)C(F)F)[nH]c2c(F)cccc12)C1(OC)CCCC1 64282,N1(C(CCNC(C)=O)=O)CCN(C(c2sc(NC(=O)C(C)C)cc2C)=O)C(C)C1C 64283,N1(C(C(CC)O)=O)CCN(C(CNC(c2cc(C(F)F)[nH]n2)=O)C(F)(F)F)CC1 64284,C1(CNC(c2ccc(CC)c(F)c2)=O)CC2(CCC2)CN1C(=O)C(C)C(C)(C)C 64285,c1(CNC(=O)NCC(=O)NC2CCNC(=O)C2)nc(=O)c2ccccc2s1 64286,C(C(C)(CNC(c1nonc1N)=O)OC)NC(C(C)OCC#C)=O 64287,C1(CNC(C2(CC(C)C)COC2)=O)COCC2(CCN(C(C3CC34CC4)=O)C2)O1 64288,C(=O)(C(F)CCC(C)(C)C)NC(C)CCCNC(c1cccnc1O)=O 64289,c1(C(=O)NC23CC(CNC(c4c(C)ncs4)=O)(C2)C3)cccn2cnnc12 64290,CCC(CC(C)C)C(=O)N1CC2C(CC(=O)NCC3CC3CC)C2C1 64291,C12(C(=O)NCC3CC(F)CN3C(=O)CC3CC=CCC3)CCN(CC1)C2 64292,N1(C(C2C(C(=O)OC)CCC2)=O)CC2CCN(C(=O)COC(C)C)CCC2C1 64293,N1(C2CC(C(=O)OC)C23CCC3)CC(NC(=O)OC(C)(C)C)CC(C)(C)C1 64294,C(=O)(C1=NOC2(CCC2)C1)Nc1c(C(=O)OCC)ncc(Cl)n1 64295,C1(C(N2CC(NC(CCNC(COC)=O)=O)CC2(C)C)=O)CN(CP(C)(C)=O)C1 64296,c1(NC(CNC(CC(CCC)C)=O)C)ncccc1[N+](=O)[O-] 64297,c1(CC)onc(C)c1C(N1CCC(OCCNC(=O)C(C)=CCO)C1)=O 64298,C(=O)(CC(F)(F)CC(=O)OC)NC(CNC(c1c(CC)n(CC)nn1)=O)C1CC1 64299,Cc1ccc(C)n1CC(=O)NCC(C)N(C)C(c1cc(C(F)F)ncn1)=O 64300,CN=c1[nH]nc(CC(=O)NCC2(NC(=O)C(C)Sc3ccc(F)cc3)CCC2)s1 64301,c1(C(N(C(Cl)C(F)(F)F)CCCC)=O)ccc([N+](=O)[O-])cc1OC(F)F 64302,c1(NCC(C)O)cc(S(=O)(=O)N2CCCC2CC(C)(C)C)ccc1C#N 64303,C1(NC(c2nc(COCC)sc2)=O)CCN(C(=O)CCSC)CC(C)(C)C1 64304,C(C)(c1cccnc1)=CC(N1CCC(C(C)(C)C)(CNC(CCCC#C)=O)C1)=O 64305,c1(CC)ccnc(C(=O)NC2C3CC2N(C(=O)COCc2nccn2C)C3)c1 64306,CN=c1nc(N2CCCC(OC3CC3)C2)[nH]c(=NCc2ccc(Cl)c(F)c2F)[nH]1 64307,c1(C(N2CC(NC(C3(C(=O)OCC)CCCCO3)=O)C2)=O)cnn2c1N(C)CC2 64308,c1(OC)ccc2c(c1)CC(C(=O)NCC(O)CCNC(=O)CC1CCOCC1)O2 64309,C1(NC(=O)CCN2CCC2)CN(C(=O)Cc2cscn2)Cc2ccnn2C1 64310,N1(C(c2cc(CC)nn2C)=O)CC2CCCC2C1C(N1CC(CO)CC(C)C1)=O 64311,C1(C(=O)NCC2CCC(NC(C3C(C)(C)C3)=O)C2)CCCC(O)C1 64312,c1(C(N2CCCC(CCNC(C(C)OCCOC)=O)C2)=O)cnc(O)cc1OC 64313,c1(C(N(C(C(=O)N(CC(COC)O)C)COC)C2CC2)=O)cc(O)ccc1C 64314,c1(CSC)cccnc1C(=O)NC1CNCC(O)C1 64315,C1(NC(Cc2nc(C)sc2)=O)CN(C(C2CCC=CCC2)=O)C2(CCOCC2)C1 64316,N1(C(C(C)NC(COC)=O)=O)CCOCC(C)(CNC(=O)Cc2ccc(C)s2)C1 64317,c1(NC(C2(F)CN(C(C(CC)=CCCC)=O)C2)=O)ccc(O)c(CO)c1 64318,N12CCOCC(C1)C(=O)N(c1cccnc1)CC(C)=CC2=O.c1(C2CC2)nc(C)n(C)n1 64319,N1(C(COCC=C)=O)CC(NC(=O)C=Cc2ccc[nH]2)CC12CCOC2 64320,C1(NC(CC2(C=C)CC2)=O)CC2CC(C1)N(C(=O)CC1CN3CCC1CC3)C2 64321,c1(C(CNC(c2cnc(C)[nH]2)=O)NC(=O)C=Cc2ncc[nH]2)ccc(F)cc1 64322,N1(C(c2c(C)con2)=O)CC2CCC(N(C(=O)Cc3cccc(F)c3)C)C2C1 64323,c1(C(=O)NCCN(C(=O)CCOC(C)CC(C)C)CCC)cc(C2CC2)n[nH]1 64324,c1(CC)ccc(C)cc1C(=O)NC1CCN(C(c2ccc(CSC)o2)=O)C(C)C1 64325,c1(N2C(C3(NC(CCC(=C)C)=O)CC3)CCC2)ncnc2c1COC2 64326,CC(=O)CCCC(=O)NCC1(O)CCN(C(=O)C(C)OC2CCCCCC2)CC1 64327,C1(O)(Cn2cc(C(C(C)(C)C)O)nn2)CCN(C(=O)COC(F)F)CC1 64328,N1(C(c2c(CC)n[nH]c2)=O)CCCC(CCNC(=O)CCCOC)CC1 64329,CC(C)C(C(=O)NCC(CNC(c1cscn1)=O)CO)NC(N)=O 64330,N1(C(C=CC)=O)CCCCCC(NC(=O)C=Cc2c(C)nn(CC(C)C)c2Cl)C1 64331,N1(C(C2CC(C)NC(=O)C2)=O)CCC2(CC1)CCN(C(=O)CC1OCCCO1)C2 64332,CC(CC(=O)N(CCCN(C)C(C1(Cc2ccccc2)CC1)=O)C)C(F)F 64333,N1(C(c2c(CCNC(C(C)OC(C)(C)C)=O)n[nH]c2)=O)CCC(C2CC2)C1 64334,C1(CN(C(=O)C(N)=O)C)CC(F)CN1C(c1cnc(N2CCOCC2)s1)=O 64335,C1(NC(=O)Cc2csc(-c3ccoc3)n2)CCCCC1CNC(c1cnsn1)=O 64336,N1(C(Cc2cn(C(C)C)nn2)=O)C2CCC1CC(N(C)C(C1CCCS1)=O)C2 64337,N1(C(=O)Cc2nc[nH]n2)CCC2CCN(C(c3csc(O)n3)=O)CC2C1 64338,N1(C(C(CC)NC(C)=O)=O)CC(O)CC1CC(=O)Nc1ccsc1 64339,C=CCC(C)(C)CC(=O)NCC(c1ccc(F)cc1)NC(=O)Cc1nccn1C 64340,c1(NC(C2(c3nn[nH]n3)CCCOC2)=O)cc(Cl)c2ccc(Br)cc2n1 64341,c1(OC)ncccc1CN1CC(F)CC1C(=O)NC(c1cccc(Br)c1)C 64342,C1(CNC(Cc2cc(C)[nH]n2)=O)CN(C(c2cc(C)on2)=O)C2CCN1C2 64343,c1(C(N2CCCC(F)C2)C(=O)NCCCSCC)ccc2nsnc2c1 64344,c1(C(=O)NC(c2ccnc(F)c2)C)cc2c(Br)cnn2cn1 64345,Cc1cccc(C=CC(N2CCC(O)CC2C(=O)N(C2(C3CC3)CC2)C)=O)c1 64346,c1(CC(=O)NCCNC(C=C(COC)C)=O)ccoc1C 64347,CS(=O)(=O)c1ccc(F)c(CNC(N2CC(CO)C(O)C2)=O)c1 64348,c1(CC)ccc(F)cc1C(=O)NCC1(C(F)F)CCN(C(c2ccnn2C)=O)C1 64349,C12(C(=O)NCCC(=O)N(C)C)CC1CCN2C(c1ccc(=N)[nH]c1)=O 64350,C1(CNC(C(C)CN(C)C)=O)CC2COCC2N1C(=O)C(F)(F)c1cnnn1C 64351,c1(C(=O)NCCN(C(c2nc(CCCCC)sc2)=O)CC2CC2)ncccc1O 64352,N1(C(c2c(C)c[nH]c2)=O)CCC12CN(Cc1cc(Cl)ccc1Cl)C2 64353,c1(C(C)C)nc(CNC(=O)C=CCNC(=O)CCC2CC2(F)F)no1 64354,c1(CCN=C(NCC2(F)CCCC2)NCC2CC2)ccc2c(c1)COC2 64355,C(C)(C(C)N(C(=O)C(c1cccs1)NC(C1(n2cccn2)CC1)=O)C)SC 64356,c1(C(=O)NC2C(NC(c3ccc(NC(C)C)nc3)=O)CC2)[nH]nc([N+](=O)[O-])c1Cl 64357,C1(C(N(C(C)CCO)C)=O)CC2CC1CN(C(=O)C(C)CN(C)C)C2 64358,Cc1ccc(OCCC(=O)NC(C)CCNC(c2c(C)cnn2C)=O)c(C)c1 64359,c1(-n2cc(OC(C(=O)NC(CCC=C)C(=O)O)C)nn2)ccc2nonc2c1 64360,c1(-c2cn(CCN(C)C(c3cccc(C(F)(F)F)c3F)=O)nn2)c(F)cccc1Cl 64361,c1(CNC(c2c(CC)cc[nH]2)=O)cccc(C(=O)NCC(Cl)Cl)n1 64362,c1(C(N(C2CC2)CC2CCCN(C(CCCOC)=O)C2)=O)cc(Cl)cnc1C 64363,c1(OC)ccc(NC(C2CC3CC3N2C(c2cnc(O)[nH]2)=O)=O)cc1F 64364,c1(C(=O)NC(C(=O)NC(C(C)O)CO)Cn2cncn2)ccccc1F 64365,Cc1ncnc(O)c1C(=O)NC1CCN(C(=O)C2=CCCCC2)C1(C)C 64366,C1(NC(C2N(C(c3cccc(NC)n3)=O)CCCCC2)=O)CCn2ncnc2C1 64367,C1(C(=O)NCCN(C(CCCN(CCCC)CCCC)=O)C)CC12CCOC2 64368,C12(NC(CN(C)CC)=O)CCC(CC1NC(c1ccns1)=O)C2 64369,C=CCC(CC)C(=O)NC(Cc1cc[nH]n1)C(=O)NC(C)CCOC 64370,c1(-c2cn(CC=C)nc2)cnc2c(C(=O)Nc3cc(OC)cc(O)c3)cccn12 64371,n1(C(C)C)cc(C(N2CC(CNC(=O)C(C)(C)C#N)C3(CC3)C2)=O)ccc1=O 64372,C(=O)(C(C)(C)CC(C)(C)C)N1CCC(CC(N2C(C)CCCC2)=O)C1 64373,N1(C(C2C(=O)NCC2)=O)CC(NC(=O)C(C2CC2)C2CC2)CC12CCCCCC2 64374,c1(C(=O)NC(C(C)NC(CCOCC#C)=O)CO)c(Cl)cccc1Br 64375,C(CCC(=O)NCC1(NC(c2csc(-c3cccnc3)n2)=O)CCC1)SC 64376,C=CC(C)(CC)C(=O)N1CC(OC)C(NC(=O)C(F)(F)c2cscn2)C1 64377,O(C1c2ccccc2CCC1F)C(c1ccc(OC)c(C#N)c1)=O 64378,c1(C(N(CC(C(=O)NCc2c(OC)nn(C)c2)C)C)=O)cn(C)c(=O)cn1 64379,C(CCC1CC1)(C(=O)N1CC(C(=O)OC)C1)NC(CC1CC(NC)C1)=O 64380,Cc1cc(O)c(F)cc1C(N1CCOC(c2cn(CC3(O)CCC3)nn2)C1)=O 64381,C1(C)(C(=O)NCC(CC(=O)N(CCNC(C(C)C)=O)C)C)CCC(=O)NC1 64382,c1(CN2CCC(NC(C3CCOCC3)C#C)CC2)csc2c1CCCC2 64383,c1(C(=O)NCCC(C)N(C(=O)CCC2CCCC(=O)N2)C)cccc(O)n1 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64613,C1(OCC)CCN(C(=O)CCNC(N)=O)C1CC 64614,C(=O)(CC(C(C)C)OC)NCC(CN(C(c1cc(CCC)c(C)s1)=O)C)C 64615,CC(C(=O)N1CCN(CC(C)(C)NC(=O)C(C)OCCC(C)C)CC1)C(F)(F)F 64616,c1(C(=O)NCCC2CCCN2C(=O)COCCF)cc2ccc(Cl)c(F)c2[nH]1 64617,c1(C(N2C3CN(C(C4CC(=O)NCC4)=O)C(CC3)C2)=O)c(Cl)ccc2c[nH]nc12 64618,C1(C)(NC(C2C(C)CCC2)=O)CCN(C(C2(c3ccccc3Br)CC2)=O)CC1 64619,C(C)(CO)(C(=O)N1CCC(OCCNC(=O)C(C)(C)SC)C1)OC 64620,C1(NC(=O)C(c2ccccc2)O)CC2CC1CN(C(C1(F)CCCC1)=O)C2 64621,C1(C)(CNC(CCNC(COC)=O)=O)CN(C(c2ccnc(C3CC3)n2)=O)CC1C 64622,n1(CC(=O)NCC2(O)CCN(C(C(C3CCCCC3)C)=O)C2)ccc([N+](=O)[O-])n1 64623,c1(C(CC)C(=O)N(C)CCN(C(=O)C(SC)SC)C)cccc(Cl)c1 64624,C1(NC(C(CSC)OC)=O)CCN(C(c2cc(-c3ccco3)on2)=O)C12CCC2 64625,N1(C(c2c(CNC(C3CC(=O)NCC3)=O)ocn2)=O)CC2COCC(C2)C1 64626,Cc1c(C(N2CC(c3ccc(C(C)C)cc3)(O)C2)=O)noc1C1CC1 64627,NS(=O)(=O)CCCCCCC(=O)NCC1CCN1C(=O)CCNc1ccncc1 64628,c1(C(N2C(C(=O)NC3CC(F)(F)C3)CSC2)=O)ccncc1Cl 64629,N1(C(Cc2ccc(CC)cc2)=O)CCN(C(=O)Cn2cc(C)cn2)C(C2CC2)C1 64630,c1(C(N(C2CC(NC(C3ON=C(CC)C3)=O)C2)C)=O)cc2c(Cl)cccc2s1 64631,Cc1scc(C(=O)N(CC(=O)NC(C(O)CO)C2CC2)C(C)C)c1C 64632,S(=O)(=O)(c1cccc(N2CCOCC(C)(C)C2)n1)NCc1cc(C)on1 64633,N1(C(CCCOCC)=O)CCN(Cc2cn(CCOC3CCOC3)nn2)CC1 64634,Cc1n[nH]c(C)c1C(=O)N(C)Cc1ccccc1CNC(C1C(C)(C)C1(C)C)=O 64635,C1(NC(CC(C)(C)NC(Cc2ccc(C)s2)=O)=O)C(O)C2CCOC12 64636,C12(C(=O)NC(CCOC)C)COC(C1)C(NC(=O)C=CC1CCCCC1)C2 64637,C1(CNC(C2=NOC(C)C2)=O)CCC2(CC1)CCN(C(c1ccc[nH]1)=O)CC2 64638,CCC(C)C(O)C(C)C(=O)NCC1CN(C(=O)CNC(N)=O)C2CCN1C2 64639,c1(C(=O)NCC2N(C(c3cn(C)nn3)=O)CCC2)c(O)cccc1O 64640,N1(C(C(=CC2CCCC2)C)=O)CC(O)CC1CNC(=O)CNC(c1ccco1)=O 64641,CC1CC(c2nc(-c3c[nH]c4ccccc34)nn2-c2ccccc2)=NO1 64642,N1(C(=O)C(F)CC2CCOC2)CCCC(F)(C(=O)NOCCC2CC2)C1 64643,c1(OC)ccc(NC(C2CCCN(C(=O)C(Cl)(Cl)Cl)CC2)=O)cc1I 64644,c1(C(=O)NCCC(C(C)C)NC(C=CSC)=O)cc2cccc(F)c2o1 64645,CC1CCC(CN2CC(N3CC(NC(=O)COC(F)(F)F)CC3=O)C2)NC1.OC 64646,N1(C(=O)CCC2CC2)CCCCC1C1CCCN(CC2(O)CCC2)C1 64647,c1(C(=O)NCC(C)NC(c2ccc(NC(C)=O)cc2)=O)sc2ccccc2c1C 64648,CCC(C)(CCC(C)C)C(=O)NCCNC(c1ccc2c(c1)CN(C)C2)=O 64649,c1(OCC(=O)NCC(C)N(C)C(c2ccc(N)c(N)c2)=O)ccc(F)c(F)c1 64650,N1(C(C(C)NC(=O)NC2CCCC2)=O)CCC2C(NC(C3CN(C)C(=O)N3)=O)C12 64651,c1(C(c2n(CC(=C)C)nnn2)NC(C(C)C)C2CC2)cnc2n1CCCC2 64652,CC1(C)CCCC(CNCC2CCCS2(=O)=O)C1 64653,CC(CCC(C)(C)C)C(=O)NC1CN(C(=O)CN2CSCC2=O)CC1O 64654,c1(NCc2c(C)nco2)ccc(C(F)(F)F)cc1S(=O)(=O)NC1C2CCCCCC12 64655,c1(C(N(CCOC(C)=O)C)=O)ccc(C(C)C)c([N+](=O)[O-])c1.N12CCC(CC1)C2 64656,N1(C(C(=Cc2ccccc2)C)=O)CCC2(CCCN(C(C3COC(=O)N3)=O)C2)C1 64657,c1(CC)nc(C)c(C(=O)NCCOCc2ccc(OC(C)=O)cc2)s1 64658,N1(C(C2C(F)(C(=O)OC)C2)=O)CCOC2(C1)CN(C(c1ccnnc1O)=O)C2 64659,CC1CC(F)(F)CN1C(=O)Nc1ccc(F)cc1-c1oncc1CO 64660,Cc1cnc2c(cnn2CC(=O)NC2CCCN(C(c3ccc(Br)o3)=O)CC2)c1 64661,c1cc(C)cc(F)c1.C(CNN(C)CC)(C(C)C)NC(C(c1ccccc1)O)=O 64662,c1(CNC(c2n(CC)nnn2)CCCC2CC2)ccccc1OCC 64663,c1(CCNC(N2CCC(CNC(CC)=O)C2)=O)ccc2c(c1)COC2 64664,C(c1cc(C)cc(C)c1)=CC(=O)NCC(CC=C)NC(=O)C(=Cc1ccco1)C 64665,C1(NC(c2oc(C)c(Br)c2)=O)C2CC3C1C3C2C(=O)N(C)C 64666,CCC(C)(CO)C(=O)N1CC(C(=O)NCCOC2CCCC2)C(F)C1 64667,C(CN=c1ccnc(N2CCC3(CCCCC3)C2)[nH]1)c1cc(O)cc(Cl)c1 64668,c1(C(=O)NCC2C(NC(c3ncc(OC)nc3)=O)COC2)cc(C)ccc1Cl 64669,CC1(C)CC(NC(C2C(O)CCN2C(=O)CC#N)=O)C12CCC2 64670,Cc1ccc(CCC(=O)NCC2CCC2NC(=O)CCC(=O)N(C)C)cn1 64671,c1(C(N2CCOC(C)(C3CC3)C2)C(=O)NC(C(=O)OC)C)ccc(C)c(I)c1 64672,C(=O)(C1=NOCC1)N(C(CCNC(C1CC(CC)C1)=O)C)C 64673,N1(C(C2CC=CCC2)=O)CC2=C(C1)CN(C(C1(O)CC(F)(F)C1)=O)C2 64674,Cc1cc(C2CCC2)ncc1C(N1CCC(NC(C2CCC(=O)C2)=O)C1C)=O 64675,N1(C(COCCCC)=O)CC(NC(=O)C(C)(C)CF)C(C(F)F)C1 64676,c1(SCC(N2CC(C)C(Nc3ncc(C(C)(C)C)s3)C2)=O)nc2ccccc2s1 64677,C#CC(C)(C)C(=O)OCC1CNCCC1c1ccc(OC)cc1 64678,c1(C(=O)NCC)cc2c(nc1O)CCCC2.C12CC(O)(C1)CN2C(C)C(=O)NC 64679,c1(CC)[nH]c(C(=O)NC(C)(CNC(C2CCOC2)=O)c2cccs2)nc1Cl 64680,O=C1CC(C(=O)NCCc2ccncc2F)N(C(C2CC2Cl)=O)C1 64681,CCCCCCCN(C(=O)C(C1CCC1)NC(C1CC1(C)C(F)F)=O)C 64682,C1(NC(C2CCC(C(C)C)CC2)=O)CN(C(C2CC2(C)Br)=O)Cc2nccn2C1 64683,Cc1ccccc1C=CC(N1CC(C(C)NC(c2cccc(F)n2)=O)C1)=O 64684,C(CN=C(NCC(c1ccccc1Cl)OC)N1CCC(C)C1)OC 64685,C1(C(=O)NC2CCN(C(CCC(C)C#N)=O)CC2)CCc2cn(C)nc2C1 64686,C(=O)(CCCCC(N)=O)Nc1c(F)ccc(NC(C2ON=C(C)C2)=O)c1 64687,N1(C(C(C)C)=O)CCC(C2CCN(C(=O)C(F)C3CCC3)CC2)C1 64688,c1(C(N2CCC(C(C)(C)C)CC2)C(=O)NC(C)C)cc(I)ccc1F 64689,Cc1[nH]cc(C(=O)NCC(n2cc(-c3ccc4c(c3)CCC4)nn2)C)c(=O)c1Cl 64690,c1(C(=O)NCC2(C(N3CCC(C=C)C3)=O)CC3(CC3)C2)cn2ccccc2n1 64691,C(CCCC(c1cn(CCCCCO)nn1)Nc1cncc(C(=O)OC)c1)NC 64692,C(=O)(CCCCCC(C)C)NCCCN(C(C=Cc1c(C)noc1C)=O)C1CC1 64693,C(=O)(C1c2ccccc2C2CC1C2)NC1CNCC(C)(C)O1 64694,CC1(C)CN(C(C2CCN(CCO)C(=O)C2)=O)CC1NC(=O)CCc1nc[nH]n1 64695,N1(C(=O)OC(C)(C)C)CC(CCNC2CCCN(CCO)C2)CC1(C)C 64696,c1(C(N2C(C)(C(N3CCN(C)CC3)=O)CC2)=O)cc(Cl)cc([N+](=O)[O-])c1 64697,Cc1cc(CN2CC3CC3(C(=O)Nc3cc(C(F)(F)F)c(Br)cn3)C2)ccc1Br 64698,c1(C(N(CCCCNC(CC2CCC(C)C2)=O)C)=O)cccc(F)c1Cl 64699,N1(C(=O)Cc2sc(-c3cccs3)nc2-c2ccccc2)CC2CCCC(C1)C2O 64700,CC1CC2CC(C(=O)N(C3CN(C(=O)CCn4cccn4)C3)C)(C2)O1 64701,c1(OC)cncc(C(=O)NCCC(C)NC(=O)C(O)CCc2ccccc2)c1 64702,c1(C(=O)NCC(COC(CC)C)=O)c(OC)cccc1F.N12CC3C(C3C1)C2 64703,Cc1cccc(C(=O)NCCCCCNC(=O)C(c2cnn(C)c2)O)c1O 64704,N1(C(C(CC=C)CC)=O)CCCCCC(NC(c2onc(C)c2C)=O)C1 64705,Cc1ccc(C)n1CC(N1CC(O)(C(C)NC(c2cnn(C3CC3C)c2)=O)C1)=O 64706,Cc1cc(=NC(CF)c2ccccc2Cl)[nH]c(C2(C(=O)OC(C)(C)C)CC2)n1 64707,C1(CNC(C2C(OC)CCC2)=O)(OC)CCN(C(=O)COCCSC)C1 64708,c1(C(=O)NC(C(=O)NCC2CCOCC2)C2CCCC2)ccc2cc[nH]c2c1 64709,N1(C(CN(C)S(N)(=O)=O)=O)C2CCC1CC(F)(CNC(=O)CC(=O)N1CCC1)C2 64710,Cc1cc(C)[nH]c(=NCc2cn3ccc(-c4cnc(OC(C)C)nc4)cc3n2)n1 64711,N1(C(Cc2c(Cl)cn(C)n2)=O)CC(NC(=O)Cc2cncs2)C(C2CC2)C1 64712,Cc1cc(=O)n(C)nc1C(N1CCCCC1CN(C(=O)CC1OCCCO1)C)=O 64713,C1(CNC(c2c(C)sc(O)n2)=O)CCN(C(=O)C(F)(F)CN(C)C)C(C)C1 64714,Cc1cc(Br)cc(C)c1CC(=O)NCC(n1cc(-c2c(O)cnn2C)nn1)C 64715,Cc1ccc(O)c(C(N2CC3CC2CN3C(=O)C(c2ccc(Cl)s2)C)=O)c1 64716,C1(CC=C)(C(=O)NC(Cc2ccsc2)CO)CCN(C(c2csnn2)=O)C1 64717,N1(C(=O)OC(C)(C)C)CCC(C(F)(F)F)CC1NC(=O)C(N1CCC12CCC2)=O 64718,C1(CNC(C23CC(C(=O)OC)(C2)C3)=O)(NC(C2COC(=O)N2)=O)CCOCC1 64719,N1(C(C(CCOC)OC)=O)CCN(C(c2sc(F)cc2C)=O)C2(CCC2)C1 64720,C(CCCCC(=O)NC1CC(CNC(=O)CC2OCCOC2(C)C)C1)NC(C)=O 64721,C1(C(=O)NCc2cc(OCC)ncc2)CC2COCC2N1c1ncncc1C#N 64722,C1(NC(c2occ(C(N3C(C(C)C)CCC3)=O)c2)=O)CC(CC(F)(F)F)CCO1 64723,CCCC(C)CC(=O)NCCC1CCN(C(c2cc(C)nc(OC)n2)=O)C1 64724,N1(C(c2cc(C(C)C)[nH]n2)=O)CC(NC(c2c(Br)cnn2C)=O)CC(C)C1 64725,Cc1cc(O)nc(C)c1C(=O)NCC(c1ccccc1)CNC(N)=O 64726,c1(CNc2c(CC(=O)NCc3ccc(F)cc3)cccc2)cnc(Cl)cc1F 64727,CC#CCC(C(=O)NCc1ccc(CC)cn1)NC(c1cncc(NC)c1)=O 64728,C1(NC(=O)CC2CC3(CC3)C2)CCN(C(=O)CS(=O)(=O)Cc2cccs2)CC1F 64729,C(CC(C(=O)NC1CC(n2cccn2)C1)NC(C1COC(C)(C)C1)=O)SC 64730,C1(CCNC(C2CC2C2CCCC2)=O)CCCN(C(=O)CCc2cn[nH]c2)CC1 64731,Cc1ccc(CCN=C(NCC(C)(C)C2CC2)NCC2CC2=CC=C(C)O)c(O)c1 64732,c1(C(=O)NC(C2(O)CN(C(c3c(SC)cn(C)n3)=O)C2)C)nc2sccn2c1C 64733,c1(C(=O)NC2COCCN(C(C(C(C)C)F)=O)C2)cccc2cnsc12 64734,S(=O)(=O)(c1ccc(Cl)cc1F)NC1CCCC(C(=O)Nc2ccc(Cl)nc2Br)C1 64735,Cc1ccc(SCC(N2CC(OCCNC(=O)C(C(C)C)N(C)C)C2)=O)c(C)c1 64736,Cn1ncc2c1CN(C(=O)C1=CCCN(C(C3CCOCC3)=O)C1)C2=O 64737,C12CC(C1)NC(=O)CC1CC(C1)OCC2=O.C1(C(C)O)CCCC1.C(C)(C)C 64738,C1(C(=O)NC(c2ccc(F)cc2)CC)CC(O)CCN1C(c1sc(C)cc1C)=O 64739,C1(C(N(C(CCC(C)C)C)C)=O)CC1C1CN(C(C2(O)CCCOC2)=O)C1 64740,CCC(C(=O)N(C1CCN(C(c2ccsn2)=O)C1)CCO)SC 64741,c1(C(N2C(C)CN(C(C3(C)CC3(F)F)=O)CC2)=O)ccc2nc(CO)[nH]c2c1 64742,c1(Cn2ccnc2)cc2ncccc2[nH]1.CC1(C)C(=O)N2CCC2CN2CC1C2 64743,C1(N(C(C(CC)C)=O)C(C)C)CCCNCC1 64744,CC1=C(C(=O)N(C2CCN(C(=O)CCC3CC(F)(F)C3)C2)C)CCO1 64745,N1(C(C=C(CC)CC)=O)CCC2CN(C(c3c(N)sc(C)c3C)=O)CCC2C1 64746,N1(C(C2CCCCC2n2cc(CCCCCO)nn2)=O)CCC2(CCNC2=O)C1 64747,c1(CC(N2CCC(N(C)C(c3ccnc(C(F)F)c3)=O)C2)=O)cc(F)ccc1F 64748,N1(C(C(=Cc2ccccc2)C)=O)CCC2(CC2NC(=O)CC23CCCC2C3)C1 64749,c1(C(=O)Nc2cc(Cl)cc(F)c2F)noc2c1CCc1sccc1-2 64750,c1(C(=O)NC2CCC(NC(CCCOCC=C)=O)CC2)nccc(F)c1Cl 64751,C=C(F)C1(CC(N2CC(C)CC2C(=O)NCC(O)C(N)=O)=O)CCC1 64752,Cc1ncsc1C(=O)NCC(=O)NC1CCC(CNC(=O)CC(=O)NCC2CC2)C1 64753,N1(CC)CCCC(Nc2cc(-c3cccc(C(F)(F)F)c3)nn2C)C1C 64754,C(=O)(C(C)(C)C(=O)N(C)C)NC1C(CNC(c2c(OCC)cncc2)=O)COC1 64755,c1(CC)sc(C(=O)NCC2CN(C(C3CC3C(F)(F)F)=O)C2)cc1Br 64756,c1(NC(C(N2CCCCC(NC(CSSC)=O)C2)=O)=O)ccc([N+](=O)[O-])c(SC)c1 64757,C1(C(=O)NCC2(C(C)(C)O)CN(C(c3cc(CC)on3)=O)C2)CCCC(F)C1 64758,CC(CC(=O)N1CC(F)(CF)C1)C(C)(C)NC(=O)C(c1ccccc1)F 64759,C1(CN(C(C=C(C)C(C)(C)C)=O)C)CC(F)CN1C(=O)COCC(F)F 64760,C1(C(=O)NCC(c2ccccc2)NC(C2C(=C)CC2)=O)CC1C1CC1 64761,c1(C(c2ccccc2OC(=O)COC)C(=O)OCC)ccc(C)cc1C(F)(F)F 64762,C1(CCNC(C=Cc2ccc(CC)o2)=O)CC(F)(F)CN1C(=O)CC1CC=CC1 64763,N1(C(CCCC(OC)OC)=O)CCCC12CCN(C(=O)C(CO)N(C)C)C2 64764,C(CC(=O)NC(C)(C)CCNC(=O)COc1ccc(Cl)c(F)c1)(C(F)(F)F)OC 64765,CCC(C)(C)C(=O)NCCN(C(=O)CCc1nc(O)n[nH]1)CC(C)O 64766,C(c1ccccc1Cl)=CC(=O)NC(CNC(C1CCOC1)=O)CC(F)(F)F 64767,C1(C(=O)NC(c2cn(C)nn2)C(=O)NCCOCC)(OC)CCC(C)C1 64768,N1(C(c2c(C(=O)OC)n(C)nc2)=O)CC(NC(C2CNC(=O)C2)=O)CC2(CC2)C1 64769,c1(OC)n[nH]cc1C(=O)NC(c1cn(C)nn1)C(=O)N(C1CCOCC1)C 64770,c1(C(=O)NCCNC(C(C)C)=O)csc(CNC(=O)C(=O)NC2CC2)c1 64771,c1(OC)cccc(CCC(=O)NCC=CCNC(c2cncn2C2CC2)=O)n1 64772,N1(C(c2cc(CNC(c3cn4ccccc4n3)=O)sc2)=O)CC2(CNC(=O)N2)C1 64773,N1(C(C2C3CC(NC(C4(C5(C)CC5)CC4)=O)C(C3)C2)=O)CC2CCC(C1)C(=O)N2 64774,C1(C)(CNC(Cc2ncc(C)o2)=O)CCCN1C(c1csc(Cl)n1)=O 64775,C1(C(N2CCC(C(=O)NC)C2)=O)CCN(C(C2CCCCC2)=O)C(C)C1 64776,N1(C(c2c(C)n(C)nc2)=O)CCN(C(=O)CCN2C(=O)CCC2=O)CC1C1CC1 64777,C(=O)(C(O)CC[S+](C)C)NCC1CC(NC(C(C)Cc2cccc(Cl)c2)=O)C1 64778,N1(C(C2(C=C)CC2)=O)CCc2c(CNC(=O)CCCC3CC3)cccc2C1 64779,CON(C(=O)C1CC(=O)NC(C(C)C)C1)C(C)c1ccccc1Cl 64780,C1(CNC(C(=O)NC(c2cscn2)C)=O)(CO)CC2CC2C1 64781,C(=O)(C(C)(F)C(C)(C)F)NC1CC(CCNC(C(C(=C)C)(C)C)=O)C1 64782,C1(NC(CCN(C)CCO)=O)CCCCCC1C(=O)NCC1CCSC1 64783,Cc1ccc(-c2ccc(CN(CC(O)CO)C)cc2)cc1F 64784,C1(CN(C(C2CC(O)(CC#C)C2)=O)C)CCCCN1C(C1CCOC1C)=O 64785,c1(C(N(CCCCNC(CC2C(OC)CC2)=O)C)=O)cnn(CCC#N)c1C 64786,c1(-n2c(C)nnn2)ccc(C(=O)NC2CN(C(C3CCN(C)CC3)=O)CC2O)cc1 64787,C1(N(C)C)CCC(C(=O)NCC(CO)NC(c2sccc2C#N)=O)CC1 64788,n1(C(=O)OC)ccc2cc(Cc3onc(C)c3Cl)ccc12.N12CC(O)CC1C2=O 64789,c1(CN(C)C)nccc(=O)n1C.C12CCCC1NC(=O)NC2 64790,CC1CC=C(C(=O)N2CCC(F)(F)C(CNC(C3CCCO3)=O)C2)CC1 64791,N1(CC(N2C(C(=O)OC)CCC(F)C2)=O)C(=O)C(=O)N(C(C)C)C1=O 64792,CC1(C)CC(C)(CO)CN1C(C1CC(=O)CN1C(C1CCCC(=O)C1)=O)=O 64793,Cc1cn(C)c(C(c2nnnn2C2CCCC2)NCCCCCCN(C)C)n1 64794,C1(c2nccn2C)CCN(C(C=CSC)=O)CC1 64795,N1(CCC(=O)N(CCNC(CC2CC(=C)C2)=O)C)C(=O)C2CCCCC2C1=O 64796,N1(C(CSCCC)=O)CC(NC(c2[nH]c(C)c(C(C)=O)c2C)=O)CC1(C)COC 64797,Cn1cc(Cl)c(C(=O)NCC2CC(NC(c3ocnc3-c3ccccc3)=O)C2)n1 64798,c1(C(CN(C(C(=O)NC(C)CC2(O)CCC2)=O)C2CC2)O)ccc(Cl)cc1 64799,Cc1nc(C(=O)NCC2CCCC2NC(C2C(Cl)(Cl)C23CC3)=O)sc1C 64800,C1(NC(Cc2nc(C)[nH]n2)=O)CCCCC1CNC(C1(C)CCN(C)C1)=O 64801,C1(C(=O)NCC(CC=C)(C)C)CCCN(C(C2CCCN2CCC)=O)CC1 64802,C(C)(c1cnn(C)c1)=CC(=O)NC(c1ccc(OCC#N)cc1)C(=O)OC 64803,c1(C(NNC(=O)NCCCSC(F)F)=O)c(Br)cc(Br)c(O)c1Br 64804,CC(C(C)C(=O)NCC(O)CN(C(=O)C=Cc1cccc(CO)c1)C)S(C)(=O)=O 64805,CC1CN(C(=O)Cn2ncnn2)CC1NC(c1conc1C(F)(F)F)=O 64806,c1(CC(=O)NCCC2N(C(c3c(OC)n[nH]c3)=O)CCC2)ccc(Cl)cc1F 64807,C1(C(=O)NCCCOC)CN(C(=O)CC2(O)CCOCC2)CC(C)O1 64808,C1(C(=O)NCC(=O)OCC=C)CN(C(=O)C=C(CC)CC)CCO1 64809,C(=O)(CC(C)CC(C)C)N1CCN(CC(C)NC(C=Cc2ccc(C)o2)=O)CC1 64810,Cc1c(C(=O)NCC(N2Cc3cccc(O)c3C2)=O)cc([N+](=O)[O-])cc1Br 64811,c12cc(ncn1)N1CCN(CC1)C(C)CN2C.c1(CSC)noc(C2CC2)n1 64812,c1(CC)nocc1CNC(=O)NC(C)Cc1ccccn1 64813,n1(CC)cnc2nc(=NCC3(S(C)=O)CC3)[nH]c(NCCn3nc(C)cc3C)c12 64814,N1(C(CCOCC#C)=O)CCCC12CCN(C(=O)C(c1c(C)noc1C)C)C2 64815,Cc1nc(CC(=O)N(C2CCCN(C(c3ccc(C)n3C)=O)C2)C)c(Cl)s1 64816,CC(=O)CC(C)(C)CC(=O)NCC1CCCN1C(=O)C(F)(F)CCc1ccsc1 64817,Cc1cn2c(n1)CCC(NC(=O)NC(c1ccnn1Cc1ccccc1)C)C2 64818,c1(C(=O)NC2CC(CNC(C(C#C)(C)C)=O)C23CCC3)cccc2sccc12 64819,c1(NC(=O)NCC2(C)CC(C)(C)C2)ccc2ccc(Br)cc2c1 64820,c1(OC)nccc(=NC2CN(C(=O)C(C)CSC(F)(F)F)CC2C)[nH]1 64821,C1(NC(C(C(C)C)F)=O)CCC2(CC1)CCN(C(=O)CCC1CCOCC1)CC2 64822,N1(C(CCN(CCC)C)=O)CC(NC(c2cc(C)oc2C)=O)C2CCCCC12 64823,CC1CCC(CC(N2CCC(C(C)(C)NC(=O)Cn3ccc(C4CC4)n3)C2)=O)C1 64824,c1(CC)conc1CNC(C1(NC(=O)COCCSCC)CC(O)C1)=O 64825,N1(C(c2c(C)n(C(C)C)nn2)=O)CCCC(NC(c2cc(Cl)cs2)=O)CC1 64826,S(=O)(=O)(c1ccc(F)cc1Cl)N1CCC2(OCC(NC(COC(C)C)=O)C2)CC1 64827,C1(NC(C2CC(NC(C=C(C)c3ccco3)=O)C2(C)C)=O)CC2CC1C(O)C2O 64828,O=CN1CCN(C(C2CC23CN(C(=O)CCc2ccc(Br)cc2F)C3)=O)CC1 64829,N1(C(C2C3(CCN(C(C4N(C)CC(F)C4)=O)C3)C2)=O)Cc2ccc(O)cc2C1 64830,CC(F)(F)C(C)(C)CS(=O)(=O)N1CCOCC1c1ccc2c(c1)OCO2 64831,c1(C(=O)NC2C(CNC(c3cnn(CC)n3)=O)CCC2)cccc(OC)c1OC 64832,c1(SC)cc(C(=O)NCCCN(C(=O)CCC2(C)CCC(=O)N2)CCO)oc1C 64833,c1(NC(C)=O)n[nH]c(NC(=O)C(N)CC2CCCO2)c1Br 64834,Cc1nc(C)n(CCC(N2CCC(CO)(CNC(c3c[nH]c(=N)s3)=O)C2)=O)n1 64835,N1(C(Cn2cnc(=N)[nH]2)=O)CCCC(CNC(=O)CCc2ccc(O)nc2)CC1 64836,CC1CN(C(c2ccc(OC3CCOCC3)nc2)=O)Cc2nncn21 64837,CC1OC(C)CC1CC(=O)N(C)CC1CCCN1C(c1occc1Br)=O 64838,c1(OC)cc(C)nc(CC2CCN(C(=O)NC3CCC(OC(F)F)C3)CC2)n1 64839,Cc1ccc(C(=O)NC(C)CNC(c2cncc(OC(F)F)c2)=O)c(C(C)C)n1 64840,C=CC(C)(O)CC(=O)NC1CCC(NC(=O)CS(=O)(=O)NC)C1 64841,N1(C(CC2CC(CC)C2)=O)C(C(=O)NCC2CCN2CCOC)C2CC(O)C1C2 64842,N1(C(C(C)NC(CC)=O)=O)CCC2(CC1)CC2(C)C(N1CCNC(=O)CC1C)=O 64843,C1(CNC(C(CCC)OCC)=O)CC2(CCN(C(=O)CC3CCCCO3)C2)CO1 64844,c1(C(N2CCN(C(Cc3cc(C)[nH]n3)=O)C3C2C3)=O)ccc2c(c1)C(=O)C(=O)N2 64845,N1(C(c2cc(CCC)[nH]n2)=O)C(C)CC2CN(C(c3cc(COC)[nH]n3)=O)CC12 64846,C1(C)(C(N(CCCCN(C(C(c2nc(C)sc2)=O)=O)C)C)=O)CCC(C)C1 64847,Cc1cnc(C(=O)NC(CNC(c2cnc(=N)[nH]c2)=O)CO)c(F)c1 64848,c1(N(CCC)C)nc2ccc(S(=O)(=O)N3CCC4(CCSC4)C3)cc2s1 64849,N1(C(CN(C(C)C)C)=O)CCC(CNC(=O)COc2ccc(Br)cc2)C1(C)C 64850,c1(CNC2CCC(C(=O)NC(C3CCCCO3)C)C2)cc(C#N)ccn1 64851,c1(C(=O)OC)ccc2c(n1)CCCN2C(c1ccc(-c2cnnn2C)cc1)=O 64852,c1(C(=O)NCC2COC(CNC(=O)C(F)n3ccnc3)C2)ccnc2[nH]ncc12 64853,N1(C(CC(c2c(N3CCC(SN)C3)cccc2)=O)=O)CCCOC(C(=O)OC)C1 64854,N1(C(C(C)S(N)(=O)=O)=O)CC2(CCC(CNC(c3ccncc3C3CC3)=O)O2)C1 64855,c1(N2CCC(c3nc(=N)[nH][nH]3)C2)c(I)cnc(Cl)c1F 64856,N1(C(c2ccc(C(C)=O)cn2)=O)CCC2(NC(=O)CC3CC3(C)C)CCCC12 64857,C(=O)(C(CO)C(C)(C)C)N1CCN(CC(=O)Nc2n(C(C)C)ncc2)C(=O)C1 64858,O=C(C#CC1CCOC1)NC1CC2CCC1CC2NC(=O)C(F)OC(F)(F)F 64859,c1(N2CCC(NC(C)C(C)(C)C)CC2)ccc2nncn2n1 64860,C(=O)(C#CC1CCCOC1)NC1CC(CNC(C2(SC)CC2)=O)OCC1 64861,c1(CC)cc(C(=O)NCCC(C)NC(=O)C(C)NC(c2cccs2)=O)ccc1F 64862,CC(CC(=O)N(C1(C(N2CCOC(C#N)C2)=O)CC1)C)C(F)F 64863,C(N=c1nc2scnc2c(NCCCF)[nH]1)C1C(C)(C)C1C(F)F 64864,c1(NCc2ccc(OC)c(Br)c2)nccc(=NC(CC)CC(C)CO)[nH]1 64865,C#CC1CN(C(=O)C(C)C(CC)CC)CCN1C(=O)CCCOC(C)=O 64866,c1(C(N2CC(O)(CNC(C(C)OCc3ccccc3)=O)C2)=O)nc(=O)n(C)[nH]1 64867,c1(C(=O)NC2(C)CCN(C(COCCOC)=O)C2)ccc2cc(C#N)ccc2c1 64868,CC(C(=O)N1CC(NC(c2ccc(C(C)(C)C)c(Cl)c2)=O)C2(CC2)C1)C(C)(F)F 64869,S(=O)(=O)(c1cccnc1C(=O)Nc1oc(C(=O)OC)cc1C)NCC 64870,N1(C(CC2CCC(=O)CC2)=O)CC2(CCC2)CC1CNC(=O)CCN1CCCC1 64871,CC(C)CCCC(=O)N1CCC(O)(CCNC(C2(O)CCSC2)=O)CC1 64872,c1(C(=O)NC2CCN(C(C3ON=C(C)C3)=O)CC2)cccc2c1CCC2=O 64873,C#CCCCC(C)C(=O)N(C1CN(C(c2ccc(F)o2)=O)C1)C 64874,c1(C(N(CCCNC(=O)CC(O)C2CC2)C(C)C)=O)ncccc1OC(F)F 64875,c1(OC)ccnc(Nc2nc(CC(=O)O)cs2)n1.c1(C2CN2)ccsc1 64876,CC1(C)CC(CNC(=O)CN2C(=O)CNC2=O)CN1C(C1CCC1C#N)=O 64877,N1(C(c2cc(OC)c(I)cc2)=O)CC2(CCN(C(=O)CCC(C)C)C2)C1 64878,c1(OC)cc(OC)c(C(=O)NCCCNC(=O)C(C)Sc2ccccn2)cc1Cl 64879,CC1CCCC1C(=O)NCC1(Cn2cc(-c3nccn3C)nn2)CC1 64880,c1(Cn2cc(C(CC)(C)O)nn2)ncccc1C(=O)N(C)CC1CCC(C)CC1 64881,C#CCC(CC(=O)N1CCC(C)(O)C1)NC(c1cn(C(C)C)cn1)=O 64882,C1(CCNC(CCN(CC)CC)=O)CCCN1C(=O)CSC1CC1 64883,C=CCCC(C(=O)NCC(O)CC(C)C)NC(c1cccnc1O)=O 64884,C1(F)(C(=O)NCC(C)(C)CNC(C2(c3ccccc3F)CCC2)=O)CCCOC1 64885,c1(C(=O)NC(CC=C)CNC(=O)Cc2cncn2C)cccnc1C(F)F 64886,N=c1[nH]c2cc(C(=O)NCC3C4CN(C(=O)CCc5cc[nH]n5)CC34)ccc2o1 64887,c1(-n2c(OCOC34CCCNCC3C4)ccc2)c(F)cccc1Cl.O=CO 64888,c1(C(=O)NCC2CCCC(NC(CCC#CC)=O)C2)csc2c1CCCCCC2 64889,C(C1=CCCCC1)(c1nnnn1CCCCCC)NCC(CC#C)(C)C 64890,c1(OCC(=O)NC2CC(C)(NC(c3ccn(C(C)(C)C)n3)=O)C2)cccc(F)c1 64891,CC1(NC(c2ccc(C3CC3)s2)=O)CCN(C(=O)CC2(C)CCOC2)C1 64892,C1(CC(=O)Nc2cccc(N3CCC3)c2)CC(F)CN1C(c1cn[nH]c1)=O 64893,Cc1n[nH]c(C)c1C(=O)NCC(c1ccc(F)cc1)NC(C1CCOC1)=O 64894,c1(N(C2CN(C(=O)CCc3ccc(F)cc3)C2)C)ccc(Br)cc1[N+](=O)[O-] 64895,C(CCN=c1[nH]c(=N)[nH]c(=NC2CCOC2C)[nH]1)(c1ccccc1)OCC 64896,c1(C(=O)NC2C(OC)CN(C(C3(C4CC4)CC3)=O)CC2)cc(Cl)c(F)c(Cl)c1 64897,c1(CC(=O)NC2C=CS(=O)(=O)C2)ccc2c(c1)CCCS2(=O)=O 64898,C(C(=O)N1CCCCC1CNC(=O)CC1CCC(C2CC2)O1)(C(C)C)SC 64899,c1(CC(N2C(CC)CN(C(=O)C(=O)NC3CCC3)CC2)=O)nc2c([nH]1)CCCC2 64900,C1(CC)C(CC(=O)NCCC(Cc2ccccc2)NC(=O)CNS(N)(=O)=O)C1(F)F 64901,C1(C2CCCN(C(=O)C(C)C#N)C2)(NC(c2ccn(C(C)C)c(=O)c2)=O)CC1 64902,C(CN1C(=O)Cc2ccccc21)NC(c1cn(C)nn1)c1nnnn1C(C)(C)C 64903,C1(NC(C2CC(SC)C2)=O)CN(C(c2cnn(-c3ccc(F)cc3)c2)=O)CC1F 64904,Cc1oc(C)c(C(=O)N(C)CC2CCN(C(=O)Cc3nnc(O)s3)C2)c1C 64905,c1(N2CCC(N(C(c3scc(C)c3C)=O)C)C2)ncnc2c1cnn2C 64906,C1(CNC(c2c(CC)nc(C)[nH]2)=O)CC2(C1)CN(C(=O)Cn1nc(C)cc1C)C2 64907,C=CCN=C(NCCNc1cn2c(n1)SCC2)N1CN(C)C(=O)C1C 64908,N1(C(COCCCC)=O)CCC(C2OCCC2NC(=O)CN2CC=CC2)CC1 64909,CCC(C(O)C(C)C)NC(=O)NC(C)CCc1ccc(Br)cc1 64910,C1(CN(C)C(=O)NCc2nnc3ccc(Cl)cn23)Cc2ccccc2N1C 64911,c1(SCC(=O)N(CCCN(C(C)C(=O)NC2CC2)C)C)ccc(Br)cc1 64912,C#CCC(CC(=O)NC1CCCC(O)CC1)NC(=O)C(O)c1ccsc1 64913,C=CCCCC(=O)N1CC2C(NC(=O)C(c3ccccc3C)C)C2C1 64914,N1(C(C(n2ccc(C(F)(F)F)n2)C)=O)CCCCC1CNC(c1c[nH]nc1F)=O 64915,C1(OC)CCC12CC(C(N1CCC(C(C)NC(=O)C3=COCCC3)CC1)=O)C2 64916,CN1CC(NC(C2CN(C(=O)NCC(=O)CC3CCC(C4CC4)O3)C2)=O)CC1=O 64917,c1(SC)nn(C)cc1CNC(=O)CC1CCC(=O)N1 64918,CCC(C)C(C(=O)NCC1=CCN(C(c2ccc(NC)cc2Cl)=O)CC1)OC 64919,C1(NC(C2(NC(c3c(OC)nccc3)=O)CCOCC2)=O)CN(C)CC1(F)F 64920,c1(COC)cccc(CNC(=O)CC2CCN2C(c2ocnc2C)=O)c1 64921,c1(SCC)ccc(OCC(N2CCCC(CN(C(=O)CSC)C)C2)=O)c(OC)c1 64922,N1(C(C(C)OC)=O)CCOC(C23CC(CNC(=O)CCOC4COC4)(C2)C3)C1 64923,c1(CCC(=O)OC(C(=O)Nc2c(C)ncc(C)n2)(C)C)cc(C)ccc1[N+](=O)[O-] 64924,c1(C(=O)NCCCN(C(=O)Cc2c(C)nn(C)c2C)CC)sccc1S(N)(=O)=O 64925,N1(C(CCc2c(OCC)cccc2)=O)CCCC(C)(CNC(C2(O)COC2)=O)C1 64926,n1(CC(=O)NCC(COC)NC(=O)Cc2cn(C)nc2C)cccc(C)c1=O 64927,C=CCC(CC)C(=O)NCC1CCCN1C(=O)Cc1cccc(NCC2CC2)c1 64928,C(=O)(CCC(C)NC(C1(C#N)CC=CC1)=O)NCC(CSC)OC 64929,C1(c2ccc(F)cc2)(C(=O)NCCN(C(C=CC(CC)C)=O)CC)CCOCC1 64930,CCC1c2cc(Cl)cc(Cl)c2CCN1Cc1cnc(-c2ccccc2)o1 64931,C(CNC(=O)CCc1nc[nH]n1)(C(=O)N(C)C(C1(C)CC1)C)OC 64932,C(C(C(=O)N(C(C)CC(C)C)C)NC(=O)Cn1cc(C)cn1)OCC 64933,c1(N2CCN(C)C(CN(C)C)C2)nc(N2CCCC(C3CC3)C2)nc2c1CCC2 64934,C1(CC)(CO)CCN(C(C2(C)CCCN2C(c2nccnc2N)=O)=O)CC1 64935,CC1COc2c(C(=O)NCC(O)CNC(c3ccccc3Br)=O)cnn2C1 64936,CC(C)C(O)CC(=O)N1CCN(C)C(C(=O)NCC2OCCC2(C)C)C1 64937,c1(CNC(CN(C(C)=O)C)=O)cnn(C)c1C(=O)NCCC1CCCC(C)C1 64938,N1(C(c2c(C)nc(O)cc2)=O)CCCCCCC1C(=O)NC1C2CCC(F)(F)C12 64939,C1(NC(c2cc(C(C)C)no2)=O)CCCCCN(C(=O)C(=Cc2c[nH]cn2)F)C1 64940,c1(C(N2C(CC)C(C(=O)NCc3ncnn3C)CC2)=O)ccc(C#N)cc1 64941,c1(CN2CCC(C(=O)Nc3cc(C)c(I)cn3)CC2)cccc2cccc(C)c12 64942,C1(F)(CNC(c2c(Cl)cc(C)s2)=O)CCCN(C(=O)C(O)C2CCC2)C1 64943,S(=O)(=O)(c1c(F)cccc1F)NC1C(C(=O)Nc2cncc([N+](=O)[O-])c2)C1 64944,CS(=O)(=O)c1cccnc1C(=O)NCC1(CNC(C2CC23CC(O)C3)=O)CC1 64945,c1(NC(=O)OC)ccc(N(C)C(=S)NCCCCF)cn1 64946,c1(NC(CC2C=CC(NC(c3c(CCC)nco3)=O)C2)=O)cnc(OC)cc1C 64947,C=CCC(CC(=O)Nc1cnc(C2CC2)nc1)NC(C1CC(=O)N(C)C1)=O 64948,c1(C(=O)NC(C(CO)NC(C(CCCOC)C)=O)C)nnc(O)c2ccccc12 64949,C(=O)(CC(C)P(C)(C)=O)N1CCCC(CCNC(c2cc(C)cc(N)c2)=O)C1 64950,Cn1c(C(=O)NC2CC(CNC(=O)CC3CCCC(=O)C3)C2)cnc1O 64951,C1(COC)CC(O)CN1C(=O)C(C1CCCO1)NC(c1nccnc1N)=O 64952,n1(CC)ncc(C(N2CCCCC2CNC(=O)Cc2csc(NC=O)n2)=O)c1Cl 64953,C1(CNC(CC(C=C)CC)=O)CC2(CCN(C(=O)C(C)C(C)CC)CC2)CO1 64954,COn1cnc(C)c1C(=O)NCC1CCC1NC(c1cc(F)ccc1C1CC1)=O 64955,c1(C(=O)NC2CCC(C)(CNC(CCOCCC)=O)C2)cc(S(N)(=O)=O)sc1C 64956,C#CCCCCC(=O)N1CCC(NC(=O)CCc2cccc(OC)n2)C(F)C1 64957,N1(C(c2c(CC)nco2)=O)CC(NC(C2CCCC2C(C)C)=O)C(C)C1 64958,c1(CN2CC3C(C(N4CCC(=C)CC4)=O)(C3)C2)c(C)cccc1C 64959,c1(CNC(N2CCCC(OCC3(CO)CCC3)C2)=O)cc(Cl)ncc1O 64960,c1(C(N(C)CC2N(C(Cc3cc(C)sc3)=O)CCC2)=O)cc(Cl)c2n[nH]cc2c1 64961,CCC(C)CC(=O)NC(C1CC(NC(c2sc(C)nc2C)=O)C1)C 64962,C(=O)(CC1CCc2ccccc21)NCCCN(C(C1CC(C(C)C)C1)=O)CC 64963,n1(CC(=O)NC2C(CC)CN(C(=O)C=C3CCC3)C2)nc(C)c(F)c1C 64964,N1(C(Cc2c(C)cnn2C)=O)CCC2CC2(C(=O)NCC2(O)CC=CC2)CC1 64965,Cc1[nH][nH]c(=N)c1C(N1CCC(CN(C)C(c2cnc(C(C)(C)C)[nH]2)=O)C1)=O 64966,N1(C(C2(C#C)CN(C(C3CCC(F)(F)C3)=O)C2)=O)CCN(C)CC1C 64967,C1(C(=O)N(C)CC2CCN(C(=O)C(C)C(C)O)CC2)(CC)CCC(O)CC1 64968,C1(CN(C)C)CCCCN1C(=O)CC=CCNC(=O)CC(O)C1CCCC1 64969,c1(C(N2C(CNC(c3ccc(SC)s3)=O)CC2)=O)occ2c1CCOC2 64970,CCC(C(=O)NC(CC1CCCC1)C(=O)N(CCCCCC1CC1)C)N(CC)CC 64971,c1(OC)cc(NCC=CCNC(=O)CCc2nncn2C)c(Cl)cc1[N+](=O)[O-] 64972,C1CC(=O)NOCC(=O)N1C.C(CC(=O)NCCCO)OCC 64973,Cc1cc(C(=O)NCc2occc2C(=O)NC(C(C)(C)O)C2CC2)c(C)cn1 64974,n1(CC)nc(C(=O)NC2CN(C(=O)CSC3CC3)CC2C)cc1C1CC1 64975,c1(C(N(CC(=O)N(CC)CC)C)=O)ccc(CNC(=O)C(C)N(C)C)cc1 64976,C(=O)(C#CC(C)(C)CNC(C1(C)CCCC1O)=O)NC(C(=O)N(C)CC)C 64977,C(=O)(C(C)C(F)(F)C(F)F)NCCC1CCCN(C(c2c(N)ccc(C)c2)=O)C1 64978,C1(C(=O)NCC2CC(NC(C3CC=CCC3)=O)C2)CCC([N+](=O)[O-])CC1 64979,c1(NC(C2CCC(C)(N(C)C)C2(C)C)=O)cccc2c1COC(=O)N2 64980,c1(C(N2C(CC(C)C)CCCC2)C(=O)NC2COC2)cccn2ccnc12 64981,N1(C(C(CC)CN(C)C)=O)CC2(C)CC1(C(=O)NOCc1cncs1)C2 64982,N1(C(C(CCC)C)=O)CCN(C(=O)CSCC(C)C)CC1C 64983,N1(C(C(COC)OC)=O)CCN(C2CN(C(C3COCCN3C)=O)C2)CC1 64984,C1(C(C)(C)O)(CNC(=O)C=CC2CCC2)CN(C(=O)CC2C=CCC2)C1 64985,N1(C(c2cc(CC)on2)=O)CCN(C(=O)C=Cc2ccc(SC)cc2)C(CF)C1 64986,c1(C(=O)NCCOC)ccc(CC2CCN(C(C3(F)CC=CC3)=O)C2)cc1 64987,c1(C(=O)NCC(N2C(C(N(CC(OC)OC)CC)=O)CCC2)=O)ncccc1F 64988,N1(C(CCCN(CCC)CCC)=O)CCC2(CCCN2C(=O)C(C)SCC)C1 64989,Cc1cc(Cc2nc(C3(c4ccc(F)cc4)CCC3)no2)c(C)cc1Br 64990,Cn1cnc2ccc(C(N3CCN(C(c4ccon4)=O)C(C4CC4)C3)=O)cc12 64991,CC1(NC(C2C3CC4C(C3NC(c3cnc(C(C)C)o3)=O)C24)=O)CCCCCC1 64992,C1(C)(C(=O)NC2(CSC)CCC2)CC(OCC)CN1C(=O)CCC(C)C 64993,Cc1cc(C(=O)NC(CCN(C)C)C(=O)NCC2=NOC(C)C2)c(C)nn1 64994,C1(C(C)NC(=O)CC2(O)CCCOC2)CCN(c2nnc(C(F)F)s2)CC1 64995,C1(CC(=O)NCCOCCN(C(COCCCCCC)=O)C)COC(C)(C)C1 64996,c1(C(=O)NCCC2CCC(NC(=O)Cc3cccs3)C2)cc(F)c2[nH]nnc2c1 64997,c1(C(=O)NC2C(NC(C(c3ccccc3)OCC)=O)CCC2)ccc(C)cc1 64998,C1(C(N(C(C)C)CCNC(C2CCC2C)=O)=O)CCCN(c2ccnc(Cl)n2)C1 64999,C(C(F)(F)C(=O)NCCN(C(c1cc(-c2cccnc2)on1)=O)C1CC1)OC 65000,C(CN=c1[nH]c2ccc(F)cc2s1)C1CC(NC(C(C)O)=O)C1 65001,C1(NC(C2C3CN(C(C(C)=C4CCCC4)=O)CC32)=O)CCCOC12CCC2 65002,c1(C(N2C(C)CCC(CNC(=O)Cc3cccs3)C2)=O)cncc2c1CCC2 65003,N1(C(C(C)=CC2CC2)=O)CCCC(CO)(NC(c2cncc(Cl)c2)=O)C1 65004,C#CC1CN(C(C23CC(CN(C(c4cn(C)nc4C)=O)C2)C3)=O)CCO1 65005,c1(C(=O)NC2CCN(C(C(CC)n3cncn3)=O)C23CC3)cccc2c1COC2 65006,C1(NC(C2C(c3ccc(C)c(Br)c3)C2)=O)CC2(CCC(NC(C)C)CC2)C1 65007,C(CCC(C)(C)C(=O)N1CC(O)C(O)CO1)NC(c1c(NC)cnnc1)=O 65008,Cn1[nH]c([N+](=O)[O-])nc1=NCCN1CC2CC2C1 65009,N1(C(c2cnc3n2CCOC3)C(=O)NC(C)C)CCC2(COC(C)C2)C1 65010,N1(C2CN(C3(C(=O)N(C)C)CC3)C2)CC2CC2(SC)C1 65011,c1(C(N(C(=O)CN2CCC3(CCO3)C2)CC)=O)ccc(-c2cccs2)cc1F 65012,c1(OC)cc(C(N2CC(O)(C3(CNC(=O)C(F)OC)CC3)C2)=O)c2c(c1)CCO2 65013,C1(C(=O)NCC(CCC)OC)CC=CCN1C(=O)CCc1nncs1 65014,N1(C(C(C)OCC)=O)CC2CC1CN(C(c1cn(C)nc1Cc1ccco1)=O)C2 65015,CCC(C(=O)NCC1CCN(C(C2CCN(CC)C2)=O)C1)n1cncn1 65016,c1(C(N(CC(=O)NC)CC)=O)ccc(C2COCCN2C(c2ccsc2Cl)=O)n1C 65017,C1(C(N2CC(NC(C3(CC)COC3)=O)C2)=O)CCOC(C)C1 65018,CN1CCOC(C(=O)N(C2CN(C(c3cc(C4CC4)n(C)n3)=O)CC2O)C)C1 65019,N1(C(CC(=C)Br)=O)CCN(C(=O)Cc2cccc(OC)c2Cl)CC(O)C1 65020,C1(COC)CN(C(=O)NC2CCN(CC(C)(C)O)CC2)CC1O 65021,c1(CC)occc1C(=O)NC(CNC(c1cnc(C)s1)=O)CCOC 65022,C1(CNC(C2C(OCC)CC2)=O)CCC2CN(C(c3ccc(CC)s3)=O)CC12 65023,N1(C(C)C)CCC(C(=O)NC(C)CC2CCN(C(=O)CC=C(Cl)Cl)CC2)CC1 65024,C(=O)(CC(O)Cc1ccccc1)N1CC(CC(=O)NCC(C2CCCC2)OC)C1 65025,n1(CC(N2CCNC(C)C2C)=O)nc2n(c1=O)CCCC2 65026,c1(C(=O)NCCN(C(=O)C(C(C)CC)OC)CCC)cc2cc(Cl)ccc2n1C 65027,c1(N2C(CCNC(C3C(C)C3c3ccccc3)=O)CCC2)ncc(I)cn1 65028,c1(CC)cccc(C(N2CC(F)CC2CN(C)C(c2ccc(F)s2)=O)=O)c1O 65029,c1(C(=O)NC2CCN(C(C3(OC)CCOC3)=O)C2)cc2cccc(Cl)c2nc1C 65030,c1(OC(C)C(N2CCCCC2CNC(=O)C(F)(F)CC2CC2)=O)cccc(F)c1 65031,C1(CNC(C(C)(C)c2ccccn2)=O)CN(C(C2CCCS2)=O)CCC1(F)F 65032,c1(NC(C2C(C)(C)CN2)=O)cc(Cl)cn2ccnc12 65033,c1(C(=O)OCC)cc(C)sc1NCc1cn(-c2ccccc2OC)cn1 65034,C1(CNC(c2c(C)cn(C)c2)=O)CN(C(c2occ(C)c2C)=O)CC(C)(C)C1 65035,C(CCCCCC(=O)N1CC2CC=CC1C2)NC(c1nccc(Cl)c1F)=O 65036,C1(C(N(CCCN(C(=O)CCn2cnnn2)C)C)=O)CCCNC1=O 65037,C1(NC(C(C)OC)=O)C2CN(C(=O)CCC(=O)N(C)C)CC12 65038,c1(C(=O)NC2CN(C(C(CC(C)C)OC)=O)CC(C)C2)scc2c1OCCO2 65039,c1(C(N2CC(C)N(C(=O)C=CC3CCOC3)CC2)=O)cc(Cl)c(F)c(Cl)c1 65040,C12(NC(C(C)=CC)=O)CN(C(=O)C(C3CCCCC3)O)C(COC)(C1)C2 65041,C1(NC(CN(CCOC)C(c2conc2C)=O)=O)CCCC1C#N 65042,N1(C(c2[nH]cc(C#N)c2)=O)CC2CCC1C(Nc1ncnc(Cl)c1Br)C2 65043,C(C(CC)(CC)CC)(c1n(CCCOC)nnn1)NCC1CCCC12CCC2 65044,c1(C(=O)NC(C(=O)NCCc2cnc(C)[nH]2)Cc2ccoc2)cnc(Cl)n1C 65045,Cc1nnc(C(=O)N(C(C)CCNC(C2CC2(C)C(F)(F)F)=O)C)s1 65046,C1(C(N2CC(C)(NC(C3C(Cl)(Cl)C34CC4)=O)C2)=O)CCCCC(=O)N1 65047,Cc1ccc(C(N2CCN(C(=O)C=CCCC(C)C)CC2C(C)C)=O)c(=O)n1C 65048,N1(C(c2ncc(F)cn2)=O)CC2CCC1CN2C(c1ccc(Cl)cc1)=O 65049,N1(C(CCC)=O)CC2(NC(c3ccc(F)cc3CC)=O)CCC1C2 65050,Cc1ccc2c(=NCC(C)CN(C)C)[nH]c(N(C)CC3CC4(CC4)C3)nc2c1 65051,c1(OC)cc(NC(C2CC2C(N2CCC(F)(CO)C2)=O)=O)nc(C)n1 65052,C=CC1(C(=O)NCc2c(C)coc2C)CCN(C(=O)CCN(CC)CC)C1 65053,c1(C(N2CC(F)CC(NC(C(CC)C(C)C)=O)C2)=O)cccc2c(C)c(C)[nH]c12 65054,c1(C(N(CCC(C)NC(C2CC(CC)C2)=O)C)=O)cn2cc(Cl)cnc2n1 65055,N1(C(C(C2CCCC2)OC)=O)CC(F)(F)CC1CNC(c1cnn2ccsc12)=O 65056,c1(-c2cn(CC3N(CC(=O)Nc4ccc(Cl)nn4)CCC3)nn2)sc(O)nc1O 65057,C(=O)(C1CCc2nccn21)NC1CCC(NC(CCc2cn(C)nc2)=O)C1 65058,C1(NC(c2cc(C)nn2C(C)(C)C)=O)CC2CN(C(c3cnc(Cl)n3C)=O)CC12 65059,c1(OC)c(C)cc(C(=O)NCCCCNC(=O)CC(C)C)cc1Cl 65060,c1(C(=O)OC)cccc(C(C(=O)NCCC#N)N(C)Cc2ncccc2Br)n1 65061,N1(C(C(C)(C)C)=O)CC(NC(=O)CCOC(=O)NC(=O)C(C)(C)C)C(F)C1 65062,c1(CCNC(c2c(CCC(=O)OC)cccc2)=O)c(Cl)cc(Br)cc1Cl 65063,C1(CCOC)CCCCN1C(C1CCN(C(c2cc(C)no2)=O)C1)=O 65064,c1(C(=O)N(c2nc(C(=O)C(=O)CO)cs2)c2ccccc2)cccc2c(Br)cccc12 65065,N1(CC(=O)NC2(CO)CN(C(CC3CCC(C)C3)=O)C2)CCCNS1(=O)=O 65066,C(CC(C)(C)C(=O)NC1CC1NC(=O)Cc1cccc(OC)c1Cl)OC 65067,CN(CP(C)(C)=O)C(C1COCCC1NC(C1(C)CC1)=O)=O 65068,C(=O)(C1Cc2c(Cl)cccc21)N(CCCCNC(CCC(=O)NC)=O)C 65069,c1(C(=O)NCCN(C(CC(C(C)C)c2ccon2)=O)C)ccc(N)cc1[N+](=O)[O-] 65070,CC1CCCCC1OCC(=O)NCC1CC(NC(C2(CC(F)F)CCC2)=O)C1 65071,Cc1cc([N+](=O)[O-])cnc1N1CC(CNC(C2(Cl)CC2)=O)OC2(CCC2)C1 65072,N1(C(=O)NCC(c2ccccc2Cl)C)CCCC(NCCOn2cnnn2)C1 65073,CC1(C)C(CNC(c2cc(C3(O)COC3)on2)=O)CCN1C(=O)C=C(Cl)Cl 65074,c1(NC(C2CC2c2nn[nH]n2)=O)cc(Cl)nn1-c1ccc(F)cc1 65075,C(CCCCCCCO)=CC(N1C(CNC(C2CCC2(C)C)=O)CC(C)(C)C1)=O 65076,N1(C(Cc2c(C)non2)=O)CCCC(CNC(c2cc(C(N)=O)no2)=O)C1 65077,C(CC(C)C(=O)NC(Cc1ccoc1)C(=O)NCCCc1ccsc1)=CCC 65078,N1(C(CCCC=C)=O)CCC(NC(=O)C(O)CCCCC)CC(C)(C)C1 65079,CC1(C)C(NC(c2ccn3nnnc3c2)=O)C(C)(C)C1NC(=O)C(F)=CCCF 65080,N(C(=NCc1nccs1)N1CCC(F)(C#N)C1)CC1(CSC)CC1 65081,N1(Cc2scc(C(=O)OC)c2)CC(C)CC1C(N1CC2CCC1C2)=O 65082,C#CCC(CC(=O)OC)NC(=O)C(C1CCN(C(=O)C(O)CN(C)C)CC1)(C)C 65083,c1(C(=O)NCc2[nH]nc(C3CCN(C(C)=O)CC3)n2)ccc(CN(C)C)c(Cl)c1 65084,CCC(CO)(C(=O)NC1CC(CNC(=O)Cn2cccc2)C1)OC 65085,C(=O)(C(C)=NOCC#N)NC(CC(=O)N(C)Cc1ccn(CC)n1)C1CC1 65086,C1(CCNC(C=NOC)=O)CCN(C(=O)C(=Cc2cn(C)cn2)F)C(C)C1 65087,Cc1nnc(O)c(C(=O)NCC(CC(F)(F)F)NC(=O)CC(C)(F)F)c1C 65088,C1(C(=O)NC2C(NC(CC3(C=C)CC3)=O)COC2)CCCCN1CCC 65089,c1(C(N2CC3C(N(C(CC=C)=O)C)C3C2)=O)cc(C(F)(F)F)cc(N)c1 65090,C(=O)(C1=CCN(C(c2ccc(F)c(F)c2)=O)C1)NC1CCN(CC)C1 65091,c1(C(N2CC(C)(NC(C(c3ccc(C)o3)C)=O)C2)=O)ccn(C2CC2)c1C 65092,Cc1ccnc(C(C)(C)C(=O)NCC(C)(O)CNC(C2CCCC2(C)C)=O)c1 65093,C1(CC(C)NC(=O)Cc2nncn2C)CCCC(C)(C)CC1 65094,c1(CC)ccc(C(N2CCC3(NC(c4cnn(C)c4C)=O)CC3C2)=O)c(O)c1 65095,C1(C)(c2cn(C3C(C)(C)C3(C)C)nn2)CCN(C(c2occc2C2CC2)=O)CC1 65096,C1(C(=O)NC2C(NC(C)=O)CCCC2)CC12CCCCCC2 65097,c1(OC)cc(C(=O)NC2(CNC(=O)CCC(C)C#N)CCCC2)c(OC)cc1Cl 65098,O=C(C1=CCCSC1)NC1C2CN(C(=O)CC3CCCO3)CC12 65099,N1(C(c2c(C)ncnc2)=O)CCC2(CO)CN(C(=O)C=CC3CCC3)CC2C1 65100,C1(N(C(COCC(=O)NC)=O)C)CC2CC1N(C(c1csc(C(C)(C)C)n1)=O)C2 65101,C1(CN(C(=O)C(C2CCN(C(=O)Cc3ccc[nH]3)C2)F)C)CCCC1(C)C 65102,Cc1cc(F)cnc1CNC(C1CC1c1ccccc1Cl)=O 65103,C1(CNC(c2ccc(OC)s2)=O)(CO)CCN(C(c2c[nH]c(C#N)c2)=O)CC1 65104,c1(C(=O)NC(C(=O)N(C)CCC2CCOCC2)Cc2cnc[nH]2)sccc1C#N 65105,N1(C(C(c2ccccc2)OCC)=O)CCN(C(=O)CS(=O)(=O)NC)CC1C(C)C 65106,CC(CC(C)(C)C)C(=O)N1CCC(N=[N+]=[N-])(C(=O)NCCCOC(=N)O)C1 65107,C1(NC(C(C)NS(CC)(=O)=O)=O)CC2CCC1N(C(c1c(C)nsc1N)=O)C2 65108,Cn1nc(C(=O)NCCN(C(=O)CSC(F)F)C2CC2)cc1OC(F)F 65109,N1(C(c2c(OC)scc2)=O)CCN(C(=O)C(F)CC(C)C)CC(C)(C)C1 65110,c1(C(=O)NC2C3C(C)N(C(C4CCCCN4C)=O)C2C3)ccc2nc[nH]c2c1 65111,C1(NC(CNC(COCC)=O)=O)CC2(C1)CC2(F)F.C12CCN1CC2 65112,c1(CC)cc(C(=O)NCC2CC2NC(=O)Cc2ccccc2CC)cc(OC)n1 65113,C12(NC(Cc3cnc(C)s3)=O)CCCC1N(C(=O)CCOC1COC1)CCC2 65114,N1(C(=O)CCCC(F)(F)F)CC2C3CCC(C2C1)N(CC1CCCO1)C3 65115,c1(CCC(=O)NC2C=CC(NC(CNC(CCCCC)=O)=O)C2)nnc(O)nc1O 65116,c1(OCCC)ccc(Cl)cc1C(=O)NC1CN(C(=O)C(C)(O)CC)CC1O 65117,C1(C(=O)Nc2cccnc2O)CC12CCN(C(c1cc(Cl)c(Cl)s1)=O)CC2 65118,C(C)(c1ccco1)=CC(=O)NC(C1C(CC(=O)NCC2C(=C)C2)CC1)=O 65119,c1(C(N2CCN(C(CC=CC)=O)C(CCC)C2)=O)nnc2ccccc2n1 65120,N1(C(C2C(C=C)OCC2)=O)CC2(CC2)CC1C(=O)NCC1CC2CCC2C1 65121,N1(C(CN(C)Cc2cncn2C)=O)CC2(CCCC(CNC3CCS3(=O)=O)O2)C1 65122,C(=O)(C(C)(CO)NC(=O)C=CC1CCCN1C)NCCC(COC)O 65123,C(=O)(CCC(=O)NCc1nc(C)c(C(=O)N(CCC(O)CO)C)o1)NCCC 65124,C1(C(=O)NCCC2(C)CCCO2)CCC(CNC(c2ccc[nH]2)=O)CC1 65125,C1(NC(=O)Cc2cnns2)CCCCC12CCN(C(=O)C1=CSCS1)C2 65126,c1(OC)nc(C(N2CCC(OCC(=O)NC3CCOCC3)CC2)=O)ncc1F 65127,n1(CCNC(N2CCN(CCC)CC2)=O)nc(C)c([N+](=O)[O-])c1C 65128,N1(C(C2(CC#C)CCOC2)=O)CC(N(C(=O)CSC2CC2)C)C(O)C1 65129,c1(CC(=O)NC(CC)CN(C)C(C2C(CC3CC3)C2(F)F)=O)ccccc1F 65130,Cc1nc(O)ccc1C(N1CCC(N(C(=O)CCCN(C)C)CCO)C1)=O 65131,N(C(=NCCn1cnnn1)NC1CCOc2ccc(F)cc21)C(CC)CC 65132,S(=O)(=O)(c1ccc(COC)s1)NC(CC)C(c1cc(C)ccc1C)(F)F 65133,Cc1ncc(C(=O)NC2CCC(C(=O)NCC(c3ccccn3)O)C2)c(=N)[nH]1 65134,C1(O)(C(C)NC(CSC)=O)CN(C(C2CCC(c3ccccc3)O2)=O)C1 65135,C1(C(=O)NC(C(=O)NC(C)C)C)(CO)CCN(C(c2c[nH]c(=S)cn2)=O)C1 65136,C1(CNC(C(CO)OC)=O)CCCCN1C(C1(C)CC1C)=O 65137,C1(OC)CN(C(c2cccn2C)=O)CC1NC(=O)CCCNS(C)(=O)=O 65138,C1(C(=O)NCCCCNC(c2[nH]cc(C)c(=O)c2)=O)CCCC1S(C)(=O)=O 65139,C1(C(=O)NCCCOCCN(C(=O)CC2C=CCCC2)C)C2CCCCC12 65140,N1(C(CC2(C(=O)OC)CC2)=O)CC(CNC(=O)CC2CCCS2(=O)=O)OC(C)(C)C1 65141,N1(C(CC(CC=C)NC(c2coc(CCC)n2)=O)=O)CC=CC12CCOCC2 65142,C1(C#N)(C(N2CCC(NC(c3cnc(SC)s3)=O)C(F)C2)=O)CCN(C)CC1 65143,N1(C(c2c(CC)n(CC)nc2)=O)CCCC(C)(CNC(=O)COCC(F)F)C1 65144,C1(C(=O)NC2(C)CCCO2)COC2(CNC(CN(CC(C)(C)C)C)=O)CC1C2 65145,C1(CC)CN(C(C2(c3cccc(Cl)n3)CC2)=O)CCC1NC(=O)CC1CCSC1 65146,c1(C(=O)NCCC(C)NC(=O)CC2CCCOC2)csc2c1CCCC2 65147,n1(CC(=O)NCC(C)C(=O)NC2CCC3CCC23)cc(C#N)cn1 65148,C1(C(=O)OC)SCCCN1C(N1CCC(Cc2nccn2C)CC1)=O 65149,c1(CNc2n(CCOc3ccc(Cl)cc3)ncc2)cccc2c1B(O)OC2 65150,c1(CCCNC(C(C)=CC)=O)ncc(-c2ccccc2)[nH]1 65151,c1(C(N2C(CNC(C3COCC(C)(C)O3)=O)CC2)=O)ccc(C#N)c(F)c1 65152,CC1(C)CN(C(C2CC3(CC(NC(c4cccnc4S)=O)C3)C2)=O)CCN1 65153,N=c1ccc(C(=O)NC(CC2CCOCC2)C(=O)NCC(O)CF)n[nH]1 65154,C1(c2nnc(C(C(=O)OC(C)(C)C)NO)o2)(OC(=O)OC)CC(F)(F)C1.C(C)(C)C.N 65155,C(=O)(C1Cc2ccc(Cl)cc21)NC12CC(NC(CN(C)C(C3CCOC3)=O)=O)(C1)C2 65156,c1(CC)cc(Br)ccc1C(N1CCCC(F)(C(N2CCC(CO)C2)=O)C1)=O 65157,c1(C(N=S(C)(=O)C2CCCC2)=O)c(CN)ccc2ccccc12 65158,C=CCC(CC=C)C(=O)NC1(C)CCN(C(=O)CCCNC(c2ccsc2)=O)C1 65159,CCCCC(C)CCC(=O)N1CC(CNC(c2cccc3c2CCN3)=O)C1 65160,C1(C(=O)OC)COC2(C1)CN(S(=O)(=O)CC1CCN(C3CC3)C1)C2 65161,C1(C(N(CC2=CCCOC2)C)=O)(NC(=O)Cn2cc(CO)nn2)CCC(C)(C)C1 65162,C1(NC(CN2CC(=O)NCC2)=O)C2CC(NC(=O)CN3CCCCCC3)CC12 65163,C(=O)(C1SCCc2sccc21)N(CCC)CCNC(=O)CCc1ccsc1 65164,N1(C2CN(C(C(C)n3cccn3)=O)C2)CCN(C(=O)CCCc2cncs2)CC1 65165,n1(CCC)ccc(C(N2CCC(CCNC(C3(c4n[nH]cc4C)CC3)=O)C2)=O)n1 65166,c1(CC)nc(C)ncc1C(=O)NCC=CCNC(C1CCOC(=O)N1)=O 65167,c1(NC(c2ccnc(F)c2)c2n(CCC3(C)CC3)nnn2)cncc(Cl)c1 65168,Cc1ccc2snc(C(=O)NCC3(NC(C4C(F)(F)C45CCC5)=O)CC3)c2c1 65169,C12(CNC(CCC#C)=O)CCCC1N(C(c1ccc(NS(C)(=O)=O)nc1)=O)CC2 65170,N(C=CC(=O)C(F)(F)F)CC1CCCC(CC)C1 65171,C(=O)(CCCCC(OC)OC)OC.C1C(CC(C)C)C(=O)O1 65172,Cc1cc(NC(=O)C(=O)NC(C2CCC2)C2CC2)cc2n[nH]cc12.C1C(=O)N1 65173,CC(C(C)(C)NC(=O)Cn1nccc1Cl)NC(C1CN(S(=O)(=O)C2CC2)C1)=O 65174,C(=O)(CC(C(F)(F)F)OC)NC(CCC)CCCNC(c1ccnnc1O)=O 65175,CC(C)CCC(C(=O)O)NC(=O)COCCc1cn(C(C)(C)C(=O)O)nn1 65176,c1(C(N(CC(C)NC(=O)C(C)c2cc[nH]n2)C)=O)c(Cl)ccc(O)c1N 65177,S(=O)(=O)(c1cccc(Cl)c1F)N1CCC(F)(C(=O)Nc2c(N(C)C)nccc2)C1 65178,c1(NC(CSC(C)=O)=O)cccc(F)c1CC(=O)Nc1cccc(C(C)O)c1 65179,C(=O)(C1=C(C)N(C)c2nnnn2C1)N1CCN(C(CCCCSC)=O)CC1 65180,n1(CC(=O)NC(C)C(=O)NCCC2(NC(=O)CO)CCC2)ncc2ccccc12 65181,c1(C(=O)NC(CC)C)cccc(-c2nc(COCCOC)n(-c3nccn3C)n2)c1 65182,N1(C(c2cc(OC)n[nH]2)=O)CCCCC2(C1)CN(C(c1ccc(C)cc1O)=O)C2 65183,c1(C(C)(C)NC(N(CCNC(=O)OC(C)(C)C)CCO)=O)cc(Cl)ccc1O 65184,C1(NC(C=COCC)=O)CC(O)CN(C(=O)Cc2ccnc(C(F)(F)F)c2)C1 65185,n1(CC(N2C3CC(C(=O)Nc4cccc(C)c4O)C2CC3)=O)cnc2ccccc12 65186,N1(C(CNC(C(CC)C)=O)=O)CCOCCC1C(=O)NCc1cnc(F)cc1C 65187,C12(NC(C(C)Oc3ccccc3)=O)CCCN(C(C3CCS(=O)(=O)N3)=O)CC1C2 65188,c1(C(=O)NC2CCN(C(c3c(OC)nsc3OC)=O)C2)ccc2nnc(O)n2c1 65189,N1(C(CC=CC(C)(C)C)=O)CCC2CN(C(=O)CCC3CCOCC3)CC2C1 65190,c1(C(=O)NCC(CC)NC(=O)C2=CC(C)(CC)C2)ccc(OC)c2ccncc12 65191,CC(CN(C)C)CC(=O)NCC1(NC(=O)CC(C)c2cccnc2)CCCC1 65192,C=CCC(C(=O)NCC1C=CCN1C(c1csc(CS(C)(=O)=O)n1)=O)C(C)C 65193,C(=O)(C(C(=O)NC1(CF)CN(C(C2CCCN2C2CC2)=O)C1)C(C)(C)C)OCC 65194,C(=O)(C(=O)C(C)CC)N1CCC(C(N2CC(C)(CC=C)C2)=O)(OC)C1 65195,CC1CC(CNC(C2(C)CNC(=O)C2)=O)CN(C(C2(C(F)F)CCCCC2)=O)C1 65196,N1(CCO)CCc2cncnc21.n1(C2CN(C=O)C2)nccc1C(F)(F)F 65197,CC1(C)CCCN(C(=O)C(C2CCOCC2)=O)C1C(N1CC2(C=CCO2)C1)=O 65198,C1(O)(CCNC(C2CC(=O)C2)=O)CCN(C(=O)CCc2cc[nH]n2)C1 65199,C1(C)(CN(CCC(=O)Nc2ccnn2C)CC)CCS(=O)(=O)CC1 65200,C(CCC(=O)NCCNS(C)(=O)=O)NC(C=CCCC)=O 65201,C12(C(=O)NCCC(C)NC(C34CC(CO)(C3)C4)=O)CC3CC1C2C3O 65202,C1(O)(CC(=O)N(C2COCC2N2CCCC2)C(=O)CCC2CC2)CCCCCC1 65203,c1(OCC)cnc(C(c2nnnn2C2(C)CC2)NC(c2cn(C)cn2)C)nc1 65204,C(CC(C(C)(C)C)NC(C1CCC1OC)=O)N(C(CC(COC)C)=O)C 65205,C1(CN(C(C2CCN(C(C)=O)C2)=O)C)C(=O)NCCN1C1CCCC1 65206,C1(NC(c2n[nH]c3c2CCCC3)=O)CN(C(C2CC2F)=O)C2CCCC12 65207,N1(C(c2noc(CC)c2C)=O)CCC2(CC1)CN(C(c1c[nH]c(C)c1)=O)C2 65208,C=CCC(CNC(=O)CC1COC(=O)C1)NC(=O)CC1CC(SC)C1 65209,c1(NC(C2N(C(c3c(Br)cnc(C)n3)=O)CCOC2)=O)cccc2ccoc12 65210,c1(CC)cc(C(N2CCC(C(C)C(=O)NCCc3ccns3)C2)=O)cc(O)n1 65211,C=C1CC2(C1)CC(C(=O)NCC1CC(F)(CNC(=O)CC3CCCCC3O)C1)C2 65212,O=C(CN=c1cc[nH]cc1)NCCC1CCCN1C(=O)CCCc1ccncc1 65213,N1(C(C(C(C)C)O)=O)CC2CCCC(C1)N2C(C1(C)CC2CCC(C1)S2)=O 65214,c1(OC)cc(C)ccc1C(N1CCC(=CCNC(=O)C(F)OC(F)(F)F)CC1)=O 65215,C1(C(=O)NCCCCOCC)CCC(C)(C)N(C(=O)C2=C(C)OCC2)C1 65216,N1(C(C(C)SC)=O)CCCC2(CCCN2C(c2cnn3ccncc23)=O)C1 65217,CC(C)CC(C)C(=O)N(C1CCN(C(=O)Cc2nnc(-c3cccs3)n2C)C1)C 65218,c1(C(N(C(C)CNC(C2(F)CCOC2)=O)CC)=O)c(C)cccc1Cl 65219,C1(NC(c2c(C)cnn2C)=O)CCOC2(CCN(C(c3ccoc3Cl)=O)CC2)C1 65220,C1(C2CCN(C(=O)CC(=O)OC(C)(C)C)CC2)(NC(C2CC(OC)C2)=O)CC1 65221,S(=O)(=O)(c1ccc(N(C)Cc2ccno2)c(C#N)c1)NC(COC)CC(C)(C)C 65222,C1(C)(COC)CN(C(c2cc(CNC(c3cnc(Cl)s3)=O)[nH]n2)=O)C1 65223,C#CC(C)(C)C(=O)N1CC(NC(c2cccc(OC(F)F)n2)=O)C(C)C1 65224,c1(C(=O)NC2C(C)CN(C(=O)CCc3nnc(O)nc3O)C2)ccc2ccnn2c1 65225,CCCC(C)(C)CC(=O)NCC1(OC)CN(C(c2nc[nH]c2C(F)(F)F)=O)C1 65226,C=CCCC(C)(C)C(=O)N1CC(CCNC(C2CCOC2)=O)C2(CC2)C1 65227,c1(OC)ccnc(C(N2CC(NC(=O)C(C)(C)n3cnc(C)c3)CC2C)=O)c1N 65228,c1(C(=O)NCCc2cscn2)cccnc1CNC(C1(O)CCOCC1)=O 65229,c1(C(=O)NC(C)CNC(=O)CSC2CCOC2=O)cncc2c(O)nccc12 65230,C1(C(=O)NCC(CNC(C2(C=C)CCCC2)=O)(C)O)CCC2(CC1)OCCO2 65231,Cc1cccc(Cl)c1OCC(=O)NCC1(O)CN(C(=O)C(F)=CC2CC2)C1 65232,N1(C(c2c(CCC)[nH]cc2)=O)CCCOC(CNC(C2(C3CCCO3)CC2)=O)C1 65233,C1(C)(C(=O)Nc2c(OC)c[nH]n2)CCN(CC(=O)OC2CC3CC3C2)C1 65234,c1(OC)cccc(C(=O)NC2CC(O)(CNC(=O)CCc3cnco3)C2)c1OC 65235,n1(CC=C)nnnc1C(c1cccn1-c1cccnc1)NCC(=O)OC(C)C 65236,c1(C(=O)NCC2CCC(NC(c3n(C)c(S)nn3)=O)C2)cc2ccoc2cc1F 65237,CCCC(CC1CCCC1)C(=O)N1CCC(C(c2cc(O)nc(C)n2)=O)CC1 65238,c1(CNC(=NCCOC)NCc2nnc3n2CCC3)nc2ncccn2n1 65239,c1(CN(C)C)ccc(C(=O)N(CCCNC(=O)CC2CC3CCC2O3)C)cc1 65240,C1(C#N)(C(=O)NC(CC)CN(C(=O)CNC(=O)C(F)(F)F)CC)CCOC1 65241,c1(C(C(=O)NC(C)CCCNC(=O)CCc2cncn2C)C)cccc(C#N)c1 65242,c1(-c2cn(CCOC)nc2)ccc(C(CC(=O)O)NCc2cnn(C)c2)cc1 65243,c1(C(=O)NC2CC2C(=O)Nc2cnn(C3CC3)c2)cccc(O)c1F 65244,c1(C(=O)NC(C(=O)NC(COCCOC)C)CC2CC2)cc(C)cc(F)c1 65245,CC1CCOCCN1C(C1(NC(c2csnn2)=O)CSC1)=O 65246,C1(C(N2CCCC(CCNC(=O)CC3CCCCCO3)C2)=O)CC2CCC1CC2 65247,c1(OC)cncc(C=CC(=O)NCC23CCC(CC2)N3C(C2CCSCC2)=O)c1 65248,C(=O)(C(F)(F)CCn1cccn1)NC1CCC(C(C)NC(c2n[nH]c(=N)s2)=O)C1 65249,C12(CNC(c3ccnnc3O)=O)CCCC(CN1C(C1Cc3nncn3C1)=O)C2 65250,c1(C(N2C3C(NC(CSCC)=O)(CCC3)CCC2)=O)cc(O)c2ccccc2c1 65251,C(=O)(C(CC(=O)OC(C)(C)C)C(C)=O)N1CC(CNC(=O)NC2CC(=C)C2)C1 65252,Cc1c(C(=O)NC2CN(C(C3CC3F)=O)CCC2O)oc(=O)c2ccccc12 65253,c1(OCC)cccc(NC(C2CN(C(c3cccn3C)=O)CCO2)=O)c1 65254,C1(CC(=O)N(CCCCCC)CCNC(=O)CCC)CC(OC(C)=O)C1(C)C 65255,c1(CC(=O)N(C(C)CC(=O)NCCOCCO)C)ccnc(O)c1 65256,C1(NC(C2(COC)CN(C(c3cn(CC)nc3C)=O)C2)=O)CCCCC1OC 65257,c1(N2CCC(c3cccc(C)c3)C2)nc2ccccc2nc1NCCC(C)C(F)F 65258,C(=O)(C1=CCC(C)(C)CC1)NCCC(C(=O)NC1CCOCC1C)OC 65259,C12(C(N(C(C)CNC(C3COC(C)(C)C3)=O)C)=O)CCC(C(F)(F)F)(CC1)CC2 65260,C=CC(C)(CC)C(=O)NCc1cc(C)c(C(=O)N(CC(O)CO)C(C)C)o1 65261,CCC(CNC(=O)CC1CCCC1O)(CC)C(=O)N1CC(N2CC(O)C2)C1 65262,CCC(CC(=O)NC1(CCC)CCCN(C(=O)CC(F)(F)F)C1)CC(F)(F)F 65263,N1(C(c2c(CC)occ2)=O)CC2CC2(CNC(=O)CCCN2CCCC2)C1 65264,c1(C(N2C(CNc3cc(COC)ncn3)CCC2)=O)ccc(Br)c2ncccc12 65265,N(C(=NCCC(C)=O)NCCn1ncnc1CC)CC1CCCC1CCC(C)C 65266,C(=O)(C1=C(C#N)CCC1)N1CC(NC(CC(C=C)c2ccccc2)=O)C(O)C1 65267,C(CCC(C)C(=O)NC1C2CC3C(C2)C13C(N1CC(O)(C(F)(F)F)C1)=O)OC 65268,C1(C(=O)OC)CCCC(NC2CCN(c3ccn(C)n3)C2=O)CC1 65269,c1(C(=O)NC2C(NC(c3oc(C)c(Br)c3)=O)CC2)cc(O)ccc1Br 65270,CCCCCCCCCC(O)C(=O)N(CC(C)CNC(c1nccnc1C)=O)C 65271,C12(C(=O)NCc3nc(C)c(C(=O)NCC4CC(F)C4)o3)CCCC1C2(F)F 65272,C1(NC(c2cn(CCC)nc2)=O)CCN(C(=O)CCCCC(N)=O)CCC1(F)F 65273,CC(C)CC(C)CNC(=O)C(O)CNC(=O)CSC(F)(F)F 65274,N1(C(CCCC#C)=O)CC(CCNC(c2cnc(OCC)c(Cl)c2)=O)OC(C)C1 65275,N1(C(C(C(CC)(C)C)=O)=O)CCC2(C1)CN(C(=O)CCC(C)(F)F)CC(C)O2 65276,c1(C(CC(=O)NC(CC)CN(C(=O)Cn2cc(C)cn2)C)C)cccc(C)c1 65277,C1(NC(Cc2c(C)con2)=O)CC(C)N(C(=O)C(C)CSc2ccccc2)C1 65278,CS(=O)c1ccccc1C(N1CC2(C1)CN(C(c1cnc(F)c(F)c1)=O)C2)=O 65279,C1(C(=O)NCCC2CCCN(c3ccnc(C)n3)C2)CCCC(C)(C)C1 65280,Cn1cnc(CCNC(c2occc2CNC(=O)C(F)n2ccnc2)=O)c1 65281,c1(C(=O)NC(C)CN(C)C(C2CCCN2c2cnccn2)=O)ccc(Cl)cc1O 65282,CCCS(=O)(=O)C(C)C(=O)NC1CCCC1NC(c1cnc2n1CCCC2)=O 65283,C1(C(=O)NCC2C(CNC(=O)Cc3sccc3Cl)C2)CC=CC(O)C1 65284,C1(C(=O)Nc2cccc(CS(CCOC)=O)c2)CCC2(CCCC2)C1 65285,C(C1=CCN(C(=O)C(C)S(C)(=O)=O)CC1)NC(C(c1scc(C)n1)(F)F)=O 65286,N1(C(c2n(C)ncc2)=O)CC(F)CC1CNC(C1(F)CCCC1)=O 65287,C1(N(C(=O)CN(C(=O)CCC2CC2C)C2CC2)C)CCOCC1NC1CCC1 65288,C1(CNC(C(C)c2ccsc2)=O)C2CC1N(C(c1ccccn1)=O)C2 65289,C1(CC)C(C)CCN1C(=O)CN(C(c1ccnn1COC)=O)CCF 65290,C1(c2onc(COCC)n2)N(C(=O)Oc2ccc(Cl)cc2Cl)CCCC1(C)C 65291,c1(NCCN2C(C)CCC2)cc(NCCNS(=O)(=O)C2CC2)ncn1 65292,C1(CNC(c2ccnc(F)c2Cl)=O)CN(Cc2ncsc2Br)CCC1(F)F 65293,CCCCC(C)CCC(=O)NC(C)(CNC(=O)C=Cc1cccc(O)c1)C(C)C 65294,C#CCC(C)(CC)C(=O)NCC(C(=O)N(C)Cc1nc(C)ns1)C(C)C 65295,N1(C(c2cn(CC)nc2)=O)CCCC1(C)CNC(=O)COCCc1ccccn1 65296,CCC(F)(F)C(=O)NC(c1nc(C(=O)NC(C)C(F)(F)F)co1)C 65297,C(C)(C(=O)N1CCC1CNC(=O)Cc1cnc[nH]1)NC(C)=O.C1C(=O)N1 65298,C1(C(=O)OC(C)(C)C)CCCC2(CN(c3ccc([N+](=O)[O-])c(Br)c3)C2)O1 65299,c1(C(=O)NC2CN(C(C3CCC3(F)F)=O)CC2CC2CC2)ccc(F)cc1F 65300,C1(NC(C2C(C=C)OCC2)=O)CCN(C(=O)CCC2CC(C)C2)CC1O 65301,C1(NC(=O)CCC(F)F)CN(C(c2cnc(Cl)c(C(F)(F)F)c2)=O)CCC1CO 65302,CC(=O)C(C)CC(C)C(=O)NCC(O)CC(N1CC2(COC(C)C2)C1)=O 65303,c1(C(=O)NCC2CCN(C(C(C(C)C)OCC)=O)C2)cccc2nc[nH]c12 65304,C(Cn1cc(CCSCC)nn1)(CC(=O)NNc1ccc(F)cn1)OC 65305,c1(NC(c2cnn(C)c2Br)c2n(C(C)C)nnn2)cc(Br)cc(C#N)c1 65306,N1(C(c2cc(CNC(CCC(C)C)=O)on2)=O)CCC(O)C12CCC2 65307,c1(CC(C(C)C)NC(=O)NCC2CC(F)CN2)ccccc1C(F)(F)F 65308,C(=O)(C1=COCCO1)NCC1(NC(=O)Cc2cnc(C(F)(F)F)s2)CCOCC1 65309,C1(NC(C(N2CC(CCOC)OCC2)C)=O)Cc2ccccc2C1OC 65310,c1(OC)cc(C(=O)NC2CCC2CNC(=O)C(C)NC(C2C=CCC2)=O)ccn1 65311,C1(C)(C(=O)NC2(COC)CN(C(=O)C=Cc3nccn3CC)C2)CCCC1(F)F 65312,C1(O)(C(=O)NCCC2CCC(NC(C=CCCC)=O)C2)CCOCC1 65313,Cc1cc(NC(C2(C(=O)C3CC3)CC2)=O)ccc1NC(=O)C(N1CCCC(C)C1)=O 65314,C(=O)(CC(O)CNC(C1COCC1C(N)=O)=O)NCCc1cc(C)ns1 65315,c1(CC(C)C)ccccc1NC(=O)CC1CCCN1Cc1ccc(F)cc1 65316,C=C(Cl)CC(C(=O)NCC(=C)C)NC(C1C=CCS1)=O 65317,C=CC(C)CC(=O)NCC1CC1CNC(=O)C(c1ccn(C)c1)C 65318,N1(C(C(c2ccccc2)SCC)=O)CC2C(CNC(C3CCOC(C)C3)=O)C2C1 65319,c1(CC(N2C(C(C)NC(CCCC(C)C)=O)CCC2)=O)cnc2ccccc2c1 65320,C1(C(=O)NC2C(CNC(c3c(C)nco3)=O)CC2)CN(C)CCO1 65321,C#CC1(C(=O)NCCCc2ccccn2)CCN(C(c2ccc(Cl)cn2)=O)C1 65322,C(c1ccc(C)c(C)c1)=CC(=O)NCCNC(C(C1(O)CCCCC1)CC)=O 65323,CC(CC(=O)N1CCCCC1c1n[nH]cc1NC(c1ccccc1)=O)C(C)(C)C 65324,C1(C(=O)NC(C2CCC2)C)CCCCN1C(c1cc(CO)ccn1)=O 65325,C1(C(=O)NC(C=C)C)(CC)CCN(C(=O)Cn2ncnn2)C1 65326,N1(C(c2c(Cl)nn(C)c2Cl)=O)CCC2CN(C(=O)C3=CCCOC3)CCC2C1 65327,C(=O)(C(CC)(CC)CO)NCC(CC)NC(C1C(C)OCCN1C)=O 65328,CN1CCN(C(C2C=CCCN2C(=O)C(C2(O)CCCC2)F)=O)CCC1=O 65329,C1(C(N(CCCNC(C(C)OC(C)(C)C)=O)C)=O)CCC(O)C1 65330,N(C1CCSc2ccc(Cl)cc21)Cc1c(C)nn(CC(F)F)c1 65331,C(CCCCC(=O)NC1CCN(C(=O)COCc2cc(C)on2)C(C)C1)=CC 65332,c1(C(N2C(CC(=O)NC3CCN(CC)C3)CC(F)C2)=O)ccc2[nH]nc(Cl)c2c1 65333,c1(CNC(=O)NCCn2c(CC)ncc2)cccc(N)c1C 65334,C1(NC(CSCc2ccc(C)cc2)=O)CC(NC(C2(C3CC3)CC2)=O)C12CCC2 65335,c1(C(=O)NCC2C(NC(CC=C)=O)CC2)ccccc1-c1nc(C)no1 65336,c1(CC)c(C)nc2ncnn2c1N1CCC(NC(C2(C)CSC2)=O)C(C)C1 65337,c1(OC)ccc(CN2CCC(CC(N3CCC4(CCC4)C3)=O)CC2)c(Cl)c1O 65338,C(C(C)(C)C(=O)N(CC(O)CN(C(=O)CN1CCS(=O)CC1)C)C)OC 65339,N1(C(C(CC)(CO)OC)=O)CC2(C=C(C(=O)N3CC=CC(O)C3)CO2)C1 65340,c1(C(=O)N(C2CC2)CC2CC3(CC3)C2)cnc(C2CC2)nc1.C1(CC2CC2)C(=O)N1 65341,c1(C(=O)NCC2(O)CCN(C(=O)Cc3ccccc3)C2)ccc(Cl)c(Cl)c1 65342,c1(CC)cccc(C(N2CCC(O)(CNC(C3CC3CC)=O)C2)=O)c1F 65343,C(=O)(C(C#N)C(C)(C)C)N1C(CC(=O)NCC2C(CC)CCCC2)C2CCCC21 65344,N1(C(c2c(CC)ocn2)=O)CCCC(N(C(=O)CC2(O)CCCCC2)CCO)C1 65345,Cc1cc(CN2CCC2C(=O)Nc2cc(F)c(F)cc2I)c(O)c(C)c1 65346,CC(C)(C)S(=O)(=O)CC(=O)N1CCN(C(=O)CC2CCOC2=O)CC2(CC2)C1 65347,C1(NC(C2CC3C=CC2N(C(c2cnc(Cl)s2)=O)C3)=O)CN2CCC1(F)CC2 65348,C(=O)(C(C(C)NC(c1ccc2[nH]ccc2c1)=O)C(C)C)NCC(C(C)(C)C)OC 65349,Cc1cnc(C(=O)NC2CC3CC2N(C(c2nc(Cl)ccc2N)=O)C3)cc1C 65350,N1(c2nnc(C3(Cl)C(C)(C)C3)n2CCC#N)Cc2[nH]nc(CO)c2C1 65351,CC(C)(C)C(CNC(=O)C(C)(C)c1ccc(Cl)s1)NC(c1cn(C2CC2)nn1)=O 65352,c1(COC)nc(Cl)cc(=NCC2(CCNC(c3c(OC)ncnc3C)=O)CC2)[nH]1 65353,CCCCC(C(=O)NC(C(N1CC2(CCC(=O)NC2)C1)=O)C(C)OC)C(C)C 65354,CCC(CC(=O)NOCC(=O)NCC1CCC(=O)O1)CC(C)C 65355,c1(OC)cc(Br)ccc1C(c1nnnn1C(C)C)NCc1cccc(Br)c1 65356,c1(NC(C(N2CCC(C)(C)C2)=O)=O)ccc(F)c(S(=O)(=O)OC(F)(F)F)c1 65357,CCC1=NOC(CNC(C2CCC(NC(=O)Nc3cn(C(C)C)nn3)CC2)=O)C1 65358,N1(C(COC(C)C)=O)CC2CCN(C(=O)CCCF)CC12 65359,C#CC(CNC(=O)CC1CCN1C(=O)CCc1cscn1)CC 65360,c1(C2(C(=O)NC3CN(C(c4c(C)[nH]cc4)=O)CC3F)CC2)ccc(Cl)c(F)c1 65361,N1(C(Cn2nc(C)oc2=O)=O)CCC(C2CC2)C1C(N1CC(c2nc(=O)o[nH]2)C1)=O 65362,c1(C(N2CCC(C(C)NC(=O)CCc3cnc(O)[nH]3)C2)=O)sccc1Cl 65363,c1(N(CC(CCC)O)C)ncc(C)cc1S(=O)(=O)NCC#CC1CC1 65364,c1(C(=O)OCC)cccc(-c2nc(OC3CC3c3nn[nH]n3)n(C)n2)c1 65365,c1(CN(C(=O)OCCC(C)C)CC2(C)CCC2)ccc(S(=O)(=O)N(C)C)s1 65366,Cc1nc(C(N2CC(NC(=O)CN3CCSCC3)C(O)C2)=O)cn1C(F)F 65367,N1(C(C2N(CC)CCC2)=O)C2CCC(C(=O)Nc3ccc4occc4c3)C1CC2 65368,N1(C(C(C)SC)=O)CCN(C(c2cc3n(n2)CCN(C)C3)=O)CC(C)(F)C1 65369,c1(-n2cc(C3(O)CN(C(C4N(CC)CCCC4)=O)C3)nn2)cccc2ccnn12 65370,C1(CN(C(c2nnc(-c3ccccc3)s2)C(=O)NCC(F)F)C)CCCSC1 65371,c1(C(=O)NCCNC(c2c(OC)csc2)=O)cc(F)c(Br)c(C)c1N 65372,CC(C(C)C(=O)NCC(F)F)NC(C1COC(=O)N1C)=O 65373,c1(C(=O)NCC(C(=O)NCC(CC)(C)O)CC2CCCC2)n[nH]cc1[N+](=O)[O-] 65374,C1(NC(C(C)OCC#C)=O)CC2CC1N(C(c1ccc(Br)c(N)c1)=O)C2 65375,C12(CNC(=NCCOCC)NCC3CCOC(C)C3)C3CC(CC13)C2(F)F 65376,c1(CC(C)C)ccnc(NC(=O)CSc2ncccc2F)c1 65377,N1(C2CCN(C(c3ccc(C)c(N)c3)=O)CC2C)CC(C)C12CCOCC2 65378,Cc1cc(C(=O)NC2CN(C(=O)C#CC3CCCOC3)C2)cc(S(C)(=O)=O)c1F 65379,C(c1ccccc1OC)=CC(=O)NCC(=C)CCNC(c1cnsn1)=O 65380,c1(CC(N2CCC(O)(CNC(CCS(C)=O)=O)C2)=O)ccc2c(c1)OCO2 65381,CCN=c1[nH]c(C(=O)NC(C2CCN(C(=O)CNC(C)=O)C2)C)cs1 65382,CC1CN2CCN1CC2C(=O)NCC1CCCCN1C(c1cnco1)=O 65383,C(C)(C(=O)NC1CC1NC(=O)Cc1cncs1)OCC(C)C 65384,c1(CC)ccsc1C(C(=O)NCc1ccco1)N(CCF)C1CC1 65385,C(=O)(C(C(C)C)C(C)C)N1CCCC(C(=O)NC(C#C)C2CCC2)(COC)C1 65386,c1(C(C)=O)cn(C)nc1C(N1CCC(NC(=O)CC23CC(C2)C3)C1)=O 65387,c1(CC(N2CCCC(NC(C(CCC)NC(C)=O)=O)C2)=O)cc(Cl)cc(Cl)c1 65388,C(N=c1[nH]c2c(c(=NCC34CC(CO)(CO3)C4)[nH]1)COC2)c1c(C(C)C)n[nH]c1 65389,Cc1cnc(C(N2CCC3(CC3C(=O)NCCOCC(F)F)C2)=O)c(C)c1 65390,c1(CCC(=O)NCC2(CN(C(C3C(CC)CC3)=O)C)CC2)ncccn1 65391,c1(NCC(C)NC(c2cc(F)c(CO)c(F)c2)=O)ncccc1S(C)(=O)=O 65392,C(C)(C(CC(=O)NCCOC1CC1)NC(C1CC(C(C)C)=NO1)=O)OC 65393,C1(CC(=O)NC(C(=O)N(CCCOC)C)Cc2cn[nH]c2)CC(=O)NC1=O 65394,n1(CC(N2CC(CNC(C(CC(=C)C)C)=O)C2)=O)c(=O)n(CC)c2ccccc12 65395,c1(C(N(C)CC2CCCN(C(=O)CCS(C)=O)C2)=O)ccc2oc(N)nc2c1 65396,CC1C(NC(C2CC(=O)N2)=O)CCCN1C(C1CCCCC1O)=O 65397,CNS(=O)(=O)N1CCN(Cc2ccc(OCC(F)(F)F)nc2)CC1 65398,N1(C(C(CNC(c2ncn(CC)c2)=O)(C)C)=O)Cc2ccc(C)cc2C1 65399,c1(-c2cncc(OC)c2)cccc2c(NC(C3(C4CC4)CC3)=O)cccc12 65400,c1(CCC(=O)OC)c(C(c2c(OCC)cccc2)=O)c(O)nc2ccccc12 65401,CC(C)C1CN2CCC(CC2)CCNC1=O.C(C(C)(C)C)NC(N)=O 65402,C1(NC(CCN2CCN(C)CC2)=O)COCCN(C(=O)CC2CCCC(=O)N2)C1 65403,N1(C(CC2(C#N)CCC2)=O)CCCC(N(C(=O)COC(F)F)CCF)C1 65404,CN1CC=C(CC(=O)N2C3CCCC2CC(NC(=O)CC2(C)CCCO2)C3)CC1 65405,CCC(C)(C)C(O)C(=O)N1CCC(CO)(CNC(C2CC3(CCCO3)C2)=O)C1 65406,C1(CC)(CC)CCCN1C(c1sccc1CNC(C1CC2(CC2)CO1)=O)=O 65407,c1(C(N2C(CNC(c3cccc(F)n3)=O)CC2)=O)ccc2cc[nH]c2c1 65408,C1(C(=O)NC(CNC(c2cc(CC)on2)=O)C2CC2)(COC)CCCNS1(=O)=O 65409,c1(C(N(CCNC(C(CC#C)O)=O)CC)=O)n[nH]c2ccc(F)cc12 65410,N1(C(C2N(C)CC(F)C2)=O)C(C(=O)NCC2CC3CCC3C2)CCC12CC2 65411,N1(C(=O)C=Cc2ccoc2)CCC2C(CCN2CC(O)CCc2ccccc2)C1 65412,C1(CC(N2CCCC(CCNC(=O)CC3OCCCO3)C2)=O)CN2CCN1CC2 65413,C1(C(N2CCCC(NC(C3C(c4n(C)ncc4)C3)=O)C2)=O)CCS(=O)(=O)CC1 65414,Cc1cc(C(=O)NC(C2CCOC2)CNC(c2cc(CO)n(C)n2)=O)ccn1 65415,C(C)(C)(CC(=O)NOC1CCOC1)N(C(=O)CC1CCCO1)C 65416,Cc1cc(C)c(C#N)c(NC(=O)Cc2csc(C)n2)n1 65417,C1(CNC(C(C)(O)c2ccsc2)=O)CC(C(=O)N2CCC(CO)(CSC)CC2)=NO1 65418,CCC(C(=O)N(C(C)CN(C)C(c1cnn(CC)c1)=O)C)N(C)C 65419,Cc1sncc1C(=O)NCCCNC(C1CC1(C)C)=O 65420,c1(-c2c(F)ccc(C)c2F)cccc2c1CCN(Cc1c(C)nn(C)c1C)C2 65421,C1(C(=O)NCC(C)OC)(OC)CCN(C(c2ccc(Br)cc2F)=O)CC1 65422,c1(N(C2CSC2)C(N2CCC(F)(C(F)(F)F)C2)=O)cnc2n1CCC2 65423,CC1(NC(=O)CC2CCCC(=O)N2)CCN(C(=O)Cc2ccsc2Cl)CC1 65424,S(=O)(=O)(CC(=O)N1CCC(C)C1CNC(c1cccc(NS(N)(=O)=O)n1)=O)NC 65425,c1(C(=O)NCC(CC(C)C)NC(=O)C2=C(Cl)CCC2)ccc2c(c1)CCCC2=O 65426,c1(C(N2CC(CC(C)NC(C3CCN(CC)C3)=O)C2)=O)cc2cncn2c(O)n1 65427,N1(C(C(N2CCOCC2)C)=O)CCCC(O)(CNC(=O)C2=CSCCO2)C1 65428,CC1CC(CNC(=O)CCn2ccnn2)CN(C(=O)CSc2cccs2)C1 65429,CC(CCCNC(C1CCCN1N=O)=O)N=c1nc(C2CCOCC2)[nH]s1 65430,N1(C(CCC(C)OC(F)(F)F)=O)CC2(CCCN2C(c2sccc2N(C)C)=O)C1 65431,c1(CC(N2CCC(N(C(C(CC=C)CC)=O)C)C2)=O)nsc2ccccc12 65432,c1(CC)nc(C)c(C(N2CCCCC2CN(C(=O)Cn2cnnn2)C)=O)c(C)n1 65433,N1(C(c2csc(Br)n2)C(=O)NC2(C)CC2)CCCCC1CCn1ccnn1 65434,C(=O)(C(O)(C(F)(F)F)c1ccccc1)N1C(SC(C)(C)C)CN(S(C)(=O)=O)CC1 65435,N1(CC(=O)NC(C2CCOC2)CNC(C(C)(C)C2CC2)=O)Cc2ccccc2C1 65436,N1(C(C(C2(O)CN(C(C(C)(CO)OC)=O)C2)F)=O)CCN(C)CC1C 65437,n1(CCOC)cc(C(=O)NCC(C)NC(=O)C=Cc2ccc(C(N)=O)o2)c(C)n1 65438,N1(CC)CC(C(=O)C2CC2)CC1=O.C(CCC1CC1)(C(=O)NCC1(CO)CCC1)N 65439,N1(C(c2c(CC)cco2)=O)CC(NC(c2csc(-c3ncccn3)n2)=O)C2CC12 65440,Cn1cc(-c2cn(CC(C3CN(C(=O)COC(=O)N(C)C)C3)F)nn2)cn1 65441,N1(C(c2cc(C)sc2C)=O)CCC(CNC(=O)CCOCCN(C)C)C12CC2 65442,C1(CCC)CN(C(=O)Cn2cc(Cl)cn2)CCN1C(=O)CN1CCC(C)(C)C1 65443,CCC(CC)C(F)C(=O)NC1CC2CCC1CN2C(C1CN2CCN1CC2)=O 65444,N1(C(C=C(C)c2ccccc2F)=O)CCCCC2(CCN(C(C3CCO3)=O)C2)C1 65445,c1(C(N2CC3CC(NC(C4(C)CCN(C)CC4)=O)C3C2)=O)n[nH]c2c1COCC2 65446,CC1=NOC2(CCN(c3cc(C(F)(F)F)ncn3)CC2)C1 65447,C1(Nc2ccc(C(=O)OC)cn2)(CNC(=O)Cn2cnnc2)CCCCC1C 65448,c1(C(n2ccnc2)CNC(N(C(c2ccccc2)C)CC)=O)cc(Cl)ccc1Cl 65449,c1(NC(c2c(C)nc(C(=O)Nc3c(C)nsc3)s2)=O)ncc2[nH]ncc2n1 65450,C(=O)(CCC(=O)N1CCC(C(C)(C)NC(C23CC(F)(C2)C3)=O)C1)OCC 65451,C=CCCN=C(NCC(C)(CO)OC)NCc1nnc(C)s1 65452,C1(NC(c2cnc(C3CC3)nc2)=O)CCCCC12CCN(C(=O)C=CI)C2 65453,c1(CC(=O)N(CCCNC(C2C(CC)OCC2)=O)C)ccc(O)cn1 65454,C=CCC(CC(C)C)C(=O)NC1COCC1CNC(=O)CCCn1cncn1 65455,C(=O)(CCCCC1CC1)NC1(CC)CN(C(C(C)OCC#C)=O)C1 65456,C1(CNC(C2N(CC#C)CCC2)=O)CN(C(c2cc(COC)on2)=O)CCN1C 65457,c1(OCC(n2cc(CC3CCCNC3)nn2)C)ccnc(NC(C2CCCC2)=O)c1 65458,N1(C(C(CCC)OCC)=O)C2CCC1CN(Cc1nc(Cl)sc1Cl)CC2 65459,N1(CCCC(=O)NC2CC(F)(CNC(C(C(C)O)C)=O)C2)CCc2ccccc21 65460,c1(C(N2CCCC(NC(C(CC)(C)O)=O)C2)=O)ccc(NC(C)=O)c(Cl)c1 65461,CC1CC(NC(=O)CCP(C)(C)=O)CN(C(=O)COc2ccc(Cl)nc2)C1 65462,N1(C(C2CC2NCc2cc(Cl)cc(Cl)c2)=O)CCN2CCOCC2C1 65463,c1(C(=O)NC2CC(NC(c3nnc(CO)s3)=O)C2)ccccc1-n1cccc1 65464,N1(C(C(CSC)O)=O)CC2(CCCC2NC(=O)Cc2ccnc(F)c2F)C1 65465,CC(C)C(C)(C)C(=O)NC1CC(CNC(C2(C)CC3CCC2C3)=O)C1 65466,Cc1nccc(Cl)c1C(=O)NCCC1(O)CN(C(=O)CC2CCCCC(=O)N2)C1 65467,CON1CC(C(=O)NC(C)C=CC(=O)N(CCC(=O)OC)C)CC1=O 65468,CON(CCC(=O)N1CCC2(CCCN2C)CC1)C(=O)CC1(C#N)CC1 65469,C1(NC(COCCOCC)=O)CC2CN(C(c3nc(O)c(C)s3)=O)CC2C1 65470,C1(NC(C=CC=CC)=O)CCCC1NC(=O)CC(=O)NCC(F)(F)F 65471,O=C1CC(C(=O)NCCCNC(C2(F)CCCOC2)=O)c2ccccc21 65472,c1(OC)cccc(C(C(=O)NC2CC(NC(c3sc(C)cc3Cl)=O)C2)OC)c1 65473,N1(C(CCC2CC(NC(c3nnn(C)c3N)=O)C2)=O)CC(S(C)(=N)=O)C1 65474,c1(C(=O)NCCN(CCC)C(C2CC(O)C2)=O)cc2ccc(C)cc2nc1C 65475,c1(-n2c(C)nnn2)ccc(NC(N2CCC(CO)C2(C)C)=O)c(F)c1F 65476,C(=O)(C1=NN2CCCN=C2N1)NC(C(C)NC(=O)Cc1csc2nccn12)(C)C 65477,c1(OC)ccc(C=CC(=O)NC2(C3CN(C(=O)C(C)O)C3)CC2)c(OC)c1 65478,C(CC(=O)NCC1CC(SC)C1)N(C(=O)CC1CC1(C)C)CC 65479,c1(OC)ccc(C(=O)NCC2CC(C)N(C(=O)Cc3ccnc(OC)c3)C2)cc1 65480,CC(C)C(C(C)NC(=O)CCCCC1CC1)NC(=O)C(C)(F)F 65481,Cc1cc(O)ncc1C(N1CC(C2CC2)(C(=O)NCC2CC(C#N)C2)C1)=O 65482,Cc1ccc(C(=O)OCCOC2CC(C(F)(F)F)N2)c([N+](=O)[O-])c1 65483,C1(NC(CC2(OC)CCOCC2)=O)CCC2(CC1)CN(C(=O)C(C(C)C)SC)C2 65484,c1(CC)nc(N2CCCC(C3CCCCN3C(c3cnoc3)=O)C2)cc(C#N)n1 65485,N#Cc1ccc(C(O)C(=O)NC2CC(NC(=O)C(F)=CCCF)C2)cc1 65486,N1(C(C2(CN)CC2)=O)CC2CC2(CNCCc2nccs2)C1 65487,C1(C(=O)Nc2cccc(NC(C(CC)(C)CC)=O)c2)CC2CCCCN2C1 65488,C1(CNC(c2c(Cl)cc(C)nc2)=O)CN(C(c2c[nH]ccc2=O)=O)C2CCN1C2 65489,C1(NC(c2c(C)coc2)=O)CCCC1(C)CNC(c1ccoc1Cl)=O 65490,c1(CC(=O)NC2CC(N(C(c3c[nH]c(=NC)o3)=O)C)C2)c(OC)cccc1Cl 65491,C1(NC(C(C)SCC)=O)CC2(CCCCN2C(=O)CCCCC(F)F)C1 65492,C1(C(=O)NC2(CCCNC(CN(C)C(N)=O)=O)CC2)CNC(=O)CC12CCC2 65493,N1(C(CC2(C=C)CC2)=O)CCC(C2CC2NC(C2(C)CS(=O)(=O)C2)=O)CC1 65494,C#CC1(O)CCCN(C(=O)CNC(=O)CNC(c2ccsc2)=O)C1 65495,C(=O)(C#CC1CCCCO1)NCCCC1OCCN(C(c2c(C)nc(O)[nH]2)=O)C1 65496,CC1(C)C(C(=O)NCC(O)CNC(C2(C)COC(=O)N2)=O)CCS1(=O)=O 65497,[N-]=[N+]=NCCC(=O)NC(C(=O)NCC(F)Br)C1CC1 65498,Cc1cnn(CC(N2CCC(C)(CNC(=O)COCC3CC3)C2)=O)c(=O)c1 65499,Cc1ccc(C(N2CC(N(C)C(c3ncn4c3CCCC4)=O)C2)=O)c2c1CCC2 65500,c1(-c2cc(C(=O)NC(Cc3n(C)ncc3)C(=O)O)no2)cccc(F)c1O 65501,C(CC(=O)NOCc1cn(C)nn1)(C1CC1)NC(C1(CC)CCCO1)=O 65502,N1(C(c2cncc(C)n2)=O)CCCC2C(CCCN2C(=O)COCC(C)(C)C)C1 65503,C1(C(=O)NCC(C)(C)OC)CCN(C(=O)C(N=[N+]=[N-])OC(C)(C)C)C12CCC2 65504,N1(C(C2(C)CC2)=O)CC2(CC2)CC1CNC(C1CC2(CCC2O)C1)=O 65505,Cc1cc(C(=O)NC(CO)C(C)NC(=O)C(O)CC2CCCC2)c(Cl)cn1 65506,c1(C(=O)NCC(C2CC2)NC(CCSCC)=O)csc(C(=O)OC)c1 65507,C(c1ccccc1[N+](=O)[O-])=CC(N1CC2(N(C(C3C(CC)C3)=O)CC2)C1)=O 65508,C(=O)(C1CCCc2nncn21)N1CCN(CCNC(C2(C)CC=CCC2)=O)CC1 65509,N1(C(CCCCCSC)=O)CCN2C(=O)C(NC(c3cc(C)n(C)n3)=O)CC2C1 65510,O=C1CC(CC(=O)Nc2ncc(C3CCOCC3)o2)c2ccccc2N1 65511,c1(CCC(=O)NC(CNC(CNS(CC)(=O)=O)=O)(C)C)ccccc1 65512,C(=O)(CC1=CCOCC1)NC1CN(C(CCOCCCOC)=O)C1 65513,c1(C(N(CCNC(=O)C=CC=C(Cl)Cl)CC2CC2)=O)cccc2nccn12 65514,C(c1cnc2ccccc2n1)=CC(=O)NC(C)(CNC(c1ccnnc1)=O)CO 65515,N1(C(Cc2cn(CC)nn2)=O)CCCC(NC(=O)C(C)(C)C(C)C)CC1 65516,CCC(=O)CCC(=O)N1CCOCC1CCNC(=O)CCc1cccc(C)c1 65517,C1(C(N2CCC(C(C)(C)O)C2)=O)(SC)CN(C(=O)Cc2ccccc2)C1 65518,Cc1ccc(C(N2CCC3CCCC23CNC(c2csnn2)=O)=O)c(=O)n1C 65519,CC1CN(C)CC(C(=O)NCC2CCN(C(c3cn(C)nc3-c3cccs3)=O)C2)O1 65520,c1(CCC)n[nH]c(=NCC(C)(C)NC(c2cnc(O)nc2O)=O)s1 65521,Cc1ncsc1C=CC(N1CCC(N(C(=O)C(C)CF)C)C1)=O 65522,N1(c2ccc(N(C)C(c3ncncc3Cl)=O)cc2)CCc2ccccc2C1 65523,N1(C(CC(C)OC)=O)CC(C2(NC(c3ccc(Cl)cc3C(F)F)=O)CC2)C1 65524,S(=O)(=O)(c1c[nH]c2ncc(Br)cc12)N(c1ccccc1)CC1(C)CCN(C)C1=O 65525,Cc1ccc2nc(C(=O)NCC3CCCC3NC(=O)COCCF)ccc2c1 65526,N1(CC)CCOC(C(N2CCC(CNC(c3cc(C)sn3)=O)C2)=O)C1 65527,N1(C(c2c(C)cccc2Br)=O)CC2(CCN(C(=O)CC(C)(C)O)CC2C(=O)O)C1 65528,C1(NC(C(=O)NCCOC)=O)C2CCC1N(C(=O)C(c1ccc(OC)cc1)C)C2 65529,C(=O)(C(C)(F)C(=O)Nc1nc(OC)cc(N2CCN(CCO)C(=O)C2)n1)OCC 65530,CS(=O)(=O)C1(C(=O)NCC2(NC(C3CC(=C(F)F)C3)=O)CCOC2)CC1 65531,C(=O)(C(C)(C)C)NCC(=O)NCCOCCNC(C1C(CC)C1)=O 65532,N1(C(c2cc(F)ccc2F)C(=O)NCCSC)CCN(C)C2(CC2)C1 65533,N1(C(=O)C=CC2CCCO2)CCOCC(NC(=O)C(F)(F)Cl)C1 65534,C(C1=CCCN(C(=O)CN2CCCCC2)C1)OCc1ccc(OC)cc1 65535,C1(NC(C2C(C(C)(C)C)CC2)=O)CCCCCN(C(=O)C=CCO)C1 65536,c1(C(N2C(CNC(=O)Cc3cncnc3)CC2)=O)ccc2c(c1)NCCC2 65537,C1(OC)CC(C)CN(C(=O)C(F)C(C)CNC(c2occc2C)=O)C1 65538,Cc1n[nH]c(C)c1CC(N1CCC(NC(C2(n3cncn3)CC2)=O)CC1)=O 65539,N1(C(c2c(C)n(CCO)cc2)=O)CCCN(C(C2C3CN(CCO)CC23)=O)CC1 65540,CCCC(C(O)C(=O)N1CCOCC1)NC(c1c(F)ccc(F)c1F)=O 65541,N1(C(CCCC#C)=O)CCCCCC1CNC(c1cc(C)nnc1CC)=O 65542,N1(C(C2NCCN(C(c3scc(C)c3C)=O)C2)=O)CCCC(C)(O)C1 65543,N1(C(c2c(C)cccc2)=O)CCC2CCC(NC(=O)C(c3ccccc3)F)C1C2 65544,C(=O)(C1=CC2(CCOCC2)C1)NCC1(C(N)=O)CN(C(CCCC(CC)C)=O)C1 65545,c1(C(N2CC(C)C(NC(c3cccnn3)=O)CC2)=O)c(Cl)ccc(Cl)c1O 65546,c1(C(C(=O)NCCC)N(CC2CCCCCC2)CC2CC2)cccc(OC)c1F 65547,N1(CCOC)CC(C(=O)NCCc2cccnc2OC)CC1=O 65548,Cn1ccnc1CN1CCCCC1.C(=O)(C(N)CC1CCOC1)N 65549,C(=O)(C(C)CC(F)(F)F)NC(CC(C)C)CNC(=O)C1=CCSC1 65550,N#Cc1c(F)cc(NC(N2CCN(CC3CC3)CC2)=O)cc1Br 65551,CC1C(C(=O)NCCCCCCF)CCCN1C(C1CCCC(=O)N1C)=O 65552,CC1CC(NC(=O)COC(F)F)CCN1CCOc1ccccc1C(N)=O 65553,C1(CC)(CO)CN(C(=O)CC2CCC(NC(=O)CCC3CC3(F)F)C2)C1 65554,C1(C(N2CCC(COC(C)(C)C)C2)C(=O)NCC)CCOCC1 65555,C(=O)(C(C)(O)CC(F)(F)F)N1CC(NC(CCCC(C)(C)OC)=O)C(O)C1 65556,c1(CCC(=O)NC2CN(C(C3(COC)CC3)=O)C2)ccccc1Br 65557,N1(C(CN(C)C(=O)C2CC2)=O)CCCCC(NC(C2CCCCC23CC3)=O)C1 65558,c1(C(=O)NC2C(NC(C3(C)ON=C(C)C3)=O)C2)c(Cl)ccc(F)c1N 65559,CC(CCCCNC(=O)COC(C)(C)C)NC(=O)C=CSc1ccccc1 65560,C#Cc1cccc(CC(=O)NC(C(=O)NCC(=O)OCC)C2CCCO2)c1 65561,n1(CC(N2C(CNC(C(C)OCC=C)=O)CC2)=O)nnc(C2CC2)n1 65562,Cc1ccc(C=CC(=O)NCC23CCCC2CCN3C(=O)COC(C)C)cc1C 65563,C1(C(=O)NCC(C#C)C(C)C)CC2CN(C(=O)C=CC(=O)N(C)C)CC12 65564,c1(C(N(C(C)CNC(c2cc(O)nc(O)c2)=O)C)=O)ccc(F)c2ccncc12 65565,Cc1cc(Cl)c(Br)cc1S(=O)(=O)N(C1Cc2ccccc2N1)C1CCN(C)CC1 65566,c1(C(=O)NCC(CNC(=O)C(F)(F)c2nccs2)OC)cccc(F)c1N 65567,c1(NC(C(=O)NCCC2CN(C)C(=O)C2)=O)cccc2c1COCC2 65568,CC1CCCC1CC(=O)NCC(C)(F)CNC(=O)Cc1cccs1 65569,C(CS(=O)(=O)CC(=O)NC1CCC1NC(c1c(C)ncn1O)=O)OC 65570,C1(=O)CCCCNC2(CC2)C(=O)NC(C(=O)OCC)Cn2cc1nn2.C(N)(=O)SC 65571,N1(C(C)=O)CC2CC2(C(=O)NC(c2ccccc2)c2cnsn2)C1 65572,c1(OC)ccc(C(C)C(=O)NCCCCCNC(=O)CSC2CC2)c(C)c1 65573,c1(CN2CCC(C(N3CC(=O)NCC3)=O)C(O)C2)ccc2nc[nH]c2c1 65574,C(=O)(C(C)(C)CCC#N)N(CC(C(N1CC(C(=O)NC)OCC1)=O)C)C 65575,c1(C(N(C(C)CNC(=O)C=Cc2ccnn2C)CC)=O)ccc(C(C)C)cn1 65576,C1(C(C)NC(C(C)(C)NC(=O)NCC=C)=O)CCCN(C(c2cc(Cl)c[nH]2)=O)C1 65577,CCC(CC(=O)NC1CC2CCC1CC2NC(c1cn(C)[nH]c1=N)=O)C(C)C 65578,FCCCC(N=c1[nH]c(=NCCC(F)(F)Cl)[nH]c2c1SCC2)c1ccccc1 65579,c1(-c2cccc(NC(C3N(CC)CCCC3)=O)c2)cnn2c1NCCC2 65580,CN1CCC(F)(CNC(=O)C(C)(CO)NC(=O)CC2CNC(=O)O2)C1 65581,CC1OCCCC1C(=O)NCc1nnn(C)c1C(N1CCC(C)(C(N)=O)C1)=O 65582,C1(O)(CCNC(C2CC(=O)N(C3CCCCC3)C2)=O)CCN(C(=O)CCF)C1 65583,Nc1ccc(-c2nc(C(N3CCCC3)=O)n(-c3ccnc(Br)c3)n2)nc1 65584,CCCC(CNC(=O)CC(C)n1cccn1)C(=O)NC1(C2(OC)CCC2)CC1 65585,c1(CC(=O)NCC2(NC(C(CCC)NC(C)=O)=O)CC2)ccc(C(C)C)c(C)c1 65586,C=CCCCCCCCC(=O)NC(C1CCN(C(=O)CCC(=C)C)C1)(C)C 65587,c1(CCC(=O)NC(C(C)NC(C(C)OCCOC)=O)C)cccc2c1OCO2 65588,C1(C(N2CCOCC2)=O)(NC(C=C(C)C)=O)CCCCC1.c12cccc(c1)C2 65589,N1(CC)CCC(=O)N(CCc2ccc(F)cc2C)C1=O.C1CCN1S(C)(=O)=O 65590,C1(CN(CCC(=O)OCC)C2CC2)CCS1(=O)=O 65591,CN1CCc2[nH]c(=NCC3CCCN3C(=O)CSCC(F)(F)F)c(C#N)cc2C1 65592,c1(OC(C(=O)NCCNC(C2C(C(C)C)OCC2)=O)(C)C)ccc(Br)cc1 65593,N1(C(=O)CC2CC3(CCC3)CO2)CC2CN(C(C34CCC(C3)C4)=O)CC2C1 65594,N1(C(C(C(C)C)C#N)=O)CCc2nc(CNC(=O)CCn3ccnn3)sc2C1 65595,c1(C(=O)NC2C(CN)CCC2)cnn(-c2cccc(F)c2)c1C(F)(F)F 65596,Cn1cnc2[nH]c(C(=O)NCC3CC(NC(C4CC5COCCN5C4)=O)C3)cc12 65597,C1(NC(C)=O)CCN(C(C2COCC2NC(=O)C(=CC2CCCC2)C)=O)C1 65598,c1(N(C)Cc2nc(CC)sc2)cc(C)c(S(=O)(=O)N2CCCC(C)CC2)cn1 65599,C1(C(=O)NCCC2CCOC2)CC2(CC2)CN1C(=O)C=CC(F)F 65600,C=CCC(C)(C)CC(c1nnnn1CCSC)NC1CC(C)C1 65601,Cc1nnc(CCC(=O)NCC(C)CNC(=O)C(F)(F)CF)n1C 65602,N1(C(CS(CCC)(=O)=O)=O)CCC2CCN(C(C3CCCS3(=O)=O)=O)C2C1 65603,c1(OC)cn(C)c(C(N2CC3CN(C(C4CC5CCC4O5)=O)CC3C2)=O)cc1=O 65604,C1(Cc2cn(CCC=C)nn2)CCCCN1C(c1scnc1C(F)F)=O 65605,c1(C(=O)NCCN(CCC)C(C2CCCCN2C(C)=O)=O)ccc2ncccn12 65606,N1(C(C(C2CCCC2)NC(CCCCC)=O)=O)CC2(CCC(=O)NC2)C1 65607,c1(C(N2C3CN(C(c4c(C)nccc4)=O)CC2CC3)=O)c(Cl)c([N+](=O)[O-])nn1C 65608,CC1=NOC(C(=O)NC(CNC(C2CC(NS(C)(=O)=O)C2)=O)CC(C)C)C1C 65609,N1(C(c2c(C)nc(COC)s2)=O)CCC(C2CC2)C1CNC(C1CC1C(C)O)=O 65610,c1(COCC(=O)N(CCC(C)NC(C2CC(Cl)(Cl)C2)=O)C)nnc(S)n1C 65611,C(=O)(N=c1[nH][nH]c2ccccc12)C1N(C(C(c2ccc(O)cc2)C)=O)CCSC1 65612,N1(C(c2cnc(OC)s2)=O)CCCCC1CCNC(=O)CCc1cc(Cl)cs1 65613,c1(C(=O)NCC2CC3(CN(C(C=CC)=O)C3)OC2)ccc2c(c1F)CCC2 65614,CCC(C)(C#N)C(=O)N1CCC(NC(c2cc(Cl)ccc2OC(C)C)=O)CC1 65615,c1(-c2ccc(C)c(OC)c2)ccccc1S(=O)(=O)N(CC(O)CN)C 65616,N1(C(C(N2CCN(C)CC2)C)=O)CC(NC(C23CCCN2CCC3)=O)CCC1C 65617,N1(C(=O)CCC2CCCC2)C(C(=O)NCC2(CF)CCC2)CCC1C1CC1 65618,C1(C(N2CC(OC)(CNC(c3cc(C4CC4)no3)=O)C2)=O)CC(C)OC1C 65619,c1(CCC)cc(C(=O)NC(c2cccc(C)c2)CNC(=O)C(C)SCC)c(C)o1 65620,C1(C(=O)NCC(C(CC)C)(C)O)CC(C)(C)CCN1C(=O)Cn1nccn1 65621,c1(C(N2CCOCC(C)C2)C(=O)NCCC2(C)CC2)ccc(F)c(Br)c1F 65622,C1(C)(C(N2CC(NC(C(C)=C(C)C)=O)C(CO)CC2)=O)CCC2(CC1)OCCO2 65623,c1(OC)nn(C)cc1C(=O)NCC1(C)CCCN1C(=O)C=CCCc1ccccc1 65624,C(CC(=O)N1CC2(CSC2)C1)(C(F)(F)F)NC(c1n(CCC)ncc1)=O 65625,Nc1ccnn1CC(N1CCCC1CNC(C1(CC2CC2)CC1)=O)=O 65626,c1(SCC(=O)NCc2nnc(-c3ccc(F)c(Cl)c3)o2)nc2cnccc2s1 65627,CN=c1[nH]c(N(C(C2CC(=O)N(C(C)C)C2)=O)CC2CC2)ncc1Cl 65628,N1(C(CC2C(=O)OCC2)=O)CC2(CC(C(=O)NCC34CCC(CC3)CC4)CO2)C1 65629,Cc1cc(Br)c(Cl)cc1C(=O)Nc1cncc(C(F)(F)F)n1 65630,C1(OCC)CC2(C1)CC2C(N1CC(OCC)C1)=O.N1(CC(=O)N)CCC1C.C1CO1 65631,C#CC1(C(N2CCOCCC2C)=O)CCN(C(=O)CCC(C)(F)F)CC1 65632,CC1CCCC(CC(=O)NC(C2CCN(C(c3ccn(CCF)n3)=O)CC2)C)O1 65633,c1(C(=O)NCC(c2ccccc2)CNC(CSC)=O)cc(C2(O)COC2)on1 65634,C(C(CNC(c1cc2n(n1)CCC2)=O)C(F)(F)F)NC(CSCCOC)=O 65635,C1(F)(CNC(CC(C)NC(C)=O)=O)CCN(C(=O)C(C)C(C)(C)C)CC1 65636,C1(C(=O)NC(C)C)CC12CCN(C1CCC(=O)N(Cc3ccccc3)C1)CC2 65637,CN=c1cc(C(=O)N(CCCCN(C)C(C2CCC3C2C3(F)F)=O)C)cc[nH]1 65638,N1(C(=O)CCc2cccnc2)CC2(C1)CN(C(C1(CCF)CC1)=O)CCO2 65639,c1(C(c2nnnn2C2CCC2)NC(c2ccccc2)CC)cn(C)nc1C(F)F 65640,CCC(C(=O)Nc1cccc(C(C)(C)C)n1)C(C)C 65641,C1(C(N2CCN(C(=O)Nc3ccc(F)cc3F)CC2)=O)CCc2cncn2C1 65642,Cc1ccc(N(C(=O)NCC2CC2c2ccco2)Cc2ccncc2)cc1 65643,C1(NC(C=CC(C)(C)SC)=O)COCCC1NC(=O)C(C)(O)C1CC1 65644,c1(C(=O)NC2(CCOC)CCN(C(=O)C3=CCCO3)C2)cc(Cl)ccc1C 65645,C1(C2CC(NC(=O)Cc3cnc[nH]3)C2)CCN(C(C2(C3CC3)CCCO2)=O)CC1 65646,C1(CNC(c2ccc(Br)o2)=O)CCC2(CN(C(c3c(O)cccc3F)=O)C2)O1 65647,CC1CCCC1C(N1CC(C)(CC(=O)NCc2ccc(Cl)s2)C1)=O 65648,C1(CC(N2CCC(CCNC(C3(CC)CCOCC3)=O)C2)=O)CCCS(=O)(=O)C1 65649,Cc1ncnc2c1CC(NCc1cn(C3COCC3OC(=O)N(C)C)nn1)CC2 65650,C1(N(CC#C)C(C2CC=CCC2)=O)CCN(C(c2ccnc(C(C)C)n2)=O)CC1 65651,C(=O)(C(C)=NOCC#N)NCC(CNC(=O)CNC(=O)CC(C)C)OC 65652,N12CC(=O)N(C1=O)CN2C.Cn1cc(CC2CCC2)c(C2(C(=O)O)CCCC2)n1 65653,N1(C(CC(=O)NCC)=O)CCCC1(C)C(=O)NC(C1(OC)CCC1)C 65654,Cc1cc(=O)oc(C)c1C(=O)NCCc1ocnc1CNC(=O)C=CC1CCC1 65655,C1(F)(C(N2CCC(C)(CCNC(C3(C#C)CCC3)=O)C2)=O)CCCN(C)C1 65656,c1(C(=O)NCCCN(C(=O)C(C)(O)C2CCOC2)CC)scnc1Cl 65657,c1(C(=O)NCC2CN(C(c3cnc(COC)s3)=O)CC2C)cnc(Cl)cc1Cl 65658,CCCC(CCC)C(=O)N1CCC(C(=O)NC(C)CC(C)C(F)F)O1 65659,C1(CNC(C2CC(=O)NC2)=O)CCCCN1C(=O)CCNc1cncnc1 65660,c1(OCCC(=O)NCC(C)CN(C)C(C2CC(F)C(=O)N2)=O)cccc(Cl)c1 65661,c1(-c2cc(N3CCN(C(CCC(C)N(C)C)=O)CC3)n[nH]2)ccc(F)c(C=O)c1 65662,N1(C(C(N2CCN(C)CC2)C)=O)CCC(C2CCCN(C(C3(CF)CC3)=O)C2)C1 65663,C(CC(F)F)(C(=O)NCCN1CCCCC1C)NC(CC=C)=O 65664,c1(C(=O)NCC(CCOC)NC(c2oc(C)nc2C)=O)ccc(C(C)C)nc1O 65665,N1(C(c2nnc(C)o2)C)CCC(NC(c2cccc(F)c2Cl)=O)C(C)C1 65666,C(CNC(c1cncnc1)=O)(CC(F)(F)F)NC(c1cnc(SC)s1)=O 65667,C=CC(C)(CC)C(=O)NCc1ccc(CNC(=O)C(C)NC(=O)CC)cc1 65668,n1(CC(=O)NC2CCCN(CCC)C2)cc(Br)ccc1=O 65669,c1(C(N2CC(C(C)NC(C3C4CCCCCC34)=O)C2)=O)cccc2c1COC2 65670,c1(C(=O)NCC2(NC(C3CC(C)C3)=O)CCCCC2)cc2n(c1)CCOC2 65671,C1(NC(c2ccnnc2)=O)CC2(C1)CN(C(c1cn(-c3ccccc3)nn1)=O)C2 65672,C(=O)(CC(CC)C(C)C)NC(CCC)CNC(=O)CCOC 65673,C1(CC)CN(C(=O)Cc2occc2C)CC1NC(c1ccc(C(C)(F)F)cc1)=O 65674,C12CCN(C1)C(=O)CO2.c1(SCCNC(C2CC(=C3CCC3)C2)=O)cccnc1 65675,Cc1c(C(=O)NCCC2(C(=O)NC3COCCN(C)C3)CCC2)cncc1F 65676,CCC(C)CC(C)C(=O)NCC(C(C)C)NC(c1n[nH]c(C)c1Cl)=O 65677,c1(C(=O)NC2CCC(N(C(C(CC)n3ccnc3)=O)C)C2)ccc(F)c(C)c1O 65678,Cc1cnc2n1CC(C(=O)NCC(F)CNC(c1csc(Br)c1)=O)CC2 65679,C(=O)(CCP(C)(C)=O)NC(C(=O)NCC#CCOC)CCOC 65680,c1(NC(C)=O)ccc(Cl)c(C(N2CC(CN(C(=O)CC3CCCO3)C)C2)=O)c1 65681,c1(SC(c2ccc(Br)cn2)COCC)cccc(Br)c1F 65682,C(=O)(CCC(O)C(C)(C)C)N(CCC(C(C)C)NC(c1csc([N+](=O)[O-])c1)=O)C 65683,C(=O)(C#CC1(C)COC1)NC(C(C)NC(c1c(C)nn(C)c1Cl)=O)C 65684,N1(C(c2c(C)con2)=O)CCC2(CCCN2C(=O)C=CBr)C1 65685,N1(C(CCC(C)SC)=O)CCCC2(CCN(C(c3c(C)ccnc3C)=O)C2)C1 65686,c1(C(N(C2CCN(C(C3(CO)CCC3)=O)CC2)CCCC)=O)nnc(O)nc1O 65687,CC1CCCC1(C(=O)NCCc1cc[nH]n1)NC(=O)COCCN(C)C 65688,Cc1cc(C(N2CCC(C)C(CNC(=O)CC3(C)CCOC3)C2)=O)cc(C#N)c1 65689,c1(C(N(C(CNC(C2(C(=O)OC)CC2C)=O)C2CC2)C)=O)ccc(F)cn1 65690,C(c1ccc(C)c(Cl)c1)=CC(=O)NCC1CN(C(CC(=O)NCC)=O)CC1(F)F 65691,Cc1cccc(CC(N2CCCC(NC(=O)C(F)n3ccnc3)C2)=O)c1Cl 65692,C(=O)(C(CCC)CC(C)C)N1C(CC(=O)NC2(C#C)CC2)CC(F)C1 65693,C(=O)(C1CCCc2n[nH]cc21)N1CCC(COC)(NC(c2c(C)ncn2O)=O)C1 65694,C1(c2ccc(OC)cc2)C(C(=O)OC)=C(C2CCOC2)N(C)C(=O)N1C 65695,c1(C(N(C(c2ccccc2)CNC(C(C)=C2CC2)=O)C)=O)ccc(Cl)c(C)c1Cl 65696,CC(N=c1[nH]c(=NC2CN(C3CCC3)C2)[nH]c2c1CCCC2)c1cn(C)nn1 65697,N1(C(C2CC(OC)C2)=O)CCC(NC(=O)C2=C(Cl)CC2)C2(CCC2)C1 65698,CCC(CC(F)(F)F)C(=O)N(C)CC1CCCN1C(=O)C(F)(F)c1cnnn1C 65699,c1(OC)cc(CNC(=O)C(C)OC(c2ccn(C)c2C(C)C)=O)ccc1OC 65700,N1(C(C(C(C)C)c2cnc(C)s2)=O)CCC2(CC2NC(=O)CC=C(Cl)Cl)C1 65701,C1(C(N2CC(OCC(=O)NC)C2)=O)CC(F)CCN1C(=O)CCCN=[N+]=[N-] 65702,CC1(C)C2CCC1(C(N1CCC(c3ccccc3)C(O)C1)=O)C2 65703,c1(CNCC(c2cccc(F)n2)C)ccc2cccnc2c1Br 65704,Cc1cc(N)ccc1C(N1CCCC(N(C)C(C2CN(C3CCC3)C2)=O)CC1)=O 65705,C(C1=NOC2OCCC12)OC(C1CS(=O)(=O)CC12CC2)=O 65706,n1(CC(=O)NCC2(OC)CN(C(=O)CC3NC(=O)NC3=O)C2)c(C)c(C)sc1=O 65707,c1(C(N2CCC(NC(c3c(CC)ocn3)=O)C(C)C2)=O)nccn2cc(C)nc12 65708,c1(COC)cnc(OC)c(C(c2cc(-c3ccc(C)s3)n(C)n2)=O)c1 65709,c1(OC)ncc(C(N2CCC(C(=O)Nc3cnc(Br)c(Cl)c3)C(O)C2)=O)cc1Br 65710,N1(C(C)=O)CCCC1C(n1cc(Cl)cn1)C(=O)O.C1CCC(=O)NC1=O 65711,c1(C(=O)NC2C(C)CN(C(=O)C3CC3)C2)ccc2nnn(C(C)(C)C)c2c1 65712,c1(C(N2C(C(N(CCCC)CCO)=O)CC3CC32)=O)ccc([N+](=O)[O-])cc1O 65713,c1(C(=O)OCC)cc(N2CCC(NC(C3CC(F)C3)=O)C(O)C2)nc(C)n1 65714,N1(C(CN(c2ccncc2)C)=O)CCCCC1CNC(C1(CN(C)C)CC1)=O 65715,C1(C)CC(=O)N1.CC(=O)NCC(=O)NCCN(C)C 65716,C1(NC(C(=O)N(CCNC(C)=O)CCOCCO)=O)CNC(=O)C1 65717,Cc1cc(C(N2CCOCC2CCO)=O)cn(C)c1=O.C12CCN(C1)C(=O)C2 65718,c1(C(N2CCC(NC(C(CC)(C)O)=O)C(O)C2)=O)[nH]c2ccc(F)cc2c1C 65719,CCCC(C(=O)NCC(C)(C1CC1)NC(c1sc(C(C)C)nc1C)=O)N(C)C 65720,N1(C(CCN(C(=O)CCC2CCCO2)CC2CC2)=O)C2C=CCC1CC2 65721,c1(CN(C2CCCC(O)C2)C)cc(Cl)cnc1O 65722,C1(CCNC(C2(F)CCCCC2)c2n(CCCSCC)nnn2)CCC(C)CC1 65723,N1(C(C(C)(C)C#N)=O)CCCC2CN(C(c3cnc4sccn4c3=O)=O)CCC12 65724,C12(N(C)C)CCC(C(=O)NCCC(C)(C)NC(=O)Cc3cnnn3C)(CC1)CC2 65725,C1(C(N2CC(N(C)C(C3(C)CCOC3)=O)C2)=O)CCCCC(C)(C)C1 65726,c1(C(=O)NCC2N(C(c3nn(CC)c(O)c3)=O)CC2)cc[nH]c2nccc1-2 65727,C1(F)(CNC(c2cc(C3CCC3)[nH]n2)=O)CN(C(C2CCCSC2)=O)C1 65728,c1(CC(=O)NC2C(CC(=O)NCCC(C)C)OCC2)ccnc(O)c1 65729,CCC(CC(=O)NC1CN(C(=O)C(=O)Nc2cnn(C)c2)C(C)(C)C1)C(C)(C)C 65730,c1(C(=O)OCC)cnc(NC(C2CC3(CCO2)CC3)=O)c(N)c1 65731,C1(C(N2CCC(O)(CC(=O)OC)C2)=O)CC(CN)CCO1 65732,c1(NC(c2ccc(NCc3ccco3)cc2)=O)nc(Br)c[nH]c1=O 65733,C(C(C)CC(=O)NC1CC(NC(=O)C=Cc2ccc(-c3ccccc3)o2)C1)OC 65734,C(=O)(CS(=O)(=O)C1CC1)N(CCC(C)(F)F)Cc1cc(NC(C)(C)C)nc(Cl)c1 65735,C1(C(=O)NC2(C)CCOC2)C2CN(C(=O)CCc3nc[nH]n3)CC12 65736,c1(C(=O)NCC(C)(O)CNC(C2(Cl)C3CCC(=O)C23)=O)cc[n+]([O-])cc1 65737,C1(CNC(CC(C)SC)=O)CC(F)(F)CN1C(=O)C=C(C)C1CC1 65738,CC(c1ccc(F)cc1F)=CC(=O)NC(C)C(CO)NC(=O)C(C)(C)C(C)O 65739,C1(NC(C2C(=C)C2)=O)CCC12CCN(C(c1ccc3nn(C)cc3c1)=O)CC2 65740,N1(C(C2(SCC)CC2)=O)CCC2(CCCN(C(=O)C(C3CCC(=O)N3)C)C2)C1 65741,N1(C(c2cc(OC)n(C)n2)=O)CC(NC(=O)Cc2sccc2Cl)C2CCCC2C1 65742,c1(OC)cc(=O)n(C)cc1C(N1CC(NC(=O)C(O)C(F)(F)F)C(CC2CC2)C1)=O 65743,N1(C(C2CC(C)OC2)=O)CCCCC12CC(NC(c1cccc(CF)c1)=O)C2 65744,CCC(C)CCCCC(=O)NCC1(CNC(=O)C(C)CC(F)F)CCCCC1 65745,C1(C(=O)Nc2cnc(N(C)C)c(Br)c2)CCC2(CC1)CS(=O)(=O)C2 65746,c1(C(N2CC(Cn3cc(-c4ccc(Cl)c(F)c4)nn3)C2)=O)cc2n(n1)CCCC2 65747,c1(NC(C(C2CC2Cl)N(C(CC)CC)C)OC)ccccc1CC 65748,C1(CNC(CN(CC)CC)=O)CC2CCC1N2C(c1cc(F)ccc1OC)=O 65749,C1(CNC(c2cnn(CCO)c2)=O)CCN(c2nc(Cl)ncc2Cl)CCC1(F)F 65750,N1(C(CC(=O)NCC#C)=O)CC2(CC2)CC1C(N1CCC(CC(N)=O)C1)=O 65751,C12(NC(C=Cc3c(C)cccn3)=O)CCCN(C(=O)C=CC3CCOC3)CC1C2 65752,C(=O)(CCCCC(C)=O)NC1CCC(N(C(CC(CC)(C)C)=O)C)CC1 65753,CC(C)(C(=O)N1CC2(CCC2NC(=O)CCCCCN2CCCC2)C1)C(N)=O 65754,C1(C(NOCC(COC)O)=O)CCOC1NC(=O)C(C)CO 65755,c1(C(=O)NC(CC=C)CNC(C2(C)CC=CCC2)=O)cc2nc(C)cc(C)n2n1 65756,Cc1ocnc1C(N1CCCC1CCNC(=O)CCC1CNC(=O)N1)=O 65757,N1(C(NOCCC)=O)CCC(CO)C(O)C1 65758,N1(C(CC(C=C)C)=O)CCOCC(F)(CNC(c2cc(OC)nc(Cl)c2)=O)C1 65759,C1(CC=C)(NC(c2ccnc(OC(F)F)c2)=O)CCCN(c2nc(SC)ns2)C1 65760,Cc1cscc1C(C(=O)NCCCC1CC1)N(C1CC1)C(c1ccccc1)C1CC1 65761,c1(-c2nc(C(c3c(OC)cccc3)C)on2)cc(C)cc(O)c1 65762,C1(CC)(NC(C2(C3CCCO3)CCCC2)=O)CCCN(C(=O)CN(C)C(C)=O)C1 65763,N1(C(c2ccn(CCCC)n2)=O)CCC(C2CC(NC(C3CC3(F)Cl)=O)C2)CC1 65764,CC1CC(C)CN(C(C2CC(F)(F)CN2C(C2CCC3(CCC3)O2)=O)=O)C1 65765,c1(C(N2CCC(NC(CCCC=C)=O)C2C2CC2)=O)ncc(P(C)(C)=O)cn1 65766,CCC(C)C(=O)N(C(C)CCNC(c1ccn(C2CCC2)n1)=O)C 65767,c1(S)ccccc1OC.N1(C(=O)NC2C(CC)C2)CCCC1C1CCC1 65768,CCCC(CCNC(=O)CN(CC(C)C)C(c1cncc(OC)n1)=O)C1CC1 65769,C1(NC(C(=O)NCC)=O)CC2CCC1N(C(C1(N(C)C)CCCC1)=O)C2 65770,N1(CCC)CCCC(C(N2CCC(CNC(=O)CSc3c(C)n[nH]c3C)C2)=O)C1 65771,C1(NC(=O)C(F)OC(F)(F)F)C2CC(CN(C(=O)COC(F)F)C2)C1CO 65772,C1(C(=O)NCC(C(=O)NC2(CC)CCCCC2)O)CC(=O)CC12CCC2 65773,N1(C(c2c(C)[nH]cc2)=O)CC2CCCC2C1C(=O)NCCCN1CCOCC1 65774,c1(C(=O)NCC2(C)CCN(C(CC(C)n3cccc3)=O)C2)n[nH]c2c1CSCC2 65775,CN1CCN(C(c2ccccc2CC#N)=O)CC1CNC(=O)C(O)CC(N)=O 65776,c1(C(=O)NC2(C(=O)NC(C=C)CO)CCC2)ccc(C)cc1 65777,C(=O)(C(O)CC(C)C)NCCN(c1ccccc1C(=O)NCCCSCCC)C 65778,N1(C(C23C(C)OC(CC2)C3)=O)CC2(CC(NC(=O)CCS(C)(=O)=O)CO2)C1 65779,C(CCC(C)C)(C(=O)NCCN1CCCCC1=O)NC(CC(CCC)C)=O 65780,N1(C(c2cc(C(C)=O)n(C)c2)=O)CCC2(CNC(c3sncc3C)=O)CCCC12 65781,C1(NC(CC2CC(=C)C2)=O)CN(C(C2(CCCC)CCC2)=O)CC2(CCC2)C1 65782,C12(C(=O)NC(C(C(=O)NC(C34CC(CO3)C4)C)C)C)CCC(C1)OC2C 65783,C1(NC(COCC(c2ccccc2)C)=O)CCC2CC1CN2C(=O)Cn1cnnc1 65784,C1(C(N(CC(C)NC(c2ccnc(C)n2)=O)C)=O)CC12CCc1ccccc12 65785,C1(C(F)F)(CNC(c2scc(OC)c2)=O)CCN(C(C2CN(C(C)C)C2)=O)C1 65786,C(=O)(CCC(C)(C)[N+](=O)[O-])N1CCC(C(C)NC(c2c(C)onc2C2CC2)=O)C1 65787,CC(C(=O)NC1CC(Nc2nccc(-n3ccnc3)n2)C1)C(C)(C)C 65788,CC1CC2=C(C(=O)N1)C(c1sccc1S(C)(=O)=O)NC(=S)N2C1CC1 65789,N1(C(c2ccc(CCC)cc2)=O)CCN(C(C2C(C)(C)C2(F)F)=O)CCC1C 65790,C=CCC(C)(C)CC(=O)NCC=CCNC(=O)CC1CCC(=O)NC1 65791,C1(NC(C2C(C=C)CC2)=O)CCCCN(C(c2ccc(Cl)cc2Cl)=O)C1 65792,C1(CN(C=O)Cc2c(OC(F)F)cccc2F)CCC2(CC2)CO1 65793,c1(C(N2C(CNC(c3c[nH]cc(Cl)c3=O)=O)CC2)=O)cc2c(Cl)ccnc2s1 65794,C1(C(N2CC(NC(CN(C(C)C)C)=O)(CF)C2)=O)CCc2nncn2C1 65795,c1(C(=O)NC2(CCCNC(Cn3ncc(CC)c3)=O)CC2)ccc(N)cn1 65796,C12(C(=O)NC(CC=C)C)CCCC1CCN2C(=O)Cc1ccoc1 65797,C1(NC(=O)CCCc2ccccc2)CC12CCN(C(=O)CCC1OCCO1)CC2 65798,CCCS(=O)(=O)C(C)C(=O)NCCNC(c1ccc(Br)c(OC)c1)=O 65799,c1(C(=O)NC(CNC(C(C)SC(C)C)=O)C2CCC2)c(C)cnnc1O 65800,c1(CC(=O)N(CC(C)NC(C=CCOCCOC)=O)C)c[nH]nc1C(F)(F)F 65801,CCC(C(C)(C)O)NC(=O)C(C1CN(C(=O)CCC(=O)NC)C1)OC 65802,CC1(C)CCC(CCNC(c2c(C(=O)NCc3cn[nH]c3)cnn2C)=O)C1 65803,C1(C(N(CCC(C)(C)O)C)=O)CCCCC1NC(C1(C2CC2)CC1)=O 65804,O=C1COC2(CCN(c3nc(NC4CCC4)c4ncn(CCO)c4n3)CC2)N1 65805,C(=O)(C(C)(C)CC(C)(C)C)NC1CN(C(C(CC)CC(F)F)=O)CC(C)(C)C1 65806,N1(CCC(=O)N(C)CCNC(C2(C)CC2Br)=O)CCOCC1 65807,C12(NC(=O)CSc3ccncc3)CC(C1)N(C(c1cccnc1O)=O)C2 65808,N1(C(c2ccc(CSC)cc2)=O)CC2CC(NC(=O)CCC3CCCO3)CC1C2 65809,C12COCCC1NC2=O.C1(C)(OC)CN(C(=O)C=CC(C)(C)SC)C1 65810,C1(COC)(CNC(C2CC(C(C)C)C2)=O)CCN(C(=O)C(c2ccc(Cl)s2)=O)C1 65811,C(=O)(CCC(C)NC(=O)Cc1cnoc1)NCC1(CC)CCOC1 65812,c12cc(cc([N+](=O)[O-])c1)c1nc2no1.CC1=NOC2(C1)CCC2.C(F)(F)F 65813,c1(N2CCC(N(C(C=C(CC)CC)=O)C)CC2)cc(C)nc2nc(C)nn12 65814,N1(C(C(C)O)=O)CC(CNC(=O)CNc2ccc(Br)cc2)C2(CCC2)C1 65815,Cc1cc(C(=O)NCC(O)CNC(C2NC(=O)OC2C)=O)ccc1C1CC1 65816,N1(CC(N2CC3C(NC(C4C(C)CCO4)=O)C3C2)=O)CCc2sccc2C1 65817,N1(C(C(COC)(F)F)=O)CCC(NC(c2ccc(F)cc2F)=O)C2(CCC2)C1 65818,C1(NC(=O)CCC2CC2(F)F)(CO)CCN(C(=O)Cc2cnn(C(F)F)c2)C1 65819,C(=O)(CCC(C)(C)C)N1CC(CC(C)NC(CCn2c(C)csc2=O)=O)C1 65820,N1(C(c2n(CC)ncc2Cl)=O)CC2CCC2(NC(=O)CCc2cnn(C)n2)C1 65821,c1(SCC(=O)NC2CC3(C(=O)OCC)C2C3)nn(C)c(C)c1Br 65822,c1(C(=O)NC2(CNC(C(C)Sc3ccccc3Cl)=O)CCC2)cnc2n1CCC2 65823,c1(CN2CCC(NC(c3c(C)nc(OC)s3)=O)C(F)C2)ccc([N+](=O)[O-])cn1 65824,Cc1ccc(C)n1CC(=O)NCC1CC(C)N(C(=O)CCc2ccccc2O)C1 65825,CCC(C)(COC)C(=O)NC(C)CCCNC(c1ccn(COC)n1)=O 65826,C1(C(=O)NC(C2CCCN2C(c2cnc(O)s2)=O)C)CS(=O)(=O)C1 65827,C1(C)(C(CC)C)CCN(C(=NCCF)NC(C)(C)C)CC1 65828,Cc1cc2c(CC(=O)NC3CC(NC(c4cc(C(=O)OC)sn4)=O)C3)csc2s1 65829,C=CCC(CC(=O)NCCCF)NC(c1coc(N(C)C)n1)=O 65830,C12(NC(C(C)c3cccs3)=O)CCCC1N(C(c1ccc3n[nH]cc3n1)=O)CC2 65831,C12CC(F)CN1C2=O.c1nc(C)oc1C.C(CC(F)(F)F)ONC(C)=O 65832,N1(C(C=C(C)C(F)F)=O)CCN(C(c2cccnc2Cl)=O)C(CCO)C1 65833,C1(C(N2CC(Nc3ncnc(C)c3F)C2)=O)Cc2cccc(F)c2O1 65834,c1(C(N(C)CC2COCCN2C(C2CC23CCC3)=O)=O)cc2c(nn1)CCCO2 65835,c1(C(=O)NCCN(C)C(C2C=CCCC2)=O)nn(C(C)(C)C)cc1Br 65836,c1(C(N2CC(OC)(CNC(=O)CNS(=O)(=O)CC)C2)=O)cc(NC)ccc1C 65837,CC1=C(C(=O)NCC2CC3COCC3N2C(=O)CC(C)CC(C)C)CCS1(=O)=O 65838,c1(C(=O)NC2(CCNC(=O)CCOC3CCOC3)CCC2)cc([N+](=O)[O-])c[nH]1 65839,C(=O)(C1COc2ccccc21)N1CC(CNC(CC(C)NS(C)(=O)=O)=O)C(C)C1 65840,C12(NC(c3cc(Cl)cs3)=O)CCCN(C(C3CCCSC3)=O)CC1C2 65841,c1(OC)ccc(Cl)cc1CC(=O)NC1CCN(C(c2cccnc2Cl)=O)CC1C 65842,C1(C(=O)NC(C2(CNC(=O)C=Cc3ccco3)CC2)C)CCN2CCOCC12 65843,C=CCCC(F)(F)C(=O)NCC1CCC(NC(=O)COC(C)C)C1 65844,c1(C(=O)NC(C(C)C)C(=O)NCCNS(N)(=O)=O)cc2cc[nH]c2cn1 65845,N1(C(=O)C=Cc2cncc(O)c2)CC2CCC1CN2C(C1CC1(CC)CF)=O 65846,Cn1c(C(N2CCOC(c3ccnn3C)C2)C(=O)NC(C)(C)C)cccc1=O 65847,N1(C(CC2CCCN(C)C2)C(=O)NC2CCCCCC2)CCCCC2(CCC2)C1 65848,C1(C(=O)OC(C)CF)CC2CC1N(C(=O)OC(C)(C)C)C2 65849,N1(C(C(=C(C)C2CC2)F)=O)CCC(NC(c2cnn(-c3nccs3)c2)=O)C(F)C1 65850,Cc1cccc(C(C(=O)O)NC(=O)NCC(c2cccc(O)c2)O)c1C 65851,[N-]=[N+]=NC1CN(C(C2CCCCC23CC3)=O)CC1NC(=O)Cc1cccnc1Cl 65852,C(CC(C)(O)C(=O)NOCC(N1CCC(c2nn[nH]n2)C1)=O)N(C)C 65853,N1(C(C(CC)OCC)=O)CCC(C)(CCNC(c2cnc(C)[nH]2)=O)C1 65854,Cc1cocc1C(N1CC(CCCCNC2(CO)CCCC2)C1)=O.C(=O)C=CCO 65855,C(C)(CCN=c1[nH]c(=N)[nH]c(=NCc2cocn2)[nH]1)CCc1ccc(C)cc1 65856,c1(C(=O)Nc2n(C)c(C3CCCNC3)nn2)ccc(Cl)c(F)c1F 65857,N1(C(c2c(CC)ncs2)=O)CCC(C2CC2)(CNC(=O)C(C)CO)C1 65858,C(C)(C(C)C(=O)N1CCOC(C)C1)NC(C1(C(C)C)CCC1)=O 65859,c1(C(N(C2CCN(C(=O)CC3CCNC3=O)C2)CCC)=O)ccc(CC2CC2)s1 65860,c1(C(N2CCC(C(C)NC(c3ncccn3)=O)C2)=O)sc2sccc2c1Cl 65861,C(=O)(CCCCCCCCC1CC1)N1CCCC(NC(C(C)CC(N)=O)=O)CC1 65862,C#CCCCCC(=O)NCC(CC1CC1)C(=O)N(CCCCC=C)C 65863,N1(C(CC23C(CN(C(c4c(CC)con4)=O)C2)CC3)=O)CCC(C#N)CC12CC2 65864,C1(C2(O)CN(C(c3cc(C)nc(O)c3)=O)C2)(CNC(CCOC)=O)CC1 65865,N1(C(c2c(CC)onc2C)=O)CC(C)CN(C(=O)CC(O)CN(C)C)C(C)C1 65866,C(=O)(C1CCCc2ncccc21)N1CCC(OCCCNC(CCC=C)=O)CC1 65867,c1(C(=O)NCCN(C(C(CC)(C)C)=O)C)cncc(Br)c1Cl 65868,N1(C(C2CC(CNC(C(C(C)C)=O)=O)C2)=O)CCN(C)C(CO)C1 65869,c1(N2c3nc(c(C)s3)C2)cnn2c1C(=O)NCC2.c1(C2(CC)CC2)nnnn1COC 65870,N1(C(c2ccc(SC)o2)=O)C2CCC1CN(C(C1(C#N)CC1(C)C)=O)C2 65871,C(=O)(CCCCCC(C)C)NCC(CNC(=O)C#CC1CCOC1)OC 65872,C(CS(C)(=O)=O)N(C)C(C1CCC1NC(=O)CCC1CC1)=O 65873,c1(C(=O)NC(C)CCCNC(=O)C=Cc2ccco2)cccc(Br)c1 65874,CCC1=NOC(C(N2CCCC(N(CCF)C(c3cn(C)cn3)=O)C2)=O)C1 65875,N1(C(c2c(C)nn(C3CC3)c2)=O)CCN(C(=O)CSc2nccn2C)C(C2CC2)C1 65876,c1(OC)cc(C(=O)N(C)CCN(C)C(c2cc(N)ccn2)=O)cc2cnn(C)c12 65877,c1(NC(=O)NC2CCN(C(c3cc(O)cc(Br)c3)=O)C2)ccc2c(c1)C(=O)CC2 65878,CONC(=O)C(=O)NCC(O)CN(C(=O)C(CC)n1cncn1)C 65879,C1(C(=O)NC2CN(C(CCC(=C)C)=O)CC2(C)C)CC2CCCC(C1)C2 65880,CC(C)CC(=O)C(=O)NC1CCCC(CC(=O)NCC2(O)CC2(C)C)C1 65881,c1(C(N(CC(=O)N(CC2CC(=C)C2)C(C)C)C)=O)n[nH]c2c1COC2 65882,C1(C(=O)NC(CC)COCC2CC2)CN(C(=O)C(C#N)C(C)C)CCN1C 65883,CC1CC(NC(c2nccnc2Cl)=O)CN(Cc2ncccc2C(F)(F)F)C1 65884,CCC(CC)C(C)C(=O)N(CC(=O)NCc1coc(C)c1)CC(C)C 65885,CC(C)C(C(=O)NC(CCC#N)c1ccccc1)N(C)C 65886,c1(SC)cc(C(=O)NC(C)C(C)NC(c2conc2-c2ccccc2)=O)c(C)o1 65887,Cc1ccc2nc(C(=O)NCc3ccc(C(F)F)cn3)[nH]c2c1 65888,CC(C)(CNC(c1cc(O)ccc1F)=O)CC(=O)NC(C(N)=O)C1CC1 65889,C(C(C)(O)CC(=O)NCC1(CNC(=O)CC(F)F)CC1)OC 65890,c1(C(N2CCC(CNC(c3cc(C)on3)=O)C2)=O)cc2ccccc2c(O)n1 65891,C1(NC(=O)CCc2ccccc2F)CN(C(c2cnc(S)nc2)=O)C2(CCC2)C1 65892,c1(C(N2CCC(N(C(=O)OC(C)(C)C)CC)C2)=O)cccc(Br)c1Br 65893,CN1CCn2cc(C(=O)NCC3CCCN(C(C4CCSC4)=O)CC3)nc2C1=O 65894,C1(C)(CNC(C2(SC)CC(=O)C2)=O)CN(C(c2cc(Cl)n(C)n2)=O)CC1C 65895,c1(C(=O)NC2CC3(CC(NC(C(CC)C(C)C)=O)C3)C2)csc2c1CCC(C)C2 65896,C(C(C(C)(C)C)NC(=O)Cc1cc(C)on1)NC(Cc1ccc(C)o1)=O 65897,CCC(C)C(O)C(=O)N1CCC(F)C(NC(c2cc(Br)cs2)=O)C1 65898,c1(C(=O)NC2CCN(C(c3cc(Br)n[nH]3)=O)CC2)cc2ncccc2s1 65899,N1(C(C2CCC(OC)CC2)=O)CC(NC(C2CCOC(C)(C)C2)=O)C(C)(C)C1 65900,N1(C(c2cc(OCC)n[nH]2)=O)CC2(CCN2C(C2CCC(=O)C(C)C2)=O)C1 65901,Cc1[nH]cc(C(N2CC(NC(C3(O)CC4CCC3C4)=O)C2)=O)c(=O)c1Cl 65902,CC1=NS(=O)(=O)NC=C1C(=O)N1CC2CC1C2NC(=O)CC(O)C(C)C 65903,C1(=O)CC(C)(C)CCN1.C(C)(C(=O)NCC(C)N(CC#CC)C)=CC 65904,N1(C(c2c(C)c(C(F)(F)F)n[nH]2)=O)CCN(C(=O)C(Cl)=CCl)C(C)C1C 65905,CC(CC(=O)N1CCOC(CN(C(=O)Cc2ccn(C)n2)C)C1)P(C)(C)=O 65906,c1(NC(C2C(C(=O)OC)C2)=O)ccc(I)c(C(c2cc(F)ccc2Br)OC)c1 65907,C(=O)(C(C)(O)C(F)(F)F)N1CCCC(CC(=O)NCc2c(OCC)cccc2)C1 65908,C1(SC)CCCC1NC(C1(CNC(=O)C=CCO)CCC1)=O 65909,CC1CC2CN(C1)C(=O)N2.C1(NC(=O)OC(C)(C)C)CCC=CC1OC 65910,n1(CCCC)ncc(C(=O)N(CCC)CCNC(=O)CC(C)SC)c1C 65911,CCC(O)C(C)C(=O)NCCN(C(=O)C(c1ccc(F)c(F)c1)(F)F)C 65912,N1(C(C=NOC)=O)CCCC1C1CCCN1C(c1c(OC)ccnc1F)=O 65913,N1(C(Cn2cc(-c3cccc(CC)c3)nn2)=O)CCC2(CC1)OCCO2 65914,c1(C(=O)NCC2C3CN(CCC=CCC)CC32)cc(C(F)F)ccc1C 65915,c1(C(F)(F)F)cnc(F)c(-c2nc(NCc3cncc(F)c3Cl)cs2)c1 65916,N1(C(CC(C(=O)OC)C)=O)CCC(C)(C)CC1C(=O)NCC1NC(=O)CC1(C)C 65917,c1(C(=O)NCCN(C(=O)C(C)C(C)O)CCOC)c(Cl)oc2ccccc12 65918,C1(NC(C2CCC(C)S2)=O)(CNC(c2cncc(F)c2Cl)=O)CC2CCC1CC2 65919,c1(NC(CC2N(C(C(CSC)O)=O)CC(F)C2)=O)ccc(O)cc1C 65920,Cc1cc(CC(N2CC(NC(c3c(Cl)cncc3Cl)=O)CC(C)C2)=O)cc(C)c1 65921,C(=O)(CC(O)C(C)C)NCCN(C(=O)Cn1ccc(O)nc1=O)CC 65922,N1(C(C2CC(=C)C2)=O)CCC(C)C1CNC(c1cnc(C2CCC2)nc1)=O 65923,Cc1ccc(CCCC(=O)NCC(CC(C)C)NC(C23CCC2C3)=O)cc1C 65924,c1(C(=O)NC2CCCN(Cc3ncccc3C(=O)O)C2)ccc2nnc(Br)n2c1 65925,N1(C(CSCCC)=O)CCN(C(c2cn(CCC)nc2C)=O)CC(O)C1 65926,C1(CNC(CSCC=C)=O)COCC1NC(=O)CSCCC#N 65927,C(=O)(C(C)(F)C(=O)N1CCC(=CCNC(c2ccc(CO)c(C)c2)=O)CC1)OC 65928,CC(C)C1=CCC(NC(C2(NC(=O)C=CC3CC3)CCN(C)C2)=O)CC1 65929,C(=O)(CC#CC(C)(C)O)N1CCC(O)(CNC(C(CC(C)C)F)=O)CC1 65930,C1(CNC(C(C)CC(N)=O)=O)CC2(CO1)CN(C(=O)CC(F)F)C2 65931,C(=O)(CCC(C)(C)F)N(CCC(C)(C)NC(C1CCCC1(F)F)=O)C 65932,n1(CC)ncc(CO)c1C.N12CCN(CC1)C(=O)N2CCOCCO 65933,N1(Cc2cc(OC)cc(Cl)c2)CCC2C1CCCN2c1nc(OC)cc(C)n1 65934,N1(C(c2c(OC)n[nH]c2)=O)CC(NC(c2ccc(Cl)c(F)c2N)=O)C2(CCC2)C1 65935,N1(C(C(N2CCOCC2)C)=O)CCCCC(N(C(=O)C=C(C2CC2)C2CC2)C)C1 65936,CC1CC(C(=O)NCC2(F)CC(CNC(C3(C4CC4)CC=CC3)=O)C2)CCC1C 65937,N1(C(C(C)OCCCC)=O)CCN(C(c2ccc(C(F)(F)F)s2)=O)CC1CCC 65938,C1(C#N)(C(=O)NCC2(OC)CN(C(c3cncc(SC)c3)=O)C2)CCN(C)CC1 65939,c1(OC)ccc(CNc2cnc(F)cc2C(=O)Nc2ncc[nH]2)cc1[N+](=O)[O-] 65940,N1(C(C2C(C)C2)=O)CC2(CC2)CC1CNC(c1ncc(C(F)(F)F)cc1Cl)=O 65941,NS(=O)(=O)N1CCCC(C(=O)NCC(O)CNC(c2c[nH]c(C(N)=O)c2)=O)C1 65942,c1(C(C)NC(N(CCC(C)C)CCCC)=O)scnc1C 65943,CCCCCCCCCCCN(C(=O)C(=O)NC(c1cc(C)ns1)C)C 65944,Cc1ccccc1C=CC(=O)NCC(=O)NC1CCN(C(=O)C#CC2CC2)CC1 65945,c1(C(=O)NC2CCC(N(C(CN(C)C(N)=O)=O)C)CC2)cccc2c1OCCO2 65946,c1(SC)cc(C)c(C(N2CC(CNC(C3(C)CCOC3C)=O)C(O)C2)=O)o1 65947,CC1N(C(=O)C(Cc2ccoc2)NC(c2cccnn2)=O)CCOC1(C)C 65948,CCCCC(C(=O)NCC(CC(N1CC(CO)CC(C)(C)C1)=O)OC)C(C)C 65949,C(C)(CC(=O)NCC(C)(C)CNC(c1cc(N)c(F)cc1F)=O)(C(F)F)N(C)C 65950,C1(CNC(CCN(C)C)=O)CC2(CCOCC2)CN1C(=O)CC1CC2CCC1C2 65951,C1(NC(C(C(C)C)C)=O)CCC(O)CN(C(=O)COc2ccc(F)cc2F)C1 65952,n1(C2N(C(COc3cc(C)cc(F)c3)=O)CCCC2)ncc2c1CCCC2 65953,C1(NC(C(CC)c2ccccc2)=O)CCCC(C(=O)Nc2ccc(Br)cn2)C1 65954,CC1(C)CN(C(=O)NCc2cc3cccnc3s2)C2CCCC12 65955,N1(C(c2c(C)ncs2)=O)CCC2(CC1)CCN(C(c1csc(C)c1C)=O)C2 65956,c1(C(C)N(CC(C)C#N)C(=O)CN(C)C)ccc(Cl)s1 65957,Cn1ncc(Cl)c1C(=O)NCC1CC2CC2N1C(=O)Cn1nnnc1C1CC1 65958,C=CCC(CC(F)F)C(=O)N1CC(CNC(C2(NC(C)=O)CC2)=O)CC1(C)C 65959,C12(NC(CC(C(C)C)C)=O)CC3CC(C1)CC(NC(=O)Cn1cnnn1)(C3)C2 65960,c1(C(CN(C(CCCSCC)=O)C)=O)ccc(F)cc1[N+](=O)[O-].C(N)(=O)OC 65961,C(=O)(NNc1nccnc1C)c1cnc2onc(C)c2c1 65962,c1(C(N(C2CC2)CC2N(C(C(CC)n3cncn3)=O)CCC2)=O)ncccc1C 65963,Cc1cccc(C)c1C(=O)NCCC1COCCN1C(C1CC1C)=O 65964,C1(C(N2CCC(O)(CNC(COCC#C)=O)C2)=O)CCc2nnn(C)c2C1 65965,c1(C(=O)NC2C(C)(C)CCN(C(CC=C=C)=O)C2)cc(C)cc2c1OCC2 65966,C#CCC(C)(CC)C(=O)NC1COCCC1C(N1CCOC(C)C1)=O 65967,CCC(CC(=O)N1CCC(CCNC(=O)C(C)(C)CF)C1)c1ccc(OC)cc1 65968,c1(CNC(C(C=C=C)C)=O)nc2c(s1)CN(C(C1(C(=O)OC)CC1C)=O)CC2 65969,c1(CCC(=O)NC2CC2CNC(C2(F)C3CCCC23)=O)ccc2ncccc2c1 65970,CC1(C)CCOC(Cn2nnnc2N2CCC(C3CC(C(N)=O)CCO3)CC2)C1 65971,O=C(CCC1CC1C(F)(F)F)NCC1CC1NC(=O)CC1CCC1 65972,c1(C(=O)NCC2(F)CCN(C(C3CC(OCC)C3)=O)C2)ccc(C)c(C)c1 65973,C12(C(=O)NCCC(C)(C)CNC(C3CN(C(N)=O)C3)=O)CCCCC1OCC2 65974,C1(NC(CN(C(C)=O)C)=O)(CNC(c2nccn2C)=O)CCC(C)CC1 65975,C(CC(O)CO)N(C)C(=O)NC1C(c2ccccc2)C1(C)C 65976,C1(NC(=O)CCCCN2CCCC2)CC(F)(F)CC1C(=O)O 65977,C1(CNC(Cn2cnc(C(N)=O)n2)=O)CN(C(=O)COC2CC=CC2)CC1C 65978,C1(NC(C(C)(C)CF)=O)CCN(C(C2(O)CC(F)(F)C2)=O)CC1c1ccccc1 65979,c1(N(C)CCC2CCCCN2C(=O)CC2(CSC)CC2)cnc2ccccc2n1 65980,C1(C(C)C)CN(C(=O)C=Cc2cnccn2)CCN1Cc1nc(Cl)ccc1Cl 65981,C(CCC1CC1)(C(=O)N1CCCC1CNC(N)=O)NC(c1cc(C)sn1)=O 65982,c1(OC)cc(CO)ccc1C(=O)NCC1(C)CCCN1C(c1cnco1)=O 65983,c1(N2CCC(N3CCC(=O)NC3=O)C2)cc(=O)n2ccccc2n1 65984,C1(O)(CNC(C2CC(=C)C2)=O)CCCN(C(c2ccc(Br)c(C)c2)=O)C1 65985,c1(OCC)cc(C(=O)NC(CCN(C(=O)C(C)OC)C)C(C)(C)C)oc(=O)c1 65986,N1(C(c2ccn(C(C)C)n2)=O)CCCC(NC(C2CC2c2cnn(C)c2)=O)C1C 65987,c1(Cn2cccc(C(C)NCc3ccncc3)c2=O)ccc2c(c1)CN(C)C2=O 65988,c1(C(N2CCC(NC(c3cncc(C(C)(C)C)c3)=O)CC2)=O)nnn2c1CCC2 65989,c1(CC(C(=O)N(C(CC#C)C)C)NC(=O)C(C)CC=C)cnn(C)c1O 65990,Cn1cc(C(=O)NC2C3CC(NC(=O)CCC4CCCC4)CC23)ncc1=O 65991,c1(OCC)ncccc1CC(=O)NCC1CCN(C(C2(n3nccn3)CC2)=O)C1 65992,C(=O)(C1=CCCCC1C)NCC(C)(C1CC1)NC(c1occ(C)c1)=O 65993,Cc1nc(Cl)ccc1S(=O)(=O)NCC1CN(Cc2cccc(O)c2O)CCO1 65994,c1(-c2c(OCCC)ccc(F)c2)ccc2c(c1)CN(C(=O)C(C)=O)CC2 65995,Cc1cc(F)c(Cl)cc1C(=O)NCC(C)CN(C)C(c1ccc(C#N)nc1O)=O 65996,c1(C(=O)NCC(CO)NC(c2ncc(C)c(C)c2)=O)cc(C#N)c(C)cn1 65997,N1(C(C=CCC)=O)CCN(C(c2cnn(CCC)c2CC)=O)C(CC)C1 65998,c1(NC(C2(OC)CCC(C)CC2)c2nnnn2C)ccc2nn(C)c(C)c2c1 65999,C1(C(=O)NC2(C(=O)NCC3C4CC5C(C4)C35)CCOCC2)CCC2CC1CO2 66000,CN1CC(CC(N2CC(NC(C3CC(N4CCCC4)C3)=O)C2)=O)C1 66001,C1(CCC)(NC(c2n[nH]cc2Cl)=O)CCCN(C(C2CC3(CC3)CO2)=O)C1 66002,c1(OC)cc(C#N)ccc1CN1CC2CC(C1)C(C(=O)O)O2 66003,C(=O)(C1CCc2snnc21)N(C(C)C)CCNC(c1cnn(C(F)F)c1)=O 66004,c1(-c2c(CC)cno2)nc(-c2cccc(OC)c2)nn1C(C)COCC 66005,C1(CNC(CCc2nc(C)sc2)=O)CCCCN1C(C1(C)CCCC1)=O 66006,C1(NC(CC)=O)CC(OC)C12CCN(C(c1c(OC)cccc1Br)=O)CC2 66007,Cn1cc(C(=O)NCC2CN(C(c3ccsc3)=O)CC(C)(C)C2)c(O)nc1=O 66008,C1(CC=C)(C(=O)NCc2nn[nH]n2)CCN(C(C2CCS(=O)CC2)=O)C1 66009,N1(C(c2ncn(CC)c2)=O)CC2(C(=O)N(C)Cc3cnc(C)s3)CCC1CC2 66010,C=CC(C(=O)NC(CNC(C1CCN(CC)C1)=O)C(C)C)OC 66011,S(=O)(=O)(c1ccc(Br)s1)NC(CC(N1CC(C)CC(C)C1)=O)Cc1ccc(F)cc1 66012,N(C(=NCCC(=O)C(=O)CC(F)(F)F)NCC(c1ccccc1)CO)CC.NC 66013,C12(NC(c3cc(COC)cn3C)=O)CCC(C1)N(C(=O)CC1CCCC(=O)N1)C2 66014,N1(C(COC(CC)C)=O)CCN2CCN(C(c3cc4c[nH]cnc-4n3)=O)CC2C1 66015,CC(=O)CCC(=O)N(CC(C)N(C(=O)CCCNC(c1ccccc1)=O)C)C 66016,c1(-n2cc(CNC(C(C)(C)C)C3CC3)nn2)ccc(F)cc1I 66017,c1(CC)ccsc1C(=O)NC(CNC(=O)Cc1ccc(Cl)s1)C1CCC1 66018,C(=O)(C(=O)N=S(C)(C)=O)N1CC(NC(CC2CCC(C)CC2)=O)C(CO)CC1 66019,N1(C(c2n(C)ccc(=O)c2)=O)CCOC2(CCCCC2NC(C2CC2(F)Cl)=O)C1 66020,N1(C(C=C(C)C(C)C)=O)CCC(NC(c2cccc(N)c2F)=O)C(F)(F)CC1 66021,N1(C(c2cc(CC)no2)=O)CC(NC(=O)C(C)SC)C2(CCS(=O)(=O)CC2)C1 66022,N1(CC(C2CCOC2)F)CCC(NCC(F)(F)F)CC1 66023,N1(C(C)C)CCCC1CC(=O)NC(C)CNC(C1(C)CC1C)=O 66024,CC1CN(C(C2(O)CCSC2)=O)CC1CNC(c1cc(-c2ccoc2)on1)=O 66025,c1(-c2cn(C)nc2)ccccc1NC(C1CN(c2ccc(F)cc2)C1)=O 66026,N1(CCC(=O)OC)CC(NC(N2CCC(CO)C(C)C2)=O)CCC1=O 66027,C1(NC(CC(CNC(CCCOCCC)=O)O)=O)CC2C(C1)C2(F)F 66028,C1(C(CNC(C=CC(CC)C)=O)F)CCN(C(=O)C(F)(F)C2CC2)CC1 66029,c1(CC(C(=O)N(C(C)CNC(C2CC2F)=O)C)C)ccc([N+](=O)[O-])cc1 66030,Cc1cccc2[nH]cc(CCC(=O)NC34CC3CN(C(=O)C(C)C3CCC3)C4)c12 66031,C(=O)(C1=NOC(C)C1C)N(C1(CC(=O)NCC(CC)(C)OC)CCCCC1)CC 66032,C1(C(=O)NC(C(C)C)C2CCC2)CCN(C(=O)CC(=O)NC2CC2)CC1O 66033,C1(C(=O)NC2(C)CCN(C(c3ccc(O)nn3)=O)CC2)CSc2ccccc2O1 66034,c1(CC(=O)NCC(CNC(CC2(C)CC2)=O)O)ccc(C(N)=O)cc1 66035,N1(C(c2c(CC)noc2)=O)CCN(C(=O)Cn2c(C)csc2=O)C(CC(F)F)C1 66036,c1(SC)nccc(=NC(CNC(c2n[nH]cc2C(F)(F)F)=O)C(C)C(C)C)[nH]1 66037,CC(=O)CCN=C(NCC1(C2CC2)CC1)N1CCC(CC(C)(C)C)C1 66038,c1(NC(COC)CO)nc(N2CCOC(C3CC3)C2)nc2sccc12 66039,C#CCC(CC(F)F)C(=O)NC1COCCC1c1ccccc1 66040,O=C(C1c2c[nH]nc2CN1C(C1C2COCC12)=O)N1CC2CC2C1 66041,c1(NC(=O)NCC2(C(=O)OC)CCCNC2)ccc2c(c1)C(CC)C(=O)N2C 66042,C(=O)(C1=CCCSC1)NC1C(NC(CCc2ccc(OC(C)C)cc2)=O)CCC1 66043,C1(NC(c2ccnc(OCC3CC3)c2)=O)CCOCC1F 66044,CCC(C)CC(=O)NCC1CCC(NC(=O)C(C)(Cl)Cl)C1 66045,N1(C(CCCc2c(C)ccs2)=O)C(C(=O)NCCOC2CCC2)CC2CC12 66046,C#CC1(O)CCCN(C(=O)CC2CCCN(C(=O)C(F)CN(CC)CC)C2)C1 66047,C12(C(=O)NC(CC)(C)CO)CCC(CC1)N(C(=O)CC1CC3C=CC1C3)C2 66048,C1(CNC(c2ncn(C)n2)=O)CN(C(=O)CC(Cl)Cl)CCO1 66049,C1(C(=O)N)CCC(C#N)C1.C12CC(O)(C1)CO2.n1(CC2(C)COC2)cc(C)nn1 66050,CCCCC(C)CCC(=O)NC1(CNC(=O)C(F)(F)C2CC2)CCCCC1 66051,C(=O)(C(F)CCC(C)(C)C)NCC(C(N1CCC(C(=O)NC)C1C)=O)CC1CC1 66052,C1(C(=O)NCCC2(C(NOCCOC)=O)CCC2)CCCC1C 66053,Cc1nnc(O)c(C(=O)NC2CN(Cc3cccs3)C2)c1C 66054,C1(N(C(CC(CC)N(C(=O)C(C)=NOCC#N)C)=O)CC)CCCCCC1F 66055,c1(C(=O)NCCCCCNC(C2CCC(NC(CC)=O)C2)=O)ncc(F)cc1N 66056,C1(C(N2CCCC(C(C)SC)C2)=O)(C(=O)NC(c2cccnc2O)=O)CCOCC1 66057,N1(C(C(C=C)(C)CC)=O)CCOC2(CCN(C(c3cccnc3)=O)C2)C1 66058,N1(C(c2c(C)onc2-c2ccccn2)=O)CC2CC1CN2C(c1csc(Cl)c1)=O 66059,N1(C(CN(C(C)=O)C)=O)CCC(F)(C(=O)NC(CC2CCC2)CO)CC1 66060,N1(C(c2n(C)nnc2)=O)CCN(C(=O)C(F)=CC2CC2)CC1c1ccccc1Cl 66061,C1(NC(Cc2scc(C)c2)=O)CCN(C(c2cc(C)cnc2Cl)=O)CC1(C)C 66062,C1(C2(O)CCN(C(c3cscc3Cl)=O)CC2)(NC(=O)COCC2CCOC2)CC1 66063,C1(C(=O)NC(C)CCC#N)CCCN(C(C2CCCCC2O)=O)C1 66064,N1(C(CCC=C(C)C)=O)C2CCC1CN(C(=O)Cc1ccc(O)c(O)c1)C2 66065,c1(CC)ccnc(N(C)C(=S)NCC(c2ccc(F)cc2)O)c1 66066,N1(C(CC2C=NN(C)C2=O)=O)CC(NC(=O)CCn2ccccc2=O)CC(F)C1 66067,c1(N(C)C)c(F)cc(C(=O)NC2CC2C(=O)NCc2nc(Br)cs2)cc1F 66068,CCCCC(O)CC(=O)N1CC(C)(C)CC1C(=O)NC1CCCC1N=[N+]=[N-] 66069,N1(CCNC(COCCC=C)=O)CCC(NC(c2sccc2OC)=O)CC1 66070,c1(NC(C2N(S(CCC)(=O)=O)CCC2)=O)cc(C(=O)OC)cc(C(F)(F)F)c1 66071,C(CCC(O)C(=O)N1CCC(n2cnnn2)C1)NC(c1cnnc(O)c1)=O 66072,S(=O)(=O)(c1cccnc1NCCC1CC1(Cl)Cl)NC(C(C)(C)C)c1ncccn1 66073,C1(NC(C2(C=C)CCC2)=O)CCCN(C(c2ocnc2-c2ccccc2)=O)C1 66074,C(C(CO)C(C)CC)NC(c1cc(CNC(C(C=C=C)C)=O)nn1C)=O 66075,c1(C(N2CCC(CNC(C3(N(C)C)CC3)=O)C2)=O)cccc2c1CCCC2 66076,C(=O)(C(F)C1=CCCCC1)NCCN(C(C(Cc1c(C)cccc1)C)=O)C(C)C 66077,N1(C(c2c(CCC)[nH]cc2)=O)CC2CC1CN2C(C1CC1F)=O 66078,N1(C(c2c(C)oc(C(C)C)c2)=O)CC(NC(=O)CC2OCCC2(C)C)C2(CC2)C1 66079,c1(C(=O)NC(CC)CCC(=O)NC2CCN(C)C2)cc(C)cc(C#N)c1 66080,c1(C(N2C(C(=O)NCCSC)CCC2)=O)cccc(-c2ccco2)n1 66081,N1(C(C2CC(OC(C)(C)C)C2)=O)CC(NC(C2C=CCC2)=O)C(O)C1 66082,c1(CNC(N2C(c3cc(=N)[nH]cc3)CCC2)=O)nc2ncccc2o1 66083,c1(C(=O)NCc2c(C3CN(C(C(C=C)O)=O)C3)ocn2)ccc(C2CC2)cc1C 66084,Cc1n[nH]cc1C(=O)N(C1CCC(NC(=O)CC2(CN(C)C)CCCC2)C1)C 66085,CC(C)C(CC(=O)NCC12CCCCC1C2)OC(=O)C(C)OC1CCCC1 66086,c1(CC)nc(C#N)cc(=NCC2(NC(C3CCOC3C)=O)CCCC2)[nH]1 66087,Cc1nc(C)c(C(=O)NC2CCCC(NC(c3cnc[nH]c3=N)=O)C2)o1 66088,Cc1n[nH]c2nc(O)c(C(=O)NC3(CNC(=O)C=CC(F)(F)F)CCOC3)cc12 66089,N1(C(C2CCC(OC)CC2)=O)CC(F)(F)CCC1C.C(=O)N 66090,N1(C(C2N(C)CCC2)=O)CC(O)C(O)C1CNC(C1CC(=C(F)F)C1)=O 66091,N1(C(C2(CNC)CC2)=O)CCCC1C(=O)NC 66092,CC1(C)C(CNC(=O)C(C2CCOCC2)O)CCN1C(c1ccc(F)c(F)c1)=O 66093,C1(N(C(c2cc(SC)oc2C)=O)C)CC2CCC(C1)N2C(=O)CCc1cnc[nH]1 66094,c1(OC)cncc(C(=O)NC(C2CCN(C(=O)CC3CCC(=O)N3)C2)(C)C)n1 66095,c1(OC)ccc(C(=O)N(C2CCCN(C(C3CC(C)(C)C3)=O)C2)CCF)c(Cl)c1 66096,c1(C(N(CCCOCCNC(c2c(C)ocn2)=O)C)=O)sc2ccccc2c1Cl 66097,CC1C(NC(=O)CC(C)(C)C(F)F)C(C)CCN1C(=O)CCOCC(F)F 66098,CC1CC(N=c2[nH]c(=NCc3cc(C(N)=O)no3)c3ncccc3[nH]2)CCS1(=O)=O 66099,c1(C(=O)NC2C(OC)CN(C(=O)C=CBr)C2)nc(C)c(C)[nH]c1=O 66100,N1(C(c2cc(Br)cs2)C(=O)NCC(C)C)CC(C)(C)OC2COCC12 66101,N1(C2CN(C(CCN(CC(C)C)C(C3CC3C(C)C)=O)=O)C2)CCCC1C 66102,C1(NC(c2cccc(CCN(C)C)c2)=O)CCN(C(C2CC(CF)C2)=O)CC1O 66103,C1(CC)CN(C(C2(O)CCCCC2)=O)CCC1NC(C1CCC(=O)N(C)C1)=O 66104,c1(NC(C2(C)CCCN(CC(c3n(C)ccc3)=O)C2)=O)cc(Cl)cnc1Br 66105,C1(C(CC)C)CCCN(C(c2cncc(CNC(=O)C=CC3CCC3)c2)=O)C1 66106,C(N=c1[nH]cnc2c1SCCC2)C1OCCN(C(C=C(C)C2CC2)=O)C1 66107,C(C(O)CCNC(c1csc(-c2nc[nH]n2)n1)=O)NC(=O)CCc1cnn[nH]1 66108,c1(NC2CCN(C(N3C(CC(=O)OC)CCCC3)=O)CC2)ccc(Br)cc1F 66109,C1(C(C)NC(=O)Cc2nnc(O)s2)CN(C(c2ccc(C(F)F)o2)=O)CCO1 66110,c1(C(=O)NC2C(NC(CCN(CC)CC)=O)CC2)cnc(O)cc1O 66111,c1(CC(=O)NC2CCC(CNC(Cc3ccn(C)n3)=O)C2)c(F)cccc1C#N 66112,Cc1ccnc(C(N2CCCC2C2(NC(=O)C=CCN3CCCC3)CC2)=O)n1 66113,C12(C(C)NC(=O)C(C3(C)CC3)NC(=O)C=Cc3ccnn3C)CCC(CO1)C2 66114,N1(C(C(=O)NCC)=O)CCC(C)(C)C1C(=O)NC1CCC(C)(C)C1 66115,c1(NC(C2CN(C(c3n(C)c(S)nn3)=O)CC2F)=O)cccc2c1CCO2 66116,C1(C)(CNC(C(C2CCCCC2)C)=O)CCN(C(c2csc(F)c2)=O)CC1 66117,CCC(C(=O)NCC(C(=O)NC1CCC(=O)NC1C)N(C)C)C(C)(C)CC 66118,c1(C(=O)NCCC(Cc2cccs2)NC(CC=C(C)C)=O)ccc(C#N)cn1 66119,c1(C(=O)NC2(CNC(C3CCNC(=O)C3)=O)CC(OC)C2)n[nH]c2c1CSCC2 66120,c1(CN(CCNC(=O)CC2(C)CCC2)C(=O)NC2(SCC)CC2)cccc(Br)c1 66121,c1(C(N(CC(F)(F)F)C)=O)ccc2c(c1)B(O)OC2.C12CCCN(C1)C2=O 66122,N1(C(CCC#C)=O)CCC(CCCNC(c2cnc(O)n2C)=O)CC1 66123,CC1CN(C(c2cc(CNC(c3ccon3)=O)[nH]n2)=O)CCC1O 66124,C1(CNC(C=C=C(C)C)=O)CCCCCN1C(=O)COCc1ccccc1 66125,C1(C(=O)NCCCCN(C(c2cc(OCC)n[nH]2)=O)C)CCCC1S(C)(=O)=O 66126,N1(C(CCOC)=O)CC(NC(c2ccc(F)c(C(F)(F)F)c2)=O)CC2(CC2)C1 66127,C(C(F)C(=O)NCC(O)CCNC(C1(C#N)CCC1)=O)N(CC)CC 66128,C1(CC(=O)NCC2(CO)CCN(C(=O)CC3CC4(CC4)C3)C2)CC2C=CC1C2 66129,C(=O)(C(C)(C)COC)N1CC(C)(C(N(CCCCC=C)C)=O)C1 66130,C1(C(=O)NC(C)CNC(c2cncc(Cl)c2)=O)CCC2(CC1)CC2(F)F 66131,N1(C(C(c2cccc(C)c2)O)=O)CC2CC(C1)C2NC(C1CC1C)=O 66132,c1(C(N2CC(COC)(CNC(C3CCC=CCC3)=O)C2)=O)ncnc2ccsc12 66133,C1(C(=O)NCC2C(CNC(=O)C=Cc3ccncc3)C2)CCC2(CCC2)O1 66134,c1(NC(c2n[nH]cc2NC(c2ccnc(Cl)c2F)=O)=O)cc(Cl)cc(Cl)c1Cl 66135,C1(NC(=O)C=Cc2ccsc2)(CF)CCN(C(C2CCC(=O)N2)=O)C1 66136,N1(C(CC(C)CF)=O)C2CCC1CN(C(=O)Cc1cc3ccccc3o1)CC2 66137,C1(C(=O)NC2C=CC(CC(=O)N(C(CCC)C)CC)C2)C2CC3C(C2)C13 66138,N1(C(CC2CCN(C)C2=O)=O)C2CCC1C(F)C(NC(=O)CCn1ccnn1)C2 66139,CCC(CC(=O)N1CCCC(N2CC(C)(C)C2)C1)c1ccccc1 66140,N1(C(CCOCCC)=O)CC(CNC(=O)CNC(=O)C(C)CC)CC1C 66141,c1(CC(=O)NCCC2N(C(c3cc(C)ns3)=O)CCC2)ccccc1OC(F)F 66142,C1(CC(=O)NCc2c(C(=O)N(C(CC=C)(C)C)CC)cco2)OCCCC1(C)C 66143,C1(CC(=O)NCCCN(C(c2coc(C3CCCCC3)n2)=O)CC)COC(=O)N1 66144,C1(C(C)C)CN(C(C2CCC3(CCC3)C2)=O)CCN1C(c1cncs1)=O 66145,Cc1noc(N)c1C(N1CCC1CNC(=O)Cc1ccc(F)nc1)=O 66146,C(CC(C)C(=O)N1CCC(NC(=O)CC2CC(SC)C2)C1CC)=CC 66147,N1(C(=O)C=CC2CCCC2)CCCC2CN(C(=O)CC3CCCCC34CC4)CC12 66148,Cn1nc(C(=O)NC(CC(N)=O)c2cn(CC3CC4CC4C3)nn2)cc1F 66149,N1(Cc2ccc(C(=O)NCC(=O)O)cc2)C(=O)NC2(CCOC2)C1=O 66150,N1(C(CCC(=O)NC)=O)CCCC12CCN(C(=O)Cn1nc(C)c(Cl)c1C)CC2 66151,CC(C)(C)C(C#N)C(=O)NC1COCCC1NC(c1cnc(S)n1C1CC1)=O 66152,C1(CCC(=O)OC)CC(CO)N(C(=O)Cc2ccc(C(=O)O)cc2)C1 66153,C(=O)(C1=NOC(C)C1)NCCC1(C(=O)NC(c2nc(C)sc2)C)CCC1 66154,n1(CC(N2CCC(O)(C(C)NC(c3cocn3)=O)C2)=O)cnc2sccc2c1=O 66155,N1(C(C2C(c3cc(C)no3)C2)=O)CC(NC(=O)Cc2cccc(N)c2)C(C)(C)C1 66156,N1(C(c2c(O)ccc(CC)c2)=O)CC2CCC(C1)N2C(C1COCCC1(F)F)=O 66157,N1(C(Cc2c(C)ocn2)=O)CC2(CCN(C(=O)C(c3ccc(O)cc3)(C)C)C2)C1 66158,N1(C(c2ccc(F)cc2Cl)=O)CCCC2(CCN(C(=O)C(F)C3CC3)CC2)C1 66159,CC1COc2c(C(=O)N(CCCCN(C)C(C3C=CCCC3)=O)C)cccc21 66160,C1(C(=O)NCC(CO)NC(c2c(COC)nn[nH]2)=O)CC2C(C1)C2(F)F 66161,c1(C(N2CCCC2C2CC2NC(=O)CCc2csnn2)C)ccccc1Br 66162,C(N=c1[nH]c(C(C)(C)C)nc(=N)[nH]1)C1C(C)CCN(C(C2(Br)CC2)=O)C1 66163,CC#CCCCC(=O)N1CCC1C(=O)NCC1(OC)CC1 66164,N1(C(CNS(C)(=O)=O)=O)CC(NC(=O)C(c2cccc(F)n2)(F)F)C(SC)C1 66165,C1(OCC)CC2(C1)CC2C(=O)NCC(C)CN(C)C(c1sc(C2CC2)nc1C)=O 66166,c1(OC)ccc(CNC2CCN(Cc3ccccc3)CC2C)c([N+](=O)[O-])c1OC 66167,c1(NC(C2CCCC(c3nc(-c4cn(CC)nc4)on3)C2)=O)cncc(C#N)c1 66168,c1(C(=O)NC2(C3N(C(COCCOC)=O)CCCC3)CC2)cnn(C2CC2)c1C 66169,c1(NC(C2C3CN(C(Cc4c(C)noc4C)=O)C2C3)=O)cnc(C#N)nc1 66170,c1(C(CC)C)nc(C)cc(=NC2CC(NC(=O)CC3CC4CCC3C4)C2)[nH]1 66171,C1(N(C(C(C)N(C)C)=O)C)CCCN(C(c2cnn3c2CCC3)=O)CC1 66172,N1(C(C(n2ncc(C)c2)C)=O)CCN(C(c2cc3n(c2)CCC3)=O)C(CO)C1 66173,N1(C(C2(OC)CCC2)=O)C2CCC1CN(C(c1ccc(C)c(CO)c1)=O)C2 66174,Cc1[nH]nc2c1CC(C(N1CCC(F)(CNC(C3(CCCF)CC3)=O)C1)=O)CC2 66175,n1(CC(=O)N(c2ccccc2)CC=C)nnnc1N(C(=O)CCC1CCOC1)C 66176,C12(CNC(C3C(CNC(C(C)=CC(C)(C)C)=O)C3)=O)CC=CC(C1)OC2 66177,c1(CC(C(=O)N(CCCNC(C2C(OCC)C2)=O)CC)O)ccccc1Cl 66178,c1(CN2CCN(CC(CC)(C)Nc3ccc(F)cc3)CC2)ncc(Cl)cc1Cl 66179,C1(CNC(c2ccc(SC)s2)=O)CN(C(C2C(C)(C)C2(F)F)=O)CCC12CCC2 66180,CCCC(CC)CCC(=O)N1CCC(N(C)C(c2cc(N)ccc2O)=O)C1 66181,c1(C(=O)NC2C(C)N(C(c3cnc4sccn34)=O)CC2)ccc([N+](=O)[O-])s1 66182,CC1CC2CCC(C(=O)NCCC(C)NC(c3ncc(Cl)n3C)=O)CN2C1 66183,c1(OC(C)C)cc(CONC(c2csc(-c3ccc(O)cc3)n2)=O)ccc1F.NC 66184,c1(C(=O)OC)cnc2c(cnn2Cc2ncoc2-c2ccc3c(c2)OCO3)c1 66185,c1(C(N2C(CN(C)CC34CCC(CC3)C4)CCC2)=O)cnc2c(c1)N(C)CCO2 66186,N1(C(C(C2CCOC2)OCC)=O)C2CCC1CC(CNC(C1CC(F)(F)C1)=O)C2 66187,CC1CN(C(C2(C#N)CCCO2)=O)CC1CC(=O)NCC(C)S(N)(=O)=O 66188,CC1CCCC(NC(c2csc(-c3cccc(Cn4cccn4)c3)n2)=O)C1 66189,N1(C(CCSCCCC)=O)CCC(CO)C(NC(C2CCCCC2(C)C)=O)C1 66190,Cc1cnccc1C=CC(=O)N(CCCNC(c1cc(O)n(C)n1)=O)C(C)C 66191,Cc1cc(C(=O)NC2(C)CC(C(=O)NCc3ccc(C)o3)C2)nc(O)n1 66192,C(=O)(C1=C(C)CCC1)NC(C(N1CC(C(CC)C)C1)=O)C1CC1 66193,C1(NC(CCCOC)=O)CCC(NC(C23CC(CN2C2CC2)C3)=O)CC1 66194,C12(NC(=O)OCC)CCCN(Cc3cnc(C4(C)OCCO4)s3)CC1C2 66195,C1(NC(CSCCN(CC)CC)=O)CCN(C(c2cnnn2C)=O)C1C 66196,C1(C#N)(C(=O)NCC(CC)(CC)NC(=O)Cc2cc[nH]n2)CC2C=CC1C2 66197,C1(C(=O)NCCCCN(C)C(C23CCC(C)(CC2)C3)=O)CC12CCCOC2 66198,C1(C(=O)NC2C(CNC(C=NOC)=O)CC2)(CNC(=O)C(C)C)CCCCC1 66199,C1(NC(C2(CC#C)CCCC2)=O)CN(c2cc(COC)ncn2)CC2(CCC2)C1 66200,CN1CC(C(=O)NC2(CNC(C3CCOC3)=O)CC2)CC1=O 66201,C1(CCCNC(C(C)c2ccco2)=O)CCCCN1C(=O)CSc1nncs1 66202,N1(C(c2nc(CC)sc2)=O)CCC2CCN(C(C3(C)CCOC3)=O)CC12 66203,C#Cc1cccc(C(=O)NC(CNC(=O)Cc2ccc(C)nc2)CCCC)c1F 66204,c1(C(=O)NC(CN(C(=O)C(C2CCOCC2)O)CC)C)ccc(Cl)s1.C 66205,c1(C(=O)NC2CC(F)(CNC(C)=O)C2)cnc(C(F)(F)F)c(F)c1 66206,C1(N(C(C(Br)=C(C)C)=O)C)CN(C(c2cncc(N)n2)=O)CC1(C)C 66207,c1(C(c2n(CC)nnn2)NCc2ccc(C)cc2OC)cc(F)c(F)c(OC)c1F 66208,CC#CCCC(=O)NC(C)(CNC(=O)CSCC1CCCO1)C(C)C 66209,C(=O)(CC(O)CC(C)(C)C)N(CCC(N1CC(C#C)OCC1)=O)CCO 66210,CCC(O)C(F)(F)C(=O)NCC(CCNC(C1(n2nccn2)CC1)=O)OC 66211,C1(NC(c2cc(C(=O)OCC)no2)=O)CCCC(N(C)C(c2[nH]cnc2CC)=O)C1 66212,N(C(=NCCCN(c1sccc1C)C)N1CCCC(Nc2ccccc2)C1)CC 66213,CCCC(C)(CC)C(=O)NC1CCC(NC(=O)C(C2CC2)SC)CC1 66214,CN(C#N)C(=O)C(=O)NC(C)(CNC(=O)Cc1cc(O)nnc1O)CO 66215,C1(CNC(CC(CC)NC(c2cnc(=N)[nH]c2)=O)=O)OC(=O)CC1(C)C 66216,C1(NC(=O)NCC(C(C)C)c2cnn(C)c2)CC2(C1)CC21CCC1 66217,C(C(O)C(F)F)NC(CCNC(c1cncnc1)=O)=O 66218,c1(C(=O)NC2CCN(C(c3c(C)c[nH]n3)=O)C2(C)C)ccc(Br)c(F)c1F 66219,c1(C(N(CC(C)NC(c2cc(C)cc(C)c2)=O)C)=O)cc2c(Cl)cncc2o1 66220,c1(C(=O)NC(CNC(C(CC)=CC)=O)C)ccccc1C1CC1(F)F 66221,C1(O)(C(=O)NCC(C(N2CCC(N(C)CC)C2)=O)N(C)C)CC(C)(C)C1 66222,CC1CC(C)(C(N2CC(O)(CNC(=O)CCn3ccccc3=O)C2)=O)CC(C)O1 66223,c1(C(N(C2CCN(C(C(CCC)C)=O)CC2)C)=O)ccc2nc(C)n(C)c2c1 66224,C(=O)(CCCCC(=O)NC(CNc1nn2cc(C)nc2s1)C1CC1)NC 66225,N1(C(C(C)OC)=O)CCC(F)(CNC(=O)Cc2cncc(C#N)c2)CC1 66226,CCC(C)C(O)C(=O)NCCC(C(C)C)NC(C1CCOC1)=O 66227,C(=O)(C1=CCCOC1)NC(C)C(CO)NC(C1(Cc2cccc(Cl)c2)CCC1)=O 66228,C1(NC(CC2(C=C)CN(C(=O)CC(=O)N(C)C)C2)=O)COC2(CCC2)C1 66229,n1(C(C)C)ccc(CC(=O)NC2CCC2NC(=O)CC(C)C2CC2)n1 66230,c1(C(N2CC(CN(C(CCCC)=O)C)OCC2)=O)cc([N+](=O)[O-])oc1C 66231,c1(OC)c(C(=O)N(C2CCCCN(C(=O)Cn3nnc(=N)[nH]3)C2)C)ccnc1F 66232,N1(C(c2cccc(C(C)=O)c2)=O)CCN(C(=O)C(c2ccccc2)C)C(CO)C1 66233,Cc1c(NCC(C)(C)C)cccc1C(=O)NC1(O)CCN(C(=O)CCF)C1 66234,C1(CNC(C2CC(N(C(c3cc(C(=O)OC)no3)=O)C)C2)=O)CCCC12CCC2 66235,N1(C(CC(C)C)=O)CC(C(=O)NC(C)Cc2cn[nH]c2)OC(C)C1 66236,c1(OCC(=O)NCC2CC(C)CN(C(C3(N(C)C)CC3)=O)C2)cc(F)ccc1F 66237,C1(CNC(C(C)OC)=O)CCCCCN1C(c1nc(C)ncc1Br)=O 66238,CCC(C)C(O)C(C)C(=O)NCCC1CCN(C(=O)CCC(=O)N(C)C(C)C)C1 66239,C(=O)(C(F)(F)C(O)C(C)C)NCC1C(NC(C2CN(C(C)=O)C2)=O)CCC1 66240,C1(CCOC)(NC(C2CCCCC2O)=O)CCN(C(=O)CNc2nccs2)CC1 66241,c1(N2C(CNC(C(c3cnn(C)c3)OC)=O)CCC2)ncc(C#N)cc1Cl 66242,C(=O)(C1=CCOCC1)NC(C)CN(C)C(c1cc(Br)c(C2CC2)s1)=O 66243,C1(NC(C(CC)=CC)=O)CCCN(C(C2CC23CCCC3)=O)CC1 66244,C1(c2n(CCCC)nnn2)(NCC2(c3cccs3)CCCC2)CCOC(C)C1 66245,CCC(CCCC(=O)NCc1cnn2ccccc12)NC(=O)CSC 66246,CN1CC2CCN(C(=O)C(=O)NCCCN3CCN(C(C)(C)C)CC3)C2C1 66247,C(=O)(C(CC(N)=O)NC(=O)CC(C)CN(C)C)NC(COC)C(C)C 66248,C1(=O)N=C2C=C(N(C)N2)C(=O)NCC12CCC2.C(C(=O)NCC=C(C)C)(OC)OC 66249,C1(C(=O)NC(c2cn(-c3c(C)ccc(C)c3)nn2)C)CCc2nc(C)sc2C1 66250,c1(C(=O)NC2C(NC(=O)CC3C=CCCC3)CCC2)ccc2c(c1)CC(=O)NC2 66251,Cc1cc(C(=O)NC2CCC2CNC(c2cncc(NC(C)C)c2)=O)ccn1 66252,CCCCCC(=O)NC1CCC(NC(=O)CC(CC)c2ccccc2)C1 66253,CCCCCCC(F)C(=O)NCC(C)(C(C)C)NC(c1cc2ncccn2n1)=O 66254,C1(C(=O)NCCC(CC)(C)OC)CNC(=O)CN1C(=O)COCC(=O)OC 66255,Cc1ccc(CC(N2CCCC(N(C(=O)C(C)CO)C)CC2)=O)c(C)c1 66256,Cc1cccc2[nH]cc(C(N3CCCC(N(C(=O)C4=CCSC4)C)CC3)=O)c12 66257,C(C(N=c1ccc2ncc[nH]c-2n1)C(C)C(C)C)NC(COC(CC)C)=O 66258,C(C(C)(C)C(=O)N1CCC(C)(CNC(C2(c3cnn(C)c3)CCCO2)=O)C1)OC 66259,c1(C(N2CC(CNC(C3CC(CCC)OCC3)=O)C2)=O)cnc(Cl)c(Cl)c1 66260,CC1(C)CC(=O)c2cc(OCCNC(N3CCOCC3C3(C)CC3)=O)ccc2O1 66261,c1(OC)cc(C(=O)NCC(C)NC(=O)Cn2ccc(C)n2)[nH]n1 66262,c1(C(=O)NC(C2CCCN2C(c2ccc(F)cn2)=O)C(C)C)cn(C)ccc1=O 66263,C(=O)(C(CC)C(=O)NCC1C(C(N2CC(C)(CC)C2)=O)CCN1C)OCC 66264,Cc1ccc(C)c(OCC(=O)N(CC(C)NC(=O)C(C(C)(C)C)C2CCC2)C)c1 66265,c1(C(=O)NC2CCN(C(c3cncc(NC)c3)=O)CC2O)ccc2c(c1)COC2 66266,C1(NC(C(C)OCCOCC)=O)CC(OC)CN(C(=O)Cc2ccsn2)C1 66267,CCCCC(F)C(=O)NC1CCC(C)(CNC(c2cnoc2C)=O)C1 66268,c1(CC)nn(C)c(Cl)c1C(=O)NCCCC1(NC(c2cnc(O)c(F)c2)=O)CC1 66269,N1(C(C2C(C)(C)COC2)=O)CCOC2(CCN(C(=O)CCc3cnoc3)C2)C1 66270,C1(N(C(CCC(=O)OC)=O)CCC(=O)N2CC(F)C2)C2CCC1CNC2 66271,c1(SC)cc(Br)ccc1C(=O)NC1CC(C)(NC(=O)C2=CCCCC2)C1 66272,c1(N(C)C)cccc(CCC(=O)NCC2CCCN2C(=O)C(F)C2CCOC2)c1 66273,N1(C(c2cccc(OC)c2OC)=O)CC2C3CCC(C2C1)N(C(C)C)C3 66274,N1(C(c2ncc(F)cn2)=O)CC2(CCCN(C(c3ccnc4c3CCC4)=O)C2)C1 66275,C1(NC(NCCS(CC)(=O)=O)=NCCCCl)Cc2n[nH]cc2C(C(F)(F)F)C1 66276,c1(C(=O)NC(c2c(C)cccc2)CF)cc2ccc(Br)cc2[nH]1 66277,c1(C(=O)Nc2c(C)noc2C(C)C)coc2c1CN(C(C1(C#N)CCCO1)=O)C2 66278,CCC(C)(C#N)C(=O)N(C)CCNC(=O)C(C)O 66279,C1(NC(CCOCCN(C(C2CC(C)(CC)C2)=O)C)=O)CCc2nncn2C1 66280,N1(C(Cc2c(C)occ2)=O)CC(CNC(c2ccsc2C#N)=O)CC1C 66281,C1(CNC(c2c(CC)nn(C)c2)=O)CCN(C(c2cc(O)cs2)=O)C1(C)C 66282,Cc1cn(C)nc1C(=O)NCC1CN(C(c2cc(CO)on2)=O)CC1C(F)(F)F 66283,C1(NC(CC=CC(C)(C)C)=O)COC2CN(C(C3CC(C)(C)CO3)=O)CC12 66284,Cc1cc(F)c2ncc(C(N3CCC(NC(=O)CC(C)O)C34CC4)=O)cc2c1 66285,C1(F)(CNC(C23CC(C)C2C3)=O)CCCN(C(C2(S(C)(=O)=O)CCC2)=O)C1 66286,C1(n2cc(CC(N(OC)C)=O)nn2)CON(C(=O)C2CCC(=O)CC2C)C1 66287,C1(C(=O)OCCC2OCCC(C)(C)C2)CC12CCc1ccccc12 66288,c1(N(C)C)ccc(C(N2CCC(NC(C3(C)CS(=O)(=O)C3)=O)C(F)C2)=O)cc1F 66289,c1(CN2CCCC(C)(C(=O)NC=Cc3ccccc3)C2)ccc2c(c1)CNC2=O 66290,C1(CCOC)CN(C(=O)CC2CCCC(C)(C)C2)CCN1C(c1cc(F)n[nH]1)=O 66291,c1(C(=O)NCC(CN(C(C(c2ccc(CC)cc2)C)=O)C)C)cc(C)cc(Cl)c1 66292,C1(C2N(C(C3N(C)CCCC3)=O)CCOC2)CN(C2CCc3ccc(Cl)cc32)C1 66293,c1(C(=O)NCCCCNC(CCCC(CCC)C)=O)sc2nccc(C)c2c1C 66294,N1(C(c2ccn(CCOC)n2)=O)CCC2(CCN(C(=O)Cn3ccc(C)n3)C2)C1 66295,c1(C(N(C(c2ccccc2)CNC(C2CC2F)=O)C)=O)cccn2nccc12 66296,C12(NC(c3c(C)nsc3)=O)CCCC(NC(=O)C3=COCC3)(C1)C2 66297,c1(CNC(C(C)n2ccnc2)=O)ccoc1C(N1CC(N2CCC2)C1)=O 66298,N1(C(CC2CC(CC)C2)=O)CC2C(CC(N3CCCC(C(C)(C)O)C3)=O)C2C1 66299,c1(C(=O)NCCC(CNC(CCC2C(C)=NNC2=O)=O)O)cn(C)c(C)cc1=O 66300,c1(OC)ccc(C(N)=O)cc1.C1C(C)(C)CN(C2CC2)CC2C(C2)NC(=O)CS1 66301,S(=O)(=O)(c1nc(N2CCC(C)(C)CC2)ccc1Br)NCCCSC 66302,N1(C(C2(C#N)C(C)C2)=O)CC=C(C(=O)NCc2cocn2)C1 66303,N#Cc1ccc(C=CC(=O)NCc2nc(CNC(=O)CC3CC(F)C3)cs2)cc1 66304,c1(CCC(N2CCN(C(C3C(=C)C3)=O)CC2C)=O)cccc2oc(C)nc12 66305,N1(C(Cc2cnc(C)s2)=O)CCCC(O)(CCNC(C2(C)CSC2)=O)C1 66306,CCC(C(=O)N1CC(O)(COC)C1)N(C(=O)C(C)C1(O)CCC1)C 66307,N1(C(CCNC(C2C(C)C2)=O)=O)CC(O)(C(F)C(=O)N(C)Cc2ncccn2)C1 66308,CCC(CC)C(C)C(=O)N1CCC(CNC(c2cccn2C(C)C)=O)C1 66309,c1(NCc2ncnn2C)nc2ccccc2nc1CC1CCN(C(=O)NC)CC1 66310,c1(-n2cc(C34CN(C3)C4=O)nn2)c(F)cc(Cl)cc1F.CN(C)C1CC1 66311,C(c1ccsc1)=CC(=O)NCCN(CCOC)C(c1nscc1C)=O 66312,C(N=c1[nH]c(=NC(C)c2ccc(F)c(F)c2)[nH]c2ccccc12)C1CC(SC)C1 66313,C(=O)(C(F)C(C)(F)F)NC(CCOC)C(=O)Nn1cc(-c2nc(O)ccc2C)nn1 66314,CC1COc2c(NC(N3CCc4cc(Br)ccc43)=O)cnn2C1 66315,N1(C(CC=CC=C)=O)CC2CCN(C(C3CC(=O)N(O)C3)=O)CC(C2)C1 66316,CC(C(=O)NCC1(CNC(c2cc(N)c(F)c(F)c2F)=O)CC1)C(C)C(C)(C)C 66317,c1(-n2c(C(=O)NCc3ccccc3Cn3cncn3)ccn2)ccc(F)cc1 66318,n1(CC)nccc1C=CC(=O)NCC(C)(C)CNC(c1cc(=O)cc[nH]1)=O 66319,C(CCSC)(C(=O)N1CC(N(CCO)C(c2cc(-c3ccoc3)[nH]n2)=O)C1)OC 66320,C1(CC(=O)NCC2C(CC(N3C(COC)CC3)=O)C2)CCOC1=O 66321,c1(CCC(=O)N(CC(C)N(C(C(C)O)=O)C)C)ccc(Cl)cc1Cl 66322,CCC(C)(C)C(O)C(=O)N(CCNC(C1CCC2(CCC2)C1)=O)CC1CC1 66323,N1(C(CCCCC)=O)CCc2c(ncn2C)C12CCN(C(=O)CC(C)COC)C2 66324,C1(CC(=O)NCCCN(C(=O)CCC2CCCO2)C(C)C)CCCOCC1 66325,c1(C(=O)OC)cc2c([nH]1)CCN(C(=O)C(c1ccc(N)cc1)(C1CC1)OC)C2 66326,C1(NC(=O)CCC2CCOC2)CCSC12CN(C(=O)C=Cc1cncnc1O)C2 66327,C12(C(=O)NC(c3n(CC)ccn3)C)CC(CN1C(c1cc(O)cs1)=O)C2 66328,C1(C(CNC(C(C)N2CCC2)=O)(C)C)CCCCN1C(c1cn(C)c(O)n1)=O 66329,N1(C(C)C)CC(C(=O)N(CCCNC(=O)C(C)(C)n2cncn2)C)CC1=O 66330,C(C(C(C)(C)C)NC(=O)CC1CCOC1)NC(CC(=O)NCC#C)=O 66331,C1(C(=O)NCCCOCCNC(CC2CC(SC)C2)=O)CC2(CCC2)C1 66332,C(=O)(C(C(C)C)N1CCCS1(=O)=O)N(CC(CC)NC(C1(O)CC(CF)C1)=O)C 66333,c1(C(=O)NCC(CNC(C2(OC)CCCOC2)=O)O)ccc2c(n1)NCC2 66334,CC1CCc2n[nH]cc2C1C(=O)NC1CCN(C(=O)CN=S(C)(C)=O)C1(C)C 66335,N1(C(CCCC)=O)CCC(NC(=O)Cc2ccon2)C1C(C)(C)C 66336,Cc1ccc(-n2ccnc2)c(C(=O)N(C2CCC3CNCC23)C)c1 66337,c1(SC)ccc(C(=O)NC(CNC(=O)CNC(=O)C(F)(F)F)C(C)C)cc1C#N 66338,C1(C(C)Nc2ncc(F)cn2)CCCCN1C(=O)C(C)Cn1ccnc1 66339,c1(CNC(=O)NCCCCNC)nccc2ccccc12 66340,C1(C)(CC)CCN(C(c2cc(CNC(C3CN(C(=O)NC)C3)=O)cs2)=O)C1 66341,CC1C(NC(=O)C=Cc2ccnn2C)C(C)CCN1C(c1cnn(C)c1N)=O 66342,N1(C(CCC#CC)=O)CCCCC1C1CCCN1C(=O)CC1(OC)CCC1 66343,C#CCC(CC(F)F)C(=O)NCC1(C(=O)NOCC(F)F)CC2(CC2)C1 66344,C1(CC(=O)NCCC2CN(C(=O)C3CC3)C2)SC2=NCCN2C1=O 66345,C1(C(N2CC(C)(C)C(Nc3ncnc4sccc34)C2)=O)CCCC(F)(F)CC1 66346,N(C1CCCc2ccnc(Cl)c21)C(=O)C(=O)NC(C1CCOCC1)C1CCCCC1 66347,C1(C(=O)NCc2n(CCC)ncn2)CC(N=[N+]=[N-])CN1C(=O)C(C)C1CCCC1 66348,C12(C(=O)NCC(CNC(C3N(C(C)=O)CSC3)=O)O)CCN(CC1)CC2 66349,CC1CCC(C)(C(=O)NCC2(C)CCN(C(=O)Cn3cncn3)C2)C1 66350,c1(-c2ncc(C)o2)cccc(C(N2CCSCC2CCNC(=O)CN(C)C)=O)c1 66351,C(C)(C(CC(=O)NCC1(C)CC(C)(C)C1)NC(=O)C(C)C(F)(F)F)OC 66352,CC1CN(C(c2ccc(Br)o2)=O)CC1NC(c1cn(C(C)(C)C)nn1)=O 66353,C12CC3CCC(C1)N3CC(=O)NC2.C1(c2c(C)cccc2)OC(=O)NC1(C)C 66354,N1(C(C(COC)COC)=O)CC(NC(=O)CCC(C)(C)OC)CC12CCCOC2 66355,N1(C(c2n(CC=C)ccc2)=O)CC(O)CC1CNC(=O)C(=O)NCCNC(C)=O 66356,c1(CC(=O)NC(CNC(Cc2ccn(CC)n2)=O)C2CC2)ccccc1Br 66357,C12(CNC(CC(CC)(F)F)=O)COCCN1CCN(C(C1(C)CC(F)(F)C1)=O)C2 66358,N1(C(C(=O)NCC(F)F)=O)CCC(C(N2CCC(n3ccnn3)C2)=O)(CF)C1 66359,c1(OCC)cc2ccccc2cc1C(N1CCC(N(C)C(C2C=C2C)=O)CC1)=O 66360,Cc1n[nH]c2cnc(C(=O)NC3CC(CNC(=O)C=C4CCN(C)CC4)C3)cc12 66361,N1(C=O)CCC(NC(CSN(C2CC(C#N)C2)N(C)CC)=O)C1.c1(C=O)cscn1 66362,c1(C(N(CC(C)NC(C2(CC#C)CC2)=O)C)=O)cnc2c(cnn2C)c1N 66363,c1(C(N(C2CCC(NC(c3onc(CC)c3C)=O)C2)C)=O)cncc2c1CCC2 66364,C1(NC(C(CC)Oc2cccc(F)c2)=O)CCN(C(C2(C)C=CCC2)=O)CC1C 66365,C1(CC)C(NC(=O)CCN(S(C)(=O)=O)C)CCCN1C(=O)C(C)CC(N)=O 66366,N1(Cc2ccc(OC)nc2C)CCC(=O)N(CC2(n3cncn3)CC2)C1=O 66367,N1(C(c2ccc(OC3CC3)cc2)C(=O)NCC)CCN(CCOC(C)=O)C(C)C1 66368,c1(CC)ncccc1C(=O)N(C)CC1CCCN1C(=O)CCC1CCCCCC1 66369,C1(C)(C(N(CCCCNC(=O)CCc2ccncc2)C)=O)COC(=O)OC1 66370,CCCCCC(O)CC(=O)NC(CNC(C1(CC)CC(F)(F)C1)=O)(CC)CC 66371,C1(NC(c2cc(Cl)sc2Cl)=O)CCC2CCN(C(c3cnc(Cl)cc3Cl)=O)C1C2 66372,CCCCCCN(CC(=O)NC1CC(C(F)F)(CNC(=O)CC23CC(C2)C3)C1)C 66373,c1(C(N(CCCN(C(C2CC(SC)C2)=O)C)C)=O)c[nH]c2cccc(F)c12 66374,C1(N(C(C2(CCC=C)CC2)=O)C)CCCCC1N(C)C(c1ccccc1Cl)=O 66375,CCC(=O)CCC(=O)N1C(CC(=O)NC(C2CCOC2)CC)C2CCCC12 66376,N1(C(C(C(C)C)SC)=O)CC2CCCC(C1)N2c1nccc(CO)n1 66377,c1(C(C(C)NC(c2cscn2)=O)N)ccccc1 66378,N1(C(c2cnc(Cl)[nH]2)=O)CCCC(NC(C2CCC(Nc3nccs3)C2)=O)C1 66379,N1(C(CC2(C)CC2(Cl)Cl)=O)CC(NC(c2ccnc(OC(F)F)c2)=O)CC1CO 66380,C1(N(C(CCNC(COC)=O)=O)C)CN(C(c2ccc(C#N)[nH]2)=O)CC12CC2 66381,c1(-c2cc(C(N(CCCC)CCCC)=O)ncc2)ccc2oc(O)nc2c1 66382,C(=O)(C(O)C(F)(F)F)N1C(CN(C(C2CC23CC3)=O)CC2CCOCC2)CCC1 66383,C12(CNC(=O)C3=NOC(CC4(O)COC4)C3)CCCC1CCN2C(c1cnsn1)=O 66384,N(C(=S)N1CCC(C2CCC2)CC1)C1C(C)CCCC1 66385,c1(C(=O)NCC(CC)NC(c2cnn(C)n2)=O)cnc(SC)cn1 66386,Cc1cccc(C)c1SCC(N1CCCC(N2CC(F)(F)C2)C1)=O 66387,C(CC(C)C(=O)NC(C)CCCNC(=O)C=Cc1csc(C)n1)=CC 66388,N1(C(c2c(Cl)cn(CC)n2)=O)CCCC(CCNC(=O)CN2CC(C)(C)C2)CC1 66389,C1(CC(=O)NC(CC)CNC(C2(c3cc[nH]n3)CCC2)=O)CC(C)(C)CO1 66390,CC1CN(C(=O)C=CCF)CCC1NC(c1nn(C)nc1Br)=O 66391,c1(C(=O)NCC(COCC#C)OC)cc(C)cc(OC)c1OCC(=O)OCC 66392,Cc1cc(C(=O)NC2CSC(C)C2)nc(N(C)C)n1 66393,N1(C(C(CC)C)=O)Cc2ccccc2C(NC(c2cc(C)c(C)[nH]2)=O)C1 66394,c1(C(N(CCCNC(=O)C2=COCC2)CCO)=O)ccc2nn[nH]c2c1 66395,N1(C(CC=CCCCCC)=O)CCCC1C=CC(=O)NCCc1nnc(C)o1 66396,CC(C)S(=O)(=O)CCCNC1CCCC1CNC(=O)C=CI 66397,C1(NC(C2(C(C)NC(c3cnc(S)nc3)=O)CC2)=O)CCN(C)CC1C#N 66398,c1(C(=O)NC2CCN(C(C(C3CCOC3)OCC)=O)C2)scc(C)c1OC 66399,C1(NC(C(c2ccncc2)C)=O)CCC2CC1CN2C(C1CCCNS1(=O)=O)=O 66400,n1(CC(N2CC(SC)C(NC(C3(C)CCCO3)=O)C2)=O)cnc([N+](=O)[O-])c1 66401,CC1(C)CCCCC1C(=O)NCC1CC(NC(C2CCC23CCC3)=O)C1 66402,N1(C(=O)NCCCc2scc(C)n2)CC=CCC1C(F)(F)F 66403,Cc1[nH]nc(C(=O)N(C)CCOCCN(C)C(C2CC23CCOC3)=O)c1Cl 66404,C1(F)(CNC(C(C)SC)=O)CCN(C(=O)C(C)(O)C2CC2)CC1 66405,C(=O)(C(C)(C)CCC#N)NC(C1CCCN(C(c2[nH]ccc2C2CC2)=O)C1)C 66406,N(C1CCc2ccccc21)C(C1N(C(CNC(=O)OCC)=O)CC(O)C1)=O 66407,c1(C(N2CC(OCCC(=O)NCCOCC(F)F)C2)=O)nc2cc(F)ccc2s1 66408,N1(C(C(C(C)C)SC)=O)CC2(C1)CN(C(C1CCC(=O)NC1)=O)CC2CO 66409,C1(C(N(C)CCN(C)C(C2COCCC2(F)F)=O)=O)CCn2cncc2C1 66410,Cc1cccc(C(F)C(=O)NCC(C)N(C(=O)CN2CC3CC3C2)C)c1 66411,Cn1ncc2c(NCC3C4CN(C(c5cnnc(Cl)c5)=O)CC34)ncnc12 66412,c1(C(=O)NC(C)CSC)cccnc1OC1CCN(C(=O)OC)C1.C(CO)O 66413,Cc1ccc(C(=O)NCCCN(C(C2CCS2(=O)=O)=O)C2CC2)cc1 66414,N1(C(c2c(C)noc2C)=O)C2CCC(C(=O)NCCC3CCCCC3)C1CC2 66415,C(=O)(CCN=c1cc[nH]c2ccccc12)NCC(=C)c1ccccc1 66416,N1(CC)N=C(C(=O)NCC(C)NC(c2cc(C)nc(N(C)C)n2)=O)CCC1=O 66417,c1(C(N2CC(NC(C3CN(C(N)=O)C3)=O)(CO)C2)=O)cc2ccc(Cl)cc2c(O)n1 66418,C(=O)(C(CC(C)C)NC(=O)CC(COC)NC(N)=O)N1CC(C(CC)C)C1 66419,c1(C(=O)NCCCN(CC)CC2CC2C)cc(-c2ccns2)on1 66420,CCCCC(C)(F)C(=O)NC(C)CCCC(=O)NCc1cnc(CC)s1 66421,c1(NC(C(CCNC(=O)C=Cc2cocn2)OC)=O)ccc2n[nH]cc2c1 66422,c1(CC(=O)NCC(C)CN(C(=O)C(C)(C)C2CCCC2)C)ccn(C(F)F)n1 66423,N1(C(c2sc(C(F)F)nc2Br)C(=O)NC)CC(O)C(O)C1CF 66424,N1(C(C(CC)(C)O)=O)CCCCC(CNC(=O)CCc2csc(=N)[nH]2)C1 66425,N1(C(C(=O)NCCOC)=O)CCN(C(=O)CNC2CCN(C)CC2)CC(O)C1 66426,Cn1cccc(C(=O)NCC(=O)NCC(N2CCC(F)(CO)C2)=O)c1=O 66427,C#Cc1cccc(CC(=O)NC(CCC=C)C(=O)NC(CCF)C(=O)OC)c1 66428,Cc1ccccc1-n1nc(C(C)O)nc1CCc1nc(C2CC2)n[nH]1 66429,c1(C(C(=O)NCCC)N(C(C)CC(C)C)C)ccc2c(c1)C(=O)NCC2 66430,C(=O)(C1=NOC2COCC12)N1CCN(C(c2c(C)oc(C)c2C)=O)CC1CCO 66431,N1(C(CCC=CCC=C)=O)C(CNC(=O)C(CC2CCC2)SC)CC2CCCC12 66432,c1(C(N(CC(CN(C(C2(CC(C)C)CCC2)=O)C)O)C)=O)ccc(Cl)nn1 66433,C(=O)(CCC(C)(C)N(C)C)NCCC1(C(=O)NC2C(C)N(C)CC2)CCC1 66434,c1(C(N(C(CCNC(c2cc(C(C)C)[nH]n2)=O)C)C)=O)cc2cccn2c(O)n1 66435,C1(CNC(Cc2ccn(CC(C)C)n2)=O)CCN(C(=O)COCCCF)C1(C)C 66436,CCC(C)C(C)(O)CNC(=O)C(C)(CNC(=O)Cc1cc[nH]c1)CC 66437,N1(C(C(CC(C)C)Cc2ccccc2)=O)CCCC2CN(C(C3(C)CC3)=O)CC12 66438,C(=O)(C1=C(C(F)Cl)N(C2CCC2)C(=S)NC1c1ccc(F)c(C#N)c1)OCC 66439,c1(-c2ccccc2)nccc(C(=O)NC2C(NC(CCOC)=O)CCC2)n1 66440,c1(C(=O)NC(C2CN(C(C3(C)CCCCO3)=O)C2)C)ccc(F)c(F)c1F 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66583,C1(C)(CC)CCN(C(C2CCCCC2(C)NC(=O)CN=[N+]=[N-])=O)CC1 66584,C1(C(=O)NCCNC(c2c(C)occ2)=O)CN(C)CC1c1ccccc1 66585,C1(CNC(CC2CCCC(C)C2)=O)CC(C)(C)CN1C(=O)CC1C=CCC1 66586,N1(C(C(C=C)O)=O)CCN(C)CC1C(=O)NCCC12CC(CO1)C2 66587,c1(OCC(N2Cc3nnsc3C2)=O)cc(Br)cc(F)c1F 66588,C(=O)(CC(C(F)(F)F)c1ccon1)NCCCNC(C1=NOC(C)C1)=O 66589,c1(CC)[nH]c(C(=O)NC2C3CC2N(C(=O)CNC(=O)C(C)(C)C)C3)nc1Cl 66590,c1(C(=O)NCc2c(C(N3CC(C)C(F)C3)=O)cco2)ccc2c(c1)CC2 66591,CC1CCOC(C(=O)N(C(C(=O)N2CC(n3ccnn3)C2)C2CC2)C)C1 66592,C1(CNC(C2C(C)CC2)=O)CCC(F)(CNC(=O)CC2CC3(CCC3)C2)CC1 66593,C1(CNC(CC(CC)C)=O)CC2(CCN(c3nc(Cl)ncc3C(C)C)CC2)CO1 66594,c1(C(=O)NC(c2ccccc2)C(C)NC(CCSC)=O)cc2scc(C)c2[nH]1 66595,c1(CC)nccnc1C(=O)NC1C=CCN(C(=O)CC2(C)CCCCC2)C1 66596,C(=O)(C(C)CCCC(C)C)NCC(CC=C)NC(C1CC(=O)NC(=O)N1)=O 66597,CC(C)CS(=O)(=O)N1CC=CC1C(=O)NCCC1CCCN1C 66598,N1(C(c2cccc(NC(C)=O)c2)=O)C2CCC1CN(C(=O)C1=CC(C)(C)C1)CC2 66599,O=C(NNC(=O)C1CCCC1O)NCCN1CCCCCC1 66600,C12(CN(C(C)C)C(=O)Nc3ccc(C4COC(=O)N4C)cc3)CCC(CC1)OC2 66601,C1(NC(C(CCC)O)=O)CCCCCN(C(=O)C(=Cc2ccccc2)OC)C1 66602,Cc1ccc(C)c(C(=O)NCC2(C(=O)NC(CO)C3(O)CC3)CC2)c1 66603,C1(CNC(CC(C(C)C)C)=O)COC(C)(C)CN1C(c1cc(O)cc(O)n1)=O 66604,C1(C(=O)NCC(=O)OCCCC)CCC(C)(C)N(C(=O)CCOC)C1 66605,Cc1ccn(CC(C)(O)C(=O)NCC(O)CNC(c2ccc(C#N)[nH]2)=O)c(=O)c1 66606,c1(CC)cc(C(N2CCCC2CC)C(=O)Nc2ccc(F)cc2)cc(F)c1 66607,S(=O)(=O)(c1cc(C)c(Br)cc1C)NS(CC1CC2(CC(OCC)(OC)C2)C1)(=O)=O 66608,C#Cc1cnn(C)c1C(N1CCCC(C(=O)NCCC(O)CCC)CC1)=O 66609,C1(C)(CC)CC(NC(C23CC2CN(C(C2CC=CC2)=O)C3)=O)CCO1 66610,c1(C(=O)NCCN(C(C2CC(n3cnnc3)C2)=O)CC2CC2)sccc1C(F)F 66611,N1(C(=O)CSC(F)(F)F)CCN(C(C2(CCF)CC2)=O)CC(O)C1 66612,C1(NC(c2c(OC)n[nH]c2)=O)CN(C(c2cnc(C)[nH]2)=O)CC1O 66613,C1(C(=O)NC(CNC(=O)C(F)(F)c2cnccn2)C2CC2)CCc2nc[nH]c2C1 66614,C1(OCC)CC(CCC(=O)N(C(C)CNC(=O)COCCC(C)C)C)C1 66615,N1(C(CSC)=O)CCCC(CN(C(=O)Cc2ccc(OC(F)(F)F)cc2)C)C1 66616,C1(NC(C2CN(C)C(=O)CC2)=O)CCN(C(=O)CCc2cnc[nH]2)CC12CCC2 66617,C1(NC(c2ccnc(Cl)c2)=O)CN(C(=O)Cc2cccnc2)CC1(F)F 66618,c1(OC)ccc(CO)cc1-c1ccc(C(=O)NCC2(C(=O)O)CCC2)o1 66619,CCCCC(C)N(C(=O)C(C)CN(C(=O)Cc1ccn(C)c1)C)C 66620,c1(C(=O)NC2CCN(Cc3cncc(Cl)c3)CC2F)ccc2ncsc2c1 66621,N1(C(C2CC2C(F)F)=O)CCC(F)(CNC(C2CCC(n3ccnn3)CC2)=O)C1 66622,Cc1cc(Cl)ccc1CC(=O)NCC1COCCN1C(c1cn(C)cc1C)=O 66623,C1(NC(CN(C(c2n(CC#C)ccc2)=O)C2CC2)=O)CN(C)NC1=O 66624,Cc1c(C(=O)NC2CCC(c3cn(CC(C)(C)C)nn3)CC2)cccc1C1CC1 66625,Cn1cc(C(N2CCC(C)(CNC(c3nsnc3O)=O)C2)=O)ncc1=O 66626,N1(C(C2(NC(C3C(C)(C(F)F)C3)=O)CCSC2)=O)CC2(CO)CCC1CC2 66627,C(=O)(C(CC)C(C)C)NC1C(NC(CSCC#C)=O)CCCC1 66628,CC1(C)CCCCC(C(=O)NC2CCCN(C(c3ccc(Br)cc3)=O)C2)C1 66629,C1(C(N2CCCC2c2cccs2)=O)CCCC2CC12 66630,Cc1cc(C(N2CCOC(CNC(C3CCN(C)C3C)=O)C2)=O)c(C)n1C(C)C 66631,C(=O)(CCCCN=[N+]=[N-])N1CC(C(N2CCC(OCC)C2)=O)OC(C)C1 66632,N1(C(C2(C)CCC(C)C2)=O)CC(C(=O)NC(C)(C)C(F)F)C2(CCC2)C1 66633,C1(S(C)(=O)=O)(C(=O)NCC2CCN(C(CC=C(C)C)=O)CC2O)CCOCC1 66634,Cc1cnc(O)c(CNC(C2COCCN(C(C3(C#N)CC(F)(F)C3)=O)C2)=O)c1 66635,c1(NC2CC3CN(C(C4CC5(C4)CC5(F)F)=O)CC32)ncc([N+](=O)[O-])cc1Br 66636,C1(C(=O)NC2(CC=C)CCOC2)C=CCN(C(c2cccc(O)n2)=O)C1 66637,N1(CCC)CC(C(=O)N(CCCCNC(c2ccc(C(=O)OC)[nH]2)=O)C)CC1=O 66638,c1(OC)ccc(N2CCC(Cc3ccc(OC(F)F)nc3)C2)cc1 66639,N1(C(C(CC)OCC)=O)CC2CCC1C(CNC(c1cc(C3CC3)[nH]n1)=O)C2 66640,CCC(CC)CC(=O)N1CCN(C(c2csc(-c3ccccc3)n2)=O)C2CC12 66641,c1(C(N2CCN(C)C(CNC(=O)COCC3CCC3)C2)=O)cc2ccncc2s1 66642,N1(C(C(C)(C)SC)=O)CC(NC(c2csnn2)=O)C(c2nccn2C)C1 66643,C1(S(N)(=O)=O)(C(N(C(c2ccccc2F)CNC(=O)Cc2ccoc2)C)=O)CC1 66644,N1(CC2CC3(C(NC(=O)OC(C)(C)C)CC3)C2)CCCc2c(CO)cccc21 66645,C1(N(C(C=NOC)=O)CC)CCC(NC(c2ccnc(OC)c2)=O)CC1 66646,c1(N2CCN(C(=O)OC)CC2)nc2c(c(=NC3COCC3F)[nH]1)CSC2 66647,c12ccc(Cl)cc1NC2.c1(CC)cnc(CC(=O)N(CCOCCCO)CC)[nH]1 66648,n1(CC(=O)NCC(CCNC(C2(CC)CC(C)(C)C2)=O)O)nnc2c1CCCC2 66649,N1(C(c2ccc(C)c(CN3CCCCC3)c2)=O)CCCNC(=O)C(F)(F)C1 66650,c1(NC(N(C(CC(CC)C)C)CC)=O)cnc2ncnc(O)c2c1 66651,c1(C(N2CCC(CNC(c3nn(C)c(F)c3)=O)C2(C)C)=O)ccc2ncsc2c1 66652,Cc1cc(N)cnc1C(=O)NCCCCN(C)C(C1CC(C)(C)C1)=O 66653,CC1SCCN(C(c2ncc(F)cc2F)=O)C1C.C12CC(C1)NC(=O)CN2C1CCC1 66654,C=CCC(C)(C)C(=O)NC1CC(CC(N2CCC3CC23C)=O)C1 66655,c1(C(=O)NC(C(C(C)C)C)CNC(c2cnsn2)=O)c[nH]c2ncccc12 66656,C1(C(N2CC(N(CCC)CC)C2)=O)CN(C(=O)C(CC)OCC)CC(C)(C)C1 66657,c1(OCC)cc(-c2cccc(NC(c3cnn(C(C)(C)C)c3)=O)n2)ccn1 66658,CCCC(C(=O)OC)C(=O)NC(C)CN(C)C(c1sc(C)c(C)c1C)=O 66659,N1(C(C(CNC(COC(CC)C)=O)CC(C)C)=O)CCC(N(C)OC)CC1 66660,c1(C(=O)NC(C2(O)CN(C(C3(C4CCCCO4)CC3)=O)C2)C)cccn(C)c1=O 66661,C1(O)(CCNC(CCOCC#C)=O)CCCN(C(=O)CC(=C)Br)C1 66662,CC1(C)C(NC(c2ncccn2)=O)CC1N=c1nc(C2CCOCC2)[nH]s1 66663,Cc1cc(C(=O)NCC2CCC(C(=O)N(C(C)CCC(C)C)C)C2)c(C)s1 66664,C(C(C)C)(C(O)C(=O)N1CCC(OCC(N2CCC(=O)N(C)CC2)=O)C1)OC 66665,c1(OC(C)C)ccc(Cl)nc1C(=O)NC1(CCCNC(=O)C(C)O)CC1 66666,C1(NC(C(C)NC(=O)NCC)=O)CN(C(=O)CO)CC2(CCC2)C1 66667,N1(CC(=O)NC(C=CC(=O)NC(c2ccnc(F)c2)C)(C)C)C(=O)CNC1=O 66668,C1(NC(CCCc2n(C)cnn2)=O)CCN(C(C2CC3(CCC3)C2)=O)CC1F 66669,c1(C(N2CC(CNC(CCCCCOC)=O)C(F)(F)C2)=O)c[nH]c2ccncc12 66670,C1(NC(c2ccc(C=C)cc2)=O)CCN(C(c2cnn(C)c2C)=O)C12CCC2 66671,N1(C(c2n(C)c(C#N)cc2)=O)CCC2(CC(NC(=O)C(C)(C)c3cnsc3)C2)C1 66672,N1(C(C(C(C)C)F)=O)CCCC(C(=O)NCCC(F)CN=[N+]=[N-])CC1 66673,c1(C(N2CC(CCNC(CC3(OC)CCC3)=O)(OCC)C2)=O)ccc(C)cc1 66674,c1(-n2cc(C(C(C)C)NCC3CCCC3O)nn2)ccc(I)c(Cl)c1 66675,C(C(C)(C)C(=O)NCCC1CCN(C(C2CN(C(C)C)CCO2)=O)C1)OC 66676,N1(C(C(C=CC)O)=O)CCN(C(c2cnsc2)=O)CC1C.c1(C)ccccc1 66677,c1(N2C(CCNC(=O)CC34CNC(=O)C(C3)C4)CCCC2)nc2ccccc2o1 66678,CCC(CC(=O)NCc1ccc(CNC(=O)C(O)CCOC)cc1)C(C)(C)C 66679,c1(C(=O)NCC(CO)NC(C(C)OCC)=O)ccc2ccc(Br)cc2c1 66680,c1(CC(c2n(CCC)nnn2)NC23CC(F)(C2)C3)ccc(OC)c(C)c1 66681,CON(C)CCNC(C1(C2CCCN2C(c2n[nH]cc2Cl)=O)CC1)=O 66682,C(=O)(N=c1[nH]c(Cl)ncc1O)C1C(C(=O)Nc2c(C)cc(F)c(C#N)c2)C1 66683,N#Cc1ccc(O)c(CNC23CC(C(=O)NC(=O)C(F)Cl)(C2)C3)c1 66684,c1(CC(=O)N(C(=O)C(C)(C)CF)C)ccccc1CNC(=O)C(C1CC1)C1CC1 66685,Cc1cc(C)c(C(N2CC(NC(=O)C(O)CC(F)(F)F)C(C(F)F)C2)=O)c(=O)o1 66686,c1(C(=O)NCC(CO)NC(c2[nH]cc(OC)c(=O)c2)=O)ccc(C)c(Cl)c1F 66687,c1(C(N(CCNC(c2cnn(CCC)c2C)=O)C)=O)cnc2ccc(Br)cn12 66688,CC(C)CC(C(=O)N(C)C)N(CC(F)(F)F)C.C1(=O)C(C)NC(=O)N1 66689,N1(C(C(C)(C)CN2CCOCC2)=O)CCCOC(CCNC(C2SCCS2)=O)C1 66690,N1(C(c2cc(OC)cc(C)n2)=O)CCC(C)N(C(C2CCCC(=O)CC2)=O)CC1 66691,C12(CNC(C3C(=C)C3)=O)CCC(C1)N(C(=O)CCC(=O)c1ccccc1)C2 66692,C(C(C(=O)N1CCCC1CNC(=O)Cn1cnc(C(F)(F)F)c1)N(C)C)N(C)C 66693,C(=O)(C1=CCCN(C(=O)Cc2ccc(C#N)cc2)C1)NCC1C(C=C)C1 66694,c1(CCNCCNC(c2ccsc2CO)=O)nccc(Cn2cc(Cl)cn2)n1 66695,Cc1nc(C2CCC2)oc1C(=O)NC(C)(C)CNC(C1(C#N)CC1C)=O 66696,CC1(C)C(CNC(=O)C(Cc2ccoc2)NC(=O)CC2CNC(=O)O2)C1(C)C 66697,N1(C(C2=CC(O)C(NC3CCCN(C(C)=O)C3)C2)=O)CCCC(C2(C)CC2)C1 66698,C1(O)(C(N2CCCC(CNC(=O)CCc3ccsc3)C2)=O)CN2CCC1CC2 66699,CCC(C)CC(=O)C(=O)NCC(CC)N(C)C(c1cccn1CC)=O 66700,Cc1nnc(NNC(=O)N(C2CC(O)C2n2cccn2)C2CC2)n1N 66701,c12cc(ccc1F)CC1CCN(C1)C2=O.c1(SCC)ccccc1O.CO 66702,N1(C(C(C)=C(C)C)=O)CCC(F)(F)C(CNC(c2cnoc2-c2ccco2)=O)C1 66703,CCC(CS(=O)(=O)c1ccccc1)OC(c1ccc(C2CCOC2)cc1)=O 66704,C1(NC(=O)COC2CCC2)CN(C(C2(F)C3CCCCC23)=O)CC1C1CC1 66705,n1(CC)nc(C(=O)NC2(C(=O)NCC3N(C(C)=O)CCC3)CCCC2C)cc1C 66706,N1(C(Cc2c(C)ncnc2C)=O)CC2(CC(NC(=O)C(C)O)c3nccn32)C1 66707,N(C(=NCCF)N1CCC2(O)CCOCC2C1)CC1(C)CCCCC1 66708,CC1CCCCN1S(=O)(=O)N1CCN(C(=O)NC2(C#N)CCCCC2)CC1 66709,c1(C(N2CC(C(=O)NC)C2)=O)ccc(CCNC(c2cnn(C)c2C)=O)cc1 66710,c1(C(N2CCCC(NCC(n3cc(Cl)cn3)C)C2)=O)c(Cl)cccc1[N+](=O)[O-] 66711,C1(NC(c2nc(CC)oc2)=O)CCC2CCN(C(c3cnoc3C3CC3)=O)C1C2 66712,CC1CCC(NC(=O)C=Cc2ccc(C(N)=O)o2)CN1C(c1nnn(C)c1N)=O 66713,c1(NC(C(C)NC(C)=O)=O)cc(Br)ccc1NC(=O)c1c[nH]nc1OC(C)C 66714,C1(CNC(c2cc(C(F)F)cc(F)c2)=O)CC2C(O)CC2O1 66715,CC12CCCC1N(C(c1cnc(C(F)F)nc1)=O)CCN(C(c1ccsc1)=O)C2 66716,Cc1cc(C(=O)NC2CCN(C(C3CS(=O)(=O)C3)=O)CC2C)nc2[nH]nc(O)c12 66717,C1(C)(C(=O)NC2(CC(=O)NC(C3CCCCC3)C)CCC2)CC(F)C1 66718,C#Cc1cccc(CNC(C2(NC(=O)Cn3nccn3)CC(CO)C2)=O)c1 66719,C1(NC(c2cc(C(C)=O)[nH]n2)=O)COC2(CCN(C(C3(C)COCCO3)=O)C2)C1 66720,c1(C(=O)NCCCNC(C(C)CN(C)C)=O)ccc(C2CCC2)cc1 66721,Cc1c(CNC(=O)CSCc2cn(CC3CCOC3)nn2)oc2ccc(Br)cc12 66722,N1(C(c2c(C)[nH]cc2C(F)(F)F)=O)CCCC(NC(c2csc(O)n2)=O)C1C 66723,c1(C(N2CC(CNC(C(Br)=C(C)C)=O)C3(C2)CC3)=O)cc2cccn2cn1 66724,N1(C(c2cc(OC)c(Cl)cc2)C(=O)NC2CC2)CCCC2(CCNC2=O)C1 66725,c1(C(N2C(C)CN(C(c3occc3F)=O)CC2)=O)nc2ccccc2cc1Cl 66726,C1(C(CNC(CCC)=O)(C)O)CCN(C(=O)C#CC2CC2)CC1 66727,c1(CNC(C2(C)CCN2C(c2cc(Br)co2)=O)=O)cccc(F)c1Br 66728,c1(CC(C(=O)NCC(CO)NC(C2(C)CC=CCC2)=O)N(C)C)ccccc1F 66729,c1(CC)nc(=N)[nH]cc1C(=O)NC1CC(F)CN(C(=O)CC(C)F)C1 66730,CC(CC(F)F)C(=O)NC1CC2C1CCN2C(c1ncccc1Br)=O 66731,Cc1cc(C(N2Cc3ccccc3C2)=O)c2c(c1)CCCN2 66732,C1(NC(c2n(CC)ccn2)=O)(COC)CCN(CC=Cc2ccc(C)cc2)CC1 66733,C(=O)(CCCC(C)NC(=O)CCC1CCC(=O)C1)Nc1cc(C)sc1C 66734,C1(C(=O)NCCCCNC(C2SCCS2)=O)C2(CCC2)C12CCC2 66735,N1(C(CCC(C)SC)=O)CC2(C(=O)Nc3ccc4c(c3)OCC4)CCC1CC2 66736,c1(C(=O)NCC2CC(OC)CN2C(C2CC(SC)C2)=O)ccc2nc(C)nn2c1 66737,CC(O)CC(C)(C)CNC(C1(CNC(=O)CC2CCSCC2)CC12CCC2)=O 66738,c1(C(N2CC(N(C(Cc3cnc(C)o3)=O)C)C2)=O)cc2nn[nH]c2cc1F 66739,N1(C(=O)NC2CCN(Cc3ccccc3)C2)CCC(C#CBr)CC1 66740,C1(N(C)C(c2cc(CF)on2)=O)CC2CCC(C1)N2C(c1cccc[n+]1[O-])=O 66741,Cc1cc(C(N2C(C(=O)NC(c3cc(Cl)ccc3O)C)CCC2C)=O)cc(O)n1 66742,C1(OC)CC(C(N2CCC(NC(c3c(C4CC4)cnn3C)=O)CC2)=O)C12CCC2 66743,C1(NC(c2n(CC)cnn2)=O)C(C)CCN(C(c2cnc(C(C)C)s2)=O)C1C 66744,C1(OC)(CNC(c2cc(SC)nn2C)=O)CCN(C(c2cnn(C)c2)=O)C1 66745,N1(C(=O)NCC(c2cccc(F)c2)C(F)(F)F)CC2CC3CCCN3C2C1 66746,C(=O)(C1=CN=C2N=CNN2C1)NCC1N(C(C2N=C(C)SC2)=O)CCCC1C 66747,N1(C(CCCC(C)NC(C2N(CC)CCCC2)=O)=O)CCC2CN(C)CC2C1 66748,c1(OC)cccc(C)c1C(=O)NCCCC1CCCCN1C(=O)C(O)C(C)(C)C 66749,Cc1ncc(C=CC(N2CC=CC2CNC(c2c(C)ccnc2O)=O)=O)c(O)n1 66750,CC1(C)C(CNC(N2CCC(OCC3CC3)CC2)=O)CC1Cc1ccccc1 66751,n1(CCCCCNC(c2ccns2)C)c(S)nc2c(Br)cccc2c1=O 66752,N1(C(=O)NCC(CCSC)OC)CCCCC(OC(C)C)C1 66753,c1(CNC(NN(CC2(OC)CCOCC2)C)=O)ccc2c(c1)NCCO2 66754,C(=O)(CC(C(F)(F)F)OC)NCc1cccc(CN(C(CCC=C)=O)C)c1 66755,Cc1cc(N2CCC(NC(=O)CC3CCS(=O)(=O)C3)C2)c([N+](=O)[O-])c(C)n1 66756,C(=O)(CC(O)CC1CC1)NC(CNC(C=CCC)=O)(C)Cn1cccn1 66757,C12(CN(C(CO)CCSc3ccccc3)CC=C(C)C)CCCC1CCC2 66758,Cc1noc(C)c1CC(N1CSCC1C(=O)NC1CC(CCC(N)=O)C1)=O 66759,CC1(C)CCC(NC(C2(C(N)=O)CC2)=O)C(CNC(=O)Cc2ccccn2)C1 66760,c1(Cn2cc(C(C)(C)F)nc2)cc([N+](=O)[O-])ccc1Br 66761,CC(C)(C)C(=O)C(=O)N1CCC(C)(NC(=O)C(CCc2ccccc2)C2CC2)C1 66762,C1(C(=O)NC(C(C)(C)C)CNC(C2CC(C(F)F)C2)=O)CN(S(N)(=O)=O)C1 66763,c1(C(N2CC3C(NC(c4cc(C)c(N)cc4)=O)C3C2)=O)ccc2cccnc2n1 66764,Cc1nc2ccccc2n1C1CN(C(=O)NN2C(C)CCC2C)C1 66765,C1(C(=O)NC(CC2CC2)C(=O)NC2C3COCC23)CC2(CCC2)CO1 66766,N1(C(C(C=C)(C)O)=O)CC2(C1)OC1(C)CC2(NC(C2CCN3CCCC3C2)=O)C1 66767,N1(C(c2cnc(C)s2)=O)CC2CC(NC(C3CCCC(F)C3)=O)CC1C2 66768,CC1(C)CC(C(=O)NC2(C(=O)NC34CCCC3C4)CC(O)C2)=NO1 66769,N1(C(=O)NCc2nn(C)c(=O)o2)CCCC(C)(CN2CCCC2CCC(=O)O)C1 66770,c1(CC)nc(C(=O)N(C2CC(NC(=O)CC(C)OC)C2)C)c(C)o1 66771,C1(CC=CC(=O)NC(C)C(C)NC(=O)CCN2CCOCC2)(OC)CCCC1 66772,C1(C(=O)NC(C)CCNC(=O)C(O)C2CCC2)C(c2ccncc2)C1(C)C 66773,c1(NC(C2CN(C(=O)CCc3ccnc(F)c3)C2)=O)ccc2scnc2c1 66774,c1(NC(C2CCN2C(c2cc(Cl)cc(Cl)c2)=O)=O)ncc(F)cc1Br 66775,C12(C(=O)NC(CCNC(C3CN(C(=O)NC)C3)=O)C)CCCCN1CCC2 66776,C1(NC(Cc2c(C)nc[nH]2)=O)CCN(C(c2sc(F)cc2Cl)=O)C(C)C1 66777,c1(C(c2n(C)nnn2)NC(C)(CCF)C(=O)O)cc(Cl)c(Br)cc1F 66778,c1(C(=O)NC2CCN(C(C3=NNC(=O)C3)=O)CC2F)ccc(F)c2ccsc12 66779,S(=O)(=O)(c1ccc(C2SCCS2)cc1)NC(CN(CCNCC1CC1)CC)=O 66780,C12(C(=O)NC3CCCN(C(COC)=O)CC3)CCCC(=O)N1CCC2 66781,C(=O)(C(C(C)Cc1ccc(CC)cc1)N1CCCC1COC)NCCC 66782,CCCCCS(=O)(=O)CC(=O)NC1(CNC(=O)C(c2ccccc2C)C)CC1 66783,c1(C(N(CCOC)CCNC(=O)CC2COCC2O)=O)cc(F)ccc1C(F)F 66784,N1(C(C2CC(OC)(OC)C2)=O)CC2CC(NC(c3cncc(C4CC4)c3)=O)C1C2 66785,C(C(C)(Cn1cccn1)N=c1[nH]nc(C)s1)NC(C(CC=C)(C)C)=O 66786,C=C(C)C(C)(C)C(=O)N1CCC(C2CCCN2C(c2c[nH]c(C)cc2=O)=O)CC1 66787,CC1(C(=O)NCCNC(c2ccc(F)c(F)c2N)=O)CC2CCC(C1)S2 66788,c1(NC2CCCN(c3c(F)cncc3F)C2)ccnc2c(Cl)cnn12 66789,CC(C)(CNC(c1cc([N+](=O)[O-])c[nH]1)=O)CC(=O)NCCCOCC1CCC1 66790,C1(CNC(C(C)NC(C)=O)=O)CC2(CCC2)CN1C(=O)C=Cc1cocn1 66791,c1(-c2cc(C(=O)Nc3c(C)ccnc3Br)ncc2)cc(F)cc(C)c1O 66792,C12(NC(C(C)OCC#C)=O)CCC(C1)N(C(=O)CCCC(=O)NC)C2 66793,Cc1ccc2c(C(=O)NCC3CCN(C(=O)C#CC4(C)COC4)C3)cnn2c1C 66794,C1(OC)CCC(CC(=O)NC(C)C(C)(C)NC(C2CC(=C3CCC3)C2)=O)CC1 66795,CC1CC(C(=O)N2CCC(CCNC(c3ccn(C)n3)=O)C2)c2ccccc2N1 66796,c1(CCC(=O)NCCC2CCCN(C(C(CC)F)=O)C2)nc2cnccc2[nH]1 66797,c1(OC)ccc(CN2CCOC(CC(=O)Nc3nccnc3Br)C2)cc1[N+](=O)[O-] 66798,C1(NC(C2(C(=O)OCC)CC2)=O)CCN(C(c2ccc(N(C)C)nc2)=O)C1C 66799,N1(C(c2ccc(C(CC)C)cc2)=O)CC(NC(c2nc(C)no2)=O)C(C)(C)C1 66800,c1(C(=O)NC2CC2CNC(C2CCS(=O)(=O)CC2)=O)cc2ccccc2c(O)n1 66801,c1(OC)cc(OC)c(F)c(NC(C2CC2NC(c2cnccc2C#N)=O)=O)c1 66802,c1(C(=O)NC2C(CC)N(C(c3ccc(C4CC4)s3)=O)CC2)ccc(N=[N+]=[N-])cc1 66803,c1(C(=O)NC2(CCNC(CCNC(=O)NC)=O)CCC2)ccc(Br)c(F)c1 66804,Cn1ncc(Cl)c1C(=O)NC1C2CN(C(C3CC3Sc3ccccc3)=O)CC12 66805,C(C)(CC(C)(C)O)NC(C(C)N(C(=O)C(c1ccnn1C)C)CCC)=O 66806,N1(C(=O)CCNc2ccccc2)CCCC(NCCN2CCCS2(=O)=O)C1 66807,N1(C(C2C(NC(CC(CC)CN(C)C)=O)CCO2)=O)CC2CC(C)(C)C2C1 66808,C(C(O)CC(=O)N(C1CC1C)C)NC(c1c(C)ocn1)=O 66809,c1(C(N2CCC(NC(C(C)SCCOC)=O)C2)=O)ccc(-c2ccco2)nc1C 66810,CC(C)C(C(=O)N(CCCCN(C(=O)CNS(C)(=O)=O)C)C)NC(N)=O 66811,C(CC(C)C(=O)NC(C1CCCN1C(=O)C(=O)NC1CC1)C)=CC 66812,N1(C(C2C=CCS2)=O)CCC2CN(C(=O)CSC3CC3)C2C1 66813,C1(Nc2nnc(C)c(C)n2)CCCC2CN(C(C3(F)CCC3)=O)CC12 66814,Cn1cc(C2CC2NC(c2c[nH]nc2CNC(c2cnn[nH]2)=O)=O)cn1 66815,c1(OC)ccccc1-c1noc(C(C)SC2CCCC(c3ccc(Cl)cc3)C2)n1 66816,C1(C)(C(N2CC(C(C)NC(c3c(OCC)n[nH]c3)=O)C2)=O)CCCN1C 66817,c1(OC)cc(C(N2CCC(NC(c3ccc(N)cc3Cl)=O)C2)=O)cc([N+](=O)[O-])c1 66818,Cc1cccc(O)c1C(N1CCCC(C)(NC(=O)CCC(F)F)C1)=O 66819,CC1CN(C(=O)C(Cl)=CCl)CC(C)N(C(c2ccnc3c2ccn3C)=O)C1 66820,C1(C(=O)NC2C(N(C)C)CCOC2)CCOCC1NC(C1CC2(CSC2)C1)=O 66821,c1(C(C)N(C)C(=O)NCC2COC3(CNC3)C2)cccc([N+](=O)[O-])c1 66822,CC1CN(C(C2CCCN2C(C23CCCN2CCC3)=O)=O)CCCO1 66823,N1(C(c2n[nH]c(=N)[nH]2)=O)CCCC(F)(C(=O)NCCCS(C)(=O)=O)C1 66824,C(=O)(C1=CCCCC1C)N1CC(NC(c2c(C)nc(C3CCC3)o2)=O)C1C 66825,c1(CC=C)ccccc1NC(=O)C(=O)NCC(C1CCOC1)NC(=O)CC 66826,N1(C(c2c(C)nc(CCC)o2)=O)CC2(CCCC2NC(C2CCCN2CC)=O)C1 66827,Cc1cc(C(F)(F)F)cc(C(F)(F)F)n1.c1(C(C)(C)N)nc(C(C)(C)N)no1 66828,C(=O)(CC(C(C)C)NC(=O)Cn1c(C)ccc1C)NC(C(=O)OCC)C1CC1 66829,C1(C(=O)Nc2ccccn2)CC2C1CCN2C(C1CCN(C(=O)C2CC2)CC1)=O 66830,Cc1nc(C(=O)NC2CCC(NC(=O)C(C)C3CCC3)C2)sc1C 66831,CCCC(CC(C)C)C(=O)NC(COC(C)C)C(N1CC(CO)C1(C)C)=O 66832,Cc1cc(=NCC(N(C(=O)CCN(CC(F)(F)F)C)C)OC)[nH]c(C)c1C#N.C1CC1 66833,c1(C(c2nnnn2C(C)CC)NCCCC(=C)C)c(O)nsc1OC 66834,CC(C)CC(O)CC(=O)NC1(Cc2ncc(F)cn2)CC1 66835,C12(OC)CCC1CN(C(=O)CC1CCN(C(=O)CCCC3CCCC3)C1(C)C)C2 66836,Cc1c(C(N2CCSCC2CCNC(C2CN(C)C2)=O)=O)sc2nccn12 66837,N1(C(=O)NC2(CO)COCC23CCC3)CCc2cc(Br)c(F)cc2C1 66838,c1(C(N(C2CCN(C(c3cnco3)=O)C2)CC#C)=O)nocc1C 66839,c1(C(=O)NCC2C3N(C(C4C(CC)C4)=O)C(CC3)C2)cc(Br)cc(C)c1F 66840,O=C(CCCCCO)Nc1nc(-c2ccc(O)nc2)cs1.C12CC(F)CN(C1)C2=O 66841,N1(C(CCCC#C)=O)CCC(C2CCCN(C(=O)CCC(=O)C(C)(C)C)C2)CC1 66842,N1(C(CC2CCC(=O)NC2)=O)CCN(C(c2cccc(Cl)c2F)=O)CC(CO)C1 66843,Cc1cccn(CC(=O)NC(C2CCCN2C(c2cc[n+]([O-])cc2)=O)C)c1=O 66844,CN=c1ccc(C(N2CC(O)CC2CC(=O)NCC(=O)N2CCCO2)=O)c[nH]1 66845,O=C(CS(=O)(=O)C12CC(C1)C2)NC1(CNC(c2sccc2Cl)=O)CCC1 66846,c1(N(CC)CC)nnc(C2CCC2)n1CCC(c1ccccc1)C 66847,CCCCCC(O)C(=O)NC(C1(O)CN(C(C2CN(C(C)=O)CCO2)=O)C1)C 66848,C1(C(=O)OC)CCC(C)(C(=O)NCCN(C(=O)CSCCC#N)C)C1(C)C 66849,C1(C(=O)NCC(CN(C(CC(C)NC(N)=O)=O)C)O)CCC(=O)N1C 66850,C1(C(CO)NC(C(C)CF)=O)CCN(C(C2(F)CC2(Cl)Cl)=O)CC1 66851,S(=O)(=O)(c1cccnc1)N1CC(NC(C2CCN(CCOCC)CC2)=O)C(O)CC1 66852,N1(C(c2scnc2C)C(=O)NCCCCCC)CCC2(O)CCOCC2C1 66853,c1(NCC(=O)NCC(F)F)cc(NC2(n3cccn3)CCC2)ncn1 66854,CC(C(=O)Nc1c[nH]nc1C(=O)NC(C1CC1)C1CC1)S(C)(=O)=O 66855,c1(NC(C2OCCN(C(C(C)(C)C)=O)C2)=O)ccc2c(c1)OCC2 66856,N1(C(CCCCOCC)=O)C2CCC1CN(C(c1cc(C)n(C(F)F)n1)=O)CC2 66857,N1(C(c2ccc(SC)s2)=O)CC2CCN(C(=O)C(c3cccc(F)c3)O)CC2C1 66858,N1(Cc2nnc(C)c(C)c2-c2ccnn2C)CCc2cc(Br)c(Cl)cc2C1 66859,C1(C(N(CCN(C(c2cncc(OC)c2)=O)C)C)=O)CC2(COC(=O)N2)C1 66860,N1(C(C(C)OCC=C)=O)CCCN(C(c2cnc(Cl)nc2)=O)C(C)C1 66861,Cc1nc(C=CC(=O)NC2COCCN(C(C3SC4C=CC3CC4)=O)C2)[nH]c1C 66862,CN1CCCCC1C(N1CCC1C(=O)NC1(CO)CC1)=O 66863,c1(OCC)ccc(C(=O)NC(C2(CNC(c3cc(C#N)c[nH]3)=O)CC2)C)cc1 66864,C1(C(=O)Nc2c(CCNC(CC(=O)NCC)=O)ocn2)CCCCN(C(=O)OC)C1 66865,C1(C(=O)NCCNC(C2(OCC)CC2)=O)CC12CCOCC2 66866,C(=O)(C1CCc2c[nH]nc21)NCC(CO)NC(c1ccn(CCF)n1)=O 66867,c1(NC(N2CC(C)OC(C)C2)=O)ccc(O)c2ncccc12 66868,C1(NC(C2C(OC)CCCC2)=O)CCC2(CC1)CN(C(=O)CS(=O)(=O)C1CC1)C2 66869,Cc1cc2occ(NC(=O)Nc3ccc(N(C)C)cc3C(F)(F)F)c2cc1C 66870,Cc1cc(C(=O)NCC2CN(C(C3CC3C3CC3)=O)CC2(C)C)c(Cl)cn1 66871,n1(CC(=O)NC)cc(C(=O)NCCC2CN(C(C3CC3Cl)=O)C2)nn1 66872,N1(C(c2c(C(C)C)occ2)=O)CCC(C)(C(=O)NCCC(N)=O)C1 66873,C(=O)(N=c1cc(-c2ccc(F)s2)[nH][nH]1)NC(c1cccc(Cl)c1F)C 66874,c1(COC(C2CS(=O)(=O)CC(=O)N2)=O)ccc2ncccc2n1 66875,C(CC(=O)NCCCCCCF)(C(F)F)NC(CC(C)c1ccco1)=O 66876,C1(C)(C(=O)NCC(C)N(C)C(c2ccncc2O)=O)CCCCC1(F)F 66877,C1(C(N(C)Cc2cc(C)no2)=O)CCCN(C(c2nc(C)oc2C)=O)C1 66878,Cc1nccc(C(=O)NCC2CCCCN(C(=O)C(O)CC(N)=O)C2)c1C 66879,C(CC(=O)NC1(C)CC(NC(C2(O)CC2(C)C)=O)C1)(C(N)=O)NC(C)=O 66880,CC(CC(F)F)C(=O)N(CC(O)CNC(c1ccnc(CO)c1)=O)C 66881,N1(C(c2c(C)noc2C(F)(F)F)=O)CCC2CC(C)CCC12 66882,N1(C(C)C(=O)NC(C2(O)CN(C(C3CCC(=O)O3)=O)C2)C)CCCCCC1 66883,N1(C(CC(C)SC)=O)CCC2(CC1)CC(NC(c1sc(F)cc1Cl)=O)CO2 66884,C1(O)(C(C)NC(C(N2C(=O)CCC2=O)C)=O)CCN(C(=O)C2=CCC2)C1 66885,CC1CCN(C(c2conc2C2CCC2)=O)CC1NC(=O)CCc1ccccc1 66886,n1(CCCC)ncc(C(=O)NC(C2CN(C(=O)C(C)(C)C3CCCO3)C2)C)c1C 66887,N1(C(C=C(CC)CC)=O)CC(C(N2CCCC2(C)C2CC2)=O)C(F)(F)C1 66888,c1(C(C(=O)NC(C)C)N(CC(=O)NC(c2ccccc2)CO)C)ccccc1 66889,CC(C)C(O)CNC(=O)C(C)(C)NC(c1ncn(C)n1)=O 66890,C1(C(=O)NC(CN(C)C)CCO)(CC)CCCN1C(C1CC(N=[N+]=[N-])C1)=O 66891,Cc1cnc2c(C(=O)NCC(CO)NC(=O)C(c3ccc(C)o3)C)c(C)nn2c1 66892,N1(C(CCc2cc(OC)c(O)cc2)=O)CCCC12CCN(C(C1CCC1F)=O)C2 66893,c1(C(N2CC(C#C)C2)=O)cncc(CNC(=O)COCc2nc[nH]n2)c1 66894,c1(N2CC(C(C)NC(Cc3c(OC)cccc3)=O)C2)ncnc2c1CCC2 66895,C1(C(N(CC(C)(C)C)C)=O)CCCN(C(=O)Cc2cnn(C)c2)CC1 66896,CC(CC(F)F)C(=O)NC1CC=CCC1C(N1CC(O)(CCO)C1)=O 66897,c1(C(=O)NCC=CCNC(c2cccc(C)c2)=O)ccc2nc(N(C)C)[nH]c2c1 66898,c1(OC)c(F)cc(NC(=O)CN2CCN(C(=O)Cc3cnc(C)s3)CC2)cc1F 66899,c1(OCC)cccc(C)c1NC(C1CN(Cc2cccc(OC)c2Br)C1)=O 66900,CN1CC2CC2(C(=O)NCC2CC(NC(=O)OC(C)(C)C)C2(C)C)S1(=O)=O 66901,N1(C(C2(F)CCCC2)=O)CCC2(CC1)CN(c1ccnc3ncnn13)CCO2 66902,c1(OC)ccc(C(=O)C(=O)N2CC(N3CCCC3)C2)cc1.C12CC1C(=O)N2 66903,Cc1ccc(CN2CC(F)CC2C(=O)Nc2ccnc(-n3cccc3)c2)cc1 66904,Cc1cnc(NCC2CC3C=CC2O3)c(S(=O)(=O)NC(c2ccco2)C)c1 66905,C1(C)(C(=O)NCCCNC(C2(NC(C)C)CC2)=O)CCOC1 66906,n1(CC)ccc(C(=O)NCC2(NC(=O)C=CC(=O)NC3CC3)CCOC2)c1C 66907,C1(CC(c2nnnn2C2CC2)(C)NC2CCN(c3ccccn3)C2)CCOCC1 66908,c1(SCC2CC(C(C)OC)C2)cc(F)c(F)c(Cl)c1 66909,C1(NC(C(C)Cc2ccco2)=O)CC(NC(=O)Cc2cnoc2)CC1O 66910,N1(C(C2CCCN(C)C2)=O)CCC2(CC(NC(C3(C)CSC3)=O)C2)C1 66911,C1(NC(c2cc(OC)ncn2)=O)CCCN(C(C2CCSC2)=O)C1C 66912,c1(C(=O)NCC(C2CCC2)NC(Cc2cc(C)sc2)=O)sc(N(C)C)nc1C 66913,CCCCCCC(C)(C)C(=O)OCC(=O)C(C)(C)[N+](=O)[O-] 66914,N1(C(c2c(CC)nccn2)=O)CCCC2(CCN(C(=O)C(C)NC(C)=O)CC2)C1 66915,C1(C(N2CC(CC)N(C(=O)Cc3c[nH]nc3O)CC2)=O)CC12CCC1(CC1)CC2 66916,c1(OC)c(CNCC2CCCN2C(=O)CCC(N)=O)cc(F)cc1F 66917,CC1CC=C(C(=O)NCCC2(CNC(=O)C(=O)C3CCCC3)CC2)CC1 66918,C(=O)(C(C(C)(C)C)OC)N(CC(C)NC(C12CC(c3ccccc3)(C1)C2)=O)CC 66919,N1(C(CN2CC(=O)NCCC2)=O)CC2CC(F)(F)CCC2(C(=O)O)C1 66920,C#Cc1cccc(OCC(=O)NC2(F)CCCN(C(=O)C3=C(C)OCC3)C2)c1 66921,c1(C(N(CCCN(C)C(c2ccc([N+](=O)[O-])o2)=O)C)=O)cnc(N)c(N)c1 66922,C1(c2nc(-c3ccc(OCC)cc3)nn2CC2CCOC2)CC2C(C1)C2(F)F 66923,Cc1cc(C)n(CCc2nc(C3CC3C(=O)O)nn2-c2ccc(Cl)cc2)c(=O)n1 66924,Cc1nc(C#N)ccc1C(=O)N(CC(C)NC(c1ccnn1CC(C)C)=O)C 66925,c1(C(=O)NCC(COC)NC(=O)C(C)n2cccn2)conc1C1CCCC1 66926,N1(C(C(c2cccc(Cl)c2)C)=O)CCC2C(C1)CN2C(C1CCCN1C)=O 66927,C1(NC(c2ccc(Br)o2)=O)CCC(CNC(c2cccn2C(F)F)=O)C1 66928,C1(O)(C(=O)NCC2(CCNC(C3(C)COCCO3)=O)CC2)CN2CCC1CC2 66929,C1(c2n(CCC=C)c(N(CCC3CC3)CC)nn2)COc2ccccc2O1 66930,C1(C(=O)NCC(Cc2ncn(C)c2)O)CC12CCSCC2 66931,C1(NC(c2cc(C)c(Cl)s2)=O)C2CC1N(C(=O)C(O)Cc1ccccc1)C2C 66932,c1(OC)c(C(=O)NCC(C2CCCC2)NC(c2cnncc2O)=O)csc1C 66933,c1(C(=O)NC(CNC(C(COC)COC)=O)(C)C)cc2n(n1)CCCC2 66934,Cc1csc(C(N2CCOC(CN(C(=O)CN(CC(C)(C)C)C)C)C2)=O)c1Cl 66935,c1(C(N2CCC(C)(C)C2CNC(c2csnn2)=O)=O)cc2ccc(Cl)cc2[nH]1 66936,CCCCCC(C(=O)NC1CCC(F)(F)CC1)N(CCCC1CC1)C 66937,N1(C(Cc2nc(C)[nH]n2)=O)CC2CC(NC(=O)Cc3cc(Cl)cc(Cl)c3)C(C2)C1 66938,C1(C)(CCNC(COCC(C)C)=O)CCN(C(=O)CSC(F)F)CC1 66939,CCC(C#N)C(=O)N1CC(COC)CC1CNC(=O)C1=CCCC1 66940,CCCC(CC)C(=O)NCC1CC2CC2N1C(c1cnn(CCOC)c1)=O 66941,O=C1CN(CCC(N2CC(O)CC3(CCCC3)C2)=O)c2ccccc2N1 66942,c1(C(=O)NC2C(C)CN(C(=O)CC3CCNC3=O)C2)ccc2c(c1)C(C)CN2 66943,N1(CC)CCOCC1CC(=O)OC(CCC1CC(C(=O)Oc2ccccc2)C1)=O 66944,N1(C(C=CCCC=C(C)C)=O)CCC12CN(C(c1cc(C)c(Cl)cn1)=O)C2 66945,C1(CC)CC(C(=O)NCCCC(C)NC(c2ccc(F)s2)=O)CCC1=O 66946,C(=O)(CCCCC(F)(F)F)NC1CN(C(CC2CN(C(C)=O)C2)=O)CC(C)C1 66947,c1(C(N2CCC(c3cnco3)C2)C(=O)NCCn2cccn2)ccc(C(F)(F)F)o1 66948,N1(C(C(CC)n2cccn2)=O)CC(C2CCN(C(=O)C3=NOC(C)C3)CC2)C1 66949,C1(NC(c2ccn(CCC)n2)=O)CCCCN(C(c2ccc(O)nc2)=O)C1 66950,Cc1cnc(CCC(=O)N)[nH]1.C(=O)(CCC1CC1)N(C)CCN(C)C 66951,CCC(CC(=O)NC1CC2CC1N(C(c1c(F)cccc1F)=O)C2)C(F)F 66952,c1(COC)nc(NCc2cncn2C)cc(=NC2CCC(C(=O)N(C)C)CC2)[nH]1 66953,c1(C(=O)NC2C3CN(C(C(CC)=CC)=O)C2CC3)cc(S(=O)(=O)NC)ccc1F 66954,c1(C(N(C(C)CNC(c2onc(C)c2C)=O)CC)=O)cc(CO)ccn1 66955,C1(CNC(C(COCC)C)=O)CN(C(=O)CCCF)CCC1(C)C 66956,C(=O)(C1=CC(C)(C)C1)NC(C)CCNC(=O)Cn1nnc(C2CC2)n1 66957,c1(NC(C2CC(O)CN2)=O)n[nH]c2c1CN(C(C1CCC(O)CC1)=O)CC2 66958,c1(NC(C(CCNC(CN(C(C)C)C)=O)O)=O)cc(O)cc(F)c1 66959,N1(C(C2C(C)OC(C)C2)=O)CCC2(CNC(=O)CC3CSC3)CCCC12 66960,N1(C(CNC(=O)NC)=O)CCC(C(=O)NCC2CN(C3COC3)C2)C1 66961,N1(C(CC(C=C)(C)C)=O)CCC2CC(C1)CN(C(=O)C(c1ccccc1F)C)C2 66962,c1(C(=O)OC)ccc(-c2ccc(-c3cn[nH]c3)cc2)n1C 66963,N1(C(C(c2cncc(F)c2)C)=O)CC2CC(NC(C3(n4ccnn4)CC3)=O)C(C2)C1 66964,C1(C(N(CC(=O)N(CC(C)C#N)C)CCC)=O)CCS(=O)CC1 66965,N1(C(CCCCC#C)=O)CC2CN(C(=O)C(C)=C(C)CC)CCC2(CO)C1 66966,C(C(N=c1[nH]c(=NCC(C(C)C)OC)[nH]c2ncn(C)c12)c1ccco1)OC 66967,N1(C(C2C(OC)CN(C(C3(CO)CCCCC3)=O)C2)=O)Cc2cnn(C)c2C1 66968,C1(C(=O)OC)(NC(C2CC2C(=O)NCCC2CCC(C)CC2)=O)CCCCC1 66969,N1(C(c2c(CCC)n(CC)nn2)=O)CC2CC1CN2C(=O)CCc1ccncc1 66970,C12(NC(=O)CSC(F)F)CC1CN(C(c1sc(N3CCCC3)nc1Cl)=O)C2 66971,C1(C(NC(C(CCC)C)=O)NC(=O)C(C)(C)C)CCCCN(C(=O)CSC)CC1 66972,c1(C(=O)NC(C(C(=O)NCCOCCC)C)C)cccc(F)c1C 66973,NC(=O)CCC(C(=O)NC1CC=CC1)n1cc(Cn2cc(Br)cn2)nn1 66974,N1(C(C(CCOC)N(C)C)=O)CC2(CCN(C(=O)CC3CCOC(C)(C)C3)C2)C1 66975,C1(CC(=O)N(C2CCCC(NC(C3(C(C)C)CCC3)=O)C2)C)CN2CCN1CC2 66976,N1(C(c2coc(Br)n2)C(=O)NC(C)C)CCC(CCF)(C(N)=O)C1 66977,N=c1[nH]c2ccccc2cc1C(N1CC(NC(=O)C(=O)NC=O)CC(F)(F)C1)=O 66978,C1(NC(C2(C)CCCN2C(=O)CCCN2CCCC2)=O)CC1C1CCCC1 66979,CC1(CNC(C2(C3CC3)CN(C(c3csc(F)c3)=O)C2)=O)CCCCC1O 66980,N1(c2nnc(CCC)s2)CC2CC(NC(c3ccn(C(C)(C)C)n3)=O)CC1C2 66981,c1(C(=O)Nc2nc(-c3ccccc3C(F)(F)F)cs2)ccncc1Cl 66982,C(C(F)(F)C(F)F)NC(C(CO)NC(c1ccccc1F)=O)=O 66983,C12(NC(c3cnn4c3OCCC4)=O)CCCC1N(C(=O)C1=CCCCO1)CC2 66984,N1(C(C2(F)CCC(C)CC2)=O)CCOC2(C1)CN(C(=O)CC1(C)CCOCC1)C2 66985,C(=O)(C1=NOC2(CCOC2)C1)NC1C2CN(C(C3CCC(C)C3)=O)C1C2 66986,N12CCCC(C)(C)C1CNC(=O)CN(c1ccccc1)CC2=O.CCOC 66987,C1(c2cn(C)nc2)CC(NC(=O)NCCC2CCOC2)CC(=O)N1 66988,N1(C(c2cc(SC)c(N)cc2)=O)CC2CCN(C(c3snnc3C(C)C)=O)C2C1 66989,c1(CC(=O)OC)cccc(NC(C2CN(C(=O)Cc3cc(C)[nH]n3)CC2C)=O)c1 66990,c1(C(=O)NC2CN(C(c3cc(C)ns3)=O)C(C)C2)cc(C(C)C)n(C)c1C 66991,N1(C(C23C(NC(C4=CC(C)(C)C4)=O)C4CC2C3C4)=O)CCCC(C2(C)CC2)C1 66992,C(C)(C(=O)N1CC(CNC(c2cocc2C)=O)CC(C)C1)(C(C)C)OC 66993,N1(C(c2c(C)noc2)=O)CCN(C(c2nocc2Br)=O)C2CC12 66994,C(=O)(C(CC1CCCC1)N(C1(C)CC(C(N)=O)C1)C)NCCSC 66995,CCC(C)CC(C)C(=O)N1CC(NC(=O)CCOc2ccccc2Cl)C1 66996,C1(C(=O)Nc2ccc(C)cc2F)CN(C(c2cc(C#N)oc2C)=O)CC12CCC2 66997,c1(C(=O)NCC2(F)CC3CCC(C2)N3)cc(F)c(F)c(F)c1F 66998,N1(C(CCc2cccc(C)c2)=O)CCCCC(NC(c2nn(C)cc2Br)=O)C1 66999,C1(C(=O)NC(C(=O)NCC(CC)NC(=O)C(C)(C)C)(C)C)COCCN1C 67000,NS(=O)(=O)CCC(=O)NC1CN(C(C2(F)CCCOC2)=O)C1 67001,C1(N(C(c2cnc(C(C)OC)s2)=O)C)CCN(C(=O)Cn2cncn2)CC1 67002,c1(NC(c2nc(C)n(-c3nc[nH]n3)n2)=O)ccc2nccnc2c1I 67003,c1(C(=O)NCC2C=CC(NC(c3c(CCC)nns3)=O)C2)n[nH]c2c1CCC2 67004,C1(C(=O)NCC(C)(CO)NC(CCS(=O)(=O)NC)=O)CCc2ccnn2C1 67005,CC1(C)CCCC(CC(=O)NC2(C)CCN(C(C3(O)CC3)=O)CC2)O1 67006,C1(C#N)(C(=O)NC(C(C)NC(Cc2ccc(C(=O)OC)nc2)=O)C)CCCOC1 67007,C1(NC(CCN(C(C(C=C)O)=O)C(C)C)=O)CCNC(=O)CC1 67008,N1(C(C(C)c2cc[nH]n2)=O)CCN(C(C2C3CCCC23)=O)CC1CC(F)F 67009,c1(NC(C(CCNC(=O)CCCc2cnn[nH]2)O)=O)ccc(O)c(F)c1 67010,Nc1cc(Cl)cc(F)c1C(N1CC(CNC(=O)C=Cc2ccc(C(N)=O)o2)C1)=O 67011,c1(C(=O)NC(CNC(C2(CC#N)COC2)=O)CO)cc(Cl)cc(F)c1Br 67012,S(=O)(=O)(c1cncn1C)NC(C)Cc1nccn1C 67013,C1(NC(C2C(=O)NCCCC2)=O)CCC(O)CN(C(C2(C(F)F)CC(=O)C2)=O)C1 67014,C1(NC(CC(=O)NCC#C)=O)CS(=O)(=O)CC1NC(c1nccc(N)c1Cl)=O 67015,c1(C(=O)NCC2C(NC(CCCN(C(C)=O)C)=O)C2)c(Cl)nsc1Cl 67016,C(=O)(C(O)CCC(C)C)N1CC2C(NC(c3ccc(OC)c(C4CC4)c3)=O)(C2)C1 67017,c1(NCCN(C(=O)CC2CCCCC2(F)F)CC)ncn(C)c(=O)c1Br 67018,c1(C(C(=O)NC)N(CCC)C)ncc2c(n1)CCN(C(=O)OC(C)(C)C)C2 67019,C=C(CC)CN=C(NCC1CC1)N(C)Cc1ccccn1 67020,C1(NC(C2(C)CCC(=O)N2)=O)CCC(O)CN(C(=O)Cn2ccc([N+](=O)[O-])n2)C1 67021,C(C(CC(=O)Nc1cnn(C(C)(C)C)c1)NC(C1C=CCCC1)=O)OC 67022,O=C1CN(CCC2CCN2CC2CCCOC2)C(=O)N1Cc1ccccc1 67023,c1(C(=O)NCC(CC(C)C)NC(=O)C(O)c2ccsc2)csc2ccc(F)cc12 67024,C(=O)(C#CC(C)(C)C(F)F)N(C)CCNC(C1CCCN1c1nccs1)=O 67025,C1(C(C)NC(=O)Cc2sccc2Cl)CN(C(=O)CC2CC2C)CCO1 67026,Cc1ncc(Cl)c(C(=O)NC2(c3nnnn3CC3CCOC3)COC2)n1 67027,N1(CC(=O)NCCC2CCN(C(c3cnn[nH]3)=O)C2)CCC(n2cccc2)CC1 67028,C1(CC)CCN(C(=O)Cc2ccsc2C)C(C(=O)N(CC(O)C2CC2)C)C1 67029,C(C1C(C(=O)NCCC(C)N(C)C(C2CCC=CO2)=O)C1(C)C)=C(C)C 67030,C(=O)(C(CCC(N)=O)n1cc(CCO)nn1)NC(c1cscn1)C 67031,C=C(C)c1cncc(C(=O)OCCOCC)c1 67032,N1(C(C(C)c2ccco2)=O)CCCC(NC(c2ncc(Cl)nc2Cl)=O)C1C 67033,Cc1ncnc(C)c1C(N1CCCC(C(=O)NCC(C)(O)C2(C)CC2)C1)=O 67034,N1(C(C(CC)(C)OC)=O)CCCC2(C1)CN(C(C1CCO1)=O)C2 67035,c1(CC)noc(C)c1CNC(C1C2CN(C(c3ncc[nH]3)=O)CC12)=O 67036,c1(C(N2CCSC(C)C2)C(=O)NCCOCC)ccc(-n2cccn2)cc1.C1CC1 67037,Cc1cccc(Cl)c1CC(N1CC2C(N(C(=O)COC3CCCC3)C)C2C1)=O 67038,C1(CC)CNC(=O)CN1C(=O)C(C1(CC)CCCC1)NC(=O)C(C)c1ccco1 67039,CCC(CC(=O)NCC1(OC)CCN(C(c2ccccc2C(C)(F)F)=O)C1)SC 67040,C1(NC(C(C)OCCCC)=O)CCCC(CNC(c2cnc[nH]c2=N)=O)C1 67041,c1(C(N2CC(C)C(NC(C3CCCC(CF)C3)=O)C2)=O)nn(C)c(Cl)c1Cl 67042,N#Cc1ccc(C(=O)CCCCCN2CC(=O)N(CCP(=O)(O)O)C2=O)cc1 67043,Cn1c(NC(=O)CC(O)c2ccccc2)nc2cc(Br)c(Cl)cc12 67044,C(C(=O)NC1CCN(C(=O)C(C)SC(C)C)C1)(C(C)C)NC(C)=O 67045,CCC(CCOC)C(=O)NC(C)CCCC(=O)N1CC(F)(C2CC2)C1 67046,N1(C(CN(C(=O)OC)C)=O)CCN(C(=O)COC2CCCCC2)C2COCC12 67047,c1(OCCC(=O)N(C2CCN(C(C34COCC3C4)=O)CC2)CC)ccccc1O 67048,C#Cc1ccc(C(=O)NCC2CC2CNC(C2CC(C)(F)C2)=O)c(F)c1 67049,C(c1ccc(S(=O)(=O)N2CCCC2)cc1)=CC(=O)NCC1(CC(=O)O)CCOC1 67050,CC1(C(=O)NCc2cc(C(=O)NC3C(O)CC3O)on2)CCOC1 67051,C1(C(=O)NCC(CC)NC(c2scnc2C)=O)CCCNS1(=O)=O 67052,N1(C(C(C=C)(C)CC)=O)CC2CC(NC(c3ccc(Cl)cc3Cl)=O)C(C2)C1 67053,N1(C(CSCC(C)C)=O)CC2CCCC1(CNC(c1coc3c1COC3)=O)C2 67054,C(=O)(C#CC1(C)CCCO1)NC.C1(NC(CN(CCC)C)=O)CCCC1C 67055,C1(NC(Cc2c(C)cc(C)s2)=O)CCN(C(c2cnc(CC(C)C)s2)=O)C12CC2 67056,C1(CNC(c2c(C)oc(CO)c2)=O)CC2(CCN(C(C3(C)CC3(F)F)=O)C2)CO1 67057,c1(C(=O)NCC2N(C(C3C(C)C3C)=O)CC(C)(C)OC2)c(F)cc(F)c(F)c1F 67058,Cc1ncc(C(=O)N(CCCNC(C2(OC(=O)N)CC2)=O)C)cn1.C(C)(C)C 67059,c1(C(N(CC(C)NC(CCCCCC)=O)CC)=O)cc2cc(F)cc(F)c2[nH]1 67060,C1(NC(c2cc(Br)n3c2CCC3)=O)CN(C(=O)CCC2CC2)CC2(CC2)C1 67061,c1(C(=O)NCC=CC(=O)NCC2CCCOCC2)cnn2c1CCC2 67062,N1(C(Cc2cc(OC)c(F)cc2)=O)CC2CCC1CC2NC(C)=O 67063,O(N1CCC(NC(C2(C)CC(NC(=O)C(C)N=[N+]=[N-])C2)=O)CC1)CC 67064,CC1CCC(NC(=O)C(C2CCCO2)C2CC2)CN1C(=O)CC1COCCO1 67065,c1(CCC(=O)N(C2CN(C(C3(CC45CC(C4)C5)CCCC3)=O)C2)C)ccc(F)cc1 67066,N1(C(c2cc(C(C)=O)[nH]n2)=O)CCOC2CN(Cc3c(C)cc(Br)cc3C)CC12 67067,CC1(C)C(=O)NC2CCC(C(=O)NCC3CCN3C(c3cnc(Cl)[nH]3)=O)CC12 67068,C1(CNC(c2cn(C)cc2C(F)(F)F)=O)CCN(C(C2(CC3CC3)CC2)=O)C12CC2 67069,c1(C(C)NC(C2CCN(C(CC(C)O)=O)C2)=O)ccc(C(F)(F)F)cc1 67070,C1(OC)(OC)CC(C(=O)Nc2c(C(N3CCC(c4ncco4)C3)=O)n[nH]c2)C1 67071,CCS(=O)(=O)CCN=c1nc(N(C)C)[nH]c(=NC(C)c2cc(F)ccc2F)[nH]1 67072,c1(CC(=O)NC2C(NC(CC3CC(SC)C3)=O)CCC2)ccc(C)cc1 67073,N1(C(C2C(CC)C2)=O)CC2(COC(CNC(c3nnc(C)s3)=O)C2)C1 67074,S(=O)(=O)(c1ccc(C#N)c(NCCS(=O)(=O)CC2CC2)c1)N(C1C(C)CCC1)C 67075,C1(CNC(C2CC23CC3)=O)CN(C(=O)CC2CCCOCC2)CCC12CCOC2 67076,C1(NC(CCC(C)OC)=O)CN(C(=O)CCn2nc(C)cc2C)CC2CC12 67077,C1(NC(Cc2c(C)n(C)nc2)=O)CCCN(C(c2cc[n+]([O-])cc2)=O)C1C 67078,c1(OCc2cn(C3CCN(C(CC)=O)C3)nn2)cc(N)cc(S(C)(=O)=O)c1 67079,N1(C(C(C2(C)CC2)NC(=O)COCc2nnc(O)o2)=O)CCCC(C(N)=O)C1 67080,N1(C(C=Cc2c(C)coc2C)=O)CC2CN(C(=O)C(C)(F)F)CC(C1)O2 67081,c1(C(=O)NCC2(F)CN(C(=O)CCC3CC(F)(F)C3)C2)cncc([N+](=O)[O-])c1 67082,CN1C(=O)CN(CC(N2CC3CC2CC3CNC(=O)C(C)(C)C2CC2)=O)C1=O 67083,c1(C(=O)NC(C2(O)CN(C(=O)CN3CCC(C)(O)C3)C2)C)ccc(N(C)C)cn1 67084,C(=O)(CC(C)C(=O)OC)NCCN(C(C1CC1c1cc(F)ccc1F)=O)CC 67085,C12(O)CN(C1)C(=O)C(C)OCC2.C1(CC)(NC(C2(CSC)CC2)=O)CCC1 67086,C(=O)(C(C(C)(C)SC)C1CCCCO1)NC1C(CC)CN(C(=O)OC(C)(C)C)C1 67087,c1(CC)[nH]c(=N)sc1C(=O)NCC(O)CN(C)C(c1ccno1)=O 67088,c1(C(C)C(=O)NC2CCCN(C(=O)C=CCO)C2)ccc(S(=O)(=O)N(C)C)cc1 67089,N1(C(Cc2ccc(C)o2)=O)CC(C(N2CCC(C(F)F)CC2)=O)CC(C)C1 67090,c1(CC)ccc(C)cc1C(N1CCC(NC(=O)CCC2NC(=O)NC2=O)C1)=O 67091,Cc1c(Br)ccc(N2CCN(C(C34CC(C)(C3)OC4C)=O)CC2C)c1[N+](=O)[O-] 67092,Cc1cc2cc(C(=O)NCC(C)NC(C3(CO)CCCCC3)=O)c(Cl)cc2[nH]1 67093,C1(C(=O)NC2CCC(C(=O)NCC(C)CC3CCC3)C2)(OC)CCOC1 67094,C(=O)(CC1CC(C)(OC)C(=O)N1)N1C(CCC#C)CCC1.C1CC1 67095,N1(C(COCCCCC)=O)CC2(C1)C(NC(c1cc(C)oc1C)=O)CCS2(=O)=O 67096,C1(C)(OCC)CCN(C(C23C(NC(C4C5CCC(F)C45)=O)C4CC2C3C4)=O)CC1 67097,Cc1nc2sc1C(=O)NC2.C1(C(=O)Nc2nccs2)CCOC(C)C1 67098,N1(C(C2Cc3c[nH]cc3S2(=O)=O)=O)CCCCC2(C1)CN(C(C1CC1F)=O)C2 67099,C1(C(C(=O)N(CC=C)CCOC)NC(c2cnco2)=O)CC=CCC1 67100,c1(CC(=O)NCC#CCNC(c2c[nH]nc2[N+](=O)[O-])=O)ccc2ccccc2c1 67101,N1(C(C(C)OCOC)=O)CC(NC(=O)C=CCCC(C)C)CCC1C 67102,c1(N(C(C2(NC(C(CC3CCC3)OC)=O)CCSC2)=O)C2CC2)ccccc1C 67103,Cc1nc2cccc(C(=O)NC3COCC3CNC(C3CCN3S(C)(=O)=O)=O)c2[nH]1 67104,c1(C2C(NC(C3(F)CCN(Cc4cnc(Cl)nc4)C3)=O)C2)ccc(F)cc1 67105,c1(NCCCC(=O)Nc2nc(COC)nc(O)c2)ccc2c(c1)CCO2 67106,C1(COC)(C)CC(NC(=O)C(=O)NC(C)COc2ccc(C#N)cc2)C(O)C1.SC 67107,C1(CC(=O)NCC2N(C(C(F)=CCC)=O)CCC2)COC2CC1C2 67108,c1(OC)c(N(C)CC2CCCN(C(c3ccc(F)o3)=O)C2)ncnc1Cl 67109,N1(C(c2n(OC)cnc2C)=O)CCC2(CC1)CC(CNC(=O)C(F)C1CCC1)C2 67110,S(=O)(=O)(CCCCCl)N1C(NC(C2CC(N(C)C)C2)=O)CC(F)C1 67111,C12(CNC(CC3C(C)CCN(C(C4(O)CC4)=O)C3)=O)CCC(CC1)C2(C)C 67112,C=C1Cn2c(C(=O)NCC3CC4CN(C(=O)C=CSC)CC34)nnc2S1 67113,C1(NC(c2c(OC)n(C)nc2)=O)COC2(CCN(C(=O)CCC3CC3)CC2)C1 67114,N1(C(C(C)OCc2ccccc2)=O)CC(C)N(C(=O)CC(F)(F)C(C)C)CC1C 67115,CC1C(C(=O)NC(=O)CNCC(C)(C)C)CCCN1c1ccc(C(F)(F)F)cn1 67116,N1(C(CC(=O)N(C)C)=O)CC2(CC(CNC(C3(C#N)CC3)=O)C2)C1 67117,N(C(=NCCCCC(C)(F)F)NC(c1cnnn1C)C)C(CC)CC 67118,C1(CNC(CC)(Cc2ccccc2)c2nnnn2C)CC(C2CC2)=NO1 67119,CC(C)C(O)CNC(=O)C(CC1CC1)NC(=O)CSC1CC1 67120,c1(OCC=C)ccc(Cl)c(NC(C2CCN2CC2CCCC2)=O)n1 67121,N(C1CN(C(=O)C2=CCCOC2)Cc2ccccc21)C(Cn1c(C)nnn1)=O 67122,CC1CCCC(CC(=O)NCC(C2CCCCC2)NC(C2CC(F)C2)=O)C1 67123,CC(C(=O)NCCCCC1CN(C(c2ccc(F)c(N)c2)=O)C1)C(F)(F)F 67124,c1(N2CCC(NC(C(COC)OC)=O)C(O)C2)cc(C#N)nc(C2CC2)n1 67125,c1(C(N2CCN(C(CCCOC)=O)C(C)CC2)=O)cc2ccc(F)c(F)c2o1 67126,C1(c2cn(C(C)C)nc2)CN(C(=O)C(c2cnn(C3CC3)c2Cl)=O)CCO1 67127,C1(NC(CCC(C)NC(c2c(C)ncs2)=O)=O)CN(C)CC1(F)F 67128,C(=O)(CCN(CCO)C(C1(C)CC1)=O)NC(C1C(C(=O)OC)C1)C 67129,C1(CCC)CN(C(c2cnc(=N)[nH]c2)=O)CC1C(=O)NC1(C)CCSC1 67130,C1(COC)(NC(c2coc(C3CCC3)n2)=O)CCN(C(C2COC2)=O)C1 67131,Cc1cccnc1C(C(C)(C)C)NC(=O)C(=O)NC12CC(c3ccccc3)(C1)C2 67132,C(C)(CCCC(=O)NCCCC(F)F)NC(Cc1c(C)scc1)=O 67133,C1(NC(C2(C)CCCCCC2)c2n(CCOCC)nnn2)CCCC(C)(C)C1 67134,N1(C(CNC(CCC(C)C)=O)=O)CCC(NC(=O)CC2CNC(=O)C2)C12CCC2 67135,c1(C(=O)NCC2N(C(CN(C)C(c3ccco3)=O)=O)CCC2)c(N)cccc1Cl 67136,N1(C(Cc2c(C)occ2)=O)CC2CN(C(=O)COc3ccc(F)cc3)CC2(C)C1 67137,c1(C(=O)NC2C(C(N3CCN(C)C(=O)C3)=O)C2)ccc2nc(Br)sc2c1 67138,C1(C(=O)NCC(CCC)O)CCN(C(=O)C#CC2(C)COC2)C12CCC2 67139,C1(=CC(=O)NCC(CN(C(C(CC)O)=O)C)O)CC2CCC(C1)N2C 67140,N(C(=NCCCNCC(F)(F)F)NCC1CCCCS1)CC(C)(C)C 67141,CC1=C(C(=O)NC2CC3CC(NC(c4cc(O)nc(C)n4)=O)CC23)CCCC1 67142,CC1CCCN(C(=O)CC2(C)CCCO2)C1.c12ccccc1C(=O)N2 67143,c1(C(N2CC(CNC(c3n(CC)nnc3C)=O)OCC2)=O)c[nH]c(C)cc1=O 67144,Cc1c(C(N2CC3(CC3)CC2CNC(=O)CCOC(C)C)=O)sc2ccccc12 67145,C(CC(C(=O)N1CC(O)C(O)C1)NC(=O)CC1CCCN1C)SC 67146,c1(C(CC)NC(C)C(=O)NC(C)C)nc(C(F)(F)F)n[nH]1 67147,C1(C)(CNC(CC2C=NN(C)C2=O)=O)CN(c2ccnc(Cl)n2)CCO1 67148,CC1CCN(C(=O)CCc2c(Cl)cncc2Cl)CC1NC(=O)C=CC1CC1 67149,c1(C(=O)NCC(C)NC(c2ccc(F)o2)=O)ccnc(O)c1Br 67150,C1(CNC(C(C)OC)=O)CCCC1NC(C1CCC2CC12)=O 67151,c1(C(=O)NCC23CCC(CC2)N(C(C2CC2(Cl)Cl)=O)C3)ccc(F)cc1[N+](=O)[O-] 67152,c1(C(=O)NC(C(C)NC(CC(C)C)=O)C)cc2c(cc1[N+](=O)[O-])OCCCO2 67153,C1(CNC(CC=CC)=O)CC(NC(c2cn(C)cn2)=O)C12CCC2 67154,N1(C(C2CCOCC2)=O)CCC(NC(C2(C(C3CCCO3)=O)CC2)=O)C(F)C1 67155,C(=O)(C1=CCCOCC1)N(C)CC1(CNC(C(N2CCCC(C)C2)=O)=O)CC1 67156,N1(C(C2(C=C)CC2)=O)CCCC2(CCN(C(c3ccc4nonc4c3)=O)C2)C1 67157,C1(NC(c2ccc(Br)cc2Br)=O)CN(S(=O)(=O)C2CC2)CC1(F)F 67158,c1(CNC(=O)Nc2nc(Cc3ccccc3)ns2)cc(Cl)ccc1Br 67159,C(=O)(C(F)C(CC)CC)N1CCN(CC(C)NC(c2nc(CC)oc2)=O)CC1 67160,C(=O)(C1=CS(=O)(=O)CCC1)NC(C)CCCCNC(=O)CC1C=CCCC1 67161,n1(CC)cnc2nc(N3CCN(C(C)C(F)(F)F)CC3)nc(NCC(C)F)c12 67162,CCC(CCCC(=O)N1CCOC(C)(C)C1)NC(C1CC(O)C(F)C1)=O 67163,CCS(=O)(=O)CC(=O)N(CC(C)(C)NC(=O)CCCC(=O)c1ccccc1)C 67164,CCC(CNC(=O)CN(C(=O)CCC(=O)N(C)C)C1CC(C#N)C1)C(C)C 67165,C1(CNC(C(C)(O)CCc2ccccc2)=O)CC2CCC1N(C(=O)CCCF)C2 67166,C1(NC(CSCC(=O)OC(C)(C)C)=O)CCCN(Cc2ccc(O)c(O)c2)CC1 67167,C(=O)(C(C)(C)CC(F)(F)F)NC(C(C)NC(CCc1onc(CC)n1)=O)C 67168,c1(C(=O)NC2C(C)(C)CN(C(c3occc3C3CC3)=O)C2)ccnc2c1CCN2 67169,C(=O)(CN=c1[nH]c2ccccc2s1)NC1CC(C)(NC(C2CC23CCOC3)=O)C1 67170,N1(C2CN(C(=O)NCC(c3ccco3)SC)C2)CCCS1(=O)=O 67171,c1(OC)ccc(C(C(=O)NC2CCOC2=O)OC)cc1Cl 67172,c1(NC(C(F)OC)=O)cccc(NC(c2cn(CCO)nn2)=O)c1 67173,C1(C(C)C)CN(C(=O)CC(C)c2cnn(C)c2)CCN1C(c1ccoc1Cl)=O 67174,C1(C(N(CC(C)NC(C2COC(=O)N2)=O)C)=O)CCCN1C(c1ccccc1)=O 67175,C(=O)(C(F)C(C)(C)O)N(CC(CC)NC(c1cc(N(C)C)ccc1N)=O)C 67176,CN1CCC(C(=O)NC2(CNC(C3CCC(F)C3)=O)CCC2)CC1=O 67177,N1(C(CCCCCOC(C)C)=O)CC(C#N)(S(C)(=O)=O)C1 67178,C(c1ccc(F)nc1)=CC(=O)NCC(CNC(c1c(C)nc(N(C)C)s1)=O)C 67179,C1(NC(c2ccc(CNC(C)=O)s2)=O)CCCN(C(C2COC(=O)O2)=O)CC1 67180,C(=O)(CC(C)(C)CNC(c1cc(Cl)n[nH]1)=O)NCC(C)CC1CCC1 67181,C(=O)(C(C)(O)C(F)(F)F)NCCC1CN(C(C2CC(OC)C(OC)C2)=O)C1 67182,C(CCC(CCC)N(C(C=CCC)=O)C(C)C)NC(c1n[nH]c2c1CCC2)=O 67183,C1(CNC(C(C)SCC)=O)(CO)CCCN(C(C2CCCN2C(C)=O)=O)C1 67184,C(=O)(CC1=CCOCC1)N1CC(C(=O)Nc2cc(C)c(O)cc2)C(C)(C)C1 67185,Cn1ccc(=O)c(C(=O)NCCCN2CCN(C(C3CCS(=O)(=O)C3)=O)CC2)c1 67186,Cc1cc2ccccc2nc1C(N1CC2CCN(C(c3csnn3)=O)CC2C1)=O 67187,C(CCCCC(=O)N1CC(NC(=O)CSC)CC(C)C1)OCC 67188,c1(C(NNC(c2cccc(CS(C)=O)c2)=O)=O)cc2n(n1)CC(O)CO2 67189,CC1(C)CC(CC(=O)NC(CNC(C2(CO)CCCO2)=O)C2CC2)CO1 67190,N1(C(CCS(=O)(=O)NC)=O)CCC2(CC1)CC2NC(=O)C(c1cccc(C)c1)F 67191,c1(C(=O)OC)cc(NC(c2sc(NC(C3CCCO3)=O)nc2C)=O)c(C)cc1Br 67192,c1(C(N2CC(C)OC(CCNC(=O)C(C)(C)C(N)=O)C2)=O)cc(C#N)ccc1F 67193,c1(C(=O)NC2(C)CCN(C(CC3ON=C(CC)C3)=O)C2)cc(C)nc2ccnn12 67194,N1(C(c2c(C)nco2)=O)CCCC(O)(CN(C(=O)C(C)CN2CCCCC2)C)C1 67195,C1(C(=O)NC(C(=O)NC2CC(O)C2)c2cccs2)CN2CCCC1C2 67196,CC(CC1CCCO1)N=c1[nH]c(=NC(C)c2cn(C)cn2)[nH]c2c1CCCCC2 67197,Cn1ccc(-n2cc(CN(CCC(=O)O)C(=O)CO)nn2)cc1=O 67198,C1(C(=O)NCCCN(C(CC(=C=C)C)=O)CC)CCOC1C(=C)C 67199,c1(C(=O)Nc2cc(Br)ccc2CO)cccn2c(-c3ccnc(O)c3)cnc12 67200,C1(C(=O)NC2CN(C(CC(C)n3ccnc3)=O)C2)CC(=O)c2ccccc2O1 67201,c1(CN2CC3CN(C(=O)CCc4ccccn4)CC32)ccc(I)c(F)c1F 67202,C(=O)(C#CC1(C)CCCO1)NC1CN(C(C(CC(C)C)N(C)C)=O)CC(F)C1 67203,CCC(C)C(C)(O)CNC(C1CCOCC1NC(=O)C(CC(C)C)OC)=O 67204,N1(CCN(C(CN(C(=O)C(C)NCC)CCC)=O)CC)CCCCC1 67205,CC1CCCC(O)(CNC(C2CC(n3cc(CC4CCOC4)nn3)C2)=O)C1 67206,N1(CCCCCCNC(C(CCC)C)=O)CCCC(C)(N(C)C)C1 67207,c12ncccc1C(=O)NC2.C(CO)(C(=O)NCCCCOC(C)C)OC 67208,N1(C(c2c(CC)ocn2)=O)CC(NC(c2cc(O)ncn2)=O)C2CCCCC12 67209,Cc1ccc(Cl)c(C(=O)NCC2CCN(C(C34CCC(CC3)C4)=O)CC2C)c1N 67210,C1(OC)CC(CNC(=O)CC(C)(C)C)N(C(=O)CCn2cncn2)C1 67211,CCCC(O)C(CO)NC(=O)CC1(NC(C2CCCC(=O)CC2)=O)CC1 67212,C(=O)(C(F)C(C)(C)O)NCCC(C)NC(C1CCN(CC(F)(F)F)C1)=O 67213,N1(CCC)CCCCC1C(=O)N(C)CCC1CCCCN1C(c1cnc(C)s1)=O 67214,N(C(=NCc1cccs1)NC1CC12CCCC2)C(CC)C1CC1 67215,CCCC(CCO)NC(=O)CC1(N(C(=O)C(CC)OC)C)CC1 67216,c1(OC)cc(C(=O)NCCc2ccccc2O)cc(C)c1 67217,c1(CCC(=O)NC2C(OC)CN(C(=O)COC3CCC3)C2)ccc(Cl)cc1Cl 67218,C12(CNC(C(C(C)O)C)=O)CC(NC(=O)CC3CC3)(C1)C1(CCOCC1)O2 67219,N#CC1CN(C(C2NCC23CCOCC3)=O)CCC1(F)F 67220,C1(NC(=O)C=C2CCCCC2)(CF)CCN(C(=O)C(c2cccc(F)c2)O)C1 67221,N1(C(C2(CCCC)CC2)=O)CCCC(C2CCCN(C(C3C4COCC34)=O)C2)C1 67222,N1(C(CP(C)(C)=O)=O)CCOCC(NC(c2ccccc2Cl)=O)C1 67223,N(C(=NCCC1CC(F)C1)NCC(N1CCCCC1)=O)C1C(C)C1 67224,CS(=O)(=O)c1cnn(CC(=O)NC2CCCC(NC(c3cnco3)=O)CC2)c1 67225,c1(N(c2ccccc2)CCN2CCC(OCCN(C)C)C2)cncc(Cl)n1 67226,C1(C(N2C(CNC(c3cnco3)=O)CCC2)=O)CC(F)(F)C12CCC2 67227,Cc1cc(Cn2cc(-c3cnn(C(C)C)c3)nn2)cc(C(F)F)c1 67228,CCCC(CC)CC(=O)N1CC2CCC(C1)N2C(c1nc(Br)c[nH]1)=O 67229,C1(CNC(C2(NC(C)C)CC2)=O)CN(C(=O)C(C)C(F)F)CC1(F)F 67230,N1(C(c2c(CC)cno2)=O)CCC2CC2C1C(=O)N1CCC(C(=O)OC)O1 67231,C1(NC(c2c(C)nc(OC)s2)=O)CN(C(=O)CN(C)C)CCC1CO 67232,C1(COC)CC(CNC(C2CC2C(C)(C)C)=O)N(C(=O)COCC(C)C)C1 67233,c1(CN(C)C(C23COCC(C2)C3)=O)ccccc1CNC(C1(F)CC=CCC1)=O 67234,c1(C(N2CCC(CNC(c3on(C)c(=O)c3)=O)C23CC3)=O)nnn2c1COCC2 67235,C(=O)(C(C)(C)C(C)(C)C)NC1CN(C(CC2C(C(=O)OCC)C2)=O)C1 67236,Nc1ncc(C(N2CC(CNC(c3ccco3)=O)C2)=O)cc1Br 67237,c1(C(=O)NC(CNC(CC2CC(=C)C2)=O)C2CCC2)nccc(N)c1Cl 67238,c1(C(=O)NC2CN(C(C3CC4CCC3C4)=O)CC2O)cc(F)cc2nccnc12 67239,Cc1c(C(=O)NCC2CC3CC2CN3C(=O)CC(C)(C)O)cncc1F 67240,C1(NC(=O)CC2(C#N)CCC2)(NCCC2CN(C(C(=O)N(C)C)=O)C2)CCSC1 67241,C(=O)(C(C)(C)CNC(C1CCCCO1)=O)N(CCO)CC 67242,C1(CNC(c2ccc(OC)o2)=O)CCC(CNC(=O)C(O)C2CC2)CC1 67243,Cc1cc(Cl)c(Cl)cc1C(N1CCCCC1CNC(c1cn(C2CC2)nn1)=O)=O 67244,C1(C(N2CCC(N(C(=O)CC(C)(C)C3CC3)CCC)CC2)=O)CC(C2CCC2)C1 67245,c1(COC)ccoc1C(=O)NC(C)(CNC(=O)CCOCCOC)CC 67246,Cc1[nH]c2ccccc2c1C(N1CCC2(C1)CN(C(C1C(F)(F)C13CC3)=O)C2)=O 67247,C=CCC(C(=O)N1CC(CNC(c2cc(Br)cnc2C)=O)(OC)C1)C(C)C 67248,c1(CNC2CN(C(CCc3c(C)noc3C)=O)CC2C)cc(F)cc(C#N)c1 67249,c1(N(CCNC(C2CC2C(=O)OC)=O)CC)cc(SC)nc(C)n1 67250,N1(C(C(C)N2CCCC2)=O)CCCCC(CNC(=O)CN(c2ncccn2)C)C1 67251,N1(C(CC=C)=O)CC(CN(C)C(c2cc(Br)ccc2C)=O)C2(CC2)C1 67252,C1(N(C(c2cc(OC)ns2)=O)C)CCN(C(c2cccc(C)c2O)=O)CC12CC2 67253,C1(CNC(C2(OCC)CCOC2)=O)(CNC(=O)CC(F)F)CC12CCC2 67254,C(CCC(C)(C)C(=O)NCCC1CCC(C)C1)NC(c1c(=O)cc(C)[nH]c1)=O 67255,N1(C(C=CC(=O)N(C)C)=O)CCCC(N(C(=O)C(F)Cc2ccccc2)C)C1 67256,c12ccccc1CCn1c(SCC)nnc1N1CCC(CC1)C2.NC 67257,CC(C)CCC(C(=O)NCc1ccnc(F)c1F)NC(c1cnn[nH]1)=O 67258,CC1CN(C(C2(O)CCC2)=O)CC1NC(c1cc(C2CCCC2)nn1C)=O 67259,c1(C(=O)NC2CCN(C(c3cc(C)c(C)o3)=O)CC2C)cccc2c(C)csc12 67260,N1(C(CCOC(C)C)=O)CCC2CCN(C(c3cc(C(F)(F)F)n(C)n3)=O)C2C1 67261,c1(CNC(=O)Cc2cccc(C3CC3)c2)ncc([N+](=O)[O-])cn1 67262,c1(OC)cccc(CN2CCC(CNC(c3csc(C)n3)=O)C2)n1 67263,c1(C(=O)NCC(C)(C2CCC2)NC(c2cscn2)=O)ccc(-n2ccnn2)cc1 67264,n1(CC(=O)NCC2(C)CCN(C(C3CC(S(C)(=O)=O)C3)=O)C2)ncc(O)nc1=O 67265,C(CCNC(c1cnc(COC)s1)=O)(C(C)C)NC(c1ccc(CCC)[nH]1)=O 67266,Cc1csc2ccc(C(=O)NC(C)CCCNC(C3CCC(O)C3)=O)cc12 67267,C(N=c1cc(NCc2cocn2)nc(C2CC2)[nH]1)c1nccc(CC)c1 67268,C1(C(=O)NC2C3CCN(C(C4CN(C)C4)=O)CCC32)COc2ccc(F)cc2C1 67269,C1(C(=O)NCCCN(C(=O)CN(C)C(=O)C2CC2)CC)CC=CCC1 67270,C(CC(C(C)(C)C)NC(C1CC(C(F)F)C1)=O)N(C)C(c1ccnc(CO)c1)=O 67271,N1(C(C(C)SC(C)C)=O)CC2(CCCN(C(C3CC(=O)NC(=O)C3)=O)C2)C1 67272,Cc1ccc(NC(=O)NC2CCC(C)(C(C)C)C2)cc1C(=O)N(C)C 67273,Cc1nc(C(N2CCC(CCC(C)(C)C)(NC(C3C4CCC34)=O)C2)=O)oc1C 67274,C#Cc1ccc(C(=O)NCCC(CNC(=O)CN2CCC(=O)CC2)OC)cc1 67275,C1(NC(c2cn(CC=C)nn2)=O)CCC(C(=O)NCc2cc(C)[nH]n2)CC1 67276,Cc1cc(F)c(F)cc1C(N1CC2CC2(C(=O)Nc2ncc(Br)nc2Cl)C1)=O 67277,c1(CC)cc([N+](=O)[O-])ccc1C(=O)NC1(COC)CCN(C(=O)C(CC)CO)C1 67278,C1(CC)CN(C(=O)Cc2ccoc2)CCC1NC(c1ccsc1C#N)=O 67279,N1(C(CCS(=O)(=O)N(C)C)=O)CCOC2(C1)CN(C(C1CC13CCOC3)=O)C2 67280,c1(C(N(CC(O)CN(C)C(C2CCCN2N=O)=O)C)=O)ccn(C)c(=O)c1O 67281,C1(CC(=O)NCC(CO)NC(=O)CNc2ccccc2)CCCCCC1 67282,Cc1cccc(C(N2CC3CC3(C(=O)Nc3ncc(Br)cc3Cl)C2)=O)c1F 67283,C1(NC(C(C)N(CCN(C)C)C)=O)CC2(CC2)CN1C(=O)CC1(C)CCCCC1 67284,N1(C(CCN(C)CC)=O)CCC2(CCCCN(C(C3(Cl)CC3(C)C)=O)C2)C1 67285,N1(C(CCc2cn(Cc3nc(C)sc3C)nn2)=O)CC(C)(C)OC2(CCOC2)C1 67286,c1(C(N2CC3CN(C(C(C)(C)C(F)F)=O)CC3C2)=O)nc2ccc(Cl)nn2n1 67287,N1(C(C2C(C#N)C2)=O)CC2CS(=O)(=O)CC2(NC(=O)Cc2ccc(F)cc2F)C1 67288,N1(C(C2C(C)OCC2)=O)C2CCC1CN(C(=O)C(c1ccccn1)N)C2 67289,c1(OC)c(C(=O)NC2(C)CN(C(C3(C)CC3(F)F)=O)C2)ccnc1Cl 67290,C1(NC(Cn2c(C)nnn2)=O)CC2CC(C1)N(C(=O)CC1CC(F)(F)C1)C2 67291,Cc1cc(C(F)(F)C(=O)N(CC(O)CNC(C2CCC(C)O2)=O)C)cc(C)c1 67292,C1(C(=O)NC2CC3CC(NC(c4cc(C)oc4)=O)C2C3)CCC(=C(F)F)CC1 67293,c1(C(=O)NCC2(C(=O)NNC(=O)OC(C)(C)C)C(C)C2)nccc2[nH]ccc12 67294,c1(OC)ccc2c(c1)C(O)CCN2C(c1ccc2[nH]c(=N)sc2c1)=O 67295,c1(C(=O)NC2(CCNC(CCc3cn(C)nc3)=O)CC2)cnc2[nH]ccc2n1 67296,C(CN=C(NCCOc1ccccc1)NCCc1cnccn1)C1CC(F)C1 67297,C1(CNC(C(Cc2ccccc2)N(C)C)=O)CN(C(=O)C=C2CCC2)CCO1 67298,CC(C)C(C)C(C)CC(=O)NC1(CF)CCN(C(=O)CC2(CO)CCOCC2)C1 67299,c1(NC)cccc(C(=O)NCCCCOC)n1.N12CC(O)(C1)C(F)C2=O 67300,C(C(N=c1[nH]c(=NCc2cnn(C)c2Br)[nH]c2c1CCCCC2)C1CC1)OC 67301,c1(C(=O)NC2CCN(C(c3n(CC)nnc3C)=O)C2)cc(C)cc(Br)c1O 67302,c1(C(N2CC(C(C)NC(C(CCC)(C)C)=O)C2)=O)cnc(O)c2ccccc12 67303,N1(C(C(=O)NCC2(C)C(C)C2)=O)CCC2(CC1)CC(=O)c1ccccc1O2 67304,c1(CCC)c(C(N2CCC2C(N)=O)=O)nnn1-c1cccc(C(F)(F)F)c1 67305,c1(C(C(=O)NC2CC(N(C(c3ccc(C#C)o3)=O)C)C2)(F)F)cccc(Cl)c1F 67306,C1(C)(CC)CC(C(=O)NCC(C)(C)OCC(N2CC(COC)C2)=O)C1 67307,c1(C(N2CC(C)C(NCc3nc(Br)cs3)C2)=O)ccc2sccc2c1 67308,N1(C(CSCC=C)=O)CC2=C(C1)CN(C(c1cc(C)sc1Br)=O)C2 67309,CC(CCO)C(=O)N1CCCCC1Cc1cn(-c2cccc(F)n2)nn1 67310,C1(CC(=O)NCC2C(C(=O)NC(C=C)CC)C2)CCCCO1 67311,N1(C(c2cc(C)[nH]n2)=O)CC2CCC(NC(c3cnnc(C4CC4)c3)=O)CC2C1 67312,C1(C(=O)NC2(CC(=O)NC3CCCC(CO)C3)CCC2)(OC)CCCCC1 67313,c1(C2CC(C(N(C(CNC(C(C)Cn3cccn3)=O)C)C)=O)C2)ccc(O)cc1 67314,N1(C(C2CC(OCC)C2)=O)CC2CCN(C(c3ccc(CC#N)cc3)=O)C(C2)C1 67315,O=C(C1=NOC2(CCC2)C1)N1CC(C2CC2C(=O)NCC23CCC(CC2)CC3)C1 67316,c1(C(N2CCC3(N(C(C4C(C(C)C)C4)=O)CCC3)C2)=O)ccc2nc(=N)[nH]n2c1 67317,C(c1cncnc1O)=CC(N1C(CNC(C(CC)n2ccnc2)=O)COCC1)=O 67318,C1(NC(c2nc(CCC)oc2)=O)CC(N=c2[nH]c3cccnc3s2)C1 67319,C12(C(=O)NC(C(=O)NCC(C)(C)O)CC3CCOCC3)CCC(CC1)C2 67320,CCS(=O)c1ccccc1C(=O)NC(C)CN(C)C(c1cc(OC)n[nH]1)=O 67321,c1(C(N2CCC(CNC(C(c3cccc(Cl)c3)CC)=O)C2)=O)ccc(F)c(N)c1 67322,c1(CC(N2CCCC(NC(C(C)OCC)=O)C2)=O)ccc2nsnc2c1 67323,Cc1cc(Cl)cc(C(=O)NC2(C)CC(NC(c3cn(CC(N)=O)nn3)=O)C2)c1N 67324,C=CCC(C)C(=O)NCC=CC(=O)NCC1(CC)CCCO1 67325,CCC(O)C(C)(C)C(=O)NCC1(O)CC(C(=O)N(CCC(F)(F)F)C)C1 67326,C(=O)(CC(C)(C)C(F)F)NCC1N(C(c2ncn(CC)n2)=O)CCN(C)C1 67327,Cc1c(C(=O)NCC2CN(C(=O)C=CC3CC3)CC2C)noc1-c1ccccc1 67328,C1(CNC(c2c(C)cc(C)[nH]2)=O)CC2(CC2)CN1C(C1CC1c1nccn1C)=O 67329,c1(C(=O)NCC23CC(NC(C(C)OCC4CC4)=O)(C2)C3)ccc2nccn2c1 67330,C1(C(=O)NCc2ncn(C)c2)CCCN1NC(=O)C1CCC1(F)F 67331,c1(CC(=O)NC(C)(C)CNC(C23CCCC2C3Br)=O)c[nH]c2cnccc12 67332,N1(C(c2c(NC)cccc2)=O)CCC2C(CCCN2C(C2(C)CCCC2)=O)C1 67333,CC1(F)CCC(C(N2CCCC2Cc2cn(C3CCC(F)(F)CC3)nn2)=O)CC1 67334,C1(C(=O)NCCN(CCC)C(c2cc(C)ccc2OC)=O)CCC2C1C2(F)F 67335,CC1CN(C(C2OCCCC2(C)C)=O)C(C)CN1C(=O)Cn1cnnc1O 67336,N12CCC(COC)(C1)C(=O)OC(CCC)C2.C(C)(C)(C)OC(=O)NC 67337,c1(NC2CCC(NC(C(C3CCOC3)OC)=O)CC2)ccc(F)cc1[N+](=O)[O-] 67338,C1(NC(C(CN(C)C)O)=O)CN(C(c2cc(F)c[nH]2)=O)CCC1CO 67339,C(=O)(C1CCCc2cc(O)ccc21)NCCCNC(C1CCN(CC(C)C)C1)=O 67340,N1(Cc2cn(-c3n(C)nnc3)nn2)CCN(C(N)=O)CC1.C1CC(=O)N1 67341,C1(C(C)C)CN(C(C)=O)CCC1N(C(C1(C2CC2)CC1)=O)Cc1ccccc1 67342,c1(CNc2nc(-c3ccc(OCCC)nc3)sc2)ccc2[nH]c(C)cc2c1 67343,N1(C(c2c(C)cn(C)n2)=O)CCC(O)(C(C)NC(=O)C(C)n2ccnc2)CC1 67344,C(=O)(CCCCC(C)(C)C)N(CC(C(=O)NCc1c(C)ccs1)C)C 67345,C=CCC(CC)C(=O)NCC(c1ccccc1)NC(C1(O)CC(C)(C)C1)=O 67346,C1(CNC(CC2N(CC)CCC2)=O)CCN(C(=O)CCCCOC)CC1(F)F 67347,CN1CCC2CCN(C(=O)C(O)CCCNC(c3ccc(F)c(F)c3)=O)C2C1 67348,N1(C(Cn2cc(CCCC=C)nn2)=O)CCC(O)C1CC 67349,C(=O)(CCC(=O)N(C)C)N(C1CCN(C(C23CC(CC(F)F)(C2)C3)=O)C1)CCC 67350,C=CCCCCC(=O)NC(CC(=C)C)C(=O)NCCc1cn(C)nn1 67351,C(C(=O)N1CC(F)(F)C1C1CC1)(C(C)(C)C)n1cc(-c2c(C)nccc2)nn1 67352,Cc1c(Br)ccc(F)c1C(=O)NC(C)CCNC(=O)C(O)c1ccco1 67353,N1(C(CC2CC(=O)NC2=O)=O)CC(NC(=O)Cc2ccon2)CC(F)C1 67354,O=C1CNC(=O)C(CC(=O)NCCN2CCN(C(=O)CNC=O)CC2)N1 67355,C1(C)(C(N2CC(SC)C(n3cc(CC4CCOC4)nn3)C2)=O)CCCCNC1=O 67356,C(CC(C)C)(C(=O)NC1(CF)CCN(C(c2cscc2C(F)(F)F)=O)C1)OC 67357,C1(OC)CN(C(C2CCN(C3COC3)CC2)=O)CC1NC(c1cnco1)=O 67358,N1(C(C2CC(F)CN2C(=O)Cc2ccc(Cl)c(F)c2)=O)CCCC2CCCCC12 67359,c1(C(=O)Nc2nc(C(=O)NC3CCCC3)cs2)ccc2nc(Br)sc2c1 67360,C(=O)(C(F)C(C)(F)F)NCc1ccc(C(N(CC)CC2CCOC2)=O)s1 67361,C1(C(N(C2CN(C(C3(C#N)CCCOC3)=O)C2)C)=O)C2CC3CC(C2)CC1C3 67362,C1(NC(C(N2CCCCCC2)C)=O)CCCC(NC(=O)OC(C)(C)C)C1 67363,C12(CC(N3CCC4CCC34)=O)CCC1CN(C(c1cccc(CO)n1)=O)C2 67364,C1(C)(C(=O)NCC2(O)CC(C)(C)C2)CCCN(C(=O)Cn2cnc(C#N)n2)C1 67365,c1(NC(C2N(C(CN3C(C)CCCC3)=O)CC(F)C2)=O)c(F)cccc1Cl 67366,C(=O)(C(F)(F)Cn1cc(C(N2CCNCC2)C)nn1)Nc1ccc(OCC)cn1 67367,C(=O)(CN=c1ccc(Cl)n[nH]1)N1CC(CNC(c2ccc(C)o2)=O)CC12CCC2 67368,CCC(C)C(C(=O)NCCc1cnc(C)o1)N(C(=O)CCCC1CC1C)C 67369,C#CCC(C)(C(=O)NCC(C)N(C)C)NC(=O)CC1CC(=O)NC1=O 67370,c1(C(N(C2CCN(C(C(CC)C(C)O)=O)C2)C)=O)cc(OC)cc2ccccc12 67371,C1(C2CCN(C(C3CCCOCC3)=O)C2)(NC(c2cccc(CC#N)c2)=O)CC1 67372,C1(CNC(CCCC=C)=O)CN(C(=O)CN2CCC(=O)NC2=O)CC1(C)C 67373,c1(C(N2CC(CCNC(=O)CC3CC3(C)C)(OC)C2)=O)c(F)cncc1Cl 67374,C1(C(=O)NC2CCC(NC(c3c(C)scn3)=O)CC2)CC2CSCC(C1)C2 67375,N(C(=NCCC1CC1)N(C)Cc1cc(F)c(F)c(F)c1)CCC1CCCC(C)C1 67376,C#CC1(C(N2CCCC2)=O)CCN(C(c2nn(C)cc2SC)=O)C1 67377,Cc1c(Br)noc1C(=O)NCC1CCN1C(c1cc(Br)sn1)=O 67378,C(=O)(C1=CC2CCC(C1)C2)N1CC(C(=O)NC2COCC2O)C(F)(F)C1 67379,c1(C(=O)NCC(CNC(c2cc(CCC)nn2C)=O)(C)C)cc2occc2[nH]1 67380,N1(C(C(C)CC(N)=O)=O)CCCCCC(Nc2ncnc(C(C)(C)C)n2)C1 67381,N1(C(CC(=C)C)=O)CCCC(CCCCNC(C2(Cl)CC2(F)F)=O)C1 67382,c1(SC)c(C(=O)NC(C2CCCN2C(=O)C(C)O)C)cccc1F 67383,c1(NC(C(N2CCN(C(c3cc(C)c(C)o3)=O)CC2)C)=O)ccn2nccc2n1 67384,CC(=O)C(C)CC(C)C(=O)N(C1CC(NC(=O)OC(C)(C)C)C1)C 67385,c1(NCC(C2CC2)NC(C2(OCC)CCCCC2)=O)ncc(Cl)c(C)c1C#N 67386,c1(N2CCCC(CNC(C)=O)C2)ccc(S(=O)(=O)N(CCCCO)C)c(Cl)c1 67387,CCS(=O)(=O)CC(=O)N1CCC(F)(C(N2CCCC2c2nn[nH]n2)=O)C1 67388,N1(C(C(CCC)N(C)C)=O)CC2CCCC1(CNC(c1cn(C)nc1C)=O)C2 67389,N1(C(c2ccnc(Cl)c2O)=O)CC2(C1)CN(C(C13CC(CCO1)C3)=O)CC2CO 67390,Nc1c(C(=O)NC2CC2NC(C2CCC(N(C)C)CC2)=O)cccc1[N+](=O)[O-] 67391,c1(CC2(C(C)Nc3ccc(C)cc3)CCC2)c(C)nn(-c2ccc(Cl)cc2)c1C 67392,C=C(C)C(O)CC(=O)NCC1CN(C(=O)CCCc2sccc2C)CCO1 67393,c1(C(=O)NCC2CC2NC(c2cc(F)c(F)cc2Cl)=O)cc2n(n1)CCNC2=O 67394,c1(C(N2CCN(C(c3ccon3)=O)C3C2C3)=O)nc2ncccn2n1 67395,c1(NC(C2(CNc3c(C)cncn3)CC2)=O)cc(C(F)(F)F)ccc1I 67396,C(=O)(CC(CC)C(F)F)NC(CCC#C)C(=O)NC(C)Cc1ncn(C)n1 67397,C(=O)(C(F)CCC(C)(C)C)NCC1(OC)CCN(C(C(CC)F)=O)C1 67398,C#CCC(CC(F)F)C(=O)NC(CCC)CC(=O)NC1(C(F)(F)F)CC1 67399,N1(C(c2cnc(N(C)C)o2)=O)C(C(=O)Nc2sncc2C#N)CC2CC12 67400,CN(C(=NCC1C=CCCCC1)NCc1ccccc1)CCC1CCCCO1 67401,c1(C(=O)NCC(CC)(C)NC(C2(OC)CCC2)=O)n[nH]c2c(C)cccc12 67402,c1(C(N(C2CCC23CN(C(=O)CCC2CC2(C)C)C3)C)=O)[nH]nc2ncccc12 67403,c1(-c2nc(C(C3CC3)OC)nn2Cc2ccc(F)c(CO)c2)cnn2c1CCCC2 67404,C(=O)(C(C)(CC#C)NC(=O)C(=O)CCC)NCCC#C 67405,CC1=C(C(=O)NCCCCCNC(C2(C)CNC(=O)N2)=O)SCCO1 67406,c1(C(c2n(CCC)nnn2)NC2CC(CC(=O)OCC)C2)nc(C)c(C)s1 67407,N(C(=NCCOCc1ccc(N(C)C)cc1)Nc1ccc(F)cc1)C(CSC)C 67408,Cc1cccc(C)c1CC(=O)N(CC(O)CNC(c1ccc(O)c(F)c1)=O)C 67409,Cc1ccccc1-n1cc(C(=O)NCC2CC2NC(C2CC(C)(C)CO2)=O)nn1 67410,c1(C(=O)NC(CN(C(C(CC)n2nccc2C)=O)C)C)cnc2c(C)nsc2c1 67411,Cc1cccc(N2CCC(N3CCC(n4cc(-c5cnn(C)c5N)nn4)C3)C2=O)c1 67412,C(F)(c1ccccc1)=CC(=O)NCCC(C)(C)NC(C1CCC(F)(F)C1)=O 67413,c1(C(C(N2C(CN(C(c3c(CC)ocn3)=O)C)CCC2)=O)C)ccncc1C 67414,N1(C(CC(CC)C2CC2)=O)CC2CC(NC(=O)C3=CCCCCC3)CC1C2 67415,CC(C)C(F)C(=O)NCCN(C(C1CC(=C(F)F)C1)=O)C(C)C 67416,C(CN=c1cc[nH]c(-c2nccs2)n1)c1cccc(NC(CC(CC)CC)=O)c1 67417,c1(C(N(CC(C)NC(=O)C(C(C)O)N(C)C)CC)=O)cnc(N)c(Cl)c1 67418,N1(C(c2nnc3n2CCC3)C(=O)NC)CCC2CN(C(=O)OC(C)(C)C)CC2C1 67419,C(=O)(C1=NOCC1)NCc1c(C(=O)NC(COC(C)C)(C)C2CC2)occ1 67420,c1(CCC(=O)NC(C2(CCC(=O)OC)CC2)=O)cccc(C#N)c1 67421,CCC(C#N)C(=O)NC(C1CN(C(=O)CCOc2cccc(OC)c2)C1)C 67422,C12(CNC(N3CCN(CC(=O)OC)C(=O)C3)=O)CCCC(CN)(C1)OC2 67423,C(CCS(C)(=O)=O)(C(=O)NCCCN(C(c1ncccc1O)=O)C1CC1)OC 67424,C12(NC(CNC(=O)OC)=O)CCCC1CN(C(=O)C(C)CN1CCOCC1)C2 67425,Cc1ccccc1CCNC(C1CCCN(C(C(C)Cc2cncnc2)=O)C1)=O 67426,C1(OC)(CNC(c2cc(C3CC3)on2)=O)CCN(C(C2CCCCS2)=O)CC1 67427,Cc1ccc(C)c(C(=O)NCC2(C)CCCN(C(=O)CCC3CCC(=O)N3)C2)n1 67428,C1(CNC(C(CC=C)OC)=O)COC(C)(C)CN1C(c1ncc(F)cc1F)=O 67429,Cc1cc(C(=O)NCCC2CCCCN2C(c2ccc(F)s2)=O)cc(O)n1 67430,c1(C(N(CCN(C(C2CCC(C)NC2=O)=O)C)C)=O)cccc2c1CCN2 67431,n1(CC(N2CCC(N(C(CCNC(C)=O)=O)C)C2)=O)nc(C)oc1=O 67432,c1(CC)cc(C)c(NC(C2CC2C(=O)Nc2cnc(OC)cn2)=O)c(Br)c1 67433,C(=O)(CCS(=O)(=O)Cc1ccccn1)NC(C)CN(C(=O)C#CC1CCC1)C 67434,Cc1cc(CC(=O)NC(C)CCCNC(C2CCC2Cc2ccccc2)=O)on1 67435,N1(C(C(C(C)(C)C)O)=O)CCC(C2CC2)(CNC(=O)CC2CC2)C1 67436,C1(N(C)C(C2CCCCN2C(=O)C(C)(C)C)=O)COC(C)(C)OC1 67437,CCCCS(=O)(=O)CC(=O)N(C1CCN(C(=O)C(CO)OC)CC1)C 67438,C1(C(N(CC(C)N(C(Cc2scc(C)c2)=O)C)C)=O)C(C)(C)C1(F)F 67439,C(=O)(CCCCCN(C(=O)CC1CC(F)(F)C1)C)NC1CCN(C)C1 67440,c1(N2C(CNC(c3ccc(F)cc3)=O)CC(F)C2)nc2cc(F)cc(F)c2o1 67441,C1(C(N(CCNC(C2(CF)CC2)=O)CC)=O)CC2C(C1)C2(F)F 67442,CCCC(O)C(=O)NC(CNC(c1sccc1COC)=O)CC 67443,n1(CC#C)c(C)cc(C(=O)NCC2(O)CN(C(c3cn(C)nc3C)=O)C2)c1C 67444,C1(C(=O)NC(CNC(C(C)n2cncn2)=O)C2CCC2)CN(CP(C)(C)=O)C1 67445,c1(C2(C(=O)OC(c3ccccc3)C)CC2)ccc(Br)cc1F 67446,C(c1ccc(C(C(=O)NCC2CC2)N(C)Cc2nc[nH]n2)cc1)=CC(=O)OC 67447,c1(CCC(=O)NC2C(NC(C3CC(C)(C)C3)=O)C2)ccncc1Br 67448,CCC(CC)C(C)C(=O)N(CCC(=O)NCc1csc(C)c1)CCCO 67449,N1(C(C(C)SC)=O)CCCC(CCNC(c2c[nH]nc2-c2ccccn2)=O)C1 67450,C(CS(=O)(=O)CC(=O)N1CC(NC(c2cc(C)sn2)=O)CC12CCC2)OC 67451,C1(NC(c2c(C)cnnc2)=O)CC2CC1N(C(=O)CCc1ccncc1)C2 67452,c1(CN(C(C2CC23CCC3)C(=O)NC2CCS(=O)(=O)CC2)C)nnc2n1CCC2 67453,CC1CCCC(C)N1C(C1CC1C(=O)NCc1ccc(Cl)c(Br)c1)=O 67454,N1(C(CNC(CNC(c2c(NC)nccn2)=O)=O)=O)CCc2nocc2C1 67455,c1(CCC(N2CC(O)(C(C)NC(C=CC=CC)=O)C2)=O)ccnc(C)n1 67456,c1(OCC)cccc(Cl)c1CNC(=O)C(CC(C)C)Oc1ccccc1 67457,C1(CNC(c2csc(C)c2C2CC2)=O)C(C)CCCN1C(c1cnns1)=O 67458,c1(CC(=O)NCC2N(C(C(CC(=C)C)C)=O)CCOC2)csc2nc(C)cn12 67459,c1(N2CCCC(C=C)C2)ccncc1S(=O)(=O)N1CCCC(c2ccncc2)C1 67460,CC(C(C)(C)NC(=O)CSc1ccccc1)NC(=O)COc1cn[nH]c1 67461,c12nnc(n1CC1(C)CC1)CN2C.c1(CC2CCCC2)ncn(C)n1 67462,C(=O)(C1=CCC(C)(C)CC1)NCC1C(C)CN(c2ccn3ccnc3n2)CC1 67463,c1(C(=O)NC2C(NC(C3(CC)COC3)=O)C2)ccc2ccn(C)c2c1 67464,N1(C(CCSCC(C)C)=O)CC(NC(c2cnc3cc[nH]c3c2)=O)C(C2CC2)C1 67465,C1(NC(c2nc(C)oc2)=O)C2CC1N(C(c1c[nH]nc1OCC(F)(F)F)=O)C2 67466,Cn1nnc2c1CCN(C(=O)CCCCCNC(=O)C(C)(F)C(C)(C)F)C2 67467,Cc1c(C(=O)NC2CCN(c3ccnc(C4CC4)n3)CC2)ccc(F)c1F 67468,C1(C(=O)OC)C(C)CCN1C(C1CC(NC(=O)CSC(F)F)CCO1)=O 67469,C1(C(N2CC(O)(CNC(C3CC(CCC)C3)=O)C2)=O)CCc2cnn(CC)c2C1 67470,c1(OC(C(=O)NC(C(C)C)CNC(C2CSC2)=O)C)cccc(Br)c1 67471,N1(C(C(C=CC)O)=O)CCC(NC(c2cccc(Br)c2)=O)C1(C)C 67472,N1(C(CC(=O)N(C)C)=O)CC(NC(C2COC3COCC3O2)=O)CC12CCCC2 67473,c1(C(=O)NC2CC(CNC(C3CC(CCC)OCC3)=O)C2)ccc([N+](=O)[O-])s1 67474,N1(C(C(c2cccc(Cl)c2)(C)C)=O)CC2CCN(C(C3CCCS3)=O)CCC2C1 67475,C1(NC(c2c(OC)n[nH]c2)=O)CCN(C(=O)CN2CCCC2=O)CC1O 67476,C1(C(=O)NCCc2onc(C)n2)CC(C)CN1C(=O)C(N1CCOCC1)C 67477,C1(C(=O)NCc2scc(CNC(C(C)SCC)=O)n2)CC2CCCC(C1)C2 67478,c1(-n2ccc(C(=O)NC3C(NC(=O)C=Cc4cscn4)C3)n2)ccccc1Cl 67479,c1(SCCC)cccc(C(=O)NC(C)CNC(c2oc(CC)cc2C)=O)c1 67480,C(C(=O)N1CCC(NC(C2CCOCC2)=O)CC1C)(C(C)(C)C)NC(C)=O 67481,c1(C(=O)NC2C3CC(NC(C(C)SCCCC)=O)CC32)cc(C)cc(C)c1N 67482,C#CCC(CC(=O)NC1CCC(NC(=O)C=CC(C)(C)C)C1)c1ccccc1 67483,C(=O)(CCCC(C)(C)C)N1C(CCNC(c2cnn(CC)c2C)=O)COCC1 67484,c1(C(=O)NCCN(C(c2c(O)cc(C)nn2)=O)C2CC2)c(C)nc2ccccn12 67485,CCCCC(O)C(C)C(=O)NCCN(C(=O)CCC1CC(F)(F)C1)C(C)C 67486,CC1CCCCCC1NC(=O)CCCCN(C)C(c1cc2occc2[nH]1)=O 67487,c1(N(CCC)C(C)=O)cc(CN2CCCC2c2cccs2)cc(F)c1 67488,N1(C(c2cc(CC)[nH]n2)=O)CC(C)N(C(C2(C)CCOC(C)C2)=O)C(C)C1 67489,C12(C)CCC(C1)NC2.C(CS(C)(=O)=O)C1CN(C(=O)NC(C2CN(C3CC3)C2)C)C1 67490,c12ccc(Cl)c(c1)NC(=O)C(C)SC2.c1(CCOC)oc(CN)cc1C 67491,c1(OC)cc(OC)cc(NC(=O)C(c2cnc(C(C)O)s2)N(c2ccsc2)C)c1 67492,C1(N(C)C(c2cc(F)cs2)=O)CN(C(c2cccc(N)c2)=O)CCC1O 67493,CC1(NC(c2cnn(CC3CCCCC3)c2)=O)CN(C(C2CC2(F)F)=O)C1 67494,c1(C(=O)NCC(=O)NC(C2(O)CN(C(C3CC=CCC3)=O)C2)C)cnc(O)nc1O 67495,C1(C)(C(N(CC(CC)NC(=O)CCOCCN(C)C)C)=O)CC2CC2C1 67496,c1(N2CCCC(CN(C(C3(COC)CCCC3)=O)C)C2)ncccc1[N+](=O)[O-] 67497,CCC(CC)(CCNC(=O)OC(C)(C)C)NCC1CCCOC1CC(C)C 67498,CCC(C)CCCCC(=O)N1CCC(NC(C2CCCC(C)(C)C2)=O)C(C)(C)C1 67499,N1(C(C(C(C)C)c2cccnc2)=O)CCOCC(NC(c2cccnc2)=O)C1 67500,C1(C(N2CC(c3ccccc3)(NC(CC(C)OC)=O)C2)=O)CCCCC1(C)C 67501,c1(N2CCC(CC)OCC2)nc(N2CCSC(c3cccs3)C2)c2c(n1)CCS2 67502,Cc1nc(NC(c2nccn2C)c2nnnn2C2CCOC2)cs1 67503,c1(C(N2C(C(C)(C)NC(=O)CCC3CC3)CCC2)=O)ccc2nc[nH]c2c1F 67504,C1(N(C(CSCCCC)=O)C)CCN(C(=O)CCCc2cccs2)C1 67505,C(C(F)(F)C(C)(C)O)NC(C1(CNC(C(CN(C)C)O)=O)CC(C)(C)C1)=O 67506,CC(O)(C(=O)N1C2CN(C(=O)Cc3ccc(C(F)(F)F)cc3)CC12)C(F)(F)F 67507,C(=O)(CS(=O)C(F)(F)F)N(C)CCN(C)C(C1CCN1C1CCCC1)=O 67508,CCCCCC(F)C(=O)NC(C)(C)CCNC(c1cnn(CC)c1C)=O 67509,CN1CCCC2C1CCN2C(=O)Nc1cccnc1-c1ccccn1 67510,N1(C(CC)=O)C2CCCC1CN(C(c1c([N+](=O)[O-])ccc(C)c1F)=O)CC2 67511,CC1(C)CC(CC(N2CC3(CCC3O)C2)=O)CN1C(c1ccco1)=O 67512,CCC(O)C(C)(C)C(=O)NCC(CC(=O)NCC(CSC)OC)OC 67513,n1(CC2C(C)CCC2)ncc2cc([N+](=O)[O-])ccc2c1=O 67514,c1(C(N(C)CC2CN(C(C(C(C)O)C)=O)C2)=O)cn2cc(Cl)cnc2n1 67515,C1(COC)(NC(=O)CNC(N)=O)CCN(C(c2ccc(C#N)cc2)=O)CC1 67516,C1(CC#C)(C(N2CC(F)CC2CNC(=O)C(C2CCCCC2)C)=O)CCCCO1 67517,Cc1ccccc1C(C(N1CCC(F)(C(=O)C2CC2)C1)=O)NC(=O)OC(C)(C)C 67518,CC#CCC(C(=O)NCCOC1(C)CCC1)NC(c1cc(C#N)n(C)n1)=O 67519,O=C(CC=C(Cl)Cl)NC1CCCC1CNC(=O)C=Cc1cc[nH]n1 67520,c1(C(N(C2CN(C(=O)CCCC#N)CC23CC3)C)=O)cc2ccsc2n1C 67521,N1(C(CCC2C(C)=NNC2=O)=O)CCC(NC(=O)CCC(C)(C)C)C12CC2 67522,N1(C(CC)=O)CCC(C)C1C(=O)N(C)Cc1ncc(Br)cn1 67523,C1(C)(C(N(CCC)CCNC(=O)CC2CCCC2)=O)CCCC1O 67524,S(=O)(=O)(c1ccc(Br)cc1C(OC(F)F)=O)N(CCNNC(c1ccccc1)C)C 67525,c1(C(N2CCN(C(c3c(C(C)C)nns3)=O)CC2)=O)cccc(Cl)c1O 67526,C(CNC(c1c(C)noc1CC)=O)(C(C)C(C)C)NC(CCCC=C)=O 67527,C#CC1(C(=O)NC(C)Cc2ccnn2C)CCN(C(c2cscn2)=O)C1 67528,C1(CNC(C(CCOC)NC(c2cnncc2O)=O)=O)CC2CCCC2C1 67529,Cc1ccc(C#CC(=O)NCC2CCOCO2)cc1 67530,C1(NC(c2cncc(OC)n2)=O)CN(C(C2SCCCS2)=O)C2CCCC12 67531,C(c1ccncc1)=C(C)C(=O)NC1(CCO)CN(C(C2(Cl)CC2(F)F)=O)C1 67532,O=C(C1=NOC2(CCOC2)C1)N1CCC2CCN(C(=O)C(F)(F)C(F)(F)F)CC12 67533,c1(OCC(=O)NCC2CN(C(C=CC(=O)OC)=O)C(C)C2)ccc(Br)c(F)c1F 67534,c1(CNC(CSCCC)=O)cnn2c1CN(C(c1cncc(C)c1C)=O)CC2 67535,N1(C(CCCOCCOC)=O)CC(NC(=O)C(F)(F)CO)CCC(O)C1 67536,c1(C(C)(C)C)nc(=NC2CC(NC(C3CC3c3ccccc3)=O)C2)s[nH]1 67537,Cc1c(Cl)sc(Cl)c1C(=O)OCC(C1C=CCC1)=O 67538,C1(C(C)SC)CC2CCC1CC2.C1(OC)CCN2C1C1C(CCO1)NC(=O)C2=O 67539,N1(C(c2cc(OC)n[nH]2)=O)CCCC(CCCCNC(c2[nH]ccc2CC)=O)C1 67540,C1(CC#C)(C(=O)N(C2CCOC2=O)C)CCN(C(=O)CN2CCNC(=O)C2)C1 67541,c1(NCC=CCNC(Cc2c(C)ncnc2C)=O)cc(=O)n(C(C)C)c(O)n1 67542,C1(C(N(CCCNC(=O)C(=O)N=S(C)(C)=O)C)=O)CC2CCCC(C1)C2(F)F 67543,N1(C(CC(C)CN(C)C)=O)C2CC1CN(C(=O)C(C)C#N)C2 67544,N1(C(CCN(CC)CC)=O)CCC(CO)C(NC(=O)CC23COCC(C2)C3)C1 67545,C1(CC2C(OC)CCC2)COCCN(n2cc(-c3c(N)c(C)nn3C)nn2)C1 67546,CC1CCOC(C(=O)NC2CC(C(C)NC(c3cc(=O)cc[nH]3)=O)C2)C1 67547,C1(NC(c2ccnc(N3CCCC3)n2)=O)CCCN(C(c2ccoc2)=O)C1 67548,C1(C(=O)NCC2CCC(C)C2)(OC)CCN(C(=O)C=NOC)C1 67549,N1(C(=O)OC(C)(C)C)CCCC1C1CCCCN1C(C1C(CN=[N+]=[N-])C1(C)C)=O 67550,C(=O)(CCCCC1CC1)NC(CC)CNC(=O)CNC(=O)Nc1ccccc1 67551,N1(C(c2c(SC)snn2)=O)CCN(C(=O)C(C)C(F)(F)F)C(CN(C)C)C1 67552,N12CC3CCC3(C1)NC2=O.C1(N(C(C)(C)C)C)C(=O)NCC1(C)C 67553,N1(c2cc(C(=O)OCC)ncn2)CCCN(C(=O)CC(C)c2cnn(C)c2)CC1 67554,c1(OCC(=O)N(CCCCN(C(C(CCC)O)=O)C)C)c(C)cccc1Cl 67555,c1(C(N(CC(O)CNC(=O)C(F)C(F)(F)F)C)=O)ccc(C#N)cc1 67556,C1(NC(C2N(C)CCC2)=O)CC2(CCCCN2C(=O)CCC(N)=O)C1 67557,N1(C(=O)CSCc2ncc[nH]2)CCC2(CCCN(C(=O)CC3CCOC3=O)C2)C1 67558,CCC(C)C(=O)NCCN(C(=O)C(C)(O)C1CCOCC1)CCOCCO 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67576,c1(CC(N2CC(NC(C(CC=CC)C)=O)C(OC)C2)=O)ccc(C)c(F)c1F 67577,c1(OC)ccc(C(N2CC(O)(C3CCCN3C(=O)CC(C)OC)C2)=O)cn1 67578,C12(C(=O)NCC(C)CNC(=O)Cc3ccsn3)CCCCC(F)(C1)C2 67579,c1(C(N2CC(C)C(CNC(=O)CCn3cnnn3)C2)=O)nn2cccnc2c1Cl 67580,c1(C(=O)NC2C(C)CN(Cc3ncccc3Cl)C2)cc2ccccc2cc1O 67581,C12(C(N(CC(C)NC(C3C(OCC)CC3)=O)C)=O)CC3CC(C(=O)N1)C2C3 67582,C(=O)(C1CC(=O)c2ccccc21)N(CCCC(=O)NC1(C)CCCC(C)(C)C1)C 67583,C1(NC(=O)Cn2ccnn2)C=CC(CNC(c2csc(O)n2)=O)C1 67584,c1(OC)ccc(C(N2CC(NC(c3ccc[nH]3)=O)CC(C)C2)=O)c(F)c1 67585,C1(NC(C2OCC(C)C2)=O)CCC2CN(c3nc4cccnc4s3)CCC2C1 67586,c1(NC2C(CNC(=O)Nc3ncccc3C(F)(F)F)C2)cc(C(F)(F)F)ccn1 67587,C(CC(=O)Nc1cccc(Cl)c1O)(C(C)(C)C)NC(c1cnc(C)o1)=O 67588,CC(C)CC(CNC=O)CC(=O)NCC(C1CCCC(C)(C)CC1)=O 67589,CCC(O)(C(=O)NCCN(C(=O)CC(C)(O)c1ccccc1)C)c1ccccc1 67590,C1CC(=O)N1CC#C.C(C(O)C1CC1)NC(C1CCC1)=O 67591,Cc1c(N(C2CCCCC2)C(=O)CN2CCCC(C(C)O)C2)cccc1Cl 67592,C1(N(C(C(C)NC(CC)=O)=O)CCO)CCCN(C(c2cc(CF)on2)=O)C1 67593,c1(C(N2CCC(O)(C(N3CC(C)C(O)C3)=O)C2)=O)cccc2ncoc12 67594,N1(C(CCCCC=CC)=O)CCC(NC(=O)COc2cccnc2)C(CO)CC1 67595,N1(C(c2ccc(C(C)C)cn2)=O)CC(CNC(=O)CP(C)(C)=O)C2(CCC2)C1 67596,c1(CN(C(c2csc(CO)c2)C(=O)NCC=C)C)ccc(OCCC)c(Cl)c1 67597,C1(C(=O)NC(c2nc[nH]n2)CC)CCCN1C(=O)CC1CCSC1 67598,N1(C(C2(C)CCC(=O)N2)=O)CCC2CC(NC(c3ccc(F)cc3)=O)CCC2C1 67599,C1(NC(C2CCC(F)(F)CC2)=O)CN(C(C2CC2(Cl)Cl)=O)C2(CCOCC2)C1 67600,c1(C(N2CC(N(C(=O)Cc3cccc(O)c3)C)C2)=O)ccnn(C)c1=O 67601,C1(N(C(C=CC(=O)OCC)=O)C)CCCCC1N(C)C(C1CC1F)=O 67602,c1(SC(C)C(=O)NCC(C)(O)CNC(=O)CCc2ccn(C)n2)ccccn1 67603,n1(CC(N2CCN(C(C)CNC3CC4CC4C3)CC2)=O)ncc2ccccc12 67604,N1(C(C2CN(C(CNC(C)=O)=O)CC(F)C2)=O)Cc2ccccc2C1 67605,C1(CC(=O)NC2CCCN(C(CC3(C)CC3(F)Cl)=O)CC2)CC2(CCCC2)CO1 67606,Nc1cc(Cl)cc(F)c1C(N1CCCN(C(c2cccc(O)n2)=O)CC1)=O 67607,CC1CN(C(C2CC(C(C)(C)C)=NO2)=O)c2cnccc2N1 67608,C1(CN(C(C2N(C(CC)=O)CSC2)=O)C)COCCN1C(=O)Cc1ccsn1 67609,C(=O)(C(C)CCCC(C)C)N(CCNC(c1c(N)ccc(OCC)c1)=O)C(C)C 67610,N1(C(c2ccc(C)s2)=O)CCC12CCCN(C(c1cccc(B(O)O)c1)=O)C2 67611,c1(C(N(CCOC)CCNC(C2(C)CC2(F)Cl)=O)=O)ccc(C)cc1[N+](=O)[O-] 67612,c1(C(N(CCCCNC(C2CC(F)C2)=O)C)=O)cc(N)cc(F)c1 67613,CCC(C)CCCC(=O)N1CC2CCC(C1)N2C(C1CCCO1)=O 67614,c1(CCC)nc(C)c(C(=O)N(C)CC2CCCN2C(=O)C(C2CCCCC2)O)s1 67615,C(=O)(C(CS(=O)(=O)C(F)(F)F)NC=O)NC(CC=C)C(=O)OC(C)(C)C 67616,C(C)(CC(=O)NCC1CC(F)CN1C(=O)Cc1ccccc1F)(C(F)F)N(C)C 67617,N1(C(CCCC2C(C)C2)=O)CCN(CN2CCN(C(=O)CCC3CC3)CC2)CC1 67618,N#CC1(C(N2CCC(NC(C3CCCC(C(N)=O)C3)=O)C2)=O)CCCO1 67619,N1(C(CNC(=O)NC)=O)CCC(O)(C2(NC(=O)CC3CC=CC3)CC2)CC1 67620,CN1CCCCCC1C(=O)Nc1ccc(Oc2cccc(C#N)c2)cc1 67621,c1(C(=O)O)ccnc(CNC(CC2CCCC2)Cc2ccc(F)cc2)c1 67622,C#CC1(C(=O)NC2COCC(C)(C)C2)CCN(C(c2ccoc2CC)=O)C1 67623,C1(NC(=O)CCc2ccccn2)CCOCC1NC(c1cncnc1)=O 67624,C1(NC(C(C=C)O)=O)CCCC12CCN(C(=O)COCC(=O)OC(C)(C)C)CC2 67625,CC1CN(C(=O)C2=COCC2)CC1CCNC(C1OCCC1c1ccccc1)=O 67626,c1(C(=O)NCCCCNC(C2COCC(C)O2)=O)ccnc(C(F)(F)F)c1F 67627,c1(C(=O)NCC(CC=C)NC(c2ccnc(SCC)c2)=O)nnn(C)c1N 67628,N1(CC(=O)NCCC(C)N(C(=O)C=Cc2cscn2)C)CCC(CO)CC1 67629,C12(NC(C(C)OCCCC)=O)CC3CCC(C1C2)N3C(C12CCOC(C)(C1)C2)=O 67630,c1(OC)cc(C(N2CCC(NC(c3cccs3)=O)C2C)=O)ccc1OCC(N)=O 67631,Cc1nccnc1NC(=O)NC(CCc1cn(C2CCN(C)CC2)nn1)C(=O)O 67632,c1(C(=O)NCC2C(C)CCN(C(=O)C(C)(C)C3CCC3)C2)ccc(C#N)nc1O 67633,C#Cc1cccc(CC(N2CC3CC(N(C)C(c4cc[nH]n4)=O)C2C3)=O)c1 67634,C1(NC(C(C2CC2)OCC)=O)CCN(C(c2ncc(C)cc2OC)=O)CC1CC 67635,c1(C(c2nnnn2CC(F)F)NCC(=C)CC)c(N(C)C)ccnc1Br 67636,N1(C(C2C3(CCN(C(c4c(C)c(C#N)[nH]c4)=O)C3)C2)=O)CCC(O)CC(C)C1 67637,C(CCN=C(NC1(C(=O)NC)CCCC1)N1CCSC(C(F)(F)F)C1)OCC 67638,C12(C(=O)NCC3C(NC(CCC(=C)Cl)=O)CCCC3)CCCCC1C2(F)F 67639,N1(C(C2(CC)CC(=C)C2)=O)CC2(CC(CC(=O)NCc3ncoc3C(C)C)C2)C1 67640,N1(C(c2ccc(C(=O)OC)cn2)=O)CC(C)CN(C(c2c[nH]ccc2=O)=O)CC1C 67641,C1(Nc2ccc(C(c3ccccn3)N(C)C)cn2)CCC(F)(F)CC1 67642,c1(N(C(c2c(CNC(c3c(CC)nc(C)o3)=O)cc[nH]2)=O)CC)ccc(C)c(C)c1 67643,c1(N2CCN(CC)CC2)nc(N2CCC3(CCCN3C)C2)nc2c1CSC2 67644,c1(C(N2CC(CNC(Cc3c(C)ncs3)=O)C2)=O)cc(C)c(C)o1 67645,C1(CNC(Cn2ncc(CC)c2)=O)CN(C(=O)CSC(F)F)CCC1C 67646,CC1(C)C(Nc2ccnc(N3CCC(c4ccc(Cl)cc4)CC3)n2)CC1O 67647,C(=O)(CC(C)CCC=CC)NC(CCCC)CNC(=O)Cc1cc(C2CC2)no1 67648,CCC(C)C(=O)C(=O)N1CC(C(=O)NC2CCN(C3CC3)C2=O)C(F)(F)C1 67649,C1(NC(C(CN(C)C)O)=O)(CO)CCCN(C(=O)CCCC2CCCC2)C1 67650,c1(N(C(CC)=O)CC)ccc(O)c(C(N2CCN(C(=O)Cc3ccco3)CC2)=O)c1 67651,C1(C(=O)NCC2N(C(c3c[nH]c(=N)s3)=O)CCC2)CCN(CCF)CC1 67652,C#CCCC(C(=O)NCC1CC12CC2)NC(c1cc(F)c[nH]1)=O 67653,c1(CC(=O)NCC2(O)CCN(C(C(C)CF)=O)C2)ccc(Br)c(F)c1 67654,C=CC1(C(=O)NCc2ccc(C(N3CCC3CC)=O)s2)CCCC1 67655,N1(C(C2CCN(C(C3(COCC)CCCC3)=O)C2)=O)CCC(CC(C)O)CC1 67656,C1(C(N(C)CC2CN(C(c3cnn(C)c3N)=O)CCO2)=O)CCN2CCOCC12 67657,C1(NC(c2ccc(=O)n(O)c2)=O)COC2(C1)CN(C(c1c[nH]nc1[N+](=O)[O-])=O)C2 67658,N1(C(CNC=O)=O)CCN(C(CNC(=O)CC2CCC(=O)N2)C(F)F)CC1 67659,C1(NC(C(C)N2CCCC2)=O)CCCN(C(C2(O)CC2(C)C)=O)CC1 67660,CC1CCCCC1(CNC(=O)COCCF)NC(c1cc(C(N)=O)cs1)=O 67661,Cc1nnc2n1CC(C(=O)NCCOC1CN(C(c3ccncn3)=O)C1)C2 67662,C1(C(=O)Nc2ccc(OC)c(N3CCNC3=O)c2)Cc2ccc(F)cc2C1 67663,C1(N(C(C=C(CC)C)=O)C)CCCCC1N(C)C(C1CCC(C)(C)C1)=O 67664,c1(CC)nn(C)c(C(N2CC(NC(=O)CC3CC(=O)C3)CC2(C)COC)=O)c1Cl 67665,c1(C(=O)NCC(C(=O)NCC(COC)O)C)cnn2ccccc12 67666,N1(C(CC2ON=C(CC)C2)=O)CC(CNC(c2ccc(Cl)cc2)=O)C2(CCC2)C1 67667,C1(COC)(CNC(=O)C=CC(C)C)CCCN1C(=O)CCc1nnc(C(F)F)o1 67668,C1(CN(C(=O)CN2CC3C=CC2C3)C)C(C2CC2)CCN1C(=O)CC1CC(F)C1 67669,c1(C(N2C(C)CC(CNC(=O)CCc3cnn(C)n3)C2)=O)cc2ncccc2o1 67670,N1(C(CNC(C(CC)CC)=O)=O)CCC(NC(=O)Cc2ccc(Cl)cc2)C(C)C1 67671,c1(C(=O)NCCN(C(CCSC)=O)CCCN(C)C)ccn2cc(C3CC3)nc2c1 67672,N1(C(C(CCOC)OC)=O)CCN(C)CC1C(=O)NCc1ccnc(O)c1 67673,c1(C(=O)NC2C(OC)CN(C(C3(C(N)=O)CCC3)=O)C2)c(F)ccc(F)c1F 67674,C=CC(C)(CCOC)C(=O)N1CC(F)(CNC(=O)CC(O)CCCC)C1 67675,N1(C(C(COC)CC(C)C)=O)CCCC(C)(C)C1C(N1CC2(CC(O)C2)C1)=O 67676,CCS(=O)CCNC(=O)CC1(N(C)C(c2cccn2C2CC2)=O)CC1 67677,c1(NC(=O)Nc2ccc(C3(O)COC3)cc2)c(F)ccnc1F 67678,Cc1coc(C(C)C)c1C(=O)NCC=CCNC(=O)CSCc1cccnc1 67679,N1(C(C2N(C(C)(C)C)CC2)=O)CCC(NC(=O)CC2CCCCC2O)CC1 67680,C1(NC(C=CC(N)=O)=O)CCC2CN(c3ccnc(C4CC4)n3)CC2C1 67681,Cc1[nH]c(=NCCC2(C(F)(F)F)CCC(C(=O)NC3CC3)C2)ccc1C#N 67682,N1(C(n2cnc(CC)c2)=O)CCC(=CCNC(=O)CCC(C)N(C)C)CC1 67683,N1(C(c2c(N)cn(C)n2)=O)CC2CCC1CN2C(c1nnn2c1CSCC2)=O 67684,C1(C(=O)NCC(C(=O)NC2CC(O)C2)O)Cc2nccn2C1 67685,Cn1nnc2c1CCN(c1nnnn1CC1CC13CCC3)C2 67686,C1(NC(C(F)=CC)=O)CCN(C(c2ccc(C)cc2C(C)=O)=O)CCC1CO 67687,c1(CN(C(CC2CCN(c3ncc(Br)s3)C2)=O)C(C)=O)ccc(F)c(Br)c1 67688,N1(C(COCC)=O)CCC(C(C)NC(C2CC23CCOC3)=O)CC1 67689,c1(C(N2C(CNC(C(C)OCc3ccccc3)=O)CC2)=O)cc2occc2n1C 67690,C1(C(=O)NC(c2ccncn2)C)CN(C(=O)CCC2CCCOC2)C2(CCC2)C1 67691,C(C(=O)N1CC(CCNC(=O)C(C)(C)CN(C)C)C(C)C1)(C(C)C)SCC 67692,CC1(C)OC(=O)NC1C(N1CC(C(O)C(=O)NC2CCCOC2)C1)=O 67693,CC(CCC(=O)NC1CC1)NC(C1CCCN1C=O)=O 67694,N1(C(Cn2cc[n+](C)c2)=O)CC2CC2(NC(=O)CC2CC=CCC2)C1 67695,C(=O)(C=CS(F)(F)(F)(F)F)NCCN(C(CC(CC)(C)C)=O)C 67696,C1(NC(C2C(C)C2C)=O)CN(C(C2CCC(C(N)=O)C2)=O)C2CCCC12 67697,N(C(=NCCSC)NC1CCCC1)CC(c1ccc(CC)cc1)C 67698,C1(C(C2CCCN2C(c2ccsc2Br)=O)C(=O)N2CCCC2)CCC2CC12 67699,N1(C(CCc2cncc(C)c2)=O)C(C)CN(C(C2C3CCC(F)(F)C23)=O)CC1C 67700,C(C)(CCC(F)(F)F)NC(CCN(CCCO)C(c1n(CC)nnc1)=O)=O 67701,c1(C(=O)Nc2cn(C)c(C(N3CCCC3C(F)(F)F)=O)n2)c(CO)ccc(Cl)c1Cl 67702,CCN(OC)C(=O)CNC(c1cc(C(=O)OC)sn1)=O 67703,c1(OC(C)C)ccc(C(=O)NC(C2CCCN2C(=O)C(F)C(C)C)(C)C)nc1 67704,c1(C(=O)NCC(CNC(CC2CCN(CC(C)C)CC2)=O)C)cc(O)cc(O)c1 67705,C(=O)(C(C)(C)C(C)(F)F)NC(C(N1C(CCC)CCC1)=O)c1cccs1 67706,Cc1[nH]nc(CO)c1NC(=O)C(N1CCC(NC(=O)CCc2cncs2)CC1)=O 67707,c1(C(N2CC(C)N(c3nnc(C4CCCC4)s3)CC2)=O)ccc2c(c1)OCO2 67708,CCCC(CC(=O)N(C1CCCC1)CC)NC(C1CC(CC)=NO1)=O 67709,CC1CN(C(C2CC2c2ccccc2)=O)CC1CNC(C1CC(F)(F)C1)=O 67710,N1(C(c2ccc(N3CCCC3)cc2)=O)CCN(Cc2ccc(I)c(O)c2)C2CC12 67711,c1(C(N2CCC(N(C(=O)CCn3ccnc3C)CC)C2)=O)cc(Cl)cc(F)c1N 67712,c1(C(=O)OC)cnc(CNC(=O)NC2CC(CSC)C2)n1C 67713,C(=O)(CCCCC(N)=O)N(C1CCCC1)CCNC(Cc1c(C#N)cccc1)=O 67714,C1(CC(=O)NCC(=O)NC2C(N(C(C3CCC3)=O)CCO)CC2O)OCCNC1 67715,C1(OC)CC(CNC(=O)Cc2cc(C3CC3)no2)N(C(C2CCC(F)(F)C2)=O)C1 67716,O=C(COC(C1CC2(CCC2)C12CCC2)=O)N=c1cc[nH]cc1 67717,c1(C(N2C(CNC(COCC#C)=O)C=CC2)=O)nn(CC)cc1[N+](=O)[O-] 67718,CC1C(NC(=O)C2=CCC2)CCCN1C(c1csc(C(F)(F)F)c1)=O 67719,N1(C(CC2(C)CC2(F)F)=O)CCCC(c2n[nH]c(CNC(=O)CSCC#N)n2)C1 67720,n1(CCOC)cc(C(=O)NC2CC2CNC(C2CC2F)=O)cn1 67721,C(CC(=O)NCC(F)CNC(c1cc(C)ccn1)=O)(C(C)C)OCC 67722,C1(C)(NC(C(C)SCCCC)=O)CCCN(C(=O)Cn2ccc(C)cc2=O)C1 67723,N1(C(c2cnccc2Cl)=O)CCCC12CN(Cc1ccc(Cl)nc1Cl)C2 67724,C1(C(C)C)CN(C(=O)C2=CCCSC2)CCCN1C(=O)CCCN(C)C 67725,c1(N(CCCOC)CCOC)ccc(S(=O)(=O)NC(C)CCC2CC2)c(Cl)c1 67726,c1(C(N(C(C)CNC(c2cnc(C)n2C)=O)CC)=O)cc(C)c2nc(C)cn2n1 67727,C1(CNC(CCCN(CCC)CCC)=O)CN(C(C2(C(=O)OC)CC2)=O)CCO1 67728,c1(C)cccc(O)c1C.C(CCCC(=O)NC(C1CCCN1C=O)(C)C)OC 67729,N1(C(CN(C)C)=O)CCC2(CCN(C(c3ccc(C4CC4)s3)=O)CC2)C1 67730,C1(NC(C2C(C)=C2)=O)CCOC12CCN(C(c1nc(C)c(C)s1)=O)CC2 67731,O=C(CCCC(F)(F)CO)NC1CC2CCC(C1F)N2C(C1CC2CCC2C1)=O 67732,CC(O)C(C)(C)CNC(C1CC(CNC(=O)C(O)CCN(C)C)C1)=O 67733,c1(C(=O)NC2CC(CNC(=O)CCCN3CCCCC3)C2)ccnnc1Cl 67734,C1(C)(CNC(c2c(CC)noc2)=O)CCN(C(=O)CC2CC2(Cl)Cl)C1 67735,CC(C)(C)C(=O)N1CSCC1CNC(Cc1cccs1)=O 67736,CCCCCCC(=O)N1CCCC(N(C)C(c2nccc(C(F)(F)F)n2)=O)C1 67737,c1(C(N2C(CNC(CC=C(C)C)=O)C=CC2)=O)ccc(C)c(S(C)(=O)=O)c1 67738,C1(C(N(CCCC)CC)=O)OCCC1NC(C1CC1Cl)=O 67739,Cc1cc(Br)cc(Cl)c1NC(=O)NCc1nccn1C 67740,c1(OC(C(=O)NCC(=C)CCNC(=O)C(O)CCSC)C)ccc(Cl)c(C)c1 67741,c1(CC(=O)NCC23OCC(NC(CCSC)=O)(C2)C3)cc(Cl)ccc1Cl 67742,N1(C(C(C)C(=O)N2CCOCC2)=O)CCCC(C)(NC(C2CC2F)=O)C1 67743,N1(C(C2N(C(c3cn(C(C)C)nc3)=O)CC(O)C2)=O)CCCCC(CO)C1 67744,C(=O)(CC(C)(C)CNC(c1scc(C)c1C)=O)N1C(C(N)=O)CC(OC)C1 67745,CC1(CNC(C2CCNC2=O)=O)CCN(C(C2SCCCS2)=O)C1 67746,CCC(C)CCCCC(=O)NCCCCCN(C)C(C1(OC)CCC(C)(C)C1)=O 67747,C(=O)(C1=CCC(NC(=O)CC2COCCO2)C1)NC(c1cncs1)C 67748,N1(C(CCC=C(C)C)=O)Cc2[nH]nc(C(N3CCCCC3C3CCC3)=O)c2C1 67749,C1(NC(CCS(=O)(=O)NC)=O)(CNC(c2ncccc2Cl)=O)CC2CCC1CC2 67750,c1(OC)ccc(OC)c(CCC(=O)N2CCC2CNC(C2Cc3nccn3C2)=O)c1 67751,C12(C(=O)NCc3ccc(COC)c(F)c3)CC3CC(C1)C(=O)C(C3)C2 67752,C1(N(C)CC)CN(c2nnc(Cc3cc[nH]n3)n2CC2CC2)CC1C 67753,N1(C(c2cccc(NC(C)=O)c2C)=O)CCCC12CN(Cc1ncsc1C)C2 67754,C1(C)(OCC(=O)NC(CNC(c2c(C)nsc2)=O)C(C)C)CCOCC1 67755,N1(C(CNC(CNC(C)=O)=O)=O)CC2CC1CCN2C(c1ncc[nH]c1=O)=O 67756,c1(C(N2CC(c3cn(CCN4CCOCC4)nn3)C2)=O)cnc(O)o1 67757,C1(CCN(C(CCCC)=O)CCOC)CCCCN1C(=O)Cc1scnc1C 67758,CCC(CC)C(C(=O)N1CCC(C(=O)NCCCC2CC2)(CC)CC1)OC 67759,CC1CCN(C(c2cnn(C)c2C(F)F)=O)CC1NC(C1CC(F)(CO)C1)=O 67760,c1(C(N2CCCC2CCNC(C2CC(O)C2)=O)=O)cc(Cl)c2[nH]c(O)nc2c1 67761,c1(C(=O)NCc2c(C)cco2)ccnc(CNC(=O)COc2ccsn2)c1 67762,c1(C(c2n(C3(C)CC3)nnn2)NCC2CCC3(CC3)C2)cccc2sccc12 67763,c1(C(N(CCCN(C)C(C2(NC(N)=O)CC2)=O)C)=O)ncc(Cl)cc1F 67764,c1(NC(NNC(=O)C(N2CC(O)(CCC3CCOC3)C2)=O)=S)cc(F)ccc1F 67765,c1(C(=O)NCC2CCCN(C(C(CC=CCC)C)=O)C2)sc2ccccc2c1Cl 67766,C1(C(=O)NC2(C)CN(C(=O)CO)C2)C2Cc3ccccc3C12 67767,c1(C(=O)NCC(CNC(Cc2cn(CC)nc2)=O)(C)C)noc2cc(F)ccc12 67768,CC(CC(=O)NC1COCC1CNC(=O)CC1CCCSC1)N(C)C 67769,CCCC(CCC)C(=O)N(C1CCN(C(C2(CCOC)CCCC2)=O)C1)C 67770,c1(OC)ccc(C(N2CCC(NC(=O)CSC)C2(C)C)=O)c(C)c1OC 67771,c1(C(=O)NC(C2(CNC(C3(O)CC3)=O)CC2)C)cc2c(cc1N)CCCC2 67772,N1(C(=O)CCCC(N)=O)CCC2(CC1)CCN(C(C(COCC)C)=O)C2 67773,CC(C)C(C)(O)CNC(=O)C=CCC(C)(C)NC(=O)C(F)CC1CCOC1 67774,Cc1nc2c(s1)CCN(C(c1cnccc1C)C(=O)NC1CCC1)C2 67775,C1CC(C)CC(C)C1.C(C(=O)NCCCC1(NC=O)CC1)SCC 67776,C#Cc1cn(C)nc1C(=O)NC(C1CCCN1C(c1cccc(O)c1C)=O)C 67777,c1(C(=O)NCCCOCCC(=O)N(CCCC)CCCO)cc(C(C)(C)C)n[nH]1 67778,n1(CC(N2CC(C)(NC(CC=C)=O)C2)=O)cc(C)c(O)nc1=O 67779,C(=O)(CCC(C)(C)F)NCC(CC(C)O)c1ccccc1 67780,C(=O)(CCCCC(C)C)NCCN(C(C1CC(CCC)OCC1)=O)CC 67781,N1(C(CCCOC)=O)CCN(C(=O)CCc2nnc(S)nc2O)CC12CC2 67782,C1(CC)CN(C)CCCN1C(=O)C(C(C)C)NC(c1c[nH]c(=NC)s1)=O 67783,C=CC1CCCN(C(c2ccc(CNC(=O)CN(C)CCOC3CC3)nc2)=O)C1 67784,CCCCC(C)(F)C(=O)NC1(CCCC(=O)NC)CCC1.C12CC1CNC2 67785,N1(C(c2ccc(SC)o2)=O)CC(CC(=O)N(C)C)C2(CC2)C1.c12ccoc1CN2 67786,Cc1cc(N(C(=O)CC2(NC(c3cnc(S)nc3)=O)CC2)C)cc(C)c1 67787,c1(C(N2CC(CNC(C3(Cl)CC3)=O)C(O)C2)=O)cc(F)c(C(F)(F)F)c(F)c1 67788,C=CCC(CC)C(=O)NC(CNC(=O)C(O)Cc1cnc[nH]1)CCCC 67789,C1(N(C(=O)C(C)(C)CC(F)F)C)CC2CCCC1N2C 67790,CCCC(C)CC(=O)NCC(C)(CC)C(=O)NCc1cc(C(C)C)n[nH]1 67791,n1(CC(=O)NCCCCNC(=O)Cn2cccn2)nnc(-c2ccccc2)n1 67792,CC(Cc1cnc[nH]1)C(=O)N(C1CCN(C(=O)C(F)(F)c2cscn2)C1)C 67793,c1(OC)ccc(C(=O)NC(C)C(C)NC(=O)CC(C)(C)C)cc1F 67794,c1(CC(=O)NC2(CC=C)CCN(C(=O)CC3CC3(C)C)C2)ccc2occc2c1 67795,CC1(C)OCC(CC(N2CCN(CCCNC(=O)C(F)n3cccn3)CC2)=O)O1 67796,c1(C(N(CCCNC(=O)CC2(C)CC2F)CC)=O)cnc(SC)nc1O 67797,N1(C(C(c2cccc(Cl)c2)CC)=O)CCCCCC1CNC(c1cnc(S)[nH]1)=O 67798,C1(CNC(c2nc(CCC)sc2)=O)CN(C(c2nocc2Cl)=O)CCC12CCC2 67799,C1(C(=O)NCC=CCNC(COC(C)C)=O)CCCC(C2CC2)O1 67800,N1(C(C2N(CC(c3ccc(O)cc3)=O)CCOC2)=O)CCOC(C(F)F)CC1 67801,c1(OCC)ccc(OC(N2CC3C(C(=O)Sc4ccc(F)cc4)C3C2)=O)cc1 67802,C(CC(=O)NC1CC(C)OC1=O)(C(F)(F)F)NC(Cc1cc(CC)no1)=O 67803,C(C1CCCN1C)=NC1(n2cc(CNC(C(C)CN3CCCCC3)=O)nn2)CC1 67804,c1ccc2ccc(Br)cc2n1.N1(Cc2n(CC)nnc2)CCC2(CC=CCO2)C1 67805,N1(C(C2(C)C(C)OCC2)=O)CCC(CNC(C2(c3cc[nH]n3)CC2)=O)C(O)C1 67806,C(CCCC(=O)N1CCOC(CCO)C1)NC(C(C=C)O)=O 67807,c1(CNC(C2C(CNC(c3c(CC#N)c[nH]n3)=O)C2)=O)ccnc(F)c1F 67808,C1(CCC(N2C(C(=O)NC)CC2)=O)CCC(NC(c2cc(C(C)=O)on2)=O)C1 67809,c1(C(=O)NC(C(C)NC(=O)CSC(F)F)CO)ccccc1-n1nnnc1C1CC1 67810,S(=O)(=O)(c1cccs1)NC(C)C(=O)NCC(=O)Nc1cc(F)ccc1O 67811,C1(CNC(Cc2scc(C)n2)=O)CN(C(=O)C(F)(F)C(F)F)CCC1(C)C 67812,C1(OC)COCCC1CC(=O)NCC(C)(C)CNC(c1scc(C)c1Cl)=O 67813,C1(CC(=O)N(CC(N)=O)CC)CN(C(=O)C(C)c2ccco2)CC1C 67814,CC(C(=O)N1CC(NC(=O)C=CC(F)F)C(CC2CC2)C1)S(C)(=O)=O 67815,C1(NC(c2ccc(Cl)o2)=O)C2CN(C(=O)Cc3ccccn3)CC12 67816,C(c1ccc(NC2CCN(S(C)(=O)=O)C2)cc1)=CC(=O)Nc1c(CC)noc1 67817,N1(C(CN(CCCCCC)C)=O)CC2CC1C2CNC(=O)CC(C)(C)O 67818,c1(OCC)nc(C(=O)NC2(C(=O)NC3CC(C(N)=O)C3)CC2(C)C)co1 67819,CC(C)C(CNC(c1cc(Cc2ccccc2)c[nH]1)=O)NC(=O)CCC#N 67820,N1(C(C2=CC(C)(CC)C2)=O)Cc2ccccc2C(NC(C2(F)CCCC2)=O)C1 67821,CC1CN(C2CCCN(c3ccccc3OC(F)F)C2=O)S(=O)(=O)C1 67822,N(C)(C1=S=C(C(=O)NC(=O)OC(C)(C)C)CCC1)C(C)Cc1cccc(F)c1F 67823,C1(N(C)C(=O)NC(CC2CCCCC2)Cc2ccccc2)CC2CCC1O2 67824,c1(C(N(CC(C)NC(C2CC2C(F)F)=O)C)=O)ccc2c(c1)C(=O)CCS2 67825,C1(C2CC2)(CNC(CC2C(C)(C)CC2)=O)CCN(C(c2ccc(Cl)cc2O)=O)C1 67826,C1(NC(c2ccn(CCCC)n2)=O)CN(C(=O)CCn2cccnc2=O)CC1O 67827,c1(CNC(=O)C(N2CC(O)CC2c2cccc(F)c2)C2COC2)ccccc1Br 67828,c1(C(=O)Nc2cncc(-c3ccc(OC)cc3)c2)ccc(Br)cc1O 67829,C12(C(=O)NCC3N(C(C(C)(C)SC)=O)C4C(C3)C4)CC3CC(C1)CC(O)(C3)C2 67830,C(=O)(CC1CCc2ccccc21)NC1CC(CNC(c2cc(C)nc(O)c2)=O)C1 67831,C1(C(=O)NCC2CCC(O)C2)CC2CC2N1C(=O)CO 67832,c1(CC(=O)NC2C(NC(C3(C(N)=O)CC3)=O)C2)ccc(Br)cc1Cl 67833,C(=O)(CCP(C)(C)=O)NC(C(=O)NC(c1cncn1C)CC)CC1CCC1 67834,c1(OC)ncccc1C(N1CCC(C)C1CNC(=O)CCc1ccncc1F)=O 67835,N1(C(CCCC=C)=O)CCN(C(=O)C(C)OCCN(C)C)CC1CCCC 67836,c1(NC2C(NC(C(C)SCC)=O)CCCC2)ncnc2cnccc12 67837,c1(-c2n(CCCC)nc(Cn3cccn3)n2)c(SC)ccc(Br)c1F 67838,C1(NC(c2cccc(F)c2O)=O)CC2CC(NC(C3CCCCS3)=O)C1C2 67839,C12CC3CCC(C1)N3c1cnc(cn1)C(=O)NC2.CC1(C)CC(C(=O)N(C)C)CO1 67840,c1(OC)ncccc1-c1cn(-c2cc(-c3ccccc3OC)on2)nn1 67841,C1(c2nnnn2C2CCC(C(C)C)C2)(Nc2c(Br)ncc(C)c2)CC2COCC2C1 67842,C(=O)(CC1=NN(C)C(=O)C1)NC1CCC(CNC(CC2CCCN(C)C2)=O)CC1 67843,c1(C(=O)NCC2CC(O)(CNC(C(C(C)C)O)=O)C2)cscc1S(C)(=O)=O 67844,C(C)(C(C)(C)C(=O)NC1C(C)(C)C1(C)C)NC(c1ccc(CC)s1)=O 67845,N1(C(c2c(C)snc2)=O)CCC2CCN(C(c3cc4n(c3)CCCC4)=O)C2C1 67846,CC1Cc2cccc(C(=O)NC3(CNC(c4ccc(F)cc4)=O)CCC3)c2O1 67847,C1(C(N(C2CCN(C(=O)Cc3ccc(OC)nc3)C2)CC)=O)CC(O)CN1C 67848,C1(NC(C2CC2Cc2ccccc2)=O)C=CCN(C(=O)C2=COCC2)C1 67849,C(CN=c1[nH]c(=NC(C)c2cc(C)on2)[nH]c2c1SCC2)OCCOC 67850,CCC(O)CC(=O)NCC1CCCN1C(c1cccc(C2CC2)n1)=O 67851,N1(C(c2n[nH]c(C)c2C)=O)CCCC12CCCN(C(C1CCCCC1(F)F)=O)C2 67852,C1(NC(Cc2c(C)nc(Cl)cc2)=O)CN(C(=O)C(C)(C)NC(N)=O)CC1C1CC1 67853,C(=O)(CCC(C)(C)c1ccccc1)N(C1CCCC(O)C1)CC 67854,c1(C(=O)NC2CN(C(c3c(CC)non3)=O)C(C)CC2)cnc(O)c([N+](=O)[O-])c1 67855,C1(=O)C2=CC(O)C(C2)N1.N1(CCNC(=O)CC2CCCCCC2)CCS(=O)CC1 67856,c1(C(=O)NC(CCNC(CCSC)=O)(C)C)cn(C)c(-c2ccccn2)n1 67857,CN1CC2(CN(C(=O)C(C3(O)CCC3)NC(=O)CCc3ccc[nH]3)C2)C1 67858,N=c1ccc(C(=O)NC2CC(CNC(c3cc(-c4ccco4)no3)=O)C2)n[nH]1 67859,C1(NC(CCc2ccc(C)s2)=O)CC2(C1)CC(CNC(C1(C)CCSCC1)=O)C2 67860,CCS(=O)C1CCCCC1NC(=O)C(=O)N(C1CCOC1)C 67861,N1(C(CCC#CC)=O)CCN(C(=O)C=C(C)C(F)F)CC2CCCCC12 67862,N1(C(c2cn(CC=C)nc2)=O)CCC2(CCN(C(=O)C(F)=C3CCCC3)C2)C1 67863,C1(C2CN(C(C(n3c(C)ccn3)C)=O)C2)CN(C(C2CCCS2)=O)CCO1 67864,C(=O)(C(F)(F)c1ncc[nH]1)NC(C1CCN(C(c2c[nH]nc2C2CC2)=O)C1)C 67865,c1(C)ccc(Br)c(Cl)c1F.Fc1ccccc1OCCn1cc(CO)nc1 67866,c1(C(=O)NC(CC=CC)C(=O)N(C(COC)CC)C)cccc(C)c1O 67867,c1(C(c2cn(CCNC(C3(C)CNC(=O)C3)=O)nn2)C)cc(F)ccc1F 67868,C1(C(=O)NC(C(=O)NCC(C(C)C)(C)F)C2CCC2)CC2(CCC2O)C1 67869,C(=O)(CC1=CCOCC1)NCC1C(C(=O)NCc2cccc(OC)n2)CC1 67870,N#Cc1ccc(Br)cc1CNCC12CC1CN(C(c1c(F)cc(F)cc1Cl)=O)C2 67871,c1(C(N(C2CCN(C(C3CC3(F)Cl)=O)CC2)CC)=O)cc(Cl)cc(Cl)c1N 67872,C1(CNC(C)=O)CC2(C1)CN(C(=O)CCc1csc(-c3ccco3)n1)C2 67873,c1(C(=O)NC(c2cccs2)C)cnc2ncc(-c3ccc(F)c4[nH]ncc34)cn12 67874,C(C(C(=O)NCC1(F)CC(CO)C1)NC(C1C=CCC1)=O)OC 67875,c1(-c2cn(CC3(C)CCC3)nn2)nc2ccccc2s1 67876,CC1CCC(NC(c2nc(Cl)ccc2F)=O)CN1c1ncc(F)cn1 67877,CCCCCCC(CC)(CC)C(=O)N(C)CC1CCCN1C(=O)C(F)C(C)(C)O 67878,N1(C(C23CCC(N=[N+]=[N-])C2C3)=O)CC(S(N)(=O)=O)CC12CCCC2 67879,CC(=O)N1C(=O)C(NC(C23C4CC(CC24)C3(F)F)=O)c2ccc(Br)cc21 67880,c1(C(N2CCC(CNC(COC(CC)C)=O)C2)=O)cc(N)cc([N+](=O)[O-])c1 67881,C(=O)(C1=Cc2ccc(Cl)cc2OC1)N(C1CCN(C(C2CC(=O)NCC2)=O)C1)CCO 67882,c1(OC)ccc2c(c1)CC1(CC1)N(C(C1C3CC(N)CC13)=O)C2 67883,C(=O)(CC(O)CC(C)C)N1C(CN(C(C(CC)C(C)C)=O)C2CC2)CCC1 67884,C(=O)Nn1cnnc1C.N1(C(C(C)N(C(C)=O)C)=O)CC(=O)NCC1C(N)=O 67885,CCC(C)CCCCC(=O)NCCN(C(C1CC2CCC1C21CC1)=O)C1CC1 67886,C1(C(=O)NCC(C)Cn2cccn2)CC(=O)CN1C(C1OCCC1(C)C)=O 67887,N1(C(C(COC)(C)OC)=O)CCC(CNC(=O)CCCN=[N+]=[N-])C(C)C1 67888,c1(C(C(=O)NC)N(CC(=O)OC)C)cn(C)nc1N(CC(C)C(C)C)C 67889,N1(C(CN(CC#C)C(C2CN3CCN2CC3)=O)=O)CC2CC(N(C)C)C(C2)C1 67890,c1(CC)cc(C(=O)NCC(C)N(C)Cc2cccc(Cl)c2F)cc(O)n1 67891,C1(C)(C(N2CCCC(CN(C(=O)C=CC=C(Cl)Cl)CC)C2)=O)CCC(=O)CC1 67892,C(=O)(CC(C(F)F)NC(=O)Cc1ccns1)NCC(C)SC 67893,Cc1ccc(-c2ccsc2C(=O)NCCCCC(C)NC(=O)CC(C)(C)F)cc1 67894,c1(OCCC=C)cccc(CC(=O)N(CCCNC(=O)CCOC(C)=O)C(C)C)c1 67895,Cn1cncc1C(=O)NCC1CC1CNC(c1cc(-c2ccco2)on1)=O 67896,c1(C(=O)NC2CN(C(C(CCC)N(C)C)=O)CC2C)cncn(C)c1=O 67897,c1(OC)cccc(CCC(N2CC=CC(NC(=O)Cc3cc(Cl)cs3)C2)=O)n1 67898,c1(C(=O)NCCCC2N(C(C(CN(C)C)O)=O)CCC2)c[nH]nc1[N+](=O)[O-] 67899,CCCC(C)(C)C(=O)NC1CCCC(CNC(=O)C=Cc2ccnn2CC)C1 67900,c1(C(CNC(=O)CC2CC(C)(C)C2)NC(c2c(C)snc2)=O)ccc(F)cc1F 67901,Cc1cc(C(=O)N)c(C)n1CCn1cncn1.N12CCCC1C2c1ccncc1 67902,CC(C)C(F)C(=O)NCCCCCNC(=O)CC1CCCC(O)C1 67903,N1(C(C2C(C(=O)OCC)C=C2)=O)CCN(C(=O)Cc2ccccc2F)C(CO)C1 67904,c1(C(=O)NCCC2CCN(C(C3CCC(C(F)F)O3)=O)C2)ccc(C(F)(F)F)nc1 67905,C1(NC(c2n(C)nc(O)c2)=O)CCN(C(c2c(Cl)cccc2Cl)=O)CC(O)C1 67906,C1(NC(C(CCC)OC)=O)CN(C(c2scc(C)c2Cl)=O)CC1N=[N+]=[N-] 67907,C(=O)(C#Cc1cccs1)N(C)C.Cc1c2cccc1N2 67908,c1(C(=O)OC)cc(C)c(CSC)cc1C(=O)CN1CC(NC(C)(C)C)CC1(C)C 67909,C1(NC(c2coc(Br)c2)=O)CCC2CCN(C(=O)CCC3CCCO3)C12 67910,CC1=C(CNC2CN(Cc3ccccc3)C(C)(C)C2)SCCO1 67911,c1(C(=O)NCC2(C)CCN(C(C3C(C#C)C3)=O)CC2)cc(C)c(F)cc1F 67912,c1(C(N2C(CNC(C(C)OCC3CC3)=O)CC2)=O)ccc(O)cc1[N+](=O)[O-] 67913,N1(C(Cn2c(C)nnn2)=O)CCN(C(=O)COc2ccc(O)cc2)C(CCO)C1 67914,C1(C(=O)NCC(=O)OCCCC)CC(O)CN1C(c1ccn(C(F)F)n1)=O 67915,C(=O)(C(C)(C1CC1)NC(C1CCCO1)=O)NCCN(C1CCN(C)C1)CC 67916,N1(CC=C)C(=S)NC(c2csc(C3CCCCC3)n2)C(C(=O)NC2CC2)=C1C 67917,CC1CN(C(=O)CCCF)CC1(C)CNC(c1ccc(CNC(N)=O)cc1)=O 67918,C12(OCC)CCC(C(N3CCC(CF)(NC(=O)CSCC(N)=O)C3)=O)(CC1)C2 67919,N1(C(Cn2c(C)ccn2)=O)CC(=O)NCC1C(N1CC(CO)CC1CO)=O 67920,N1(C(=O)N(C2CCCCC2N2CCCC2=O)CCC)CC(OC(C)=O)CCC1C 67921,c1(C(N2CCC(C(CNC(CC(C)SC)=O)F)CC2)=O)n[nH]c2c1CCCCC2 67922,c1(OCCOC)ccc(NC(=O)C(c2cnn(CC(C)C)c2)C)cc1 67923,C1(CCn2c(C3(C(=O)OCC)CCCC(C)C3)nnn2)C2CC3CC(C2)CC1C3 67924,c1(C(N2CCC(N(C(=O)CN3CCC3C)CC#C)CC2)=O)ccc(O)c(F)c1 67925,C12(NC(C(c3c(C)cccc3Br)NC(C(CSC)O)=O)=O)CC1COC2(C)C 67926,Cc1nn2cc(C(=O)NCC3CN(C(=O)C(C)N4CCC4)C(C)(C)C3)nc2s1 67927,C1(O)(CC)CCN(C(C2C(NC(=O)Cc3cc[nH]c3)C2(C)C)=O)CC1 67928,C1(C(=O)OC2CCN(CC)C2=O)CCN(c2ccccc2)CC1C 67929,C12CCCN(C1)C2=O.c1(C2N(C(C3CN(C(=O)OC)C3)=O)CCC2)cc(C)oc1C 67930,C(CC(=O)NCCS(C)(=N)=O)(CC(C)C)NC(c1c(C)cc(C)nc1)=O 67931,C(=O)(CC(O)C(C)(C)C)N1CCC(F)(CNC(c2c(C)n(C)cn2)=O)CC1 67932,C=CCC(CC)C(=O)NCC1(NC(=O)CC2(O)CCOC2)CCOCC1 67933,c1(C(=O)NCC2(C)CCC(NC(C=C(C)C(C)C)=O)C2)ccc2cc[nH]c2n1 67934,CCC(C(=O)N(CCNC(c1cc(O)cs1)=O)CCc1ccccc1)N(C)C 67935,C(=O)(C(C)(C)SC)N1C(C(=O)NC(C=C)C2CCC2)CC1 67936,N1(C(C2C(C)CC2)=O)CCC(CO)(CNC(C2CC(n3cnnc3)C2)=O)CC1 67937,N1(C(COC2(C)CCC2)=O)CC(NC(=O)Cn2cc([N+](=O)[O-])cn2)C2(CC2)C1 67938,C1(CNC(C=CC(C)NC(C=CC(C)(C)SC)=O)=O)CCOC(C)C1 67939,C(=O)(C1=CC2(CCOC2)C1)N1CC2C(CNC(c3c(C)nncc3)=O)C2C1 67940,N1(Cc2c(Br)ccc(OCC)c2)CC2CCN(C(c3cc(C(C)=O)c[nH]3)=O)C2C1 67941,c1(C(N2C(C)CCC(NC(c3csc(C#N)c3)=O)C2)=O)ccn2nccc2c1 67942,c1(OC)cc(C(N2CC(CC(N3CCC(Br)C3)=O)C2)=O)c([N+](=O)[O-])cc1F 67943,C1(CNC(C(c2cccc(F)c2)C)=O)CN(C(C2CC(=O)C2(C)C)=O)CCCO1 67944,Cc1cnc(C)c(C(=O)NCCC(C)CCNC(=O)CN2CCC(O)CC2)c1 67945,N1(C(c2ccc(-c3csc(C)n3)s2)C(=O)NC)CCCN(C2CCC2)CC1 67946,Cc1ccncc1C(N1CCC(N(CC(N2CCC(C(=O)N(C)C)CC2)=O)C)C1)=O 67947,c1(OC)ccc2c(c1)OCC(C(=O)NC(CNC(c1ccc(C)s1)=O)CO)C2 67948,CC(C)CN=C(NCC(C)(C)C(C)(C)C)N1CCC(C)(F)C1 67949,n1(CCC(=O)N(C(C)CNC(=O)Cc2cnsc2)C)cnccc1=O 67950,c1(C(N2CCC(NC(C(C)SC(C)C)=O)C2C2CC2)=O)cc(N)ccc1O 67951,CCCCC(C(=O)N1CC(CNC(c2cccnc2N)=O)C1)NC(N)=O 67952,C1(CNC(Cc2cc(C)sc2C)=O)N(C(=O)C(C)CC(C)C)CCC1(C)C 67953,C(=O)(C1=CCN(C(=O)CC2(O)CCCCC2)CC1)NC(c1nccn1C)C 67954,c1(CC)ccc(C(=O)NC(CNC(C2CC2(Cl)Cl)=O)CC)cc1[N+](=O)[O-] 67955,c1(NC(c2cccnc2SCc2cc[nH]n2)=O)cccc2c1oc1ccccc21 67956,C1(CNC(C(CSC)OC)=O)(OC)CCN(C(C2C3CC4C(C3)C24)=O)CC1 67957,CC(C(=O)NC1CN(C(=O)CC2CSCCO2)CC1n1ccnn1)C(C)(C)C 67958,C(=O)(CCCCC(OC)OC)NC(CC)CN(C(=O)Cc1ccc(Cl)cn1)C 67959,CC1(C(=O)NC(C2CCCCC2)CNC(C2CCCCS2)=O)CC2(CCC2)C1 67960,O=C1CCC(O)CN1Cc1cn(CC2CCN2C(=O)CSc2cccnn2)nn1 67961,CCC(C)CC(C(=O)NCCCn1cc(C)cn1)NC(c1cnc2n1CCC2)=O 67962,C(N=c1[nH]ccnc1F)C1CN(C(C2(C)CCCOC2)=O)CC1C(F)(F)F 67963,C12(NC(c3cc(Br)co3)=O)CCCN(C(c3cc4cccnc4[nH]3)=O)CC1C2 67964,N1(C(C(c2ccc(Cl)cc2Cl)C)=O)CCC12CN(C(c1ncccc1O)=O)C2 67965,CC(C)CC(O)CC(=O)NC1CC(CNC(c2cccc(C(C)C)n2)=O)C(O)C1 67966,C1(C(=O)NCC(C)(C)NC(=O)CSCC(N)=O)CC2(C1)CC21CCC1 67967,N1(C(C(C(C)C)O)=O)CC2(C1)SCCC2NC(c1ccc(-n2cncn2)nc1)=O 67968,C1(C(=O)NCCN(C(=O)Cc2sccc2Cl)CCC)(N(C)C)CCCCC1C 67969,CCC(C(=O)N(C)CCOCCCN(C(=O)C(C1CCCCC1)OC)C)OC 67970,C1(NC(CC(CC)CC)=O)CCCC2CN(c3nn(C)cc3[N+](=O)[O-])CC12 67971,C1(C(=O)NC(CCCNC(CCCC#CC)=O)(C)C)CCCCC12OCCO2 67972,CCC(O)C(=O)NC(C1CCN(C(=O)CCNC(c2ccoc2)=O)C1)C 67973,C(=O)(C(C)C(O)CCCC)NC1CCC(CC(=O)NCC(CCC)O)CC1 67974,c1(CC(=O)NCC(C)N(C(c2c(CC)n[nH]c2)=O)CC)ccnc(C(F)(F)F)c1 67975,N1(C(Cc2cnn(C)n2)=O)CCC2CCCN(C(=O)C=CC3CCC3)C2C1 67976,N1(C(Cc2ncc(C)s2)=O)CCC(C2(NC(C34CCCC3C4(F)F)=O)CC2)CC1 67977,C=C(C)C1OCCC1N=c1nc2c(ncn2C)c(NCC2CC2C2CC2)[nH]1 67978,c1(CC(=O)NC(c2ccccc2F)CNC(CC=C=C)=O)cn(C)nc1C(F)F 67979,c1(OC)ccc(C(N2CC(NC(C3CC(O)(C(F)F)C3)=O)C2)=O)cc1 67980,C=C1CCN(C(c2cccs2)=O)C(C(=O)NCc2cc(C)ccc2O)C1 67981,C#CCC(C)C(=O)N(CC(C)(C)NC(c1cn(CC2(CC)COC2)nn1)=O)C 67982,c1(C(=O)Nc2cccc(F)c2I)cc(Cl)c2cnccc2c1 67983,c1(C(=O)NCCCC)cc([N+](=O)[O-])c(C(=O)N(CC(=O)C2(Cl)CC2)C)cc1OC 67984,C#CCC(O)C(=O)N1CC(C(=O)NCCc2ccn(C)n2)C(CC)C1 67985,c1(OC)nc(C(=O)NC2CN(C(=O)C=Cc3cncnc3O)CC2O)cc(O)n1 67986,C1(C(=O)OCC(=O)Nc2c(C(C)=O)cc(OC)cc2)CCC2(CCC2)C1 67987,N1(C(c2cc(C)[nH]c2)=O)CCCC(O)(CNC(c2c[nH]cc(F)c2=O)=O)C1 67988,c1(C(=O)NC2CN(C(=O)CCc3nccs3)CC2O)ccc(F)cc1Br 67989,c1(C(=O)NC2CCCC(NC(C(C)CC(N)=O)=O)C2)cc(Cl)c(F)cc1O 67990,c1(C(N2CCCC(NC(c3c(OC)oc(C)n3)=O)C2)=O)c(C)cc(C)cc1C 67991,CC1(CNC(c2cc(C#N)c[nH]2)=O)COCCN(C(=O)CN2CSCCSC2)C1 67992,c1(C(=O)NCCC(C)NC(C(CC)N(C)C)=O)cnc2ccnn2c1 67993,c1(C(=O)NC(C(C)C)CNC(=O)Cc2ccccc2F)ccc2[nH]ccc2n1 67994,CC1(C)CCCCC1=CC(=O)NCC=CCNC(=O)CC1CCC(=O)O1 67995,C1(C(N(CC(C)(C)C(=O)NCC2SCCS2)C)=O)CCC(C2CC2)C1 67996,C1(NC(COc2c(C(C)=O)cccc2)=O)CCN(C(=O)CC2CCCO2)CC1C 67997,C1(c2nnnn2Cc2ccco2)(NCc2n(CC)ncc2)COCCO1 67998,c1(C(N2C(C)(CNC(COCC)=O)CCC2)=O)ccc(=O)n(C)n1 67999,Cn1[nH]c(=NNC(=O)C2CN(S(C)(=O)=O)C2)s1.c1(N)ccc(Cl)cc1 68000,C1(NC(Cc2scc(C)n2)=O)CC(NC(=O)Cc2ccn(C)n2)C12CCOCC2 68001,c1(C(N2CCN(C(c3c(C)cns3)=O)CC2C)=O)ccc(S(C)(=O)=O)s1 68002,N1(C(CCC2(C)CC2(F)F)=O)CCC12CCNC2=O 68003,c1(C(C(N)=O)N(C(c2cccc(Cl)c2)C(=O)NCC)C)ccccc1I 68004,C1(C2CCN(C(c3cccnc3N)=O)C2)(NC(C(C2CC2)SC)=O)CC1 68005,C1(C)(CNC(C2CC(N(C)C)C2)=O)CCCN(C(c2cc(C3CC3)on2)=O)C1 68006,Cc1ccc(C(CO)NC(=O)NC(C2CCC(C)O2)C2CC2)c(Br)c1 68007,C1(CC(=O)NC2(CCOC)CC2)CC2(CC2)CN1C(=O)CC1CCC=CCC1 68008,C1(NC(Cn2c(C)nc(C)n2)=O)COC2(CCN(C(c3nnn(C)c3C)=O)C2)C1 68009,C(N=c1[nH]c(N2CCC3CC3C2)nc(=N)[nH]1)C1(SC)CC1 68010,C(=O)(C1=Cc2ccccc2C1)NC1C2(CCN(C(CCSCC)=O)C2)C1 68011,C(c1ccc(-c2ccccc2)cc1)=CC(=O)NC1CC(NC(C=CS(C)=O)=O)C1 68012,C(=O)(C1CCCc2ncccc21)N1CC=C(CNC(C2C(C)CCCC2)=O)CC1 68013,C1(NC(c2cnc(O)s2)=O)CCN(C(c2ocnc2C2CC2)=O)CCC1(F)F 68014,N1(C(CC2C(C)(C)CC2)=O)CC(NC(=O)CCC2CCCCCC2)C2(CCC2)C1 68015,C=CCCN=C(NCc1ncnn1C(C)(C)C)NCc1ncc(C(F)(F)F)s1 68016,N1(C(c2c[nH]c(=NC)o2)=O)CCC2(CC2NC(=O)CN2CCCC2)C1 68017,CC1(CNC(C2CCCCN2C(N)=O)=O)CCN(C(=O)C2=CCCSC2)CC1 68018,c1(CCC)c(C(N2CC(CNC(=O)CCN3C(=O)CNC3=O)C2)=O)cnn1C 68019,N1(C(COCCC)=O)C2CCC(C(N3CC(OC)C(OC)C3)=O)C1CC2 68020,C1(N(C(c2nc(C)oc2)=O)C)CCCN(C(=O)COC2CCCCCC2)C1 68021,C(CC)(C(=O)N(CCc1ccccc1)CCc1cccnc1)OCC 68022,N1(C(=O)CC2CN(C(c3ncccc3Br)=O)CCO2)CCn2nccc2C1 68023,N#Cc1cccc(OCC(N2CCCC2c2nc(C(=O)O)co2)=O)c1 68024,Cn1nc2c(c1NC(C1CSCCN1Cc1cc(F)ccc1Br)=O)CCC2 68025,N1(C(C(C2CC2)OC)=O)CC(O)(C2(CNC(C3(Cl)CCC3)=O)CC2)C1 68026,C(=O)(C1=CC(C)(CC)C1)NCC(CN(C(=O)Cn1cc(C)cn1)CC)(C)C 68027,C(CCCCC(=O)N1CC(NC(=O)C=Cc2ccccn2)C(C)C1)=CC 68028,C1(O)(CN(C(C2(OC)CC2)=O)C)CCN(C(C2CCCOC2C)=O)CC1 68029,C1(C(=O)NCC#CCNC(c2cccc(C3CC3)c2Cl)=O)CC2CCC1CC2 68030,C(=O)(CCCC(F)F)NCCC1CCCN(C(C2CCCN(S(C)(=O)=O)C2)=O)C1 68031,C1(NC(CCCCCSC)=O)CCCOC12CCN(C(c1cc(F)n[nH]1)=O)CC2 68032,C(C)(c1cccnc1)=CC(=O)NCCN(C(=O)C(F)C(F)(F)F)CCC 68033,S(=O)(=O)(c1[nH]c(=NCc2c(C)cccc2Cl)ccc1Br)NCCOC 68034,C1(=O)CC(=O)N2CCC(C2)N1CC#C.C(=O)(C(=O)NC1CCCC1)NC 68035,C(=O)(CN=c1ccc(C#N)c[nH]1)N1CCCC(N(C(C(CCC)C)=O)C)C1 68036,C(=O)(CC(F)(F)C(F)(F)F)N1C(CNC(c2cncs2)=O)CCC1 68037,CCC(CC(=O)NC1CC(CNC(c2cnns2)=O)C12CCC2)CC(C)C 68038,CC(CCNC(c1cc(Br)co1)=O)CCNC(C1CCS(=O)CC1)=O 68039,CCCCC(C)CCC(=O)NCC1CCC(C(=O)NC(C2CCCC2)C)O1 68040,O=C1COC2(CCN(C(c3ccc4nsnc4c3)=O)C2)CN1 68041,C1(F)(CNC(C2C(C)=CCS2)=O)CCC(NC(c2nccnc2C)=O)C1 68042,N12CC=CC(C1)C2=O.N1(CC)CCC1C(=O)NCC=CCC1CCCC1 68043,Cc1c(C(N2CC(NC(c3cnn[nH]3)=O)CCC2C)=O)sc2nnc(S)n12 68044,C(CC(C)C)(C(=O)NC1CCN(C(=O)C(c2ccccc2Cl)C)C1C)OC 68045,C1(CCC)(NC(c2ccc(C(F)F)o2)=O)CCCN(C(c2cccc(C)n2)=O)C1 68046,C1(OC)CCN(C(=O)CNC(N2CCCC2)=O)C1NC(c1ccoc1C1CC1)=O 68047,c1(C(=O)Nc2c(F)cc(C)c(Br)c2)ccc2nnc(C(F)F)n2c1 68048,C(C(CNC(C1(CC(C)C)CCC1)=O)OC)NC(C1C(CCC)C1)=O 68049,N1(C(C(CC2CCC2)NC(c2ccco2)=O)=O)CCC(C(F)F)CC1 68050,C1(C)(NC(C2C(C(=O)NCC#C)C2)=O)CCN(C(c2oc(C)nc2CC)=O)CC1 68051,CC(C)C(CCNC(=O)C(C)O)NC(=O)C(C(C)O)c1ccccc1 68052,CC1CN(C(C2(F)CCOCC2)=O)CCC1N=c1[nH]c(Cl)ncc1Br 68053,c1(C(N(C2CCN(C(c3cnc(=N)[nH]c3)=O)C2)CCC)=O)cccc(F)c1CC 68054,C1(C(=O)NCCN(C)C(C2CC(C)(C)O2)=O)CC2(CC2)C1 68055,C1(F)(C(N2CC(CNC(C3(CC)CCC3)=O)OCC2)=O)CCC(C)CC1 68056,c1(-c2c(C(=O)NC3CCN(C(C=CCN(C)CC)=O)C3)nco2)ccccc1F 68057,CC1=C(C(=O)NC(C(=O)NCc2cc(F)ccc2F)C2(O)CCC2)SCCO1 68058,Cc1nc2c(N3CCN(C(c4c(F)cncc4F)=O)C4CC34)ncnc2[nH]1 68059,N(C1CCc2ccccc21)C(CCCCNC(CC=C)=O)=O 68060,c1(C(=O)NCC2CC(C(N3CC=C(C)CC3)=O)C2)cc(C#N)n(C)n1 68061,c1(C(N2C(C(C)C)CCC2)=O)cccc(S(=O)(=O)N(C(=O)Cc2cc[nH]n2)C)c1 68062,c1(C(=O)OCC)nc(C(N2CCC(C(C)NC(=O)CC3CCC3)C2)=O)cs1 68063,c1(C(N(C2CCCN(C(=O)CCC3(C#N)CCC3)C2)C)=O)nn(C)cc1Br 68064,c1(C2C(Cl)(Cl)C2)nc(CCN2CCCC2)nn1CC1CCCCO1 68065,N1(C(c2c(C)cnn2COC)C(=O)NCCCC)CCN(C(C)CC)CC1 68066,Cc1ccc(C#N)c(NC(C2CC(NCc3cncs3)C2)=O)c1 68067,N1(C(C(=O)Nc2ccc(F)cc2C2CC2)=O)CCc2ccc(Cl)nc2C1 68068,c1(OC)c(C)csc1C(N1CC(F)CC1CN(C)C(c1cnc(C)[nH]1)=O)=O 68069,c1(C(=O)NC(C2CN(c3snc(C(C)(C)OC)n3)C2)C)ncc(F)cc1F 68070,c1(NCN(CCNC(CCC)=O)CC)ccc(C#N)c([N+](=O)[O-])c1.C1(=O)CN1CC 68071,C1(NC(C(C=C)(C)CCOC)=O)CCC2(CC1)CCN(C(c1cnc(C)[nH]1)=O)C2 68072,C1(CNC(c2ccc(N(C(C)=O)C)cc2)=O)CCC(C)N(C(=O)CSC(C)C)C1 68073,CCC(C(=O)OC(C)(C)C)C(=O)NCCN(C(=O)C(C(C)(C)C)OC)C 68074,c1(OC)ccc(C(=O)NC2CCN(C(=O)CC3CC34CC4)CC2)c(F)c1Cl 68075,C(=O)(CC(CNC(C1C=CCCC1)=O)C1CCC1)N(CCC#C)C 68076,C12(C(=O)NC3CC4(C(NC(CCCC#N)=O)C4)C3)CC3CC1(CO)CC3C2 68077,c1(C(=O)NCC(C)(C2CC2)NC(c2cc(CC(F)(F)F)c[nH]2)=O)ncc(F)cn1 68078,N1(C(C(C=C)c2ccccc2)=O)CCC2CCN(C(C3(C)CC(C)C3)=O)CC12 68079,C12(C(N(CCNC(=O)CCSCC(C)C)CC)=O)CC(C)C1C2 68080,c1(C(=O)OC)cnc(F)cc1NCC(S(=O)(=O)OC)COC 68081,C1(NC(C=CCOC)=O)CN(C(C2CCCN2C(=O)CCC)=O)CC1F 68082,C1(O)(C(C(=O)NC2C(O)CC2O)NC(N)=O)CCCCC1 68083,C(=O)(CCCCCC(C)(C)C)NC(c1ccnc(N2CC(OC)C2)n1)=O 68084,CC(CCCNC(c1csc(O)n1)=O)NC(c1csc(O)n1)=O 68085,c1(C(=O)NCCC(=C)CNC(=O)CC2CCCOC2)ccccc1SC 68086,C1(C(=O)O)(CO)CCC(F)(F)CC1.C1(NC(=O)C=Cc2cc[nH]n2)CCCC1O 68087,C(CCC(C)CC(=O)NC(C1CN(C(c2cnn(C)c2C)=O)C1)C)=C(C)C 68088,N1(C(C=CCCC)=O)CCC2(CCCC2NC(c2cnc(N(C)C)o2)=O)C1 68089,c1(C(=O)NC2C(NC(c3n(CCC)ncc3)=O)C2)nn(C)c2c1CCC2 68090,C1(C(=O)NC(CNC(=O)CC2(O)CCC2)C2CCC2)(CC)CCCCC1 68091,C(=O)(C1c2c[nH]nc2CCC1C)NC1C(S(CC)=O)CCCCC1 68092,C1(C(=O)NCC2(F)CN(C(C(CSC)C)=O)C2)CC2C(C1)C2(C)C 68093,C(=O)(C(O)C(CCC)NC(c1cnc(Cl)n1C)=O)NCCC#C 68094,n1(C(CC)C)nc(C(=O)NC(C)CNC(=O)C=Cc2csc(C)n2)cc1C 68095,C(=O)(C(F)C(C)CNC(=O)C(C)(C)C(F)F)NCCc1c(C)ncs1 68096,c1(C(=O)NC2C(C(=O)Nc3cncc(OC)n3)C2)csc2ccc(Br)cc12 68097,c1(NC(C2C(NCc3c(C(=O)O)cccc3)C2)=O)nc(Cl)c(Br)cc1O 68098,c1(N(C2CCCN(C(CCC(C)SC)=O)C2)C)snc(C)c1C#N 68099,C1(N(C)C)CN(C(c2cocc2Br)C(=O)NC2CCOCC2)CC12CC2 68100,c1(C(=O)NC2C(F)CCN(C(C=Cc3c(C)ncs3)=O)C2)ccc2c(c1)CCC2 68101,c1(OC2CCN(C(N(c3cc(F)ccc3Cl)CC)=O)CC2)cccc2[nH]ccc12 68102,Cc1c(C(=O)OCC(=O)Nc2ccccc2)cccc1O.c12ccccc1C(=O)N2 68103,C(N=c1[nH]c(=NCCC(C)CO)c2c(F)cccc2[nH]1)c1ccc(C)cn1 68104,c1(C(=O)NC(CCCCNC(C(C)(C)OC)=O)CO)ncc2ccccn12 68105,C1(NC(c2c(C)onc2)=O)(CNC(C2(C)CCCO2)=O)CC2CCC1CC2 68106,C1(CC(=O)NC)CN(C(=O)Cn2cc(Cl)cn2)CCN1C(=O)C(C)CC1CC1 68107,C1(C(=O)NCC(n2cccn2)C)CCOCCN1C(c1ccc(C#N)o1)=O 68108,c1(C(=O)NCC2C(NC(C3(C)C=CCCC3)=O)CCC2)cc(F)c(F)c(O)c1F 68109,c1(C(=O)NCCN(C(C2CCC(=O)NC2)=O)CC)coc2ccccc12 68110,C=Cc1cc(C(=O)NCC2(C)CCN(C(c3ccc(C(C)C)s3)=O)C2)cc(F)c1 68111,c1(COC)nn(C)c(Cl)c1C(N1CCCC1CNC(C1CC(C)(C)C1)=O)=O 68112,Cc1ccc(C=CC(=O)NCC(C2CC2)NC(=O)C(n2nccc2C)C)cc1Cl 68113,C1(CC(=O)NCC(CC)C(C)C)CCN(C(=O)CC2CCC(=O)C2)C1(C)C 68114,c1(NC(Cc2nc(CCC(CCC)O)on2)=O)cc(N(C)C)cc2cccnc12 68115,N1(C(CSC)=O)Cc2ccccc2C(CNC(c2cnc(NC(C)=O)o2)=O)C1 68116,C1(CNC(C=C(C)C(C)(C)C)=O)CC2CN(C(C3(C#N)CC4CC4C3)=O)CC12 68117,CCC(CC(=O)NC(C)(C)CC(F)C(=O)N(CC(=O)NC)C)CC(C)C 68118,N1(C(=O)Cn2cnc(Br)c2)CCC2CCCC(C1)N2C(C1C2COCC12)=O 68119,C1(CC(=O)NC(C)C(C)(C)NC(c2cocn2)=O)CS(=O)(=O)CCO1 68120,C1(C(N2CC(CNC(C=CCC)=O)C2)=O)CC(C2CCOCC2)=NO1 68121,CC(C)(O)C(F)C(=O)N1CCOC(C2CN(C(c3cncc(N)n3)=O)C2)C1 68122,N1(C(Cc2ccc(OCC)nc2)=O)CCC(C2(NC(C3CC3COC)=O)CC2)C1 68123,CC1(C)CN(C(c2ccon2)=O)CC1NC(c1cc(-c2ccco2)cs1)=O 68124,CCCCS(=O)(=O)NC(N(C)CCCc1cn(-c2ccccc2Cl)nn1)=O 68125,N1(C(c2c(OCCC#C)cccc2)=O)CC2(C1)CN(C(=O)C=CC=CC)C2 68126,C1(NC(C(CSC)(C)C)=O)CCCN(C(c2cc3sccc3s2)=O)CC1 68127,CN1CCC(C(=O)NC(CNC(C2CN(C(=O)OCC(C)(C)C)C2)=O)CO)CC1 68128,C1(C2CCN(C)CC2)(CC2CC(C)N2C(=O)CCC(N)=O)CC1.c12cn(nn1)C2 68129,CC1CCCC(OCCNC(=O)NCc2ccsc2)C1 68130,CC1(C(=O)NCc2cccc(Cl)c2F)CCCN(Cc2nccs2)C1 68131,c1(CC(=O)NC2CC(CCNC(CCSC)=O)C2)ccc(OC(F)(F)F)c(F)c1 68132,c1(OC)nc(C(N2CCCC(CNC(=O)CCC3CCCN(C)C3)C2)=O)sc1C 68133,c1(C(N(C)Cc2c(OCc3c(OC)cncc3)cccc2)=O)nc(Cl)ccc1F 68134,N1(C(c2n[nH]cc2C(F)(F)F)=O)CC(N=c2[nH]nc(C(F)F)o2)C2(CCC2)C1 68135,N1(C(C)=O)CCCC(O)(CC(N2CC(O)(CNC(=O)CNc3ccsc3)C2)=O)C1 68136,CCC(CC)CC(=O)NCC1CN(C)CCN1C(c1cc(C)nn1C(F)F)=O 68137,n1(COC)nccc1C(N1CCC(OCC(=O)NC(C)Cc2ccnn2C)C1)=O 68138,CC1(CNC(=O)C2=CCOC2)CCCN(C(=O)C(C2CCOCC2)F)C1 68139,C(=O)(CC(=O)NCC1CC(N(C)C(c2c[nH]nc2C(C)C)=O)C1)OC 68140,N1(C(C)=O)CCN(C(=O)CCCn2cc(CCOC(C)=O)nn2)CC1 68141,Cc1nn(C)c(C)c1C(N1CC(NC(=O)CN2CCCS2(=O)=O)CC(O)C1)=O 68142,N=c1[nH]cc(C(=O)NCC(O)CNC(c2cscc2F)=O)c2cc[nH]c12 68143,C1(C(N(CC(CN(C)C(c2cnncc2O)=O)O)C)=O)CCC(O)CN1C 68144,N1(C(CC=Cc2ccc(C)cc2)=O)CC2(CCC1C(=O)O)OCCO2 68145,c1(C(=O)NC2CCCN(C(C(CC)NC(C)=O)=O)CC2)cc(=O)c(OC)cn1C 68146,c1(NC)snc(C)c1C(=O)NCC12CC1CN(C(=O)COCC1CCOCC1)C2 68147,c1(C(=O)NCCN(C(CCC2CC(OC)C2)=O)C)ccc(N)c2ccncc12 68148,C1(C2(O)CCOCC2)(C(N2C(C(=O)OCC)C(O)CC2)=O)CC1 68149,c1(OCC)cccc(C=CC(=O)N(C(C)CNC(=O)Cc2c(C)noc2C)C)c1 68150,c1(C(=O)NC)cccc(CCNC(=O)NC2CCC2C(C)(C)C)c1 68151,Cc1cnc(C(C)NC(=O)C(C2CCCCC2)C2CCNCC2)s1 68152,N1(C(CC=C(C)C)=O)CCC(NC(c2cc(C(F)(F)F)ccc2N)=O)CC1C 68153,C(=O)(C(C)(CC)CO)NCCCC.c12nc(cc(O)n1)CN2CC 68154,CC1CCCN(C(c2ccccc2)CNC(=O)Nc2conc2C2CCNCC2)C1 68155,C(=O)(C(O)C(C)(C)C)N1CC(C)C(NC(=O)Cc2ccncc2Cl)C1 68156,C#CCC(C)(CC)C(=O)N1CCCC(CC(N2CCc3sccc3C2)=O)C1 68157,C(c1ccc2occc2c1)=CC(=O)NCC1C(NC(C(C(C)O)C)=O)CCC1 68158,C(=O)(CC(C)CC(F)(F)F)N1C(CCNC(C=C(C)C2CC2)=O)CCC1 68159,CCC(CC)(C(=O)N=c1ccn(C(C)C)[nH]1)Oc1ccccc1 68160,C1(C(=O)OCC)COCC1C(=O)N(CCCCNC(=O)C(c1cccs1)SC)C 68161,c1(NC(C(=O)NCCN(C(CC)C)C)=O)ccc2c(c1)C(=O)OC2(C)C 68162,C(CNC(c1ccc(CO)nc1)=O)(CC(F)(F)F)NC(COCCOC)=O 68163,c1(C(N2CCC(C(=O)NCC)CC2)=O)ccc(F)c(-c2c(C)cccc2F)n1 68164,c1(CNC2C(CC(=O)OC)CC2)nnc(-c2ccccc2)s1 68165,C1(NC(C(CC)C)=O)CN(C(C2(Cc3ccccc3)COC2)=O)CC1(C)C 68166,c1(CC(C2CCOC2)NCCCCOC(C)=O)cc(C)nn1C 68167,N(C(=NCC1CCOC1C1CC1)N1CCC(c2ccccn2)C1)CC(C)(C)OC 68168,Cc1cc(C)n2nc(C(C)NCCOc3cccc(Br)c3)nc2n1 68169,c1(SCC)ccc(Cl)cc1C(=O)N(CC(CC)NC(=O)C(F)CC1CCC1)C 68170,C12(NC(C(COC)COC)=O)CCC(F)(F)CC1CN(C(=O)C(F)C(C)(C)O)C2 68171,CC1CN(C(=O)CN(C2CC(C#N)C2)C(c2csc(C#N)c2)=O)CCCO1 68172,c12cc(Br)ccc1S(=O)(=O)NN2.C12(NC(CN(CC)CC)C)CC(C)(CCO1)C2 68173,C1(NC(C(C)C)=O)CCN(C(c2csc(C(C)(C)C)c2)=O)CC1CO 68174,C#CCCCCCC(=O)NCC1(F)CN(C(c2c(C)csc2C)=O)C1 68175,C12(CNC(C3N(C)CCC3)=O)CCCC(CN(C(=O)C(F)C3CCC3)C1)C2 68176,O=S(=O)(c1cccc(COCCCC(F)(F)F)c1)NCCF 68177,c1(NC(=O)Nc2cnn(C)c2C(F)(F)F)c(F)ccc2c1OCC2 68178,C12(CNC(CC3N(C(C)C)CCC3)=O)CC1CN(C(C1CC(C)CCO1)=O)C2 68179,C(=O)(CCCCCOC)NCC1C(C(N2CCC(=C)C2)=O)C1 68180,c1(C(=O)NC(C(C(C)C)NC(=O)Cc2cn[nH]c2)C)cc(=O)c2ccccc2[nH]1 68181,C1(NC(=O)NCCC2(O)CNC2)COCC1n1cccn1 68182,CC(Cc1ccccc1)(C(F)F)NC(=O)OCC(F)(F)F 68183,c1(C(=O)NCC2CN(C(CC(C=C)C)=O)CC2O)n[nH]c2c1CS(=O)(=O)CC2 68184,c1(C(N2CCCC(CNC(CCC3CC(C)C3)=O)C2)=O)cn(C)c(=O)n(C)c1=O 68185,N1(C(C=C2CCC(C)CC2)=O)CCC(O)(C(C)NC(=O)CC(C)(F)F)CC1 68186,c1(Cn2c(C(CC)NC(C)CCC(C)C)nnn2)cc(C(F)(F)F)ccc1C#N 68187,C#CC1(C)CCN(C(C2(CC=C)CCCN2C(C2CN3CCC2C3)=O)=O)CC1 68188,CC(C)(C)C(CNC(=O)CN1CCOCC1=O)C(=O)NCc1ncc(CO)o1 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68206,C(C)(C)(CCCNC(C1CCC(C)O1)=O)NC(c1c(C(C)C)ncs1)=O 68207,C1(CNC(C(C=CCCC)O)=O)CCCN(C(=O)CNC(=O)CCC(C)C)C1 68208,N1(C(C(C=C)(C)O)=O)CC(NC(C2CC3(CCOCC3)C2)=O)CC2(CCC2)C1 68209,C1(NC(C=C(C)C(C)C)=O)CCN(C(C23CC(C)(CCO2)C3)=O)CC1C(C)C 68210,Cc1cc(C(c2ccco2)NCc2cn(C3CCOC3)nn2)on1 68211,c1(N2C(CC(=O)Nc3cc(CCC)no3)COCC2)ncc2cccc(Br)c2n1 68212,C1(C)(CCNC(C(C=C)C)=O)CCN(C(=O)COc2ccsc2)C1 68213,c1(C(N(C(CNC(C(C)CC2CCC2)=O)C)C)=O)c[nH]c2nccc-2c1 68214,C1(CNC(c2ccn(CCC)n2)=O)CC(NC(=O)C(O)CC2CCCC2)C(O)C1 68215,N1(C(CCOCC)=O)CCN(C(C23CC(C2)S(=O)(=O)C3)=O)CC1C 68216,c1(C(N2CCCN(C(CC(=C)C)=O)CC2)=O)cc(F)c2cn[nH]c2c1 68217,Cc1nc(CC(=O)NC2(C(=O)NC3CC3C)CSC2)cs1 68218,N1(C(C)=O)CCC(C#N)(NC(C2(CO)CCNCC2)=O)C1 68219,c1(C(N2C(CNC(C3C(C(C)(C)C)C3)=O)CCCC2)=O)cc(N)nc(Cl)c1 68220,N1(C(CNC(CCC(C)C)=O)=O)CCC(NC(=O)CN2CCC2)C(C)(C)C1 68221,CC1(C(N2CCCC(CNC(=O)CCCc3ncco3)CC2)=O)CCCNC1=O 68222,c1(COC)cnc(OC)c(C(=O)NCC(C)CNC(=O)COC2CCCOC2)c1 68223,C(=O)(C1=C(Cl)CCCC1)NC1(O)CCN(C(CCOC(CC(C)C)C)=O)CC1 68224,CCC(CC)C(C)C(=O)NCC(C)(CC)NC(=O)CSc1nncn1C(C)C 68225,c1(CN(C(CN(C)CC)=O)C)ccc(CC2(C(=O)NC)CC2)cc1 68226,N1(C(c2scc(C)c2Cl)=O)CCC(CNC(=O)CC2CCC(C)O2)C(F)(F)C1 68227,c1(C(N2CC(c3cn(C4(C(=O)OC)CC4)nn3)(C)C2)=O)ccnnc1C 68228,C(=O)(C1CCc2cccnc21)NCC#CCNC(C1CCC(=O)O1)=O 68229,N1(C(c2cnc(CC(C)C)s2)=O)CC2CC(NC(=O)CC3=NNC(=O)C3)CC1C2 68230,CCCC(C)(CC)C(=O)N1CCCCCC(C(=O)N2CC=CCO2)C1 68231,O=C(C1=COCC1)NCC1CN(C(=O)Cc2cccc(OC3CC3)c2)CCO1 68232,C1(CC#C)(C(=O)NC(CN(C(=O)C(C)(C)F)C)Cc2ccccc2)CCOCC1 68233,C1(OC)CCC(C(=O)OC2(C(=O)NCc3ccc(Br)cc3)CCOC2)CC1 68234,C12(C(=O)NCC3C4CN(C(C(C)(C)N(C)C)=O)CC43)CCC(C)(C(=O)O1)C2(C)C 68235,Cc1nc(N2CCC3(CC3C(=O)NC(C)(CO)CO)C2)c2sccc2n1 68236,c1(C(=O)NCCOCCNC(=O)C(F)C2CCOC2)cccnc1N1CCC1 68237,CC1CC(NC(C2(F)CCC2)=O)CCN1C(=O)C(C)C1CC1 68238,C1(C(N2CCC(C)(NC(c3nc(C(C)C)oc3)=O)C2)=O)CC12CC(F)(F)C2 68239,N1(C(C2(c3ccccc3)CC2)C)C(C(N2CCC(C)C2)=O)CC2CC12 68240,C1(C(=O)Nc2ccc(CO)cn2)CN(C(C2(C3CC3)CC2)=O)CC1C1CC1 68241,C(=O)(C(O)CCC(F)(F)F)NC(C1CCCC1)CNC(CC(COC)(C)C)=O 68242,c1(C(N2CC(NC(Cc3c(C)cccn3)=O)C(C)C2)=O)c(C)nc2cccnn12 68243,C1(CNC(c2ccc(Cl)cn2)=O)C2CN(C(=O)CCc3cncc(F)c3)CC12 68244,N1(C(c2c(CC#N)ccs2)=O)CCC(O)C(O)c2ccccc21 68245,c1(CNC(C)=O)c(F)cccc1Br.c12ccc(s1)C(=O)N1CC(C1)CO2 68246,Cc1ccc(C=CC(N2CCN(C(=O)Cn3ccnc3C)C(C)C2C)=O)cc1Cl 68247,C1(CC=C)(C(=O)NC(C2CN(C(C3CCC(F)C3)=O)C2)C)CCCCC1 68248,CCCCC(CC)CC(=O)N1CC(F)CC1CN(C(=O)CC(C)(C)C(F)F)C 68249,C1(NC(C2C(C)CN(C(c3cnc(O)n3C)=O)C2)=O)CCN(C)CC1C#N 68250,C(CC(C(=O)N(C)CCN(C(=O)C=Cc1cocn1)C(C)C)NC=O)[SH](C(C)C)C 68251,C(=O)(CC1=NNC(=O)C1)N1C2C(NC(CN(C)C(N)=O)=O)C(C2)C1 68252,O=C(C#CC1CCOC1)NCCCN(CCO)C(C1CCOC2(CCC2)C1)=O 68253,C=CC1CCCC(c2nnnn2C2COC2)(NCCc2nc(COC)no2)C1 68254,C(CC(=O)NC1CN(C)CC1OC)(C(C)OC)NC(c1c(CCC)nco1)=O 68255,C1(c2n(CC(=C)C)nnn2)(NCc2ccccc2-n2cncn2)CC(C)N(C)C1 68256,c1(C(=O)NCC(C(=O)NCC(COCC)C)O)ccc2[nH]ccc2c1 68257,Cc1cscc1C(=O)NC(C(=O)NCCc1cn(C)nn1)C1CCCO1 68258,c1(NC(C2N(C(c3c(COC)cco3)=O)CC2)=O)ccc(O)c(OC)c1 68259,C1(NC(CCN2CCC(C)CC2)=O)CN(C(=O)CNS(=O)(=O)C2CC2)C(C)(C)C1 68260,c1(C(=O)NCCOC2CCN(C(C3(OCC)CCOC3)=O)C2)c(C)ncn1C 68261,C(=O)(C(C(=O)NC12CC(C1)N(C(C1(CO)CC1)=O)C2)C(C)C)OCC 68262,c1(C(=O)NCC2(C)CCN(C(C(C(C)C)NS(N)(=O)=O)=O)C2)cccc(=O)n1O 68263,C1(CC)COCCN(C(C2CCCN(C(c3cnn(CC)c3C)=O)C2)=O)C1 68264,c1(C(=O)NC2CCCCN(C(C(C(C)C)(C)C)=O)C2)cc2c(nc1N)CCC2 68265,c1(C(=O)NCC2N(C(C(C)Oc3cccnc3)=O)CC2)cnccc1C1CCC1 68266,N1(C(C)C)CC(C(N2CC=CC(NC(=O)C(=O)NCC(F)(F)F)C2)=O)CC1=O 68267,C1(C(=O)NCc2c(C(=O)NCC(C3CC3)SC)con2)CCC(C)=C(C)C1 68268,C1(C(COC(c2n(CC#C)ccc2)=O)=O)CCCN(C(=O)C(C)(C)C)C1 68269,C(C(O)C(=O)NC1CC(F)(CNC(c2cscc2Cl)=O)C1)SC 68270,C1(NC(C2C(c3nc(C)[nH]n3)OCC2)=O)CCN(C(C23CC2C3)=O)CCC1(F)F 68271,C(=O)(C(C)(C)CS(N)(=O)=O)NCC1(F)CC(NC(CC(=O)NCC#C)=O)C1 68272,C(=O)(CC1=CCN(C(C2CCN(C(C)=O)C2)=O)CC1)N(C(C#C)C1CCC1)C 68273,Cc1cccc2nc(C(=O)NCC(O)CNC(C34CCCCC3C4)=O)cn12 68274,C1(F)(CNC(C2C(OC(C)=O)C2)=O)CC(CNC(C2(F)CC2)=O)C1 68275,c1(C(N(C(C)CCNC(=O)C=Cc2ncc[nH]2)C)=O)cc(F)c(F)c(N)c1Cl 68276,c1(CC)ncc(C(=O)NCC(n2cc(CN3CCNC(=O)C3)nn2)C)c(C)n1 68277,CC1CCN(C(c2cc3sccc3s2)C(=O)NCC(=O)NC2CCCCC2)CC1C 68278,c1(CC)nn(C)c(C(=O)NC2CCN(C(=O)C(C)(C)Cl)C2)c1Cl 68279,N1(C(=O)OC)CCN(C(C2CCCN2Cc2csc(C(C)=O)c2)=O)CC1 68280,CCC(C)C(CC(=O)N1CCn2nncc2C1)NC(=O)CSCC(F)F 68281,c1(OCC(=O)NC2C(CN)CN(C(=O)CO)CC2)ccc(F)c(F)c1 68282,C(=O)(CCCCNC(N)=O)NCC(C)(C)CNC(C1(C)CCNC1=O)=O 68283,C1(NC(=O)C2=CC(c3ccccc3)C2)CCC2(CC1)CC2NC(C1CC1(F)F)=O 68284,C=CC(C)CC(=O)NC(CNC(=O)CC1CNC(=O)O1)C(C)C 68285,C1(C(=O)NC2(CC)CCOC2)CCN(C(C2CCCN2C)=O)CCO1 68286,N1(C(CCCC2C(C)C2)=O)CCCC(NCCC2CC(F)C(=O)N2)C1 68287,Cc1ccc(-n2nnnc2N2CC(NCC)CC2C)cc1.C1(C)(C=O)CCC(C)C1 68288,c1(N2CCC(F)(CNC(c3ccc4nccn4c3)=O)CC2)ncnc2[nH]cnc12 68289,c1(C(=O)NCCCCNC(C(CC)c2cccnc2)=O)ccc(Cl)nc1O 68290,c1(NC(C)=O)ccc(C(=O)NCCN(C(=O)CCC(N)=O)C2CC2)c(O)c1 68291,C1(C(=O)NC2(CO)CN(C(C(=Cc3cnc[nH]3)C)=O)C2)CCS(=O)(=O)N1 68292,c1(CC(=O)NCCNC(c2cn(C3CCC3)nn2)=O)ccc(F)cn1.C1(N)CCSC1 68293,CCC(F)(C(=O)OC)C(=O)NCCNC(c1ccc(CCF)cc1)=O 68294,N1(C(C(C)CCN(C)C)=O)CCC(C2CC2)C1CNC(=O)C=CC1CC1 68295,Cc1noc(C)c1C(C)C(=O)NCCN(C(C)C)Cc1ccc(C(F)(F)F)nc1 68296,C12(COC)CCC(C(=O)N(C)CCNC(C3(C#N)CCCO3)=O)(CC1)CO2 68297,CN1CC(C)(C(N2CC=CC(NC(=O)CN3CCC(O)CC3)C2)=O)CC1=O 68298,C1(NC(C2C(NC(C3CCCN3CC(F)F)=O)C2)=O)CCCCCCC1O 68299,c1(CCNC(CC(C)CC2CCC2)=O)ccccc1[N+](=O)[O-] 68300,C1(N(N2CCC(C(F)F)CC2)C)COC2(CNC2)C1 68301,C12(NC(c3cc(Cl)c[nH]3)=O)CC3CCC(C1C2)N3C(c1c[nH]c2cnccc12)=O 68302,N1(C(C2CC=C(C)CC2)=O)CCC(C)(C(=O)Nc2ncc(C)c(Cl)n2)CC1 68303,CN1CCCC1(C)C(=O)NCC1CCN1C(=O)Cn1[nH]cnc1=N 68304,C(N=c1[nH]cnc(Cl)c1CO)C1CCC(NC(c2ccc(C(=O)NC)nc2)=O)C1 68305,n1(CC(=O)N(CC(CC)NC(=O)C(C)n2cccc2)C)nc(C)cc1C 68306,N1(C(CCCC#C)=O)CCCC2C(NC(c3cc(O)cc(C#N)c3)=O)C(C)(C)C12 68307,C=CCCC(=O)N(CCCCCNC(=O)C(C1CCCC1)OC)C 68308,c1(CNC(CNC(C2C(C)C2)=O)=O)ncc(C(=O)NCCCS(N)(=O)=O)cn1 68309,c1(C(N(CCC)CCNC(C2(CCC)CCC2)=O)=O)cc(Cl)cc(Cl)n1 68310,c1(CC(=O)NC2CN(C(c3c(OC)nsc3)=O)C3C2C3)cc2ccccc2o1 68311,c1(C(=O)NC2COCCN(C(C3CC(C(C)C)C3)=O)C2)cn2ccccc2n1 68312,N1(C(C2ON=C(C)C2)=O)CC2C(c3cn(CCc4ccccn4)nn3)C2C1 68313,C(=O)(C(C(C)(C)C)NC(=O)CC1CCCC(=O)C1)NCCCc1c(C)n[nH]c1C 68314,c1(C(N2CC(O)CC(NC(C3SCCS3)=O)C2)=O)cnn2c(Cl)cccc12 68315,C(=O)(C#CC1CCCC1)NC1(CC2CC2)CN(C(c2cnn(CC)c2Br)=O)C1 68316,CCC(C)C(CC(=O)N(CC(F)F)CC)NC(C1CCC2(CCC2)C1)=O 68317,c1(C(N(C)CC2CN(C(C3C(C(=O)OC)CCC3)=O)C2)=O)c(C)cccc1O 68318,C1(C(N(CC(=O)NCC2(F)CC2)C)=O)CCCN1C1CC1 68319,C(C(=O)NCCC1CC1)(C1=Cc2cc(Br)ccc2OC1)N(C(C=C)C1CC1)C 68320,Cc1c(C)n(C)c2ccc(C(=O)NCC3CN(C(=O)C(C)(F)F)CCC3C)cc12 68321,C1(OC)CC(CNC(=O)C(C)(C)n2cnnn2)N(C(=O)CC2CS(=O)(=O)C2)C1 68322,N1(C(CCOCC)=O)C2CCCC1CN(C(=O)C(c1ccccc1)=O)C2 68323,Cc1cncc(C(=O)NC2CC(C)N(C(=O)COCCC(C)C)C2)c1 68324,C(=O)(CCC(CC)NC(c1c[nH]c(C)cc1=O)=O)NC(CSC)C 68325,C1(NC(=O)NCC=CCC)CC(=O)N(CC(C)C)CC1 68326,C1(NC(Cn2nc(C)c(Cl)c2)=O)CN(C(C2(C)CC(C#N)C2)=O)CC1(C)C 68327,CCC(C(=O)NCC(C)(C)NC(C1CC1c1cncn1C)=O)SC 68328,C1(C(=O)OCC)CCCN1N(C)C(=O)C1C(c2ccccc2)C1(C)C 68329,Cc1ccc(F)cc1C(=O)C(=O)NCC1(F)CC(NC(c2cnc(C)n2C)=O)C1 68330,c1(C(N2C(CN(C(COC(CC)C)=O)C)CCCC2)=O)ccnc2ncsc12 68331,C(=O)(CN=c1cc[nH]cc1)N(C(C(=O)NCC(CC#C)(C)CO)C1CC1)C 68332,C1(N(C(CCC=C)=O)C)CCC2N(C(=O)C(CC)=CC)CC12 68333,C(=O)(CCCCCOC)NC1CCN(C(CNS(CCCC)(=O)=O)=O)C1C(C)C 68334,C#CC1CN(C(=O)Cn2cccc2C(=O)O)CCN1C(=O)CCc1ccoc1 68335,C1(NC(c2c(C(C)C)noc2)=O)CN(C(C2COC(=O)N2C)=O)CC1O 68336,CC(C)(C)CCCCCC(=O)N1CCn2ncc(CNC34CCN(CC3)C4)c2C1 68337,N1(C(c2cccc(C)c2F)=O)CCC2(CCCN2c2nc3ccc(F)cc3o2)C1 68338,C(=O)(CS(=O)(=O)CCC)N1CCCC(c2cn(C(C3CC4(CCC4)C3)CC)nn2)C1 68339,C1(O)(CN(C(Cc2ccc(C)nc2)=O)C)CCN(C(=O)C(C)(C)CC#N)CC1 68340,N1(C(c2cc(Cl)c(Br)c(Cl)c2)=O)CCC2C(CCN2C(=O)CC2CCOCC2)C1 68341,C1(C(=O)NC2C3CN(C(CC(CC)CC)=O)C2CC3)CCc2nnnn2CC1 68342,Cc1nn(CC(=O)N(C)CC2CCCCN2C(=O)C(O)C2CCC2)c(=O)o1 68343,n1(CC)nnc(-c2nc(CC(C)CC)nn2-c2ccc(OCC(C)C)cc2)c1C 68344,C=CCC(C)C(=O)NCC1CC(COC)CN1C(c1cnn(C(C)(C)C)c1C)=O 68345,c1(C(N(C)CC2(NC(C(F)=CCC)=O)CC2)=O)cn2c(n1)CCC2 68346,C1(C(N(CC(CSC)C)C)=O)C2CC1N(C(=O)COC(C)=O)C2 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68365,N1(C(C=CCC)=O)CCCC(O)(CCNC(=O)CNC(c2cccc(Cl)c2)=O)C1 68366,c1(N(C)C)ncc2c(n1)CN(c1cc(NC(=O)NCCCl)ncn1)C2 68367,c1(C(N(CCCNC(C2=C(C)CCC2)=O)C)=O)cc(C)cc(Cl)c1N 68368,C1(C(C)C)CC(NC(C2CC(C)(O)C2)=O)CO1 68369,Cc1cccnc1CCC(=O)NC(CN(C(=O)C=CC(C)C)C)(CO)CO 68370,c1(-c2c(OC)ccc(-c3nccn3CC(O)CO)c2)cc2cccc(OC)c2o1 68371,C(CC(C(=O)N1CC(C(=O)NCC2(F)CCCCC2)(SC)C1)OC)OC 68372,c1(SC)ccccc1CC(=O)NCCC1(O)CN(C(c2cccc(NC)n2)=O)C1 68373,N1(C(Cc2c(N(C)C)nccc2)=O)CCN(C(=O)C=CCF)CC1C1CCC1 68374,C(CCCCCCC(=O)NCCOCCNC(C1CC2CCC1O2)=O)SC 68375,C1(C(c2cccc(Cl)c2)CC)CC2(CN(C(=O)CN3CCCC3)C1)OCCO2 68376,C1(NC(C(C)n2cncn2)=O)C=CCC(C(=O)N(C)Cc2cncs2)C1 68377,Cc1ccc2cc(CN3CCC(NCC4CCC(C(F)(F)F)C4)C3)n(C)c2c1 68378,n1(CC(=O)NCC(C)(C(C)C)NC(C(c2cccnc2)SC)=O)nc(C)c(C)c1C 68379,C1(CC)CN(C(=O)C(c2c(C)n[nH]c2C)C)CC1NC(=O)COCCCF 68380,N1(C(c2c(C)ocn2)=O)CC2(CCOCC2C(=O)Nc2cc(CO)ccc2F)C1 68381,c1(OCC)ccc(C(=O)NC(C)C(C)NC(=O)C2=C(C)CCC2)cc1OC 68382,c1(CC(=O)NC2CC(CNC(Cc3c(C)ncs3)=O)C2)sc(O)nc1O 68383,N1(C(CC(C=C)C)=O)CCCC(C)(C)C1CNC(c1c(C)cc(Cl)cc1N)=O 68384,c1(-c2cn(C)nc2)ccc(NC(=O)CC(c2ccccn2)NC(C)(C)C)cc1 68385,CC(CC(C)(F)F)C(=O)NC(c1cn(CCN2CCNC2=O)nn1)(C)C 68386,Cc1cnncc1C(=O)NC(CC1CC1)CC(=O)N1CCN(C2CC2)CC1 68387,C1(C(N(C2CCN(C(=O)Cc3sccc3C)C2)CC)=O)Cc2nccnc2C1 68388,c1(C(=O)Nc2cc(CCC)cc(C)c2)cc(Cl)c(OC)nc1C 68389,c1(C(C(=O)NCC(CCOC)NC(c2sccc2C)=O)(F)F)ccc(C)cc1 68390,N1(C(C2=C(C)OCCC2)=O)CCOC2(C1)CN(C(=O)CC13COC(CF)(C1)C3)C2 68391,c1(NC(=O)NC(C)CCC2CCCCC2)ncc(Br)cc1Cl 68392,c1(OC)cc(OC)c(F)c(C(=O)NC2CC(C)CN(C(C3CCCS3)=O)C2)c1 68393,c1(C(=O)NC2C(CNC(=O)C=Cc3cccs3)COC2)cnnc(C2CC2)c1 68394,Cc1nc2ncnn2cc1C(=O)NC1CCCCC1NC(=O)Cc1cccnc1 68395,C1(C(=O)NCC2N(C(CC(CC(=O)OC)C)=O)CCC2)CCn2c(cnc2C)C1 68396,c1(C(c2n(CC)nnn2)NCc2cc(F)cc(Br)c2)ccc(S(N)(=O)=O)cc1Cl 68397,C1(CC)(NC(=O)C(C)C(C)(F)F)CCN(C(=O)C(C)Cc2ccncc2)CC1 68398,C1(CNC(CC2C(C)CCO2)=O)CN(C(c2ccc3c(n2)NCC3)=O)CCN1C 68399,C1(CC)CN(C(c2ccccc2Br)C(=O)Nc2cccc(OC)c2)CCO1 68400,C(C(O)C(=O)NC1(C)CC(NC(c2cc(C3CCC3)[nH]n2)=O)C1)=CCCC 68401,c1(OCC)cncc(C(=O)NC2CC(CO)N(C(=O)Cc3cc(Cl)cs3)C2)c1 68402,CC1CCc2[nH]c(C(N3CCOC(CN(C)C(c4ccnnc4)=O)C3)=O)cc2C1 68403,c1(C(=O)NC2C(C(N(CCCC(O)CO)C)=O)COCC2)ccc([N+](=O)[O-])[nH]1 68404,c1(C(=O)NCCC(C)N(C(C(CC)OC)=O)C)ccn(C)c(=O)c1 68405,CC(C)C(CC(=O)NCC1CC2CCC1CC2)NC(C1CC2(CCO1)CC2)=O 68406,c1(C(N2CC(C)(CNC(CCCCOCC)=O)OCC2)=O)c(F)ccc(C)c1Cl 68407,C1(C(C)C)CN(C(c2cc(-c3cccnc3)no2)=O)CCN1C(=O)CC(F)F 68408,C(=O)(C1CCCc2nncn21)Nc1nnc(CC2(NC(C3CCCCC3)=O)CCC2)s1 68409,C(=O)(C(CN(C)C)CC)NCCCN(CCCNC(C(C)OCC)=O)C 68410,c1(N(CC(C)C)C)ccc(C(=O)NCCC(C)(C)CNC(=O)C(C)(C)O)cc1 68411,C(CC(C)CC)(C(=O)NCCC(=O)NCC)NC(CCCC)=O 68412,c1(N2CCCC(CCNC(COC(CC)(C)C)=O)C2)nc(CO)nc2[nH]ccc12 68413,N1(C(C2(CNC(c3c(C)scn3)=O)CC3(CC3)C2)=O)CC2CC(C)C2C1 68414,C(=O)(CCCC(=O)NC)c1ccc(OC)cc1.C1(CNC=O)COCCN1C 68415,c1(OC)ccccc1C1(C(=O)NC2CC2NC(c2nocc2C)=O)CCC1 68416,C(C1=NOC2CCCC12)NC(=O)NCC(C1CCCOC1)OCC 68417,C1(N(C)S(N)(=O)=O)(CC(N)=O)CCN(C(=O)NC(C2CC23CC(F)(F)C3)=O)CC1 68418,C(C(C)(C)C(=O)OC)(c1n(CCC)nnn1)NCC1(c2ccccc2)CC1 68419,c1(C(N2CCC(C)(CC(=O)NC(C(F)(F)F)C3CC3)C2)=O)cc2ncccc2[nH]1 68420,C1(NC(C(C)(C)NC(=O)OC)=O)C2CCC(C2)C1C(=O)NCc1cncnc1 68421,c1(C(=O)NC2CC(CCNC(C3(Cl)C(C)(C)C3)=O)C2)cc2cn[nH]c2cn1 68422,c1(C(=O)NC2C=CC(CNC(c3c(C)cns3)=O)C2)cc(C(F)F)ncn1 68423,c1(CNC(C23N(C(c4oc(CC)c(C)c4)=O)CCC2C3)=O)ccc(C)nc1O.C1CC1 68424,C1(C)(NC(C(C2CCCCC2)NC(c2c(C)snc2)=O)=O)CCC2(CC1)CC2 68425,C1(C(=O)NC2CCC(NC(CCC)=O)C2)COCCN1C1CCCC1 68426,C1(CN(C(=O)C2=CCSC2)C)CN(C(=O)C(C)(C)C2CCC2)CC12CC2 68427,C=C1CC2CC1CN2C(=O)C(C1(O)CN(C(=O)C(F)F)C1)F 68428,c1(C2C(C(=O)NCC(CNC(c3cccc(N)c3)=O)OC)C2)cccc(F)c1 68429,C(CC(=O)N1CCCC1)NC(COCC(=O)NC)=O.C1C(=O)N1 68430,C(CC)(C(=O)N1CC(CC(C)NC(=O)CC2CC(Cl)(Cl)C2)C1)=CC 68431,N1(C(c2cc3sccc3s2)=O)CC2(CCN(C3CCc4c(F)cccc43)C2)C1 68432,c1(C(=O)NCC(CC)NC(C2CCCCC2C(N)=O)=O)ccnc(OC)n1 68433,N1(C(c2cc(CC)ncc2)=O)CCN(C(C23CC(C(C)(C)C)(C2)C3)=O)CC1CC 68434,N(C1CCc2c1ccc(Br)c2F)C(N(c1ccc(F)cc1F)C(CC)C)=O 68435,N1(C(C2(CC)CCCO2)=O)CC(CNC(c2cc(C)ncn2)=O)C(O)C1 68436,Cc1nc2n(c1C(N1CCC(Oc3cccc(C(=O)O)c3)CC1)=O)CC(C)CC2 68437,c1(C(=O)NC2CCCN(C(CCCCCSC)=O)C2)cccc2c1NCC2 68438,CC(C)C(C)C(=O)N1CCOC(CNC(=O)Cc2cncnc2O)C1 68439,N1(C(C2C(Cl)(C(=O)OC)C2)=O)CC2CCC(CNC(C3CC(C(C)C)C3)=O)(C2)C1 68440,C(=O)(C(CC(F)F)N1CCCC1Cc1ccc(F)cc1F)NCCOC 68441,C1(NC(c2ccc(-c3ccccc3)s2)=O)CCCN(C(c2ccncc2)=O)C1 68442,C1(C(=O)NC2CC(C)CN(C(=O)CCC=CBr)C2)COc2ccccc2C1 68443,N1(C(C(CC2CCOCC2)NC(c2cnsc2)=O)=O)CC2COCC2C1 68444,N#CC1(C(=O)NC2CN(C(=O)CCCc3ccncc3)C2)CC2CC2C1 68445,C(CCCCC(=O)NC(CO)C(=O)N1CC(C(=O)NC)C1)OCC 68446,C#CC1(C(=O)N(CC(C)COC)C)CN(C(=O)C(=C2CCCCC2)F)C1 68447,C1(F)(CNC(COC(C)C)=O)CCN(C(C2CCC2F)=O)CC1 68448,N1(C(NN(C(C(C)NC2CC2)=O)C)=O)C(=O)Cc2ccccc2C1=O 68449,N1(C2C(COC(c3scc(CNC(C)=O)c3)=O)CCC2)CCN(C)CC1 68450,C1(CNC(=O)NC(C)C2CC2)CCCC(C(F)(F)F)C1 68451,c1(N(C2CNC2)C(c2cc(F)c(C)c(Br)c2)=O)ncc2c(n1)NC(=O)C2 68452,c1(C(N2C(NC(C(C)OCCOCC)=O)C=CC2)=O)cccc2c1CC(C)(C)C2 68453,Cc1ccc(Cl)c(OC(C)C(=O)NC2CN(C(=O)C3=NOC(C)C3)C2)c1 68454,C1(c2cn(C)nc2)CN(C(C2CC23CCCCC3)=O)CCN1C(=O)CCC(F)(F)F 68455,C1(C(=O)NCC2(C)CCCN2C(c2ccncn2)=O)Cc2ccccc2S1(=O)=O 68456,N1(C(=O)NC2CCN(c3ccc(F)cc3F)C2)CC2CCCCCC2C1 68457,C1(NC(c2sc(F)cc2Cl)=O)CCCC12CN(C(C1CCCC1)=O)C2 68458,C(=O)(CC(C(=O)N1CC(N(C(=O)C=Cc2ccsc2)C)C1)NC(C)=O)OC 68459,c1(SC2CCCCC2)cncc(C(=O)N(C2CC2c2ccccc2C)CCC)c1 68460,Cc1cc2[nH]c(C(N3CC4=C(C3)CN(C(C3(C)CCCCN3C)=O)C4)=O)cc2o1 68461,c1(C(=O)NCC(C)NC(=O)CC2COC(=O)N2)ncc(Cl)nc1Cl 68462,Cc1cccc2c1CC(C(N)=O)N(C(=O)NCC1CCS(=O)(=O)C1)C2 68463,CCCC(O)CN=c1[nH]c2cc(C)c(S(=O)(=O)NC(CSC)CC)cc2s1 68464,C(=O)(C1=NNC(=O)CC1)NC(C)CC1CN(C(=O)CCc2ncnn2C)C1 68465,C=CCC(CNC(=O)CNC(c1ccco1)=O)NC(=O)COC.C(C(F)F)OC 68466,N1(C(CC(C)F)=O)CCCCC(CN=[N+]=[N-])C1.C1(C2CC2)(C(=O)N)CC(=O)C1 68467,N1(C(c2ccc(OC)nc2Cl)=O)C2CCC1C(F)C(NC(C1OCC1(C)C)=O)C2 68468,c1(C(=O)NC23CCC(CN(C(c4ccnnc4)=O)C2)C3)cnc(O)c2cncn12 68469,Cc1csc(=NCC(=O)N(C2CN(C(C3CS(=O)(=O)C3)=O)C2)C)[nH]1 68470,N1(C(=O)Cn2ccc(C3CC3)n2)CCN(C(C2CC3(CCC3)CO2)=O)C(CO)C1 68471,N1(C(C2C(O)CCN(C(CN(C(C)C)C)=O)C2)=O)CCC2COCC2C1 68472,c1(N(C)CC2(OC)CCOC2)[nH]c(=NC(C)c2cnn(C)c2)nc2sccc12 68473,Cc1cc(C(=O)NCCC2CC(NC(C3(C)CSC3)=O)C2)c(Cl)cc1F 68474,C1(NC(=O)NC)CCC12CCCO2.c1(CNC(=O)OC(C)(C)C)c[nH]nc1CO 68475,c1(N2C(C)(C)C(NC(=O)Cn3cncn3)CC2)cc(C#N)ccc1[N+](=O)[O-] 68476,N1(C(c2ccn(COC)n2)=O)CCN(C(c2cc(COC)on2)=O)CC1CF 68477,C(C)(CC(C)NC(c1ccnn1C1CC1(F)F)=O)NC(COCCOCC)=O 68478,c1(C(=O)NC2(CNC(C3CCC(CC)C3)=O)CCCC2)cc(C)nc(O)c1 68479,N1(C(C2C(CCOC)C2)=O)CCN(C)C(C(=O)NCC2(CO)CC3CC3C2)C1 68480,CCCC(C(=O)N1CC(NC(c2ccc(S(=O)(=O)NC)o2)=O)C(O)C1)C(C)C 68481,Cc1[nH]c(C#N)cc1C(=O)NC(c1nocc1C(=O)NCCOCC(F)F)C 68482,C1(C(N2C(C(C)NC(Cn3c(C)c(Cl)cn3)=O)CCC2)=O)CCn2cnnc2C1 68483,N1(C(c2scc(C)c2C)=O)C2CCCC1CC(NC(C1C=CCCC1)=O)C2 68484,N1(C(C(CC)O)=O)CC2(CCC2)CC1CNC(c1ccnc(-c2ncc[nH]2)c1)=O 68485,Cc1cc(C)n(CC(=O)NCC2(O)CCN(C(c3[nH]c(O)nc3C)=O)C2)n1 68486,C1(NC(C2(COC)CC2)=O)C=CCN(C(=O)C(C23CCC(CC2)C3)C)C1 68487,N1(C(Cc2c(OC)cccc2)=O)CCCC(C)(NC(=O)CC2CCSC2)C1 68488,C(CC)(CCCC(=O)N1CC2COCC2(C(N)=O)C1)NC(C(CC)O)=O 68489,C1(C(=O)NC(C(=O)OCC)C)CN(C(c2ccc(N3CCNCC3)cc2)=O)CC1F 68490,Cc1cccc2c(=O)n(CC(=O)NCC(C)NC(=O)CSC3CC3)cnc12 68491,CCC(F)(C(=O)OC)C(=O)NC12CCC(CC1)N(C(=O)COc1cn[nH]c1)C2 68492,Cc1cncc(C(N2CCC(C(F)F)(CNC(C3CC(F)C3)=O)C2)=O)c1 68493,C1(N(C(c2c(CC)[nH]cc2)=O)C)CCN(C(=O)C=Cc2cncc(O)c2)CC1C 68494,c1(CC)cc(N)ccc1C(N1CCN(Cc2ccco2)CC1CC(F)F)=O 68495,CCCCC(O)CC(=O)N1CC2C(CNC(=O)C=C(Cl)Cl)C2C1 68496,Cc1ccc(F)c(CNC(C2(CNC(C3CCS(=O)CC3)=O)CCOCC2)=O)c1 68497,C1(NC(CN(C)CCO)=O)CCN(C(=O)Cc2cnn(C(F)F)c2)CCC1CO 68498,c1(C(=O)NC2(C(=O)OC)CCC2)ccc(NC(C2(CCCF)CC2)=O)cc1F 68499,N1(C(C(C(C)C)C(C)C)=O)CCCC2(NC(c3nccnc3C)=O)CCCC12 68500,C1(NC(COCc2c(C)ncs2)=O)CCCN(C(c2cccc(F)c2F)=O)C1C 68501,C1(NCC2(F)CCC(C(=O)O)CC2)CCSC2(CCC2)C1 68502,C(CCCCNC(=O)C(C)c1cncs1)NC(C(c1ccccc1)NC(C)=O)=O 68503,Cn1cc(C(=O)NCC2(NC(=O)CC3=CCOCC3)CC2)c2ccccc12 68504,CC(c1ccccc1F)=CC(N1CC(N(C)C(C2COCCN2C)=O)C1)=O 68505,C1(CNC(C2(C(C)C)CCOCC2)=O)CNCC(C)(C)C1 68506,N1(C(CCCNC(N)=O)=O)CC2CCC1CC2NC(=O)CC1CCCSC1 68507,C1(C(CO)NC(C2(NC(=O)COCC3CCC3)CC2)=O)CCCCC1 68508,c1(C(N(C)C)=O)ccc(CNC2(c3ccncc3)CNC2)cc1[N+](=O)[O-] 68509,C1(CNc2cc(N3CC(CCC)OCC3)ncn2)CC2CCC(C1)S2 68510,c1(CCC(N2CC(C(C)NC(=O)C(CC)N3CCCC3=O)C2)=O)c(C)noc1C 68511,C1(NC(=O)CC2(O)CCC2)CC2CCC1CN2C(C1CNC(=O)N1)=O 68512,C#CCCC(C(=O)Nc1cccc(C#N)c1)NC(c1[nH]nnc1C)=O 68513,C(=O)(CC(C)CC(C)(C)C)NCCC(=O)NCc1ncc(C)cn1 68514,Cc1ccc(CNC2CCCCC2C(=O)NCC2CCCOC2(C)C)c(F)c1 68515,N1(C(C(C(C)NC(=O)C(N2CCNC2=O)C)(C)C)=O)CCC2CCCC2CC1 68516,C1(C(=O)NCC23C(CN(C(CNC(=O)OC)=O)C2)C3)CCc2nc(C)[nH]c2C1 68517,Cc1nc(CNC(=O)CC2C3CN(C(=O)CCc4cccnc4F)CC23)oc1C 68518,c1(C(N(C(C(=O)NC(CCC)c2nn[nH]n2)C)C2CC2)=O)snc(C)c1N 68519,CN1CCC(NC(=O)C(C2CC2)N(C)C(c2cc3occc3[nH]2)=O)C(C#N)C1 68520,C(=O)(C(C(C)O)NC(C)=O)NCCN(C(c1cc(CC2CC2)ns1)=O)CC 68521,c1(COC(c2c(OC)c(Cl)ccc2)=O)c(F)cc([N+](=O)[O-])cc1F 68522,c1(C(N2CCCC(CCNC(C(C)=CC)=O)C2)=O)cccc2c1OC(C)C2 68523,CCC(C)(C(=O)N1CC(CO)(NC(c2ocnc2C)=O)C1)OC 68524,N1(C(C=CCC)=O)CC(NC(=O)CCC=Cc2cccc(F)c2)CC1(C)COC 68525,CC(=NO)C1CC(C(N2CCC(C(C)Nc3cc(Cl)nc(C)n3)CC2)=O)C1(C)C 68526,c1(C(=O)NC(CC2CN(C(c3cc(C)[nH]n3)=O)C2)C)cc2sccc2s1 68527,O=C(C#CC1CCOC1)N1CCCOC(CN=c2cc[nH]c(-c3nccs3)n2)C1 68528,N1(C(C(CC)N(C)C(c2ncnc(C)c2C)=O)=O)CCCC(C)(C)C1C 68529,N1(CC2CC(CC)OCC2)CC2CCC1CN2C(=O)COCCCC(C)C 68530,N1(C(C(C(C)OC)NC(=O)Cc2ccco2)=O)CCC(O)CC(C)C1 68531,N1(CC)CCN(C(C2(CF)CCN(C(=O)CSC(F)F)C2)=O)C(C)C1 68532,c1(CC(=O)NC(CCCCC)C)ccc(C#N)nc1 68533,N1(C(c2c(C)nc(O)[nH]2)=O)CC(CNC(=O)C2=NOC(C)C2)CC1(C)C 68534,CCCC#CC(C)(C)NC(=O)C(CN(C)C)NC(=O)C(C)(C)COCC 68535,CN1CCC(C(N2CCC(N3CC=CC3)C2)C(=O)NCc2ccco2)CC1 68536,c1(OCC)cc(CNC2CC(NC(c3cc(Cl)ccc3Br)=O)C2)cc(F)c1 68537,C1(NC(c2cncc(F)c2)=O)CN(C(=O)C#CC2CCCO2)C2(CCC2)C1 68538,C1(CN(C(=O)C(C)N2CCCC2)CC)CCCN1C(=O)C(C1CC1)SC 68539,C1(C2CC2)(CNC(CN(C2CC2)CC)=O)CCN(c2nc3ccccc3o2)C1 68540,c1(C(=O)NC2C(CNC(COCC(=O)NC)=O)C2)cc2ccc(Cl)c(F)c2[nH]1 68541,N1(C(CC(=C)C)=O)CCCC2CN(C(C3CCc4c(nnn4CC)C3)=O)CCC12 68542,C1(C#CC(=O)NC2CC(CC(N3CCC(CN4CCCC4)C3)=O)C2)(C(C)=O)COC1 68543,N1(C(c2nn(C(CC)C)c(C)c2)=O)CC(NC(=O)C=CS(C)(=O)=O)CC2(CC2)C1 68544,C1(CC=C)(C(=O)NC(CCCOC(F)(F)F)=O)CN(C(=O)CC(C)C2CC2)C1.NC 68545,c1(CC(N2CCC(C(C(C)C)NC(=O)CC(F)F)CC2)=O)c[nH]c2ncccc12 68546,Cn1c(O)nc2cc(C(=O)NC3CN(c4cnc(C#N)cn4)CC3(C)C)ccc12 68547,Cc1noc2ncc(C(=O)NC3CC4CC3N(C(c3ncccn3)=O)C4)cc12 68548,CC1(C)CC(O)(CC(N2CC(CCCCNC(c3nn[nH]c3Cl)=O)C2)=O)CO1 68549,c1(Nc2n(CCOC)ncc2)cc(Br)ccc1S(=O)(=O)N1CCOC(OC)C1 68550,Cc1cc(Cl)c(C(N2CC(CCNC(=O)CN3CC(C)C3)C2)=O)cc1F 68551,C(=O)(CC(C)CC(C)(C)C)N(C1CCN(C)CC1)C(C1ON=C(C(C)C)C1)=O.N 68552,Cc1cc(C(=O)NC2CN(C(C3CCOC(=O)N3)=O)CC2F)oc1C 68553,C(=O)(C1=CC2C=CC1C2)N1C(C)(COC)CC(NC(=O)C#CC(C)C)C1 68554,C1(NC(CN(C(C)=O)C)=O)CCC(C)(CNC(=O)Cc2csnc2C)C1 68555,C1(=CC(=O)NC(CCC)CCCNC(=O)C(C)CF)CC2CCC(C1)N2C 68556,C#CCCCCCCC(=O)NC1CC(NC(c2ocnc2CC)=O)CC1O 68557,N1(C(CC(=O)Nc2nccs2)=O)CCN(C(c2cnsn2)=O)C2CCCC12 68558,C(=O)(C1=CS(=O)CCC1)NC(c1cn(CCC=C)nn1)=O.C123CCC(CO1)(C2)C3 68559,c1(C(N2C(CCNC(CC3ON=C(C)C3)=O)COCC2)=O)ccc(Cl)cc1O 68560,c1(C(N(C)CC2(NC(=O)CCc3cn[nH]c3)CC2)=O)ccnc(Cl)c1Cl 68561,c1(C2(OC)COC2)cccc(C(c2cccc(Cl)c2)c2nn[nH]n2)c1.C1(=O)CN1 68562,N1(C(C(C(C)C)n2ccc(C)c2)=O)CC(O)C(O)C(O)C1COC 68563,C1(C(N2CCC(O)(CC=C)C2)=O)COCCN(C(C2(C(=O)OC)CC2)=O)C1 68564,c1(N(C)C)ccc(F)c(C(N2CCC(C)(NC(C3CN(S(N)(=O)=O)C3)=O)C2)=O)c1 68565,c1(C2CC(CNC(C(c3cccc(F)c3)N)=O)C2)ccc(F)c(F)c1 68566,c1(CC(N2CC(F)(CNC(CC3(COC)CCCC3)=O)C2)=O)cc(F)ccc1C 68567,C1(NC(C=C(C)CNC(=O)CN2CCSCC2)=O)C(=O)NCCC1C 68568,C1(C2CC2)(C(N2C(C)CC2(C)C)=O)CN(C(=O)CC2CC3C=CC2C3)C1 68569,c1(CC(=O)NC2CN(Cc3n(C)nnc3)CC2O)ccc2c(c1)OCO2 68570,CC(C)(C)CC(O)CC(=O)NC1CCCCC1NC(c1cc2cccnn2c1)=O 68571,C(C)(N=c1ccnc(NCc2ncc(Cl)n2C)[nH]1)n1cccc(CC)c1=O 68572,CCC(C)CCC(=O)NCC=CCNC(=O)C(c1ccc(F)cn1)(F)F 68573,CCC(CC(=O)NCCOCCOC(C)(C)CNCC1COC(C)(C)C1)C(F)F 68574,C(=O)(C#CC(C)(C)CNC(=O)C(C)CC)NC(CCC)CC 68575,C(=O)(C1=C(Cl)CCC1)N1C(C(C)NC(=O)CCOCC(F)F)CCC1 68576,C1(CCC(=O)N(C2CC(=O)NC2=O)C)CCN(C(c2cn(C(C)C)cn2)=O)CC1 68577,CCCCC(C(=O)NCC1(CC(C)C)CCC1)NC(c1cn(C)nn1)=O 68578,CC(C)CCCC(C)C(=O)NCCC1(CNC(c2cc(F)c(F)c(F)c2)=O)CC1 68579,N1(C(CCSCCCC)=O)CCN(C(C2CC23CCOC3)=O)CC(O)C1 68580,Cc1c(C(=O)NCC2C3CCC(C3)N2C(c2csc(C(C)C)n2)=O)cncc1N 68581,C=CCCCCCC(=O)NC1(C2CN(C(=O)C(C)C(C)(C)C)C2)CC1 68582,N1(C(c2c(C)ccc(=N)[nH]2)=O)CC2CCCC2(NC(=O)CCC2CCOC2)C1 68583,C1(CC(=O)N(C2CCN(C(=O)CCC(C)SC)C2)CC)C(C)(C)C1(C)C 68584,N1(CC(=O)NC2CCC(C)(NC(=O)C=CC3CCCC3)C2)CCS(=O)(=O)CC1 68585,C1(CCC)COCCN1C(C1CCCCC1NC(c1ccncc1OC)=O)=O 68586,Cc1cc(=N)[nH]cc1C(=O)NCC1CC1NC(=O)C(C)(C)C(C)C 68587,c1(CC)nc(C(=O)NCCC2CCN(C(C3(CC)COC3)=O)C2)c(C)o1 68588,N1(C(c2c(OC)nn(C)c2)=O)CCC(NC(c2cc(F)ccc2OC)=O)C(C)C1 68589,C(C1NC(=O)c2ccccc21)[NH+].C(N=c1ccnc(NCC)[nH]1)c1cccc(C)c1Br 68590,N1(C(CC=CCC)=O)CC(O)(C2CCN(C(c3cc(C)c(C)cc3Cl)=O)CC2)C1 68591,N1(C(CC2CN(C(c3c(C)ncs3)=O)C(C)(C)C2)=O)C2CCC1CC(=O)NC2 68592,c1(C(N2CC(CC=C)(NC(=O)CC3CSCCS3)C2)=O)c(C)oc(C)c1C 68593,N1(C(c2c(OC)nsc2)=O)CC2=C(C1)CN(C(=O)CC1C=NN(C)C1=O)C2 68594,c1(NC(C(C)Sc2scc(C)n2)=O)cccc(NC(C2(F)CCCC2)=O)c1 68595,C1(NC(C(C)(C)NC(C=COC)=O)=O)CN(C(c2cnc(SC)s2)=O)CC1F 68596,C1(C)(CC)CCC(C(=O)N(C)CC2CC(CN=[N+]=[N-])C2)O1.C12(CC1)C(=O)N2 68597,c1(OC)cc(NC(C2(F)CCN(C(c3c(Cl)ccnc3Br)=O)C2)=O)nc(Br)c1 68598,c1(CN2CCC(NC(c3ccncc3F)=O)CC2)c(F)cc(I)cc1F 68599,c1(C(N2CC(CNC(COC(C)(C)C)=O)OCC2)=O)ccnc2[nH]ncc12 68600,C(=O)(C#CC1CCCC1)N(CCOCCNC(C(CCC)(F)F)=O)C 68601,C(C(C)(C)CC(=O)NCCOc1ccccc1)NC(C(C1CC1)OC)=O 68602,C#CC(C)(C)C(=O)N1CCC(C(CO)NC(C2CCCO2)=O)CC1 68603,C1(NC(c2ccc(CC)cc2)=O)CN(C(=O)CNS(=O)(=O)CC)C2CCCCC12 68604,N1(C(c2cnc(CC)s2)=O)CC2CC(NC(=O)CNS(=O)(=O)NC)C2C1 68605,c1(C(=O)NCC(CC(F)(F)F)NC(C(C)C2CCC2)=O)ccc(P(C)(C)=O)cn1 68606,Cc1nn(C)c(C)c1NC(C1CCN(C(c2ccc(C(F)(F)F)cc2I)=O)C1)=O 68607,C1(NC(C(C2CC2)NC(CCOC(C)=O)=O)=O)CN2CCC1(C)CC2 68608,N1(C(C(c2ccc(OC(F)(F)F)cc2)SC)=O)CCc2cc([N+](=O)[O-])cc(Br)c21 68609,CC1CN(C(=O)C#CC(C)(C)C)CCC1NC(c1cccc(NS(N)(=O)=O)n1)=O 68610,c1(C(=O)NCc2c(CN(C(C(C)C)=O)C3CC3)cccc2)cc2n(n1)CCCC2 68611,N1(C(CCC2(NC(CSCCC(C)C)=O)CCC2)=O)CCOC(C(C)C)CC1 68612,c1(C(=O)NC2C(OC)CN(C(c3cnc(Cl)s3)=O)C2)cc(C)n(CC2CC2)c1C 68613,C(=O)(C1=NOC(C(C)(C)C)C1)N(C)CCNC(=O)CC(C)(C)c1ccc(F)cc1 68614,C1(CNc2ccc(N3C(=O)OCC3)cc2)CC2OC1C1CC21 68615,Cc1cccc(C(N2CCN(Cc3ccc(F)c(F)c3)C(C)C2)=O)c1C 68616,c1(OC)cc(C(N2CCC2CNC(C2CC(C)(C)C2)=O)=O)cc(OC)c1C 68617,C(C(C(=O)NC1CCC1C)C(C)C)NC(CCC(=O)NCCC)=O 68618,C1(NC(c2cccc(C3CC3)c2)=O)CC1C1CCCN(C(c2cccnn2)=O)C1 68619,c1(OC(C(=O)N(CCN(C(c2cc(CCC)on2)=O)C)C)C)ccc(Cl)cc1C 68620,C1(OC)CC(CNC(=O)CN2CCCOC2=O)N(C(=O)CN2CCCC2(C)C)C1 68621,N1(C(C=CCOC)=O)CC2CCCC2(CNC(=O)CCCCCN(C)C)C1 68622,c1(C(N(C2CCCN(C(C3CCCC4CC34)=O)CC2)C)=O)nc2ncccn2n1 68623,N1(C(CC(=C)C)=O)CCC(CCNC(c2cncc(NS(C)(=O)=O)c2)=O)CC1C 68624,c1(OC)ccc2oc(C(N3CC4CC3C4C(=O)Nc3ccc(O)nc3)=O)cc2c1 68625,c1(NC(C2CCN(C(=O)Cn3ccc(O)nc3=O)C2)C)ccccc1[N+](=O)[O-] 68626,N1(C(C#C)=O)CCn2cc(C(=O)NCCNCCO)nc2C1 68627,CC1CC(CNC(=O)C(=O)NC2CC2)CN1C(=O)Cn1cnc(C#N)n1 68628,O=Cc1cccc(CN2CC3(CCC(C(=O)NC4CSC4)O3)C2)c1Br 68629,C1(C(=O)NC(C(=O)NCC2CC=CC2)C2(C)CC2)(C2CC2)CCCO1 68630,c1(CS(=O)(=O)NC(c2nncs2)CC)cccc(F)c1 68631,N1(C(C2(CC)CCCCC2)=O)CC(C)(C)C(O)C1(C)C 68632,C12(NC(c3c(CC)nn(C)c3)=O)CCC(CC1NC(C1(F)CCOC1)=O)C2 68633,C1(NC(CC2N(CC)CCOC2)=O)CCN(C(c2cn(C)nn2)=O)CC(C)(C)C1 68634,C1(CC=C)(NC(=O)C(c2ccc(C)cc2)N(C)C)CS(=O)(=O)C1 68635,c1(CN2CCC(NC(c3cccc(-c4nc[nH]n4)c3)=O)CC2)c(Cl)cc(Cl)cc1Cl 68636,C(=O)(C1=NOC2COCC12)N1C2C(N(C(c3cc(OC)ncc3)=O)C)CC(C2)C1 68637,c1(CC)nc(CC(=O)N(C2(CC(C(=O)C(C)NC3CCCC3)=O)CC2)CC)cs1 68638,CC1CCN(C(C2CCCC2(C)C)=O)CCN1C(c1cnco1)=O 68639,CCCCC(C(=O)NCCC1CCCCN1C(=O)CN(C)C)C(C)C 68640,n1(CC(N2CC(CNC(C(C)=C3CC3)=O)C2)=O)nnc(C2CC2)n1 68641,C(CCCCCNC(c1c(Br)noc1C)=O)NC(C(CC)OC)=O 68642,C(CCCC(=O)OC)(C(=O)NCc1cccc(Br)c1)N1CCCC(COC)C1 68643,C(=O)(C(C)CC(C)C)NCc1c(C(=O)NC(CCCC)(C)C)occ1 68644,Cc1cc(CNC(=O)C(=O)N(C)CCOCCOCCO)c(C)o1 68645,C(=O)(C1CCc2c(Cl)cccc21)OCC(=O)NC(Cc1ccc(C)cc1)C(=O)O 68646,N1(C(C)=O)CCC2(CC1)CN(CCn1cncn1)Cc1ccccc12 68647,CC1=CCCN(C(=O)NCCCC2CCCO2)C1 68648,S(=O)(=O)(c1cn(-c2ccccc2)nn1)NCC1(CO)C(C)(C)C1 68649,C(=O)(C(O)CC(C)(C)C)NC1C(CNC(c2c(C)[nH]c(C#N)c2)=O)CC1 68650,C1(C(=O)NCCC(=O)NC(CC)C)CCOCC1NC(C1OC2CCC1C2)=O 68651,c1(C(=O)NC2C(CNC(C3(Br)C(C)(C)C3)=O)C2)ccn2c(O)nnc2c1 68652,C(C(COC)C(=O)NC(CO)C(C)NC(C1(N(C)C)CCC1)=O)OC 68653,c1(CCC(=O)NCCN(C(=O)C(c2nc(C)cs2)C)CC)ccc(Cl)cc1F 68654,C12(COC)CC(CNC(c3ccc(Cl)o3)=O)(CN1C(C1(C(F)F)CCCO1)=O)C2 68655,C1(NC(C(C2(C)CC2)NC(CCC(CC)OC)=O)=O)CC2CC1C(O)C2O 68656,C1(CNC(C2(OC)CCOCC2)=O)CN(C(C2CCO2)=O)CCC1C 68657,N1(C(c2ccc(C3CC3)nc2O)=O)CC2CCCN(C(=O)Cc3cccs3)C2C1 68658,Cc1cc(C(=O)NCC(C)CN(C)C(c2c(C(F)F)cnn2C)=O)sc1C 68659,C(C(=O)NCc1cn(C2CN(C(=O)CC(C)C)C2)nn1)(C(C)(C)C)NC(C)=O 68660,N1(C(C(C(C)CNC(c2coc3c2COC3)=O)F)=O)CCCCN(C)CC1 68661,c1(-c2occ(CC(=O)NCCN(C(c3c(CC)nco3)=O)C)n2)ccc(O)cc1 68662,Cc1cc(C(=O)NCC(C)(C(C)C)NC(=O)CC2CCCC(C)(C)O2)nc(O)c1 68663,C1(N(C(=O)CN(C)C(N)=O)CC)CN(c2nnco2)C1 68664,c1(C(=O)NC2C(NC(c3sc(CC)c(C)c3)=O)CC2)ccc(F)c(F)c1C 68665,C1(C(N(CCN(C(CN2CCN(CC)CC2)=O)C)C)=O)CC(C2CCCC2)C1 68666,c1(OC)cc(O)ccc1NC(C1CC2CC2N1C(=O)Cc1cnc(C)s1)=O 68667,C1(=O)C(CCSC)N1.c1(CCN2CCC(OCC)C2)ccc[n+]([O-])c1 68668,C=CCCCCCCCC(=O)NCC1CCCN(C(=O)C(O)CC(C)C)C1 68669,N1(C(CCCCC(C)C)=O)CCC2(CCCCC2NC(c2ccccn2)=O)CC1 68670,N1(C(C2(C=C)CCN(C(=O)CN(C3CCC3)C)C2)=O)CC2CC(C)(C)C2C1 68671,O(C=CC(O)(CNC(c1ccccc1)=O)C(F)(F)F)CC.C1(=O)C(C)(C)O1 68672,c1(OC)c(C(=O)NCCC2CCCCN2C(=O)CCN(C)CCO)cccc1F 68673,Cc1cc(C(N2CC(NC(C3C4COCC34)=O)C(n3cccn3)C2)=O)nc(C)n1 68674,C(C)(CCC(=O)NC1CC1CNC(=O)CC1CC1(C)C)OC 68675,Cc1nc(-c2ccc(CN3CCC(NC(F)(F)CF)C3)cc2)nc(O)c1C 68676,CC(=O)CCCC(=O)N1CCC(C(F)(F)F)C(NC(=O)Cn2nc(C)cc2N)C1 68677,C#CC1CCCC(NC(=O)C(CCOC)NC(c2cc(C#N)c[nH]2)=O)C1 68678,N1(C(Cc2cnc(C)[nH]2)=O)CC2CCC2(CCC2N=N2)C1.C(=O)C=CC(C)C 68679,N1(C(C(C)NC(N)=O)=O)CC(NC(=O)CCN(C)CCO)C(c2ccccc2)C1 68680,C(=O)(C1=NOC2COCC12)N1CC=C(C(=O)NCCC(C=C)C)CC1 68681,c1(CC(=O)NC2CC(CNC(COCCC(C)C)=O)C2)ccc2ccoc2c1 68682,C1(CNC(C(CC)(F)F)=O)C(C)CCCN1C(=O)C(=O)NCCC(N)=O 68683,C(CNS(C)(=O)=O)(C(=O)NCCNC(C1CCCO1)=O)N(C)C 68684,S(=O)(=O)(c1cccc(Br)n1)N1C(C)(C(=O)NCc2cncc(Br)c2)CCC1 68685,C1(NC(C(CCC)C)=O)CCC12CCN(C(c1c[nH]c(=NC)s1)=O)CC2 68686,C1(NC(C2(SC)CC2)=O)CCCC2CN(C(c3noc4cc(F)ccc34)=O)CC12 68687,N1(C(COCCOC)=O)CC(C)CCC1CNC(=O)C(=O)NCC1CC1 68688,CCCCCCC(=O)N1CCCC1CNC(c1cccc(Cl)c1OC(F)(F)F)=O 68689,C1(NC(c2cocn2)=O)COC2CN(C(=O)Cc3ccc(F)cc3F)CC12 68690,O=c1cc(C(C)NC2CCCC(Sc3ccc(Cl)cc3)C2)nc2n(C)ccn12 68691,Fc1cncnc1Cc1nnc(N2CC3CCC2C3)n1CC(c1ccccc1)F 68692,c1(OCC)ccc(C(=O)NCC2CC(O)CN2C(=O)Cc2cc(C)cs2)cc1Cl 68693,c1(C(=O)NC2CC(C(=O)N)C2)ccnc(CN2CCC(C(F)(F)F)C2)c1.CO 68694,Cc1nc(Cl)nc(N2CCCC2CNC(=O)CCC2CCCC(O)C2)c1[N+](=O)[O-] 68695,CC(C)(C#N)CCC(=O)NC1(CNC(c2cc3ccccc3o2)=O)CCOC1 68696,C1(CC(C)(C)C)CN(C(C2(Cl)CC23CCC3)=O)CCN1C(c1sccc1CO)=O 68697,C1(C(NOCC(CC)C)=O)CCC(C)N1C(c1ccc(C)n1C)=O 68698,c1(C(=O)NCC2C(NC(C3CC=C(C)CC3)=O)C2)cn(C)cc(Br)c1=O 68699,C=CC(C)(C)CC(=O)NC1(CNC(=O)COCc2ccnn2C)CCCCC1C 68700,c1(C(N2CCC(OCc3cnccn3)CC2)=O)cc(Cl)c([N+](=O)[O-])cc1F 68701,CC1=NOC(C)(CNC(=O)C(CC2CCCC2)NC(c2cc(C)oc2C)=O)C1 68702,c1(CCOC(c2ccc(Cc3ccccn3)cn2)=O)ccccc1F 68703,CC1CC(NC(=O)C(C)NC2CCC2)CC(C)(C)C1 68704,c1(NC2(CNC(C(C)C3CC3)=O)CCC2)ccc(Cl)cc1Cl.C1(C(=O)N)C2CCCC12 68705,C(C(O)C(=O)NCCN(C(=O)C(C)N(C)C)CCSC)SC 68706,C1(CC(C)(C)C)CN(C(C2CC3CC3C2)=O)CCN1C(c1ccoc1C1CC1)=O 68707,C1(CC(C)NC(C=C(C)C(C)C)=O)CCN(C(c2cc(C3CC3)no2)=O)CC1 68708,CCC(CCCC(=O)NCCN1CCOCC1=O)NC(=O)C(CC)(CC)CO 68709,C#Cc1ccc(CNC(N2CCC3(CC2)COC3)=O)cc1OC 68710,C1(CNC(CSCC(C)C)=O)CC(F)CN1C(=O)CC1CCCO1 68711,C=CCCCC(C(=O)N(CC(C)C(C)C)C)NC(c1cc(C)on1)=O 68712,n1(CC)nnnc1C1(NC2(c3cnn(C(F)(F)F)c3)CC2)CCCC1 68713,c1(C(N2CC(F)(CNC(c3nc(C)oc3C)=O)C2)=O)cc(S(=O)(=O)N(C)C)c[nH]1 68714,c1(C(=O)NCC(=O)NCCC(C)NC(c2cccc(=O)o2)=O)ccc(N)cc1 68715,C(C)(C)(C(C)CC(=O)N1CCC2CC12)NC(CC(C)CN(C)C)=O 68716,Cn1c(NC(=O)CO)c(C#N)c(=O)n(C)c1=O.N12CC(CC1=O)CN1CC2C1 68717,CCCC(C)CC(=O)N(CCC)CCNC(C1(c2ccccc2C)CCCC1)=O 68718,C1(CCC(=O)NC2(COC)CCC2)CCN(C(=O)CCn2ccnn2)C1 68719,Cc1cc(C(N2CCCC(NC(=O)CN(C)C3CC3)C2)=O)c(F)cc1N 68720,C1(NC(c2scc(OC)c2OC)=O)CC2(C1)CN(C(C1CCOC1(C)C)=O)C2 68721,C1(OC)CCC2(CCN(C(c3ccc(CNC(=O)C4=CCOCC4)s3)=O)C2)C1 68722,c1(C(=O)NC2C(C=C)CN(C(c3ccc(CC)nc3)=O)C2)cccc2ccoc12 68723,c1(CNC(C2CC2(Cl)Cl)=O)csc(C(N2CCC(C(C)(C)OC)C2)=O)c1 68724,C(=O)(CS(=O)c1ccc(Cl)cc1)N(C1CN(C(C(=O)CCN2CCCC2)=O)C1)C 68725,c1(C(N(C(C)CNC(C2CC2F)=O)CC)=O)ccc(NS(C)(=O)=O)cc1O 68726,CN1CCN(C(=O)CCCCc2ccc(C#N)cc2)CC1CNC(C1(F)CC1)=O 68727,C1(CNC(=O)OC(C)(C)C)CC(CN(C2CC23CCCC3)C(=O)NCCO)CO1 68728,N1(C(CC2ON=C(C)C2)=O)CC2(CC(C(=O)NCCN3CCOCC3=O)CO2)C1 68729,C1(C)(NC(C(CC(F)F)NC)=O)CCc2ccccc2C1 68730,n1(CCC(=O)NCCOCC(=O)NCC(C)(C2CC2)OC)ccnc1C 68731,N1(C(C(CC)C)=O)CCC(NC(C2(CCOCCO)CCC2)=O)C1C 68732,Cc1ccc(C)c(CC(=O)NCC2CCN(C(c3cnc(C)cn3)=O)CC2)c1 68733,C1(CNC(C2CCC(C)S2)=O)CCN(C(=O)Cc2cccnc2)CC1 68734,N1(C(CCN(C)CC)=O)CCC(C)(CCNC(C2CCC(F)C2)=O)CC1 68735,C1(CNC(CCOCC)=O)CN(C(=O)C(c2ccccc2)NC(N)=O)CC1O 68736,CON1CC(C(=O)N(C2CCCCC2NC(=O)CCn2cnnn2)C)CC1=O 68737,C1(NC(c2snc3ccccc23)=O)COC2(C1)CN(C(c1ccon1)=O)C2 68738,CC1(C(N2CCC2CNC(C23C=CC(CC2)C3)=O)=O)CC2CCC1CC21OCCO1 68739,C(C)(C)(CCCCC(=O)NC1CCC(NC(c2cscc2OC)=O)C1)OC 68740,C(CC1CC1)(C(=O)N(CCCO)CC)NC(CN(C(=O)OCC)C)=O 68741,c1(C(N(CCNC(C2(C#C)CC2)=O)CCOCCO)=O)nnn2c1CCCCC2 68742,C1(F)(C(N2CCN(CC3(NC(c4c(C)ccs4)=O)CC3)CC2)=O)CCC(C)CC1 68743,c1(CC(=O)NCC(CNC(=O)C(O)C(F)F)OC)cc(F)c(F)c(F)c1 68744,N1(C(c2cncc(C#C)c2)=O)CCC(C(=O)NCCSCCO)CC1(C)C 68745,c1(SCC(=O)NC(CNC(c2nc(C(C)OC)oc2)=O)C)ccccc1O 68746,C(=O)(C#CC1CC1)N(Cc1c(C(N(c2ccccc2)CC=C)=O)occ1)CC 68747,C(=O)(C(C(=O)NC(C1CCCCC1)C(=O)N(C)Cc1cncn1C)OC)OC 68748,C(CC1CC1)(CC(=O)O)Sc1ccc(N)cc1.c12cn(nn1)CN(C)CCC2 68749,c1(C(=O)NCC2CC(NC(COC)=O)C2)ccc(NC2CC2)cc1O 68750,c1(C(=O)NCc2cc(OC(CC)C)ncc2)c(C)cc(Br)cc1F 68751,C1(CNC(C(CC)C)=O)CCCCN(C(=O)CCc2ccc(O)cc2)C1 68752,c1(CNC(=O)NCCOc2cn(C)nc2C(N)=O)cccc(C#N)c1Br 68753,c1(NC2(C)CC(NC(c3nc(CCC)sc3)=O)C2)ncnc(C)c1F 68754,c1(CNC(C(Cc2ccccc2)OC)=O)cccc(NC(C2CC(F)(F)C2)=O)c1 68755,C1(NC)CC2CCC1CC2.C1CCCCCNC(=O)N1.C1(OC)CC1 68756,C12(OC(N(CCC(=O)NCC)C)=O)CC1CN(C(=O)CCCOC)C2 68757,C(CC(C)C)(C(=O)NC(C(=O)N(CC1=CCCOC1)C)C1(O)CCC1)OC 68758,CN1CCC(NC(=O)NC2CCCC2O)C1C(F)(F)F 68759,Cc1[nH]nc(Cl)c1C(c1nnnn1C)NCCCc1cnoc1 68760,C1(NC(C2C(CC)CCC2)=O)CC12CCN(C(=O)CCc1ccccn1)C2 68761,N1(C(CC2CC(SC)C2)=O)CC2CCC1CC2NC(c1ncnc(C)c1C)=O 68762,C1(C(N2CCC2(C)C(=O)N(C)C)=O)(CC)CCCN(C(c2ccsc2C)=O)C1 68763,c1(C(=O)NCCCN(C)C(c2cnn(C)c2)=O)ccc(OCCOCC2CC2)nc1 68764,N1(C(c2c(OC)scc2)=O)CC(C(=O)NCC2(C)CCC2)C(C(C)C)C1 68765,Cc1cnc(CCC(=O)NCC2CCCN2C(c2nncn2C(C)C)=O)[nH]1 68766,c1(CC(N2CCC(O)(CN(C(c3cnc(Cl)s3)=O)C3CC3)C2)=O)cnccc1Cl 68767,Cc1cc(C(=O)Nc2cc(F)ccc2C(=O)NCC(F)(F)F)cc2c1CCC2 68768,c1(C(=O)NCCn2cc(C(N(C)Cc3nc(=O)o[nH]3)=O)nn2)cc(C#N)cn1C 68769,c1(CN(C(C)C)C)ccc([N+](=O)[O-])cc1.c12ccccc1-c1cc(ccn1)NC2 68770,C(CC(=O)NCC1CCN1C(=O)OC(C)(C)C)(C(F)(F)F)N(C)C1CC1 68771,O=C(C1=C(Cl)CCC1)NCCC1COCCN1C(C1CCC(F)(F)C1)=O 68772,CC1CCCN(C(c2c[nH]nc2C(F)F)=O)C1CCNC(c1ccc(C#N)[nH]1)=O 68773,C1(C2CCCCO2)(C(N(C)CCO)=O)CCCO1 68774,C1(CCC)CCCC1C(=O)NCCC(O)CNC(=O)C=CCOC(C)(C)C 68775,C1(C(=O)NCC(=O)NC(C)C)CCN(C(=O)COc2ccn(C)n2)C1C(C)C 68776,C(=O)(CCCC(C)NC(C1(OC)CCOC1)=O)N(CCCN(CC)CC)C 68777,c1(OC)ccc(N2CCC(NC(=O)C(=O)NC(c3cccnc3)(C)C)CC2)cc1 68778,N1(C(CCC=CC)=O)CCOCC(CNC(=O)C(C)SC)C1 68779,c1(SC(C)C(c2c[nH]cc(Cl)c2=O)=O)ccc(Nc2ncc[nH]c2=N)cc1 68780,C1(CC(=O)N(CCC(C(C)C)NC(=O)C(C)(C)CO)C)SC2=NCCN2C1=O 68781,c1(C(N2CCC(NC(C(C(C)C)OC)=O)CC2)=O)ncnc(O)c1Br 68782,c1(SCC(N2CCC(CNC(C(CC)F)=O)CC2)=O)ccc(F)cc1F 68783,C(=O)(CC(C)CC(=O)OC)N(C(CC)C(=O)NC1COCC1O)C 68784,c1(NC(CC2N(C(c3cc(C)[nH]c3)=O)CCC2)=O)ccccc1C(C)(C)C 68785,c1(N(CC(C)NC(c2csc3nccn23)=O)C)ncnc2c1ncn2C 68786,C=CCC(CC(C)C)C(=O)N1CC2(C1)CN(C(C1CC(O)CN1C)=O)C2 68787,C12(C(N3C(CN(C)C(c4cnc(Br)s4)=O)CCC3)=O)CCC(C)(C1)OC2 68788,N1(C(CC(C)C)=O)CCCC(C)C1CCNC(c1c(Cl)sc(C)c1C)=O 68789,c1(C(=O)NCCCCC2CN(C(C3CCC(C)O3)=O)C2)c(F)ccc(F)c1F 68790,N1(C(C2CCc3nnc(O)n3C2)=O)CCC2C(CCCN2C(=O)C2=CCCC2)C1 68791,C(=O)(C(=O)N=c1ncn(-c2ccccc2)[nH]1)NC1C(C)C2CCC1C2 68792,Cc1ccc(CNC(C2CCC2CNC(=O)C=CCN2CCC2)=O)cc1F 68793,C1(N(C(=O)C(C)OCC(F)(F)F)C)CCCN(C(=O)CSc2nccn2C)CC1 68794,C12(NC(C(C)SC)=O)CCCC1N(C(=O)CC=CC(C)(C)C)CC2 68795,CN1CC(C)(C)CC1C(N1CC(C(N)=O)(CNC(c2cc(F)ccc2N)=O)C1)=O 68796,CN1CCN(C)C(C(N2CCOC(CNC(=O)CCC(C)(C)C)C2)=O)C1 68797,Cc1ccc2c(C(=O)NCC(C)(CO)NC(C34CCCC3C4(F)F)=O)onc2c1 68798,c1(OC)cc(C(F)(F)F)ccc1-c1cc(CN2CCC(Br)CC2)ccn1 68799,C(=O)(C(F)(F)F)NCC(=O)NCCCN(C(=O)CNc1cccnc1)CCO 68800,C=CC1CN(C(=O)C(C)P(C)(C)=O)CC1NC(c1cnc(-c2ccccc2)[nH]1)=O 68801,c1(C(=O)NC2CCC(C)N(C(C3CCC(=O)N3C)=O)C2)cccc2c1ncn2C 68802,C1(NC(CCc2onc(C)n2)=O)COCCN(C(=O)CC2COCCO2)C1 68803,N1(C(CC2C(COC)CC2)=O)CCCC(O)(CNC(c2cn(C)nc2OC)=O)C1 68804,O=C(NNc1cccc2c1OC(F)(F)O2)c1c(Br)ccc(F)c1I 68805,c1(C(=O)NCCCN(C(c2c(C)sc(O)n2)=O)C)cnc(Cl)c(N)c1 68806,N1(C(C(C2CCCC2)OC)=O)CCCC2(C1)CN(C(C1(C3CCCO3)CC1)=O)C2 68807,C12(C(=O)NCC3(CCNC(C(C4CC4)OCC)=O)CC3)CC(C)(C1)OC2C 68808,C12(C(=O)NCC(CNC(C3(CS(N)(=O)=O)COC3)=O)O)CCCC(=O)N1CCC2 68809,C1(NC(C=C(C)C(C)C)=O)CC2CN(C(c3csc(CC(C)C)n3)=O)CC12 68810,N1(C(C(CCC)N(C)C)=O)CC(C)N(C(=O)CC(C)(C)COC)C(C)C1 68811,C1(C(=O)NC2(CF)CCN(C(C3N(C(=O)NC)CCC3)=O)C2)CC2C(C1)C2(F)F 68812,C1(NC(C(CC)NC(N)=O)=O)CC(OC)CN(C(=O)Cc2c(O)ncnc2O)C1 68813,C1(C(C(=O)N(CC(CC)O)CC)F)CCN(C(=O)CC2(CC)CCC2)C1 68814,Cc1cnc(NC(C2CCN(Cc3ccc(Cl)cn3)CC2O)=O)nc1Cl 68815,c1(CN=[N+]=[N-])ccc(CNC2(C3CC3)CCCC2)cc1 68816,c1(CN2CCC(CC(=O)NC(c3c(C)noc3C)CC)C2)c(O)cc(O)cc1O 68817,CC(C)CC(CC(C)C)C(=O)Nc1cccc(-c2ccc(S(C)=O)cc2)c1 68818,c1(SC)cc(C(=O)N(C)CC2CCCN(C(=O)CC3COCC3O)C2)nn1C 68819,c1(C(C)C)nncn1C(C)C.N12CCCC1CCCNC(=O)CNC(=O)C2C 68820,N1(CCCNC(C2C(=C)CC2)=O)CC(NC(C2(CCOC)CCC2)=O)CC1=O 68821,Cc1ccc(C(=O)NC2CC3CC(NC(=O)C4=CCCSC4)C3C2)nc1F 68822,N1(C(C(C)(Cl)Cl)=O)CCC(CF)(NC(c2c[nH]cc2Br)=O)C1 68823,C(=O)(CCCC(F)(F)F)N1C2(C(=O)NC(c3n(CC)ncn3)C)CC(C)(C1)C2 68824,N1(C(c2cn(CCOC)nc2)=O)CC2CCC1CN2C(=O)C(=O)NCC(F)(F)F 68825,N1(C(c2snc(OC)c2I)=O)C(CO)CCCC1CO 68826,c1(C(=O)NCC2N(C(CC(C(C)C)O)=O)CC(O)C2)ncn2ccccc12 68827,c1(-c2cccc(OC)c2OC)cccc2c(NC(=O)C(C)=O)cccc12 68828,c1(OC)ncc(C(=O)NC2CCC(NC(c3scc(C)c3Cl)=O)C2)cc1Br 68829,N1(C(C(C)SC)=O)CC=C(CC(=O)NCC2CCN(C3CC3)C2)CC1 68830,N1(C(c2c(C)noc2C)=O)CC2CC(O)C1C2NC(c1ccc(CO)cn1)=O 68831,C=CC(F)(F)C(=O)NC(CN(C(=O)C(CC)=Cc1cn[nH]c1)C)CC 68832,C1(O)(CC(=O)NCC2(C(=O)NCCN(C(C)C)C)CC2)CCCC1 68833,C1(NC(C2(N(C)C)CCCC2)=O)CC2CC(NC(=O)Cc3cnoc3)CC12 68834,C=CCCC(F)(F)C(=O)NCCOCCN(C)C(c1cn2cc(C)nc2s1)=O 68835,CC1c2nncn2CCN1C(c1ccc(CNC(=O)CSc2cn[nH]c2)s1)=O 68836,C1(NC(c2n(CC)nc(C)c2)=O)CCN(C(C23CC(C)(CO2)C3)=O)C12CCC2 68837,C=CCCC(CC(C)C)C(=O)NCC1CCN(C(c2cc(Cl)cc(C)c2C)=O)C1 68838,N1(C(c2cc(C(F)(F)F)c[nH]2)=O)CC2(C1)CN(C(C1(N3CCCC3)CC1)=O)C2 68839,C(C(C)(C)CC(=O)NC(C)CCO)NC(Cn1c(C)nc(C)n1)=O 68840,c1(CC)cccc(N(C)C(C2COCC2NC(=O)CCc2ccn(C)c2)=O)c1 68841,N1(CC)CCCC(C(=O)NC(C)(C)C(C)NC(C2CC(SC)C2)=O)C1 68842,S(=O)(=O)(c1c[nH]c(=NCCC#N)cc1C)NC(CC)C(C)O 68843,CN1CC2CCCN(C(=O)CCn3cc(CCCN4CCOCC4)nn3)C2C1 68844,C1(C(=O)NCC(C(C)C)NC(=O)CCCC2CC2)CCC(C(=O)N(C)C)CC1 68845,CC(C)(C)C#CC(=O)NCC(CC(=O)NCC1OC(=O)CC1(C)C)OC 68846,c1(CNC(=O)NC2CC3(CC(C)OC3)C2)ccc2c(c1)CN=S2(C)=O 68847,c1(C(N2CCC(O)(CNC(C3CCCN(C(C)=O)C3)=O)C2)=O)c(C)cc(C)nc1O 68848,C1(CC)(NC(C2CCCCC2NC(=O)C(C)C(O)CC)=O)CCCCCC1 68849,C12(CNC(CCCC)=O)CCC(CC1)N2C(=O)C(N1CCCCCC1)C 68850,c1(CC(=O)NC(CN(C(c2csc(C3CC3)n2)=O)CC)C)ccccc1C 68851,C1(NC(CSC(C)=O)=O)CCCC2CN(C(c3ccnc(F)c3F)=O)CC12 68852,N1(C(C2CCCN(C(C3CC4CC(=O)C3O4)=O)CC2)=O)CCOCC(C2CC2)C1 68853,c1(CC(C)C)cccc(C(N2CCC(C(C)(C)NC(c3c[nH]c(Br)c3)=O)C2)=O)c1 68854,C(C)(C)(CCCNC(=O)C=CC=C(Cl)Cl)NC(C(CC)n1ccnc1)=O 68855,C1(C)(NC(COCC(=O)OC)=O)CCCN(C(C2(CS(C)(=O)=O)COC2)=O)C1 68856,C1(C(N2C(C)CCC2)=O)C2CC1N(Cc1ccc(O)nc1)C2 68857,Cc1cc(C(=O)N(C)CCC2CCCCN2C(=O)CN2CCSCC2)ccc1O 68858,c1(C(=O)NC(C2CCCN(C(CNC(CC)=O)=O)C2)C)c(F)c(F)cc(F)c1F 68859,C(CC(C)C)(CC(C)C)NC(CCNC(CN(C(COC)=O)C)=O)=O 68860,C(=O)(C(CC(C)C)C(N)=O)CCC1N(C(C(CC#C)C2CNC(=O)N2)=O)CCOC1C 68861,N1(C(CSCC(=O)OC)=O)CCCC(CCNC(c2cccn2C)=O)C1 68862,N1(C(c2ncc(CC)cn2)=O)CCC2CN(C(=O)CCS(N)(=O)=O)C(C)C12 68863,c1(OC)ccc2c(c1)C(C)(C)N(C(=O)CC(C)C(C)C(F)(F)F)CC2 68864,CCCCCCC(C)CC(=O)NC1CCC2(CC1)CN(C(c1ncnn1C)=O)C2 68865,C1(C(N(C(C)C(N)=O)C)=O)CC12CCN(C(=O)Cn1cnnn1)CC2 68866,CC(C)(C)CCC(=O)NC1(CO)CCN(C(=O)CC2CCC(C)(C)CC2)CC1 68867,c1(C(=O)NCC2CC(NC(C(C)C3CCCO3)=O)C2)cc(Br)cs1 68868,CC(c1ccc(F)cc1F)=CC(=O)N(CCCCNC(C1CC2CC2C1)=O)C 68869,C#CC1(C(N2CCC(C(C)O)CC2)=O)CCN(C(c2cc(Cl)c[nH]2)=O)C1 68870,C(CN=c1cc(-c2cccs2)nc[nH]1)NC(CC1CC(C)(C)OC1)=O 68871,c1(C(CC)=O)cccc(NC(N2CCCC(N(C)C(C)=O)C2)=O)c1 68872,c1(CC)cccnc1C(N1CCC(CCC(=O)NCC(C2CCC2)OC)C1)=O 68873,CCC(C)C(CC(=O)N(C1CCOC1=O)C)NC(c1ccn(COC)n1)=O 68874,N1(C(C2(CCOCC)CCC2)=O)CCC2(CC1)CC2NC(=O)C1=CSCS1 68875,c1(-n2cc(C3N(C(CS(C)(=O)=O)=O)CCCC3)nn2)cccc2c1CCCC2 68876,C1(CNC(=O)C2CC2)CC2(CCN(C(=O)CCOc3ccccc3)C2)CO1 68877,C=CCC(C(=O)NC1(C)CC(NC(C2CC2c2ccc(F)cc2Cl)=O)C1)C(C)C 68878,N1(C(C=CC)=O)CCC(O)(C(C)NC(c2c[nH]c(C)cc2=O)=O)CC1 68879,C(C(O)C(F)(F)F)N(C(C1(NC(c2cc(C)[nH]c2)=O)CCSC1)=O)C 68880,c1(OCC)cc(C(=O)NCC(CNC(=O)CCC(C)OC)CO)ccc1C 68881,CC#CCCCC(=O)NCC1CN(C(=O)CCCOC2CCOCC2)CCO1 68882,c1(CC)nn(C)cc1C(=O)N(C(CC)C(=O)NCC1=CCCCC1)C 68883,C1(NC(c2c(CC)nns2)=O)CCCC12CN(C(c1cc(O)c(F)cc1N)=O)C2 68884,C(=O)(C(CNC(C1CC1C(F)F)=O)CC(C)C)NC(c1nc[nH]n1)CC 68885,c1(-c2c(C(=O)NCC#CC)cccc2)ccc(C(C)NC(C)=O)c(F)c1 68886,N1(C(C(C(=O)OCC)CO)=O)CC(n2cc(OC3CCC3)nn2)C2(CCC2)C1 68887,Cc1nc(O)sc1C(=O)NC(Cn1cccn1)C(=O)NCCC(C)(C)C1CC1 68888,CC1CN(C(=O)Cc2ccccc2O)CC1CNC(c1ccoc1C(F)(F)F)=O 68889,c1(C(=O)NC2CCCN(C(CCSC)=O)C2)ccc([Si](C)(C)C)s1 68890,C1(C(=O)NC(C)CCCNC(=O)C(C)OCC2CC2)C(C(F)(F)F)C1[N+](=O)[O-] 68891,N1(C(C2N(C(c3c(CC)nn[nH]3)=O)CCC2)=O)CCC(C)(C2CC2)C1 68892,C=CC(C)(O)CC(=O)N(C(CNC(=O)C(C)Sc1ccccn1)CC)C 68893,N1(C(CNC(=O)OC)=O)CCN(C(c2cn3ccncc3n2)=O)CC(O)C1 68894,CCN=C(NCc1ccc(CC2CCCCC2)o1)N1CCC2CCCOC2C1 68895,C1(C(=O)Oc2cccc(N(CC)CC)c2)CC2CCCC(C1)C2 68896,C(C)(C)(CCC(=O)N1CCC(C)(C(=O)NCC2(C)CCC2)C1)N(C)C 68897,C=CC1COCC1NC(C1CSCN1C(=O)C(C(=O)OC)OC)=O 68898,C1(NC(C=Cc2scc(C)n2)=O)CCCC12CCN(C(=O)Cc1ccon1)C2 68899,N1(C(=O)OC(C)(C)C)CCC2CC12CC(N1CCN(c2ccsc2C#N)CC1)=O 68900,c1(C(C)=O)ccc(C(=O)NCC2CCCN2C(=O)Cc2cc(C)no2)cc1 68901,C1(C(=O)NC2CCN(C(C3COC(=O)O3)=O)CC2)CCc2ncncc2C1 68902,C1(CNC(c2n(CC)ccn2)=O)CC(C)N(C(c2sccc2F)=O)C1 68903,C1(C(=O)NC2C(C=C)CN(C(=O)CC(=C)Br)C2)CCCCCS1(=O)=O 68904,C1(SC)CC(N=c2cc(C)nc(N3CC=CCC(C)(C)C3)[nH]2)C1 68905,N1(C(c2c(C)cc[nH]2)=O)C2CCC(C2)C1C(=O)NCC(O)C(F)F 68906,c1(C(=O)NCc2cn(C)nc2)ccc(Cl)cc1NCc1cn(CC(C)(C)C)nn1 68907,c1(C(=O)NCCC(=C)CNC(C2OCCC2C)=O)cccc2c(C)[nH]nc12 68908,C1(C(=O)NC(C2(O)CCCCC2)C)CCCN(C(c2ccc(Br)nc2C)=O)CC1 68909,C(=O)(C1c2c[nH]nc2CN1C(=O)CC(C)n1ccnc1)Nc1ccc(C)c(F)c1 68910,C1(OC)CN(C(C23CC(C2)C3)=O)CCC1NC(c1cc(B(O)O)co1)=O 68911,N1(C(C(C=C)O)=O)CCC(C(=O)NCC(O)C(=O)OC)(CC)C1 68912,CCCC(C(O)C(=O)NCCC1CCCC1)NC(=O)C(CC)C(C)C 68913,N1(CCN(C)C(C2(NC(C3CCC3(F)F)=O)CCSC2)=O)CCOC1=O 68914,C12(C(=O)NC3C(C)CN(C(c4cncn4C4CC4)=O)C3)CCC(CF)(C1)OC2 68915,C1(C(CNC(C(C)(C)SC)=O)(C)C)CCN(C(c2oc(C)cc2C)=O)CC1 68916,N1(C(C=Cc2c(C)n(C)nc2)=O)CCCC(NC(=O)Cc2cncn2C)C(F)C1 68917,C1(C)(C(=O)NCCNC(c2cc(SC)oc2)=O)CCCCCC1 68918,c1(C(=O)NCCN(C(=O)CC2(O)CCCC2)CCC)ncc(C(C)(C)C)o1 68919,C1(CC(=O)NCCCOC=C)CCN(Cc2cn(C)nn2)C1 68920,CCCCCCC(=O)NCC(C(C)C)NC(=O)Cn1cc(C2CC2)nn1 68921,Cc1ncc(CC(=O)NC2CC2NC(c2sccc2SC(F)F)=O)s1 68922,c1(NC(C)=O)ccc(F)c(N(C2CC3CNC2C3)C(=O)C(C)(F)F)c1 68923,C1(CNC(c2c(C)n[nH]c2C)=O)CCN(C(C2CC2c2nccn2C)=O)CC1C 68924,C1(C(N2C(C)C(NC(=O)C(F)(F)c3cscn3)CC2)=O)CSc2ccccc2O1 68925,N1(C(C(CCC)CC(C)C)=O)CCC(C2(O)CCN(C(=O)CNC(=O)NC)C2)CC1 68926,C1(OC(C)(C)C)CC(C(=O)OCC2CC(F)C2)C1 68927,c1(C(=O)NCC(CNC(CNS(N(C)C)(=O)=O)=O)F)ccc2c(c1)CCO2 68928,N1(C(C2CC(NC(c3ccc(C#C)o3)=O)C(O)C2)=O)CCCCC(C)C1 68929,C1(C(=O)NCCC(C(=O)OC)C)CC(C)(C)CN1C(c1ccn(C(F)F)n1)=O 68930,C(CCC(C)CC(=O)N1CC(NC(C2(C)CCC2)=O)C2CC2C1)=C(C)C 68931,C1(CCNC(c2c(CC)occ2)=O)CN(C(=O)C(c2cccc(C)c2)O)CC1C 68932,C1(NC(CC2(CC=C)CCCC2)=O)CN(C(=O)NCc2ccccc2C)CCO1 68933,N1(C(c2c(CC)ccc(F)c2)=O)CC2(CCCC(CNC(=O)OC(C)(C)C)O2)C1 68934,C1(NC(C2(C)CC(C)(C)C2)=O)CCN(C(=O)CC2CC(F)(F)C2)CC1O 68935,C1(c2nnnn2C2CC2)(NC(COC)C)CSC(C)(C)C1 68936,CSC1=C(C(=O)NC2CN(C(=O)C3=NOC(C)C3)CC(C)(C)C2)CCCC1 68937,c1(N2CC(CN(C(c3n(CC)nnc3)=O)C)OCC2)nc(C(C)C)nc(C)c1Br 68938,C1(N(C)C(c2cnc(SC)s2)=O)CN(C(C2(C(F)F)CCCC2)=O)CC1F 68939,C1(c2c(OC)cccc2)C(NC(c2cccc(C3CNC3)c2)=O)CC(=O)N1C 68940,N1(C(c2n(CC#C)ccc2)=O)CC(NC(=O)C(C2CCCCC2)OC)C(CO)C1 68941,c1(CCCC(=O)NCC2(O)CCN(C(=O)C3CC3)CC2)c[nH]c2ccccc12 68942,C1(NC(c2cn3ccnc3s2)=O)CN(C(C2CC=CC2)=O)C2(CCCOC2)C1 68943,C(=O)(C=C1SCC(=O)N1C)NC12CCCN(C(CC3C(C)CCCC3)=O)CC1C2 68944,C(=O)(C(C)(C)CC(F)F)NC(CNC(CCCC(=O)NCC)=O)(C)C1CC1 68945,C1(NC(C(C)(C)Cc2cccc(Cl)c2)=O)CC2CC(C1)N(C(=O)CCC1CC1)C2 68946,c1(CC)ccc(C(=O)O)cc1.C1(N(C(C)=O)CC)(CO)CCOC1 68947,c1(CC)nnc(C)cc1C(=O)NC(C)CC1CN(C(c2cnn(C(C)C)c2)=O)C1 68948,N1(C(C2(NC(C3(CC(C)=O)CC3)=O)CC(O)C2)=O)CCOC(C2CC2)CC1 68949,C1(O)(CNC(CCC2C(C)C2)=O)CCN(C(c2ccc(=N)[nH]c2Cl)=O)CC1 68950,Cc1cc(=NC2CC(C)N(C(=O)CCOCC(F)F)C2)[nH]c(C(F)(F)F)n1 68951,CC1(C)CN(C2(c3cn(-c4cccnc4)nn3)CC2)CCC1c1cc[nH]n1 68952,C1(CNC(=O)Cc2coc(C(F)F)n2)CCCC1NC(=O)CC1C=CCC1 68953,CN(C)S(=O)(=O)N1CCC(C(=O)NC2C=CCN(C(=O)CC3CC3)C2)CC1 68954,c1(-n2c(C(C)OCC)nc(-c3cccc(Br)c3)n2)ccc(Cl)c(F)c1 68955,c1(C(N2C(CCC(N3CCC(=O)NCC3)=O)CCC2)=O)ccc2c(c1)CCCO2 68956,C(C(C(C)C(C)C)NC(C1(C(F)(F)F)CC(F)(F)C1)=O)NC(CCOCC#C)=O 68957,CCC(C)CCC(=O)NCCNC(=O)C(c1ccc(C(C)(C)C)cc1)=O 68958,c1(NC(CC2CC(C)C(C)CC2)=O)cccc2c1C1CCC2CC1 68959,C(=O)(C1CCc2cccnc21)NCC(CNC(c1ccc(C)cc1Cl)=O)(C)C 68960,C12(CNC(c3c(COC)scc3)=O)CCCC1CN(C(=O)CCC(C)(C)F)C2 68961,Cc1cccnc1C(=O)NCCC1CCCN(C(=O)CCn2cnnn2)C1 68962,N1(CC(N2C(C(C)NC(=O)C=C3CCSCC3)CCC2)=O)CC2CCC1C2 68963,c1(CC)ncccc1NC(=O)CCNC(=O)C(C)=C(C)C 68964,C1(C(=O)NC2(CN(C)C(C34CC(CC(F)F)(C3)C4)=O)CC2)CCOCC1(C)C 68965,N1(C(C(=O)NC2(Cl)CC2(F)F)=O)CCC2(CCOC2)C1 68966,Cc1nccc(C(N2CCCC(NC(C3CC(C4CCC4)C3)=O)C2)=O)c1N 68967,c1(CN2CCC(C(N3CC4(CCC4)C3)=O)C2)c(O)cccc1F 68968,N#CCCCCC(=O)NC1CCN(C(C23CC(CO)(C2)C3)=O)C(C2CC2)C1 68969,C#CCC(CC(F)F)NC(c1cn(CCNC(C2CC2C(=O)OC)=O)nn1)=O 68970,C1(CCNC(C2N(CC)CC2)=O)CCCN(C(=O)C(C)(C)c2ccccc2)CC1 68971,c1(CCOC(CCC2=CCCN(C(=O)OC(C)(C)C)C2)=O)cn2cccnc2n1 68972,c1(CN2C(C)(C(=O)NCC3CCC(F)C3)CC2)cc(C#N)ccc1F 68973,CON=Cc1ccc(C(=O)NC(C2CCOC2)CNC(C2(C(F)F)CC2)=O)cc1 68974,c1(OC)ccc(C)cc1C(N1CCC(C(C)NC(=O)C(C)n2cccn2)C1)=O 68975,c1(C(N(CCCNC(=O)CCC2CC2)C2CC2)=O)ccc(=O)n(CCF)n1 68976,Cc1[nH]c2ccc(F)cc2c1C(=O)NCCNC(=O)CCCc1ccc(Cl)cc1 68977,c1(C(C)C(=O)NC2CCC(CCNC(=O)OC(C)(C)C)C2)ccc2c(c1)OCO2 68978,c1(C(N2CCC(CNC(Cc3nn(C)c(Cl)c3)=O)C2)=O)cc(N)cnc1Cl 68979,CC1CCCc2nc(C(=O)NC(C)CCCNC(=O)CSc3n[nH]c(=N)s3)cn21 68980,C1(C(=O)NCC2(C)CCN(C(=O)C=CC3CCCCC3)C2)CC(C2CCCC2)C1 68981,N1(C(C2(N(C)C)CCC2)=O)CCC2(NC(c3cccc(=O)o3)=O)CC2C1 68982,C1(C(N(C(C)CCNC(=O)CCC2(C)CC2)C)=O)CCN(c2nccn2C)C1 68983,C1(CC(N2CCC(N(C(=O)CCSCC)CC)C2)=O)CCc2ccccc2C1=O 68984,C(=O)(CCCCCC#N)N1C(C)CC(CCNC(=O)CCC(N)=O)CC1 68985,C(=O)(CCCN=[N+]=[N-])NC1(C)CCN(C(c2csc(-c3ncccn3)n2)=O)C1 68986,Cc1cc(NC2CCN(C(C3CC(C)(C)OC(C)(C)C3)=O)C2)ccc1[N+](=O)[O-] 68987,C(C)(CCC(=O)N1CCOC(CNC(=O)CCc2nnc(C3CC3)o2)C1)OCC 68988,c1(C(N2CC(C(N3CC(CCC#C)C3)=O)OCC2)=O)cccn(C)c1=O 68989,Cc1cc2ncc(C(N3CCC(C)C(NC(C4CNC(=O)C4)=O)C3)=O)cn2n1 68990,C(=O)(N1CC(O)CCO1)c1c(CNC(C2(C)COC(=O)N2)=O)n[nH]c1 68991,c1(C(=O)NCCC2CCCN(C(c3ccn(CC#N)n3)=O)C2)ccc(Cl)cc1O 68992,C(N=c1ccc(C#N)c[nH]1)C1C(NC(COC2C(CC)CCCC2)=O)CCC1 68993,c1(C(N2CC(CNC(CC=CC)=O)C(C)C2)=O)cc(C)cc2ccoc12 68994,N#Cc1ccc(C(=O)NCCCCCNC(c2cnc(S)[nH]2)=O)cc1O 68995,c1(OCC(=O)NC(CCCC)CNC(=O)CC2COC(=O)N2)cc(Cl)ccc1C 68996,C(=O)(C(CC1CCCO1)C(F)(F)F)NC(C1CN(C(=O)C(F)C2CCCC2)C1)C 68997,c1(CNC(NC(C2CCC2)C)=NCC23CCCCC2C3)ccc2c(c1)OCC2 68998,CC1CC=C(C(=O)N2CCCC2CN(c2ncccc2[N+](=O)[O-])C)CC1 68999,c1(N(C(C)=O)C)ccc(F)c(C(=O)NCC(CC)NC(=O)CCc2cnn[nH]2)c1 69000,c1(NC(=O)OC(C)(C)C)c(F)ccc(CC2CCCC3(CC3)C2)c1F 69001,C(C(C(C)C(C)C)NC(C1CN(C2CCCCC2)C1)=O)NC(c1cc(C)sc1)=O 69002,C1(C(=O)NCCCC(C)NC(c2c(OC)cc(C)cn2)=O)CCCC1S(C)(=O)=O 69003,c1(C(=O)NC2CN(C(C3C(C)CCC3)=O)C2)nn(C)cc1N 69004,N1(C(CCSCC)=O)CCN(C(c2cnn(CCOC)c2F)=O)CC1CO 69005,C1(NC(CC)=O)CCC2CN(C(C3(c4cccc(Br)c4)CC3)=O)CCC2C1 69006,c1(C(C)(C)C)cc(Br)cc(Br)c1OC(c1n[nH]cc1C(=O)N(C)C)=O 69007,C=CCCCC(C(=O)NCC(C)(O)CCO)NC(=O)C(C)N(C)C(C)=O 69008,Cc1ccc(NC(=O)COC2CCN(C(=O)CNc3ncccn3)C2)cc1C 69009,c1(C(=O)NCC2C3N(C(C=CC(C)C)=O)C(CC3)C2)cc2ncccc2o1 69010,C1(C(=O)NCC(CC)(C)C(N)=O)CN(C(C2CCN2C)=O)CC(C)(C)C1 69011,N1(CC(C)(C)NCC(=O)N(C(c2cccc(OC(C)(C)C)c2)=O)CC)CCOC(C)(C)C1 69012,S(=O)(=O)(c1cnc(N2CC3CC2CO3)c(Cl)c1)NC1C(C(N(C)C)=O)C2CCC1C2 69013,c1(C(C)C)c(C(N2CCCC(NC(=O)C=CCF)C2)=O)cnn1CCO 69014,C1(C(=O)NC(CCSCC)C)CCCCCCN1C(C1CC(N=[N+]=[N-])C1)=O 69015,CC1(C)CCN(C(=O)CC2CCSC2)C1CC(=O)NC1(C)CC2(CC2)C1 69016,Cc1cc(C)c(C(=O)NC2CCCCN(C(C3CC34CC4)=O)C2)c(Cl)n1 69017,C1(NC(C(c2ccc(OC)cc2)O)=O)CC2CC1CN(C(=O)CC1CN(C)C1)C2 69018,N1(C(C(CCOC)C)=O)CCC(CNC(=O)Cc2nc[nH]n2)(OC)CC1 69019,Cc1nc(C)c(C(=O)NC(C2CN(C(c3cocc3C)=O)C2)C)[nH]1 69020,N1(Cc2ccccc2)CCC(C(C(=O)CCc2cnc(C3CCC3)o2)C2(C)CC2)C1 69021,c1(C(N(C(CCC2CC(C)C2)=O)C)=O)ccc(=N)[nH]c1 69022,c1(-c2nc(CCCCC)nn2C(Cc2cn[nH]c2)CC)cnc(O)nc1O 69023,C(C(CC1CC1)C(=O)NCC1CC=CC1)NC(CC1N(C)CCC1)=O 69024,CC1(C(=O)NCc2ncccc2CNC(C2CCCC(=O)N2)=O)CNC(=O)N1 69025,C1(NC(c2cnnc(C)c2C)=O)CC2CCC1CN2C(C1CCOC(=O)CC1)=O 69026,Cc1c(C(=O)NS(=O)(=O)c2ccc(I)cc2)oc2cc(Cl)ccc12 69027,c1(CC)nc2sc(C)cn2c1C(N1CCC(C)(NC(=O)CC(F)(F)F)C1)=O 69028,N1(c2n(C(c3ccc4c(c3)OCO4)C)nnn2)CC(CCO)Oc2ccccc21 69029,N#Cc1cccc(F)c1CC(N1CC2CC(NC(=O)C#CC3CCC3)C1C2)=O 69030,C1(C(N2CCC(C(C)NC(c3cnc(C(F)(F)F)s3)=O)C2)=O)CCS(=O)(=O)N1 69031,C1(CC)CN(C(=O)CCOCC2CC2)CCC1NC(=O)CC1CCC=CCC1 69032,Cc1ccc(C)c(NC(=O)C(CO)NC(=O)Cc2cc(C)no2)c1 69033,N1(C(C2CN(CC)C(=O)C2)=O)CC(C(=O)NCC(=O)NC2CC2)CC12CCC2 69034,N1(C(CCCC2(NC(C3(C)CCCOC3)=O)CCC2)=O)CC2(CC(C(F)F)C2)C1 69035,c1(C(N2CCCC(CCNC(C3CC(=C4CC4)C3)=O)C2)=O)cc(F)c(O)c(F)c1 69036,C1(CCCC)CCC(C(=O)NCC(O)CNC(C2(Cl)CC2(F)F)=O)CC1 69037,C(C)(C)(C(=O)NCCC1CC(NC(C2CSCCS2)=O)C1)OC(C)C 69038,C(C)(C(=O)N1CC(OC2CCOCC2)C1)(C(C)C)SC 69039,c1(C(C)(C)C)nocc1C(=O)NC1CCCC1NC(=O)C(F)CC1CCCC1 69040,c1(C(N2CCC(C(C)NC(c3c(COC)cco3)=O)C2)=O)ccc(Cl)cc1SC 69041,Cc1nc2ccccc2cc1C(N1CCOC(C(C)(C)O)C1)C(=O)NCC(C)C 69042,C(=O)(C(C)CC(F)(F)F)NCC1(OC)CN(C(c2ccnc(-n3ccnc3)c2)=O)C1 69043,c1(NC(C)=O)cnc(N2CC(NC(=O)C3=CCCCO3)C3CC23)nc1C 69044,N1(C(c2ncc(CC)s2)=O)CC(N=c2ccn3ccnc3[nH]2)CC2(CCC2)C1 69045,C1(c2nnnn2CCOC)(NCCCC(C)(C)C)CCCC(C(F)(F)F)C1 69046,c1(CC(=O)Nc2cnc[nH]2)ccc(F)c(Cl)c1F.C12(CC1)C(=O)N(C)C2 69047,C1(C(N2CCCC(CC(F)F)C2)=O)CCCC(OC(COC(C)(C)C)=O)C1 69048,C(=O)(CCC(C)(C)C#N)NC(c1ccc(C)cc1)C(=O)NC(COC)C(C)C 69049,C(CC1=CCOCC1)C(=O)NC1C(CNC(=O)CC(C2CC2)C2CC2)CC1 69050,Cc1ccn2cc(C(=O)NC3CN(C(C4CCC(N=[N+]=[N-])C4)=O)CC3(C)C)nc2c1 69051,N1(C(CC2(C)CC2)=O)CC2CCCC(C1)N2C(=O)CC1CCCCCC1(F)F 69052,CC1CS(=O)(=O)CC(C)N1C(C1SCCS1)=O 69053,C1(NOC(C(CCC=C)NC(c2ccccc2)=O)=O)CCC2(CCC2)C1CO 69054,C(=O)(C1=CCOCC1)NCc1cc(C(N(C2CCCC2(F)F)C)=O)on1 69055,c1(C(N2CCCC(N3CCCC3)C2)C(=O)NCCCF)ncccc1F 69056,CC1(C(F)(F)F)CCN(C(=O)NCc2cccnc2)CC1 69057,c1(CNC2CN(C(c3ccc(F)c(F)c3)=O)CC(F)C2)cc(Cl)c2cn[nH]c2c1 69058,c1(-c2c(C(=O)NC(c3ccccc3)CC)c(F)cnc2)c(F)cccc1Cl 69059,c1(CC(C)C)ccccc1C(=O)NC(C)(C)CNC(=O)CCN1CCNC(=O)C1 69060,c1(C(N(CCCNC(=O)CC2CC(O)C2(C)C)C)=O)csc(S(C)(=O)=O)c1 69061,N(C1CCC(N=c2[nH]cnc(C(C)C)c2Cl)c2ccccc21)C(C(C=C)(C)O)=O 69062,c1(OCCC)c(F)cc(-c2nc(NC(=O)CNc3nccs3)cs2)cc1F 69063,N1(C(C(CC=CC)CC)=O)CC2CCCC2C1C(=O)NC1CC1O 69064,N1(C(=O)OC(C)(C)C)CCN2CCOCC2C1.Cc1cccnc1C1CN1.C 69065,C(=O)(C(=O)CC(C)CC)N(C(C(=O)NC1CC(=C)C1)C)C1CC1 69066,Cn1c(C(N2CCC(O)(CNC(=O)CC3CCCOC3)CC2)=O)cc2sccc12 69067,N1(C(=O)C=Cc2ncc[nH]2)CCC2OCCN(C(C3CCC(F)CC3)=O)C2C1 69068,c1(C(=O)NC2CCN(C(C(C)S)=O)C2)ccnc2ccc(Cl)cc12.C(=O)(C1CC1)N 69069,C(=O)(C(CC(C)C)C(N)=O)NC1CC2N(Cc3n(CCC)c(C)nn3)C(CC2)C1 69070,N(C1CCCc2occc21)C(c1n(CCOC)nnn1)c1ccsc1Cl 69071,c1(CCC)nc(C(=O)NC2(Cn3cc(C(C)(O)CCO)nn3)CC2)co1 69072,N1(C(C=CC(=O)N(C)C)=O)CC(CNC(c2ccc(Cl)s2)=O)C2(CCC2)C1 69073,Cc1nc(-c2cn(CC(C3CN(C(=O)CCc4nccs4)C3)F)nn2)sc1C 69074,C1(NC(c2n[nH]c(=N)s2)=O)CCCC2CN(C(C3CCCC(F)(F)CC3)=O)CC12 69075,O=C(N1CC(n2cc(C3CCCCO3)nn2)CO1)c1cncc(C2CC2)c1 69076,Cc1nc(O)ccc1C(N1CCC(C(=O)NCCc2c(C)n[nH]c2C)C1)=O 69077,c1(CC=C)ccccc1C(=O)NCCCCCNC(=O)C(COC)N(C)C 69078,C=CCC(CNC(c1nnn(CC)c1C)=O)C(=O)N(C(C)C(=O)OC)C1CC1 69079,C1(C(N(C(c2ccc(CC)s2)C(=O)NC(C)C)CCC)C)CCCCC1 69080,Cc1cc(C(=O)NC23CC(C2)N(C(c2cccnc2C(F)(F)F)=O)C3)cc(Cl)c1 69081,C1(NC(C2CCC(=O)O2)=O)CCCC(C(=O)Nn2cccn2)CC1 69082,C1(C(N2CC(NC(=O)C(C)(C)C)CC(C)(C)C2)=O)Cc2cc(Br)ccc2O1 69083,N1(C(CSC)=O)CC(NC(=O)CSc2cccc(Br)c2)CCC1C 69084,c1(CC)ccc(CN(C)C(c2c[nH]nc2CCNC(C2CC(C)(O)C2)=O)=O)cc1 69085,CC(C)(C)C(C(=O)N1CC(CCn2cc(CNC(N)=O)nn2)C1)NS(C)(=O)=O 69086,N1(C(c2c(C)ccnc2C)=O)CC2CCC(C1)C(NC(c1ccnnc1C)=O)C2 69087,N1(C(CCc2c(C)cccn2)=O)CC2(CCC2NC(C2CC2F)=O)C1 69088,CCC(CC)CCCC(=O)N1CC2CC(NC(=O)C=Cc3ncc(C)[nH]3)C(C2)C1 69089,C1(CC)CN(C)CCCN1C(=O)COC1(C)CN(C(=O)CC2CCCC3CC23)C1 69090,C1(C(=O)NCC2(O)CCSCC2)CCC(OC(F)(F)F)CC1 69091,C(C)(C)(CCCC(=O)NCCCC1CCCC1O)NC(c1c(C)cc(O)nc1)=O 69092,C(=O)(C(O)CC(C)C)NC(CCN(C(c1cc(OC)ns1)=O)C)C(C)C 69093,C1(NC(c2cnn(C(C)C)n2)=O)CC(C(=O)NCc2snnc2C)C12CCC2 69094,N1(Cc2ccc(OC)nn2)CC2CN(C(=O)Cc3cc(SC)cc(Cl)c3)CC12 69095,Cc1ccccc1C(C)C(=O)NCC(C)CN(C(=O)C(C1CCC1)C1CCC1)C 69096,Cc1cc(-n2cccn2)nc(=NCC2C(C)CCCN2C(=O)C(C)CN(C)C)[nH]1 69097,c1(C(N(CC(C)NC(=O)CCCC#N)C)=O)ccc(-n2cccn2)cc1 69098,c1(N2CC(C)=C(C)C2)ccc(S(=O)(=O)NCC2Cc3ccccc3CO2)cc1Cl 69099,c1(C(=O)NC(CC(C)NC(=O)CC2CCN(C)C2=O)C)cc(N)c(F)c(F)c1F 69100,c1(OCC)cc(OC)c(C(=O)NC2C=CC(C(=O)OC)C2)cc1N 69101,Cc1nc(-c2ccc(COc3ccccc3)cc2)ccc1C(=O)NC1COC1 69102,N1(C(c2cn(CC)nc2C2CC2)=O)CC(OC)CCC1C 69103,C(=O)(C(C)S(=O)(=O)C(C)C)NCC(C)(C1CCC1)NC(C1CCC(CC)O1)=O 69104,c1(C(=O)OC)c(Cl)nc[nH]c1=NCC(C)(C)NC(=O)C(C)Cc1ccccc1 69105,c1(C(=O)NC2C(C)CN(C(c3cc(Br)ccc3N)=O)C2)ccn2nnnc2c1 69106,C#CC(C(C)OC)NC(C1(C(C)NC(C2CC(CC)C2)=O)CC1)=O 69107,CC(CCC#N)(c1nnnn1CSc1ccccc1)NCCc1cccnc1 69108,Cc1nn(C(=O)N(C(C)CNC(=O)C(CO)c2ccccc2)C)cc1Cl 69109,C1(CNC(C#C)=O)CN(C(C2(C(=O)NCNC(N)=O)CC2)=O)CC1C(F)F 69110,c1(C(N2CC3CC(C2)N(C(c2cscc2Br)=O)C3)=O)ccc2nc(Br)sc2c1 69111,N1(C(C23OCC(C(C)C)(C2)C3)=O)CCC(C)(NC(=O)CCS(N)(=O)=O)CC1 69112,Cc1cc(C)c(C(N2CCCC2CCCNC(=O)CN(C)C)=O)[nH]1 69113,c1(C(=O)OCC(N2CCOCC2)C)ccn(C2CC2)n1 69114,C1(O)(CN(C)C(C2C(C)(C)C2(F)F)=O)CCN(C(C2(c3cc[nH]n3)CC2)=O)C1 69115,C(C)(C(CC(=O)NCCc1cc(C)no1)NC(c1cnsc1C)=O)OC 69116,C(N=c1[nH]c(NC2CCC2)nc2c1SCC2)C1(C)CCN(S(C(C)C#N)(=O)=O)C1 69117,N1(N2C(C)CCC(NC(c3cc4c(s3)CCOC4)=O)C2)CC2OCCN(C)C2C1 69118,N1(C(c2cc(C)sc2N)=O)CC2C=CC1C(C(N1CC(O)C(C3CC3)C1)=O)C2 69119,N1(C(C2(SC)CC2)=O)CCC(CC(C)NC(C2(CC(C)C)COC2)=O)CC1.C 69120,C(=O)(C(C(F)(F)F)C(F)(F)F)N1CC(N(C(C2CC2C(F)(F)F)=O)CCO)C1 69121,C1(Cn2cc(OS(=O)(=O)c3cc(C(F)F)cs3)nn2)CC12CCc1ccccc12 69122,C(C)(CCC(=O)NC(CNC(=O)C(C)(C)c1cnc[nH]1)CO)OC 69123,C1(C(=O)NCC(C)(C)NC(C(C(C)C)O)=O)CCC2CC2CC1 69124,N1(C(COc2cc(C)on2)=O)CCN(C)CC1CNC(C1CC(N(C)C)C1)=O 69125,n1(CC)nc2c(c1C(N1CCC(C(C)NC(=O)C(O)C(C)C)CC1)=O)CCCC2 69126,N1(C(C=CCC)=O)CCC(NC(=O)C=Cc2cc[nH]n2)C(C)C1 69127,CN1CC(F)CC1C(=O)NC(Cc1cc[nH]n1)C(=O)NC1(CCO)CCCCC1 69128,C1(C(N2CC(c3ccccc3)(NC(C(COC)C)=O)C2)=O)CCCS1(=O)=O 69129,C1(C)(C(N2CC(C)(CSC)C2)=O)CCN(C(=O)C(O)C(C)(C)C)CC1 69130,CC(C)C(C)(O)C(=O)NCC1CC(NC(c2coc(Br)c2)=O)CC1O 69131,C1(C(=O)NC)CCN(C(=O)NCCN(C)C(=O)OC)C1C(C)C 69132,C(=O)(C(C)(O)C(F)(F)F)NCC(C)NC(=O)C(O)CC1CCOCC1 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69168,c1(C(N2C3CCC(CNC(c4c(OC)n[nH]c4)=O)(C3)C2)=O)c(O)nnc(C)c1C 69169,C1(NC(C2CCCCCC2)=O)CC2CN(C(c3ccc(C4CC4)c(F)c3)=O)CC12 69170,C1(C)(NC(CCOC)=O)CC(NC(c2[nH]ncc2C(C)(C)C)=O)C1 69171,c1(C(N2CC(C)C(CNC(C3(C4(O)CCC4)CC3)=O)C2)=O)c[nH]c2ncccc12 69172,C(C(C)C(C)C(=O)NCC12COC(CNC(c3sccc3Cl)=O)(C1)C2)OC 69173,N1(C(c2n(CC)cc(Cl)c2)=O)CCC(CCNC(c2n[nH]c(C)n2)=O)C(F)(F)C1 69174,c1(CN(C)C)nn(C)cc1[N+](=O)[O-].c12nnc(n1CCn1cccn1)SC2C 69175,Cc1cc(C(=O)NCc2ncccc2C(=O)NCC(C)(O)C2(C)CC2)c(C)cn1 69176,N1(C(C(C)CC2CCCC2)=O)CCC(CC(N)=O)(NC(c2cnn[nH]2)=O)CC1 69177,c1(C(=O)NCC=CCNC(C2CCC2F)=O)ccc(-c2nc(=O)o[nH]2)cc1 69178,CC1(C#CC(=O)N2C(C(=O)NC3CCN4CCCC34)CC3CCCC23)COC1 69179,Cc1ncc(C(=O)NCC2CC2NC(C23CCC(CO2)C3)=O)c(C2CC2)n1 69180,CCCCCCC(=O)N(C(C)CCNC(=O)C(C)OCCN(C)C)C 69181,Cc1cncc(C(N2CCC(NC(C34CCCC3C4(F)F)=O)C(O)C2)=O)c1Cl 69182,C1(NC(=NCC=C)NCC(CC)(CC)SC)CCc2cc(OC)ccc2C1 69183,C1(C(=O)NC(c2ncc[nH]2)C)C2CN(C(=O)C(C)(F)F)CC12 69184,N1(C(c2cnc(COC)s2)=O)CCC(NC(=O)CC2CC(F)(F)C2)C2(CCC2)C1 69185,c1(NC(c2n(CCC(=O)OCC)nnn2)C2CCC2)ccc2nc(C)ccc2c1 69186,c1(C(C2(O)CC(NC(C=CC(C)(C)SC)=O)C2)=O)cc2n(n1)CCC2.C1C(C)N1 69187,c1(CC(=O)NCC=CCNC(C2N(CC)CC2)=O)cc(Cl)ccc1Cl 69188,C1(CC(=O)NC(CNC(C(C2CC(F)(F)C2)OC)=O)(C)C)CCC2(CCC2)CO1 69189,C1(OCC(=O)NC(C2CN(C(C3C(C)C3C)=O)C2)C)CCCCCC1 69190,c1(OC)ccc(CCCNC(=O)CCNC(N2CC(CCO)(OC)C2)=O)cc1 69191,n1(CC)nc(C2CC2)cc1C(=O)NCC12CC1CN(C(C1(O)CCSCC1)=O)C2 69192,N1(C(=O)Nc2ccc(C)cc2)CC2CCC2(C(=O)Nc2cc(F)nc(F)c2)C1 69193,c1(C(=O)NC(C2CN(C(=O)CCC3CCCO3)C2)C)nccc2ccsc12 69194,CC1(C)CCC(C(N2CC(NC(c3cnc(O)c(F)c3)=O)CC(F)C2)=O)CO1 69195,C1(C(=O)OC)CC1C(=O)N(CC(N)=O)C.C1=CCNC1=O 69196,C(C(CC(C)C)C(=O)N1CC(CNC(=O)C(C)(C)C(C)O)C(O)C1)OC 69197,C1(NC(C2C(C(C)C)(CC)C2)=O)CCCCC1NC(c1ccc(C(F)F)cc1)=O 69198,Cc1c(C(=O)NC2CC3CC(NC(C4(C)COC4)=O)C3C2)nn(C)c1Br 69199,C1(NC(CN(C)CC)=O)CCC(C)(CNC(c2ccnc(C3CC3)c2)=O)C1 69200,C(=O)(C1=CCSC1)N1C(C(=O)Nc2ccccc2)C=CC1.C12CCN1C2=O 69201,C(N=c1cc(C(=O)OCC)[nH]c(C(C)C)n1)C1CN(C(CC)=O)CC1C 69202,Cc1c(C(=O)NC2CC3(C2)CC3CC(=O)NC2CCC(C3CC3)C2)cncc1F 69203,c1(C(=O)NCCNC(c2cccc(CC)c2O)=O)ccc2cc(C)ccc2c1 69204,CC1CCN(C(=O)CCNC(C2CCCC2)=O)C1CNC(=O)C(F)OC(F)(F)F 69205,N1(C(C(=O)NCC2CC2)=O)CCC2(CCCCC2NC(=O)CCC2CCC2)C1 69206,N12CC3CCC1C(C3)NC(=O)C1CC(C1)C2=O.C1(C=O)CCCO1.CO 69207,C(=O)(CCC(C)CCCC)NC1CC(C(NOCCCC#C)=O)CC1O 69208,C1(CCOC)(NC(=O)COc2ccon2)CCN(C(=O)C(C)N=[N+]=[N-])C1 69209,N1(C(CC(C)(C)C)C(=O)NCc2cccs2)CCn2c(Br)cnc2C1 69210,c1(OC)cnc(SCc2c(C(N)=O)csc2)c(C)n1 69211,C(=O)(C1=C(CC)OCCC1)N1CC(C(N2C(CC(=O)OCC)CCC2)=O)NCC1 69212,C1(C(C)NC(=O)CC(F)(F)F)CCCN(C(=O)CCc2ncccn2)CC1 69213,N1(C(Cn2c(C)ccc2C)=O)CCN2CCN(C(=O)C(O)C(C)(C)C)CC2C1 69214,C1(CCNC(C2CSCN2C(c2ccccc2)=O)=O)CCCCO1 69215,Cc1nc2cc(NC(C3CCC(C)N3C(c3ccns3)=O)=O)cnc2[nH]1 69216,C1(NC(C2C(c3ccc(C)s3)C2)=O)C=CCN(C(c2cc[nH]c2C2CC2)=O)C1 69217,C1(CNC(CC(C(C)C)C)=O)CC2CCC1N(C(=O)CC1C=CCCC1)C2 69218,c1(CC(=O)NCC2N(C(c3ncc(OC)nc3)=O)CC=C2)cc(F)ccc1C 69219,c1(C(N2CC(C)C(CNC(C3CCC3(F)F)=O)C2)=O)cccc2c1CC(=O)N2C 69220,C=C(C)CCCC(=O)NCC(C)(C)OCC(=O)NCc1ccccc1F 69221,CCC(CC(=O)N(CCCC(=O)NCC1C=CCCC1)C)C(F)F 69222,C=C(C)CC(C)C(=O)NCC1CC(OC)CN1C(c1cc(F)cnc1Cl)=O 69223,C1(C(N(C)CCNC(c2cnc(Cl)cc2N)=O)=O)CCc2ncncc2C1 69224,C1(C(=O)NCCC(CNC(C(C)n2cccn2)=O)C)CC(=O)CCO1 69225,c1(OC)ccc(C(=O)NCCOCCNC(C2CC2CN(C)C)=O)c2[nH]ccc12 69226,c1(C(N2C(C)CC(CNC(c3n(CC)ccc3)=O)C2)=O)occ2c1CCC2 69227,CC(CC(C)(F)F)C(=O)NCC(O)Cn1ccnc1 69228,C(=O)(CC(C)(F)F)N1CCC(n2cc(CNC(CN(c3ncccn3)C)=O)nn2)C1 69229,CC(=O)CCCC(=O)NCCOCC(N1CCC(C2(C)N=N2)C1)=O 69230,c1(NC(CCN(S(CC)(=O)=O)C)C)cccc(C(=O)OC(C)(C)C)c1 69231,N1(C(Cc2cc(C)sc2C)=O)CCCC(N(C)C(C2CCCC(C#N)C2)=O)CC1 69232,C(C)(CCN=c1[nH]nc(-c2ccon2)s1)NC(Cc1cccc(CC)c1)=O 69233,N1(C(C(C)OCOC)=O)CC=CCC1C(N1CCN(C2(C)CC2)CC1)=O 69234,c1(N(CCC)C(=O)NCCCCc2ccccn2)ccc(C2CCC(=O)N2)cc1 69235,C(=O)(C(O)C(C)(C)C)N(CCN(C(c1sc(CCC)c(CC)c1)=O)C(C)C)C 69236,c1(CC(=O)NCC(CO)NC(CCc2ncc(C)[nH]2)=O)ccnc(Cl)c1F 69237,C1(OCC=C)CCN(C(=O)C(C2CCCO2)NC(c2nccn2C)=O)C1 69238,C1(NC(C(COCC)CC)=O)CCN(C(=O)CCCOC)CC1(C)C 69239,N1(C(C2C(C)(CC)C2)=O)CCOC2(C1)CN(C(C1(OC)CC1)=O)C2 69240,N1(CCNC(C2(C)C(C)C2)=O)CCC(NC(=O)CC2CCC2(F)F)CC1 69241,C(=O)(C1=NOC2(CCOC2)C1)NCC(CNC(CC1CC(NC(C)=O)C1)=O)OC 69242,C1(C(=O)NCC(c2ncccn2)C)CCC2(CC2)N1C(=O)CCC1CC1C 69243,C1(NC(C(C(CC)C)OC)=O)CCCC12CN(C(c1ccsc1SC)=O)C2 69244,CC(C)C(C)C(=O)N1CC2CC2(NC(c2cc(-c3ccccc3F)on2)=O)C1 69245,CCC(C)(C)C(C#N)C(=O)N1CCCCC(NC(c2cccc(CSC)c2)=O)C1 69246,C(=O)(C#CC1CCC1)NCC(C)CN(C)C(C1C2CCCC12)=O 69247,CC1CC2(CCN(C(C3CCN(S(=O)(=O)c4ccc(Cl)cc4)CC3)=O)C2)CO1 69248,n1(CC)nncc1CNC(=O)C(C)CNC(=O)CCCNC(C)=O 69249,c1(N2CCN(C(=O)NCCC(C)N(C)CC)CC2)ccc(C)c(F)c1 69250,C1(C(=O)NC(CC)CN(C(=O)CC2OCCC2(C)C)CC)CCC2(CCCC2)C1 69251,N1(Cc2cn(C=C)nc2)CCCCC(C)C1.c12cn(nn1)C(C)C(=O)N2 69252,C#CC1(OCC(=O)NCC(C)NC(=O)C(c2cnn(C)c2)=O)COC1 69253,C1(NC(=O)CCc2cccc(Cl)c2)CC2CCC(C1)N2C(C12COC(C1)C2)=O 69254,CCCCCC(O)CC(=O)NC(C)CCC(=O)NC1(CSC)CCC1 69255,c1(NC2CC(C#N)C2)ccc(S(=O)(=O)NCC(=C2CCCCC2)F)cc1F 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69273,c1(C(=O)NCc2cc(CN3CCCCC3)on2)nccc(=NCc2cnco2)[nH]1 69274,N1(C(C(C)(C)OCC)=O)CC2CCOCC2(NC(c2nc(C(C)C)oc2C)=O)C1 69275,c1(C(N2C(C(=O)NC(c3ccsc3)C)CC(O)C2)=O)cccc([N+](=O)[O-])c1 69276,C1(C2CC2)(C(=O)NC23CC(CNC(C(C)NC(=O)NC)=O)(C2)C3)CCC1 69277,C1(NC(C2(C)CCNC2)=O)CC2(C1)CN(C(c1cc(Br)ccc1OC(F)F)=O)C2 69278,c1(C(N2C3CC(CNC(CC(C)SC)=O)C2CC3)=O)coc2c(F)cc(Cl)cc12 69279,N1(C(C(CC)SC)=O)CCCC(C2CCN(C(=O)C(F)=CC3CC3)CC2)CC1 69280,CC(C)(CO)C(=O)NCCCN(C(=O)CCc1ccon1)CC1CCCC1 69281,N1(C(COCC)=O)CC=CC(NC(c2ccc(OCc3ccccn3)cc2)=O)C1 69282,O=C(CC(C(F)(F)F)c1ccon1)NC1(CO)CN(C(=O)C(F)OC(F)(F)F)C1 69283,C1(C(N2CCC(c3cc[nH]n3)C2)C(=O)NCC)CCC(C(F)(F)F)CC1 69284,C1(CNC(c2ccsn2)=O)CCC2(CCC2)C1NC(c1ncc(F)cn1)=O 69285,CCCCC(CNC(c1cc(-c2ccco2)cn1C)=O)NC(=O)CSCCC 69286,C=C(Cl)C(C)(C)C(=O)NCC1(CCNC(=O)CN2CCNC(=O)C2)CC1 69287,CC(C)S(=O)(=O)CC(=O)NC1CCN(C(c2cc(C#N)n(C)n2)=O)C1C 69288,N1(C(C)=O)CCN(C(c2[nH]ccc2CC2CCCCC2)=O)C(CS(C)(=O)=O)C1 69289,N1(c2ccnc(C(=O)OC)n2)CCC(CNC(=O)CC2CC=CC2)C(F)(F)CC1 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69307,C12(NC(c3cc(F)cc(F)c3)=O)CCCN(c3nccc(C(F)F)n3)CC1C2 69308,c1(-n2c(-c3scc(Cl)c3Cl)nc(CC(C)C)n2)cccc(C#N)c1 69309,C12(NC(c3c(C)ocn3)=O)CCC1CN(C(c1ccc(-n3cccc3)cc1O)=O)C2 69310,N1(C(CCOCC#C)=O)CC2CCC2(CC(=O)NC(C)Cc2ccccn2)C1 69311,C(C(C(=O)NCCN=[N+]=[N-])NC(C1CC1Cl)=O)N(C)C 69312,c1(CC(C=C)NC(=O)NCc2ncccc2C(N)=O)ccccc1F 69313,O=S(=O)(C1CCCCCC1)C1CCN(S(=O)(=O)c2cc(F)c(F)cc2F)CC1 69314,c1(C(=O)NC2(C)CCN(C(C=C3CCC(C)CC3)=O)C2)cc2cnn(C)c2s1 69315,C(N=c1[nH]c(=NCCOCCC2CC2)[nH]c2c1COC2)C1(CC)CCC1 69316,C1(CC(C)(C)C(=O)NCC2(c3cc(F)cc(Cl)c3)CC2)CC(=O)NC(=O)N1 69317,C1(OC)CN(C(=O)C=Cc2ncc[nH]2)CCC1NC(=O)Cc1ccsc1C 69318,C1(NC(CCNc2ccc(C)cc2)=O)CC12CCC(N)CC2 69319,Cn1c(O)nc(N2CC3(CCCC3NC(c3cnn4cccnc34)=O)C2)cc1=O 69320,C12(C(N(CCNC(=O)CC3CCCOC3)CC3CC3)=O)CC3CC1C2C3 69321,N1(C(C2(C(=O)OC)CC2C)=O)CCN(C(C2CCN(C(=O)C3CC3)CC2)=O)CC1 69322,N1(C(C(CSC)C)=O)CC2CCC(C1)N2C(c1cccc(C)c1NC(C)=O)=O 69323,C(=O)(CCCC(C)(C)CC)N(CC(C(=O)NCCC1CC(OC)C1)(C)C)C 69324,CCCCCCCNC(=O)C(CCN(C)C)NC(c1cc(C2CC2)on1)=O 69325,C12(NC(c3ncn(C)c3)=O)CN(C(=O)C3=CCS(=O)(=O)C3)CC1CS(=O)(=O)C2 69326,c1(C(N2C(CNC(c3c(C)nc(C(C)C)o3)=O)C(C)CC2)=O)ccc(O)cc1F 69327,N1(C(c2c(OC)n[nH]c2)=O)CCCC2CN(C(C34CC(C#N)(C3)C4)=O)CC12 69328,N1(C(C2OCC(C)C2)=O)CCC(NC(c2ccc([N+](=O)[O-])o2)=O)C12CCC2 69329,C1(C(N(C(C)(C)C)CCN)=O)C2CC(F)C(C2)N1C(C1C=CCN1)=O 69330,c1(C(N2CCCC(CNC(c3c(CC)cno3)=O)C2)=O)cnn2c1CCCC2C 69331,c1(C(N2CC(CNC(C(CC)C)=O)C2)=O)cc(F)cc(Br)c1 69332,Cc1nc(NC2CCC(CNC(c3c(C(F)(F)F)cccc3C)=O)C2)ncc1Br 69333,N1(C(=O)NCc2c(C)cno2)CCN(C2CCCC2)C(C)C1 69334,CCCC(C)CC(=O)NCc1ncccc1CNC(C12CCN(CC1)CC2)=O 69335,N(C(=NCCCOC1CCC1)NCC1(C)CCS(=O)(=O)CC1)C(C=C)C 69336,N1(C(C2N(CC)CCC2)=O)C2CCC1C(NC(c1cc(Cl)cc(Cl)c1)=O)C2 69337,C=CCCC(O)CN(C(=O)CCCN(C(=O)C(C)COC)C)C 69338,C=CCC(CC=C)C(=O)N(CC(=O)NC1COCC(C)(C)C1)C1CCC1 69339,N1(C(C2(CC)CCNC2=O)=O)CCCCCC(NC(c2c(C)coc2C)=O)C1 69340,c1(C(=O)NC(C)CCCNC(c2ccon2)=O)cc(C2CCCC2)n(C)n1 69341,N1(C(C2(C)COC2)=O)CCC(C)(CNC(=O)C=CCOCC(F)(F)F)C1 69342,C(=O)(C(F)(F)C(F)(F)C(F)F)N(C1CCN(C(C2CC23CCOCC3)=O)CC1)C 69343,C1(CNC(CCC(N)=O)=O)CCC2(CCC2)C1NC(=O)CC1=NNC(=O)C1 69344,Cc1cc(=NC(C)CNC(=O)Cc2ncncc2Cl)[nH]cn1 69345,O=C(C1=CCCN(C(=O)Cc2c[nH]c3ncccc23)C1)NCC1CCC1 69346,C1(C(=O)OC)C[Si]2(CCCC2)CN1C(CC1(C#N)CC1)C(=O)NCCC#N 69347,N1(C(CCSCCC)=O)CC(NC(C2CCCC(=O)C2)=O)C(C)C1 69348,CCCCC(C)CCC(=O)N(C(C)CNC(c1ccc(O)c(C)c1)=O)C 69349,C1(Cn2cc(-c3cn(C(CC)C)nc3)nn2)(OC)CCS(=O)(=O)C1 69350,C(=O)(CC1COc2cc(O)ccc21)NCCCC(C)NC(c1ccc(C)nc1)=O 69351,C(=O)(C(C(C)CC)NC(N)=O)N1CCC(O)(CNC(C=CCC)=O)C1 69352,N1(C(COCCCOC)=O)CCC(C)C(N(C(=O)C(F)=CC2CC2)C)C1 69353,c1(C(CC)C)ccc(NC(=O)CN2CCN(c3ncc(C)c(C)n3)CC2)cc1Cl 69354,CCCC(C(=O)OC)C(=O)N1CC(C)CC1C(=O)NCCCC(C)C 69355,Cc1ccc(-c2nc(C(c3cccnc3)C)no2)c([N+](=O)[O-])c1 69356,c1(-c2onc(C3(CC)CCC3)n2)cc2cc(Cl)ccc2[nH]1 69357,c1(NCC2CC(OC)C2)cc(=NC(C)c2ccn(C)n2)[nH]c(C(F)(F)F)n1 69358,Cc1cc(C(=O)NC2CC2NC(=O)C2=C(Cl)CCC2)cc(O)n1 69359,N1(C(c2c(C)onc2)=O)CCCC(C(C)NC(=O)CC2(c3ccon3)CCC2)C1 69360,CC1CCOC1C(C)(C)CNC(C1CC(Cl)(Cl)C1)c1nnnn1CCOCC1CC1 69361,c1(C(N2CC(CCC)N(C(c3cnnn3C)=O)CC2)=O)ccn2cccc2c1 69362,Cn1ccnc1SCC(N1CCC(OCCc2cccnc2)C1)=O 69363,C=C1CCN(C(C2CC(=O)CC(=O)N2)=O)C(C(=O)NCCCCCOC)C1 69364,C1(C(=O)NCC(CNC(=O)C(C2CCOCC2)C)CO)(CC)CCCC1 69365,CCCCC(CNC(C1CSCCN1C(=O)Cn1ccnc1)=O)CCC 69366,C(CC(C(=O)N(C)CC1CCOC1C)OC)NC(c1n(CC#C)cnn1)=O 69367,CC(F)(F)CCC(=O)N1C2CCC1C(CNC(c1ccnn1CC1CCC1)=O)C2 69368,N1(C(CCC2N(C(c3c(CC)cco3)=O)CCC2)=O)CCC(C)C2(CCC2)C1 69369,c1(CN(CCCCOC)CCC)csc(-c2cnn(C)c2)n1 69370,CC1CN(C(=O)CC(O)C2CCCC2)CCC1NC(c1cn(C)ccc1=O)=O 69371,C1(NC(c2sc(C)c(O)n2)=O)CCN(C(c2nc(C)ncc2Cl)=O)CC1CO 69372,c1(C(N(CCC(C(C)C)NC(C2C(C)C2(F)F)=O)C)=O)nc2n(c1Cl)CCCC2 69373,N1(C(CCC(=O)NC2(NC(=O)CO)C(C)C2)=O)CCC(F)(F)C(O)C1 69374,N1(C(CNC(=O)OC)=O)CC2CCC2(CC(=O)NC2CC(=C3CC3)C2)C1 69375,C1(O)(C2CN(C(CC(OCC)OCC)=O)C2)CCN(C(=O)C(C)C(=O)OCC)C1 69376,Cc1cc(C(N2C(C(N3CCC(F)(F)C3)=O)CC3CC23)=O)c(C)cc1Br 69377,C(=O)(C1CCCc2scnc21)N1C(C)(C)CC(NC(=O)CC2CCC=CCC2)C1 69378,C1(N(C(C(c2ccccc2Cl)C)=O)C)CCC(NC(=O)C(C)(C)C#N)CC1 69379,CC1CC(C(=O)Nc2c[nH]nc2Br)N(C(c2cncc(Br)c2)=O)C1 69380,c1(CC(N2C(C(=O)NC(C)CC#N)CC2)=O)ccccc1NC(=O)CC(F)(F)F 69381,N1(C(COc2cccc(CC)c2)=O)CCC2(NC(=O)C(C)(F)F)CC2C1 69382,c1(NC(c2cn(CC=C)nn2)=O)cccc(CNC(=O)CC2CC2C2CC2)c1 69383,C#CCC(C)(C(=O)NC1CN2CCC1CC2)NC(=O)CCC(=O)NC(C)C 69384,N1(C(C2CCC(OC(C)(C)C)CC2)=O)CC2CC1CCC2NC(c1cnsn1)=O 69385,N1(C(Cc2c(C)ocn2)=O)C2CCCC1CN(C(C1CCCOC1)=O)CC2 69386,N1(C(=O)NCCC2CCO2)CCN(N2CCC2)CC1 69387,c1(NCc2cc(C)ncc2)nc(C)nc(Br)c1F 69388,c1(C(=O)NC(CNC(c2c(C)ccnc2O)=O)C(C)(C)C)ccc2c(c1)OCC2 69389,N1(Cc2ccc(-c3c(-c4ccc(C)nc4)nccc3)o2)CCC2(CCCOC2)C1 69390,N1(C(c2c(OC)cc(Br)cn2)C(=O)Nc2ccccc2)CCCNC(=O)C1(C)C 69391,CC1Cc2cc(CCN=c3ccnc(N4CCC(C)(F)C4)[nH]3)ccc2O1 69392,C1(NC(C=CC)=O)CC2CN(C(c3[nH]nnc3COC)=O)CC12 69393,N(C(=NCCCC1CCC1)N1CC=C(c2cccs2)CC1)CCOC 69394,CCC(C(=O)NCCN(C1CCCC1)C(=O)COCC1CCCC1)SC 69395,C=CC1CN(C(C2CC(=O)CCO2)=O)CC1NC(C1CCCO1)=O 69396,CCC(CC(=O)NC1CCC12CN(C(=O)COc1ccc(C)c(C)c1)C2)C(F)F 69397,c1(CC)cnc(C(=O)NCC(C)CNC(c2n[nH]c(C(C)(C)C)n2)=O)nc1 69398,S(=O)(=O)(c1c[nH]c(C(=O)NC2CN(C(=O)CCc3cnn(C)n3)CC2F)c1)NC 69399,N1(C(CC=C)=O)CCCC(NC(c2nc(C)n(C3CC3)c2C)=O)C1C 69400,C(CCC(=O)N(C(=O)CC(C1(CC(C)O)CCCC1)C)C)=C(C)C.N(C)C 69401,S(=O)(=O)(c1cnc(NCC2CCC2(F)F)c(Cl)c1)NCC(C(CC)CC)O 69402,N1(C(C(C2CC2)OC)=O)CC(CNC(=O)CSc2ccccn2)C2(CC2)C1 69403,CC1CCCCC1CNC(=O)CC(c1cccc(Br)c1)C 69404,Cc1ccc(F)c(C(=O)NCc2cccc(CNC(c3cn(C)cn3)=O)c2)c1F 69405,C(=O)(C(CNC(C1(CO)COC1)=O)C(C)(C)C)N(CCC)CC 69406,CC1CCC(NC(=O)Cn2cnc(=N)[nH]2)CN1C(=O)CC1(CO)CC1 69407,N1(C(C2(NC(C)=O)CCC2)=O)CCN(C(c2cnc(C3CC3)o2)=O)C(C)C1 69408,CC1(C(=O)NCC2(O)CCN(C(=O)CCCn3cccc3)C2)CCCNS1(=O)=O 69409,N1(C(c2cn(CCC)nc2)=O)CCOC(CN(C(=O)Cn2[nH]cnc2=N)C)C1 69410,c1(C(=O)NC2(C)CCC(NC(C(C)(C)OC)=O)CC2)cc(C)c(F)cc1N 69411,c1(C(=O)NCC2N(C(C3CCN(C)C3)=O)CCOC2)cncc2c(F)cccc12 69412,c1(C(=O)NC2CN(C(C(CCC)(C)C)=O)CC(C)C2)n[nH]c2c(C)cccc12 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69449,C(=O)(CC(O)CNC(=O)C(C)(CO)NC(=O)C(n1ccc(C)n1)C)OC 69450,c1(SC)cccc(C(N2CCC(NC(c3occc3C)=O)C(F)C2)=O)c1[N+](=O)[O-] 69451,C1(CNC(C(C(CC)O)C)=O)CN(C(C2CC3(CCCC3)C2)=O)C2COCC2O1 69452,c1(C(N2CC3(CCN(C(C4ON=C(CC)C4)=O)C3)C2)=O)cccc2nc(O)oc12 69453,C1(CC#N)CN(Cc2ccc(Br)nc2Br)CCN1C(c1ccc(Cl)c(O)c1)=O 69454,N1(C(c2c(CC)[nH]cc2)=O)CCN(C(=O)C=Cc2nnn(C)n2)C(C2CCC2)C1 69455,N1(C(C2(CCOC)CCC2)=O)CCC(NC(=O)CC2CC(SC)C2)C(C)(C)C1 69456,c1(C(=O)OCc2cc(C(=O)NC)c(F)cc2)cnc(C)c(C#N)c1 69457,C1(CC)CN(C(=O)Cc2cccnc2)CCC1CNC(C1(S(C)(=O)=O)CCC1)=O 69458,c1(OC)ccc(OCCC(=O)NCCNC(C2COCC(C)O2)=O)cc1C 69459,N1(C(C2CCC(=O)C2)=O)CCCCCCC1C(N1CCCC1CNC=O)=O 69460,c1(C(=O)NCC(C)N(C)C(c2ccncc2Cl)=O)cccc2c1OCO2 69461,C(=O)(C(C)CCCO)CCO.CC(C)(C)CC(=O)N(CCCN)CCO 69462,C(=O)(C(C)C(C)S(C)(=O)=O)NC1CC(NC(c2c(OC)ccc(C)c2)=O)C(O)C1 69463,CCCCCC(C)CC(=O)N1CC(C(=O)NC(c2cnc[nH]2)C)CCC1(C)C 69464,c1(OC)ccc(C(C)C(=O)NCC2CCCCC2NC(c2cccs2)=O)cc1F 69465,Cc1ccc(NC(C2CCC(NC(=O)C(C)C#N)C2)=O)c(C)n1 69466,c1(C(N2C3CN(C(C4CC(C#N)(OC)C4)=O)CC32)=O)c(C)ccc2ncccc12 69467,N1(C(C(=O)N(C)Cc2ccc(Cl)nc2)=O)CCn2c(CC3CCCC3)nnc2C1 69468,C(c1ccc(C(N)=O)cc1)=CC(=O)NCC(C)N(C(C(C)C1CCC1)=O)C 69469,CCC(C)C(O)C(=O)NC1CCN(C(C2CN(CC)CCO2)=O)C1C 69470,C1(O)(CNC(C=C2CCC(C)C2)=O)CCCN(C(c2cc(Cl)c(Cl)[nH]2)=O)CC1 69471,c1(NC(CCN(C(CC(COC)C)=O)CCCO)=O)ccc(C)c(F)c1 69472,N1(CCC(C)C)CCC(C2(NC(=O)C(C)Oc3ccccc3F)CC2)CC1 69473,c1(OC)c(C(=O)NCC(C)CNC(=O)C(c2cccc(N)c2)O)ccnc1F 69474,C(CCCC(=O)NC12CC(C1)N(C(c1ccn(-c3ccccc3)n1)=O)C2)N(C)C 69475,C12(C(=O)NCCCCC(C)NC(=O)Cc3nncn3C)CCN(CC1)CC2 69476,c1(OCCC(N2CCC(C)(NC(C(CC)F)=O)C2)=O)c(C)cccc1C 69477,c1(C(C)=O)ccc(C(N2CC(N(C(=O)C3=CCCCC3)C)C3(CC3)C2)=O)c(O)n1 69478,N1(C(C(C)c2cc[nH]n2)=O)CC2CN(C(c3ccc(CCO)cc3)=O)CCC12 69479,C1(OC)CC(C(=O)NCC(C)C2CCC2)N(C(=O)COCC(C)C)C1 69480,Cc1ncc2c(n1)CCC(CNC(c1csnn1)C)C2 69481,Cc1oc(S(N)(=O)=O)cc1C(=O)NCC(C)N(C(=O)C(C)c1cncs1)C 69482,C=CCC(CNC(=O)CCCOC)C(=O)NC(c1c[nH]ccc1=O)C 69483,c1(OC)ccc(OC)c(C(=O)NCC2CCN2C(C2(OC)CCSCC2)=O)c1 69484,CCCCC(F)C(=O)N1CCC(C(=O)NCCn2cnnc2CC)CC1 69485,C1(C(=O)NC(COC)C(C)C)CCCCCN1C(c1nn(C)cc1C)=O 69486,c1(C(=O)NCC2CCN(CC(C)O)CC2)ccc(C2(F)COC2)cc1 69487,Cn1cccc(C(=O)NCCOC2CCN(C(=O)CCCC3CCCC3)C2)c1=O 69488,N1(C(C(CCC)N(C)C)=O)CCC(C2CN(C(C3(OC)CCOC3)=O)C2)CC1 69489,C1(NC(c2cncc(OCC)c2)=O)CCCC(NC(=O)CC2(C#N)CC2)CC1 69490,N1(C(c2ccc(C(C)=O)c(F)c2)=O)CC(CNC(=O)C2=CCCS2)N2CCC1C2 69491,C(CC(CNC(=O)CSCCC(C)C)NC(c1cnn(CC(F)(F)F)c1)=O)OC 69492,N1(C(C(CC(N)=O)O)=O)CCCC2CN(C(c3scc4c3CCCC4)=O)CCC12 69493,C12(NC(C=CCN(CC)CC)=O)CCC(CC1)N(C(=O)C(C)CC1CCCO1)C2 69494,CC1N(C(C2CN(C(=O)C(C3CCCCC3)F)CC23CC3)=O)CCC1(C)C 69495,c1(CC(=O)NCc2ccc(C(=O)OC)n2C)noc2ccc(O)cc12 69496,c1(C(=O)NCCC2C(C)CN(C(=O)CC3CNC(=O)O3)C2)cnc2n1CCC2 69497,C1(C(=O)NCCCC2CC2)CCCN1C(C1CC(C(F)F)C1)=O 69498,N1(C(CCN(C(=O)C(C)c2cccs2)CC=C)=O)CCCC(NC(C)=O)C1 69499,c1(C(=O)NCCN(C(C(CO)NC(C(C)C)=O)=O)C2CC2)c(C)cc(C)cc1C 69500,c1(C(N2C(CNC(c3cncc(C)c3)=O)CC(COC)C2)=O)cc(C#N)oc1C 69501,N1(C(c2ncc(C)c(Cl)c2)=O)CC2CCN(C(C3CCCC3)=O)CC12 69502,c1(C(N2C(CNC(CC(=O)NCC)=O)C=CC2)=O)cccc2[nH]nc(O)c12 69503,C(=O)(C1=NN2CCCN=C2N1)NC1C2N(C(C3CCN(C)C3)=O)CC(CC2)C1 69504,Cc1nc(C(=O)NC(C)CNC(=O)CCN2CCNC(=O)C2)cc(O)n1 69505,c1(CN=c2ccc(NC(c3c(F)ccnc3F)=O)c[nH]2)cccc2ncccc12 69506,CC1CN(C(=O)CC2CC3CC3C2)CC(C(=O)NCc2cc(C(F)F)no2)O1 69507,c1(C(N2C(C(=O)Nc3cnc(OC)c(F)c3)CCC2C)=O)[nH]nc2ccncc12 69508,Cc1ccc(S(=O)(=O)n2ccc(NC(=O)NC(CO)C(C)C)c2)cc1 69509,C(=O)(C1=NOC(C)(C)C1)N1CCCC(F)(C(=O)NCC(CCC)C)C1 69510,c1(C2(C(=O)NCC(C)CN(C)C(C3CC=CC(O)C3)=O)CCC2)cccc(F)c1 69511,C1(NC(CN(CC#C)C(C2(C)CCC(=O)C2)=O)=O)C2C3CCC(C3)C12 69512,C(=O)(N=c1cc2ccccn2[nH]1)C1CCN(C(C(C)CC2CCC2)=O)CC1(C)C 69513,N1(C(C2CCCN(Cc3ccc(CC)[nH]3)CC2)=O)CCC2(CCN(C)CC2)C1 69514,c1(C(N(C2CCC(NC(C3(CCCC)CCC3)=O)C2)C)=O)cccc(F)c1O 69515,S(=O)(=O)(c1cc(Cl)ccc1F)N1CCC(O)(C(=O)Nc2cc(F)c(Cl)cc2Br)C1 69516,CC(O)CC(C)(C)CNC(=O)CC1CCN(C(c2cc[nH]n2)=O)C1 69517,C1(OC)CCCC(CC(N2CC(F)CC2CNC(=O)CCSCC(N)=O)=O)C1 69518,c1(C(=O)NCC(CNC(c2cccc(C)c2)=O)C)ccc2nnc(C3CC3)n2c1 69519,c1(C(=O)NCCOCCNC(C2OCCN(CC)C2)=O)nccc(Cl)c1F 69520,C1(C(=O)NC2(C)CN(C(=O)CC3(C)CCOC3)C2)CCOC(=O)CC1 69521,C1(N(C(C(CSC)C)=O)CCO)CCN(C(c2cncc(C(C)(C)C)c2)=O)CC1 69522,C1(C(=O)NCC2(CNC(C=CC(C)(C)SC)=O)CCC2)C(F)(F)C12CCC2 69523,Cc1c(C(=O)NC2CC3CC(Nc4ncc(Cl)cn4)C2C3)nn2c1OCCC2 69524,C1(C)(NC(c2ccnc(C)n2)=O)CCN(C(c2cc(C(C)(C)C)ccn2)=O)CC1 69525,C(=O)(C(C)(C)C1=CCSCC1)NC(CCCC)CNC(c1cccnc1OC)=O 69526,CC(O)(CC(=O)N1CC=CC(NC(C2CC2Cc2ccccc2)=O)C1)C(F)(F)F 69527,N1(C(=O)NCc2nccnc2Cl)CC2CC(CF)C(C2)C1 69528,N1(C(c2c(C)c(C3CC3)on2)=O)CCC(O)(CNC(C2CC23CC(O)C3)=O)CC1 69529,C1(C(C)NC(=O)CCC2CCOC2)CCCN1C(c1n[nH]c(C2CC2)n1)=O 69530,CC(C)C(O)C(=O)N1CCCCC1C(N1CCCC1c1ccccc1)=O 69531,C1(CC)CCCCC1OCC(=O)NC12CC(C1)N(C(=O)CN(C)C(C)C)C2 69532,C1(C(=O)O)CC2CC(C1)N(Cc1ccccc1OCC(F)(F)F)C2 69533,C(=O)(C(=O)N=S(C)(C)=O)N1C(COC)CN(C(c2coc(C(F)F)c2)=O)CC1 69534,N1(C(c2nc(CC)oc2)=O)CC2(CC(CC(N3C(C(=O)OC)CC3C)=O)C2)C1 69535,CC1CN(C(=O)CC2CC3(CCC3)C2)CC(C)N(C(=O)CCCCN(C)C)C1 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69553,C(c1cn(C)nn1)=CC(=O)NC(COC)C(=O)N(C)Cc1cnn(C)c1 69554,CC1(C)CC(C)(CNC(c2cc3cccnn3c2)=O)CN1C(=O)C(F)C(F)(F)F 69555,CC1(C)CCC=C(C(=O)NC2CN(C(=O)CC3CCC=CCC3)CC2F)C1 69556,C(CN=c1nc(C(C)C)[nH]s1)C1(OC)CN(C(=O)CC2CCC(=O)N2)C1 69557,C1(CCNC(c2c(Cl)cn(CC)n2)=O)CCN(C(c2cc[n+]([O-])cc2)=O)C(C)C1 69558,N1(C(CCc2ncn(C)c2)=O)CCC(CNC(C2CC23CCC3)=O)C(O)C1 69559,C(=O)(N=c1cc(C)[nH][nH]1)c1nccc(NC(c2c(OC)cc(C(F)(F)F)cc2)=O)c1 69560,c1(C(CO)NC(C2CCCO2)=O)ccccc1C(F)(F)F 69561,c1(C(=O)NC2CCC(CCNC(=O)C(F)F)C2)cc(F)c2ccccc2c1 69562,c1(C(=O)NC(CC)CNC(c2cnc(O)s2)=O)cc(OC(F)F)ccc1C 69563,C1(NC(Cn2c(=N)nc[nH]2)=O)(CNC(=O)C=Cc2cccnc2)CCOCC1 69564,C(=O)(C(=O)C(C)CC)NC(C(=O)N1C(COCC#C)CCC1)CC=C 69565,N1(CC)CCC2CN(C(C3CC3C)=O)CCC12 69566,C1(C(=O)NC(C)(CNC(C2CCC(C(F)(F)F)CC2)=O)CO)COC2(CCC2)C1 69567,c1(C(=O)NCC(C2CC=CCN2)=O)c(F)cc(Cl)cc1Cl 69568,C1(NC(C2C(C(C)(C)C)C2)=O)CCC2CC1CN2C(C1CC2(C1)CC2F)=O 69569,c1(N2CCC(C)(CC)C2)ncccc1S(=O)(=O)N1CCC(CN(C)C)CC1 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69798,Cc1cc(NC2CCCCN(C(c3ccnc4c3CCC4)=O)C2)ncc1[N+](=O)[O-] 69799,n1(CC(=O)NC2CC(NC(c3ccc(Br)o3)=O)C2)cc(C(F)(F)F)nn1 69800,C(C(C)C)(C(O)C(=O)NC(C(N1CC(C2(C)CC2)C1)=O)C1CCOC1)OC 69801,c1(C(C(=O)N(C(CNC(C2CC(F)CN2C)=O)C2CC2)C)(C)C)ccc(Cl)nc1 69802,CC(CC(=O)N1CC(OCC(=O)NC(CC2CCCC2)CO)C1)C1CCCC1 69803,c1(OC)cccc(=NC(=O)Cc2cccc(CN=c3[nH]c(C)cn3C)c2)[nH]1 69804,N1(C(c2ccc(OC)cc2)=O)CC(NC(=O)CN2CCNC(=O)C2)CC(C)C1 69805,Cn1nnc2c(N3CC(C(N)=O)(CNC(=O)Cn4ncc5cccnc45)C3)ncnc12 69806,C(C(CC(C)C)C(=O)NC1CC(O)CC1O)NC(Cc1c(C)noc1C)=O 69807,Cc1n[nH]c(C)c1CCC(=O)NC1(C)CC(NC(=O)C(C2CCCCC2)C2CC2)C1 69808,C1(NC(CNC(=O)NC)=O)CN(C(c2ccc(C(C)C)c(F)c2)=O)C(C)(C)C1 69809,c1(C(C(=O)NC(COC)CNC(=O)CCOCC(C)C)O)ccc(F)c(Cl)c1 69810,N1(C(c2c(SC)cn(C)n2)=O)CCN(C(=O)CC2(O)CCCC2)CC12CC2 69811,C=CCCCC(C1CC1)NC(=O)C(C)C(C)NC(=O)C=CC(=O)OCC 69812,c1(C(=O)NC2CCN(C(C(CCC)C)=O)CC2)sc2ccccc2c1Cl 69813,C1(NC(C(CC(=C)C)C)=O)CN(C(=O)Cc2csc3nccn23)CC2CCCC12 69814,c1(CSCC)ccc(C(=O)N(C2CC(SC)C2)C)cc1.c12cncc(c1)C(=O)N2 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69833,CCCC(C)(CC)C(=O)N(C)CC1CC(F)CN1C(=O)C(C)=CC1CC1 69834,c1(OC)cc(C(N2CCN(C(=O)COC3CC(F)(F)C3)C(CO)C2)=O)cc(F)c1 69835,C1(CC(C(=O)N(CC(C)O)CCCO)NC(=O)OC(C)(C)C)COCCOC1 69836,CC1=C(C(=O)NC(C(=O)NCCOc2ccccn2)c2cccs2)CCO1 69837,C1(N(C(C2COC(C)C2)=O)CC)CCCN(C(=O)Cc2csc(Cl)c2)CC1 69838,C12(NC(Cc3cc(C)n(C)n3)=O)CCC1CN(C(=O)C(C1CCC1)C1CCC1)C2 69839,CCC(CC)(CC)C(=O)NCCC1CC(NC(c2ccc(C#N)c(Cl)c2)=O)C1 69840,Cc1cc2[nH]c(=O)c(C(=O)NC(C)CN(C)C(C3CCCC(C)CC3)=O)cn2n1 69841,C1(NC(C=CC)=O)CN(C(C2CCN(C(=O)NC(C)(C)C)C2)=O)CC2CCCC12 69842,CC(C(=O)N(C)Cc1ccc(CNC(C2CC2C(N)=O)=O)cc1)C(F)F 69843,N1(C(c2ccc(CNC(C)=O)o2)=O)CCC2CN(C(=O)Cc3cnsc3)CC12 69844,c1(C(CC)C)ccc(C(=O)NCC2(C)CCC(NC(=O)CO)C2)c(O)n1 69845,c1(OC)cccc2c1CCN2c1cc(NCC2C3Cc4ccccc4C23)ncn1 69846,N1(C(C(C)OCC#C)=O)CC(NC(=O)CCNC(c2ccoc2)=O)CC(O)C1 69847,Cc1nc(C(=O)NC(C)C(C)(C)NC(=O)CCCN(C)C)cn1C(F)F 69848,C=C=CCCC(=O)NC1CCC(C)(CNC(=O)CCN(CCCCC)C(C)C)C1 69849,C#CCC(O)C(=O)N(C1C=CCN(C(=O)CC(F)(F)F)C1)Cc1ccccc1 69850,c1(C(=O)NC2C(NC(c3n(CC)ccn3)=O)CCOC2)c[nH]c2ccc(F)cc12 69851,N1(C(=O)Cc2cc(C(F)(F)F)ccn2)CC2(CO)CCCC2(CO)C1 69852,N1(C(c2c(C)scn2)=O)CC(=O)NCC1C(=O)NCCc1nccs1 69853,CC(N=c1[nH]nc(C2CC2)s1)C1CCN(C(c2ncnc3sccc23)=O)CC1 69854,C(CC(C)(C)C)(C(=O)NCC1CCC1)NC(CC(C=C)CC)=O 69855,c1(CNC(C2CC(=O)OC2)=O)ccc2c(c1)CCC2NC(=O)C=CC=C(Cl)Cl 69856,C(=O)(C1CCCc2cccnc21)NC1CCCN(C(c2ccc(C)o2)=O)CC1 69857,C(=O)(CS(=O)(=O)CCO)NC(C)CCCNC(C1CCCOC1C)=O 69858,c1(C(CNC(C)(C)Cc2ccccc2)F)cccc(Cl)c1F 69859,N1(CCNC(Cc2cn(CC)nc2)=O)CCN(C(C2(COC)CCCO2)=O)CC1 69860,c1(C(N2CC(CNC(CC=CC)=O)C3(C2)CC3)=O)cc(F)c(Cl)cc1Cl 69861,N#Cc1ccnc(C(=O)NCC2CC(NC(c3ccc(CO)o3)=O)C2)c1 69862,C1(CC(=O)NCCCN(C(C2CC2C(C)(F)F)=O)CC)CC2CCC1O2 69863,C(CC(C)CCNC(C1CCC(n2cc(C3(O)CCCC3)nn2)C1)=O)NC(C)=O 69864,Cc1c(C(=O)OC)oc2ccc(F)cc12.c1(CC(=O)NS(C)(=O)=O)cscn1 69865,C1(C(N2CC3(CC(=C)C3)C2)=O)CCN(C(=O)C=CC2CCC2)CC1(C)C 69866,C12CCC(CC1)CCOC2=O.C1(COC)CN(C(=O)OC(C)(C)C)CC1C 69867,C1(CC(=O)NC2CN(C(C3(CC#C)CCCCC3)=O)CC2O)CC2(CCC2)CO1 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69939,C=CCC(CC=C)C(=O)N1C2CCC1C(CNC(=O)CSCc1ccccn1)C2 69940,CCC(C(=O)NC(C)CCC(=O)NCCN(C1CCC1)CC)C(F)(F)F 69941,C1(CCC(=O)NC(C2CC(NC(=O)CC(C)N(C)C)C2)C)CCOCC1 69942,CC(C(=O)NC(CC1CCC1)C(=O)NCCc1cnco1)C(F)(F)F 69943,c1(CNC(C(C)c2ccco2)=O)ccnc(C(=O)NCCN2CCCCC2C)c1 69944,N1(CC(=O)Nc2c(NC(C)=O)c(Cl)ccc2)CCC2(C=Cc3ccccc3O2)C1 69945,c1(NCc2nccc(C(F)(F)F)c2)nnc2ccc(Br)cn12 69946,N1(CCn2c(=O)cc(CCOC=C)n2C)CCC2(CCC(O)C2)C1.C(=O)OC 69947,N(C1CCOc2ccccc21)(CC(N)=O)CC(C1CC1(F)F)=O 69948,n1(CCNC(C2(c3ccncc3)CC2)=O)cc(CCCCCC2CC2)nn1 69949,N(C1CCCc2cnccc21)C(=O)NC12CCOC1CCOC2 69950,c1(C(N2C(CN(C(=O)CC(C)(C)C)C)CCCC2)=O)nnn2c1CCC2 69951,C(=O)(CC(C(F)(F)F)P(C)(C)=O)NC(C)CNC(=O)C#CC1(C)CC1 69952,c1(CNC(c2c(C(=O)NOCC3CCCC3)con2)=O)cncc(Cl)c1 69953,CCC(C)(CNC(c1csc(C#N)c1)=O)C(=O)NC1CCN(C2CC2)C1 69954,c1(CN2C(C(CC)C)CCCC2)csc([N+](=O)[O-])c1 69955,c1(C(=O)NCCCN(C(C(n2ccc(C)n2)C)=O)C2CC2)cccc(C)c1C 69956,N1(CC)CCOCC1C(=O)NC(C(=O)N(C)CCC1CN(C)C1)C1CCCO1 69957,C(=O)(C(O)CC(F)(F)F)NC1C(NC(=O)CCCn2cncn2)CCOC1 69958,N1(C(C(CC=C)(C)C)=O)CCC2(CC1)CC(CNC(C1CC(C)CC(C)C1)=O)C2 69959,CCS(=O)(=O)c1cnc(O)c(C(=O)NC2C3CN(C(=O)C(F)=C4CCC4)CC23)c1 69960,C(=O)(C#CC(=O)NCCCN(CCCCNC(=O)CC=C(C)C)C)OCC 69961,C(C(=O)NC1CCCCC1C(=O)NC1(CO)CCCC1)(C(C)C)OCC.NCC 69962,N1(C(C2C(C)CC(C)O2)=O)CCCC(N(C(=O)CC2CC(=O)C2)C)CC1 69963,N1(C(C(CCCC)F)=O)CCC2CN(C(C3CC3C(F)(F)F)=O)CC2CC1 69964,Cn1nccc1CC(=O)NC1(CNC(=O)CCOCC(F)(F)F)CCOC1 69965,C(C)(C)(CC(F)C(=O)N1CC=C(CO)CC1)NC(C(C)CO)=O 69966,c1(OC)ccccc1C(C)CC(=O)N(C1CC(NC(=O)Cc2c[nH]nc2C)C1)C 69967,c1(C(N(C2CC(NC(C3C(C)C3C)=O)C2)C)=O)cccc2c1nnn2C 69968,CC1CN(C(=O)CCc2nc(O)n[nH]2)CCC1NC(C12CC(CO1)C2)=O 69969,c1(C(=O)NC2C(CNC(C(=Cc3cccnc3)C)=O)C2)ccc(S(N)(=O)=O)cn1 69970,Cc1cc(=NC(C)CCNC(=O)C#CC2(C)CCCO2)[nH]c(C)c1C#N 69971,CCCCCC(C(C)(C)C)NC(c1ccc(S(=O)(=O)NCCO)cc1)=O 69972,N1(C(C(CCSC)OC)=O)CCCC2(C1)CN(C(=O)CC1(N3CCCC3)CC1)C2 69973,c1(C(N2CCCC(CNC(CN(C(C)C)C)=O)C2)=O)coc(S(=O)(=O)N(C)C)c1 69974,c1(N(CCNC(CCCS(N)(=O)=O)=O)CC2CC2)cc2nn[nH]c2cc1[N+](=O)[O-] 69975,C(=O)(C(C)(O)CC(F)F)N(CCCNC(c1ccc(CN(C)C)o1)=O)C1CC1 69976,c1(CC(=O)NC(CNC(C2CC(F)C2)=O)CO)coc(-c2ccccc2)n1 69977,O=C1Cc2cccc(NC(C34CC3CN(Cc3c(F)cc(I)cc3F)C4)=O)c2N1 69978,C(=O)(N(CCC(=O)N1CCC(C(F)(F)F)C1)OC)C1(CC#C)CCCN1 69979,N1(C(C2(OCC)CCC2)=O)C2CCC1C(CNC(=O)Cc1cccnc1Cl)C2 69980,N1(C(C(CN(C)C)O)=O)CCC(C(=O)NCC(C)(O)C2(C)CC2)(CO)C1 69981,c1(C(=O)NCC(C2CCCC2)NC(c2csnn2)=O)cccc2c1OCCO2 69982,c1(-c2scc(C)n2)ncc2cc(C)ccn12 69983,c1(C(N2C(CN(C)C(C3CCCOCC3)=O)COCC2)=O)cnn2ccncc12 69984,CCC(C(=O)NC(CNC(c1nccnc1OC)=O)C1CC1)C(C)C 69985,c1(C(=O)NCCN(C(C2(CC=C)CCC2)=O)CC)cnn(C=C)c1N 69986,C(=O)(C1=CCN(C(c2coc(C)c2)=O)CC1)N(C1COCC1O)CC 69987,C1(O)(CCNC(c2cc(C(C)=O)sc2)=O)CCN(C(=O)C(C)(C)C(F)F)CC1 69988,N1(C(C2(C(N(C(C)C)C)=O)CC2)=O)CC2CC(C1)N(C(C1CC13CC3)=O)C2 69989,N1(S(CCC)(=O)=O)CCc2c(C(=O)N=c3[nH][nH]cc3-c3ccccc3)n[nH]c2C1 69990,C(CC(C)C(=O)N1CCC(O)(CNC(c2nn(C)cc2SC)=O)C1)=CC 69991,N#Cc1cccc(NC(=O)C(=O)NC(C2CCOC2)CO)n1 69992,C(=O)(C(C)CC(C)(F)F)NCCCCCN(C(C1CC=C(C)CC1)=O)C 69993,C1(C(C(=O)CCn2cc(C)cn2)=O)CNc2ccccc2C1C.CO 69994,Cc1ccc(C(N2CCC(CCNC(C34CCCC3OCC4)=O)C2)=O)c(F)c1F 69995,c1(C(=O)NCCN(C(=O)CCN2CCC(F)C2)C)ccccc1F 69996,C(=O)(C=CS(F)(F)(F)(F)F)N(C1CCN(C(C2SCCCS2)=O)CC1)C 69997,c1(C(N2C(C(=O)NC(CC(=O)NC)(C)C)CC2)=O)cc(C)nc(O)c1 69998,c1(SCC)cccc(CC(=O)NC(C)(C)CNC(C2CC2C(F)(F)F)=O)c1 69999,c1(OC)nc(C2=CCNCC2)ccc1C(=O)Nc1cnn(CC(F)F)c1 70000,N1(C(=O)NC2(C(=O)O)C(C)C2)CCN2CCN(CC3CCC(=O)N3C)CC2C1 70001,C1(CNC(CS(C(C)C)(=O)=O)=O)CCC2CN(C(C3CC4CC4C3)=O)CCC2C1 70002,N1(C(c2cnc(SC)s2)=O)CC2CN(C(C3(N(C)C)CC3)=O)CC(F)(F)C2C1 70003,C1(NC(c2c(CC)nco2)=O)CCN(C(c2c[nH]nc2-c2cccs2)=O)CC1F 70004,c1(-c2cnc(SCC3CC3)nc2)nc(C2Cc3ccccc32)no1 70005,C1(CC(=O)NC2CC(C(C)O)C2)CC(C)(C)CN1C(=O)Cc1cccc(F)c1 70006,c1(C(N2CCC(C)C(N(C)C(c3ccnnc3O)=O)C2)=O)cc(C#N)ccc1F 70007,Cc1nnc(O)c(C(=O)NC2CC2CNC(=O)C(C)Cn2ccnc2)c1C 70008,N1(C(C(N2CCCC(C)C2)=O)=O)CCC(NC(C2CCCOCC2)=O)C1(C)C 70009,c1(SCCC(=O)NCC(C(C)(C)C)NC(C2C(C)C2)=O)ccc(Cl)cc1F 70010,c1(C(=O)OCC)cc(Br)c(F)cc1NC(C1CCN1Cc1cc(F)cc(Br)c1F)=O 70011,c1(C(=O)OC)cc(=NC(=O)C2(NC(C3CCCCC3F)=O)CCC2)[nH]n1C 70012,C1(C(=O)NCCCN(C(=O)C#CC2(C(F)(F)F)CC2)C(C)C)Cc2nncn2C1 70013,C12(CNC(C(CN(C(C3N(CCC)CCC3)=O)C)C)=O)CCN(CC1)C2 70014,c1(CC(N2CCC(N(C)C)CC2)=O)c[nH]c2cccc(F)c12.C12CCN1C2=O 70015,c1(C(N2CCC(NC(C(C)SC)=O)C(C)C2)=O)cccc2c1NCC2 70016,C(=O)(C(C(C)CC1CCOCC1)N(C)CC1CCCN(C)C1)NCC=C 70017,C(=O)(C1=CC2(CCOCC2)C1)N1CC(C)(NC(=O)C2=CS(=O)CCC2)C1 70018,c1(OC(C(=O)Nc2cn(CC)nc2)=O)ccc(C)c(OC)c1.C1(N)CCS(=O)(=O)C1 70019,N1(C(c2nc(CC)[nH]n2)=O)CC(NC(=O)CC(C)(F)F)CC1C 70020,C1(C(N2CCC3CN(C(C4(CF)CC4(F)F)=O)CC23)=O)CCC(=C(F)F)CC1 70021,N1(C(C2=C(C)CC2)=O)CC2(C(N3CCOC(CCO)C3)=O)CC1CO2 70022,C1(C(=O)NC(CNC(c2cc(OCC)ncc2)=O)(C)C2CC2)CC2(C1)CC(F)C2 70023,C1(CC)CN(C(C2CCCS2)=O)CCN1NC(c1cc(CC)n(CCO)n1)=O 70024,C1(C(N(C(C)C)Cc2cc(C)no2)=O)C2CN(C(=O)C(F)CC3CCOC3)CC12 70025,C1(CNC(c2c(OC)csc2)=O)CN(C(C2CCN(C3CC3)CC2)=O)CCN1C 70026,CC1CCN(C(=O)C(=O)NC(C)(C)C(C)NC(=O)CCCc2ccncc2)CC1 70027,C1(CC(=O)N(CCNC(C(C(C)C)OCC)=O)CCOC)CCCC2(CCC2)O1 70028,C12CCC(C1)NC2=O.c1(CC)ccsc1C(F)(F)F.C12(CC1)C(=O)NC2 70029,C1(C(=O)NCC(CC)O)C(CNC(c2ccoc2Cl)=O)C1(C)C 70030,c1(C(=O)NC2CC(C)(NC(CC(C)CF)=O)C2)nc[nH]c2ncnc1-2 70031,c1(CNC(C(=O)OC)Cc2ccc(C(F)(F)F)cc2)c(C)nn(C)c1C 70032,CC(N=c1[nH]c2c(c(=NCCOC3CCC3)[nH]1)CCCCC2)c1ccc(Br)cn1 70033,C1(N(C(C=CCCC)=O)C2CC2)CN(C(c2csnc2C)=O)CCC1C(F)(F)F 70034,c1(NS(=O)(=O)Cc2ccccc2I)ccccc1N1CCCCC1 70035,C=CC(C)(O)C(=O)NCC1(C(=O)NC(C)Cc2cccs2)CC1 70036,C1(NC(c2cccc(C3CCC3)c2)=O)C2CCN(C(C3CC=CCC3)=O)C12 70037,N1(C(C(C)OC)=O)CCN(C(c2ccc(-c3ccc(Cl)c(F)c3)o2)=O)C(CF)C1 70038,Cc1cc([N+](=O)[O-])c(C)c(S(=O)(=O)NC2Cc3ccc(F)cc3C2)c1 70039,Cc1cc(C)c(C(=O)NCc2cc(C(=O)Nc3ccccc3)no2)s1 70040,c1(C(=O)NC2C(NC(c3c(OC)c(F)ncc3)=O)CC2)c(C)ccc(C)c1C 70041,c1(C(=O)NC2CC(NC(=O)CCc3cccnc3Cl)C2)cccc2scnc12 70042,C1(NC(COC2(C)CCC2)=O)CC2CC(NC(=O)CSc3n[nH]c(=N)s3)C2C1 70043,C(=O)(CC(F)(F)F)N(C1CCN(C(C(Cn2ccc(C)n2)C)=O)C1)CCO 70044,C1(C(=O)NCC(C2CCCC2)NC(=O)C(F)C(F)(F)F)CNc2ccnn2C1 70045,C1(C(=O)NCCN(C(=O)C(=O)Nc2ccccc2)CC)COCCN1C 70046,CCCC(CC(=O)NCCN1CCCCC1)NC(C1CC(SC)C1)=O 70047,C(CC(=O)NC1CSC1)(C(F)F)NC(=O)C=Cc1ccccc1 70048,C1(C)(C(N(CCC)C2CC2)=O)CC12CCN(C(C)Cc1cccc(Br)c1)CC2 70049,C1(C(=O)NCC2CC(=C)C2)CC2(CCC2)CN1C(=O)Cc1ncccc1F 70050,N1(C(COC(C)(C)C)=O)CCC2CN(C(=O)C=Cc3cccs3)CC2C1 70051,CCCCCCC(C)(CC)C(=O)NC1CCC(NC(=O)CCc2nncs2)C1 70052,c1(C(=O)NC2(CNC(c3c[nH]c(=O)cn3)=O)CCOC2)cc(Cl)c(Br)[nH]1 70053,N1(C(C(=O)NC(CC)C)CC2C=CCC2)Cc2ccc(Br)cc2CC1C 70054,C(C(=O)N1OC2CCC1C2)C1CCN(C(C(N=S(C)(C)=O)=O)=O)C1 70055,C1(C2CC2)(NC(CNS(C)(=O)=O)=O)CCN(C(=O)C(C)(C)C(=O)OC(C)(C)C)C1 70056,c1(CC(=O)NCC2(OC)CN(C(=O)C=C(C)C(C)C)C2)c(O)nc(=N)[nH]c1C 70057,C1(CN(C)C(c2ccc(F)cc2)=O)CCCCN1C(c1ccnc(S)c1)=O 70058,c1(CNC(c2c(C)ncnc2)=O)nc(CNC(=O)CN2CCOCC2)cc(O)n1 70059,C(=O)(C1=C(C#N)CCC1)NC1C2C(C(=O)NC(C)CS(C)(=O)=O)C3C(C2)C13 70060,CCS(=O)(=O)CC(=O)NCC1(C(=O)NCC(C)(CO)CO)CC12CCC2 70061,CCCC(F)C(=O)NC(Cc1ccco1)C(=O)N(C(C)C(=O)N(C)C)C 70062,C(=O)(C1=CCC(F)(F)CC1)NC(CNC(C(CC)(F)F)=O)C1CC1 70063,C(CCN(C(=O)CC1CC=CCN1C)C)(C(C)(C)C)NC(C1CC(OCC)C1)=O 70064,C1(O)(CNC(C(C)N(C(C2(CCC=C)CC2)=O)C)=O)CCCCCC1 70065,N1(C(c2cn(CC=C)nc2)=O)CCCN(C(c2cnc(O)cc2C)=O)C(CO)C1 70066,N1(C(c2ccno2)=O)CC(C2CCCN(C(C3CC3F)=O)C2)C1 70067,N1(C(=O)CN(C2CCC2)C)CCCC(C)(C#N)C1.CC1=CC(=O)NC1 70068,CC1C(NC(CCC2CC3(C2)CC3(F)F)=O)CCCN1C(c1cccnc1N)=O 70069,C1(C)(NC(Cc2c(CC)con2)=O)CCCN(C(c2nc(CSC)oc2C)=O)C1 70070,c1(-c2cc(Nc3ncc(OC)cn3)ncc2)ccc(S(C)(=O)=O)cc1C 70071,C1(NC(C(Cn2ccc(C)n2)C)=O)CN(C(c2c[nH]nc2C)=O)CCC1F 70072,C1(C2N(C(C=C(C)C(C)C)=O)CCC2)CCN(C(=O)C(c2ccncc2)C)CC1 70073,c1(COC)cc(C(N2CCOCC2CNC(C2CC2c2cccs2)=O)=O)n(C)c1 70074,C12(NC(C3=NOC(C)C3)=O)CCCC1(F)CN(C(c1ccncc1Cl)=O)C2 70075,N1(C(c2c(CCC)occ2)=O)CCC(C)C1CNC(C1(CF)CC1)=O 70076,C(CC(CNC(c1ccn(C2CC2(F)F)n1)=O)NC(=O)CN1CCCC1)OC 70077,c1(OC)cc(F)c(C(=O)NC2CC(F)(CNC(=O)CC3COCCO3)C2)c(F)c1 70078,N1(C(C(C2CC2)SC)=O)CCC(C(=O)N(C(C)C(F)F)C)(CF)C1 70079,c1(C(N2CCCC(N(C(COCC=C)=O)C)C2)=O)cc(=O)n(C)cn1 70080,C(CCCC(=O)c1n(COC)ncc1)N1CCC(CC(C)(C)C)C1 70081,N1(C(C(C)Oc2ccc(C)cc2)=O)CCC2CCC(C1)N2C(C1CCCCO1)=O 70082,C1(NC(C(N2CCOCC2)C)=O)CCN(c2ccnc(Cl)n2)CC1C 70083,N1(C(COCCSC)=O)CCC(C(C)(C)NC(=O)C(O)CSC)CC1 70084,c1(C(=O)NC2(C)CCN(C(=O)CC3CCCO3)C2)cc(S(N)(=O)=O)ccn1 70085,S(=O)(=O)(c1c(F)cc(F)cc1F)N1CC2CN(C(c3cc(Cl)c(Cl)s3)=O)C2C1 70086,N1(C(CC2COCC(C)O2)=O)CCC=C(C(=O)NCCCc2cc[nH]n2)C1 70087,CC1CC(C(=O)NCCn2cncn2)CN(C(=O)Cc2ccon2)C1 70088,N1N(Cc2cn(-c3ccc(OC)cc3)nn2)CCOC2(CCOC2)C1 70089,C(CCN=C(NCCc1cccc(Br)c1)NC1CCCC1)c1c(C)cccc1 70090,c1(CC)sc(OC(C)=O)c(Br)c1C.c12cc(no1)-c1cn(nn1)C1CC(C1)NC2=O 70091,C12(C(=O)NCCOC3CCOC3)COCC1CN(C(=O)Cc1cnoc1)C2 70092,C1(NC(c2cc(CNC(c3cc(C)n(C)c3C)=O)oc2)=O)CC2CC1CC21CC1 70093,C1(CNC(COCCOC)=O)CCCCCN1C(=O)C(C1CC(C)(C)C1)OC 70094,Cc1nccc(C(=O)NC2CC(C(=O)NCC(C)(C)OC(C)C)C23CCC3)c1C 70095,CC(CS(N)(=O)=O)NC(C1(CNC(c2cnncc2O)=O)CC2(CC2)C1)=O 70096,C(C(CC1CC1)C(=O)N1CC2CC2(CO)C1)NC(C1CC(=C2CC2)C1)=O 70097,NC(=O)CC(O)C(=O)NC(CNC(=O)CCc1cc(Br)ccc1F)CO 70098,c1(CN2CCC(C(=O)Nc3c(C)nn(C)c3C)C(O)C2)ccc2c(c1)CCCO2 70099,C=CC(C)(O)CC(=O)NCC1(CNC(=O)CC2CCSC2)CC1 70100,N1(C(C(CC)NC(C)=O)=O)CC(CNC(=O)C(C)Sc2ncccn2)C(C)C1 70101,c1(C(=O)NCC(C)NC(c2c(C)csc2)=O)ccc(C2CCC2)nc1 70102,CC(CCC(C)(C)C)C(=O)NC1CCN(C(=O)CCc2cnoc2)CC(O)C1 70103,N(C1CCc2cc(C(=O)OCCc3cnc(O)nc3O)ccc21)C(=O)OC(C)(C)C 70104,C=CC(CC)CC(=O)N(CCC(C)NC(=O)CCN(C(=O)OC(C)(C)C)CC)C 70105,C1(CN(CC(=O)O)C(C)=O)CCCC(NC(=O)C(C)c2cc[nH]n2)C1 70106,CC1CCCC(CC(N2CC(O)(CNC(=O)C3=CSCS3)C2)=O)C1 70107,C1(CC(C)NC(C2(C3CC3)CCCO2)=O)CCN(C(c2ccco2)=O)CC1 70108,C#Cc1cccc(C(=O)NC2CN(C(C3COCCN3C=O)=O)CC2(C)C)c1C 70109,C(CC(C(C)C)NC(c1cc(CCNC(=O)Cn2nc(C)cc2C)on1)=O)OC 70110,C1(C(=O)NCC2(C)OCCN(C(CC(=O)NCC)=O)C2)CCn2c(O)nnc2C1 70111,C#Cc1ccc(Br)c(OCC2OC(=O)NC2(C)C)c1 70112,N1(C(c2scnc2C)C(=O)NC)CCC(O)CC12CC2 70113,N1(C(C2(C)CC(C#N)C2)=O)CCC=C(CNC(C2(C)CCCS2)=O)C1 70114,C(c1cnn(C)c1C)=CC(N1CCC(NC(C2CCC(=C)CC2)=O)C1)=O 70115,c1(CC)cccc(C(C(=O)NCC2(OC)CN(C(C)=O)C2)OC)c1 70116,C1(CCOC)CN(C(=O)C(N2CCN(C)CC2)(C)C)CCN1C(c1csnn1)=O 70117,CC(C)(C)C(CNC(C1(F)CCC1)=O)NC(=O)CC(=O)NC1CC1 70118,C1(NC(c2cc(C)on2)=O)CC(C)N(C(=O)COc2ccc(N(C)C)cc2)C1 70119,Cc1cccc(C=CC(=O)NC2CC(O)C2CC(=O)NCC(F)(F)C(N)=O)c1 70120,C1(C(N2CC(CNC(C(CC)OC)=O)C2)=O)CC(=O)N(c2ccc(SC)cc2)C1 70121,c1(C(=O)NCC2C3CN(C(C45COC(CCO4)C5)=O)CC23)ccc2cc[nH]c2n1 70122,CC1CC(CNC(=O)CC(C)(C)O)CN1C(c1cnco1)=O 70123,C#CCC(CC#C)C(=O)NCC(C)(C1CCC1)NC(C1CC1C(=O)OC)=O 70124,N1(C(CCC(=O)NC)=O)CCC2(CCN(C(=O)C(C)OCC3CCCO3)C2)C1 70125,c1(C(N)=O)cccc(O)c1NC(c1n[nH]cc1NCc1csc(Br)c1)=O 70126,c1(C(=O)NC2CCCC2CNC(c2cn[nH]c2)=O)ccc(F)c(Cl)c1F 70127,Cn1ccc(C(=O)NCC2CC(NC(c3cnnn3C3CC3)=O)C2)c1 70128,CC(C)CC(C(=O)NCC1C=CCN1C(=O)Cc1cccs1)N1CCCCCC1 70129,C(=O)(C(CCC=C(C)C)N(c1ccccc1Cl)C)NC.C1(C)C(=O)N1 70130,N1(C(C2CN(C)CC(C)O2)=O)CC(C)N(C(C23CCCC2C3)=O)C(C)C1 70131,C1(C(N(C2CN(C(c3c(OC)c(F)ncc3)=O)C2)C)=O)Cc2c(F)cccc2O1 70132,C1(NC(c2c(SC)snn2)=O)CN(C(=O)CSCC(N)=O)C2(CCCOC2)C1 70133,C(C1=CCCN(C(C2(C)CCCC2)=O)C1)NC(CCn1ncc(C)c1)=O 70134,Cc1cccc(C)c1NC(=O)C(c1ncc(Cl)s1)N(CC(C)C(C)C)C 70135,c1(C(=O)NC2(c3ccc(F)cc3)CCN(C(CCC#C)=O)C2)cc(=O)cc(Cl)[nH]1 70136,c1(C(=O)NC(C#C)CC2CC2)cc(CNC(c2coc(CC)n2)=O)on1 70137,c1(CC)cc(N2CCCC2(C)C(=O)NCCc2cc[nH]n2)ncn1 70138,N1(C(c2c(COC)cc[nH]2)=O)CCOCC1CNC(C1CC(F)(F)CS1)=O 70139,c1(COC)cc(=NCC2(O)CCN(C(C3(N(C)C)CC3)=O)CC2)[nH]cn1 70140,c1(C(N2CC(NC(CCCOC)=O)CC(C)(C)C2)=O)ccccc1C#CC1CC1 70141,C1(C(=O)NC(C2CCCC2)CNC(c2sc(C)c(O)n2)=O)COC2(CCC2)C1 70142,c1(C(N2CC3=C(C2)CN(C(C2CC2F)=O)C3)=O)cncc2n[nH]c(C3CC3)c12 70143,CCCCCC(O)CC(=O)NCC1CN(C(c2ccccc2-c2ncc[nH]2)=O)C1 70144,N1(CCC(=O)N(CC2N(C(C(C)OCC)=O)CCC2)CC)CCNC(=O)C1 70145,CC(CN1CCCCC1)C(=O)NC(C)CCNC(c1nn[nH]c1Cl)=O 70146,c1(CC(N2CCC(C(=O)O)CC23CC3)=O)ccc2cnccc2c1 70147,C#CC1(C(=O)NCCOCCOCCNC(c2ccc(CF)cc2)=O)CCCC1 70148,c1(C(N2CC(C)C(NCc3ccc(F)cc3F)C2)=O)cccc2c1CCC(=O)N2 70149,C1(NC(CNC(=O)OC)=O)CCCC(C(=O)NCCC(=O)NCC(C)C)C1 70150,c1(CC(N2CC(CCNC(C3CC(CC4CC4)C3)=O)(OC)C2)=O)ccccc1F 70151,N1(C(C2CCCN(CC)C2)=O)CC2(CC(CC(=O)NC3(CCF)CC3)C2)C1 70152,N1(C(C2N(C)S(=O)(=O)CC2)=O)CCCC2(CCCN2C(C2CC(O)C2)=O)C1 70153,c1(C(N2C3C(NC(c4n(CC#C)ccc4)=O)C(CC3)C2)=O)ccc2nonc2c1 70154,N1(C(C=Cc2ccc(C(=O)OC)o2)=O)CCCC(C2CN(C(=O)C(C)O)C2)C1 70155,C(=O)(CCC(C)(C)OC)N(CCCCN(C(C(CC)N(C)C)=O)C)C 70156,c1(N2C(CCNC(C3(C#N)CC3)=O)CSCC2)ncnc(Cl)c1F 70157,C(=O)(C(F)C(F)(F)F)N(CCC1OCCN(C(C2C(C(C)=O)C2(C)C)=O)C1)C(C)C 70158,N1(C(C(C)CC(F)(F)F)=O)CC2(C)CN(C(C3CC4C=CC3CC4)=O)CC2(C)C1 70159,N1(C(c2cn(CC(=O)OC)nn2)=O)CC2CC2(CNC(=O)C(F)(F)C2CCC2)C1 70160,N1(C(c2c(C)cc(C)c(C)c2)=O)CCC2CCN(C(=O)CSCCC#N)CC12 70161,C1(F)(C(=O)NC(C(C)C)CCN(C(=O)C=Cc2nnn(C)n2)C)CC2(CCC2)C1 70162,c1(CNC(=O)NC2(C3CC3)CCCCC2)cccc2c1OCCC2O 70163,N1(C(c2n(CC#C)ccc2)=O)CCC(O)C(N(C)C(C2CC3(CCCO3)C2)=O)C1 70164,CCCC(O)C(CO)NC(=O)CCOCCNC(=O)Cn1ncccc1=O 70165,C1(NC2CC(CCCF)C2)CC2(CCC(C(c3nnnn3C3COC3)=O)CC2)C1 70166,c1(CN2CCC(C(C)=O)C2)cccc(Cn2nc(C)cc2C)c1 70167,C(=O)(C(C(C)C)NC(=O)COCC1CCCC1)Nc1cn(C2CC(OC)C2)nn1 70168,C12(C(=O)NCC3CC(NC(=O)CCC(F)(F)F)C3)CCCC(CCC1)C2 70169,N1(C(CC(=O)NCC#C)=O)CCC(C)C(NC(=O)C(C)Cc2ccncc2)C1C 70170,CCCCC(=O)C(=O)N1CCOC(C(C)NC(C23CCCN2CCC3)=O)C1 70171,c1(C2N(C(c3c(OC)oc(C)n3)=O)CCC2)cccc(Cl)c1Cl 70172,N(C(=S)N1CCC(Oc2ccc(Cl)c(F)c2)C1)CCCF 70173,c1(N2CCN(C(=O)CCCN3CCCCC3)CC2)ncnc2ccccc12 70174,C(=O)(C=C=C(C)C)N1C(C(=O)NCCC2(COC)CC2)CC1C 70175,CCCC(C(=O)OC)C(=O)N1CCC2(C1)CN(C(C1CCCS(=O)(=O)C1)=O)C2 70176,N1(C(Cn2c(C(C)C)ncc2)=O)CCC(O)C(NC(=O)C(C)(C)c2cnco2)C1 70177,Cc1cc(O)cc(O)c1CNC1CN(C(=O)CCc2ccccc2Br)CC1C 70178,C#CC1CCC(C(N2CCOC(CNC(=O)COc3cn[nH]c3)C2)=O)CC1 70179,c1(CCC(=O)NC(C2(O)CCN(C(C3(O)CCCC3)=O)C2)C)ccc(F)c(F)c1F 70180,C(=O)(C1CCc2nccn21)N1CCCN(C(Cc2n(C)ncc2Br)=O)CC1 70181,C(C(C)(O)C(=O)NCc1cccc(F)c1)OC.C12CC(C1)NC(=O)CCNC2=O 70182,CCC(C)(C)C(=O)C(=O)NC1(CO)CCCN(C(=O)C(c2ccc(C)cc2)O)C1 70183,c1(C(=O)NCC2(C)CCCN2C(C2CCSCC2)=O)cccn2cnnc12 70184,CC(CC(F)(F)F)C(=O)NC12CCC(NC(C3C=CCCC3)=O)(CC1)C2 70185,c1(C(=O)NC(C)C(C)NC(=O)CCc2cnn(C)n2)cc(Cl)n(C)n1 70186,C1(Nc2c(OC(CCF)CC(F)(F)F)ccc(Br)c2)Cc2nc3ccccc3n2C1 70187,C1(CCC(C)C)CCN(C(C2CCCCC2)C(=O)NC2CCOC2)CC1 70188,c1(-c2cn(CC3N(C(CCCCC(=O)NC)=O)CC3)nn2)cccc2cnccc12 70189,c1(OC(C(=O)NCC2CN(C(CC3C(C)C3)=O)C2)C)cccc(Br)c1 70190,Cc1cc(C=CC(N2CCN(C(=O)C(C(C)C)N(C)C)CC2C)=O)c[nH]c1=N 70191,C1(C(N2C(CCCNC(c3cc(C)no3)=O)CCC2)=O)CCC2C(CC1)C2(F)F 70192,Nc1sc2c(c1C(=O)NC1CC(C(=O)Nc3ccc(CO)cc3)C1)CCC2 70193,CCC(CNC(C12CC(C)(C1)C2)=O)(CC)NC(=O)CCn1cccn1 70194,C(=O)(CS(=O)(=O)CC(C)C)NC1CCN(c2snc(CCOC)n2)CC1O 70195,C1(C(N(CC(C)O)CCNC(=O)COC2(C)CCOCC2)=O)CN2CCN1CC2 70196,c1(C(N2CCOCC(NC(C)=O)C2)=O)cnc2[nH]ncc2c1 70197,C1(OC)(CNC(=O)CC2(C)CCN2C(=O)C(C)OCC(C)C)CCOC1 70198,N1(C(c2cc(-c3nn[nH]n3)cc(Cl)n2)=O)CCC2(CCOCC2)C(NCCOC)C1 70199,C1(C(=O)NCC2CC(NC(c3ccnnc3O)=O)C2)OCC2CCCCC12 70200,C1(C(N(C2CCSCC2)CC)=O)CCC(C(F)(F)F)C1 70201,C1(C(N2CC(CCCCNC(C(C3CCOC3)OC)=O)C2)=O)CN2CCC1CC2 70202,C1(CNC(CCC2CCC(=O)N2)=O)CC2(CC2)CN1C(c1nc(Cl)c(Cl)s1)=O 70203,C(=O)(C(F)(CNC(=O)C(C)NC=O)C(C)C)NCCC(C(C)C)(F)F 70204,C1(C)(CC(=O)NC(CCOCC)C)CCN1C(=O)CC1CC(F)(F)C1 70205,c1(C(=O)NCCCCN(CCCNC(C(C=C)O)=O)C)c[nH]cc(C)c1=O 70206,Cc1cc(CC=O)cs1.C(C(=O)N(CC(N)=O)C(C)C)=CCNC 70207,c1(SC)cc(Cl)ccc1CO.c12cccn1CCOC2=O 70208,N1(C(=O)CCc2c[nH]cn2)CCC2(CCC(NC(C3CC(O)C3)=O)C2)C1 70209,N1(C(C2CCC(C(=O)Nc3ccc(C)cc3OC)C2)=O)CCC(COC)C(O)C1 70210,c1(C(C)C)ccc(OCCCC(=O)NCC(C)NC(c2cc(F)n[nH]2)=O)cc1 70211,C=CCCCCCC(=O)NCC1COC(CNC(c2c(C)cc(=O)oc2C)=O)C1 70212,CCS(=O)CC(=O)NCC1(C(C)NC(=O)CNC(c2ccc(OC)cc2)=O)CC1 70213,C1(CCN(C(C2(CC)CCOC2)=O)C)CCCCN1C(c1cc(C(C)C)on1)=O 70214,C(=O)(CC(CC(C)C)NC(c1cccc2nccn12)=O)NC(CC(C)(C)OC)C 70215,c1(C(=O)NC2CCC(NC(C3(C=C)CC3)=O)C2)ccnc2c1CCO2 70216,c1(C(=O)NCCC2OCCN(C(=O)OC(C)(C)C)C2)ncccc1N=[N+]=[N-] 70217,C1(C(N(CCCCNC(CCCC(C)C)=O)C)=O)CCc2n[nH]cc2C1 70218,c12cccc(c1)C2.C1(C(C)C(=O)O)CCN(C(c2cnsn2)=O)CC1 70219,C1(C)(NC(C2N(C(=O)CN3CCC(C)CC3)CCC(=C)C2)=O)CC(C)(C)OC1=O 70220,C(=O)(C(O)CC(C)(C)C)NCC(CCNC(CSc1ccc(C)cc1C)=O)O 70221,CCC(C)CCCCC(=O)NC1CC(C)N(C(c2ccc3oc(O)nc3n2)=O)C1 70222,C(c1ccc(OC)c(F)c1)=CC(=O)NCC(C(=O)OC)CC1CCCC1 70223,c1(C(=O)NCC2C(CNC(CSCCOC)=O)C2)ccc2nc(C3CC3)oc2c1 70224,O=S(=O)(c1cc(F)cc(F)c1)Nc1ccc(Br)c(Cl)c1F 70225,c1(C(N2CC(COC)(NC(c3ccc(=NC)[nH]c3)=O)C2)=O)ccn2nnnc2c1 70226,C1(C(N(CCN(CC(COCCOC)O)C)C)=O)(OC)CCCCC1 70227,C1(NC(c2cccc(N(C)C)c2)=O)C2CCC1CN(C(C1CC(=O)N1)=O)C2 70228,C=C1CCN(C(C2CC(=O)C2)=O)C(C(=O)NCC2CC2c2ccoc2)C1 70229,c1(C(C)OC)nc(-c2c[nH]ccc2=O)n(CC2CCCOC2)n1 70230,C(C(=O)NCCN1CCN(C(=O)C(=O)NCCC(N)=O)CC1)(C(C)(C)C)OC 70231,Cc1ncc(NC(C2(CCNC(C3(C(=O)NC4CC4)CC3)=O)CCC2)=O)c(C)c1C 70232,c1(C(=O)NC2CC(CNC(C3C(C)CCO3)=O)C2)c(Cl)csc1Cl 70233,CN1CCCCC1C(=O)NC1(CNC(c2cccc(C3(C#N)CC3)c2)=O)CC1 70234,CC(C)CC(C(=O)N1C2CCCC1CC(NC(=O)Cc1cn(C)cn1)C2)C(C)C 70235,C1(C(=O)NCC(C)N(C(c2ccc(F)cc2F)=O)CC)CN(CP(C)(C)=O)C1 70236,N1(C(C(C)=CC)=O)C2CCC1C(CNC(=O)CCC(=O)NCc1ccccc1)C2 70237,c1(CC(C(=O)OC)NC(=O)NCc2nnc(Br)s2)cccc(F)c1 70238,C(C(CC(=O)NC(C(C)C)C(C)C)C1CCC1)NC(C1C(C(C)C)(CC)C1)=O 70239,C#CCCCCCC(=O)NCc1cc(C(=O)NCC(C)C(C)CC)n[nH]1 70240,CCCCCC(O)CC(=O)NCC1CCCN1C(c1cnn(C)c1C(C)(F)F)=O 70241,C(=O)(C1=NOC2(CCCN(Cc3cc(Cl)sc3Cl)C2)C1)OC(C)(C)C 70242,CCC(CC(=O)NC1COCCOC1)NC(=O)C(C)C1(O)CCC1 70243,C#CCCC(C(=O)N(C(CO)C(C)C)C)NC(=O)C(C)SC(C)C 70244,C1(C(=O)NCCC(=O)NC(CC)C)CCN(C(C2CC2C(F)F)=O)C12CCC2 70245,C1(C(=O)NCC=CCNC(C2(CC=C)CCCC2)=O)Cc2nnc(C)n2C1 70246,C1(NC(CCOCC)=O)CCC(C(N2CCC2CF)=O)C1 70247,c1(C(=O)NC2CCC(NC(CC(CCC)C)=O)C2)cc2c(s1)CCCCC2 70248,C1(NC(=O)C2=CCCSC2)CCN(C(=O)CC2CN3CCN2CC3)CC12CCC2 70249,c1(-c2cncc(OCC)c2)ccc(F)c(N(C(=O)CCC=CC(C)C)C2COC2)c1 70250,c1(C(N2CC(NC(c3cn(CCC)nc3C)=O)C2)=O)ccc([N+](=O)[O-])cc1F 70251,C12(C(=O)NC(C)CCCNC(C3NC(=O)CC3C)=O)CCCCC(=O)N1CCC2 70252,N1(C(C(CC)n2nccc2C)=O)CCC(NC(c2cnc(C)n2C)=O)C(C)(C)C1 70253,c1(NC2CN(C(c3cnc(C)nc3O)=O)CC2C)cc(C(C)C)nc2ncnn12 70254,C1(C(=O)NC2CC2)CCC(NC(=O)C=C2CC(C(C(=O)OC)F)C2)C1.C1(=O)CN1C 70255,N1(C(C(C)c2cc[nH]n2)=O)CC(CNC(c2cc(C(N)=O)no2)=O)C2(CC2)C1 70256,C1(C)(C(N2CCC(CCOC)C2)=O)CCN(C(=O)C(C)CC(N)=O)CC1 70257,C12(CCNC(C=C(CCN(C)C)Cl)=O)CCC1CN(C(c1cnccc1Cl)=O)C2 70258,c1(C(N(CC(CN(C)C(c2ccc(O)c(N)n2)=O)O)C)=O)ccc2c(c1)CC2 70259,CC#CCC(C(=O)NCc1cc(C)n(C)n1)NC(=O)C(C(C)C)SC 70260,c1(C(N2CC(NC(C(CC)COC)=O)C(O)C2)=O)c(C)cc(O)nc1C 70261,C1(NC(CC(C(=C)C)OCC)=O)CC2CCC1N(C(=O)CNC(C)=O)C2 70262,c1(CC(=O)NCC2(NC(CCOC)=O)CCCCCC2)cccc2ccsc12 70263,N1(S(CC)(=O)=O)CCC2(CC(C(=O)Nc3cccc4c(O)cccc34)=NO2)C1 70264,C1(OC)CC2CC(C(N3CC(N(C(=O)COc4ccc(F)c(F)c4)C)C3)=O)CC12 70265,N1(C(CC(COC)C)=O)CCC2(CCCN2C(=O)CCc2nc(=N)[nH][nH]2)CC1 70266,c1(C(N(CCNC(CC2(COC)CC2)=O)C2CC2)=O)cnc2ncnc(O)c2c1 70267,C(=O)(C1CCCn2c(C)nnc21)N1CC(NC(c2c(C)nncc2)=O)(C(C)CO)C1 70268,N1(C(C2N(C(C(C(=O)OCC)F)=O)CC(F)C2)=O)CCCC(OC)CC1 70269,Cc1nc(NC2C3CC2CN(C)C3)c2sccc2n1 70270,Cc1ccc(F)c(C(=O)N(CCSc2ncncc2N)Cc2ccccc2)n1 70271,C12(NC(C(CCC)N(C)C)=O)CN(C(c3nc(C)ncc3Cl)=O)C(COC)(C1)C2 70272,c1(C(=O)NC2CCCC(N(C(CN3CC(CC)C3)=O)C)C2)cn2nc(C)sc2n1 70273,C1(C(=O)NC2(CNC(CCC3CCC(=O)NC3)=O)CCC2)COCC2(CCC2)O1 70274,C1(C(N2CC3C(CNC(C4CCCC4)=O)(C3)C2)=O)CCN(CCO)C(=O)C1 70275,CCC(CC(=O)N1CC2C(C(=O)NCC(C)(C)CN=[N+]=[N-])C2C1)C(F)F 70276,CCCCCCCCCC(=O)NCC1CN(C(=O)C2=NNC(=O)CC2)CCO1 70277,c1(N2CCCC(NC(C(C)(C)C)=O)C2)nc(=N)[nH]c(=NCc2csc(Br)n2)[nH]1 70278,C(C(COC)CC(=O)NCCCC(=O)NCC1COCC1O)OC 70279,c1(C(N2CCC(C(C)(C)C)(CNC(C(CC)(C)O)=O)C2)=O)ncnc2ccsc12 70280,C(=O)(C(CC(C)C)C(N)=O)NC(C(=O)N1CC(CC)C1)CCF 70281,c1(CNC(N(CC(CC)NC(=O)OC(C)(C)C)C)=O)cc(C)nc(Cl)c1 70282,Cc1nc(C(=O)NC2CCOCC2C(=O)NC2(CO)CCC2)sc1C 70283,C1(C2CC2)(C(=O)NC2CC(CCNC(C34C=CC(CC3)C4)=O)C2)CCOCC1 70284,c1(C(N(CC(F)(F)F)C(C)CO)=O)cccc(Nc2ncccc2Br)c1 70285,Cc1ccc(F)c(C(=O)NC2CC3CC2CC32CC2)c1Cl 70286,C1(CNC(C(C=C)O)=O)CCCC2CN(C(=O)CCCCC(=O)NC)CC12 70287,c1(C(N2C(CNC(CC(CCC)(C)O)=O)CC2)=O)cc(F)cc2nccnc12 70288,C1(NC(c2c(C)cc(C)[nH]2)=O)CS(=O)(=O)CC1NC(=O)CCC1CCCCC1 70289,C#CCC(C(=O)NCC)NC(=O)NC1(C)CCN(CC=C(C)C)C1 70290,C1(NC(C(CSC)O)=O)CN(C(c2ccc3ncncc3c2)=O)CC1S(C)(=O)=O 70291,C(=O)(C(O)C(F)(F)F)NC(CN(C(c1csc(-c2ccsc2)n1)=O)CC)C 70292,c1(C(N(C(CN(C(C(COCC)C)=O)C)C)C)=O)cc2n(n1)CCCC2 70293,N1(c2nc(NC(C3CCOC3)CC)c3c(n2)scc3)CCc2cccc(F)c2C1 70294,C(CN=c1[nH]c(Cl)ncc1C(N)=O)C1CCC(NC(C2OCCN(C)C2)=O)C1 70295,C=CCC(C(=O)NC1CCCCC1CNC(c1c[nH]nc1F)=O)C(C)C 70296,c1(C(N2C(CNC(c3sccc3Cl)=O)CC(O)C2)=O)ncn2c1CCCC2 70297,C1(NC(c2cnc(C)nc2C2CC2)=O)CN(C(C2CC2C(F)F)=O)CC1C1CC1 70298,N1(c2cc(OCC)ncn2)CCC(CNC(c2ccn(C)c2)=O)C(C)C1 70299,N1(C(=O)C(C2CCOCC2)F)CCN(C(=O)CCCn2ccnn2)C(CC2CC2)C1 70300,Cc1cc(C(=O)NC2CN(C(c3cc(O)no3)=O)CCC2C(F)(F)F)cnc1F 70301,N1(C(=O)CC2(O)CC2)CCC2C(C1)CN2C(C1CCOCC1)=O 70302,c1(C(=O)NCCC2CCC(NC(C(C)NC(C)=O)=O)C2)noc2ccc(Cl)cc12 70303,Cc1nc(CC(N2CCC(CCNC(=O)CCCc3ccncc3)C2)=O)c(C)s1 70304,N1(C(c2c(F)cccc2Cl)=O)CCC2C(CCN2C(=O)CCn2cncn2)C1 70305,C=CCC(C)C(=O)NC1CCC(N(C(=O)CC2C(=O)NN=C2C)CC)CC1 70306,c1(N(CC(=O)NC2(CO)CN(C(C3C4CCCC34)=O)C2)C)ccc(Cl)cn1 70307,C1(C2CC2)(CNC(c2c(C(C)C)ccs2)=O)CCN(C(=O)C(O)C2CCC2)C1 70308,N1(C(C23N(C(C(COC)C)=O)CCC2CCC3)=O)CCC2(CCCCC2)C1 70309,c1(CC(=O)NCCCN(C(=O)C(O)c2ccco2)CC)cncnc1 70310,C1(C2CCCN2C(c2ccccc2)=O)CCCN(C(C2(CN)CCCCC2)=O)C1 70311,CC1C(=O)NC(=O)CN1C(C1(C)CN(C(c2cc([N+](=O)[O-])n[nH]2)=O)C(C)(C)C1)=O 70312,C(C(CO)C(F)(F)F)NC(C(CC1CC1)NC(c1nn(C)c(O)c1)=O)=O 70313,CCC(CO)C(=O)NC(C)CC(C)NC(=O)CC(=O)OC(C)(C)C 70314,C1(CC)CCN(C(C2CC23CCC3)=O)C1C(=O)NCC(=O)NC(C)(C)C 70315,CC(CC=Cc1ccccc1)C(=O)N1CCC(NC(C2OCCO2)=O)C1 70316,C(C)(CCCC(=O)NCC1OCC2CCC1C2)NC(C(C)NC(CC)=O)=O 70317,C12(NC(CN=S(C)(C)=O)=O)CCOCC1CN(C(c1ccncc1)=O)C2 70318,C(=O)(C1CCCn2ccnc21)N1CC(NC(CCCS(N)(=O)=O)=O)C(F)C1 70319,c1(C(=O)NCCOCCN(C)C(C2(C)CCNC2=O)=O)ccc2c(n1)CCO2 70320,C1CN=C(NC(C)CNC(C2(CCCF)CCC2)=O)NC1.C(C)(C)(C)OC(C)C 70321,C(c1ccc(COC)o1)=CC(=O)OC.c1(CC(=O)N2C3C(CC3)C2)sc(C)nc1C 70322,CC(CNC(=O)CN1CCC(=O)CC1)CC(=O)N(C)Cc1nnc(O)o1 70323,C1(NC(CCC(=O)NC)=O)CC(O)CN(C(=O)CCCNC(N)=O)C1 70324,c1(C(=O)NC2C(N(C(=O)CCF)C)CCCC2)cccc2nc[nH]c12 70325,c1(CNC(c2c(C)ccs2)=O)cc(F)c(F)c(Cl)c1 70326,C1(CCC(=O)NCCS(CC)=O)CCCCN(C(C2CC3(CCO2)CC3)=O)C1 70327,C1(NC(C=CC(=O)OCC)=O)CC2C(NC(=O)C(c3ccccc3)C)C2C1 70328,N1(C(C(CC)NC)=O)CC2CN(C(c3cnc(Cl)c(C)c3)=O)CC12 70329,Cn1nnc2c1CCC(C(=O)NC1CCC(O)CN(C(=O)CC3CSC3)C1)C2 70330,N1(C(C(CCC)(C)O)=O)C2CCC1C(C)C(NC(=O)CCc1cscn1)C2 70331,c1(NC(N2CC(CCN3CCOC3=O)C2)=O)cc(Cl)ccc1I 70332,N1(CCCC)CCCCC1C(=O)N(CCCCNC(C1(CCF)CC1)=O)C 70333,CC(C)CC(CNC(=O)CCCC1(NC(=O)CCC2(C)CC2)CCC1)CO 70334,C1(NC(C=CC(CC)=CC)=O)CC1C1CCCN(C(=O)C(C#N)CC)C1 70335,C1(CNC(C(=O)NC(C)C)=O)CN(C(c2cn(C3CCC3)nn2)=O)C(C)(C)C1 70336,C(=O)(C#CC1(C)CCCO1)NC1C(NC(Cc2nc(COC)sc2)=O)C1 70337,CCCC(O)C(=O)N(C)CC1COCCN1C(=O)CC12COCC(C1)C2 70338,Nc1cc(C(=O)NCCOC2CN(C(=O)CCc3ccncn3)C2)cc(Cl)n1 70339,C1(C(N2CCCC(C(C3CCOCC3)=O)C2)=O)Cc2ccc(O)cc2CN1 70340,C1(C(N(CC=C)CCO)=O)CCC(C)(C)N(C(c2coc(C(N)=O)c2)=O)C1 70341,c1(C(=O)NCCN(CC(=O)NC2CC2)C2CC2)ccoc1I 70342,c1(CC(=O)NC(C)(C)CN2CCN(C(c3csnn3)=O)CC2)cc(Cl)cc(Cl)c1 70343,C12(COC(c3cncc(N)n3)=O)CCC(C(=O)OC)(CO1)C2 70344,c1(C(N2C(CCCNC(CN(C(C)=O)C)=O)CCC2)=O)cc(C(F)F)ccn1 70345,C#Cc1ccc(F)cc1C(=O)NC1CN(C(=O)CC(C)F)CC1n1cccn1 70346,C(=O)(C(C)C(CC)CC)N1C(C(N(CC(=C)C)C)=O)CC(=O)C1 70347,c1(C(=O)NC2(CNC(c3n(C=C)nnc3)=O)CCOC2)cc2sc(Cl)cc2s1 70348,C(C(=O)NC12CCC(C1)N(C(=O)CCc1ccsc1)C2)(C(C)(C)C)OC(C)(C)C 70349,C=C(C)C(C)(C)C(=O)NC1CN(C(=O)C(=O)NCC2CC2)CCC1CO 70350,c1(C(=O)NC2(CCNC(CCC#CC)=O)CCC2)ccc2ccnc(Cl)c2n1 70351,c1(C(N2C(C)(COC(c3c(OC)c(Cl)sc3)=O)CCC2)=O)n[nH]c2c1CCC2 70352,C#CCC(C)(C)C(=O)N1CC(C(=O)NC2CCC(N(C)C)C2)C(F)C1 70353,C(=O)(CCCCCOC)NC1(CC=C)CCN(C(c2ncc(N)nc2C)=O)C1 70354,C1(C(=O)NC2C(NC(c3c(Cl)cn(CCC)n3)=O)CCC2)CCc2nncn2C1 70355,C1(CC(N2CCC(C(=O)NCCCC3CCC3)C2)=O)CC(C2CC2)C1 70356,c1(C(=O)NC2(C)CC(NC(CC(=C=C)C)=O)C2)cc[nH]c2nccc1-2 70357,CC(C)C1=NOC(C(N2CCC(C(C)NC(C3CC(=O)C3)=O)C2)=O)C1 70358,C=C=CCCC(=O)NCCC1CCC(NC(=O)CCS(C)=O)C1 70359,C1(NC(C(C(C)C)NC(C)=O)=O)CN(Cc2ncc(Br)cc2C)CC1C#N 70360,C1(NC(C=CC(C)(C)SC)=O)CCCC1NC(=O)C(C)CC1CCC1 70361,N1(C(c2cc(C)ncc2)=O)CCC2CC2(NC(=O)COCc2ccncc2)CC1 70362,c1(C(=O)Nc2c(C#N)nccc2)ncncc1C1=CCOCC1 70363,c1(CC(=O)NCCC(CCNC(C(C)NC(=O)NC)=O)C)c(C)nn(C(F)F)c1C 70364,N1(C(C(C(=C)C)(C)O)=O)CCCC(C2CCN(C(=O)COCC)CC2)C1 70365,c1(C(=O)NC(COCC)C2CC2)ccc(NC2(C(=O)NC)CC2)c(F)c1 70366,c1(OC)ccccc1NC(=O)C(C(C)C)N1CCN(S(=O)(=O)C(C)C)CC1 70367,C(=O)(C(O)C(C)(C)C)N(CCC(C)NC(=O)COC1CCOCC1)C 70368,C1(NC(c2cc3ncccc3o2)=O)CC2CC1CN(C(c1cc(Cl)sc1Cl)=O)C2 70369,N1(C(CN2C(C)CCCC2)=O)CC2(CC(C(=O)NC3CN(C(C)C)C3)CO2)C1 70370,c1(C(C)O)ccc(C(N2CCCC2CNC(c2coc(Cl)n2)=O)=O)cc1 70371,C(CC(=O)NC1CCC12CCCC2)(C(C)OC)NC(C(COC)(C)C)=O 70372,C1(NC(c2cnc(Cl)c(Br)c2)=O)CCc2nc(NC(c3cc(Br)cs3)=O)sc2C1 70373,C(=O)(CCCCCN(C(=O)C(O)C1CC1)C)N1CC(C#C)(N(C)C)C1 70374,c1(NC(C(CCC)NC(=O)C(C)(Cl)Cl)=O)cc(C)cn(C)c1=O 70375,CC1(C)C(=O)NCC1NC(C1CC(F)CN1C(C1CC1c1cccc(O)c1F)=O)=O 70376,C(=O)(CCC(=O)NC1CC1NC(=O)CNC(c1cccc(F)c1)=O)N(C)C 70377,C1(OC)CCCC(C(=O)NCC2CCC(C(=O)N(CC(O)CO)CCO)CC2)C1 70378,C(=O)(CCCCNC(c1snc(C)c1N)=O)NCC(C(=O)NC)C 70379,N1(C(C(CC(C)C)N(C)C)=O)CCC2(CC(NC(=O)Cc3cccc(Cl)c3)C2)C1 70380,N1(C(c2cncc(NC)c2)=O)CC(O)C(O)C1CNC(C1CC1OC)=O 70381,N1(C(C=C(C)C2CC2)=O)CCN(C(C2CC3CC23)=O)CC1 70382,C(=O)(C(C(C)(C)C)N(C)C(=O)OC(C)(C)C)NCC(c1ncccn1)CC 70383,C(=O)(C(CO)C(C)(C)C)N1CC(C(C)NC2CN3CCN2CC3)OCC1 70384,CCCCS(=O)(=O)NCC(=O)NC1CCCC1CNC(C1CC(C(F)F)C1)=O 70385,C1(CNC(C2C(C)C2)=O)CC2CCCC2N1C(=O)C(=Cc1c[nH]cn1)F 70386,c1(CC)ccc(C(F)(F)F)cc1S(N)(=O)=O.N12CCCC1CCCNC2=O 70387,C1(C(=O)NCCOC2CN(C(CCc3cnc(C)s3)=O)C2)CN(C)CCO1 70388,C=CCC(F)(F)CNC(C1(CO)CCN(C(c2ccc(CC)[nH]2)=O)C1)=O 70389,N12CC3CN3C(O)=NN=C(C1)C1(CC(C)CCn3cccn3)CCN(CC1)C2=O 70390,Cc1cc(C(=O)NC(CO)C(C)NC(C2(C3CCCCO3)CCC2)=O)nn1C 70391,c1(C(N2CC=C(CNC(C3(C)CC3F)=O)CC2)=O)ccc2snnc2c1 70392,CN(C)NC(=O)CCC(=O)Nc1ccnn1CC(=O)NC1CCC(F)(F)CC1 70393,CC1(C)CNCC1CC(=O)NC(c1ccccc1)C1CC1CC(F)(F)F 70394,C1(NC(c2c(C)cc(CNC(C(C)=CC3CC3)=O)o2)=O)CCCC1C1CC1 70395,C1(CCNC(=O)Cn2ncnn2)CCCN(C(=O)C(c2ccccc2)=O)CC1 70396,c1(C(N2C(CNC(C3(CC#N)COC3)=O)CCCC2)=O)cnc(F)c(Cl)c1 70397,c1(NC(C2CN(C(c3ccc(Br)cc3Cl)=O)C2)=O)cc(F)c(F)cc1Cl 70398,c1(CN(C(=O)C(N2CCCCC2c2nnc(C)o2)=O)CCOC)ccc(F)cc1F 70399,C1(C(C)CN(C)C)CCN(C(=O)N(CCS(C)=O)CCOC(C)(C)C)CC1 70400,C(=O)(CC(C)C(F)F)NCC(C1CCN(C(c2nc(C)oc2C)=O)CC1)F 70401,Cc1cc(C(=O)NC2CCCCC2NC(c2cccs2)=O)nn1C(C)C 70402,c1(C(C(=O)NC)N(N2CCOCC2)CCC(=O)OC)cnc(C)c(C#N)c1 70403,C1(CC)CCN(C(C2CCC2COC)=O)C(C(=O)NC2C(O)CC2O)C1 70404,n1(CC(=O)NCC=CCNC(c2cccc(C)c2N)=O)cc(P(C)(C)=O)cn1 70405,c1(CC)c(C(N2CCN(C(c3ccnnc3S)=O)C3CC23)=O)cccc1C 70406,N1(C(C2CN(C(C)=O)C2)=O)C2CCC1CN(C(C1COC(C)(C)CO1)=O)C2 70407,CC1(C)OC2CC(C(=O)NC3(CNC(C4OCC5CCCCC45)=O)CC3)CC2O1 70408,Cc1ccc(-c2nc(-c3ccc(C(C)(C)C)cc3)nn2C2CCC(C)C2)c(C)n1 70409,n1(CC(=O)NC2CC(NC(CC3C(C)=NOC3=O)=O)C(O)C2)ccc(O)nc1=O 70410,c1(COC(=O)CCCCN2CCCS2(=O)=O)cc(O)nc(CSC)n1 70411,C1(NC(C2C(N(C)C)CN(C(CCCCCSC)=O)C2)=O)CC1C1CCCCC1 70412,N1(C(C=C(C)C(F)F)=O)CCC(NC(=O)COc2ccc(F)nc2)CC1C 70413,C1(C(=O)NCC2CCC(NC(C3CC(=C)C3)=O)CC2)CN(CP(C)(C)=O)C1 70414,N1(C(c2c(N)ccc(Cl)c2)=O)CCCN(C(c2ccccc2F)=O)CC1CO 70415,c1(OC(C)C)cccc(C(=O)NCC(CO)NC(c2cc(O)cs2)=O)n1 70416,CC(O)C(F)(F)C(=O)NC1CC(F)(CNC(=O)C(c2ccccc2F)(F)F)C1 70417,C1(CC(=O)N(C(C)CNC(C2CCC(N(C)C)CC2)=O)CC)CCS(=O)(=O)C1 70418,c1(C(=O)NCCN(C(=O)CC2CC(F)C2)C)cn(C)cc1C(F)(F)F 70419,c1(C2C(C(C)NC(=O)NCCCc3ccnn3C)C2)ccc(F)c(F)c1 70420,Cc1cc(CC(=O)NC2CCCC(NC(=O)CCOCC(C)C)C2)cc(C)c1 70421,c1(CCC)nc(C)c(C(N2CCC(NC(C3CC3C)=O)C2C)=O)s1 70422,c1(C(N2C(CC)C(C(=O)OC)CCC2)=O)ccc([N+](=O)[O-])c(O)c1C 70423,Cc1c(Br)ccc(O)c1C(N1CC(NC(=O)CCC2CCC(C)O2)C1)=O 70424,C1(CC(C)C)CC(C(=O)NCC2CN(C(c3coc(C(C)C)n3)=O)C2)CC(=O)N1 70425,O=C(C(=O)C(F)(F)F)N1CCC(CN(C2CCCCC2O)CCO)C1 70426,C1(CC)CCOC1C(=O)NCC1(F)CC(N2CC3(CCC3)CC(=O)N2)C1.OCC 70427,C(=O)(CCS(C)=O)N1CCC(C(C)(C)NC(=O)C(C)(C)N2CCOCC2)C1 70428,C1(NC(=O)CC2CCCC2)CCCC12CCN(C(=O)CC1CC3(CC3)CO1)CC2 70429,C1(NC(c2cc(O)nc(-c3ccccn3)n2)=O)CC2CN(C(=O)CCF)CC2C1 70430,N1(C(CNC(=O)NC)=O)CCN(C(=O)CC(C)(C)C2CC2)C(C(F)F)C1 70431,C1(C(=O)NCCN(C(=O)CCOC2COC2)C)(CC2CCC2)CCOC1 70432,C1(C(N(CC(=O)NCCN(CCC)C(C)C)CC2CC2)=O)CCCCN1C 70433,N1(C(=O)C=Cc2ccco2)CC23CCCC2(C1)CN(C(c1cc[n+]([O-])cc1)=O)C3 70434,C1(NC(c2c(CC)n[nH]c2)=O)CCC(C)N(C(c2ccc(C)cc2)=O)C1 70435,CC(C)C(C)C(CNC(c1ccc(N(C)C)nn1)=O)NC(=O)CC(C)(C)O 70436,c12cc(C)ccc1NC2=O.C1(NC(CC(=C)C)=O)CCC(OCC)CC1 70437,C1(CNC(C2CN(C(C)=O)C2)=O)CC(NC(c2n[nH]cc2Br)=O)C1(C)C 70438,c1(N2C(CCNC(=O)CN3CCS(=O)(=O)CC3)CSCC2)ncccc1[N+](=O)[O-] 70439,C(C1c2ccccc2CCN1C(c1ccc(C(N)=O)c(Cl)c1)=O)NC(C(C)C)=O 70440,c1(OC)cccnc1CN1CCC(C)(C(=O)NCC2CCO2)C1 70441,c1(CN(C(C2(CF)CCN(C(=O)CCC(=O)NC)C2)=O)CC)ccncc1OC 70442,c1(OCCNC(CN(C(C(C)N(C)CCO)=O)CCO)=O)ccccc1 70443,C1(NC(c2cccc(I)c2Cl)=O)CN(S(=O)(=O)c2cccs2)CC1(F)F 70444,c1(SC)ccc(C)c(C(N2CCC(C)(CNC(=O)C(O)P(C)(C)=O)C2)=O)c1 70445,c1(SC(C2CCN(CC(n3cnnn3)=O)CC2)C)ccccc1Cl 70446,C1(C(=O)NCC2CCN2C(=O)CSC(F)(F)F)CCCC1C(F)(F)F 70447,c1(C(=O)NC2C(NC(CCCC#CC)=O)CC2)cc2ccc(OC(F)F)cc2[nH]1 70448,CC1CC(c2nnnn2CC2CCCCCC2)(NCC(C)(C)C(F)(F)F)CCO1 70449,N1(C(c2c(C)n(C)nn2)=O)CC(CC(N2CCCCC2C(N)=O)=O)CC1(C)C 70450,C(C#Cc1cccnc1)NC(C1CCCN1C(c1cccn2cncc12)=O)=O 70451,N1(C(C(=O)NCCN(C(C2CC(OC)C2)=O)CC)C)CCCC(O)C1 70452,c1(CC)cc(C)c(C(=O)NC2CCCCC2CNC(c2cnc[nH]2)=O)o1 70453,C(C1=CCN(C(=O)CC2CCCS(=O)(=O)C2)CC1)NC(CC1CCC(C)CC1)=O 70454,N1(C(=O)OC(C)(C)C)CCC(C(=O)N(C2CCC2)CC2CC2)C1 70455,C1(C)CCC2CC2C1.C1(N(C(C2C(C(=O)OCC)C2)=O)CC)CCN(C=O)C1 70456,C1(C(=O)NC(CCC)C2CCC2)CCN(C(C2C=C(C)CS2)=O)C(C)(C)C1 70457,N1(CC(=O)NCC#CC(=O)NCC(n2cccn2)C)CCCCC1=O 70458,C1(CNC(c2c(C)nsc2)=O)CCCCN(C(=O)CCc2ccccc2)C1 70459,N(C1CCCn2nccc21)C(C1(C=C)CCN(C(c2cc(C)c(C)nn2)=O)C1)=O 70460,Cc1ccc(C(C)CC(=O)NC(C)C(C)(C)NC(c2ccsn2)=O)cc1 70461,c1(OC)ccc(-c2c[nH]nc2C(=O)Nc2ccc(F)c(OC(F)(F)F)c2)cc1F 70462,c1(OC)ccc(CO)cc1C(=O)NC(CNC(=O)CN1CCCCC1=O)C1CC1 70463,c1(C(=O)NCC(CN(C(=O)C=C2CCSCC2)C)(C)C)ccc2ccsc2c1 70464,CCC(CC(=O)NC(C(=O)N(C1CCSC1)C)C(C)O)C(F)F 70465,C12(C(=O)NCC(C)(C)O)CC(CN(C(C3C4CCC(F)C34)=O)C1)C2 70466,C1(C(=O)NCCC2(NC(C(C)N3CCCC3)=O)CCCC2)CCCC(C#N)C1 70467,N1(C(c2c(CC)cco2)=O)CCCN(CCNC(=O)Cn2cncn2)CC1 70468,Cc1c(C(=O)NCC2CC(NC(C34CC(F)(C3)C4)=O)C2(C)C)cccc1O 70469,C#CC(C)(C)C(=O)NCc1nc(C(=O)NC(C)CC(C)(C)O)c(C)o1 70470,C(=O)(CCC(F)(F)F)N(C1CCN(C(CCCC#C)=O)CC1)CC1CCCO1 70471,C#CC1(n2cc(C3(CNCP(C)(C)=O)CC3)nn2)CCCN(C(=O)CCC(=C)Cl)C1 70472,N1(C(C2CC2(F)F)=O)CCCC(C2CCCN(C(=O)Nc3ccc[n+]([O-])c3)C2)C1 70473,C1(NC(CN(C)S(N)(=O)=O)=O)CCCC12CN(C(=O)Cn1cc[nH]c(=O)c1=O)C2 70474,c1(C(c2nnnn2C2CC2)NC(c2c(F)cccc2F)C)cc(F)c(Br)c(F)c1 70475,C(=O)(C(C)CC(C)C(C)=O)N(C)CC1C(NC(C(C2CC2)OCC)=O)CCC1 70476,C1(CC(=O)NCC2C(NC(C(COCC)(C)C)=O)C2)CC2CCC1CC2 70477,c1(C(=O)NC2CN(C(c3cc(C)nc(C)n3)=O)CC(F)C2)ccc2[nH]ccc2n1 70478,N1(C(Cc2c(OC)ccc(Br)c2)=O)CCC2(CC1)CCN2C(=O)C(C)O 70479,c1(CN(C)C)ccc(C(N2CCC2CNC(c2csc(=N)[nH]2)=O)=O)[nH]1 70480,C#CCC(C)C(=O)N1CCC(C(C)NC(c2ccc(C3(C)CCO3)cc2)=O)CC1 70481,C1(C(=O)Nc2c(SC)cccc2)CCN(C(=O)CNc2nccs2)CC1C 70482,N1(C(C2N(CCC)CCCC2)=O)CCC(F)(CNC(=O)CC(C)(C)O)CC1 70483,C12CCC(C1)NC2=O.c1(C(=O)NCCNC(C2(Br)CC2)=O)ccco1 70484,c1(C(=O)NC2C(SC)CN(C(c3ccn(C)n3)=O)C2)ccc(CO)c(Cl)c1 70485,C(C)(C)(C=CC(=O)NC(C1CC(NC(=O)Cc2ccoc2)C1)C)SC 70486,c1(CC)nn(C)c(CC(N2CCCC(NC(=O)C(F)C3CCC3)C2)=O)c1Cl 70487,C1(C(N2C(CNC(c3n(C)cc(C#N)c3)=O)CC(F)C2)=O)CNC(=O)C(C)(C)C1 70488,C(C(=O)N1CC(C(N2CCC(CC(C)C)CC2)=O)C(F)C1)(C(C)C)OCC 70489,c1(-c2nc(C(C)SC)nn2C(c2cncc(F)c2)C)cc2c(OC)cccc2[nH]1 70490,C1(NC(c2c(C)ocn2)=O)CN(C(=O)C(C)OCC(C)C)CCC1F 70491,C(CCCCC(=O)NCC1CCC(C(=O)NCC(=O)NC(C)C)C1)SC 70492,Cc1nn(C)c(N)c1C(=O)NCC(C)NC(c1cccc(C(N)=O)c1C)=O 70493,CC(C)C(C(=O)N1CC(CCCCNC(C2CC3C=CC2O3)=O)C1)NC=O 70494,C#CC1(NC(=O)CCOCCN(C(=O)C2=NOCC2)C)CCOC1.OCC 70495,CCCCC(CNC(c1ccc(F)s1)=O)NC(=O)C(C)(C)n1ccnn1 70496,N1(C(CCC(C)C)=O)CCC12CN(C(C1CCCC(C)(C)O1)=O)C2 70497,Cc1c(C(N2CC(CO)(NC(=O)CC(C)F)C2)=O)nc2sccn12 70498,c1(CCCNC(CN(CCOC)C(C2C=CCS2)=O)=O)nc[nH]n1 70499,n1(CC(N2CC(C(C)NC(C34CC(CC(F)F)(C3)C4)=O)C2)=O)nc(Cl)ccc1=O 70500,CC(C)C(C)(O)C(=O)NC1CC1NC(c1cc(Cl)ncc1O)=O 70501,C1(CNC(C(C)OCCC=C)=O)CCN(C(c2cc(Br)no2)=O)CC1(F)F 70502,c1(SCC2CCN(C(N3CC(C)CC(C)C3)=O)C2)ccc(S(=O)(=O)C(F)F)cc1 70503,N1(CC)CC(C(N2CCCC(N(C(=O)C(C)Sc3ccncc3)C)C2)=O)CC1=O 70504,CCC(CC(=O)NCC(C1CC1)NC(=O)Cc1cnnn1C)SC 70505,CC(C)CC(C)C(=O)NCc1nc(C(=O)N(C2COCC2(C)C)C)co1 70506,C1(NC(C(c2cn(C)nc2)=O)=O)CC(NC(=O)CCN2CCCCC2)C12CCC2 70507,Cc1cc(C)c(C(N2CCN(C(=O)CC3COCCN3C)C(CO)C2)=O)c(C)c1 70508,c1(C(N2CCCC(OC)C2)C(=O)NCC)nc(Br)ccc1OCC(C)C.C1(C)CC1 70509,C(=O)(CC(P(C)(C)=O)P(C)(C)=O)N(C(CNC(C(CCC)O)=O)C)C 70510,c1(C(N2C(C)CCC(CNC(=O)CCC(C)(C)C)C2)=O)ccc2n[nH]cc2c1 70511,c1(C(=O)NCC(CC)N)ccc(C(N)=O)o1.c1(C(N2CC(CO)C2)=O)ccn(CC)n1 70512,C(CC)(CCCNC(=O)C=Cc1cncs1)NC(C(C)NS(CCC)(=O)=O)=O 70513,C12(NC(c3cc4n(n3)CC(F)C4)=O)CCCC1CN(C(c1cc(O)ncn1)=O)C2 70514,C=CCC(F)(F)C(=O)NCC(C)(C)CNC(C1CSC(C)=N1)=O 70515,c1(C(=O)NC2CCN(C(c3ccc(OC)s3)=O)CC2F)ccc2nc(O)oc2c1 70516,Nc1ccc(C(=O)NCC(CO)NC(C2CCCN2C=O)=O)c(Cl)c1 70517,c1(CNC(C(=O)NCC)=O)cccc(CNC(C2CCC(F)C2)=O)c1 70518,N1(C(C=Cc2cn(C)nc2)=O)CC2COCCC2(NC(=O)C(F)=C2CCCC2)C1 70519,C1(CN(C(C2CC(OC)C2)=O)C)CCN(C(=O)CCN2CCCCC2C)CC1 70520,c1(C(=O)NCC2CN(C(C(C)=C3CC3)=O)C2)ccc(C(F)F)nc1 70521,CCCC(O)C(=O)NCC(C)N(C(c1coc(-c2cccnc2)n1)=O)CC 70522,c1(C(=O)NC(CC=C)C(=O)NCC(CC)n2cccn2)cc(F)cnc1O 70523,c1(C(=O)NC2CCN(CC=C)C2=O)noc2cc(Br)ccc12.C1(C(C)C)C(=O)O1 70524,C(C(C)N=c1nc(NCC)cc(OC)[nH]1)NC(CCC(=O)NC)=O 70525,CC(C)C(C(=O)N1CC(CNC(c2c[nH]nc2-c2ccsc2)=O)C(C)C1)N(C)C 70526,CC1CN(C(C2CC(C)(C)CO2)=O)CC1C(=O)NC1C=CCC1 70527,C1(NC(c2ccn(CC)c2C)=O)CN(C(C23CCCC2C3)=O)C2(CCCCC2)C1 70528,C(CC(C(=O)NCC1CCCCO1)NC(=O)CC1CCC(=O)C1C)OC 70529,C(CCCC(=O)N(C(CCNC(C1CCCCO1)=O)C(C)C)C)OCC 70530,C=C=C(C)CC(=O)NC(CCNC(c1cccc(C)n1)=O)C(C)C 70531,C(=O)(C1=CCCCO1)N(C1CCCN(C(C2(CC=C)CCOC2)=O)C1)CC 70532,N1(C(C(C)OCCOCC)=O)CCN(C(=O)CN2CSCCSC2)C2CCC12 70533,C1(CC(=O)NC2(C)CC2C)(OC)CN(C(=O)CC2CC(C)=NO2)C1 70534,c1(OC)ccc(C(=O)NCCC(C)NC(=O)C(O)Cc2ccc(F)cc2)cc1C 70535,N#CC1CNCC12CCC2.c1(-c2cn(C3CC4(C(=O)N)C3C4)nn2)ccncc1 70536,C1(NC(C2CC(NC(c3ccoc3)=O)C2)=O)CCCC(O)CC1 70537,CC(C)(CCCO)CN=c1[nH]c(=NCc2ccc(C(F)(F)F)s2)c2sccc2[nH]1 70538,c1(C(=O)NCC2(NC(C3CCS(=O)(=O)CC3)=O)CCC2)[nH]c2ccccc2c1Cl 70539,CCCC(C(=O)NCCC1CCN(C(c2coc(S(C)(=O)=O)c2)=O)C1)S(N)(=O)=O 70540,c1(CN(C(=O)NC2CCC(C)(CC)CC2)CC)cc(Br)ccc1C 70541,c1(OC)cc(C)cnc1C(=O)NC(C(C)NC(c1cnc(C2CC2)s1)=O)C(C)C 70542,C(N=c1[nH]c2cc(Cl)cc(Cl)c2o1)C1CCN(C(c2cc(C)ns2)=O)C1 70543,Cn1cnc2ccc(C(=O)NCC3CC4CC4N3C(c3cc(Cl)ccn3)=O)nc12 70544,Cn1ncc2c1CN(C(C1(C)CN(C(=O)Cc3cc(I)ccc3Br)C1)=O)C2 70545,CP(C)(=O)c1ccc(C(=O)NCC(C2CCC2)NC(c2ncccc2F)=O)cc1 70546,CC(C)(CNC(C1CC2CC1CC2O)=O)CC(=O)Nc1cccc(O)c1 70547,N1(C(C=CCNC(=O)CCC2OCCO2)=O)CC(O)CC12CCC2 70548,N1(C(CC2CN(C)CC2O)=O)CC(NC(c2ccoc2Cl)=O)C(C)(C)C1 70549,C(=O)(CC(C(C)CC)NC(=O)CCCF)NC1(C#C)CCCCC1 70550,C1(C(N2C(C(N3CCC(O)(CC(=O)OC)C3)=O)CC2)=O)C2CCC(C2)C1C 70551,c1(C(=O)NC2CC(CCC(=O)NC3(CCCC)CC3)C2)cnc(C)n1C 70552,Cc1c[nH]c(NC(C2CC2c2ccc(C(=O)NC3CONC3=O)cc2)=O)c1C 70553,N1(C(c2ccc(COC3CCSC3)cc2)C)C(=O)CCN(CC2CC2(Cl)Cl)C1=O 70554,N1(OC)CC(C)CC(C)C1.c1(CSCC(=O)N2CCC2)ccccc1C 70555,C=CCC(CNC(=O)C(C)(C)N1CCCCC1)NC(C1CN(C(C)C)C1)=O 70556,C(C(C)C(=O)NCCNC(N)=O)N(C(C(C)SCC)=O)C 70557,c1(C(=O)NCC2C(C)CCN2c2nnco2)cc(F)cc(Br)c1F 70558,C1(C(N(CCN(C(c2ccsc2)=O)CC)CC)=O)CC2(C1)CC(F)(F)C2 70559,c1(NC(C2CC=CC2)=O)ccc(O)c2c1CCCC2 70560,C(=O)(C(CNC(C1CC=CCC1)=O)C(C)(C)C)N(C(CCSC)C)C 70561,C1(OC)CC(CNC(=O)COC2CCCC(C)C2)N(C(=O)CCCSC)C1 70562,N1(C(CC2CC(OC)C2)=O)CCC2CN(C(=O)C=CI)C2C1 70563,N1(CC(=O)NCC(CO)NC(C2(COC(C)C)CC2)=O)CCS(=O)(=O)CC1 70564,N1(C(CC(CC)C)=O)CCC(C2CC2NC(c2cc(C)cc(Cl)c2)=O)CC1 70565,Cc1cccc(C(CO)NC(C2(C3CC=CCC3)CC2)=O)c1 70566,c1(OC)cc(C)c(CNC(CCCC2CC2)C(=O)O)cc1OC 70567,N1(C(CN(C2CCC2)C(C)=O)=O)CC2CCC(N(C)C)C2C1 70568,C(=O)(C1=CCCN(C(C2(COC)CCCO2)=O)C1)NC(CCCC)(C)C 70569,CCC(CC(=O)NCCCCn1cc(CC(O)C2CC2)nn1)CC(F)(F)F 70570,S(=O)(=O)(CC(=O)NCCNC(C1C2CC2C2CC12)=O)NC 70571,N1(C(C(CC)(F)F)=O)CC2CCC(C(N3CCC=CC3C(=O)OC)=O)(C2)C1 70572,C1(C(N2CC(C(N(C(CO)C3CC3)C)=O)OCC2)=O)CC(=O)NC1(C)C 70573,C(=O)(C(C)S(N)(=O)=O)N1C(CNC(c2c(C)[nH][nH]c2=N)=O)CC1 70574,c1(NCC(=O)Cc2ccncc2)ccnc(Oc2ccccc2)c1 70575,c1(C(=O)NC2CCC(CNC(C(C)c3ccco3)=O)CC2)ccn2cnnc2c1 70576,C1(C(=O)NC2CON(CC)C2=O)CC(C)(C)CCN1C(C1CCN1C)=O 70577,C1(C(N(CC(=O)NC)C)=O)CN(C(=O)CCc2ccccc2)C2(CCC2)C1 70578,c1(C(=O)NCC(CO)NC(C(C)(CO)NC(C)=O)=O)cc(Cl)c(F)cc1F 70579,c1(C(N2CC(NC(C3(C)CC4C=CC3C4)=O)C(F)CC2)=O)ccc2c[nH]nc2c1 70580,N1(C(C(C)CC2CC2)=O)CC2(C)CC1(C(=O)NCCC1(C)CCOC1)C2 70581,C(C(CC1CC1)C(=O)N1CCC1(C)CCO)NC(C1CC(N(C)C)C1)=O 70582,C=CCC(C)C(=O)NCCCC1(NC(=O)C2=CCOC2)CC1 70583,CC(C)(CCC(=O)N1CC(C(=O)NCC(c2cnc[nH]2)O)C(F)C1)[N+](=O)[O-] 70584,c1(NC(C(CC=C)CNC(C2C3CN(C)CC23)=O)=O)cnc(C)c(C)c1C 70585,c1(CC)ccccc1CC(N1CC(C)(NC(C2CC(C)CO2)=O)C1)=O 70586,C=CC(C)C(=O)NCCONC(=O)CN1CCC(C(C)C)C1 70587,c1(C(=O)NC2(C)CCN(C(=O)CCc3cnoc3)C2)nccc2ccsc12 70588,C1(C(N2CCN(CCNC(=O)C(C3CC(F)(F)C3)O)CC2)=O)CC(=O)C12CCC2 70589,C12(C(N3CC4C(CC(=O)NC5CC6(CCC6)C5)C4C3)=O)CCCC1C2(F)F 70590,CN1CCC(C)(C(N2CCC2CNC(=O)C=Cc2ccccn2)=O)CC1 70591,c1(SCC(=O)N(CCC(C)NC(C(CCSC)O)=O)C)ncnc2[nH]cnc12 70592,CCC(O)C(C)(C)C(=O)N1CCOC(CC(=O)NC2(C)CCCC2)C1 70593,c1(OC)ccc2c(c1F)CCN(Cc1cncc(Br)c1)C2 70594,c1(C(=O)NCC2CCN(C(CC=C)=O)C23CCC3)ccc2nc(N(C)C)sc2c1 70595,C1(NC(c2c(N)ccc(OCC)c2)=O)CCN(C(=O)CCSC)C12CCC2 70596,CC1CN(C(c2cc(Br)n(C)c2)=O)CC1NC(C1CC12CC(O)C2)=O 70597,C1(C)(C(=O)NC(c2cnc(C)s2)C)C=CCN1C(c1cnn(C)c1Cl)=O 70598,C(=O)(C(F)(F)C1=CCOCC1)NCC1CN(C(C2C(C=C)OCC2)=O)CC1O 70599,c1(C(N(CC(C)O)CCNC(C(C)OCC)=O)=O)cnc(CC(C)(C)C)o1 70600,C(c1ccc(F)cc1)=CC(=O)NCC1(C(=O)Nc2ccc(F)c(F)c2)CC1 70601,C(C(CO)(CO)NC(=O)CC1(C)CCC(=O)N1)N(C(=O)C=Cc1cncn1C)C 70602,CC(C#N)C(=O)NC(Cn1cccn1)C(=O)N(C)Cc1ccsc1 70603,C(C(C)CC(=O)N1CCCCO1)NC(C=C(CCC)C)=O 70604,n1(CC(N2C(CCOC)CCC2)=O)cc2ncccc2n1 70605,c1(NCCC)ccc(C(=O)NCCNC(C2CNC(=O)C2)=O)cc1 70606,C1(C2(C)CCN(C(c3c(OC)c(C(C)C)sc3)=O)C2)CCC(F)(F)CC1 70607,C1(C(=O)O)Cc2ccccc2O1.c1(C(C)(C)C)ncoc1COC 70608,CC1C(NC(C2CCCO2)=O)CCN1C(=O)Cn1ccnn1 70609,C1(CC(N2C(CNC(c3c[nH]c(=N)o3)=O)CC2)=O)CC(C2CC2)C1 70610,c1(NC(C2N(C(CCS(C)(=O)=O)=O)CC=C2)=O)ccc2nc(Cl)sc2c1 70611,c1(C(=O)NCC2N(C(CC3CCC(=O)C3)=O)CC(F)(F)C2)nc2c(s1)CCCC2 70612,N1(C2CN(C(C3C(OC)CCC3)=O)C2)CCN(C(=O)C=C2CCCCC2)CC1 70613,CC(C(=O)NCC1(CNC(=O)CCn2cncn2)CC12CCC2)S(C)(=O)=O 70614,c1(C(=O)NC2(C)CC(NC(C(C)Cc3cnc[nH]3)=O)C2)cnc2c[nH]nc2c1 70615,Cn1nc(C(N2CC(NC(=O)C(C)(C)C)C3CC23)=O)c2c1CCOC2 70616,c1(C(=O)NCC2N(C(C(CC)NC(C)=O)=O)CCCCC2)cccc2scnc12 70617,O=C(CC1=CCCCC1)NC1CCCN(C(C2COC(=O)C2)=O)CC1 70618,C1(CS(C)(=O)=O)CN(C(C2CCCCCCC2)=O)CCN1C(C12CC(F)(C1)C2)=O 70619,C(=O)(CC(C)(C(F)(F)F)N(C)C)N1C(CCNC(c2n(CC)cnn2)=O)CCC1 70620,C1(C)(CN(C(=O)CCCNC(C(CF)CF)=O)C)C=CCCC1 70621,C(=O)(CC(P(C)(C)=O)P(C)(C)=O)NC1CN(C(C2C(C)N(C)CC2)=O)C1 70622,N1(C(c2n(C)ncc2)C2CCCC2)CCC2OCCN(C(=O)C(O)C(F)F)C2C1 70623,C=C(Cl)C(C)(C)C(=O)NCC12CC(CC)(CN1C(c1ccc([N+](=O)[O-])s1)=O)C2 70624,Fc1cncc(CSc2nc(-c3cccc(Cl)c3)nn2CCC2CCC2)c1 70625,c1(CNC(C(=O)NCC(n2cccn2)C)=O)ccc(CN2CCNC(=O)C2)cc1 70626,CC(CC(=O)NCC(CC(=O)N1CC(N2CCCOC2=O)C1)C1CCC1)C(F)F 70627,C(=O)(C(C(C)C)C(C)C)NC1C(NC(c2c(Cl)c(C)n(C)n2)=O)CCCC1 70628,Cc1nscc1C(=O)NC1(CC(=O)N(C)CC2CCCCC2)CCC1 70629,N1(C(c2c(F)ccc(C)n2)=O)CC(C(=O)NCC2OCCC2C)C2(CCC2)C1 70630,C1(CNC(=O)CCc2ccc[nH]2)CC(CNC(=O)Cc2ccoc2)CO1 70631,C1(CNC(C2(N(C)C)CCCC2)=O)CCC(NC(=O)Cc2cnccn2)CC1 70632,c1(CC)c(C(=O)NC2(CF)CCN(C(C3CCC(CN(C)C)O3)=O)C2)cnn1C 70633,CC1(C)C2CCC(CC(=O)NCCC3(O)CCN(C(=O)COC(F)F)C3)C1C2 70634,C1(CNC(c2c(CC)cco2)=O)COC(C)(C)CN1C(c1cc(N)nc(Cl)c1)=O 70635,c1(CC)cnc(C(=O)NC2(CN3CCN(C(C4CCC(F)C4)=O)CC3)CC2)cn1 70636,c1(N(CCC(C)O)C)nc(=NC(C)CC(N)=O)[nH]c2ccccc12 70637,N1(C(C(C)OCCOC)=O)CC(NC(c2cnc(N(C)C)nc2)=O)C(C)C1 70638,c1(CN(C(C)CN2CCOCC2)C)cc(C#N)ccc1F.N12CCC(C1)OCC2=O 70639,C1(CC(N2C(CO)CC2C)=O)(OC)CN(C(=O)C=Cc2ccoc2)C1 70640,c1(N2CC(CNC(=O)Cn3nnnc3C3CC3)OCC2)ncnc2[nH]cnc12 70641,C1(C(=O)NCCNC(CCN(CCOCCOC)C)=O)CCC(C)(C)C1 70642,C1(CC)C(NC(=O)CCOC(C)CC(C)C)CCN1C(C1(c2cccs2)CC1)=O 70643,CC1(C(=O)NC(C)(CNC(c2ncccc2C2CC2)=O)C2CC2)CCOCC1 70644,c1(C(N(C2CN(C(CCC=C)=O)C2)C)=O)cccc(OC)n1 70645,C#Cc1ccc(NC(=O)C#CC(C)(C)CNC(c2cncn(C)c2=O)=O)c(C)c1 70646,c1(NC(=O)NC2C(C)C2)ccc2[nH]nc(O)c(=O)c2c1 70647,CN1CCC(C(=O)NC(C(=O)NCC2(C(C)(C)O)CC2)C2CCC2)C1=O 70648,c1(CN(C(=O)CN2CCC(F)CC2)C)ccccc1CNC(=O)CC(F)(F)F 70649,c1(CC)ccccc1CC(=O)NCC(C(C)C)NC(C1CCCC1F)=O 70650,N1(C(C=C(C)C(C)C)=O)CCC(CCNC(c2cccnc2C)=O)CC1C 70651,C1(C)(CNC(C(CC)CCOC)=O)CN(C(C23CC(C)(C2)OC3C)=O)C(C)(C)C1 70652,N1(C(c2c(C(=O)OC)csc2)=O)CCC(NC(c2coc(C(N)=O)c2)=O)C(O)C1 70653,N1(C(c2cc(CC)n(C)n2)=O)CC(NC(=O)Cc2nccn2C)C(C)(C)C1 70654,N1(C(=O)OC(C)(C)C)CC2(CCN2C(=O)CCC(c2ccc(C(N)=O)cc2)=O)C1 70655,c1(C(N2CC(C(=O)OC(C)(C)C)(COC)C2)=O)cc(S(C)(=O)=O)cc(F)c1Cl 70656,CC1(C)CC(NC(=O)C(=O)NCC(F)(F)F)CN(C(=O)C(C)(C)S(C)(=O)=O)C1 70657,c1(C(=O)NCCOCCN(C(=O)C(C2CC2)C2CC2)C)ccc(Cl)s1 70658,C(=O)(CC(C)CNC(C1COCC(C)O1)=O)NCCc1cnc(C)[nH]1 70659,C1(NC(=O)COC2CCOC2)CCC(CNC(=O)COc2ccc(Cl)nc2)CC1 70660,C1(C2CN(C(=O)CNc3ccccn3)C2)CN(C(c2ccc(CO)s2)=O)CCO1 70661,O=C1CCc2nc(N3CCN(C(c4cc(=O)cc[nH]4)=O)CC3CCO)ccc21 70662,N(C1CCc2cccnc21)C(=O)C(=O)Nc1c(OCC(F)F)cccc1F 70663,c1(C(N2CCC3C(NC(C4(F)CCCCCC4)=O)C3C2)=O)ccn2cncc2c1 70664,S(=O)(=O)(c1ccc(N(C)CCc2ccc(Cl)cc2)cc1Cl)NC(C)CCCO 70665,C1(C(N2CCC(CCNC(CCCc3nc(C)sc3)=O)C2)=O)CC2CCC(C1)C2 70666,c1(C(=O)NCC(C)NC(=O)C2=CCC2)cc(Br)c2c(c1)CCO2 70667,c1(C(N2CCC(NC(C3(CC)CC3(F)F)=O)C2)=O)nc(SC)ncc1C 70668,C1(CN(C(=O)CCc2ccccn2)C)CCCCN1C(=O)Cc1cccnc1Cl 70669,C(=O)(C(O)C(F)(F)F)NCC.C1=CC(=O)NC1(C)C 70670,CCCC(C)CC(=O)NC(CNC(c1cc(C)cnc1Cl)=O)CC(C)C 70671,C1(NC(c2c(C#C)c[nH]n2)=O)CCCCCCC1NC(=O)CCCCOC 70672,N#Cc1ccccc1C(N1CCN(C(c2ccncn2)=O)C(CC2CC2)C1)=O 70673,c1(CC(=O)NC(C2CCCN2C(=O)CC2CC2(C)C)C)cn(C)nn1 70674,C1(C2CC2)(C(=O)NC(CC(=O)OC)C2CC2)CN(C(C2C=CCC2)=O)C1 70675,C(=O)(CC(C)(O)C(F)(F)F)N1CC(C)(NC(=O)Cc2csc(Br)n2)C1 70676,c1(C(N2CCOC(CNC(c3cc(CO)[nH]n3)=O)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 70677,C1(CCNC(CN2CC(C(=O)NC3(CC)CC3)C2)=O)CCN(C(C)=O)CC1 70678,c1(C(N2C(CO)CC(NC(C=C(C)C)=O)C2)=O)cc(O)c2ccccc2c1 70679,C1(C(N(CC(F)(F)F)CCC#N)=O)CCCC2C1C2(F)F 70680,c1(C(N2CC(NC(C=CSC)=O)C(CO)CC2)=O)cnc2c(c1)NC(=O)CS2 70681,Cc1cccc2cc(C(=O)N(CC(C)(C)NC(c3occc3Br)=O)C)cnc12 70682,C=CC1(C(=O)N(CCCN(C(=O)C(C)Cc2ccncc2)C)C)CCC1 70683,c1(C(C(=O)NC2CC2)N(C)CC2CCCC2O)ccc2ccc(Br)cc2n1 70684,O=C(C1=CCCCO1)NCCCOCCNC(C1COC2(CO)CC1C2)=O 70685,C1(C(=O)NC2CCOCC2C)(CC)CCN(C(c2csnn2)=O)C1 70686,N1(CCOC)CCN(C(=O)C(C)NC(c2ccnn2C)=O)CC1C 70687,O(NC(=O)C(O)C1CC1)CC(=O)NC1(CN(C)C)CCC1 70688,C#CCCC1=C(C(=O)OCC)C(c2sccc2N)NC(=O)N1CC 70689,C1(NC(C=C(NC(C)=O)C)=O)CC2CCC(C1)N2C(=O)Cc1ccccc1O 70690,C(=O)(C(C(C)C)C(C)C)NC1CCN(C(COc2cccc(C(=O)NC)c2)=O)C1 70691,c1(C(=O)NC(CC)CNC(=O)CCCCOC)ccnc2[nH]ncc12 70692,C1(NC2Cc3ccccc3O2)CCC2CN(Cc3n(C)nc(Br)n3)C2C1O 70693,c1(C(=O)NC(CCN(C(CCSCCCC)=O)C)C)ccc2nonc2c1 70694,N1(C(C(C)C)=O)C2CCC1CC(CCNC(c1cc(Cl)ccc1OC(F)F)=O)C2 70695,C1(CNC(C2CC(OC)C2)=O)CN(C(C2CCN2C2CCCC2)=O)CCO1 70696,c1(N2CCCCC(C(C)NC(c3ccc(F)nc3F)=O)C2)ncnc2c1nnn2C 70697,C12(NC(c3n(CC)ncc3)=O)CCC(C(N3CCC(C)(O)C3)=O)(CC1)CC2 70698,CCCC(CCCNC(=O)C)NC(=O)CCCOc1sccc1-n1cnnn1 70699,c1(SCC)ccc(Cl)cc1C(=O)Nc1c(OC)cncc1OC 70700,c1(C(=O)NCCOCCN(C(C(CC#C)C)=O)C)cc2c(nn1)CCCO2 70701,Cc1cc(C(=O)NC2CCCCC2NC(C2CCC(=O)O2)=O)cc(C)c1Br 70702,Cn1cc(Br)c(C(=O)NCC2(CCNC(=O)Cn3cccn3)CC2)cc1=O 70703,Cc1cc([N+](=O)[O-])c(N2CCC(C(F)C(=O)O)C2)cc1Br 70704,C#CC1CC2(CC2)CN1C(=O)C(C(C)CC)N(C)C(c1oc(C)cc1C)=O 70705,c1(CNC(c2ccccc2Cl)c2n(CC)nnn2)ccc(Cl)nc1 70706,c1(NC(C(=O)NCC(=C)F)=O)cc(C(F)(F)F)ccc1OC 70707,c1(NC(=O)CCc2noc(-c3ccccc3)n2)cc(N2CCOC2=O)ccc1F 70708,C(=O)(C(O)CC(F)(F)F)NC1(CC(N2CCC(C(=O)OC)CC2)=O)CCC1 70709,N1(C(C(CC)C)=O)CCCN(C(=O)Cc2ccc(OC)cc2C)CC1 70710,C1(C(=O)NCC(CCOC)OC)(CNCC2CCC(CO)CC2)CCC(O)CC1 70711,C1(C(=O)NC(CN(C(c2cncn(C)c2=O)=O)CC)C)CCC(C)(C)O1 70712,C1(CC)CCC(CNC(c2ccn(C3CC3(F)F)n2)=O)CC1 70713,N1(C(CCC#CC)=O)CCC(N(C(C(=O)NC(C)(C)CC)CCC)CCO)C(O)C1 70714,N1(C(c2c(C)n[nH]c2)C(=O)NCC2CCOC2)CCC(F)(F)C2(CCOC2)C1 70715,C(CCCCC(=O)N1CCCC(C(C)NC(c2cc[n+]([O-])cc2)=O)C1)OC 70716,C1(C(=O)NCC2(CN=[N+]=[N-])CC2)CN(C(C2CCC3(CC2)CC3)=O)CC1(F)F 70717,N1(c2nccc(OC)n2)Cc2ccc(NC(c3cc(Br)c(C)s3)=O)cc2C1 70718,C1(N(C(C(=O)NC(c2noc(C)n2)COC)=O)C)CCSCC1 70719,Cc1ccc(CCC(N2CCN(C(c3nnc(O)nc3O)=O)CC2)=O)cc1Cl 70720,CN1CCCC12CCN(C(=O)CC1CN(C(c3ccc(N)c(F)n3)=O)CCO1)C2 70721,C1(C(N2C(CNC(c3cc(CC)on3)=O)CC2)=O)CCOCC12CCC2 70722,Cc1[nH]c2ncccc2c1C(N1CCN(C(=O)CC2CCCO2)C(CF)C1)=O 70723,N1(C(C(CCC)CNC(=O)C(C)(C)C2CC2)=O)CC2CN(C)CC2C1 70724,c1(SCCN2CCN(C(C3ON=C(C)C3)=O)C(C)C2)nc(C)nc2sc(C)c(C)c12 70725,c1(C(C(=O)NCC2N(C(c3nccc(CC)c3)=O)CC2)SC)cc(Cl)cc(Cl)c1 70726,N1(C(C(=O)Nc2ccccc2)=O)CC2CCNCC12.c12ccc(cc1)[nH]c2=O 70727,c12cc3nn[nH]c3cc1C(=O)N(CC)C2.C1(c2cn[nH]c2)CCCN1CCC 70728,C(=O)(CC1=CCCCC1)NC(C1CCN(CC(CC)OC)CC1)C1CCCC1 70729,Cc1cc(C(=O)NC2CCN(C(=O)C(C)(C)c3cnco3)C2)n(C2CC2)n1 70730,c12cccc(c1)NC2=O.C1(NC(C2CC2C)=O)CCCC1N.CCS(=O)(=O)NC 70731,C(=O)(C(C(C)(C)C)NC(C1(Cl)CCCCC1)=O)NCC(C1CC1)OC 70732,c1(-c2cn(C3C(C)CN(C(=O)C(F)OC(F)(F)F)C3)nn2)cc(Cl)cc(Cl)c1Br 70733,C1(N(C(c2c(OC)ccs2)=O)C)CN(C(=O)CCc2nncs2)CC1F 70734,C=Cc1cnn(C)c1C(=O)NC(C1CCN(C(=O)C(C2CCCCC2)F)CC1)C 70735,c1(OC(F)F)cccc(NC(c2nnnn2CSc2ccco2)C2CC2(C)C)c1 70736,C1(NC(c2ccc(CCC)cc2)=O)CCN(C(c2cnc(N)c(O)c2)=O)CC1F 70737,C(C1=CCSC1)(c1n(CC(=C)C)nnn1)OC.C12CC(=O)N(C1)CCS2 70738,C1(N(C)C(C2CCN(c3ncccn3)C2)=O)CC1C1CC1 70739,C1(NC(C2(CC)CN(C(C(CCCC)C)=O)C2)=O)CCCCC12CCC2 70740,C1(CNC(c2scnc2Cl)=O)CN(C(c2cn[nH]c2)=O)C2(CCOCC2)C1 70741,N1(C(C(C)(C)NC(=O)NCC)=O)CCN(C(=O)C(C)c2cccs2)C(CCC)C1 70742,c1(CC(=O)NC(CC#C)COC)nc(C)ccc1Br 70743,c1(C(N2CCC(NC(c3c(OC)csc3)=O)CC2C)=O)cc(C)cc2ccoc12 70744,c1(C(N2CCC(CC)(NC(C3CC3COC)=O)C2)=O)cc(Cl)c2[nH]c(O)nc2c1 70745,c1(C(=O)NCC(CNC(C2CCN(C(=O)NC)C2)=O)OC)cc(C)n(C(C)C)c1 70746,C1(OC)CC(NC(c2cc(C3CC3)on2)=O)CN(C(c2cc(F)cc(Cl)c2)=O)C1 70747,C(C(C)(C)C(=O)N1CCC(OC2CC2)C1)N(C(C1CC(OC)C1)=O)C 70748,C(C(=O)NCC1C2CC1N(C(c1cc(C(F)(F)F)cs1)=O)C2)(C(C)C)SC 70749,c1(CC)cccc(OCC(=O)NCCC(C)(C)NC(C2CCC(C)O2)=O)c1 70750,c1(CC)ccc(C(N2CCC(C)=C(Br)C2)C(=O)NCC(F)F)cc1C 70751,C(=O)(C(C(C)C)OC(C)=O)NCC(CN(C(C1(COC)CCC1)=O)C)O 70752,c1(C(N2C3C(NC(CCN(C(C)=O)C)=O)CC(C3)C2)=O)cn2ccc(F)cc2n1 70753,C(=O)(CC(C)(C)CCC)NCC(CCC)C(=O)N(C)CCC1CC1 70754,C(=O)(N=c1[nH]nc(N(C)CC)s1)N(CC)CC1CCNC1 70755,C1(C(CNC(C(C)(C)n2ccnn2)=O)(C)O)CCN(C(C2CCCCC2)=O)CC1 70756,C(CC(CNC(c1nncs1)=O)OCC)NC(C(C)OCC=C)=O 70757,CN1CC(NC(c2cc(CNC(c3ccc(O)nn3)=O)ccn2)=O)CC12CCC2 70758,CCCCC(CC)Nc1ccccc1Br.N12CCCC(C1)COC2=O 70759,C#Cc1cc(C(N2CCC(F)C(NC(c3cc(Br)n(C)c3)=O)C2)=O)cc(N)c1 70760,N1(C(C2(COC)CC=CC2)=O)CCC(F)(CNC(C2(COC)C=CCC2)=O)CC1 70761,c1(C(N(CC(c2cccc(O)c2)O)C)=O)cccc(OCc2cccs2)c1.O=C 70762,O=C(CCC[N+](=O)[O-])N1CCOCC(CNC(C2(c3ccccn3)CC2)=O)C1 70763,c1(C(C)C(=O)NC2CC(CC(N3CCCCC3C3CC3)=O)C2)ccc(C#N)cc1 70764,CC1CCC(CCC(N2CC(O)(CNC(=O)CC34CC(C3)C4)C2)=O)O1 70765,N1(C(c2c(CC)con2)=O)CCCC(C)(C(=O)NC2CCOC2=O)C1 70766,CCCCC(C(=O)N(CC(C)N(C)C(c1cccc2[nH]ccc12)=O)C)C(C)C 70767,c1(C(=O)NCC2C(C)CCN2C(c2ccc(F)c(F)c2)=O)cnn2c1N(C)CC2 70768,c1(C(=O)NCCN(CCC)C(c2c[nH]nc2CC)=O)c(C)csc1Cl 70769,C1(CNC(C(c2cccs2)SC)=O)CC2(CCC2)CN1C(c1ncoc1CO)=O 70770,C(=O)(CC(C)(C)C(=O)N1CC2CC(NC(c3cc(Br)no3)=O)CC2C1)OC 70771,N1(C(C=Cc2ccn(C)c2)=O)CC(NC(C2CC3(C2)CC3F)=O)CC(F)C1 70772,CC#CCCC(=O)NC1(C(N2CCOC(COC)C2)=O)CC1 70773,c1(C(N(CCN(C(=O)C(F)(F)c2cscn2)C)C)=O)ncc(C(C)(C)C)o1 70774,C1(CC)CC(NC(=O)Cn2cc(-c3csc(-c4ccc(Cl)nc4)n3)nn2)C1(C)C 70775,CCC(CC)C(F)C(=O)N(CCNC(C1CCCC(C)(C)O1)=O)CC 70776,C(CC1CCCC1)(C(=O)NCC=CCNC(c1cc(Br)co1)=O)NC(C)=O 70777,CN1C(=O)CC(c2ccccc2)C1c1ccccc1.C1(C)(CCN(C(=O)OC)CC)N=N1 70778,C1(CCC#C)CCCN(C(=O)C(C)(CO)NC(=O)C(C)N(C)C(C)=O)C1 70779,C1(C(=O)NC(C(C)C)(C)CNC(=O)CN2CCC(=O)CC2)CCCCC1(F)F 70780,C1(C(N2C(C(=O)NC(C3C(C(=O)OC)C3)C)CC(F)C2)=O)C2CCC(C2)C1C 70781,c1(CC)nc(=N)[nH]c(=NCC2(CNc3cnc(OC(C)C)cn3)CC2)[nH]1 70782,N1(CC(C)O)CCCN(C(c2c(Cl)nn(C)c2Cl)=O)CC1 70783,c1(C(N(C)CC2CCN(C(C(C)c3ccsn3)=O)C2)=O)cc(Br)n(C)n1 70784,CC(C)CC(O)CN=c1cc(NC(C)C(N)=O)nc[nH]1 70785,c1(OC(C)C)ccc(NC(c2nnnn2C2CC(F)(F)C2)(C)C2CC2)c(F)c1 70786,c1(CN(C)C(C2CN(c3ccncc3)C2)=O)ccnn1C 70787,CCC(C)C(O)C(C)C(=O)N1CCOCC1CC(=O)NCc1snnc1C 70788,CN1C(=O)OCC1C(N1CCC(F)(C(=O)NC2CC2)C1)=O 70789,N(C(=NCCC(C)C)NCC(C1CCOCC1)(F)F)Cc1c(CC)cccc1 70790,Cc1cnn(C(C)C(=O)N(C(C)CN(C)C(c2[nH]nnc2C)=O)C)c1 70791,N1(C(CC=C(C)C)=O)CCN(C(c2ccc(C(F)F)o2)=O)CC1c1cn[nH]c1 70792,C(CO)(CCCCOC(C)(C)C)OC(=O)NC(c1ccc(C2CC2)cc1)C 70793,c1(N(c2nccc(C(C)C)n2)C(C2CCCNCC2)=O)ncc2ccccc2n1 70794,Cc1cc(C(N2CCC23CN(C(=O)CCC(C)(F)F)C3)=O)c(O)c(C)c1 70795,N1(CCC(=O)NC(CSC)CC2CCCO2)CCCC(NC(=O)OC(C)(C)C)C1=O 70796,C(C(C(=O)N1CC2CC2O1)OC1CC1)NC(c1ccc(OCC)cc1)=O 70797,c1(OC)cc(C)c(C(=O)NCC2(O)CN(C(C3CCCOC3)=O)C2)cc1Cl 70798,c1(C(=O)NC(CN(C(C2(OC)CCCOC2)=O)CC)C)ccc(=N)[nH]c1 70799,Cc1cc(C)n(CC(N2CCC2CNC(c2cc(Cl)c(F)cc2N)=O)=O)c(=O)n1 70800,Cc1ncc(CCC2CC2SCCCC(=O)NC(=O)CCC2CCCO2)s1 70801,c1(C(=O)NC(CNC(C(CCC)(C)C)=O)(C)CO)cnc(O)c2cncn12 70802,CCC(C(=O)NC1CC(C)N(C(=O)Cc2cc(C)n(C)n2)C1)C(C)(C)CC 70803,c1(CC#N)ccnc(NCC2CCCC2NC(=O)CCCN2CCCC2)n1 70804,c1(N2CC(C(F)(F)F)OCC2)nc2cccc(F)c2c(=NCc2cnc(O)[nH]2)[nH]1 70805,C1(CNC(C(C#C)(C)C)=O)CN(C(=O)C(c2cc(C)oc2C)C)CCCO1 70806,C1(C)(C(=O)NC(CCOC)CNC(C2CCCC2(C)C)=O)CCCN(C)C1 70807,N=c1nc(O)c(CC(N2CCCCC(NC(c3cc(Cl)ncc3Cl)=O)C2)=O)c[nH]1 70808,c1(-c2cn(C3CC(C(N(CC(=O)NCCOC)C)=O)C3)nn2)ccc(C)cc1 70809,c1(SC)cccc(F)c1C(=O)NCC1CCC(NC(c2occc2F)=O)C1 70810,c1(NC(c2n(C)cc(NC(CSCC=C)=O)n2)=O)cc2ccccc2c(C)c1Cl 70811,O=C(C(F)(F)CO)N1CCC(N2CCN(C(=O)C=C3CCCC3)CC2)CC1 70812,CCCC(C)(C)C(=O)NCC(C)CNC(C1(c2ccc(OCC)cc2)CCC1)=O 70813,c1(NC(CC)=O)cncc(C(=O)NC2CC(CNC(=O)C(C)n3cccc3)C2)c1 70814,C(CC(=O)NC(CCC)C(=O)NC)(C(C)CC)NC(C(CCC)C)=O 70815,C1(C(N2CCC(CCC)C2)=O)COCCN1C(c1cc[nH]n1)=O 70816,C(C(=O)N(C)CC1CCSC1)(C(C)(C)C)NC(c1nc(C)c(C)s1)=O 70817,c1(C(=O)NCC2CN(C(CC(C(C)C)C)=O)C(C)(C)C2)c2c(nn1C)CCCC2 70818,c1(C(=O)NCC(CNC(c2cc(CCC)[nH]n2)=O)(C)C)ccc2oc(S)nc2c1 70819,c1(C(N2C(C(C)NC(=O)CNC=O)CCCC2)=O)cc2c(Cl)cccc2[nH]1 70820,N1(C(CCSCC(N)=O)=O)CC(C2CCCN(C(c3cc(C(F)F)[nH]n3)=O)C2)C1 70821,c1(C(=O)NCc2cc(C(=O)NCCC(COC)O)n(C)n2)ncc(F)cc1N 70822,CC1CC(CNC(=O)C=CC2CCCCCC2)CCN1C(c1nn(C)cc1Cl)=O 70823,C1(C(=O)NCCSCC(=O)NCC2C=C(C)CCC2)CC(=O)OC1(C)C 70824,c1(CCCC)ccccc1-c1ccc(C(C)N(CC)Cc2nc[nH]n2)s1 70825,CC1CN(C(=O)CCC(C)(C)NC(=O)C(C2CCCCC2)O)CC(C)C1O 70826,C(=O)(C#Cc1ccc(F)cc1F)N1C(C(=O)NCc2ccncc2)CCC1 70827,Cc1ccc(-c2cnc[nH]2)s1.C1(=O)C(NC(c2cnn(C)c2)=O)CC2(CCC2)N1 70828,C1(C(NOCCCC=C)=O)CCCCCN1C(C1(CCCF)CC1)=O 70829,C(=O)(C(O)CC(C)(C)C)NC(CNC(c1c(C)cc(OC)nc1)=O)CO 70830,c1(C(=O)NCC(C(C)C)NC(C2(OC)CC(CF)C2)=O)ncn2cc(Cl)ccc12 70831,c1(OC)ccc(Br)c(CN2CCCC2c2cc(-c3ccccc3)no2)c1 70832,N(C)(C(=NCC1CC2CC1C2)NCC(C)(C)C#N)C(COC)C 70833,C(CCCCCNC(c1sccc1C(F)F)=O)N(C(C(c1cccnc1)C)=O)C 70834,c1(C(N2CCN(C(C=CCOC)=O)C(C)CC2)=O)ccc2c(c1)C(C)CO2 70835,c1(C(=O)NCCN(C(C)C)C(C2CC2(Cl)Cl)=O)ccccc1S(=O)(=O)C(F)F 70836,CC1SCCN(C(=O)CC2CCN(C(C3(C)CCCCCC3)=O)CC2)C1C 70837,N1(C(CC(=C)Br)=O)CCC2(CCN(C(c3cccc(C(C)C)n3)=O)C2)C1 70838,c1(C(=O)NCC(C2(O)CCN(C(COCC=C)=O)C2)C)cc(N(C)C)nc(Cl)c1 70839,n1(CC(=O)NCC(CC(C)C)NC(CSCCCC)=O)cc(F)ccc1=O 70840,C1(C2CCC2)(NC(C(C2CCN(C(c3csc(O)n3)=O)C2)C)=O)CC1 70841,c1(C(N2CCN(CCN(C3CN(C(C)=O)C3)CC)CC2)=O)cnn2cccc2c1 70842,c1(NC(CCOC)=O)cccc(CNC(=O)C(=O)Nc2cccc(C)c2)c1 70843,CCCCC(C(=O)NC1CC(OCC)C1)NC(=O)Cn1cc(C#N)cn1 70844,C1(C(=O)NC)C=CC(NC(=O)C(=O)NCCOC2CC2)C1 70845,C1(C#CC(=O)NCCn2cnc(C(=O)NC(C)(C)CC(C)C)c2)(CC)COC1 70846,C(=O)(C1=Cc2cc(F)ccc2OC1)N(C(C)CN(C)C(C1CCCCCC1)=O)C 70847,C(=O)(CCC(=O)NC)Nc1ccc(SC(c2cn(-c3ccccn3)nn2)=O)cc1 70848,C1(NC(C(CC(C)C)NC(=O)CCn2cnc(=N)[nH]2)=O)CCC2CCCC1O2 70849,N1(C(CC=C)=O)CCC(NC(=O)CCc2ccc(C)nc2)C(CC)C1 70850,C1(CN(C(=O)CS(=O)(=O)N(C)C)CC)CCN(C(C2OCCOC2C)=O)CC1 70851,N1(CN2C(=O)CCN(Cc3ccn(CC)n3)C2=O)Cc2ccc(F)cc2CC1C 70852,N1(C(CC2(OC)CCC2)=O)C2CCC1C(C(N1CC(c3ccc(Cl)cc3)C1)=O)C2 70853,Cc1ccccc1C=CC(=O)NCC1CC(F)(F)CN1C(=O)C(C)OCC1CC1 70854,c1(OC)cc(CN(C(=O)C(O)C(C)C)CC(C)C)cc(I)c1OC 70855,CCCC(C)(CC)C(=O)NCC(C)(C1CC1)NC(C1CCCC1C)=O 70856,N1(C(C(=O)NCC)=O)CC(OC)CC1CNC(=O)COCc1scnc1C 70857,c1(NCC(C)NC(c2coc(C3CCOCC3)n2)=O)ccc([N+](=O)[O-])cc1C#N 70858,C1(C(=O)NCC2(O)CC(CNC(=O)CC3CCCCC3)C2)Cc2nccn2C1 70859,C1(C(=O)NC2CC(C)(NC(COC3(C#C)COC3)=O)C2)CCC(C2CC2)C1 70860,C12CCC13CCN(CC3)C(=O)Cn1cc2nn1.n1(CC=C)cccc1CC1CC1 70861,N1(C(c2nc(C)oc2C)=O)CCc2sccc2C1CNC(C12CCC1C2)=O 70862,C(C(CCC)C(=O)N(C)C(C1CCCO1)C)NC(c1c(CCC)nco1)=O 70863,Cn1ncc(Cl)c1C(=O)NC1CC(N(C)C(C2CCCN(C(=O)C3CC3)C2)=O)C1 70864,c1(CC)ccc([N+](=O)[O-])cc1C(=O)NCC=CCNC(c1cnc(C)s1)=O 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70916,c1(C(N2CC3(CCN(C(C4CCC(C)C4)=O)C3)C2)=O)c[nH]c2ncc(Br)cc12 70917,CCC(C)C(C(=O)N1CCCNC(=O)C1)NC(C1CC1(C)C(F)F)=O 70918,c1(C(CC)NC(=O)C(=O)NC(C)CCc2ccco2)ccc2c(c1)OCCO2 70919,CCC(C)(COC)C(=O)NC1CC(NC(=O)C(C)N(C)C)C(O)C1 70920,c1(C(=O)NCC(C2CCCC2)NC(CN(C2CCC2)C)=O)ccoc1Br 70921,c1(OC)cc(C(=O)NCCN(C(=O)C(C)C(C)C)C)c(C(F)F)cc1OC 70922,Cc1nn(C)c2c(NCC3CC3)nc(=NCC(C(C)C)OCC(F)Br)[nH]c12 70923,N1(Cc2nc(C)on2)CCC(O)CC1C(=O)O.n12nc(C)cc1C(=O)N1CC2C1 70924,Cc1c(C=CC(N2CCC(C(C)NC(C3CC4CC3CO4)=O)CC2)=O)cnn1C 70925,Cn1cc(C(=O)NCCCC(c2ccccc2)NC(C2(F)CCCC2)=O)nn1 70926,N1(C(C2(CC(C)C)CCCC2)=O)CCN(C(=O)Cc2cncnc2)CC1CO 70927,c1(C(N2CC(CNC(Cc3c(C)ccc(C)c3)=O)C2)=O)ccc(P(C)(C)=O)nc1 70928,c1(C(=O)NCC(CCNC(C(C)CS(C)=O)=O)(C)C)scc2c1OCCO2 70929,CC(CNC(c1cc(O)cc(F)c1)=O)C(F)C(=O)NCC1(C(C)(C)O)CC1 70930,c1(C(N(CC(C)NC(COCCC#C)=O)C)=O)ccc(C(C)=O)nc1O 70931,N(C(=NCc1ccn(C)c1)NCc1cccc(OCC(F)(F)F)n1)C(C)C1CC1 70932,N1(C(C(C)SCC)=O)CCC2(CC1)CCN(C(c1cnncc1O)=O)C2 70933,c1(OC)nc(C(=O)NC2CCC(NC(c3cc(Cl)cs3)=O)CC2)cc(O)n1 70934,N1(C(CNC(=O)OC)=O)CCCC(C)(C(C)(C)NCC(c2ccncc2)C)C1 70935,c1(CN(C(C(C)NC(CC)=O)=O)C)ccc(CNC(=O)CC(C)(C)SC)cc1 70936,Cc1nc2ccccc2n1CCC(N1CC(C)(NC(c2ccnnc2O)=O)C1)=O 70937,CCC(C)(CNC(=O)C(F)C(C)C)C(=O)N1CC(O)(C(C)C)C1 70938,C1(CC(=O)NCc2n(C)ncn2)CN(C(C2CCCC(=O)C2)=O)CCO1 70939,CCCCC(CNC(c1cnccc1N)=O)NC(c1cc(CCO)on1)=O 70940,N1(C(C2(F)CCCN(C(C3N(C)CCC3)=O)C2)=O)CCc2cc(F)ccc21 70941,CCCCC(C)N=c1cc(NCCCCCOCC)nc(C)[nH]1 70942,c1(OCCCCC)ccc(C(N2CC(C)(NC(c3cncc(C)c3)=O)C2)=O)nn1 70943,C1(C(=O)NCCC2CCC(NC(C=C(C)C(F)F)=O)C2)CCCCC1O 70944,CC(C)CC(C)C(=O)N(CC(C)(C)CNC(=O)COCc1nccn1C)C 70945,N1(C2(C(N(CC(CNC(C3(C(F)F)CC(=C)C3)=O)C)C)=O)CC2)CCCCC1=O 70946,C1(NC(C(CCOC)NC(C(CC)O)=O)=O)CC2C=CC1CC2 70947,CS(=O)(=O)C(C(=O)OC(C)(C)C)C1CN(C(=O)OCC)C1.C1CCCOC(=O)CC1 70948,c1(CN(C(C(OC)OC)=O)CCCNC(C2(C)COC2)=O)ccccc1 70949,C(=O)(CCCC(C)(F)F)NC1(CCOC)CCN(C(=O)C(C)C2(O)CCC2)C1 70950,c1(OCC(=O)NC2C3(CC(NC(COCC)=O)C3)C2)ccc(C#N)cc1Cl 70951,C1(C(N2CCC(C#CC)C2)=O)CCC2CCC1N2C(=O)C=Cc1ccccc1F 70952,C(=O)(C1=CCC2CCC1N2C(=O)CC1CCC(C)(C)O1)NCC#CC 70953,C(=O)(C#CC1CCCO1)N1CCC(OCC(=O)N(C2CC(F)(F)C2)C)C1 70954,N1(C(C=CC(C)NC(C2CC(=O)N(C)C2)=O)=O)CCc2cc(F)ccc21 70955,C#CCC(C(=O)N(C1COCC1O)C)NC(c1ccnc(C)c1)=O 70956,N1(c2n(Cc3cc(C)[nH]n3)nnn2)CCC(O)c2ccccc2C1 70957,C#CC(C)(C)C(=O)N1CCC(C(=O)NCCC(=O)NC(C)C)O1 70958,c1(NC(=O)NC2C(N(C)C)CC2)cc(CC(C)(C)C)nn1C1CC1 70959,c1(CSCC(=O)NC(CNC(C2C(C)(C(C)C)C2)=O)C)ccc(Cl)cc1 70960,C1(N(C(c2c(CC)nc[nH]2)=O)C)CCC(NC(C2CCN(C3COC3)C2)=O)CC1 70961,Cc1nn(C)c2sc(C(=O)NCCC(P(C)(C)=O)C3(Cc4ccccc4)CC3)cc12 70962,c1(C(=O)NC2CN(C(c3cc(OC)c(F)cc3)=O)C2)cn(C)cc(Br)c1=O 70963,C1(N(C(=O)CC2CCOC2)CCC)CCN(C(=O)Cc2cc[nH]n2)CC1 70964,C1(C(=O)NC2CC(C)N(C(c3cnc(C4CCOC4)s3)=O)C2)CCCC(C)(C)O1 70965,C1(NC(COCCOC)=O)CNC(=O)CN1C(=O)CC1C(=O)ON=C1C 70966,Cc1sc(O)nc1C(N1CC(F)(C(=O)NC2CCOCC2F)C1)=O 70967,N1(C(CC(=O)NCC)=O)CCC(O)(C2(NC(=O)C(C)C(C)(F)F)CC2)CC1 70968,c1(C2CCN(CC(=O)N(c3cccc(N4CCCC4)c3)C)C2)ccc(F)cc1 70969,CCC(C)C(C(=O)N1CCC(NC(=O)C(Cl)(Cl)Cl)C(O)C1)NC(=O)OC 70970,C1(OC)CN(C(c2nncs2)=O)C(C)(CNC(=O)CC=Cc2ccccc2)C1 70971,c1(C(=O)NC2CCc3n(C)cnc3C2)ccc2c(=N)[nH]cnc2c1 70972,C1(CC(=O)NC(C)CN2CCN(C(c3c[nH]c(=N)o3)=O)CC2)CCCCC1(C)C 70973,C#Cc1ccnc(C(=O)NC(CC=C)C(=O)N2CCOCC2CCO)c1 70974,C1(NC(c2c(NC)nc(C)cc2)=O)CC2CC(C1)N(C(=O)Cc1scnc1C)C2 70975,C1(C(=O)NCC(=O)OCC=C)CCCC(NC(C2(N(C)C)CC2)=O)CC1 70976,c1(C(=O)NCc2cccc(NC(CCC)=O)c2)cc2cc(C)[nH]c2cc1Cl 70977,C(CC(C)CCNC(=O)CCC1CCCO1)NC(C1N(C(C(C)C)=O)CCC1)=O 70978,C1(NC(c2c(C(C)C)occ2)=O)CCC(O)CN(C(C23CC4CC2C3C4O)=O)C1 70979,CCC(CC)C(C(=O)NC=Cc1ccc(N2CCOCC2)cc1)N1CCOCC1 70980,C(C(C(F)(F)F)n1cc(C)cn1)NC(CC)Cc1cccn1C 70981,N1(C(C(COC)C)=O)CCOC2(CCCN(C(c3ccc(CN(C)C)[nH]3)=O)C2)C1 70982,C(=O)(C(C)(C)CC(C)(C)C)N(CC(C)CNC(=O)C1=CCCC1)C 70983,C1(CC)CCC(C(N2CCC2C(C)(C)O)=O)C1.C1C(=O)N1 70984,Cc1cc(C)c(C(N2CCCC(NC(=O)C#CC3(C)CC3)CC2)=O)c(S)n1 70985,C=CCCC(C(=O)NC1CCOCC1(C)C)NC(=O)COCCN(C)C 70986,C1(C(=O)Nc2ncccc2C2CC2)CC(F)CN(C(=O)CC2CCSC2)C1 70987,C=CCC(C(=O)N1CCC1(C)CC(=O)NC1CC(C)C1O)NC(C)=O 70988,c1(CC)ccc2c(Oc3cnn4ccc(O)nc34)nccc2c1 70989,C1(NC(C2(NC(C(CCSC)O)=O)CC(F)(F)C2)=O)CCn2nccc2C1 70990,c1(C(C)C)ncc(C(N2CCC(F)(C(N3CCOC(CO)C3)=O)C2)=O)cn1 70991,C1(NC(=O)C(Cl)=CCl)C(CNC(=O)C=CCN2CCOCC2)CCC12CCC2 70992,CCCC(C)(C)C(=O)N1CC(NC(C2CC2c2cc(Cl)cc(Cl)c2)=O)CC(F)C1 70993,Cc1nsc(N)c1C(N1CCC(C(C)NC(=O)C=Cc2ccoc2)C1)=O 70994,C12(C(N3CCC(CN(C(=O)CCn4ccc(=N)[nH]4)C)C3)=O)CCCC1C2(F)F 70995,c1(C(N(CC(CC)NC(=O)C(C)COC)C)=O)cc(OC)c(OC)cc1[N+](=O)[O-] 70996,c1(CC(=O)NC(CN(C(=O)Cc2cc(C)[nH]n2)CC)C)coc2cc(C)ccc12 70997,C(=O)(CC(C)CC)NCCO.N1(C(C(c2ccccc2)OC)=O)CCC(OCCN(C)C)C1.CC 70998,Cc1cc(C2CC2)ncc1C(=O)NCC1CCC(C)CN1C(c1cnccn1)=O 70999,C1(C(N2CC3(CCN(C(C4(C)CC=CCC4)=O)C3)C2)=O)CCC2(CCOCC2)C1 71000,CC1CCN(C(C2CC23CC(O)C3)=O)CCN1C(=O)CCC1CC1(F)F 71001,N1(C(C2CCC(NC(=O)OC(C)(C)C)CC2)=O)CCC2(NC(=O)CC3CC3)CC2C1 71002,N1(C(c2nn(CC)nc2C)=O)CCC(C(N2CC(O)CC2C(N)=O)=O)C(C)(C)C1 71003,CC1C(C(=O)Nc2ccc(Cl)c(Cl)c2)CCCN1C(=O)NCC(=O)N(C)C 71004,N1(C(c2ccc(SC)o2)=O)CCCC(CC(=O)NC(c2nn[nH]n2)(C)C)C1 71005,N1(C(C(CCSC)O)=O)CCOC(C)C1C(=O)NCc1cc(C(N)=O)no1 71006,c1(C(=O)NC(CNC(c2ccc(NC(=O)OC)cc2)=O)(C)C)nn(C)c(Cl)c1Cl 71007,CCCC(CC)CC(=O)NCC1COCCN1C(=O)CN(C)CC 71008,c1(CN(C)C)ncc(C(c2nnnn2C2CC2)NCCCc2cnn(C)c2)o1 71009,N1(C(=O)C=C2CCC2)CCCC2C1CCCCN2C(=O)CCF 71010,C1(C2(O)CN(C(C3CSCCS3)=O)C2)(CNC(Cn2nnc(C)n2)=O)CC1 71011,c1(C(=O)NCC(CC)NC(=O)Cc2ccn(C)n2)cnc2c(c1)NC(=O)CS2 71012,C1(NC(=O)CCN2CCCCC2)C=CCN(C(c2ccc(Cl)o2)=O)C1.C1(N)CNC1 71013,C1(NC(c2cc(C)n(C)c2C)=O)CCC2(CC1)CC(NC(=O)C(F)(F)C(C)O)C2 71014,C(=O)(CCCOCC)NCC(C=C)O.C1(=O)C(C)N1 71015,c1(CC(N2CCCC(NC(C=C3CCN(C)C3)=O)C2)=O)csc2ccc(Cl)cc12 71016,c1(C2C(C(N3C(CCNC(CN(C)C)=O)COCC3)=O)C2)ccc(C#N)cc1 71017,N1(C(C2C(C)CC(C)O2)=O)CC2CCN(C(c3ccc(=O)n(C)c3)=O)CCC2C1 71018,Cc1scc(C(N2CC(NC(=O)C(C3CCC3)C3CCC3)C(F)C2)=O)c1C 71019,Cc1ncc(C(=O)NC(C)(C)CCNC(C2CC(C3CC3)=NO2)=O)cc1N 71020,C1(C(=O)Nc2cccc(N(C)C(C3(CCF)CCC3)=O)c2)OC(C)(C)OC1(C)C 71021,CCC(C(=O)OC)C(=O)NC(C(N1CC(C)(F)C1)=O)C1CCCC1 71022,N1(C(c2ccc(N(C)C)nc2)=O)CCOCC(C(=O)NCc2ccc(Br)s2)C1 71023,C(=O)(CCCCCNC(c1ncncc1C)=O)N1C(C(C)C)CC1 71024,C(C(F)(C(=O)NCC1CC(O)C1(C)C)C(C)C)NC(C1(OCC)CCC1)=O 71025,c1(OC)ccncc1C(N1CC(N(C(=O)CNC(=O)C(C)(C)C)C)C1)=O 71026,CC(C)CCC(O)C(=O)NCC(CC(C)C)C(=O)N1CCC1C(C)C 71027,C1(C)(C(N(CC)CC2CCC2)=O)CNC(C)(C)C1 71028,c1(NCC(CSC)(C)C)cc(=NCC(c2ccsc2)N(C)C)[nH]c(C)n1 71029,c1(C(c2cnn(C)c2)NC(C(C)NC(COC)(C)C)=O)noc(C)n1 71030,c1(C(N(CCC(N2CCC(CN(C)C)C2)=O)CC#C)=O)cn(C)ccc1=O 71031,C1(C(=O)NC2(C#C)CC2)CCN(C(=O)C(C)COC)CCO1 71032,C1(C(N2CC(F)(CNC(=O)C(CO)c3ccccc3)C2)=O)(CC)CCCC1 71033,C(=O)(C1CCOc2ccc(Cl)cc21)NC1CN(C(CC#N)=O)C2(C1)CCC2 71034,c1(CC(C)NC(c2c[nH]nc2CCNC(=O)C(F)OC(F)(F)F)=O)cccnc1 71035,C#CC1CCCC(CNC(C2CCC=CC2NC(c2nccnc2CC)=O)=O)C1 71036,C12(NC(C3C(CC)C3)=O)CC1CN(C(=O)CSCC(F)F)C2 71037,C12(CNC(C(CC)O)=O)CCC(CC1)N2C(C1CCC(=C2CCC2)CC1)=O 71038,C=CC1(CNC(=O)CC2N(C(=O)CC3CCC3C)CCC2(C)C)CCOCC1 71039,CC1(C)CC(C(=O)NCC(c2ccsc2)O)CCN1C(=O)Cc1ccon1 71040,c1(CC(=O)N(CC(=O)NC(C)COC)CC#C)ccccc1C 71041,c1(OCC(=O)NC2CC(NC(C(C(C)O)C)=O)C2)ccc(Cl)c(F)c1 71042,Cc1ccc(OCC(C)NC(=O)NC2CCN(CCCO)CC2)c(F)c1 71043,Nc1nc(C(=O)NCC2CC(F)(CNC(=O)C(F)n3cccn3)C2)ccc1O 71044,CCCC(CC(C)C)C(=O)NC1CN(C(c2c(CC)nn(C)c2C)=O)CCC1O 71045,c1(OC)ccnc(C(=O)OCc2cn(-c3ccccc3I)nn2)c1 71046,c1(C(=O)NC(CNC(c2c(CCC)cccc2)=O)C)ccnc(F)c1N 71047,Cc1csc(=O)n1CC(=O)N(C1CCN(C(C23CC(C#N)(C2)C3)=O)CC1)C 71048,C1(CC)CC(C(=O)NCCC(C)NC(c2coc3c2CSC3)=O)CCC1=O 71049,c1(C2N(C(c3ccc(=O)n(C)c3)C(=O)NCC)CCC2)c(Cl)cc(Cl)cc1Cl 71050,c1(CC)ccc(C(=O)NC(CN(C)C)C(N2CCC(C)(CC)C2)=O)cn1 71051,C(=O)(C1COc2ccccc21)NCCCN(C(C1(C)CC(F)(F)C1)=O)CC 71052,n1(CC(N2CCC(O)(CN(C(C(C)C(F)F)=O)C)C2)=O)cnc2ccccc12 71053,C(=O)(CC1=CCCCC1)N1C(C(=O)Nc2cncc(OC)c2)CSCC1 71054,C(C(=O)NCCCN(C)C)N(CCC)C(C1CC1CSC)=O 71055,CCC(C)CC(C(=O)NCC1(c2noc(C)n2)CC1)NC(=O)CSC(C)C 71056,c1(C(=O)NCCC2(NC(c3c(CC)occ3)=O)CCC2)ccc(COC)cn1 71057,N1(C(C(C)CC(C)(C)C)=O)CCC2(CCCN2C(=O)C(C2CCOCC2)O)C1 71058,CCCCCCN(CC(=O)NCC(C)(CC)NC(c1coc(SC)c1)=O)C 71059,c1(C(N)=O)ccc(Cl)nc1NC(C1CCCC1NC(c1ccnc(O)c1)=O)=O 71060,O(C1CCCc2nc(C)ncc21)C(Cc1n(CC)ccc1)=O 71061,C(=O)(C(O)C(F)(F)F)NC(c1nocc1C(=O)NCC1CCCOCC1)C 71062,c1(CNC(=O)CN2CC(CC(F)C(=O)NC3C(SC)CC3)C2)cccc(F)c1C 71063,CC1CCc2[nH]c(C(=O)NCCCN(C(=O)CC(C)(C)O)C3CCCC3)cc2C1 71064,N12CCCN(CC1)C(=O)C(C)n1cc(nn1)C2.CCCCCC(=O)NCC 71065,C1(C)(CCNC(c2c(OC)ccs2)=O)CCN(C(C2(O)CCSC2)=O)C1 71066,C1(C#N)(C(=O)NC(C(=O)NC2CN(CCC)C2)c2ccoc2)CC2CC2C1 71067,N1(C(C=NOC)=O)CCc2cc(C(N3CCC(F)C(OCCOC)C3)=O)ccc21 71068,c1(C(=O)NC2C(NC(c3ccccn3)=O)CCCC2)ccc(O)nc1Cl 71069,N1(C(C2(CC=C)CN(C(c3cc4ncccc4[nH]3)=O)C2)=O)CC2NC(=O)OC2C1 71070,C(C1C(C(=O)NCC2CN(C(=O)Cn3cnnc3)CCO2)C1(C)C)=C(C)C 71071,c1(C(=O)NC2(CNC(=O)CCc3ncc[nH]3)CCC2)cc(Cl)cc2ccncc12 71072,c1(C(=O)NCCCN(C(=O)CC2C=CS(=O)(=O)C2)CCO)ccc2cncn2c1 71073,C1(C2CC2)(NC(C(C)SCC)=O)CCN(C(c2ccc(C#N)n2C)=O)C1 71074,c1(C(N2CC(F)(C(=O)Nc3n(CC)nnn3)C2)=O)cc(Br)c(C)cc1O 71075,C(C(C)(C)CC(=O)N1CC(CC(=O)NC(c2[nH]c(C)nc2C)C)C2(CC2)C1)OC 71076,c1(CC(=O)N(CCN(C(c2cc(C)n(C3CC3)n2)=O)C)C)c(F)cccc1F 71077,N1(C(C2CC(=O)C2)=O)CCOCCC1C(=O)NOCCc1ccccc1 71078,S(=O)(=O)(c1ccc(N2CC=CCC2)c(F)c1)NCC1OCC(C)C1 71079,C(=O)(C#CC1CCCOC1)NC1CCCCN(C(CC(C)O)=O)C1 71080,C1(CC(=O)N(CC#CC)C)CCCCN1C(c1cn(C)nn1)=O 71081,c1(CNC(C(CC)C)=O)ncccc1CNC(c1cc(Br)nn1C)=O 71082,C1(CCC(=O)N(CCN(C)C)C)CN(C(=O)OC(C)(C)C)CCO1 71083,C12(C(=O)N(CCO)CC3CC3)CCC(C(F)F)(CC1)CC2.C1(C(=O)N)(C)CCCO1 71084,CC(C)(C)C(C(=O)N1CC(C#N)(c2nn[nH]n2)C1)c1ccccc1 71085,c1(C(=O)NC2(CO)CN(C(C3(F)CCCOC3)=O)C2)ccc2nccn2n1 71086,c1(C(=O)NCCCN(C(C)C)C(C2CCC3CC23)=O)ccc2c(c1)CCOC2 71087,CC(CCCNC(c1cccnn1)=O)NC(C1CCCC1c1nc[nH]n1)=O 71088,n1(CC)cnc(CNC(C2CC(N(C)C(c3coc(C)c3)=O)C2)=O)n1 71089,C(=O)(C1=CC2CCC=CCCC12)N1C2(CCN(C(=O)CSC(F)F)C2)CCC1 71090,N1(CCC)CCC(C(=O)N(CC(C)O)CCNC(=O)CCC2CCC2)CC1 71091,N1(C(C2C(CNC(CNC(CCC)=O)=O)OCC2)=O)CCOCC(C(C)C)C1 71092,c1(C(N2C3CN(C(C4C(C(C)C)C4)=O)CC2CC3)=O)ccc2c(n1)CCC(C)C2 71093,N1(C(Cc2n(C)ccn2)=O)CCCCN(C(c2cccc(O)c2)=O)C1.CC=CC#N 71094,N1(C(c2cscc2Br)C(=O)NCCCSCC)CCCC2(CCNC2=O)C1 71095,Cc1nnc2n1CCC(NC(=O)NC(C)(C)C(C)c1ccccc1)C2 71096,c1(N2CC(CC(C)NC(c3ccc(CO)nc3)=O)C2)ncc(O)cn1 71097,C1(OCC(=O)NCC2CSC2)CCN(C(C2COCOC2)=O)C1 71098,N1(C(CCN(C(C)=O)C)=O)CC2(CC(NC(=O)C(C)(C)C(C)O)CO2)C1 71099,C(=O)(C(C)Cc1cnc[nH]1)NC1C(NC(CSCCC)=O)C1 71100,C12(C(N3CCCC3)=O)CCC(n3cc(-c4cnc(C5CC5)s4)nn3)C1C2 71101,C(=O)(C(O)C(F)(F)F)N1CC2C(CNC(C(CCO)N(C)C)=O)(C2)C1 71102,CCCCC(CN(C)C(C1CC(NC(C2(OC)CCC2)=O)C1)=O)CC 71103,N1(Cc2c(OC)cccc2C)CCC2(CCN(C(=O)Cn3cccn3)C2)C1 71104,CCCC(CCC)CC(=O)NCC1CN(C(c2ccsc2CC)=O)CC12CCC2 71105,c1(OCCCNC(C2(COC)CN(C(=O)CC(O)C(C)C)C2)=O)cccc(F)c1C 71106,CN1N=C(C(=O)NC2CCCC2CNC(C2COC(C)(C)CN2)=O)CCC1=O 71107,N1(C(c2[nH]nc(OC)c2Cl)=O)CC2(CCC2NC(c2ccc(CO)cc2)=O)C1 71108,C1(C(=O)NCC(C)NC(c2c(OC)cnc(Cl)c2)=O)CCOCC12CCC2 71109,c1(C(=O)NCCCN(C(c2c(C)ccc(Cl)c2)=O)C(C)C)cc2cccnn2n1 71110,N1(C(c2[nH]n(C)c(=O)n2)=O)CC2OCCN(C(=O)CCCS(C)(=O)=O)C2C1 71111,C1(C(N2CC(C#N)C(NC(c3csc(Br)n3)=O)C2)=O)CCc2ccccc2C1 71112,C1(O)(CNC(c2cc(CCC)nn2C)=O)CCN(C(C2(Br)CC2)=O)CC1 71113,c1(CN2CCC(N(C(C(C)n3cncn3)=O)C)CC2)cccc2c1CCCC2 71114,C(=O)(C(C)(CC)CCCCC)N1CCC(N(C(C2C(C=C)CC2)=O)CC)C1 71115,CC1CCCN(C(=O)C(=O)N(C)CC2(CC(=O)C(C)(C)C3CC3)CC2)C1 71116,CCC(C)(C(=O)N1CCC(O)C(NC(=O)Cc2ccc(C)nc2)C1)C(N)=O 71117,Cc1cc(C(=O)NC2C3CCC2N(C(C2(CCN(C)C)CC2)=O)C3)ncc1CO 71118,c1(CC(N2CCC(F)(C(=O)NCC(C)(C)N(C)C)C2)=O)cc(Cl)cc(Cl)c1 71119,c1(C(N2CC(CN3CCN(C(C4C(=C)C4)=O)CC3)C2)=O)nccn2c(C)nnc12 71120,CCC(O)C(C)(C)C(=O)N(C)CCCNC(c1ncoc1CC(=O)OC)=O 71121,c1(OC)ccc(CC(=O)NC2CCC(N(C(=O)Cn3cc(Cl)cn3)C)C2)cn1 71122,Cn1c(C2CCCCC2)n[nH]c1=NC(=O)N1CCN(CC2CCCO2)CC1 71123,N(C1CCCn2ncnc21)C(C(CNC(c1ccc(CC)[nH]1)=O)OC)=O 71124,Cc1ccc(Br)c(NC(=O)CNC(C)(C)C(O)c2ccccc2)c1 71125,N1(C(C(C)Cn2cccn2)=O)CCN(C(c2ccc(Cl)cc2I)=O)CC12CC2 71126,c1(C(=O)NC2C(NC(COCCCOC)=O)C2)ccnc2c(Br)cccc12 71127,c12cc(NCC=CCNC(C(CSCCC)O)=O)ccc1OC2=O.C(C)(C)OC 71128,c1(C(=O)NCC2(C)N(C(c3cc(OC)nn3C)=O)CCC2)cc(O)nc(O)c1 71129,C1(CC(=O)NCCNC(Cc2[nH]c(=N)sc2)=O)CCCC12NC(=O)NC2=O 71130,C(C)(C)(C(C)CC(=O)NC1CC1)NC(CC(CC)OC)=O 71131,C=CCCCCCN=c1nc2scnc2c(NC(c2ccn(C)n2)C)[nH]1 71132,N1(Cc2cncc(C)c2)CCC(O)CC1C(=O)Nc1cnn(C(F)(F)F)c1 71133,C1(C(N2CCCC2(C)CNC(C2CC(C)OCC2)=O)=O)(COC)CC=CCC1 71134,c1(C(=O)NC(CCCC(=O)N(C2C(OC)COC2)C)C)cccn2ccnc12 71135,N1(C(c2c(C)nsc2)=O)CCC2CN(C(=O)C(O)CC3CCCCC3)CC12 71136,C1(NC(C2CCN(C(C)=O)C2)=O)CN(C(=O)COc2cccnc2)CC1C(F)F 71137,Cc1cc(C(=O)NC(C)C(c2ccccc2)C2CCOC2)ccc1F 71138,C1(CC=C)(NC(c2ccsn2)=O)CCN(C(=O)COCc2ncc(C)o2)C1 71139,C1(C2CCN(C(=O)C3=CS(=O)CCC3)C2)(NC(Cc2nc(CC)sc2)=O)CC1 71140,N1(C(C=CC(C)C)=O)CC(O)(C(C)NC(=O)CNC(C2CCC2)=O)C1 71141,CCCCCC(CC)C(=O)N1CC(C)CC1C(=O)NOCC1CCCCC1 71142,c1(C(COC2CCN(C(C(=O)NC(CC)(C)C)=O)C2)N(C)C)c[nH]c(C(N)=O)c1C 71143,C(=O)(C1CSc2ccccc21)N(C)CCNC(=O)COC(F)F 71144,C1(C(=O)NC(CNC(CN2CC(C)C2)=O)(C)C)CC(c2ccccn2)=NO1 71145,C#CC1(C(=O)NC2CC(C)(C)OC2=O)CCN(C(C2CCC(F)CC2)=O)C1 71146,N1(c2n(CCC#N)c(-c3cnccn3)nn2)CCC2(CCOCC2)C1 71147,Cc1ccc(C(=O)NC2CCCC2NC(c2scnc2C2CCCC2)=O)o1 71148,C1(NC(CCc2n(C)ccn2)=O)CC12CCN(C(=O)CC1CC(F)(F)C1)C2 71149,c1(C(N2CC(C3OCCN(C(c4c(C)nns4)=O)C3)C2)=O)cc(Cl)cc(Cl)n1 71150,N1(C(c2c(C)ncnc2)=O)CC(C2(NC(C3CC4(C3)CC(C)C4)=O)CC2)C1 71151,c1(-c2c(C)ccc(CO)c2)cnc2[nH]cc(C(=O)Nc3[nH]cnc3C(N)=O)c2c1 71152,CCC(C)C(O)C(=O)N1CCCC1CN(C(=O)C=Cc1ccccc1)C1CC1 71153,C1(N(C(COC(CC)CC)=O)C)CCN(C(=O)C=CC2CCOCC2)CC1 71154,Cc1ccc(C(=O)NCC2C3CN(C(c4c(C)csc4Cl)=O)CC23)c(O)n1 71155,C12(CNC(C3CN(C)CCO3)C)CCC(C)(CC1)CO2 71156,c1(C(=O)NC(C(CO)NC(c2cc(C)no2)=O)C)cnc2n1CCC(C)C2 71157,C1(CN(C=O)CC(c2cc(C)c(F)cc2)O)CCS(=O)(=O)C1(C)C 71158,Cc1cc2cc(C(=O)NC3CC4(C3)CC4C(=O)NC3CCC3)oc2cc1C 71159,C(=O)(C#CC1(c2ccccc2)COC1)NC(CC#C)C1CC1 71160,c1(C(=O)OC)ccc(C(C)=CC(=O)OCCOC2CCCC(C(F)(F)F)C2)cc1 71161,C1(CC)(NC(=O)CSS(C)(=O)=O)CCCN(C(c2cncc(OC)c2)=O)C1 71162,C(c1ccncc1)=CC(=O)N(C(C(=O)NC(CC)C)C)C1CC1 71163,N1(CCNC(C2(CCCC)CC2)=O)CCCN(C(=O)CC2CC2C(F)(F)F)CC1 71164,c1(CC)nc(C)ncc1C(=O)NCC1CCC1NC(c1ccc(COC)cc1)=O 71165,CC(C)(C(=O)NCC1CCN(C(C2(c3cccnc3)CCC2)=O)C1)C1CCCC1 71166,c1(NCC2(C)CCN(C(C3CC(CCC)OCC3)=O)C2)cc(C)nc(Cl)n1 71167,c1(CN(C2CCCCC2)CCCCC2CCCCC(F)(F)C2)cccc2c[nH]nc12 71168,c1(C(C)C)nnsc1C(C)NC(=O)N(CCCCOC(C)(C)C)C 71169,N1(C(c2occ(S(C)(=O)=O)c2)=O)CC2CCCN(C(c3n[nH]c(=N)s3)=O)C2C1 71170,c1(CCC)cccc(C(=O)NCCC2CCCCN2C(=O)C(C)NC=O)c1 71171,CCCC(C)(O)C(=O)N1CCC(C)(CC(=O)NCC2(O)CCN(C)C2)C1 71172,N1(C(=O)OC(C)(C)C)CC=CC1C(=O)NCC=CC#N.C1(CC(=O)N)CCN(C)C1 71173,C1(C(=O)NC2C(C)CN(C(=O)CCc3cncc(F)c3)C2)CCC2C(C1)C2(F)F 71174,CC(C)CC(O)C(C)C(=O)N1CC(F)(F)CC1C(=O)NC1C=CCCC1 71175,C1(C(N2CCC(OCCNC(=O)CCC3CC3)C2)=O)C(C(F)(F)F)C1[N+](=O)[O-] 71176,N1(C(c2cnc3cnccn23)C(=O)NCCC2CC2)CCc2c(Br)cccc2C1 71177,c1(CC)c(C(N2CC3C(CNC(c4n[nH]c(CC)c4Cl)=O)C3C2)=O)csc1C 71178,c1(SCC(=O)N(CC(CNC(C(C)OCC(F)(F)F)=O)C)C)ccccc1 71179,C1(CC(=O)NC2(CN(C(=O)CP(C)(C)=O)C)CC2)CCC12CCC2 71180,CCCCCCCC(C)CN=c1[nH]c(=NCC2CCOC2)[nH]c2cc[nH]c12 71181,C1(C(=O)NCC(C)(C)OCCNC(c2cnc(CC)s2)=O)(OC)CCS(=O)(=O)C1 71182,c1(C(=O)NCC(=O)N(C(CC)COC)C)ccc(C)nc1 71183,c1(CC)ncnc(N2CCSCC2CCNC(C2CCCN2C(C)C)=O)c1F 71184,Nc1c(O)ccc(Cl)c1C(=O)NCC1CCCN(C(=O)C=CC2CCC2)C1 71185,C1(C)(C(=O)NCCN(CCOC)C(c2ccc[n+]([O-])c2)=O)CNC(=O)C1 71186,C(=O)(C(F)(F)C(F)(F)OC(F)(F)F)NCCC(C)NCC.C12CC(F)(C1)NC(=O)N2 71187,Brc1ccc(C2CCN(CCCCc3nccs3)CC2)nc1 71188,O=S(=O)(c1ccc(Br)c(Cl)c1Cl)Nc1cc(C2CC2)nn1-c1ccccc1 71189,c1(OC)cc(C(=O)NC2CC2NC(C2CC3C(C2)C3(C)C)=O)cc(Cl)c1O 71190,c1(C(=O)NC2(F)CCC(OC)C2)cnc2cc(C)nn2c1C.C12(CC1)C(=O)N2 71191,C1(NC(Cc2c(C)nn(C)c2)=O)CC2CCC1N(C(c1nnc(O)nc1O)=O)C2 71192,Cn1nc(C(N2CCC(NC(=O)Cc3cnns3)C(F)C2)=O)c2c1CCSC2 71193,c1(-c2cc(C)[nH]c2)nc(CCOc2ccccc2)nn1C1CCS(=O)(=O)C1 71194,C1(C(=O)Nc2ccc(-c3cn(CCOC)nn3)cc2)CCCCC1(C)C 71195,C(CC(C)C)(C(=O)NCCc1ccn(C)n1)NC(CCC(C)SC)=O 71196,c1(OC)ncccc1S(=O)(=O)NC1(c2ccc(CO)cc2)CCOCC1 71197,N1(C(CCCNC(N)=O)=O)CC2CC1CCC2NC(C1C2C3CCC(C3)C12)=O 71198,Cc1cc(O)cc(=O)n1CC(=O)N(C)CC1CCN(C(C2C=CCC2)=O)C1 71199,n1(CCNC(CN(C(C(C)=C2CCCC2)=O)C2CC2)=O)cnc(CO)c1 71200,C(=O)(C(F)(F)Sc1cnn(C)c1)NCCOCCN(C(=O)Cc1ccn(C)n1)C 71201,C(CCN(C)C(C1(C)CS(=O)(=O)C1)=O)(C(C)C)NC(c1cn(CCC)nc1)=O 71202,c1(C(=O)NCC2N(C(CSCC)=O)C3CCC2C3)ccc(Br)c(F)c1F 71203,C(=O)(C(C(C)(C)C)NC(C1CCCCCCC1)=O)N1CC(NC(=O)NC)C1 71204,C1(NC(c2ccc(-n3cncn3)cc2)=O)CCCC(C(=O)Nc2ncc(F)s2)C1 71205,Cc1cc(C)c2nc(N3CCN(C(c4cc(C(C)C)nc(Cl)c4)=O)CC3)sc2c1 71206,Cn1c(C(=O)NCC2(c3ccccc3)CC2(F)F)cnc1Cl 71207,c1(C(=O)OC)ncccc1NC(=O)NCCCCNCC1CCOCC1N(C)C 71208,c1(C(=O)NCC2(O)CN(C(=O)Cc3cccc(Cl)c3)C2)cccc2oc(O)nc12 71209,N#CCCCCC(=O)NCCNC(C1OCCOC1c1ccccc1)=O 71210,N1(C(C(C(C)C)OC)=O)CCCC2CN(c3nc(-c4ccc(Cl)cc4)ns3)CC12 71211,C(=O)(CS(N)(=O)=O)N(C)CC1(CNC(=O)CC2(C)CC2(F)F)CC1 71212,C#CCC(C)(C(=O)NCC(C)(O)C1CCCC1)NC(=O)C1=CC(C)(C)C1 71213,C1(CNC(CC(C)C)=O)CN(C)CCN1C(=O)CCc1ccc(Br)s1 71214,C1(NC(c2cccc(OC)c2)=O)CN(C(c2cc(C)ccc2N)=O)CC2(CC2)C1 71215,c1(CN(CCOC)C(=O)NC2CCCC2n2cc(Br)cn2)ccc(Cl)c(Cl)c1 71216,N1(C(C(Cc2cn[nH]c2)NC(c2cncc(OC)c2)=O)=O)CCNC(=O)CC1C 71217,c1(C(N2CC(CN(C(C(C)OCCOC)=O)C)C2)=O)n[nH]c2c1CCCCC2 71218,C1(CC(N2CCCC2)=O)CCCN(CC(O)CC(F)(F)F)C1 71219,N1(C(c2cnc(Br)n2C)C(=O)Nc2c(C)cccc2)CCCN(C)C(=O)C1 71220,CC1CCSCCN1Cc1cccc(-c2ccc(F)cc2)c1 71221,CC(C(=O)NCCC1CN(C(=O)CCc2nncn2C)CCO1)C(F)(F)C(F)F 71222,C1(CC(=O)OCC)(NCc2sc3nccn3c2C)CCCS(=O)(=O)C1 71223,C1(CNC(C2(CC(C)=O)CC2)=O)(CNc2ccncn2)CC12CCC2 71224,CC(C)CC(C(=O)N1CCOCC1)OC(C1CC(C)OC1C)=O 71225,C(=O)(C1=CCOC1)NC(C)CC1CN(C(=O)C(C)c2cccs2)C1 71226,C1(CNC(=NCCC)NCC2CCN(S(C)(=O)=O)CC2)C2CCC(C2)C1(C)C 71227,CC(CNC(=O)C=CCN1CCCC1)(CO)NC(=O)CC1CCC(=O)C1 71228,CC(C)(C)C1=NOC(C(=O)NCCC2CCCCN2C(=O)Cc2cccnc2)C1 71229,CCCC(F)C(=O)NCC(C)NC(c1cc[nH]c1C1CC1)=O 71230,N1(C(CCc2cc(C)on2)=O)CCC2CCC(NC(=O)CCc3cnoc3)C1C2 71231,N1(C(=O)NC2C(CC=C)COC2)CCC(F)C(F)C1 71232,N1(C(=O)CCC(F)F)CCN(C(=O)CSc2cccc(F)c2)C(CO)C1 71233,c1(C(=O)NCC2N(C(C3CCCCS3)=O)CCC(C)C2)cc(S(N)(=O)=O)ccn1 71234,C1(C(=O)NCc2csnc2C)(COC)CN(C(C2CCCC2OC)=O)C1 71235,C1(CNC(C(C)(C)c2cccs2)=O)CC2(CCN(c3ncc(O)cn3)CC2)CO1 71236,C1(NC(C2CCN(C(CC)=O)C2)=O)CN(C(=O)CN2CCCCC2)CC1F 71237,Cc1c(C(=O)NCC2CC(C)N(C(c3ccoc3Cl)=O)C2)cccc1C#N 71238,C1(CNC(=O)OC(C)(C)C)CCCC(CF)C1.C12CC(C1)OC(=O)C2.CCO 71239,c1(C(=O)NC2CCCN(C(CSCC(=O)OC)=O)C2)ccc(S(N)(=O)=O)[nH]1 71240,c1(NC(=O)NC2CC(OCC(Br)=C(C)C)C2)ccc(C(F)(F)F)cc1O 71241,c1(NC(C2C(NCc3c(C#N)c(F)ccc3)CCC2)=O)c(O)cccc1[N+](=O)[O-] 71242,c1(C(N2CCC(c3c(C(=O)NCC(N)=O)cccc3)CC2)=O)ccc(Cl)c(O)c1 71243,c1(C(N2C(CN(C)CC3CCC4CC4C3)CCCC2)=O)cc2sccc2s1 71244,C1(C(N2C(C)CC(NC(c3cc4c[nH]nc4s3)=O)CC2)=O)CCCC2C1C2(F)F 71245,O=C1CCCCCN1Cc1cn(CC2C=CCN2C(C2CC(C(F)F)C2)=O)nn1 71246,N1(C(c2c(CC)occ2)=O)CC(OC)CC1C(N1CCC(O)(CN(C)C)C1)=O 71247,c1(CNCCNS(N(c2nc(C)nc(O)c2)C)(=O)=O)[nH]c2ccccc2c1Cl 71248,c1(OCC)cccc(OCC(O)CN(C2CCS(=O)(=O)C2)CC(C)CO)c1 71249,CCCC(O)CC(=O)NC(CCNC(=O)CC1CCC(C)C(C)C1)C(C)C 71250,N1(c2c(F)cnc(OCC)n2)C2CCC1CC(NC(c1cc(F)ccc1Br)=O)C2 71251,Cc1ccc(O)c(CNC(=O)CC=CCNC(C2CC3CC3C2)=O)c1 71252,N1(C(COC(C)C)=O)CCN(C(C2CCC(N(C)C)C2)=O)C(C(C)(C)C)C1 71253,N1(C(c2c(C(C)(C)C)noc2)=O)CCCC(C2CN(C(=O)C=CCF)C2)C1 71254,C1(O)(C(N2CCC(O)(CCNC(C(C)CC(F)F)=O)C2)=O)CN2CCC1CC2 71255,N1(C(c2cc(C)ns2)=O)C2CCC1CC(NC(c1cncc(N3CCCC3)c1)=O)C2 71256,c1(CC(N2CC(NC(C3N(CCC)CCCC3)=O)C2)=O)cc(Br)ccc1OC 71257,C1(N(C(C(CCOC)C)=O)C)CC2CCC(C1)N2CC1CNC(=O)C1 71258,C1(OC)(CNC(=O)C(c2cccnc2)C)CCN(C(=O)CC2CCCS2(=O)=O)C1 71259,C#Cc1cn(C)nc1C(=O)NCC(CC)NC(c1ccc(N)cc1Cl)=O 71260,C1(CC)CCC(CC(N2CCCC(N(C(=O)Cn3ccnc3C)CC)C2)=O)CC1 71261,C1(CNC(c2csnn2)=O)(CO)CCN(C(c2occc2C2CC2)=O)C1 71262,Cc1cccc2c1CCOC2C(=O)NC1CCCN(C(c2nn(C)cc2Cl)=O)C1 71263,c1(C(=O)NCC2(CN=c3cc(COC)nc[nH]3)CC2)ccc2c(c1)COCC2 71264,c1(NC(=O)NC2COCCO2)cncc(C(C2CCCCC2)=O)c1 71265,c1(C(N(C2CC(NC(=O)CP(C)(C)=O)C2)C)=O)ccc(-c2ncc[nH]2)cc1 71266,c1(C(=O)NC(CC)CN(C(=O)CC2OCCO2)C)cnc(-c2cccnc2)s1 71267,c1(C(=O)NC(C)CN(C)C(c2nocc2C2CC2)=O)ccc(P(C)(C)=O)o1 71268,C(C1CCN(C(=O)C(C)C2CCCC2)CC1)=CC(=O)NC(C=C)C 71269,CCC(O)(CN(C)C(C1CCN(C(=O)COc2cccnc2)C1C(C)C)=O)CC 71270,c1(-n2cc(CC)nn2)ccc(CCC(N2CCC(OC)C(C)(C)C2)=O)cc1C#N 71271,c1(ONC(C)=O)cccc(NC(=O)CCCc2cc(SCc3ncccn3)on2)c1 71272,N1(C(CCC(=C)Cl)=O)CCN(C(c2cccc(OCC(C)C)c2)=O)C(C)C1C 71273,N1(C(C(C)C2CC2)=O)CC2CCN(C(C34CCC(CO)(CC3)C4)=O)CCC2C1 71274,c1(NC(=O)NC(c2ccc(Cl)cc2OC)CC)ncnc2c1c(Br)nn2C 71275,c1(C2(NCc3ccc(-n4ccnn4)nc3)CC(C3C(C)C3)C2)nc(Cl)ncc1F 71276,C(c1nccs1)=CC(=O)NC1(NC(=O)CSCc2nc[nH]n2)CC1 71277,C1(C)(CNC(CS(=O)(=O)N(C)C)=O)CCCN(C(C2CCCC(C)(C)O2)=O)C1 71278,C1(C(N2CCN(C3CCN(C(C4(Cl)CC4)=O)CC3)CC2)=O)C2CS(=O)(=O)CC12 71279,C12(C(=O)Nc3nccs3)CCCN1CC(O)C2.C12CC(C)(C1)NC(=O)CN(C)C2=O 71280,CS(=O)CC(=O)N1CCCC1CCNC(c1cc(C(C)(C)O)on1)=O 71281,C1(C(=O)NCCC2(C)CCN(C(CSCC)=O)C2)CCc2nc(C)nn2C1 71282,C(=O)(CC(CC)C(C)(C)C)NC1C(CCC)CN(C(c2nnn(CC)c2C)=O)C1 71283,C1(C(C(=O)NCC(C(C)C)NC(c2cnsn2)=O)C)CCCC(F)(F)C1 71284,C1(NC(CCOCCNC(CN2CC(=O)NCC2)=O)=O)CCN2CCCC2C1 71285,C12(CN(C)C(=O)NCc3cnn(C)c3)CCCC1OCC2 71286,c1(CNC(=O)NC(C2COCCO2)C(=O)O)ccc(Br)cc1[N+](=O)[O-] 71287,n1(CC)nc(C(=O)N(C2CCCN(C(C3(CSC)CCC3)=O)C2)CCF)cc1C 71288,c1(OCC(N2CCC(C)(CNC(COCCCOC)=O)C2)=O)ccc(F)c(F)c1 71289,C(=O)(CCP(C)(C)=O)NC(C(=O)NC(C(C)C)C(=O)N(C)C)C 71290,n1(C(CC)C)nnnc1C(c1ccc(COC)o1)NCC1(F)CC(CO)C1 71291,c1(C(C(=O)N(CC(c2nccn2C)(C)OC)CC)OC)ccccc1Cl 71292,C1(CNC(=O)OC(C)(C)C)CCC2(CO1)CN(C(=O)NC(C)C(C)(F)F)C2 71293,C1(NC(C=NOC)=O)CN(C(C2CC3(CC3)C2)=O)CCC1C(F)(F)F 71294,C1(C(=O)Nc2c(C)n(C)nc2)CCN(C(=O)CCn2cccc2)CC1O 71295,c1(-n2cc(C3(CO)CCOC3)nn2)ccc(-n2cccc2)cc1 71296,c1(NC(CCC)CC)ccc(S(=O)(=O)N2CCC(CO)CC2)c(Br)c1 71297,c1(OCC)cc(C(=O)NCC(c2cccc(C)c2)NC(=O)C2=CCSC2)ccn1 71298,Cc1cc(C(N2CCCC2(C)CNC(=O)CC2CNC(=O)C2)=O)c2[nH]cnc2c1 71299,c1(C(=O)NCC(CNC(c2c(C)ncs2)=O)(C)F)c(C)nn2ccccc12 71300,CC(C)(CS(C)(=O)=O)C(=O)NCCC1(CNC(c2cc3n(n2)CCCN3)=O)CC1 71301,C=CC1CCCCN1C(C1(C)CCN(C(c2nnn(C)c2C)=O)CC1)=O 71302,Cc1noc2ncc(C(=O)NC3CC(CNC(c4cccc[n+]4[O-])=O)C3)cc12 71303,C(=O)(C(C)(C)C(O)C(C)C)N(CCC(=O)NC(CC)CC(F)(F)F)CC=C 71304,c1(NC(c2nnnn2C(C)C)(COC(C)=O)C)cc(C(C)(F)F)ccc1Cl 71305,c1(C(N(CCN(C(C(C(C=C)C)C)=O)C)C)=O)ccc2c(=N)[nH]cnc2c1 71306,Cc1cc(C(N2CCCC2CNC(=O)C(C)C(F)(F)F)=O)c(O)nn1.[nH]1cccn1 71307,CC1(C)CN(C(=O)CCCS(N)(=O)=O)CC(CNC(C2CC3(CSC3)C2)=O)O1 71308,CC1=CCC=CC1C(N1CCC(CCNC(C2CCCN2C)=O)CC1)=O 71309,N1(C(c2nc[nH]n2)CC)CCc2cc(F)c(F)cc2C1 71310,c1(C2(C(N3CC(N(C(CCOCC#C)=O)C)C3)=O)CC2)c[nH]c2cccc(F)c12 71311,C=C1CCN(C(=O)CCN=[N+]=[N-])C(C(=O)NCCC(O)CO)C1 71312,C1(NC(=O)CC2CCCCC2)CN(C(=O)C(F)n2cccn2)C2CCCCC12 71313,C1(C(=O)NCCN(CCC)C(c2cscc2C)=O)CCc2[nH]nc(O)c2C1 71314,c1(CN(C)CC2CCCN(C(c3ccc(Br)c(Br)c3)=O)C2)ccc(F)c(F)c1Cl 71315,N1(C(C)C)CCCC1CC(=O)NC1CCCC1NC(=O)C(C)(C)c1ccnn1C 71316,N1(C(C(C)(C)SC)=O)CCCOC(CNC(=O)Cn2cc(Br)c(=N)[nH]2)C1 71317,CC1(C)CC(=O)NCC1C(N1CCC(OCCNC(C2CC(=O)NC2=O)=O)C1)=O 71318,N1(C(C(c2ccccn2)C)=O)CC2CCC1CN2C(=O)CSc1cccc(Cl)c1 71319,N1(C(CC2ON=C(CC)C2)=O)CCCCCC1C(=O)NCCc1cnc(C)[nH]1 71320,C12(NC(c3ncn(CC)c3)=O)CCCC1N(CC1CCCCO1)CC2 71321,C(=O)(CC(C(F)(F)F)NC(C1CC2CC2C1)=O)N(CCCCOC)C 71322,N1(C(CC2(OC)CCC2)=O)CCC(NC(c2ccc3c(c2)CCN3)=O)C(C)(C)C1 71323,CC1CC(N(C(=O)C(c2ccoc2)NC(=O)COCCCN=[N+]=[N-])C)CCO1 71324,N1(C(c2cnnc(Cl)c2)=O)CC2(CCCN2C(c2cc(F)c(Cl)c(F)c2)=O)C1 71325,c1(CC(=O)NC2CC3(C(NC(C=CS(C)=O)=O)C3)C2)ccc2c(c1)CCC2 71326,C1(C(=O)Nc2cc(-c3cc(F)cc(F)c3)[nH]n2)CCC(O)C(O)CC1 71327,N1(C(CCC(C)(C)C)=O)CCC2(CCC2NC(c2csc(C(F)F)c2)=O)CC1 71328,C(=O)(C1CCCc2nncn21)NC1CCCCN(C(c2c(=N)[nH]cnc2)=O)C1 71329,C1(C(=O)NCc2nc(C)c(C)[nH]2)COCCN(C(C2CCC(F)CC2)=O)C1 71330,n1(CC)cnc2nc(N3CCC(C)(CC)C3)nc(NCC3CC(C(F)(F)F)C3)c12 71331,N1(C(c2cncc(C)c2)=O)CCC(C)C(N(C)C(c2cn(C3CC3)cn2)=O)C1 71332,Cc1cc(=NC2CCCc3n[nH]cc32)[nH]c(N2CCC(F)(CF)C2)n1 71333,N1(C(C2(C)CCCC2)=O)CC(NC(C2CC(CC3CC3)C2)=O)C(n2cccn2)C1 71334,C1(NC(C2CC(=O)OC2)=O)CCCN(C(c2nc(F)ccc2Cl)=O)CC1 71335,N1(C(c2cc(C)nn2C)=O)CCC(CNC(=O)C(O)CC(C)(C)C)C(F)(F)CC1 71336,c1(OC)ccc(C(=O)N(CCCCNC(C2(C3CCCO3)CCC2)=O)C)o1 71337,CCN=c1[nH]cc(C(=O)NC(C)(C)CNC(=O)Cc2ccc(OC)cc2F)s1 71338,c1(CNC(CC(C(C)C)O)=O)cnn2c1CN(C(c1c(O)cccc1F)=O)CC2 71339,C12CCC(CC1)C(=O)N(c1nnc(O)s1)C2.C1(c2cccs2)(CC)CCCC1 71340,C1(C)(NC)CN(C(=O)CCC2CCC(NC(=O)C(C)OCC(C)C)C2)C1 71341,c1(CC(C)C)nc(C(=O)NCC2CCN(C(C)(C)C)C2)c(Br)s1 71342,C1(N(C(Cc2cn(C(C)C)nc2)=O)C)CCN(C(C2COC(C)C2)=O)CC1 71343,C1(CNC(=O)CNC(C2CC23CCC3)=O)CC(C2CC2)=NO1 71344,Cc1cccc(Cl)c1C(=O)NCCC1CC(NC(c2cccc(N(C)C)n2)=O)C1 71345,c1(C(=O)NCC2OCCC(NC(C3C(C)C3)=O)C2)ccnc2c1CCC2 71346,N1(C(C(c2n(C)ccc2)=O)=O)CC2CCC2(C(=O)Nc2ccc(O)cc2Cl)C1 71347,c1(CN2CCC(C(N(CCC(=O)OC)C3CC3)=O)CC2)cc(Br)c(O)c(Br)c1 71348,Cc1ccccc1-n1nnnc1C(c1nncs1)NCC(n1cccn1)C 71349,C1(CNC(C2C(C=C(C)C)C2(C)C)=O)C2CCC1CN(C(c1cc(C)[nH]n1)=O)C2 71350,N1(C(CONC(C2OCCN(C)C2)=O)=O)CCC(O)CC1C(N)=O 71351,c1(C(=O)NC)ccc(C(=O)NC2CC2NC(c2cccc(C)c2C)=O)cc1F 71352,c1(N2C(C(=O)NCc3ccncc3)CC(O)C2)cccc(F)c1[N+](=O)[O-] 71353,C(c1ccc(F)cc1F)=CC(=O)NC(C(C)NC(=O)CC(C)(C)O)C 71354,c1(OC)ccc(C(CNC(C2CC23CC3)=O)NC(=O)C=Cc2cncs2)cc1 71355,c1(C(N2C(CNC(CCCC=C)=O)C(C)CC2)=O)cc(Br)c2ncccc2c1 71356,C1(CC)(CC)CCN1C(CCC)C(=O)NCCCC(=O)OC(C)(C)C 71357,C1(NC2(C(=O)OC)CCC2)=C2CN=C(N=N1)N2.c1(C(=O)NC)cc2ccccc2[nH]1 71358,c1(CN(C=O)Cc2c(OC)c(F)c(F)cc2)cccc2c1OC(C)(C)C2 71359,N1(C(C2(NC(CC(COC)C)=O)CCN(C)C2)=O)CC(=O)NCC12CC2 71360,C1(NC(CCC=CCC=C)=O)CCCCN(C(C23COC(CF)(C2)C3)=O)C1 71361,C1(COC)(NC(C2CCSC2)=O)CCN(C(=O)CCCSC)C1 71362,C1(C(N2CCC(F)(C(=O)NC(CC#C)C(=O)OC)C2)=O)CCCC2(CC2)C1 71363,C(=O)(CCC(=O)N1CCN(C(=O)CCC2NC(=O)NC2=O)CC1)N(CCC)CC 71364,N1(C(CCOCCN(C)C(=O)NC2CC2Cl)=O)CC(=O)N(C)C(=O)C1 71365,C(c1sc2ccccc2c1Cl)=CC(=O)NCC(O)CF 71366,N1(C(c2cc(Cl)sc2Cl)=O)CC2CCN(c3ncc4[nH]ncc4n3)C2C1 71367,C(=O)(CCC(C)C)NC1C(NC(C2(C(=O)OC)CCCO2)=O)CCC1 71368,N1(C(CCCOC)=O)CC(C(=O)NCCC(F)(F)C(C)C)CC(C)C1 71369,C1(NC(C2(C)CCC(F)(F)CC2)=O)CN(C(=O)C(N)=O)Cc2nccn2C1 71370,Cc1cnc(N)c(C(=O)NC2CCC(C)N(C(c3coc(Br)c3)=O)C2)c1 71371,C=CC1(CC(=O)NCC2CN(C(=O)C=CC(C)C)CCN2C)CCCCC1 71372,C1(C(N2C(C(C)(C)NC(CNC(CCC)=O)=O)CCC2)=O)C2CCC3C(C2)CC13 71373,Cc1ccsc1CNC(C1CCCN1C(c1ncc[nH]1)=O)=O 71374,CC1(N=c2[nH]c(Cl)c(C#N)s2)CC(NC(c2ccc3c(c2)OCCCO3)=O)C1 71375,CC1CC(NC(c2ccn(C3CC3)n2)=O)CN(C(C23CCC(CC2)CO3)=O)C1 71376,c1(OC)cc(N2CC3CC2CN3Cc2cccc(Br)c2Cl)nc(OC)n1 71377,N#CC1(C(N2CC3(CO)CC3(C(F)(F)F)C2)=O)CCCCCC1 71378,N1(C(CSCCC(C)C)=O)CCCC(O)(CNC(=O)CCC2CCCN(C)C2)C1 71379,C1(CC)(NC(=O)CC2CC2(C)C)CCN(C(c2ccc(C(N)=O)nc2)=O)CC1 71380,CCC(CN(C)C)CC(=O)NCC1(NC(C2CCN(C3CC3)C2=O)=O)CC1 71381,n1(CCC)ccc(C(=O)NC(CO)C(=O)N2CCC(n3cccn3)C2)n1 71382,c1(CC)ncc(C(N2CCOCC2CNC(c2cc(Cl)ncn2)=O)=O)cn1 71383,Cc1c[nH]c2ncnc(N(C(c3cc(Cl)ccc3Cl)=O)CC3CCNC3)c12 71384,CC(C(=O)N1CC(O)(C(C)NC(c2ccc(CN(C)C)[nH]2)=O)C1)C1=CCCC1 71385,C12CCOC1NC2=O.C(C(C)CCO)OCC(=O)NC1CC(OCC)C1 71386,n1(C2CCN(C(=O)C(O)CF)CC2)cnc2c1CCN(C(C1CC(F)C1)=O)C2 71387,C1(CNC(c2c(C)nc(O)cc2)=O)CCN(C(C2CCCN(C)C2)=O)C12CCC2 71388,CCC(CC)C(=O)NCc1cccc(C(=O)NCc2ncnn2C(C)C)n1 71389,N1(C(C(CNC(c2ncccn2)=O)CC2CC2)=O)CCCC2COCC12 71390,C12(CO)CCN(C1)C(=O)c1cnc(cn1)C(=O)N2.Cc1n[nH]cc1CO.N(C)C 71391,Cc1noc(C)c1C=CC(=O)NC1CCCN(C(c2ccn(C(F)F)n2)=O)C1 71392,C1(C2CC2)(CNC(C=C(c2cn(C)nc2)F)=O)CCN(C(c2cc(F)n[nH]2)=O)C1 71393,c1(C(=O)NCC(C2CC2)NC(C(c2ccc(N(C)C)cc2)C)=O)cc([N+](=O)[O-])n[nH]1 71394,N1(C(C2C3CCC(C3)N2C(C2CCOCC2)=O)=O)CC23CCC2(COC3)C1 71395,c1(NC(C2CN(C(c3c(Br)cnc(C)n3)=O)C2)=O)ccc(C#N)cc1I 71396,N1(C(C(CCCC)C)=O)CCCN(C(c2c(OC(C)=O)ccnc2O)=O)CCC1 71397,CCCC(CCC)CC(=O)N1CC2(NC(c3cc(CC)c(C)s3)=O)CCC1CC2 71398,c1(C(C)(C)C)ccc(CN2CCC(F)(C(=O)Nc3c(Cl)cnn3C)C2)c(F)c1 71399,c1(C(=O)NCC2C3N(C(C(C)OCCC#C)=O)C(CC3)C2)c(C)ccc(Cl)c1F 71400,CSC1=C(C(=O)N(C(C)CN(C)C(C2(C#N)CC2(C)C)=O)C)CCCC1 71401,N1(C(C=C(CC)CC)=O)CCC=C(C(=O)N2CC(Cc3ccco3)C2)C1 71402,N1(C(CCOC)C)CCN(CC(N2CCCC2CCC(C)C)=O)CC1 71403,c1(C(=O)NC2CC3(C(NC(CC4(OC)CC4)=O)C3)C2)csc2nccn12 71404,C1(CCNC(c2nscc2Br)=O)CN(C(=O)C=C2CCC2)CCO1 71405,Cc1nsc2ncc(C(N3CCC(Cc4cn(C5(C(N)=O)CC5)nn4)CC3)=O)cc12 71406,C(C(C)(C)CC(=O)N1CC=CC1(C(=O)NC(C)C(=O)OC)CN(C)C)OCC 71407,C(=O)(C1=NN(c2ccccc2)C(=O)CC1)NCC1N(C(C2ON=C(C)C2)=O)CC1 71408,c1(C(=O)NC(CNC(C(=O)NCCC(N)=O)=O)CO)cc(CN2CCCC2)on1 71409,N12CCC(C)(CC1)C2=O.C(=O)(CC(C)CN(C)C)NCC(C(C)C)CNC(C)=O 71410,N1(C(C(CCCC)=O)=O)C(CO)CCC12CCC2.C1(C)C(C)C(=O)N1 71411,C(=O)(C(C)(C)C1=CCN(C(=O)CCc2ccc3c(c2)OCCCO3)CC1)OC 71412,C1(N2CC3C(C)C3C2)CCCN(CC(=O)NCC(=O)O)C1=O 71413,c1(CC(=O)NC2CCC(C(=O)NCCc3ccc(Cl)cc3)C2)ccc(O)c(Cl)c1 71414,C(CC(C)(C)C(=O)N1CCC(O)(Cn2cc(-c3ccc(F)c(C)n3)nn2)C1)OC 71415,Cc1nc(S)nc(C)c1CCC(=O)NC(CNC(C1CC(C#N)C1)=O)CC(C)C 71416,C(CCC(=O)NC(c1ccoc1)C)(C(C)C)NC(c1cc(OC)n[nH]1)=O 71417,c1(CN(C2CCN(C(C3(CCF)CC3)=O)C2)C(C2C(CC)C2)=O)cccc(F)c1 71418,C12(C(=O)NCC(c3ccccc3)N(C(=O)Cc3ccco3)C)COCC1C2(F)F 71419,C(=O)(C(C)C(O)CC(C)C)N1C2(C(N3CCC(CCCC)C3)=O)CC2CC1 71420,C12(CNC(COCC#C)=O)CC(C(N)=O)(C1)C1(CN(C(C3CCCCS3)=O)C1)O2 71421,CCCCN=C(NCC1(COC)CCOC1)N1CC(C)(C)OC2(CCOC2)C1 71422,c1(C(=O)NC(CC)CNC(C2(CO)CCCO2)=O)cc(C)cc2c1NCCC2 71423,O(NC(=O)CCCC1CCCC1)CC(=O)NCc1cc(O)cc(F)c1 71424,C=Cc1cc(C(=O)NC(C)(CNC(C2(N(C)C)CCC2)=O)CC)cc(F)c1 71425,n1(CC(=O)NCC2CCN(C(CCC3C(C)C3)=O)C2)cnc2c(cnn2C)c1=O 71426,c1(C(=O)OC)ncc(C(=O)NCCN(C(=O)CCc2cc[nH]n2)CC(C)O)s1 71427,N1(C(c2ncccc2Br)=O)CC2CCC1CN2C(c1cccc2c1CCC2)=O 71428,c1(C(C(=O)NC2(c3nn[nH]n3)CC2)N(C)CC2CC2)cc(Cl)cc(Cl)c1 71429,Cc1noc(C)c1CC(=O)NC1CCC1NC(=O)CCC1COC(C)(C)O1 71430,C1(C(C)C)CCCC(C(=O)Nc2ccnc(-c3ccc(C(F)(F)F)cc3)c2)CC1 71431,N1(CC(C)(C)OC)CC(c2ccccc2Cl)OCC1C 71432,C(=O)(C1Cc2ccccc21)NC1CCCCN(C(Cc2cc(C)cc(F)c2)=O)C1 71433,C1(NC(CCC2(C)CCCN2C(=O)COCC2CC2)=O)Cc2nccn2C1 71434,N1(C(c2ncnc3c2CCC3)=O)CCCC2(C1)CN(C(C1CCCCS1)=O)C2 71435,N1(C(c2c(C)cno2)=O)C2CCC1C(C)C(NC(=O)C(C)(C)C)C2 71436,C1(C)(NC(C(C)N(C(=O)CC2CCOC2)C2CC2)=O)CN2CCC1CC2 71437,c1(OC)ccc(CC(C(=O)OC)NC(=S)NC2CCCN(c3ccccc3)C2)cc1 71438,C(=O)(C1(C)OCCc2ccccc21)NCCN(C(c1cnn(C)c1Cl)=O)C1CC1 71439,c1(SCC(N2CCN(C(C(=O)OC(C)(C)C)=O)CC2)=O)cc2cc[nH]c2cn1 71440,N1(C(c2cc(CC(C)C)on2)=O)CC(NC(=O)CC(C)n2cccn2)CC(C)C1 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71723,c1(NC2(C)CCN(C(=O)CCOCC(F)(F)F)CC2)ncnc2cnccc12 71724,C(=O)(C1=CCN(C(c2cc(C3CC3)no2)=O)CC1)NCCc1c(C)n[nH]c1 71725,c1(OC)ccc2ncc(C(N3CCC(CNC(c4[nH]c(C)nc4C)=O)C3)=O)n2n1 71726,Cc1cnc(NC(C2C3CCC(C3)N2C(c2cc(I)ccc2Cl)=O)=O)cc1I 71727,c1(C(C2(C(=O)O)CCN(CCN3CCNC3=O)C2)C)cccc(C#N)c1 71728,c1(N2CCC(C)S(=O)(=O)CC2)nc(=NC2CCC(CC#N)C2)[nH]c2c1CCC2 71729,C1(C(=O)NCC(CO)NC(C2CC=CC2)=O)CC2CCC1CC2(F)F 71730,c1(C(=O)NCC2(NC(C3CCC(F)(F)C3)=O)CC2)cc2cc(O)ccc2[nH]1 71731,C(C)(CNC(=O)CC1CCC(=O)CC1)(C(C)C)NC(C(CCC)N(C)C)=O 71732,C1(NC(c2c(COC)cco2)=O)(CO)CCN(C(c2[nH]cc(C)c2C)=O)C1 71733,c1(CC(=O)NC(CNC(C2(C(=O)OC)CC2)=O)C2CC2)nc(C)c(C)o1 71734,CCC(CC)CC(F)C(=O)NC(C)(CNC(C1Cc2cscc2C1)=O)CO 71735,c1(C(=O)NC(c2cn(-c3cccc(Cl)c3F)nn2)CCC)cc(Cl)c(C)cc1O 71736,C1(F)(C(NOC(C)C)=O)CCN(C(C2CC2OC(C)=O)=O)C1.C(C)(C)(C)O 71737,C1(NC(C2(CSC)CCC2)=O)CC2(CCC(NC(=O)C3=CCCCCC3)CC2)C1 71738,Cc1ncc(CC(=O)NCC2(NCC(=O)NC3CCC(CC(C)C)C3)CCC2)s1 71739,c1(NC(C(C(=O)OC)c2ccccc2)c2ccccc2)ccc2ncccn12 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71898,C(=O)(C1=CCCSC1)NCC(C)(C)CC1CN(C(CNS(CCOC)(=O)=O)=O)C1 71899,C1(C)(C(N2CC(C)(C(F)(F)F)OCC2)=O)CCNCC1(F)F 71900,CC1(C)CCCC(C(N2CCC(CF)(NC(C3CC(F)(F)C3)=O)C2)=O)C1 71901,c1(C(N(CCCNC(C(C)OCCCC)=O)C)=O)cc(C(N)=O)ccn1 71902,c1(C(c2n(CC)nnn2)NCC2COC(C(F)F)C2)ncccc1C 71903,N1(C(c2n(CC)ncn2)=O)CC2CC1CCC2NC(c1cc(C)nc(C)n1)=O 71904,N1(C(C(CC2CC2)NC(C2NC(=O)CC(C)C2)=O)=O)CCCN(C)CC1C 71905,N1(C(c2n(CC=C)ccc2)=O)CCC(C)(C)C(CNC(c2ccsc2C)=O)C1 71906,N1(C(c2cc(OC)n[nH]2)=O)CCC(n2cccn2)(NC(C2CNC(=O)C2)=O)CC1 71907,c1(NCCC)ncccc1C(=O)NC1COCC1n1cc(CCN(C)C)nn1 71908,N1(C(C(C)(C)CF)=O)C2CCCC1CN(C(C1CCc3ccnn3C1)=O)C2 71909,c1(C(=O)NCCCCC(C)NC(c2c(CC)non2)=O)c(O)cc(Cl)cc1F 71910,C12(NC(Cc3nc(C)oc3)=O)CCC1CN(C(c1ncccc1C)=O)C2 71911,c1(NCC)cccnc1C(=O)NC(C)CN(C(=O)C(C)Cc1cccc(Cl)c1)C 71912,C(=O)(CN=S(C)(C)=O)NC1(C)CCN(C(=O)CNC(C2CCOCC2)=O)C1 71913,CC1(C)C(CNC(=O)C(O)C2CC2)CCN1C(=O)CCCn1cccc1 71914,C(=O)(CCCCC#N)N1CCCC(C(C)NC(CCn2c(C)nnc2O)=O)C1 71915,c1(CNC(=O)C(F)C2CC2)cccc2c1CCN(C(c1n[nH]c(C3CC3)n1)=O)C2 71916,c1(NC(=O)OC(C)(C)C)n[nH]c2c1CN(C(c1cc(F)cs1)=O)C2 71917,c1(C(N2CC(F)(CNC(c3ccn(C4CC4)n3)=O)C2)=O)ccc(Br)cc1 71918,CC(C)(C)C(O)C(C(=O)Nc1ocnc1CC(=O)O)c1ccccc1 71919,S(=O)(=O)(c1cccc(Cl)c1)NC(c1ccc(O)cc1)C.C(CC(C)C(C)(C)CC)OC 71920,C12(CNC(CN3CC(C)(OC)C3)=O)CC1CN(C(=O)CCc1n[nH]c(=N)s1)C2 71921,C(=O)(C(C)C(C)OC1CC1)NCC.C12CCC1C(=O)NCC1(CC1)C(=O)N2 71922,N1(C(C2N(C(C)C)C(=O)CC2)=O)CC(NC(C2C(C)(C)OC2(C)C)=O)CCC1C 71923,C1(CNC(C=CC(C)(C)C)=O)CC2COCC2N1C(C1(F)CC2(CCC2)C1)=O 71924,N1(C(C(CC#C)CC#C)=O)CCC2C(C1)NC(=O)CN2C(=O)CCCC(C)CC 71925,c1(NCc2ccc(C#N)s2)cnc(F)cc1C(=O)Nc1cc(Br)cc(I)c1 71926,C1(CNC(C(C)O)=O)CCC12CCN(C(c1cnc3ccsc3c1)=O)CC2 71927,N1(C(C(CC)F)=O)CC2CC1CN2C(c1ncsc1Br)=O 71928,CCC(C)(C(=O)NCC1(COC)CCN(C(CC(CCC)C)=O)CC1)C(N)=O 71929,N1(C(C2CCN(C(C)C)C2=O)=O)CCC(NC(=O)C(F)=C2CCCC2)CC1C 71930,C1(CNC(COCCNC(C=CCC)=O)=O)CCC2(CCC2)CC1 71931,C1(NC(C2CCC2F)=O)C=CCC(C(=O)NC2(CF)CC2)C1 71932,N1(C(C(C)=C(CC)C)=O)CC2CC1C2CNC(C1(N2CCCC2)CCC1)=O 71933,N1(C(CC(CNC(=O)CC2CCCCC2)OC)=O)CCC(F)(C(N)=O)CC1 71934,N1(S(C)(=O)=O)CCOC(C(=O)NC2CCC(CNC(C3CC3F)=O)C2)C1 71935,C1(C#N)(C(=O)NC(CC)CN(C)C(c2cc(SC)oc2C)=O)CCCCCC1 71936,c1(C(=O)NC2C(NC(C(Cn3ccc(C)n3)C)=O)C2)cc(C)c(C)o1 71937,C1(CNC(C(N)=O)=O)CN(C(c2ccc(-c3cnc[nH]3)cc2)=O)C2CCN1C2 71938,c1(C(=O)NC2C3CN(C(c4cc(C)c(C)s4)=O)CC2C3)cn2c(n1)CCC(C)C2 71939,c1(C(=O)NCCC(C)NC(=O)CC2CCCC3CC23)ccc(-c2ncc[nH]2)nc1 71940,N1(C(=O)C2=CCCS2)CCC2CCCC(C1)N2C(C1CCc2ccccc2C1)=O 71941,C1(NC(C2(C(N)=O)CN(C(=O)CC(=O)NC3CC3)C2)=O)CCC(C2CC2)C1 71942,O=C(C1CCCc2nccn21)NC1CC1C1CCN(C(=O)C=C2CCC2)CC1 71943,c1(OC(C)C)nc(F)ccc1-c1cc(NC(=O)C(C)(C)CCl)ccn1 71944,Cc1scc(C(=O)NCC2CCCC2NC(c2ccnc(SC3CC3)c2)=O)c1C 71945,c1(C(N2CC(C(F)(F)F)OC(C)(C)C2)C(=O)NC)cc(Cl)cc(OC)c1Br 71946,N1(C(CCC2C(C)=NOC2=O)=O)CC(NC(c2onc(C)c2C)=O)CC1(C)C 71947,Cn1cc([N+](=O)[O-])c(C(=O)NC2CC(NC(c3coc(Cl)c3)=O)C2)n1 71948,c1(C(=O)Nc2cc(C)c(OC)c(C)c2)c(C(C)=O)cc(F)cc1F 71949,N1(C(c2cc(C(C)=O)[nH]n2)=O)CC(n2cc(CN3CCCC3)nn2)CCC1(C)C 71950,c1(C(N2CC(O)(CN(C)C(C3CC=CCO3)=O)C2)=O)ccncc1N=[N+]=[N-] 71951,N1(C(C(C)CCO)=O)CC(C2CCCN(C(=O)C(C)(O)C3CC3)C2)C1 71952,N1(C(C(=O)NC(C)=O)C)CCC(NC(=O)C(c2ccc(Cl)cc2)O)CC1 71953,c1(CN2C(CC)CN(C(C3CCCN3C(C)C)=O)CC2)c(Cl)ccc(F)c1F 71954,CC(CNC(=O)CCC(N)=O)C(F)C(=O)NCCCC(C)(C)C 71955,C1(C2(O)CCN(C(=O)CCC(N)=O)CC2)(NC(c2ncc(C)nc2)=O)CC1 71956,N1(c2ccn(C)n2)CCC(N2CCOCC2c2ccccc2F)C1=O 71957,CCS(=O)(=O)CC(=O)NCC1(F)CCCN(C(c2cc(Br)ccc2Cl)=O)C1 71958,Cc1cc(CNC(=O)CC(O)CNC(C2CCOC2)=O)sc1C 71959,c1(C(=O)NCC2N(C(CN3C(=N)CCC3)=O)CCC2)ccnc(F)c1F 71960,CC(C)C(O)CC(=O)N(C(C)CCNC(=O)C(c1ccc(N)cn1)C)C 71961,c1(C(=O)NCC2CC(OC)CN2C(=O)CC=C(Cl)Cl)cc(Cl)cc(C)c1O 71962,C1(NC(c2sc(CC)c(C)c2)=O)CN(C(C2CC2C2CC2)=O)Cc2ccnn2C1 71963,CC1(CNC(C2(C(c3ccncc3)=O)CC2)=O)CCN(C(=O)C(N)=O)C1 71964,c1(C(=O)NC(CC)CNC(C2C=CCC2)=O)csc2ccc(Br)cc12 71965,CCC(O)C(F)(F)C(=O)N1CC2(CNC(c3cc(C)on3)=O)CC1CO2 71966,C1(NC(=O)C=Cc2ccccc2)CN(C(=O)C(O)CC2CC2)CCC1C(F)(F)F 71967,c1(NCC(C)NC(=O)OC)nc(N2CCOC(C)(c3ccccc3)C2)cc(C)n1 71968,C1(NC(C2(c3nc(Cl)cc(OCC)n3)CCC2)=O)CC2CCCCN2C1 71969,C(CCCCCNC(C12CC(NC(C3CC3(C)C(C)C)=O)(C1)C2)=O)OC 71970,C1(C2(C(=O)NC3C(CNC(C=CCN(CC)CC)=O)CC3)CC2)CCCOC1 71971,N1(C(c2c(C)nc(F)cc2)=O)CCC2(CC1)CCN2S(=O)(=O)c1ccc(Cl)cc1 71972,n1(CCCC)nc(COc2ccccc2)nc1-c1ccc(=O)oc1 71973,C(C(CC(C)C)C(=O)N1CCC(O)(CN(C(=O)C=CCF)C)C1)OC 71974,C(C)(CN=C(NCC(=O)NC1(C)CC1)NC1CCC1)OC 71975,C#CC1(CC(=O)N(CCC)CC2CCC(C)C2)CC(=O)C1 71976,c1(COC)nnc(N2CCOC(c3ccccn3)C2)n1Cc1occc1C 71977,N#CC1CN(C(c2ncc(F)cc2F)=O)CCN1C(c1sccc1Br)=O 71978,CC(C)C(C(=O)NCC(C)(Cn1cccn1)NC(=O)C=Cc1ccc[nH]1)NS(C)=O 71979,C1(CC=C)(C(=O)N(CC(N)=O)C)CN(C(=O)C(CC)OC)C1 71980,C(=O)(CCCCC#N)N(CCOCCNC(N)=O)C.CCCC1C(=O)N1 71981,Cc1cc(C(=O)N(C(C)CNC(=O)C(c2cccc(Cl)c2)C)C)oc1C 71982,C#CC1(C(=O)NC2CCOC(C)(C)C2C)CCN(C(=O)C(C)NC(C)(C)CC)CC1 71983,N1(C(c2c(NC)cncc2)=O)CCC2(COC(CNC(=O)C(C)CO)C2)C1 71984,c1(CNC(=NCC23CC(C)(OC2)C3)NCC2CCCCC2)cc(Cl)cnc1F 71985,C1(C(=O)NCC(C(C)O)C)N(C(=O)Cn2cncn2)CCC1(C)C 71986,C1(C(=O)NCC(CNC(C2N(C(=O)NC)CCC2)=O)O)C2CNC(=O)C12 71987,C1(C(=O)NC2(CN(C)C(c3ccc(N)cn3)=O)CC2)CCC(F)(F)CO1 71988,C#Cc1ccc(C(N2CCC(C)(C)C2CNC(C2(N(C)C)CCCC2)=O)=O)cn1 71989,c1(C(N2CCC(N(C)C(c3snc(Cl)c3Cl)=O)C2)=O)cc([N+](=O)[O-])c(F)cc1Br 71990,CC(C(=O)N1CC(CNC(C2(F)CCOCC2)=O)C1)C1OCCc2sccc21 71991,CCCCCC(=O)N(C1CCCC(NC(C2(CC)C=CCC2)=O)C1)CC 71992,c1(C(=O)NC(C(C)C)CNC(=O)CC2(C)CC2)ccccc1-c1ccccc1 71993,c1(CC(=O)NCC(CC)NC(C2(S(C)(=O)=O)CCC2)=O)cc(Cl)ccc1Cl 71994,c1(C(=O)NCC2C(C)(C)CCCN2C(=O)CS(N)(=O)=O)ccc2nc(O)[nH]c2c1 71995,N1(C(C(COC)O)=O)CCC(C)(NC(=O)COc2cccc(NC(C)=O)c2)C1 71996,c1(NC(C2CCN(C(=O)Cc3nc(Cl)cs3)C2)=O)ccc(O)cn1 71997,c1(C(=O)NC(C)(C)CC(=O)N2CCC(CCO)CC2)ccc2c(c1)CC2 71998,CC(=O)CCCCC(=O)N1CC(C(=O)NCC2CCCC(C)(C)O2)CC1(C)C 71999,c1(CN2CCCC(C(C)NC(CNC(C)=O)=O)C2)ccc(F)cc1Br 72000,c1(OC)cc(C(=O)NC2CC2NC(c2cccnc2Cl)=O)cc(OC)c1O 72001,Cc1cn2cccc(NC(C3CN(C(=O)CSc4nc[nH]n4)CCN3C)=O)c2n1 72002,c1(C(N2CCN(C(c3c(SC)nccc3)=O)C3C2C3)=O)cc2cc(F)ccc2[nH]1 72003,C12(C(=O)NCCOCCN(C)C(c3ccc(CO)s3)=O)CCOC1CCOC2 72004,C(C(=O)NC12CC(C1)N(C(=O)CCc1cccn1C)C2)(C(C)C)C1C(C)C1 72005,c1(C(N2C3CC(NC(c4occc4Br)=O)C2CC3)=O)cc2cc(F)ccc2s1 72006,Cc1nsc(NC(C2CCN2C(c2c(Cl)cccc2Br)=O)=O)c1C#N 72007,C(=O)(C(C)(C)C(C)(F)F)NC1(CNC(CCCC=C)=O)CC2CCC1C2 72008,C1(CNC(CC=C)=O)CCCCN(C(c2cnnc(C)c2)=O)CC1 72009,Cc1ccc(C(=O)NCC(C)CNC(=O)C(C2CCCCC2)F)cc1S(C)(=O)=O 72010,C1(CC(=O)NC(CCNC(C2ON=C(C)C2C)=O)(C)C)OCCCC1(C)C 72011,C#CCC(CC(=O)NCC)NC(=O)C(c1cnccn1)C1CC1 72012,C(CCC)(C(=O)NCC1C=CCN1C(c1cccc(N)n1)=O)=CCC 72013,CC12CC(CCO1)N(C(C1CC3(CCN1C(=O)C(N)=O)CC3)=O)C2 72014,C=CCC(CC)C(=O)N1CC2CC(C1)N2C(C1C=CCS1)=O 72015,C#CC1CN(C(=O)CC2CC(C)=NO2)CCN1C(c1cc(CO)[nH]n1)=O 72016,C1(NC(c2c(C)coc2)=O)CC(C)CN(C(=O)COCC2CCC2)C1 72017,C12(C(N3CCC(N(C(C=CC(CC)C)=O)C)C3)=O)CCC(CC1)C(C)(C)O2 72018,N1(C(CC(C=C)CC)=O)CC2(CCC2)CCC1CNC(=O)CSC(F)F 72019,CC1CC(C(=O)NCCOC2CCN(C(=O)Cn3ccnn3)CC2)C1(C)C 72020,c1(C(=O)Nc2ccc(CCO)cc2)cn2c(n1)CN(S(=O)(=O)CCCCl)CC2 72021,c1(C(N2CCCC(F)(CNC(=O)C3=NOCC3)C2)=O)ccc2c(c1)CCC2=O 72022,N1(CC)CCC(CNC(C2COCC2NC(C2CCCO2)=O)=O)C1 72023,c1(-c2cc(C(=O)NCCc3cccs3)sc2)cc(F)c(F)cc1O 72024,C1(OC)CC2(C1)CC(C(=O)NC1CNC(=O)CN1C(=O)COC(C)(C)C)C2 72025,CCCC(CCCO)C(=O)N1CCC(OCCNC(c2cc(O)cc(F)c2)=O)C1 72026,C1(NC(CCCC#C)=O)CS(=O)(=O)C12CCN(C(=O)C(C)CS(C)(=O)=O)CC2 72027,c1(C(=O)NCCCNC(Cc2ccn(CC)n2)=O)cc(C)oc1C(F)(F)F 72028,N1(C(CC=CC=C)=O)CCOCC(NC(=O)CN2CC=CC2)C1 72029,C#Cc1cncc(C(=O)NC2COCCC2C(=O)NCCc2cncs2)c1 72030,n1(C(C)C)c(O)nc(N2CCC(NC(c3csc(CO)n3)=O)C(CO)CC2)cc1=O 72031,c1(CC(N2C(C3CCN(C(=O)Cc4ccon4)C3)CCC2)=O)ccc(F)cn1 72032,C1(C(=O)NCCCC(C)NC(C=C(COC)C)=O)CCC(=O)N(C(C)C)C1 72033,C(C(F)(F)Cn1cc(C2COCC2O)nn1)NC(c1cccnn1)=O 72034,CC1CCC(C(=O)OC)CC1.C12CCCC1OC2=O.c1(C2C(C)N2)ccccc1 72035,S(=O)(=O)(c1cccc(F)c1F)N(C)C(c1cnn(C)c1-n1cccc1)=O 72036,N1(C(CC(C)C(F)F)=O)CCS(=O)(=O)C(CCNC(c2c(F)cccc2F)=O)C1 72037,C=CCCC(C(=O)N(CCF)CC)NC(=O)CC(C)C(F)F 72038,C(=O)(C1=C(C)Oc2ccccc2C1)N1CC(NC(CCC#CC)=O)C(OC)C1 72039,C(=O)(CS(=O)(=O)Cc1ccccn1)NCC1C(C(=O)NC2CC(O)C2)C1 72040,c1(C(=O)NCCCN(C(C2CCCN(C(C(C)C)=O)C2)=O)CC)cc(N)c(F)cn1 72041,C(=O)(CC(C)(C)c1cccs1)NCCCN(C(=O)Cn1ccnn1)C(C)C 72042,C(=O)(C1=CCCCC1)NC(CSCC)C(=O)N(C)Cc1nc(C)cs1 72043,Cc1nc(CC(C)C)sc1C(=O)NC1CCCC1C(N1CCCC1)=O.C(=O)CCF 72044,N1(C(c2c(Br)ccc(C)n2)=O)CCC2(CCN(C(C3CC3C3CC3)=O)CC2)C1 72045,C(=O)(C(C)C(F)(F)F)N1CC(C)(NC(c2c(NC(C)=O)cncc2)=O)C1 72046,C1(NC(c2nc(C)n(C)n2)=O)CCN(C(c2cc3c(s2)CCC3)=O)CC1(C)C 72047,C(CCN(C(=O)CCSc1nccn1C)C)(C(C)C)NC(c1ccc(CC)[nH]1)=O 72048,c1(C(N2C3C(CNC(C)=O)(CCCC3)CC2)=O)cc2cc(C)cc(C)c2[nH]1 72049,c1(CCC)c(C(N2CC(C(C)(C)O)(NC(=O)COCCOCC)C2)=O)nnn1C 72050,C12(CC)CCN(C1)C2.c1(CNC(=O)OC(C)(C)C)cccnc1Br 72051,C1(C(=O)NC(CC(=O)NC)(C)C)CC2(CCC2)CN1C(=O)C(C)N(C)C 72052,C12(C(=O)NCC(C)OC)COCC1CN(C(c1cc(OC)n[nH]1)=O)C2 72053,c1(C(=O)NCC2(F)CC(NC(COCC(=C)C)=O)C2)cccn(C2CCC2)c1=O 72054,Cc1cc(C(=O)NC2CC(NC(C3CC3C3CC3)=O)C2)cnc1C(F)F 72055,c1(OC)nc(C)c(C(N2CCCCC2C(=O)Nc2cnn(CCO)c2)=O)s1 72056,c1(CC)nsc(CNC(=O)C(C2(O)CCC2)NC(c2sccc2F)=O)n1 72057,Cc1cnncc1C(=O)NCC1CCCN1C(C12CC(CC(F)F)(C1)C2)=O 72058,c1(C(=O)NC2CCCCC2CNC(c2n[nH]cc2F)=O)ccc2c(c1)OCCO2 72059,N1(C(C2OCCC(NC(CC3C=NN(C)C3=O)=O)C2)=O)CC2CSCC(C2)C1 72060,C(=O)(CCC(=O)N(C1CCCCC1NC(c1nc(CC)oc1C)=O)C)NCCC 72061,N1(C(C2(C)CCN(C(C)=O)C2)=O)CCN(C(c2ccncc2Br)=O)C(C)C1 72062,C1(OC)(CNC(=O)Cc2sc(C)cc2Br)CCC(C)CC1 72063,C1(C(=O)NC(C(=O)N(CC)CC)C)CC2CCN(C3CCOC3)CC12 72064,CC(C)CC(C(=O)NCC12CC1CN(C(C1(N(C)C)CC1)=O)C2)c1ccccc1 72065,C1(c2n(CCSC)nnn2)(NCc2ccc(Cl)c(Cl)c2)CCOC2(CCOC2)C1 72066,N1(C(C2CC(O)CN2Cc2cccc(Cl)c2F)=O)CCC2(CCCO2)C1 72067,N1(C(CN(CC)CC)=O)CCC2(CC1)C(NC(=O)C#CC1CCOC1)CS2(=O)=O 72068,N1(C(CSCC=C)=O)CCCC(NC(c2ccc(CCCC)cc2)=O)C1C 72069,C1(OC)CC(CC(=O)NC23CC(NC(c4cc(C(C)(C)C)on4)=O)(C2)C3)C1(C)C 72070,N1(C(C(C)NC(C)(C)C)=O)CCN(C(=O)C=Cc2cncc(F)c2)C(CF)C1 72071,c1(OC)c(C(=O)NCCC(C(C)C)NC(C2CC=CCO2)=O)c(C)nn1C 72072,C1(NC(c2ncc(Cl)s2)=O)CCN(C(c2ccn(C(F)F)n2)=O)CC1CO 72073,C1(C(C)NC(C2CCC3CC23)=O)CN(C(c2csc(C(C)(C)C)n2)=O)CCO1 72074,CC1CC(=O)NC1C(=O)N(CCCNC(=O)CCc1cnc[nH]1)C 72075,Cn1cc(Cl)c(C(=O)NC2CC(NC(=O)CCc3cccc(NC(N)=O)c3)C2)n1 72076,N1(CC)CCCC(CN2CCC(C(=O)NCC(c3ccncc3Cl)O)CC2)C1 72077,CC#CCCCC(=O)NCCOCCC(=O)NC1(OC)CCS(=O)(=O)C1 72078,c1(C(=O)NC2C(CNC(CNC(=O)NC)=O)C2)coc(C#Cc2ccccc2)c1 72079,Cc1ccn(C)c1C(=O)NCC1CCN(C(=O)CSc2ccccc2O)C1 72080,c1(OCCOC)ccc(CNCc2cc(C(O)C(F)(F)F)ccn2)nc1 72081,CC1CC(C(=O)NCC2CCN(C(c3cc(F)ccc3O)=O)C2(C)C)=NO1 72082,N1(C(C(CN(CC)CC)F)=O)CCN(C(=O)CCOc2ccccc2)CC1 72083,Cc1c(Br)cnc(O)c1C(=O)NC(C)CNC(C1CCCC(F)C1)=O 72084,O=NN1CCCC1C(=O)NC1C=CCN(C(c2ccc(-c3cn[nH]c3)cn2)=O)C1 72085,Cc1noc(C)c1SCC(=O)NCCC1(O)CCN(C(=O)C(CO)N(C)C)C1 72086,n1(C(C)C(N2CC3(CC(CNC(=O)C(O)C(F)F)C3)C2)=O)cnc2ccccc12 72087,N1(C(c2c(CC)nns2)=O)CCOCC(F)(CNC(=O)CC2CCNC(=O)C2)C1 72088,N1(C(C2CC(=O)NC2)=O)CC2CCC1C(CNC(c1n[nH]c3c1CCOC3)=O)C2 72089,C(=O)(CCCC(=O)NC1CC(=O)N(C2CN(C(=O)Cc3cnccn3)C2)C1)OC 72090,Cc1ccc2sc(N3CCCC3CNC(=O)C(C)CF)nc2c1C 72091,c1(CC)ccc(C(C)C(=O)NCC2C(C)CCN2C(=O)Cc2n[nH]c(C)n2)cc1 72092,CCC(C)(C)CC(=O)NC1CC(F)(CNC(C2CCCCN2C2CCCC2)=O)C1 72093,C(=O)(CC(O)CNC(C1CN(C2CCC2)C1)=O)N(C1CC(F)(F)C1)C 72094,N1(C(C(C)Nc2cc(Cl)ccn2)=O)CC(NC(=O)COC2CC2)C2(CC2)C1 72095,C=Cc1ccc(C(=O)NCCN(CCC)C(c2cccn(CCF)c2=O)=O)cc1 72096,C1(C(C(N)=O)F)CCCN(Cc2ccccc2NCCO)C1 72097,c1(-c2cn(C(C(=O)NCC(CC)(C)COC)C)nn2)cccc(Br)c1F 72098,CC1CCc2ccccc2C1NCc1cc(Cl)nc2n[nH]cc12 72099,c1(C(=O)NCC2(F)CCC(CNC(CCSCC)=O)C2)cccc(Cl)c1F 72100,c1(C(C(=O)C2=CCCCC2)=O)cc(CC)cc(F)c1.CC(C)C(C)C(C)O 72101,CCCCCCC(=O)N1CCC(C(N2CC(O)C2)=O)(CO)C1 72102,C1(C(=O)NCC2CC(CF)C2)CCC(Cc2ccncc2)CC1 72103,N1(C(C(=O)NCCOc2cccc(CC)c2)=O)CC2CC2(CC)C1 72104,N1(C(C(C)NC(C)=O)=O)CC2CCC(C1)C(CNC(=O)C(C(C)C)C1CCC1)C2 72105,C(C)(CCC(=O)N1CC(OC)CC1CCNC(=O)CCc1cc(C)no1)OCC 72106,C1(C(=O)NC)CCCC1NC(=O)NCCCC1CCOC1=O 72107,c1(C(=O)OC)ccc2c(c1)C(C)(C)OC2.C12(CC1)C(O)CN2 72108,c1(C(N(C(C)CCNC(c2cnc(S)n2C)=O)C)=O)c(Cl)nc2ccccn12 72109,N1(C(C(C(C)C)C#N)=O)CCCC2(C1)CN(C(c1cc(Cl)cnn1)=O)C2 72110,CCC(F)(F)C(=O)NCCn1cc(C(=O)NCCC2CC2C)nn1 72111,Cc1ccnc(C(C)(C)C(=O)NCC(C)(C)NC(=O)CC(C)N2CCCC2=O)c1 72112,c1(OC)ccccc1SCC(C)OC(c1ncoc1-c1ccccc1F)=O 72113,N1(C(c2ccc(C)cc2)=O)CC(C(=O)N(C2CC2)CC2CC2)CC(C)(C)C1 72114,CN1CCN(C(C2(F)CCCOC2)=O)c2cnccc21 72115,C1(NC(c2ncccn2)=O)CCN(C(=O)CC23CCC(CC2)CC3)CC1F 72116,C1(CNC(c2n(CCSC)nnn2)(C)CCCl)CCCC12CCOCC2 72117,Cc1c(Br)ccc(F)c1C(=O)NC(C1CN(C(=O)C(C)(C)C#N)CCO1)C 72118,c1(CC)cc(NC(C23CC2CCN3C(c2cnn(CCOC)c2)=O)=O)cc(C)c1 72119,c1(OC)c(C)cnc(C(c2nnnn2C)NC(c2cncc(Br)c2)C2CC2)c1C 72120,c1(C(N2C(CNC(C3C(=C)CC3)=O)CCCCC2)=O)cc2c(CC)cccc2[nH]1 72121,C=CCCCC(C(=O)NCCC(F)(F)Cl)NC(C1CNC(=O)N1)=O 72122,C(=O)(C(CC(C)C)N(C)C(C1CC(SC)C1)=O)NC(COC)CCO 72123,CCCCCCC(CC)C(=O)N1CCCCNC(=O)C1C 72124,c1(C(=O)NC(CN(C(=O)C(C)Sc2ccccn2)CC)C)ccnnc1S 72125,CC(=O)CCCC(=O)N(CC(=O)N(C1CC1)Cc1ccc(C)cc1)C1CC1 72126,c1(C(N2C(CNC(CCC3CCC(=O)C3)=O)CCCC2)=O)c[nH]nc1S(N)(=O)=O 72127,C(N=c1[nH]c(=NCC2CC2(F)F)[nH]c2c1CSC2)c1ccc(N(C)C)c(F)c1 72128,c1(NC(C)C(N2CCCCC2CNC(c2ncn(C)n2)=O)=O)ccc(Cl)cc1 72129,C1(C(N(C2CC(C(N(CC(C)C)C3CC3)=O)C2)C)=O)CCC(CO)O1.C1(=O)CN1 72130,C1(COC)CCC(C)CC1n1cc(-c2nc(-c3ccc(OC)cc3)n[nH]2)nn1 72131,Cc1cc(C(N2CCN(C(=O)CC3(N(C)C)CCC3)C(C3CC3)C2)=O)cc(C)n1 72132,C1(C)(NC(CN(S(C)(=O)=O)C)=O)CC(NC(=O)Cn2ncnn2)C1 72133,N1(C(C)NCCC2c3cncc(c3)C2CC)CC(C)N(C(=O)C(C)n2cccn2)C(C)C1 72134,N1(C(CCCCN(C)C)=O)CCCC2(CCN(C(=O)COCC3CCOC3)C2)C1 72135,c1(OC)ccc2ocnc2c1CN.c1(OCCOCCO)ccc(O)cc1 72136,C(=O)(CC(F)(F)C(C)(F)F)N1CCCC(C)(CNC(C=CCCC)=O)C1 72137,C1(NC(c2cc(C)n(CC)c2C)=O)CCC2(CC1)CC2NC(=O)C1=CCCSC1 72138,N1(C(c2c(C)csc2)=O)CC2(CCCCN(C(=O)C(F)CC(C)(C)C)C2)C1 72139,N1(C(=O)OC(C)(C)C)CC(CNC(C2CC3CC2C(O)C3O)=O)N2CCC1C2 72140,Cn1nccc1C(=O)NCCC1CCN(C(c2cc(C(C)(C)C)on2)=O)C1 72141,CCC(C)C(=O)NC1CCCC1CNC(C1(C)CCC1)=O 72142,N1(C(CSCC(N)=O)=O)CCC2(CC1)CN(C(c1ccccn1)=O)CC2CO 72143,c1(SC)ncc(N)c(C(=O)N(CCNC(=O)CCc2nc[nH]n2)C2CC2)n1 72144,C1(NC(c2c(C)nc[nH]2)=O)CN(C(C2(CN(C)C)CC2)=O)CC2(CC2)C1 72145,N1(C(c2ccc(OC)c(Br)c2)=O)CC(NC(C)=O)C(C2CC2)C1 72146,N1(C(=O)NC2CCc3cc(Br)ccc3C2)CCS(=O)(=O)c2ncc(Br)cc21 72147,C1(CNC(C2C(N)CCC2)=O)CCC(NC(c2cccc(=O)o2)=O)CC1 72148,C(=O)(CCC(C)(F)F)NCC1(C)CCC(NC(c2cn(C)nc2C2CC2)=O)C1 72149,C1(C(N2CCC(COCC)C2)=O)CC12CCN(C(C1(O)COC1)=O)CC2 72150,n1(CC(=O)OCC)ccc2c(NC(=O)Cc3cnc(Cl)c(C)c3)cccc12 72151,N1(C(C(CC=C)OC)=O)CC2(CC(CN(C)C(C3CCCO3)=O)C2)C1 72152,C1(NC(N2CCOC(c3c(F)cc(F)cc3F)C2)=O)CC2CCC(C1)C2O 72153,C12(C(=O)NCC(COC)(C)C)CCCC1CCN2C(=O)CCN1CCCCC1 72154,c1(OCCC)ccc(C(=O)NC2CC(NC(=O)C(C)(C)CF)C2)c(OC(C)=O)c1 72155,C1(CC)(NC(c2cc(C(F)(F)F)[nH]c2C)=O)CCN(C(C2CC(C)CO2)=O)CC1 72156,c1(C(=O)NC2CCN(C(c3c(C)cc(Cl)cc3)=O)C2C)cnc2c(c1)nnn2C 72157,c1(OC)cncnc1C(=O)NCC1CCC(NC(c2ccc(C3CC3)cc2)=O)C1 72158,Cc1ccc(OCCC(=O)NCC2CN(C(C3CCC(C)(C)CO3)=O)C2)c(Cl)c1 72159,C1(C2CCN(C(=O)COCCN(C)C)C2)(NC(CCCC)=O)CC1 72160,CCC(CCCC(F)(F)F)NC(=O)C(=O)NC1CCS(=O)(=O)CC1 72161,c1(N2CCCC3(CC(=O)NC3)C2)nc2c(c(=NCC3CC34CC4(F)F)[nH]1)COC2 72162,C(=O)(C1=CCC(NC(=O)C#CC2CC2)C1)Nc1cccc(C(C)F)c1 72163,CC(C)(F)C(=O)NC1CCCC1CNC(c1cn(CCF)nn1)=O 72164,c1(C(=O)NC(CCC)CCCNC(=O)CC(C)(C)O)ccc(F)c(C)c1C#N 72165,Cc1ccc(NC(c2n[nH]cc2NS(=O)(=O)C(F)(F)F)=O)c(C)c1 72166,C(C(=O)N(CCCNC(=O)C(F)=C1CCC1)C1CC1)(C(C)C)OC 72167,C=CCCCCCCCCC(C(=O)NCCC)N1C2CCCC1CC(O)C2 72168,Cc1cc(=NC2CCC(N3CCOCC3)C2)[nH]c(=NCC2COC(C)(C)C2)[nH]1 72169,CC(C)C(CC(=O)NC1(CCNC(=O)CCc2ncc[nH]2)CC1)C(C)C 72170,C(c1cccc(C)c1)=NC(C1(CCOC)N(C(n2cnnc2CC)=O)CCC1)=O 72171,C1(CNC(C(C(C)C)OC)=O)CCN(C(c2ccc(Cl)c(O)c2)=O)C12CC2 72172,CC1CN(C(c2ccc(-c3cccc(Br)c3)n2C)=O)CCC1O 72173,c1(C(=O)NC2CN(C(C(C(=C)C)(C)C)=O)CC2C)cc(C)cc([N+](=O)[O-])c1N 72174,c1(CNC(C(COC)N(C)C)=O)cccc(C(N2CCC(c3ncc[nH]3)C2)=O)n1 72175,c1(C(c2nnnn2-c2ccc(Br)cc2)NCC=CCSC)cc(C)oc1C 72176,c1(C(N2CCC(CN(C)C(c3cc(C(F)(F)F)on3)=O)C2)=O)cccc(F)c1 72177,c1(C(=O)NC(C2CN(C(CCCOCC)=O)C2)C)cncc(C)c1C 72178,C1(CC(=O)O)CC2(C1)CN(C(=O)Nc1nscc1Br)C2 72179,Cc1cccc(NC(=O)C(=O)Nc2ccc(-n3ccnc3C)nc2)c1C 72180,C(CCCCCN=c1[nH]c(Cl)c(C#N)s1)NC(CSc1cccc(C)c1)=O 72181,N1(Cc2ccc(OCC)c(O)c2)CCC2(CC1)CC(C(=O)NC(C)CC)CO2 72182,CCCC(C(O)C(=O)NCCCc1cccnc1)NC(C1CC(O)C1)=O 72183,C1(C(=O)NC2(C(=O)NCCC(C=C)(C)C)CCCC2)CC(=O)NC(=O)C1 72184,C1(CN(CC2N(C(C(CC)NC(C)=O)=O)CCC2)CC)CCCC(NC)C1 72185,N1(C(CCc2ncn(C)c2)=O)CC2(C1)CN(C(=O)C(O)CCc1ccc[nH]1)C2 72186,c1(N2CC(NC(C3(CC#C)CC=CCC3)=O)CC3(C2)CC3)ccc([N+](=O)[O-])c(C)n1 72187,C(Br)(C(=O)N(C1CCCC1)CCCNC(c1cnc[nH]1)=O)=C(C)C 72188,C(CCCOC)(C(=O)N1CC(c2nn[nH]n2)C1)NC(CCC=C)=O 72189,N1(C(C(C)OCCC(C)C)=O)CCCC1C=CC(N1CC(O)(CCO)C1)=O 72190,N1(C(C(C)Cc2ccccn2)=O)CCN(CCNC(=O)CC2CCCCC2)CC1 72191,n1(CCC(=O)N(CCC(C(C)C)NC(C(C)SCC)=O)C)cnc(C)cc1=O 72192,c1(C(=O)NCC2CCN(C(C3(CF)CC3(F)F)=O)C2)ccc(-n2cncn2)cc1 72193,C12(NC(CNC(CNC(C)=O)=O)=O)CCC(CC1NC(=O)C=CC1CCC1)C2 72194,c1(OC)ccc(C(=O)NCC(CNC(C2CC(F)(F)C2)=O)OC)c(F)n1 72195,c1(CCC(=O)NC2CN(C(c3c(C)csc3)=O)CC2F)cccc2c1OCO2 72196,C(CCCCC(=O)NC1CC2COCC2C1)N(C(=O)CCCCCF)C 72197,Cc1ccc(C(=O)NCC(C2CCC2)NC(=O)CN2CCN(C)CC2)cc1 72198,CC1(CNC(c2cc(C3(O)COC3)on2)=O)CCCN1C(=O)C(F)CC1CC1 72199,N1(C(CCN(C(C2CCC(C)O2)=O)C)=O)CCN(C)C(=O)C1 72200,c1(CNC(c2c(C)con2)=O)ccc2c(c1)CCC2NC(=O)C(O)CCC(C)C 72201,C(=O)(C(C)CC(C)(F)F)N1CCC(N(C(=O)Cn2nc(C)n(C)c2=O)CC)CC1 72202,C1(C(=O)NC2(C)CCN(C(c3cccc(C(=O)NC)n3)=O)C2)CC(O)C12CCC2 72203,c1(CN(C(=O)NC(C)CCc2cn[nH]c2)C2CC2)nn(C)cc1Br 72204,c1(C(N2CCCC(CCC=C)C2)=O)coc2c1CN(C(=O)CC1CCCN1C)C2 72205,c1(CC(=O)NC(CN(C(C(CC)Oc2cccc(C)c2)=O)C)C)ncccc1C 72206,Cc1c(C(=O)N(C)CCNC(C2(C(=O)OC(C)(C)C)CCC2)=O)nnn1C 72207,C(=O)(C(O)CC(C)(C)C)NC(CCCNC(c1ccc(SCC)nc1)=O)(C)C 72208,C1(C)(C(=O)NC2CCC(CN(C(c3c(C)cncc3)=O)C)CC2)CCN(C)C1=O 72209,C1(COC)(CNC(=O)CC2CC2C)CCCN1C(=O)CCSC 72210,c1(CC(N2C(C(C)(C)NC(=O)CCc3cscn3)CCC2)=O)cccc2nonc12 72211,c1(CC)cccc(OCC(=O)NCC2CN(C(c3ncccc3N)=O)CC2O)c1 72212,C=CC(C)(CCOC)C(=O)NCCN(C(=O)C(c1c(C)cccc1C)O)C(C)C 72213,c1(CC)cc(C(=O)NC2CN(C(=O)COC3CCOCC3)CC2C)ccn1 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72231,c1(C(=O)OCC)nc(=NCC(C)CNC(=O)Cc2cn[nH]c2)c(F)c(Cl)[nH]1 72232,C1(NC(C=CCOC)=O)CCC12CN(C(=O)CC1(O)CCCC1)C2 72233,c1(C(N(C2CCN(Cc3ccc(Br)cc3Cl)C2)C)=O)ccc2cccc(Br)c2n1 72234,N1(C(c2cnc(C#N)s2)=O)CCC2(CC1)CC2CNC(C1(NC(N)=O)CC1)=O 72235,c1(NC(=O)N(CC(N2CCCCCC2)=O)CC2CCOC2)ncc(F)cn1 72236,c1(OCC(=O)Nc2c(F)ccc(O)c2O)ccc2ccoc2c1 72237,C(=O)(C(O)CCC(C)C)N1C(CNC(C2C(OC)CCCC2)=O)CC2CC21 72238,C1(C2(O)CCOCC2)(C(N2C3CC(NC(c4ccc(C)o4)=O)C(C3)C2)=O)CC1 72239,CCCN=C(NCCC1CN(C(C)=O)C1)N1CCC2(C1)CC2(F)F 72240,c1(C(N2CC(O)(CNC(C(C)C(F)F)=O)C2)=O)cc2c(Cl)ccnc2s1 72241,N1(C(C2CC(=O)NCC2C(F)(F)F)=O)CC2CC1CN(C(=O)COC(F)F)C2 72242,C=CCC(C(=O)N1CCOC(C)C1C(=O)N(CCCC)C)OC 72243,c1(OC(c2cccnc2)C(=O)NCC2CC3CC2C3)cc(F)ccc1F 72244,n1(CC)ncc2c1CCCC2NC(=O)C(N1C2CCC1COC2)=O 72245,c1(OC)cc(C=CC(=O)NCC2(O)CCCCCC2)ccc1OC(F)F 72246,C(C1c2ccsc2CCN1C(=O)C=C1CCC1)NC(C1CC2CCC2C1)=O 72247,N1(C(C2(CC#C)CCCO2)=O)CCC2C(C1)CN2C(=O)CCc1nc(C)c(C)o1 72248,N1(C(C2CCCC(NC(CC(C)O)=O)C2)=O)CCC(O)C(C)C1 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72370,C(=O)(CC(C)(CN(C)C)C(F)(F)F)N1CC2CN(C(CCCC(C)C)=O)CC2C1 72371,C(=O)(C1=COc2ccccc2O1)NCCC1CC(C)(C)OCC1 72372,Cc1sc(C(=O)N(C2CCN(C(=O)CCC3CCCCCC3)C2)CCO)nc1O 72373,CCC(O)C(=O)NC1(CCNC(=O)C(c2cncn2C)O)CCC1 72374,Cc1cc(=O)c(C(=O)NCC2CCCN2C(=O)C(n2cnc(C#N)n2)C)cn1C 72375,CC1CC(C(=O)CSCC(=O)N(CC(N2CC(SC(C)(C)C)C2)=O)C)CO1 72376,C(=O)(C(CC(F)F)c1ccccc1)Nc1cccc(NC(c2n(C)nnc2)=O)c1 72377,C(=O)(C1=CC(O)CCC1)NC(C)CCNC(c1c(Cl)csc1Cl)=O 72378,c1(CN(C(C(=O)NC)C2CCCC2)CC)ccc(Br)s1 72379,C1(NC(CN(C(COC)=O)C)=O)CC2CCC1N(C(c1cc(C)nnc1O)=O)C2 72380,N(C(=NCC1COCCO1)NC(CC(F)(F)F)C)Cc1ccc(C(C)C)cc1 72381,CCC(O)C(C)(C)C(=O)NC1CC(F)(F)CC1NC(=O)COCCCOC 72382,N1(C(C)C(=O)NCC2CC2)CCN(C(C2CC=CCO2)=O)CC1 72383,CCCC(C(=O)NC(C)Cn1cccn1)NC(=O)CN(C)CC1CCOC1 72384,N1(C(C2(CC#C)CCOC2)=O)CC2CC(C1)N2C(c1cn(C2CCOC2)nn1)=O 72385,N1(C(C=CCCC)=O)C2CCC1CC(NC(=O)Cn1ccc(Br)n1)C2 72386,N1(C(C(C)(C)OCC)=O)CCCC(CCNC(=O)CCC2(C)CCC(=O)N2)C1 72387,C1(C)(C(=O)NC2CN(C(COC3(C#C)COC3)=O)C(CO)C2)CC2(CCC2)C1 72388,O=C(CC1=CCCCC1)NCCC12CCC1CN(C(C1CC(=O)NC(=O)N1)=O)C2 72389,C(CCCC(C)(C)NC(C1CCCN1C(N)=O)=O)NC(C(C=C=C)C)=O 72390,C(C(=O)NC(C(=O)NC1CC=CC1)C1CCC1)(C(C)C)OC 72391,c1(-c2nc(-c3[nH]n(Cc4nc(C)sc4)c(=O)c3)on2)ccc2c(c1)COC2 72392,CC1CN(C(c2nc(N(C)C)nc(=N)[nH]2)=O)CCN1C(=O)CCN1CCC(F)C1 72393,Cn1nc(CC(N2CC3CC3(NC(C34CC(F)(C3)C4)=O)C2)=O)cc1C(F)(F)F 72394,N1(C(c2cccc(C)c2C)=O)CCC2CN(C(c3ccc(=N)[nH]c3Cl)=O)CC12 72395,N1(C(CCC(CC)C)=O)CCOC2(CCN(C(=O)C(C)C3CCC3)CC2)C1 72396,C(=O)(C(CC)C(=O)OC)NCC1(CNC(c2n(CC#C)cnn2)=O)CC1(F)F 72397,C(CC(C)(C)CNc1ccncc1Cl)NC(CNC(COCCC(C)C)=O)=O 72398,c1(OC)sccc1C(C(=O)NCCc1cn(CCN(C)C)nn1)N(C)C 72399,Cc1c(O)cc(C(N2CCC(O)(C(=O)NCC(C3CCCC3)=O)CC2)=O)cc1O 72400,C=C1CCN(C(C(COC)(C)O)=O)C(NC(=O)C(N2CCC(C(C)O)CC2)=O)C1 72401,C1(CNc2ncc(C)cn2)CC(C)(C)CCC1NC(=O)C1=NOCC1 72402,N1(C(C)=O)CCCC1(C)C(C)Nc1ncccc1OCc1ccccc1 72403,N1(C(C2(OC)CCOC2)=O)CCN(C(=O)C=C(C2CC2)C2CC2)C(CC(F)F)C1 72404,c1(CNC2CC(C(=O)Nc3c(C#N)scc3)C2)c(I)ccnc1Cl 72405,C1(NC(c2c(CC)ncs2)=O)CCN(C(c2cccc(C)c2)=O)CC(C)(C)C1 72406,S(=O)(=O)(c1cc(C(=O)O)c(Cl)cc1Cl)CN1C(C#C)C(C)(C)C1 72407,N1(C(c2c(OCC#C)nccc2)=O)CCN(C(c2csnc2Cl)=O)C(CCO)C1 72408,C1(NC(C2C(C(=O)OC)C2)=O)CCCN(C(c2cc(C)co2)=O)CC1 72409,CCC(c1ccc(OC)cc1)=CC(=O)N(C)CCNC(c1ccc(C)n1C)=O 72410,C=CCCC(C(=O)NCC1(O)CN(C(c2ccc(N)cc2Cl)=O)C1)c1ccccc1 72411,C1(C(=O)NCc2nc(CC)[nH]n2)N(C(=O)C(O)CSC)CC12CCCC2 72412,N1(C(c2c(C)nc(CO)s2)=O)CC(N=c2[nH]nc(C3CC3)s2)CC(C)(C)C1 72413,C(=O)(CCC(CC)CCC)NC1C2(CCN(C(C(=O)NCC)=O)C2)C1 72414,c1(C2(C(N3C(C)(CO)CCC3)=O)CCCC2)ccc(F)c(F)c1 72415,c1(CCC)nccn1CC(=O)NC1COCC1N1CCOCC1 72416,N1(C(c2cn(C)nc2)=O)CC(C)(C)CC1CNC(=O)C(O)C1CC1 72417,CC1(C)C(CO)CCN1C(c1ncc(C(F)(F)F)s1)C(=O)NC1CCOC1 72418,c1(C(=O)NCCCC(CCC)NC(c2nc(OC)oc2)=O)n[nH]c(C)c1[N+](=O)[O-] 72419,N1(C2C(NC(c3ccco3)=O)CCC2)CCN(C(=O)CSC2CCOC2=O)CC1 72420,c1(C(N(CCN2CCN(C(C(C)OC)=O)CC2)C)=O)cc2cccnc2[nH]1 72421,c1(OC)ccc(C(N2CC(CNC(=O)C(O)CCC(C)C)C2)=O)c2ccoc12 72422,C(=O)(C1=CC(C)(CC)C1)N1C(COC)(CNC(=O)C(c2cccnc2)C)CCC1 72423,C(CC1CC1)(CN=c1ccc(Br)c(S(=O)(=O)NC2CC23CCC3)[nH]1)OC 72424,N1(C(c2c(CC)cns2)=O)CCCCC1C(=O)NCC1(O)CCCOC1 72425,C1(c2occc2)C(Cc2cnc(C3CC3)[nH]2)CCN1CC1CCNC1 72426,C1(CC(=O)N(c2ccccc2)CC)(OC)CN(C(=O)CC2CCC2C)C1 72427,N1(C(CCCOC)=O)CCC2CCCC(C1)N2C(C1CCC2(CC2)C1)=O 72428,c1(-c2c(NC(c3c(C)ncc(Br)c3)=O)cc(C3CC3)nc2)ccccc1[N+](=O)[O-] 72429,c1(C(=O)NC2CC(NC(C(C)OCCC=C)=O)C2)c(F)cncc1Cl 72430,c1(CN2CCC(C)C(C(F)(F)F)C2)cc(P(C)(C)=O)cs1 72431,N1(C(c2cc(CC)on2)=O)CCN(C)C(CNC(C2CCSC2)=O)C1 72432,C(=O)(CCCC(C)(C)C#N)NCCC(CC)(C)NC(c1sc(C)nc1C)=O 72433,c1(C(=O)NC2(CCOC)CCN(c3snc(Cl)c3C#N)C2)cnc(C)cc1C 72434,N1(C(C2C(OC)CCCC2)=O)CC2CCC1C(NC(=O)C=CCn1cncn1)C2 72435,c1(C(C(=O)NCCF)N(CCOCCOCC)C)sc(CC)cc1Br 72436,N1(C(C(CCC)C)=O)CC(NC(=O)CCc2cnc[nH]2)CC2(CCC2)C1 72437,c1(C(=O)OC)cnc(=NCCC(C)(C)NC(c2c(C3CC3)cnn2C)=O)[nH]c1 72438,CC1CCN(C(C2CCOCCN2C(=O)CC(C)O)=O)CCS1 72439,Cc1cc(C(=O)NC(CNC(=O)CSc2ccccc2O)CO)c(C)n1C 72440,c1(C(=O)N(c2ccc(Cl)c(I)c2)C2CC3CNC2C3)cccc2c(Cl)ccnc12 72441,CC(CC(=O)NOCCCCC(=O)N(C)CCN(C)C1CC1)C1CC1 72442,c1(C(=O)NCCNC2(C3CCCO3)CCCC2)ccnc(CC2CC(O)C2)n1 72443,N1(C(c2cc(CC(C)C)c(N)cc2)=O)CC2(CCCC2NC(C2CC2(F)F)=O)C1 72444,c1(CNC(CC2CCN(C(CNC(=O)OCC=C)=O)CC2)=O)c(C)cccc1C 72445,C(=O)(CC(C)C(=O)N1CCC(C(C)C(=O)NC2(CC)CNC2)C1)OCC 72446,C1(NC(=O)Cn2nnc(=O)[nH]2)CN(C(c2cnnc(O)c2)=O)CC1C1CC1 72447,n1(CC(=O)NC(CNC(C(C)(C)C)=O)(C)C2CC2)cc(F)ccc1=O 72448,C1(C)(C(=O)NCCCCCN(C(=O)CSCCC(F)(F)F)C)CCCNC1=O 72449,Cc1oc(C)c(C(=O)NCC2CC(CNC(=O)COCCN(C)C)CO2)c1C 72450,Cc1ncc(Br)c(N(C2CCNC2)C(c2cccc(I)c2)=O)n1 72451,C12(NC(=O)COC3CCC3)CC(C(=O)NCCc3ccon3)(C1)C2 72452,c1(-c2c(C)cc(C)c(C)c2)nc2c(s1)CCN(S(=O)CCCl)C2 72453,C12(NC(c3n(CCC)ncc3)=O)CCC1CN(C(c1cc(C3CC3)ncn1)=O)C2 72454,CC(C(=O)N1CC(O)CC1Cn1cc(-c2ccc(Cl)c(Cl)c2)nn1)S(C)(=O)=O 72455,c1(C(=O)NC2(CN(C)C(c3ccnnc3O)=O)CC2)cccc(CO)c1 72456,N1(C(C(CC=CC)CC)=O)CC2CN(C(=O)C(c3ncc(Cl)n3C)(F)F)CC2C1 72457,C(CC(=O)NCC1(C)CCCN(C(=O)C=C2CCCC2)C1)(C(F)(F)F)OC 72458,c1(CNCc2n(CCOC)ncn2)ccc(C#CCO)s1 72459,CCC(CN(C)C)CC(=O)NC1(CCC(=O)Nc2ccc(OC)c(C)c2)CCC1 72460,N1(C(=O)NCc2cnc(Br)c(F)c2)CCC(C2CC2)(CO)C1.CC(C)(C)O 72461,N1(C(c2ccc(CC)c(I)c2)=O)CC(C(=O)OC)Oc2c(C)cccc21 72462,c1(C(=O)NC(CC=C)CNC(=O)CC2(CO)CC2)ccnc(SC(C)(C)C)c1 72463,C1(CC(=O)NCCCN(C(C2CCC(CC)O2)=O)C)NC(=O)CNC1=O 72464,C(CCN=c1[nH]c(=N)[nH]c(=NC(C)c2ccc(Br)cc2F)[nH]1)OC=C 72465,CCC(CC(C)C)C(=O)NC1CCN(c2cn(C3(O)CCCCCC3)nn2)C1 72466,CCC(C)(COC)C(=O)NC1CCC(CCC(=O)NCC2(F)CC2)C1 72467,C(=O)(C1COc2ccccc21)N(C)CCN(C)C(C1(CO)CCCO1)=O 72468,c1(C(C)C)ccc(C(C)C(=O)NCC2(F)CN(C(c3ncccc3O)=O)C2)cc1 72469,C1(C)(NC(C(CC2CC2)OC)=O)CCN(C(C2CCC(C)(C)OC2)=O)CC1 72470,c1(N(CC(C)C)C(=O)CN(C)CC2(C)CCCC2)nc2ccc(F)cc2s1 72471,C1(NC(C(CC)N(C(=O)C(C)OC(C)=O)C)=O)CC(C)(OC)C1(C)C 72472,N1(S(CC(C)c2ccccc2)(=O)=O)CCN(C2CCNC2)C(C)C1 72473,N1(C(=O)Cn2cnnc2O)CCN(C(c2cncn2-c2ccccc2)=O)C2CC12 72474,CC(C(=O)NC1CC(NC(=O)Cn2nnc(C(C)(C)C)n2)C1)S(N)(=O)=O 72475,N1(C2C(C3CCC(C(C)(C)C)O3)C2)CCCC2(CCOC2)C1 72476,c1(OCC2CC(N(C(CN(CC)Cc3nccs3)=O)C)C2)ccccc1OC 72477,CC1CCCCC1(C)NC(=O)CCN(CCO)C(c1cccn1C1CC1)=O 72478,C1(NC(CC(C)OC)=O)CCC(C(=O)NCC2(CCO)CCCC2)CC1 72479,C(CC(C(=O)NCC1(OC)CCC(C)C1)NC(=O)CC1CNC(=O)O1)OC 72480,CC(CN=c1[nH]c2c(c(=NCC3CC4C=CC3C4)[nH]1)SCC2)n1cccn1 72481,C1(NC(CC2CCC(C)C2)=O)CN(C(=O)CCc2ccc(F)nc2)CC2(CC2)C1 72482,C(=O)(C(C)(CO)NC(c1ccnc(OC)c1)=O)N(CCCC)CC 72483,C1(NC(CCN(CCC)C)=O)C2CCCN(C(C3CCSC3)=O)C2C1(C)C 72484,C1(NC(c2ccsn2)=O)CCC(CCNC(c2ccnn2-c2ccncc2)=O)C1 72485,c1(C(=O)NC(C(C)C)CNC(c2cn(C)[nH]c2=N)=O)ccc2ncnn2c1 72486,c1(CC(N2CCC(C(=O)Nc3ncn(C)n3)CC2)=O)cccc(F)c1Cl 72487,N1(C(CSCCOC)=O)CCC(NC(=O)CC2CCOC2)CC1C 72488,c1(C(N2CC(CCNC(=O)C(O)CCSC)(OC)C2)=O)nn(C)c(C)c1Cl 72489,c1(C(N(CCC)CCNC(=O)CC2CCCC(O)C2)=O)c(C)[nH]c(C)c1C 72490,S(=O)(=O)(c1ccccc1F)N(N1CC(N(c2ccc(Cl)o2)C)C1)C1CC1N.C 72491,c1(OCCC(N2CCC(NC(C(C)C)=O)C2C)=O)cc(F)cc(F)c1 72492,C12(C(N3CC(N4CCN(C(c5cncnc5)C)CC4)C3)=O)CCCC1CCC2 72493,C1(CC(N2CC(OCCC(=O)NC(C(C)C)C3CC3)C2)=O)NC(=O)NC1=O 72494,C(=O)(CCP(C)(C)=O)N(C1CCCCN(C(=O)C(c2ccc(F)cc2F)=O)C1)C 72495,c1(C(=O)OCc2c(F)ccc(F)c2Br)cc(I)ccc1[N+](=O)[O-] 72496,n1(C(C2CC2)C)nnnc1C1(NCC(Cc2ccoc2)CO)CC(C)C1 72497,N1(C(c2cc(OCC)no2)=O)C(C)CC2CN(C(c3c(C)coc3CC)=O)CC12 72498,Cc1cccc(C2CCN(C(=O)CN(C(=O)CC3C=CCC3)C)C2)c1.C1(=O)CN1 72499,N12CC3CC1CN3C(C1CCC1)CC2=O.c1(C2CCC2)ccc(Cl)cc1 72500,N1(C(=O)C=Cc2cccc(CO)c2)CCC(CNC(C2(Br)CC2)=O)C(F)(F)CC1 72501,c1(C(=O)NCC2CCN(C(CCC3C(C)C3)=O)C2(C)C)ccc2c(c1)ncn2C 72502,Fc1cc2c(cc1Br)CN(Cc1cccc(Cl)n1)CC2 72503,c1(C(N2C(CO)CC(NC(C(CC(C)C)NC(C)=O)=O)C2)=O)cc(C)nc(Cl)c1N 72504,Cn1cc(Br)cc1C(=O)NCC1(NC(=O)CNC(=O)C2CC2)CC1 72505,C(=O)(C(Cc1cn(CCCCC2C(=O)ON=C2C)nn1)CC(F)(F)F)OC 72506,c1(N2CCC(C)(CSC)C2)nc(=N)nc(N2CCC(CCO)C2)[nH]1 72507,C(=O)(CC1=NN(C)C(=O)C1)N1CCC(C#C)(C(N2CCOC(CC(N)=O)C2)=O)C1 72508,N(C1CCc2ccc(Cl)cc21)C(CC1CNC1)=O.CCCCS(=O)(=O)N 72509,c1(C(=O)NC(C2CCOC2)CNC(c2ccccc2Cl)=O)ccc([N+](=O)[O-])s1 72510,c1(NC(=O)NC2(CC(=O)Nc3c(C)cc(F)cc3)CCC2)cc(F)c(F)c(F)c1 72511,C1(C(N(C2CCNC2=O)CC)=O)CN(C(=O)C(F)C(C)C)CC1C(C)C 72512,c1(C(N2CC(NC(CCNC(N)=O)=O)C3(C2)CC3)=O)cccc2c[nH]nc12 72513,CC1(C)CN(CCF)CCN1C(c1ccnc(Cl)c1F)C(=O)NC1CCOC1 72514,C1(CN(C(=O)COC(C)(C)C)C)CCN(C(=O)CCN2CCC(F)C2)CC1 72515,c1(C(N2CCCC(NC(c3ccc(Br)cc3Br)=O)CC2)=O)c(Cl)cc(F)cc1Cl 72516,C(CCC(C)C(=O)N1CC(Oc2cc(C(=O)NOCCN(C)C)on2)C1)OC 72517,C1(NC(c2c(C)c(Br)n(C)n2)=O)CN(C(=O)C(C)C#N)CCC12CCC2 72518,N1(C(C(C(=O)OC)OC)=O)CC(NC(c2ccnnc2)=O)C2CCCC12 72519,N1(C(C2CC3(CC3)CO2)=O)CCN(c2ncncc2F)CC12CCC2 72520,C1(=O)C(C)(C)CCC(=O)C(NC(C(CC)CCOC)=O)CCC(CC)N1.OC 72521,c1(N(C2CNCCC2(F)F)c2nccc(OC)n2)ncc2ccccc2n1 72522,c1(C(=O)NCC2CCCN(c3sc(C(=O)OC)c(Cl)n3)C2)c[nH]nc1S(N)(=O)=O 72523,N1(C(Cc2c(C)cccn2)=O)CC2(C(=O)NC3CCC(C4CC4)C3)CC1CO2 72524,N1(C(C(C)SCCCC)=O)CC2CN(C(=O)CN(C)S(N)(=O)=O)CC2(C)C1 72525,c1(C(=O)NC(C(C)C)CCN(C(=O)C(C)O)C)c[nH]c2c(Br)cccc12 72526,CCCCC(=O)NNC(=O)C1CCN(OC(=O)NC(C)(C)C)C1(C)C 72527,CC(CC(=O)N1CCCC1(c1cn(C2CCC(C)(C)CC2)nn1)CO)C(F)(F)F 72528,C1(C(=O)NCC(CC=C)(C)C)CN(C(c2cnc(C)s2)=O)CC1(F)F 72529,CCN=c1[nH]c(C)c(C(=O)NCC(C2CC2)NC(=O)Cc2nncn2C(C)C)s1 72530,c1(CNC(CC=C)=O)ccnc(C(=O)NCC2C=CCCC2)c1 72531,CC1=C(C(=O)NC2CCCCN(C(C3CCCCC3C(N)=O)=O)C2)CCS1(=O)=O 72532,C1(CCNC(CCOCC#C)=O)CN(Cc2ccc(C(N)=O)cn2)CCS1(=O)=O 72533,CC1CCC(C(N2CC(C(=O)O)(Nc3ccccc3)C2)=O)CN1 72534,C1(NC(C(c2cccc(C)c2)C)=O)CC(F)CN(C(c2cnnc(C)c2)=O)C1 72535,CCC1=NOC(C(=O)NCCCCN(C(=O)Cn2cccc2)C2CC2)C1 72536,c1(COCC)cc(Cl)cc2cc(NC3(c4n(CC)nnn4)COCC(C)(C)C3)oc12 72537,c1(C(N2CC(CC=C)(NC(=O)CCCC(C)=O)C2)=O)ccc2c(c1)CCS2(=O)=O 72538,CC(CC(C)(C)NC(=O)NC1C2CC3C(C2)C13)N(C)C 72539,N1(C(CS(CC)=O)=O)CC2CC1CN(C(c1cccc(NC(=O)C3CC3)c1)=O)C2 72540,N1(C(C(n2cccc2C=O)C)=O)CCC2(CC1)CCN(C(=O)C(C)(C)C)C2 72541,C1(CC(=O)NCCN(C(c2c(N)ccc(C)c2)=O)C)CCn2cncc2C1 72542,c1(C(=O)NC2(C(=O)NCCCCCCC)CCOCC2)cn2c(n1)CCC2 72543,C1(CCC(=O)N(C(CC(C)C)C)C)CCN(C(=O)Cc2ccc(F)cc2)C1(C)C 72544,c1(N(c2cc(C)ccc2C)C(C)=O)cccn2nccc12.C12CCCN(C1)C2=O 72545,C=CCCCCCC(=O)NC(C)(C)CN(C(=O)C(c1ccc(Cl)s1)C)C 72546,N1(C(CC=C=C)=O)CCC2CCN(C(c3cn(C)nc3-c3ccc(C)o3)=O)C2C1 72547,C(=O)(C(C)(C)S(C)(=O)=O)NC1CN(C(CCC(CC)OC)=O)CC2C1C2 72548,c1(C(=O)NCC2C(CNC(CCCC(C)(F)F)=O)C2)sc2ccccc2c1Cl 72549,CCC(C(=O)NC(C)(C)C(C)CC(=O)NC(c1ccccc1O)C)C(F)(F)F 72550,C1(CNC(C(C=C)CC)=O)CC2(CC2)CN1C(c1cc(CC)oc1C)=O 72551,N1(c2cc(NCCCCOC)ncn2)CCN(C(=O)OC)CC1(C)C 72552,c1(C(=O)NCCN(C(=O)C(F)n2ccnc2)CC)c[nH]c2cccc([N+](=O)[O-])c12 72553,CC(O)C(C(=O)NC12CC1CN(C(c1ccc(C3CC3)cc1)=O)C2)NC(N)=O 72554,C(=O)(C1CCCc2cncn21)NC(C)(CNC(C1CCCC1)=O)C1CC1 72555,C(CN=c1[nH]c2c(c(=NCC3COCCN3C)[nH]1)SCC2)c1ccc(F)c(F)c1 72556,N1(C(C2C(OC)CCC2)=O)CC(=O)Nc2ccccc21 72557,C1(C(=O)NCC2(C)CCN(C(C=CCN(C)C)=O)CC2)COc2ccccc2O1 72558,N1(C(CCC=CC)=O)CC2(CCN(C(c3ccc(=O)n(CCF)n3)=O)CC2)C1 72559,c1(CC)cc(F)c(C(=O)NCCC2(NC(c3ccccn3)=O)CCC2)cc1F 72560,N1(C(c2nc(CC)oc2)=O)CCC2(C=C(C(=O)NCc3ncoc3C)C2)C1 72561,C1(C(N2C(C(C)NC(=O)COC3(C)CCC3)CCC2)=O)CCc2c[nH]nc2C1 72562,N1(C(C=Cc2scc(C)n2)=O)CCN(C(C2CCCO2)=O)CC2(CC2)C1 72563,N1(C(C(=O)NC(CC=C)=O)C)CC2CCCN(C(=O)Cc3oc(C)nc3C)C2C1 72564,C(=O)(C(C(C)(C)C)c1ccccc1)N(CCc1cn(CC)nn1)C.C(CC)=C(C)C 72565,C1(NC(C(n2c(C)ccn2)C)=O)CCN(C(c2cc(C(F)(F)F)ns2)=O)CC1 72566,c1(C(N2C3C(NC(C4(CCOC)CC4)=O)C(C3)C2)=O)cccc2occc12 72567,N(C(=NCC1(C)CCCO1)NC(C)C)C(C#C)CC1CCC1 72568,c1(CC)oc(C(N2CCCC(CNC(C3(Cl)CC3C(C)=O)=O)C2)=O)cc1C 72569,S(=O)(=O)(c1ccc(N(CCC(O)CCC)C(C)C)cc1)NCC=C 72570,N1(C(c2onc(C)c2C)=O)CCC(NC(C2CC(C)CC(C)C2)=O)C12CCCC2 72571,C(CC(=O)NC(CC1CC1)C1CC1)(C(F)F)NC(c1c(C)n[nH]c1C)=O 72572,N1(C(C=C(C)C(F)F)=O)CCN(C(=O)CCC23CCC(CC2)C3)CC1C1CC1 72573,c1(C(=O)NCC2CCN(C(C(C)(C)C3CCOC3)=O)C2)cncc(P(C)(C)=O)c1 72574,CC1=NOC(C)(C(=O)N(C)CC2(NC(=O)CCC=CBr)CC2)C1 72575,c1(C(=O)OCCCCCCC)cncc2nc[nH]c12 72576,C(C#CCNC(C1(C(F)(F)F)CC1)=O)NC(CN(C(C)=O)C)=O 72577,N1(C(C2C3CN(C(c4cccn(C)c4=O)=O)C2C3)=O)CCC(N=[N+]=[N-])CC1 72578,C1(C2(C)CC2)(C(=O)NC(CNC(c2cn(CC(CC)O)nn2)=O)CO)CC1 72579,C1(CC(=O)NCc2onc(C)n2)CN(C(c2nnn(C(C)C)c2C)=O)CCO1 72580,N1(C(C(CC#C)C2CC2)=O)CC2N(C(C)(C)C1)Cc1cn(nn1)CCS2.SC 72581,c12ccc(cc1)C(=O)N(CCCN1CCC(F)CC1)C2.Cc1ncon1 72582,N1(CCNC(N(C)CC2CCCC(C#N)C2)=O)CCc2c(Cl)cccc2C1 72583,C1(NC(C(CC)O)=O)C2CCN(C(=O)C(C)CCc3cccc(F)c3)CC12 72584,C1(CC(C(=O)NCCCOCC(C)(C)C)N(CCC#N)C)CN2CCC1CC2 72585,c1(C(=O)NCC(CNC(CCSCCCC)=O)(C)F)cc(F)cnc1O 72586,CC1OCCOC1C(N1CCOCC1C(=O)NCCC1(C)CC1(F)F)=O 72587,C(C)(CCC(C)(C)C)NC(c1nncc(OCC)c1)=O 72588,N1(C(=O)CC2CC(Oc3ccccc3)C2)CC2ON=C(C(F)F)C2C1 72589,CCC(C)C(C(=O)NCCCCCCNC(N)=O)NC(=O)CN(C)S(N)(=O)=O 72590,CCC(CC)(CO)C(=O)N1CCC(NC(C2CCn3cncc3C2)=O)CC(O)C1 72591,Cc1nccc(C(=O)NCc2ocnc2C(=O)NC(C)C(N)=O)c1N 72592,N1(C(C2(C)CC=CCO2)=O)CC2=C(C1)CN(C(=O)CCNC(c1cccs1)=O)C2 72593,C(CC(C(=O)NC1(C)CC(O)C1)NC(=O)CC(C)(F)F)N(C)C 72594,C1(C(=O)NC2CCC(CNC(=O)COCC(F)F)CC2)CCN2CCCCC12 72595,c1(C(=O)NC(C)CNC(=O)C=CCO)cc2scnc2[nH]1 72596,C1(CC(=O)NC(C(=O)OC)CCF)C2CCC(C2)N1C(=O)CC1CN(C(C)=O)C1 72597,C1(N(C(Cc2ncc(C)o2)=O)C)CN(C(=O)CC2CN(C)C2)CC1F 72598,CC1(C)OC1C(=O)OCC(F)(F)Br 72599,CS(=O)c1ccc(C(=O)NCCC2CCCN2C(=O)Cc2ccc(Cl)cn2)cc1 72600,c1(CNC(C2(NC(C3CC3C(F)(F)F)=O)C(C)(C)C2)=O)ccccc1O 72601,CCC(CC(=O)N1CCC(COC)CC1)N(C)C(C1(CC(=O)OC)CC1)=O 72602,C1(C2CC2)(C(=O)NCC(CNC(CCC)=O)OC)CCOCC1 72603,C(=O)(CCC1=CCCCC1)N1CCN(C(CCCC#CC)=O)CC1CC(F)(F)F 72604,c1(C(=O)NC(C2CCN(C(c3ccc(Cl)nc3)=O)C2)C)cccc(F)c1 72605,C1(NC(C2CCCC23CC3)=O)CC12CCN(C(c1ncc3[nH]ncc3n1)=O)CC2 72606,c1(NC2C(C)CN(C(C3CCOC(C)C3)=O)C2)c(C#N)cccc1[N+](=O)[O-] 72607,C(c1cn(C(C)CNC(C2(c3ccc(Cl)cc3)CCCC2)=O)nn1)=CC 72608,C1(CNC(CCC2CCN(C(c3c(CC)cco3)=O)C2)=O)CCC(C)N1C 72609,N1(C(COCCCC#C)=O)CCCC(CCNC(=O)C(c2cccc(Cl)c2)O)C1 72610,C1(NC(C2CN(C)C2)=O)CN(C(c2cccc(CC#N)c2)=O)C2CCCCC12 72611,C(C1CCCCCC1)=CC(=O)N(CCCCN(C(C1CCC(OC)C1)=O)C)C 72612,N1(C(=O)OC(C)(C)C)CCC2C1CCCN2C(c1cc(Br)cc2nc[nH]c12)=O 72613,C(=O)(CC(C)C(=O)OCC)CC.C1(C(N2CCC(O)(CN)C2)=O)(OC)CCOCC1 72614,C1(C2CN(C(=O)C(C)Cn3ccnc3)C2)(NC(Cc2c(C)n[nH]c2)=O)CC1 72615,C1(CN(C)C(c2ccncc2)=O)CCCCN1C(=O)COCCC1CCCCO1 72616,c1(C(=O)NCC(CCNC(CCC(=O)NCC)=O)O)cnc(C)cc1Cl 72617,Cc1nn(C)cc1-c1ccc(C(=O)NC(=O)CC(C2CC3CCC2C3)N)s1 72618,C1(NC(c2c(C)sc(Br)c2)=O)CC2CC1CN2C(=O)C(N)=O 72619,Cc1ncnc(O)c1CCC(=O)N(CCNC(C1CCC2(CCC2)C1)=O)C(C)C 72620,C(CN=S(C)(C)=O)NC(c1n(CC)nnn1)c1ccnn1C(C)C 72621,CC(C)(C)C(CNC(=O)Cc1nc(=N)[nH][nH]1)NC(C1CC1Sc1ccccc1)=O 72622,c1(C(=O)NCCC2(C(=O)NCC3(OC)CCC3)CCC2)nc(C)sc1C 72623,C(=O)(C(O)(C(F)(F)F)c1ccccc1)N1CCC(CCNC(C2(F)CC2)=O)C1 72624,C(=O)(C1CCCc2n[nH]cc21)NCCCC(C)NC(C1CC1(F)F)=O 72625,N1(C(CC(C)O)=O)CCC(F)(F)C(CNC(c2cc(C3CC3)n(C)n2)=O)C1 72626,Cc1nnc(NC2CC(NC(c3sccc3C)=O)C2)nc1C 72627,c1(N2CCN(C(CCC)=O)CC2)cc(C)nc(C)c1[N+](=O)[O-] 72628,C1(C(=O)NC(C2(OC)CCC2)C)CC2CN(C(c3ncn(C)n3)=O)CC2C1 72629,C(C1CCCN1C(c1coc(CO)c1)=O)=CC(=O)N(C)Cc1ccco1 72630,N1(C(C#CC2(CC)CC2)=O)CCCC2CN(C(C3(CO)CCC3)=O)CC12 72631,S(=O)(=O)(C1(c2cn(CCC(N3CCC3(C)C(C)C)=O)nn2)CC1)NC 72632,Cc1c(C(=O)NCc2ncc(C(N3CC(C)CC3C)=O)cn2)c[nH]c1C#N 72633,CCC(C)C(O)CC(=O)N1CCOC(CC(=O)NCC(C)(F)C(C)(C)F)C1 72634,c1(C(N2CCC(CN(C(C(N3CCC(O)CC3)C)=O)C)C2)=O)cccc(Cl)c1Cl 72635,N1(C(C(C=C)O)=O)CCN(C(=O)CN(c2ccncc2)C)CC2(CC2)C1 72636,N1(C(C=CC=CC)=O)CCC(NC(c2cn(C)nc2CCC(F)(F)F)=O)C1C 72637,c1(N(C)C)nc(Cl)ccc1C(=O)OCCc1nc(C(C)(C)N(C)C)no1 72638,N1(C(CSCC#C)=O)CCCC(C(C)(C)C(=O)NCc2cnn(CCC)c2)C1 72639,C1(NC(C2CC2(F)F)=O)CCN(C(=O)C=Cc2ccncn2)CC1CO 72640,C(=O)(C(F)(F)C(F)(F)F)N1CC(NC(=O)Cn2ncc(O)nc2=O)C(O)C1 72641,C1(C(N(CC(=O)N(CCCC(C)C)C2CC2)C)=O)CNC(=O)CC1C 72642,c1(NC(C2(O)CCN(C(C=CC(C)C)=O)C2)=O)ccc([N+](=O)[O-])c(F)c1 72643,n1(CCC(=O)NC23CC(NC(C(C(C)C)F)=O)(C2)C3)nc(O)c2ccccc12 72644,C1(C(N2C(C)(COC)CCC2)=O)CC2CCCC2N1C(=O)C1=C(C#N)CCC1 72645,N1(C(C2C(C)(CC)C2)=O)CCC(C(=O)Nc2cn(C)nn2)CC1 72646,N1(C(Cc2nnc(C)o2)=O)CCN(Cc2cccc(C)c2O)C2CC12 72647,C(=O)(CCCC(=O)NCC1CN(C(=O)CC2(O)CCCCC2)CCO1)NCCC 72648,N1(C(c2nc(C)n(-c3ccccc3)n2)=O)CC2CC1CN(C(C1(F)CC1)=O)C2 72649,C(=O)(CS(N)(=O)=O)N(C(C)C)CCNC(=O)C(C)n1cnnn1 72650,N1(C(C(=O)NCCC(C)c2ccco2)=O)CCC(NCC(F)F)CC1 72651,C(C(CC)(CC)C(N)=O)NC(C1C(CNC(CCC=C=C)=O)CCC1)=O 72652,N1(C(C(C(C)C)SC)=O)CCCn2cc(Br)cc2C1 72653,c1(CC)cc(NNC(=O)NC2CCCC(C3CC3)C2)ncn1 72654,CCCCCCC(=O)NC(C(=O)N(C)CC1CCOCC1)c1ccoc1 72655,n1(CCOCC)nc(-c2cccc(C(F)(F)F)c2)nc1CCCC1CCCCC1 72656,CCC(C)C(=O)C(=O)NCC1C(C)CCCN1C(c1cnn(C(C)C)c1)=O 72657,C1(NC(C(C)CO)=O)CCC2(CC1)CN(C(c1coc(C3CCOCC3)n1)=O)C2 72658,Cc1cc(NC(=O)CN(C(=O)C(F)C(C)(C)O)C(C)C)cc(C)c1O 72659,c1(C(=O)NCCN(C(C(CC)N2CCCC2=O)=O)C(C)C)ncc2ccccn12 72660,C(=O)(C1=CC(O)C(NC(C2C(C(C)=O)C2(C)C)=O)C1)NC1(CO)CC(OC)C1 72661,c1(OCCCCC)ccc(C(=O)NCC2CCCN2C(=O)C(C)O)cc1 72662,C1(NC(C2OCCN(C(C=CCOC)=O)CC2)=O)CCCCN(C)C1=O 72663,C1(C(=O)NC(CNC(c2c(CC)csc2)=O)C2CCC2)CCCCCCC1 72664,c1(C(=O)NC(C(C)O)C(=O)O)cc(Br)cnc1O 72665,C1(NC(c2cn(C(C)C)nc2)=O)CC2(CCN(C(c3cccc(N)n3)=O)CC2)C1 72666,N1(C(C(C)=C(C)C)=O)CCCC1CNC(c1nc[nH]n1)=O 72667,N1(C(C2(C)COC2)=O)CC(C2CN(C(c3nccc(Cl)c3F)=O)C2)C1 72668,N1(C(c2cc(C)cc(F)c2)=O)CCC2(CC2)CC1C(=O)NC(C)C(C)F 72669,c1(C(=O)NCC(C)NC(Cc2c(C)cco2)=O)cc2c(n1C)CCOC2 72670,C(=O)(CC(CC(C)C)NC(=O)CCn1cnc(=N)[nH]1)Nc1cn(CC)nc1 72671,N1(C(CC(C)F)=O)CCCCC2(CCN(C(=O)Cc3ccc(Cl)cc3Cl)C2)C1 72672,C1(C(N2CC(NC(c3c(CC(C)C)cccc3)=O)C(O)C2)=O)CCN(C)S1(=O)=O 72673,C12CCCN(CC1)C(=O)CSCC(=O)OCC(=O)N2.N1(C(CC)C)CCCC1 72674,c1(C(N2C(CO)CC(NC(c3cc(C)oc3C)=O)C2)=O)ccc2c(c1)NCCC2 72675,C=C(C)C(C)(C)C(=O)NC1CCCC(CN(C)C(c2ccc(CC)[nH]2)=O)C1 72676,C1(N)CN(c2ccccc2)CC12CCOCC2.C1(F)(N(C)CC(C2(C)C(COCC)C2)=O)CCCC1 72677,C1(N(c2cccc(C(C)C)n2)C(C(c2ccccc2)C)=O)CCNCC12CC2 72678,c1(C(c2n(CCNC(C3CCCCC3)C)nnn2)OCC)nccc(Cl)c1C 72679,Cc1cnc(C(=O)NCC2(NC(c3cnn(C)c3F)=O)CCCCCC2)c(C)c1 72680,C1(CC(=O)N(CCCCN(C(=O)Cc2cnco2)C)C)OCCC1(C)C 72681,S(=O)(=O)(c1cccc(C(=O)NC(c2ncccn2)(C)CC)c1)NC(CC)C(N)=O 72682,c1(C(=O)NC2C(C)CN(C(C34CC(CC(F)F)(C3)C4)=O)C2)cc([N+](=O)[O-])ccn1 72683,N1(C(CCCC#C)=O)CCOCC(NC(=O)CCCc2ccc(C)s2)C1 72684,C1(C(=O)NC2CCCN(C(c3nccc(CC)c3)=O)C2)CNC(=O)C(C)(C)C1 72685,CC(C)C(F)(CNC(C1CCCC12CCC2)=O)C(=O)N(C)CC1CCOC1C 72686,C(=O)(C(C)(C)CC(=O)OCCOC(C)Cc1ccccc1F)OC 72687,c1(CCC)ccc(OC(=O)C=Cc2scnc2C)c(OC)c1 72688,c1(C(=O)NC2C(OC)CN(C(c3cccn3C)=O)C2)ccc2c(N)nccc2c1 72689,N(C1COc2cc(Br)cc(C)c21)C(=O)Nc1ccc(C(=O)OCC)c(F)c1 72690,C=CCCCCC(=O)NCC(C)(CC(C)C)NC(=O)CCCc1ncco1 72691,N1(N(C(c2nc(C(C)C)on2)=O)C)CCCC(n2cc(C(C)(C)F)nn2)CC1 72692,c1(C(N2CC3(CN(C(CC(C=C)(C)O)=O)C3)C2)=O)nn2ccccc2c1C 72693,CC1C(C)N(C(C23CCC(CC2)OC3)=O)CCN1C(=O)CNC(=O)CN(C)C 72694,C1(N)(C)CCCC(C)(C)C1.c1(C2C(=O)N2C)ccc(C)cc1.CO 72695,c1(C(=O)NC2CC(C)C2)cnn2cccc(-c3ccc(C4CCOCC4)cc3)c12 72696,c1(C(=O)NCCC2CC(NC(CC#N)=O)C2)ccc2c(c1)S(=O)(=O)NC2 72697,C(=O)(C(C)(C)CCC#N)NC1C(C(NOC(C=C)C)=O)COC1 72698,c1(NCC(C)(C)OC)nc(C)cc(=NC(C)c2nc(C(F)(F)F)n[nH]2)[nH]1 72699,C(=O)(C(O)CC[S+](C)C)NCCCCNC(C(C)OCC=C)=O 72700,C1(C(C)C)CCC(C)CC1(O)CNC(=O)C(C1CCCCC1c1ccccc1)=O 72701,C(=O)(NN1CCCC1C(=O)N(C1CCCC1)C)C1CC(N(C)C)C1 72702,c1(OC)cc(C2(C(=O)NCC(C)(O)CNC(C3CCCO3)=O)CC2)ccc1C 72703,c1(COCCNC2CCN(C(C(c3ccccc3)SC)=O)C2)ccnc(F)c1N 72704,N1(C(c2cnc(-c3cccnc3)s2)C(=O)NC(C)C)CCCCC(F)(F)C1 72705,c1(CC(=O)NC2CCC(CNC(C(N(C)C)C3CC3)=O)C2)cc(Cl)ccc1Cl 72706,n1(CCC(=O)NC(C(C)C)c2ncc[nH]2)cc(CNS(N)(=O)=O)nn1 72707,CCC(C)(O)CCNC(C1(NC(C2C3CCCOC23)=O)CCSC1)=O 72708,Cc1ccc2ncc(C(N3CCCC(NC(c4coc(C)n4)=O)C3)=O)n2c1 72709,c1(CN2CC(O)(C(=O)NC3CNC3)C2)cccc2c1oc1ccccc21 72710,C(=O)(CCCCCF)NC1C(C)CN(C(c2cnc(C(C)(C)C)[nH]2)=O)C1 72711,C1(C(=O)NC2C(CNC(c3c(C)n[nH]c3C)=O)COC2)CCCCCN1C 72712,CC12CN(C(=O)Cc3ncc(Cl)s3)CC1CN(C(c1coc(C(F)F)n1)=O)C2 72713,c1(C(=O)NC(C)CNC(=O)Cc2n[nH]c(O)n2)cccc(-c2ccoc2)c1 72714,C1(NC(c2c(OC)ccs2)=O)CCCC(C(=O)NCc2cnco2)C1 72715,c1(C(N(C(CCNC(C(CCCC)O)=O)C)C)=O)cc(Cl)cc(F)c1N 72716,c1(C(=O)NC(C2CCCN2C(=O)CS(=O)(=O)N(C)C)C)cc(C(=O)N(C)C)oc1C 72717,c1(N2CCCC(CNC(c3n(C)ncc3)=O)CC2)ncnc2c1ncn2C1CC1 72718,N1(C(C(C)=CC2CC2)=O)CCC2(NC(c3conc3C)=O)CC2C1 72719,C1(C(=O)OC(C)Cn2cncn2)CCN(C2CN(S(C)(=O)=O)C2)CC1 72720,c1(C(=O)NCCN(C(CCCC(=C)C)=O)CC(C)O)cncc(S(C)(=O)=O)c1 72721,c1(C(=O)NC23C(CN(C(C4C(C)(C)CCCC4)=O)C2)C3)c(Cl)cccc1[N+](=O)[O-] 72722,c1(SC2(C(=O)NC(C)CNC(C3CCC3C(F)(F)F)=O)CCC2)ccccc1 72723,N1(C(CCCOCC=C)=O)CCC(C2(NC(=O)Cc3ccc(OC)cc3)CC2)C1 72724,CC(C)CCCCCC(=O)NCC1C2CC1N(C(c1coc(Cl)n1)=O)C2 72725,C(=O)(C(C)(C)n1cccn1)NCCN(C(CCNC(COC)=O)=O)C 72726,c1(C2(C(=O)NC3CC(C(N)=O)OCC3)CC2)ccc(-c2ccsc2Cl)cc1F 72727,c1(CNC2(CC(=O)OC)CCOCC2)c(Cl)nc(SC)nc1Cl 72728,c1(C(CNc2nc[nH]n2)NC(CC2(CSC)CC2)=O)ccccc1.C1(=O)CN1 72729,CC1CN(C(=O)CC(C)CN(C)C)CCCN1C(=O)CCn1cccc1 72730,c1(OC)cccc(Cl)c1C(N1CCC(CO)(Nc2ccncn2)CC1)=O 72731,N1(C(CN(C(C)=O)C)=O)CCCC(CCNC(=O)CCNC(c2cccs2)=O)C1 72732,C(CN=c1[nH]c(N2CCN(C(C)=O)CC(C)(F)C2)nc2c1CCC2)SC 72733,c1(C(c2nnnn2CCCF)NCC2CC(C(=O)OC)C2)ncc(C)s1 72734,c1(N(C)CC(=O)Nc2ccc3c(c2)OCO3)nc2c(c(=NCCCP(C)(C)=O)[nH]1)COC2 72735,c1(OC(C)C)cccc(C(N2CC(O)CC2C(=O)Nc2nc(C#N)cs2)=O)c1 72736,C1(NC(C(C(C)C)CO)=O)CCN(C(=O)CCOc2ccccc2)CCC1CO 72737,c1(CNC(=NC)NC(c2ccc(-c3ccccc3C)cc2)C)cccnc1F 72738,c1(OCC)cccc(OCC(N2CC(C)(NC(C3(C)CC3Br)=O)C2)=O)c1 72739,c1(C(C)C)ncc(NC(=O)C(C)C(C)NC(=O)Cc2ccoc2)cn1 72740,c1(OCC#C)ccc(Br)cc1CN(c1cnc(C)cn1)C 72741,c1(C(=O)Nc2cc(C)c(C(F)(F)F)cc2)cccc(S(=O)(=O)NCCN(C)C)c1 72742,C(CC)(CCCC(=O)N(C)CP(C)(C)=O)NC(C1C(=C)C1C(=O)OC)=O 72743,CCCCCC(C)CC(=O)N1CCC(NC(=O)CCc2ccc(O)nn2)C(F)C1 72744,C(=O)(CC(C)CC(C)(C)C)N1C(C(N(C(C)C)C)=O)CSC1 72745,C(=O)(CC(F)(F)Cl)NC(c1ccc(F)cc1)CNC(C12CC(C)(C1)C2)=O 72746,CC1Cc2cc(C(=O)NC3COCC3NC(=O)Cn3cnnc3)ccc2O1 72747,C#Cc1nccnc1NC(=O)NC1CCC(COCCC)CC1 72748,N1(C(C(CC)(C)O)=O)CC(NC(c2cc(C)cc(C)n2)=O)CC(O)C1 72749,N1(C(CC(n2c(CC)ncc2)C)=O)CC2CC1CN(C(c1ccc(C)s1)=O)C2 72750,CC(Cl)(Cl)C(=O)N1CC(C(N)=O)(CNC(c2ccc(C(F)F)o2)=O)C1 72751,C1(CNC(CC2N(C(C3CN(C(C)C)C3)=O)CCCC2)=O)OC(=O)NC1(C)C 72752,c1(NC(c2n(C)cc(NCc3ccc(Br)[nH]3)n2)=O)ccc(Br)cc1C(C)(C)C 72753,c1(OC)ccc(C(=O)NC2CCN(C(c3cc(C)ccn3)=O)C(C)C2)c(F)c1Cl 72754,C1(C(N2CCOC3CC23)=O)C2CC(O)C(C2)N1C(=O)COC1CCCCC1 72755,N1(S(CC)(=O)=O)CCC(C(=O)NCc2ncc(-c3cccc(Cl)c3)[nH]2)CC1 72756,N1(C(C2(c3c(C)cccc3)CC2)=O)C2CCCC1CC(NC(=O)C(C)(C)O)C2 72757,c1(C(N2CC(C(=O)OCC)C2)=O)cnc(CNC(=O)CC2CCC(=O)C2)nc1 72758,N1(C(C(C)C2(O)CCC2)=O)CCN(C2CN(C(=O)COC3CC(F)(F)C3)C2)CC1 72759,c1(C(N2CCC(CCC(=O)NCc3cncc(Cl)c3)C2)=O)c[nH]nc1[N+](=O)[O-] 72760,C1(CNC(C(CC)F)=O)CC2(CCN(C(C34CCC(F)(CC3)C4)=O)C2)CO1 72761,c1(OC)ccc(CCC(N2CC(O)(CNC(=O)C(C)C3CC3)C2)=O)cc1 72762,C1(C(=O)NC(C)(C)C)CCCCN1C1COC1.C(CCCNC(C=C)=O)N(C)C(=O)O 72763,c1(C(=O)NC2CCCC(CNC(C(=O)NCC)=O)C2)c(C)cnnc1O 72764,c1(C(N2CC(NC(c3n(CC)ncc3)=O)CC2(C)CC)=O)ccc2n[nH]cc2c1F 72765,C(=O)(CCCC(C)(C)C)NC1C(CNC(c2ccc(C(OC)OC)o2)=O)C1 72766,c1(CNC(=NCC=C)NC(C)CCOC)ccc(S(=O)(=O)N(C)C)cc1 72767,C1(CN(C(C2C(C)=C2)=O)C)CCCN1C(C1CCC(=O)N1)=O 72768,C12(CNC(C3CC4(CCC4)C3)=O)CCCC1CCN2C(c1cc2c(s1)CCC2)=O 72769,C(=O)(CC(C)(C)C1CC1)NCCCC(C)NC(=O)CC1C=NN(C)C1=O 72770,CC1CCCn2cc(C(N3CCCC4(NC(=O)CC5CC(F)C5)CC4C3)=O)nc21 72771,c1(C(N2CC3C(CNC(c4c(CC)onc4C)=O)(C3)C2)=O)ccc(F)cc1O 72772,C1(CN(S(C)(=O)=O)C)CCN(C(=NCC2CC2)NCC2CCCOC2)C1 72773,c1(CC(=O)N(C(CNC(CC(C)O)=O)C2CC2)C)ncncc1Cl 72774,C1(NC(C(C)=CC2CC2)=O)CC(C(=O)N(C)Cc2cnccn2)C1(C)C 72775,C#CCCCC(C)C(=O)N1CCC2(CC2NC(=O)C(c2ccccc2F)C)C1 72776,C(CC(F)(F)C(C)C)NC(CC(CNC(C1COC(=O)N1C)=O)OC)=O 72777,CCC(C)CCCC(=O)NCC1CC(C(=O)NCCOCC(N)=O)C1 72778,CS(=O)(=O)c1ccc(C=CC(N2CC3CC(C2)N(C(=O)C(F)C(F)(F)F)C3)=O)o1 72779,Cc1ccc(C(N2CCCC(NC(c3cc(N)ccc3C)=O)C2)=O)c(F)c1 72780,N1(C(C2CCN(OC)CC2)=O)C2CCC1C(F)C(NC(=O)C(C)CC(N)=O)C2 72781,C1(C(=O)Nc2c(C)nco2)C2CN(C(c3coc(C(=O)N(C)C)c3)=O)CC12 72782,N1(C(C(C)Cn2cccn2)=O)CCC2C(NC(c3ccc(Cl)s3)=O)CC12 72783,C1(C(=O)OC(C)(C)C)C(C2CC2)CCN1C(=O)C(N1CCC(n2cccc2)C1)=O 72784,C(=O)(CC(CC1CC1)NC(=O)CC(O)CN(C)C)NCCc1scc(C)n1 72785,N1(C(CN(C)C2CC2)=O)CC(C2CCN(C(c3ccc(OC(F)F)cn3)=O)C2)C1 72786,N#CC1(C(=O)NCC=CCNC(=O)CC2CC2(Cl)Cl)CCC(=O)CC1 72787,CC1(C)CCCC1C(=O)NC1CCN(Cc2cn(-c3ccc(Cl)cn3)nn2)C1 72788,N1(C(C(C(C)C)O)=O)CC(NC(C23CC(c4ccccc4)(C2)C3)=O)CCC1C 72789,c1(C(N2C(C(N3CCC(N(C)CC)C3)=O)CNC(=O)C2)=O)cccc2cncn12 72790,c1(C(N2CCC(CNC(CC(C(F)(F)F)OC)=O)C2)=O)cc(O)c2sccc2c1 72791,O=C1CCC(N=c2[nH]c(NC3COCC3C(F)(F)F)nc3c2CCCC3)CN1 72792,C1(C(=O)NC(CC(=O)OCC)c2ccccc2)CCCN(C(C)CNC)CCO1 72793,C1(OC)CC(NC(=O)CCn2ccnc2)CN(C(C2(C#N)CCCC2)=O)C1 72794,C1(C(N(C(C(=O)NC)C)C)=O)CC2(CCN(C(c3cnc(O)o3)=O)C2)C1 72795,c1(C(N(CC(CC)NC(=O)CNC(C)=O)C)=O)cc(Br)cc(C)c1F 72796,C1(CNC(C2N(C(CSC)=O)CC=CC2)=O)CCCC2(CC2)C1 72797,C12(NC(CCCC(=O)NC(C)C)=O)CCC(CN(C(=O)C(F)OC(F)(F)F)C1)C2 72798,C1(CC(C)C)CC(C(=O)NCCC2CCN(C(=O)CCF)C2)CC(=O)N1 72799,C1(C(=O)Nc2cccc(OC)n2)CCN(C(c2cncc(F)c2)=O)CC1O 72800,N1(C(CCN(C)C)=O)CC(C(=O)Nc2cc(N(C)C)ccc2F)CC(F)(F)C1 72801,CCC(O)CCNC(=O)CC1(CNC(=O)Cc2ccsc2C)CC1 72802,C1(NC(C2C(C)C2)=O)CC12CCN(C(c1ccc(C(F)F)cn1)=O)C2 72803,N1(C(C2C(OC)CC2)=O)CCCC2(NC(c3coc(C(C)C)n3)=O)CC2C1 72804,c1(C(N2CCC(C)C2)=O)c(CNC(c2cc(Cl)cs2)=O)cnn1C 72805,c1(SCC(=O)NC2CCC(CC)C2)nnc2ccccn12.C12CN(C1)CC(=O)NC2 72806,c1(C(=O)NC(CC)CN(C)C(c2cc(Cl)n(C)n2)=O)cccc(F)c1C#N 72807,C(C(CC)CC)(c1n(CCOC)nnn1)NCc1cccc(OC)c1 72808,C1(C(=O)NC2C(C(=O)NC(C)C(F)F)CCC2)CCCC(=O)N1C 72809,C(=O)(C1=CCCN(C(=O)Nc2ccccc2)C1)NC(C(C)(C)C)CCO 72810,C(=O)(C1CCOc2ccccc21)N(C(CNC(Cc1c(C)nc[nH]1)=O)C1CC1)C 72811,c1(C(N2C(CNC(C3CC3F)=O)CCCC2)=O)cn2cc(Cl)cc(Cl)c2n1 72812,c1(C(N2CCC(n3cc(-c4c(N)cccn4)nn3)C2)=O)ccc2cccnc2n1 72813,N1(CC(=O)NCC(C)(C)NC(C2CC23CCOC3)=O)CCS(=O)(=O)CC1 72814,N1(C(c2cnc(C)[nH]2)=O)CCN(C(C2CC=CCO2)=O)CC1CS(C)(=O)=O 72815,CCC(CC)C(C)C(=O)NC(C)(C(=O)NCc1ccc(F)cc1C)C1CCC1 72816,CN1CCC(C(=O)NC2CC2NC(=O)C=Cc2cccc(CO)c2)S1(=O)=O 72817,c1(C(=O)NCC2CCCN2C(=O)CN2CCCC2)ncncc1Cl 72818,N(C1CC2(CN(C(C3CC(C)N(C)C3)=O)C2)n2ccnc21)C(CC(=C=C)C)=O 72819,O=C1CCC(NC(c2ccc(Cn3cc(CC4CC5(CC5)CO4)nn3)o2)=O)C(=O)N1 72820,N#CC1CCCC1NC(=O)CC1CCN1C(C1CCCSC1)=O 72821,C(CCCCC(=O)NCC(O)CC(=O)N(C)CCc1nccs1)N(C)C 72822,C1(NC(=O)C=CC2CCCC2)CCN(C(c2cc(Br)ccc2OC(F)F)=O)CC1F 72823,Cc1nc(SC(F)F)sc1CC(=O)N(CCC(C)NC(=O)CC(C)N(C)C)C 72824,CN1C(=O)CN(CC(=O)NCCCN2CCN(C(=O)C3=C(Cl)CCC3)CC2)C1=O 72825,c1(C(=O)NCC(CNC(CNS(NC)(=O)=O)=O)F)ccc(C(F)(F)F)nc1 72826,S(=O)(=O)(c1ccc(C#N)c(N(CC(C)OC)C)c1)N1CC(CC)C2(C1)OCCO2 72827,c1(C(=O)NCc2c(SC)cccc2)cnc(N)c(Br)n1 72828,Cc1c(C(=O)NCC2(NC(C3C(Cl)(Cl)C34CC4)=O)CC2)sc2ccsc12 72829,C(=O)(CCS(=O)(=O)CC(C)C)NCC1N(C(c2cc(C(C)=O)sc2)=O)CC=C1 72830,N1(C(C2(CN(C)C)CCCC2)=O)CCCC(CO)(NC(C2CC(CF)C2)=O)C1 72831,C(CC(F)F)(C(=O)N(C)Cc1ccsc1)NC(C1C(C)C1)=O 72832,C1(C(N2CCC(CCC)C2)=O)C(C2CC2)CCN1C(=O)CC1COCC(C)O1 72833,C1(NC(CNC(=O)NC)=O)CCC2(CC1)CN(C(=O)C(C)(CC)CO)CCO2 72834,N1(C(CCC=C)=O)CCC(C(=O)NC2CN(CCC)C2)=C(F)C1 72835,O=C1NCC2(CCN(C(c3cccc4ccoc34)C(=O)NCc3ccco3)C2)O1 72836,C(=O)(C#CC(C)(C)O)NC(C(NC[Si](C)(C)C)=O)C1(O)CCC1 72837,c1(N2CCN(C)CC2CNC(c2ccc(O)nc2)=O)nc2ncc(Cl)cc2o1 72838,c1(NC(C2N(C(c3ccc(OC)c(C)c3)=O)CC2)=O)sc2ccccc2c1C#N 72839,c1(C(=O)NC(CC)CN(C(=O)C(C)C2CC2)C)ccnc(N2CCCC2)n1 72840,N1(C(c2cccc(NC(c3ccc(I)c(O)c3)=O)c2)=O)CCn2cccc2C1 72841,C1(CNC(C(C)OCC#C)=O)CCN(C(c2cc(C)nn2C2CC2)=O)CC1(F)F 72842,C(C(=O)NCCCCC(C)NC(=O)C(C)Cc1cnc[nH]1)(C(C)C)SC 72843,c1(-c2ccc(C(=O)NCCOCCCNC(C3CCSC3)=O)o2)cccc(F)c1 72844,C=C(CNC(=O)CC(C)C(=O)NC)c1ccccc1F 72845,C(C(C)(O)C(=O)N1CCCC(CC(=O)NCC(C)(C)OC)C1)OC 72846,C1(CNC(=O)CCc2ccoc2)CCCCCN1C(=O)CC1CC2(CCC2)CO1 72847,C1(C(=O)NC2CC23CC(NC(c2ccc(OC)cc2)=O)C3)(CC)CC(C)(C)C1 72848,C1(NC(=O)CCc2ccccc2)CCCCCN(C(C2CN3CCN2CC3)=O)C1 72849,N1(C(c2c(SC)cnn2C)=O)CC2CCN(C(c3cc4n(c3)CCOC4)=O)C2C1 72850,C(CCCCCN(C)C(C1CC=C(C)CC1)=O)NC(C(C1CC1)OCC)=O 72851,C(C(C)(C(N)=O)NC(C1CC(NC(C2CCCOCC2)=O)C(O)C1)=O)OC 72852,N1(C(c2cc(C(N)=O)cs2)=O)CCN(C)C(CNC(C2(OC)CCC2)=O)C1 72853,N1(C(C(C=C)OC)=O)CC(NC(c2cc(C)nc(O)c2)=O)CC12CCC2 72854,C(C(C)(CC(C)C)NC(=O)Cn1cc(CO)nn1)NC(c1[nH]nc(OC)c1Cl)=O 72855,c1(C(=O)NCC2(SCC)CC2)ccc(SC2(CC#N)COC2)c(OC)c1 72856,c1(CCC(=O)N(C)CCNC(C2CC(=C3CCC3)C2)=O)ccsc1Br 72857,C1(CC)(NC(=O)CCCc2ccncc2)CCN(C(=O)C(O)C2CCCC2)CC1 72858,c1(CNCC2(C)N(C(C(c3cccc(C(C)C)c3)C)=O)CCC2)cc(O)ncc1Br 72859,C1(NC(CCOC)=O)CCN(C(c2ccc(-n3ccnc3)nc2)=O)C12CCC2 72860,C1(NC(c2ccccc2-c2ccccc2)=O)CCCCC1NC(C12CCC1C2)=O 72861,c12ccc(cc1)OC1CC=CC(C1)n1cc-2nn1.C(C(O)CCO)SCC.C1(OO)CC1 72862,c1(CNC(C2Cc3nccnc3C2)=O)cc2n(n1)CCNC2 72863,c1(CCC(N2CC(NC(c3cncc(C)n3)=O)C(C)C2)=O)ccc(C)c(F)c1 72864,Cc1cc(Br)ccc1NC(=O)C(c1cnsc1)N1CCC1C(C)C 72865,c1(C(=O)NCC2C(C)CCCN2C(C2CC(O)C2)=O)cnn2c1CCCC2 72866,c1(C(N2CCC(OC)(CNC(=O)C(CO)N(C)C)C2)=O)c[nH]c2cc(F)ccc12 72867,C12(NC(c3c(N)ccc(Cl)c3)=O)CCCC1CN(C(=O)CCCC1CC1)C2 72868,c1(CN2CC(NC(c3cc(NC(C)=O)c(F)cc3)=O)C2)c[nH]c2ncc(Cl)cc12 72869,c1(C(=O)NC2(CNC(c3cccc(C)n3)=O)COC2)cc(F)c(Cl)nc1Cl 72870,O=[N+]([O-])c1cc(CCN2CCCC(n3nccn3)C2)cc(Cl)c1 72871,C(=O)(N=c1cc(C(N)=O)n(C)[nH]1)C1C2(CN(C(CC(C(CC)C)O)=O)C2)CCC1 72872,CS(=O)CCC(O)C(=O)NCC12CC(NC(=O)CCCC3CC3)(C1)C2 72873,c1(C(=O)NCC2CC(NC(c3cn(CCO)nn3)=O)C2)c[nH]c(=S)cn1 72874,c1(OC)cccc(N(C(=O)CN2CCCC(N3CCOC3=O)C2)C(C)C)c1 72875,Cc1cc(C(N2CC(C)CC2C(=O)NC(CF)C(F)(F)F)=O)nc(C)c1 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72893,C(CN=C(NCC(C)(O)CCC(C)C)NCCO)CC=C.C1(C)(O)CCC1 72894,N1(C(=O)CNC(CSC)=O)CC(NC(C2CCCN2c2ccncn2)=O)C(C)C1 72895,c1(C(=O)O)ccc(C(c2cn(CCCCCO)nn2)O)cc1.C(=O)(C(F)C1CCC1)N 72896,c1(C(=O)NC(C(C)C)C(N2CCC(N=[N+]=[N-])C2)=O)coc2c1COC2 72897,C1(C(=O)NCC2C(NC(CC(=O)NCC)=O)C2)CCC(OC)CC1 72898,CCCCC(CC)CC(=O)NCC(C1CCCC1)NC(=O)Cc1c[nH]nc1C 72899,C=CCCCCCCC(=O)N1CCN(C(c2ccc(F)c(O)c2)=O)C(C2CC2)C1 72900,c1(C(N2CC(C)C(NC(=O)CC3CCC(F)(F)CC3)C2)=O)onc2ccccc12 72901,C1(NC(C2CCC(C)(C)C2)=O)CC2CCC(C1)N2c1nnc(C(F)F)s1 72902,CC1CCc2[nH]c(=NC(C)c3cn(C)cn3)[nH]c(=NCC3(N(C)C)CC3)c2C1 72903,C(C)(CN=c1[nH]nc(C)s1)(C1CC1)NC(C(C)OCC#C)=O 72904,C1(C(=O)NC(=O)OC(C)(C)C)CC(O)CN1C(c1cc(Br)sc1Cl)=O 72905,C1(OCC#C)CCN(C(=O)CCC2CC2C(=O)OC)C1 72906,C(=O)(CS(=O)(=O)N1CCOCC1)NCC(C)N(C)C(c1ccc(C(C)O)cc1)=O 72907,c1(-c2nc(C3CCN(C)CC3)nn2CCS(N)(=O)=O)cnc2ccnn2c1O 72908,c1(OCC)cc(C(=O)NC2CC(NCc3ccncc3F)C2)cc(F)c1 72909,c1(NC(C2CCCCCC2)CNC(C=CCC)=O)c(CC)c(C)nc2ncnn12 72910,C=CCC(C)(C)C(=O)NCC1(NC(c2cccc(-n3ccc(CC)n3)c2)=O)CC1 72911,CCC(CNC(=O)C(CN=[N+]=[N-])NC(=O)Cc1cc[nH]n1)(CC)C(N)=O 72912,c1(C(=O)NC2CCCN(C(c3ccc(CC)s3)=O)C2)cc(C)c(C)nc1C 72913,c1(CN2CCN(c3ncc(C)cn3)C(C(F)(F)F)C2)ccc2c(c1)C(=O)C(=O)N2 72914,C(=O)(C1=CCC2CCC1N2C(=O)C(CN(C)C)N(C)C)NC(C#C)(CC)CC 72915,N1(C(c2ccc(C)cc2)CC)CCN(Cc2cnn(C)c2N)CC1C 72916,c1(NCCC(C)OC)[nH]c(=NCc2cc(F)ccc2C(F)(F)F)nc2scnc12 72917,N1(C(C(=O)NCCC2CC2)C2(CC)CC2)CC(C)(C)C2COCC12 72918,C#CCC(CC(=O)NCC1CCCN1C(c1cnn[nH]1)=O)c1ccccc1 72919,C1(C(=O)NC(C2CCOC2)C#C)CN(C(=O)CCCC2CC2C)CC1(F)F 72920,c1(NC(C2OCCC(NC(C(C=C=C)C)=O)C2)=O)cc(O)ccc1OC 72921,CC1CC(c2ccccc2)CN(C(=O)C(=O)NCCN2CCCCC2=O)C1 72922,N1(C(C(C=C=C)C)=O)CC(CNC(c2nc(Br)sc2C)=O)CC1(C)C 72923,C1(C)(CNC(c2c(C)ncs2)=O)CCCN1C(c1cn(CC2CCCO2)nn1)=O 72924,Cc1cc(Cl)cc(N)c1C(=O)NCC1CC1NC(=O)C(CO)C(C)(C)C 72925,N1(C(C2C(OC)C2)=O)CCC2CN(C(c3cnc(OC)c(C(F)(F)F)c3)=O)CC12 72926,C1(F)(CNC(C(C)(C)c2cscn2)=O)CCC(NC(=O)C(N)=O)C1 72927,c1(N(CC)CC)ccc(NC(=O)C(=O)NCCCC#N)c(O)c1 72928,C(=O)(C(O)CC(C)C)NC(COC)CC(=O)N(C)CCN1CCOC1=O 72929,c1(C(N2CCC(OCCNC(C3CC(C)O3)=O)CC2)=O)cc2c([nH]1)CCCC2 72930,c1(NC(C)=O)ccc(C(=O)N(C2CCN(C(C3C(C)C3C)=O)C2)C)cc1 72931,C1(NC(=O)CC2(O)CCOC2)CCC2CC1CN2C(c1nc(F)ccc1Cl)=O 72932,c1(CC)oc(C(=O)NC(C)(CNC(c2cccc(C)c2)=O)C2CC2)cc1C 72933,c1(CC(N2CCC(C)(CCNC(c3ccc(C)cc3)=O)C2)=O)cccc(C#N)c1 72934,c1(SC)cccc(C(=O)NC(C)CCCNC(c2cc(C#N)on2)=O)c1Cl 72935,c1(C(=O)NC2C3CN(C(c4[nH]c(=N)sc4)=O)C(C3)C2)cc2cc(F)c(F)cc2[nH]1 72936,N1(C(CC(C)(C)C2CC2)=O)CC(C(=O)NOC2CCC(O)C2O)C2(CCC2)C1 72937,N1(C(=O)CC2CCCO2)CCCCC1CC1(F)CC(CNC(C23CC2C3)=O)C1 72938,N1(C(c2n(CC)ncc2)=O)CCCC(CO)(NC(=O)CN(c2ccncc2)C)C1 72939,C1(NC(C2C(C(=O)NCCO)C2)=O)CCCN(C(c2ccccc2O)=O)CC1 72940,N1(C(=O)CCc2cncnc2)CC(C2CC2)(C(=O)Nc2ccc(O)c(F)c2)C1 72941,CC(CF)CC(=O)N1CCN(C(c2cn(-c3ccccc3Br)nn2)=O)CC1 72942,C(=O)(C(C)(C)CC#N)NCCN(CC(C)O)C(=O)CN1CCCC1=O 72943,c1(C(=O)NCC(C)CNC2(COC(C)(C)C)CC2)ncccc1[N+](=O)[O-] 72944,Cc1nccc(Cl)c1C(=O)NC1CC(F)CN(C(c2nccn2C)=O)C1 72945,N1(C(C(CCC)CCNC(=O)COC2CCOC2)=O)C(C)CC2CCCC12 72946,CC1CC(CC(=O)N(C)CC2CN(C(C3CCCCC3C)=O)CCO2)C(C)O1 72947,c1(C(=O)NCC2(C)CCCN(C(=O)C(F)C3CCC3)C2)ccc(=O)n2c1CCC2 72948,N1(C(C(C)C)=O)CC2(C1)CN(C(c1cccnc1-c1ccccc1)=O)C2 72949,CCCCC(C)CC(=O)N1CCN(C)CC1CNC(=O)C=NOC 72950,c1(OC)cc(Cl)c(C)cc1C(N1CCN(C(c2ccc(C)n2C)=O)C2CC12)=O 72951,Cc1c(C(N2CCCC(CNC(=O)C=Cc3cccs3)C2)=O)nn2c1CCCC2 72952,C1(NC(c2ccsc2Cl)=O)CCCC1n1cc(C2C3COCC23)nn1 72953,C(=O)(C(COC(C)=O)NC(C1CC1(Br)Br)=O)OC 72954,C1(C(=O)NC2C(NC(C3OCC(C)(C)C3)=O)CCCCC2)CC2C=CC1C21CC1 72955,N1(C(CCC)=O)CC2C3CCC(C2C1)N(C(c1cccc(C(=O)OC)c1)=O)C3 72956,C(=O)(CC1=CCOCC1)NC1CC(CNC(C2(COC)CCC2)=O)CC1O 72957,Cc1cnc(N2CC(NC(=O)CC(=O)NCC(F)(F)F)CCC2C)nc1O 72958,c1(OCCC)c(OCCC)cc(C(C)C)cc1Cl.C1(CN)CC2(C1)CC2F 72959,N1(C(C(C)OCC=C)=O)CCC(F)C(NC(=O)CC2(OC)CCCCC2)C1 72960,c1(C(N(CC(CNC(Cc2c(C)cco2)=O)(C)C)C)=O)c(C)nsc1C 72961,C1(NC(C(C)N2CCC2)=O)COCCN(C(c2c(Cl)csc2Cl)=O)C1 72962,N1(C(CN(C)C)=O)CC(NC(C2CC(=O)N(CCN(C)C)C2)=O)CC(F)C1 72963,C(=O)(CC1OCCc2ccsc21)N(C)CCNC(=O)C(C)(C)c1sccc1Cl 72964,c1(C(C(=O)NCCN(C)C)N(CC)CC2CCC2)c(CO)nnn1C 72965,C#Cc1ccc(OCC(N2CCOCC2CNC(C2CCCN2N=O)=O)=O)cc1 72966,S(=O)(=O)(C1CCN(C2CCOC(C)(C)C2)C1)NC 72967,C(C1CCCN1C)=CC(=O)NCCCN(C(C(C)=C1CC1)=O)C(C)C 72968,Cc1cccc(C2(C(=O)NC(C)CC(C)NC(=O)CCN3CCCC3)CC2)c1 72969,c1(C(N2CC(CNC(C3CC(O)C3)=O)C3(CC3)C2)=O)cc(Cl)ccc1OCCF 72970,c1(C2C(CC(N3CC(C(C)NC(=O)CN4CCCC4=O)C3)=O)C2)ccc(Cl)cc1 72971,C1(CCNC(C2C(C)C2)=O)CCN(C(=O)OC(C)(C)C)CC1(F)F 72972,C1(O)(C(C(=O)NC(CNC(CC2C(C)C2)=O)C2CCC2)(F)F)CCOCC1 72973,Cc1cccc(C(=O)C(C)N(C)C(c2cc(-c3ccoc3C)[nH]n2)=O)c1 72974,c1(C(N2CC(C3(NC(C4N(C)CCC4)=O)CC3)C2)=O)cc(F)c2cn[nH]c2c1 72975,c1(C(=O)NC(CNC(=O)CC2CCC2)C2CC2)cc(F)cc(Br)c1 72976,O=C(C1=CCCS1)NCCCN1CCN(C(=O)COc2ccc(Cl)nc2)CC1 72977,C1(C(=O)NC2(C)CCN(C(C3CCC(CCC)CC3)=O)C2)CCC2CC1C2(C)C 72978,C1(NC(C=C(Cc2c(OC)cccc2)C)=O)CC2CC(NC(C3CC3C)=O)CC12 72979,N1(C(C(CCSC)O)=O)CC2C=CC1C(C(N1CC(NC(N)=O)C1)=O)C2 72980,c1(CN2C(C(N3CCC3CO)=O)CC3CC32)cc(F)c(O)c(F)c1 72981,N1(C(C2(C)CS(=O)(=O)C2)=O)CC2=C(C1)CN(C(c1cnn3c1SCC3)=O)C2 72982,N1(C(C(C2CCN(C(=O)C(F)=CC3CC3)C2)C)=O)CC2OC(=O)N(C)C2C1 72983,N1(C(c2ccc(N3CCC3)nc2)=O)CCSCC1CCNC(C1C=CCCC1)=O 72984,N1(C(COCCOCCOCC#C)=O)CC(CCNC(n2cccc2)=O)C1.OCC 72985,c1(CC)ncc2c(n1)CCC(C(=O)NCCCNC(c1ncnc(C)c1C)=O)C2 72986,c1(C(=O)NC(CCC(C)C)C)cccc(N=c2cncc[nH]2)c1 72987,CC(C)(F)CCC(=O)NCC1CCCC1NC(c1cnoc1-c1ccccc1)=O 72988,CCCCCCCCCC(=O)NCC(C1CC1)NC(C1CC=C(C)CC1)=O 72989,CCC(CN=c1[nH]c(N(c2cc(C)cc(C)c2)C)nc(=NC)[nH]1)N1CCCCC1 72990,c1(C(=O)NC(CNC(C=CCOC)=O)C(C)C)cnc(O)n(-c2ccccc2)c1=O 72991,N1(C(Cc2c(C)noc2C)=O)CC2CCCC2(NC(c2cc(C(F)F)no2)=O)C1 72992,N1(C(C(C)=C2CCOC2)=O)CC2CCC(CNC(=O)CCC3CCCCC3)C2C1 72993,N1(C(C=CC2(C)COC2)=O)CCC(CNC(=O)Cc2cn[nH]c2)C(O)C1 72994,C1(C(N2CCC(OCCNC(C=C(CC)C)=O)C2)=O)CCN(C2CC2)S1(=O)=O 72995,Cc1cc(Cl)cc(C(=O)NC2C3CN(C(=O)CC4CCCOCC4)CC23)c1O 72996,CCCCC(CNC(=O)CC1(C)OCCCO1)NC(=O)OC(C)(C)C 72997,C=CCC(CC(F)F)C(=O)N1CC2CC(C1)N(C(C1CC3COCC3C1)=O)C2 72998,N1(C(c2c(C)coc2)=O)CCCC(C2CN(C(=O)CCCc3ccncc3)C2)C1 72999,C1(C(C)C)CN(C(c2cc(C)cc(O)c2)=O)CCN1C(=O)CN(C)C(N)=O 73000,S(=O)(=O)(c1ccc(C(=O)OC)cc1Cl)Nc1ccc(C#C)c(Br)c1 73001,C1(CNC(CCCCN(C)C)=O)CC2CCC1N(C(c1nc(Cl)sc1Cl)=O)C2 73002,CC1CN(C(c2cc3n(n2)CCCC3)=O)CCN(C(=O)COC(C)(C)C)C1 73003,CCC(CNC(=O)C=Cc1ccsc1)(CC)NC(C1CC2CC2C1)=O 73004,c1(NC(C)CN2CCCC2=O)nc(N(C)CCn2cnnc2)nc2c1CCC2 73005,CC1CC(CCC(=O)NCC#CCNC(=O)CCc2ccn(C)n2)C(C)N1C 73006,C12CCCCCN1CC(=O)N2.C1(N(C)C)CCN(C(=O)OCc2ccccc2)C1 73007,c1(C(N(CC(CC)NC(c2ccc(CO)s2)=O)C)=O)c[nH]nc1Br 73008,c1(C(N(CCC)CCCC(N)=O)=O)cc(S(=O)(=O)NC2CCC3CC23)c[nH]1 73009,C1(NC(N2CCC(CNC(c3ccn(C(C)(C)C)c3)=O)C2)=O)CCC2(CC1)CC2 73010,C(C(CC)N=c1[nH]c2ncc(Cl)cc2o1)NC(COCCCC)=O 73011,C=CCCCC(=O)NCC=CCC(=O)NCC1CCC(C)CO1 73012,C1(CNC(C)CS(C)=O)(NC(=O)OC(C)(C)C)CC12CCC2 73013,N1(C(c2nnc(C)s2)C(=O)NCc2cccs2)CCn2ncc(Cl)c21 73014,c1(CC)ccccc1CC(=O)NCC(C)CN(C(=O)CCSc1nccn1C)C 73015,Cc1nc(CCNC(c2nnnn2CCN2CCOCC2)(C2CCOC2)C)cs1 73016,c1(C(C(=O)NCC=C)N(CC=C)C2CC2)ccc2nonc2c1 73017,n1(CC(N2C3CN(C(c4ccc(C)s4)=O)C(C3)C2)=O)cc(C(N)=O)c(O)nc1=O 73018,c1(C(=O)NC2CN(C(C3CN4CCN3CC4)=O)CCC2F)ccc2oncc2c1 73019,N1(C(C2C(C)(C)C2(F)F)=O)CCCC2(C1)OCC(O)C2O 73020,C1(CN(C(=O)CSc2cnn(C)c2)CC)CCCCN1C(=O)C=Cc1ccco1 73021,N1(C(C(CNC(c2c(C)snn2)=O)C(C)C)=O)C2CCC1CC(O)C2 73022,N1(C(C2CC(OC)C2)=O)CC(CNC(=O)C=C(C)c2ccccc2)C2(CCC2)C1 73023,Cn1ncc(C(=O)NCc2csc(CNC(C3C=CC=CC=C3)=O)n2)c1F 73024,C(=O)(CC(C)(C)C(C)=O)NC1CC(C(=O)NC(c2ncco2)CC)OCC1 73025,Cn1ccc2[nH]c(C(=O)NC3CCC(NC(=O)Cc4csc(NC=O)n4)C3)cc12 73026,c1(C(N(C(c2nn[nH]n2)C#C)C)=O)ccnc2[nH]c(C(F)F)nc12 73027,C1(Nc2cc(C)c(C(F)(F)F)nc2)CCN(C(=O)C(=O)N(C)C)C12CCC2 73028,N1(C(c2nc(CC)sc2)=O)CCOC(C)(CNC(=O)C(F)C2CCC2)C1 73029,c1(COC)cc(C(=O)NCCCCN(C)C(C2CC2c2cncn2C)=O)no1 73030,Cc1ccc(O)c(C(N2C(C(N3CCN(CCO)CC3)=O)CC3CC23)=O)c1 73031,c1(CC)[nH]c(Cl)nc(=NCC2CN(C(c3ccncc3OC)=O)C2)c1C#N 73032,c1(C(=O)NC(C)CCN(C(=O)Cc2ccccc2CO)C)ccc(N=[N+]=[N-])cc1 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73157,C(=O)(C1CCCc2scnc21)N1C(CNC(c2c(C)[nH]c(=NCC)s2)=O)CCC1 73158,CC1COCCCN1C(C1CCCC1CNC(c1ncccc1CO)=O)=O 73159,CCCC(C)CCCC(=O)NCC1(F)CCC(CNC(=O)CC2CCC2)CC1 73160,C(=O)(C(C#N)(CC)CC)N(C1CCC(NC(=O)CN2CCCCCC2)CC1)CC 73161,c1(-c2nc(=N)[nH]cc2)cc2cc[nH]c2cc1C(N1CCC2(CC1)CC2(F)Cl)=O 73162,C1(NC(C2(C)C(C)C2)=O)CCC2(CC1)CN(C(=O)Cc1ccccc1O)C2 73163,C1(COC(=O)C(F)n2cccn2)C(F)(F)C12CC2 73164,c1(NC(CC=C)C)[nH]c(=NCc2cnc[nH]2)nc2c1cnn2C 73165,C(=O)(C1CCOc2ccc(Cl)cc21)N1CC(C)CC(NC(C=CC)=O)C1 73166,C1(NC(c2cc(CNC(=O)C(F)CC3CCOC3)cs2)=O)CCC2(CC2)C1 73167,C(CC(CNC(c1cc(C)co1)=O)NC(=O)C(=CC1CCCC1)C)OC 73168,CCCCC(C)(F)C(=O)NC1CCCCC1NC(=O)CCCc1ccc(F)cc1 73169,C1(C(=O)Nc2ccc(C(N)=O)cc2)CN(C)CCN1C(=O)C(F)C(F)(F)F 73170,C(=O)(C1=CC2(CCOC2)C1)NC(C(=O)N(C(C#C)C1CCC1)C)CC1CC1 73171,c1(C(C)C)n[nH]c(=NC(C)C2CCCN(C(c3cccc(C(C)C)n3)=O)C2)o1 73172,C(=O)(C1=CS(=O)CCC1)NCC12CC(NC(CC(=O)N(C)C)=O)(C1)C2 73173,CCC(C)C(C(=O)OC(C)(C)C)OC(c1ccccc1NCC(C)S(C)(=O)=O)=O 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73208,CCCCCCCCCCCCN(C(=O)Cc1ccc(OCCC(=O)O)cc1)C 73209,C1(NC(C2(CC)CCC2)=O)CN(C(c2cccc(N(C)C)n2)=O)CC2CCCC12 73210,N1(C(c2ccc(NC(C)=O)s2)=O)CCC(C)(C)C1CNC(C1CC(=O)N(C)C1)=O 73211,c1(C(N2CCC(NC(C3CCC(=O)O3)=O)C2)=O)ncc(F)cc1F 73212,C12(C(N3CCC(NC(CNS(NC)(=O)=O)=O)C3)=O)CCC(=O)N1CCS2 73213,c1(C(=O)NC(CC)CN(C)C(c2cc(C3CC3)no2)=O)ccnnc1C 73214,C(=O)(C(C)CC(F)(F)F)NC1C(NC(c2onc(OCC)c2Br)=O)C1 73215,CC1(C)CCCC(O)(CNC(=O)Nc2ccc3ccoc3c2)C1 73216,CC1CCN(C(c2ccccc2C(=O)NC2CC(NC(C)C)C2)=O)CC1 73217,C1(CCC(=O)NC(C)C(C)NC(C2CC(OC3CC3)C2)=O)CCCOC1 73218,N1(C(C(C)CC(F)F)=O)CCC2C(CCCN2C(=O)CN2OC(C)(C)CC2=O)C1 73219,c1(CNC(c2n(CC(=C)C)nnn2)(C)CC2C=CCC2)nc2c(s1)CCC2 73220,N1(C(C2CCC(CC)O2)=O)CC2CCC2(CC(=O)NCCc2ccc(C)cn2)C1 73221,c1(C(CCC)C)cn(CC(=O)OC)nn1 73222,CCS(=O)c1ccccc1C(=O)NC1CCN(C(=O)C(=O)N(C)C)CC(C)(C)C1 73223,C1(NC(C(c2cc(C)oc2C)C)=O)CC2CN(C(=O)CCc3cn[nH]c3)CC2C1 73224,C(CCCC(=O)NC1(C)CN(C(C2CCC(C#N)C2)=O)C1)NC(C)=O 73225,C1(C(N2CC(NC(C3(C)CCCC3)=O)C2)=O)CCC(N=[N+]=[N-])C1 73226,CN1C(=O)C(F)CC1C(N1CCCCC(NC(c2ccc(C3CC3)nn2)=O)C1)=O 73227,c1(N2CC(NC(c3c(C)cn(C)c3)=O)C(C)(C)C2)c(F)cccc1[N+](=O)[O-] 73228,C(=O)(C(C)CCC(C)(C)C)NCC1(F)CCN(C(C(C)NC(CC)=O)=O)C1 73229,C1(CCn2cc(CCCC=C)nn2)CCCCN1C(C1CC1CCC)=O 73230,C1(CC(N2CC(NC(CC=CC)=O)C(n3cccn3)C2)=O)CCCNC(=O)C1 73231,C1(N(C(C2CCN(CC(C)C)C2)=O)C)CN(C(=O)CCc2ccco2)CC12CC2 73232,C1(C(=O)NC2CCCC(O)C2)CN(C(c2ccnn2C2CC2)=O)CC1(F)F 73233,N1(C(C2(N(C)C)CC2)=O)CCC(O)C1.C1(C)(CNC(COC)=O)CCCS1 73234,c1(NC2(C(=O)NCc3[nH]cc(COC)c3)CCOC2)ccc(OC)cc1 73235,N(C1CCCc2c[nH]nc21)C(C1C(CNC(c2c(C)nc(CC)o2)=O)CC1)=O 73236,c1(-c2nc(-c3scc(C)n3)nn2C2CCCSC2)cc(S(N)(=O)=O)c(C)cc1C 73237,N1(C(C(CC)CC)=O)CCC(C2(CNC(=O)C3CC3)CCOCC2)CC1 73238,N1(C(CC=C)=O)CCc2sccc2C1CNC(=O)C(C)Cc1ccccc1 73239,C1(C(N2CCC(C(=O)O)(CC)C2)=O)CCN(C)CC1C(F)(F)F 73240,CC(C)CCC(CO)NC(C1CC(CNC(c2coc(C(F)F)c2)=O)C1)=O 73241,N1(C(c2c(C)nsc2C)=O)CCC(C)C(CC(N2CC=CC2CF)=O)C1 73242,C1CCC(F)(F)CC1(C)C.Cc1onc(C)c1I.n12cc(nn1)Cn1nnnc1-2 73243,c1(C(N(C)CC2CCCCN2C(C2CCC(CO)CC2)=O)=O)ccc(O)c(F)c1 73244,c1(C)cccc(C(C)CCCOC)n1.CCS(=O)(=O)N(CCN(CC)C)C 73245,CCCCC(C(=O)N1CCC(C(C)(O)CNC(c2nn[nH]c2Cl)=O)CC1)C(C)C 73246,N1(C(c2c(CC)noc2)=O)CCCC(C2CCN(CCOC3CCCC3)C2)C1 73247,C(C1=NOC2CN(C(C3(C4CC4)CCOCC3)=O)CC12)NC(c1cccnn1)=O 73248,C(C(C)(O)C(=O)NCC1(F)CCC(NC(=O)CCSc2ccccn2)C1)OC 73249,C(=O)(C1=CCCCCC1)N(C(C)C(=O)Nc1cc(Cl)cnc1C)CC 73250,C=CC1(NC(C23CC2CN(C(C2CCC(O)C2)=O)C3)=O)CCCC1 73251,N1(C(C=C2CCN(C)C2)=O)CCC(NC(=O)CC2(C)CC(F)(F)C2)C(O)C1 73252,c1(C(N(CCCNC(C2(C=C)CCCCC2)=O)CCO)=O)cn2cccnc2n1 73253,c1(C(=O)NC2CCC(NC(C3(C4CC4)CC3)=O)CC2)cc2ccncc2o1 73254,CC(C(=O)NC1(C)CCCN(C(c2cccc(Cl)c2F)=O)C1)C(C)(F)F 73255,C(CCCCC(=O)NC1(C(=O)NOCC2(C)CC2)CCCCC1)NC(C)=O 73256,Cc1nc(S(C)(=O)=O)ccc1NC(c1ncncc1-c1c(F)cccc1F)=O 73257,C1(NC(COC(C)=O)=O)CC(F)CN(C(=O)C(C(C)C)c2cccc(Cl)c2)C1 73258,S(=O)(=O)(c1cnc(N2CCC(n3cnnn3)C2)c(Cl)c1)N(C)CC1CCC(=O)NC1 73259,c1(CC(=O)N(CCCNC(c2cn(C)c(=O)n2C)=O)C2CC2)ccc2ncsc2c1 73260,CN1C(=O)CCCC1C(=O)NC1CCCCC1C(N1CCOCC1CC(N)=O)=O 73261,c1(OCC)ncc(C)cc1C(=O)NC1CC1C(=O)Nc1ccc(C(C)(C)C)cc1 73262,N#Cc1cnc(N2C3CCC2C(CNC(c2cscn2)=O)C3)c(Cl)c1 73263,C1(C(N2CC(CC)N(C(=O)C=CC3CCOC3)CC2)=O)CC(F)(F)CCC1(C)C 73264,c1(OCCC(=O)NCC(CNC(CC=C=C)=O)F)ccccc1CC 73265,c1(N2CC(c3cc(C)no3)OCC2)ccc(S(=O)(=O)NCc2conc2C)cn1 73266,C1(C(=O)NC(CC)(CNC(=O)CC2CCC3CC23)CC)CCc2ccccc2N1 73267,CCC(C(=O)N(C)CC1(O)CN(C(=O)C=CCOCCOC)C1)SC 73268,CC(C)CC(C(=O)N1CC(O)(C(F)C(=O)NCC2(C)NC(=O)NC2=O)C1)C(N)=O 73269,C(=O)(C(CC(C)C)OC)NCc1c(CCNC(CC(=O)OCC)=O)ocn1 73270,C=C(C)CCCC(=O)NCC1COCC1NC(=O)C(C)NC(C)=O 73271,c1(OC)cc(OC)c(NC(=O)NC(Cc2ccccn2)C(N)=O)cn1 73272,C12(C(N(C)CC3CCCN3C(=O)CC(C)(C)C(F)F)=O)CCCN1S(=O)(=O)CC2 73273,CCCC(CC(C)C)C(=O)N1CCN(C)C(CNC(=O)C(C)(C)C(C)O)C1 73274,Clc1cc(C(c2nnnn2CCC2CC2)NC2C=CCC2)ncn1 73275,C1(CN(C)C)CCCN(C(C2C3CN(C(=O)CCS(C)=O)CC23)=O)C1 73276,C1(CCC(=O)NC(C)CCN(C(=O)CSC2CC2)C)NC(=O)NC1=O 73277,C1(NC(c2csc(CO)n2)=O)CCC12CN(C(=O)C(c1ccc(F)cc1)CO)C2 73278,N1(C(CCc2onc(CC)n2)=O)CC2CC(C1)N(C(=O)CCC1CCC(=O)N1)C2 73279,C(C(=O)N1CC(NC(c2ccnc(C3CCCC3)n2)=O)C1)(C(C)C)SC 73280,CC(CC(N)=O)C(=O)NCCOC1CN(C(c2nc(C3CC3)sc2Br)=O)C1 73281,Cc1cc(Cl)c(C(=O)NCCN(C(=O)CCC2CCC(C)O2)C2CC2)cn1 73282,N1(C(CN(C(C(CC=CC)C)=O)C(C)C)=O)CC2(CNC(=O)OC2)C1 73283,C1(NC(NOC(CC)=O)=O)CCCCC12CCN(C(=O)C(CC(C)C)OC)C2 73284,c1(-n2cc(CCC3(O)CN(C(CN(C(C)C)C)=O)C3)nn2)cccc(F)c1F 73285,C(C(=O)NCCSC)(C1=CCC2CC1C2(C)C)N(C1CCOCC1)CC=C 73286,C1(CNC(C2C(C)C2C2CC2)=O)CC2(CCC2)CN1C(c1cnc[nH]1)=O 73287,Cc1c(F)c(F)c(CNC(C2CCC(C)C2)=O)c(F)c1F 73288,N1(CC(=O)N(CC(=O)NCC(c2cnc[nH]2)C)CC)CCC(F)CC1 73289,CC1CCN(C(=O)C2=COCC2)C1C(=O)N(C)CCc1ccncc1 73290,C(CCCC)(C(=O)N1CC(OC(C)C)C1)NC(CCCC#C)=O 73291,Cc1nc(O)nc(C)c1C(=O)NCCC(C)NC(=O)Cc1cnn(C(C)(C)C)c1 73292,c1(N2CCN(OCc3c(C)cccc3)CC2)n[nH]c2ccccc12 73293,Cc1c(C(N2CCN(C(C3CC34CCC4)=O)CC2C(C)C)=O)cnc2nncn12 73294,CCCC(C)C(=O)NC1(CCC(=O)NCc2cn(C)nc2CC)CCCC1 73295,c1(OC)cc(C#N)ccc1N(C1CC2CNC1C2)C(=O)CCc1cnc[nH]1 73296,C1(C(=O)NCC(C)CNC(C2(C)CCSCC2)=O)CCOC(=O)N1 73297,N1(C(C2N(C(c3c(C)cc(C)o3)=O)CSC2)=O)CCCC(C)(O)C1 73298,c1(CNC(CC(C=C)c2ccccc2)=O)ccc(N2CCCC2)c(F)c1 73299,N1(C(CC=CCC)=O)C2CCC(C2)C1C(=O)NC1CCN(C(C)C)CC1 73300,CC1(C)CCCN(C(c2cc(N)cc(O)c2)=O)C1CNC(=O)CNc1nccs1 73301,C(=O)(C1=C(Cl)CCOC1)NCCC1N(C(C2(CCOCC)CCC2)=O)CCCC1 73302,c1(CC(=O)N(C(CCNC(CC=C(C)C)=O)C)C)ccc(Cl)cc1 73303,c1(SCCNC(C(=O)NC(c2ccc(F)c(Cl)c2)C)=O)ccc2c(c1)CCO2 73304,C1(CC(=O)N(C2CCN(C(=O)C(O)c3ccco3)C2)CC#C)NC(=O)NC1=O 73305,c1(CCCNSC2C(=O)NOC2)ccc(F)cc1Br 73306,C1(C#N)(SC)CN(C(=O)C(Cc2ccoc2)NC(C2CC(N(C)C)C2)=O)C1 73307,C(=O)(CC(O)C(Cl)(Cl)Cl)NC1CC(C)(NC(=O)C=Cc2cnc[nH]2)C1 73308,C1(CC)CC(C(=O)NCC(CC)(CC)NC(c2oc(CO)cc2C)=O)CCO1 73309,c1(CC)ccccc1CC(=O)N(C1CC(NC(c2ccn(CCO)c2C)=O)C1)C 73310,C1(NC(C2CCCC(=O)N2)=O)CCCC12CN(C(C1CCS(=O)(=O)N1)=O)C2 73311,C1(NC(c2nc(CC)sc2)=O)CC2CCC(C1)N2c1ncc(Br)cn1 73312,n1(CCC(=O)NC2CCN(C(CSCCCC)=O)C2CC)nc(C)c(C)c1C 73313,C1(CN(C2(C)CCN(C(C3(OC)CCCOC3)=O)C2)C)CCCCCCC1 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73436,C1(C(=O)OCC(c2[nH]c(C)c(C(=O)OC)c2C)=O)(OC)CCCC(C)(C)C1 73437,C(=O)(CC(C)(C)COC(C)=O)N1CCC(CC(N2CCC(NC(CC)=O)C2)=O)C1 73438,C1(C(=O)NOC(CC)CC)(CC#C)CCN(C(=O)Cc2cncs2)C1 73439,C1(CC)CN(C(c2ccc(Cl)cc2)=O)CCC1NC(=O)C=CC1CCOC1 73440,c1(OC)cc(C(N2CCC(O)(CCNC(c3ocnc3C3CC3)=O)C2)=O)n(C)n1 73441,C#Cc1cccc(NC(C2CCC(C)N(C(c3ccc(CC#N)cc3)=O)C2)=O)c1 73442,CC1CN(C(c2cccnc2C(F)F)=O)CC1NC(=O)C(O)C(F)F 73443,Cc1cc(C(=O)NCCC2CCN(C(=O)C(F)(F)c3ccccc3)C2)nn1C 73444,c1(C(N2C(C(=O)Nc3cccc(OC)c3O)CSCC2)=O)ccc2nc(C)[nH]c2c1 73445,Cc1noc(C)c1C(N1CC(CN(C(=O)CSCCC(F)(F)F)CCO)C1)=O 73446,c1(OC)ccn2ncc(C(=O)NCC3CN(C(=O)C(O)C(C)C)CCN3C)c2c1 73447,C#CCC(CC(F)F)C(=O)NC1C=CCN(C(=O)COCc2ccc(C)cc2)C1 73448,c1(C(N(CCCNC(C(c2cn(CC)nc2)(F)F)=O)C)=O)c(C)nnn1CC 73449,C1(N2CC(C)(c3nc(C)cs3)C2)C(N)CC1(C)C.CO 73450,Cc1nc2c([nH]1)C(Nc1cc(C)c(S(N)(=O)=O)cn1)CCC2.C=O 73451,c1(OC)cc(N2CCC(NC(c3cc4ccccc4o3)=O)C2)ccc1[N+](=O)[O-] 73452,N1(C(c2n(CCC)ncc2)=O)CCCC(C(=O)NCC2CCC3(CC3)C2)CC1 73453,C#Cc1cnn(CC(=O)NCC(C(=O)NCC#CC2CC2)N(C)C)c1 73454,C12(NC(CCN(C(CCC)C)C)=O)CCCC1CN(C(=O)Cn1cnccc1=O)C2 73455,c1(NC2(CNC(CCc3ccc(C)s3)=O)COC2)nc2cccc(F)c2s1 73456,c1(OC)csc(C(=O)N(C)CC2CN(C(C3(c4oncc4C)CC3)=O)C2)c1OC 73457,C1(CNC(CN(CCOC)C)=O)(CO)CCN(C(=O)Cc2c[nH]ccc2=O)CC1 73458,C12(C(=O)NC(CC(C)NC(c3coc(-c4ccccc4)n3)=O)C)CC(C)(CO1)C2 73459,C(C(=O)N1CCCc2nccn21)C1OCCN(C(CC(CC)C(F)F)=O)C1 73460,C12(CN(CCN(CCC)C(c3ccc(CCF)cc3)=O)C)COCC(C1)C2 73461,CN1CCCCC(C(=O)NC2(CNC(C3(C)CCCSC3)=O)CC2)C1=O 73462,c1(C(=O)NC2CCN(C(=O)CC3(C(F)(F)F)CC3)C2)nccc2[nH]ccc12 73463,Cc1c(C(=O)NC2CN(C(=O)C=CS(C)=O)CCC23CCC3)ccc(F)c1F 73464,C(=O)(C1=NOCC1)NC(C1CN(C(=O)CN(C2CCCC2)CCO)C1)C 73465,C(=O)(C(O)C(F)(F)F)NC1(CO)CCN(C(C(N2CCOCC2)C)=O)C1 73466,C1(C(=O)NC2CCCN(C(c3ccc(F)nc3)=O)C2)CCc2nnnn2C1 73467,C1(NC(CCC(CC)OC)=O)CN(C(=O)CCCNC(=O)OC)CC(F)(F)C1 73468,Cc1nc(NC2CCC(NC(=O)CC(C)n3ccnc3)CC2)cc(C#N)n1 73469,c1(C(N2C(COC)CCCC2)=O)ccc(Cl)nc1NC(c1ccc(O)cc1F)=O 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73505,CC1(C)CCC(CNC(C2CCCC(F)C2)=O)N(CC(=O)NCC2CCCO2)C1 73506,CCC(C)(CO)C(=O)N1CC(N(C)C(c2cc(O)nc(O)n2)=O)C2(CC2)C1 73507,c1(-n2c(Cn3ccc(C(F)F)n3)nc(COC(C)C)n2)ccc2ncsc2c1 73508,N1(C(C(C)=CC2CC2)=O)CCCC(C)(C)C1CNC(C1CC1C1CC1)=O 73509,C(=O)(CN=S(C)(C)=O)N1C(C)CC(NC(c2n(CC=C)ccc2)=O)C1 73510,c1(OC)ccc(OC)c(S(=O)(=O)N(CCCNC2(c3cccs3)CC2)C)c1 73511,Cc1cc(CCN2CCN(CC(C)O)CC2)cc(O)n1 73512,C(CCCC(C)NC(C1CCOCC1)=O)NC(c1nc(C(=O)OCC)sc1)=O 73513,c1(CNC(N(CCC=C)CC(=C)C)=O)c(Br)ccc2c1CCC2 73514,N1(C(C(C)(C)c2ccccc2)=O)CC2COCC2C1.c1(N)cc(O)ncn1 73515,C1(C(N2CC(CC(C)NC(=O)CCSCC(N)=O)C2)=O)(OC)CCOCC1 73516,c1(COC(N2CC(CC(C)NCCc3cc(Cl)n(C)n3)C2)=O)ccc(N)cc1 73517,N1(Cc2ccc(N(C)C)cc2)CCc2n[nH]cc2C1.N12CC3CC3(C1)C2=O 73518,C(=O)(C1=CS(=O)(=O)CCC1)NC(C1(O)CCN(C(c2ccn(CF)n2)=O)CC1)C 73519,N1(C(c2c(C)coc2)=O)CCN(C(=O)C(F)(F)Oc2ccccc2)C(C)C1 73520,c1(C(=O)NCC2C(NC(CCn3ccc(C)n3)=O)COC2)ccn2nncc2c1 73521,Cc1nc(-c2cn(CCCC(=O)N(C)Cc3nc(C(=O)O)co3)nn2)cs1 73522,N1(C(C(C)=C2CC2)=O)CCC(C)C1CNC(=O)Cc1n[nH]c(C)n1 73523,C1(C(=O)OC)CCC(CNC(C)CCNC(CC(C)SC)=O)CC1 73524,CC1CC(CC(N2CCCC2C2(C)CC2)=O)CN1C(=O)COc1ccc(F)cc1 73525,C(c1c(C)coc1C)=CC(N1C(CCNC(CC2N(CC)CCC2)=O)CCC1)=O 73526,C1(C(N2CC(CC)SCC2)=O)CC(F)(F)CN1C(=O)CCC(C)OC 73527,C(=O)(C(C)(C)CC#N)N(C(CC(=O)NCC1(C)N=C(C)SC1)(C)C)C 73528,C=CCCCCCCC(=O)NC1(CNC(c2cncc(C)c2Cl)=O)CCOCC1 73529,N1(C(C2C3CN(C(C4CC5(CC(C)C5)C4)=O)CC32)=O)CC(O)C(O)C12CCC2 73530,N1(C(C(c2ccnn2C)NC(C(C)C#N)=O)=O)CCCCCCCCC1 73531,CC(C)CCCCC(=O)NCC(C1CC1)NC(=O)C#CC(=O)N(C)C 73532,Cn1cncc1NC(C1CC(C(C)(C)NC(=O)CCCN2CCCC2)C1)=O 73533,C1(Cn2cc(C(CC)(C)C)nn2)CC(O)CN1C(c1coc(C)n1)=O 73534,O=C(C1=CCCOC1)NC1(CO)CCN(C(c2ccccc2)=O)C1 73535,Cc1cc(N2CC(C)(C)CC2(C)CNC(=O)CCC2CCCO2)ccc1[N+](=O)[O-] 73536,C(=O)(C(CC(F)F)NC(=O)Cn1cnnn1)NC(c1cncs1)C 73537,Cc1nc(C(=O)NCc2c[nH]nc2C(=O)NC2CCC2O)c(C)s1 73538,c1(-n2c(-c3ccc(C)n3C)nc(CSC)n2)ccc(Br)cc1C 73539,C=CC(C)C(C)C(=O)NC1(C)CC(NC(c2cncc(Cl)c2Cl)=O)C1 73540,CCCCCCC(C)C(=O)NCC1(S(=O)(=O)NC)CC1 73541,C1(C(C)C)CNC(=O)CN1C(=O)CCCCCn1cc(-c2ccsc2)nn1 73542,C(=O)(C(C)(C(=O)OC)C(C)NC(C1CC(=O)N(c2ccc([N+](=O)[O-])cc2)C1)=O)OC 73543,CN1CCC(CC(=O)NCC(=O)NCCNC(=O)CO)C1=O 73544,Cc1ccc2oc(C(N3CC4(CCCN4Cc4cccc(C)c4O)C3)=O)cc2n1 73545,CCCC(C(=O)N(C(C)(C)CC(=O)NCCCN(C)C)C)C(C)C 73546,C1(C(=O)OCC)CC(C)(C)CCO1.C1CCN(CCF)C1 73547,CC1(NC(=O)Cc2cnoc2)CC(NC(C2CC2C#N)=O)C1 73548,C1(N(C(c2c(C)ocn2)C(=O)NCCCF)C)CC(O)C1(C)C 73549,C1(C)(C(=O)NCC(C)(C)NC(C2(C)CC3CCC2C3)=O)CC2CCC1C2 73550,CC1(C(=O)NCC2(C)CCN(C(=O)Cc3csc(Cl)n3)C2)COC(=O)OC1 73551,C1(CNC(c2c(C)con2)=O)(CO)CCN(C(=O)Cc2cccc(C#N)c2)CC1 73552,c1(C(=O)NC(CC(=O)NC2CCCC2)c2ccccc2)ccc(I)c(Cl)c1 73553,C(CCF)(C(=O)N1CC(C(C)(C)O)C1)NC(CN(CCC#C)C)=O 73554,c1(CNC(C2CC2Nc2cc(OC(F)F)ccn2)=O)cccc(I)c1 73555,C1(CCNC(=O)CN2CCOCC2)CCN(C(c2csc(CO)n2)=O)CC1(F)F 73556,CC1OCCC1(C)NC(=O)NCCc1csc(-c2cccnc2)n1 73557,N1(C(C2CN(C(C(C)Oc3ccccc3Cl)=O)C2)=O)CCOc2ccccc21 73558,c1(C(=O)NC23C(CN(C(C(CCSC)OC)=O)C2)C3)n[nH]c2c1CSCC2 73559,CCC(CO)(C(=O)N(C)CC1CCN(C(=O)CC(C)N2CCCC2=O)C1)OC 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73577,c1(OC)ccc(C(=O)NC2COCC2NC(C2(C(F)(F)F)CC2)=O)nn1 73578,C1(C(N(C2CCN(C(c3cn(CCO)nn3)=O)C2)C)=O)CC(=O)NC(=O)C1 73579,CC(C)(CC(=O)NCc1cncs1)CC(F)F 73580,C1(CN=c2[nH]nc(C(N)=O)s2)CN(C(=O)CCc2ccccc2)C2(CCC2)C1 73581,c1(CC)c(C(=O)NCC2CC(F)CN2C(C2CCC(C)(C)O2)=O)cccc1C 73582,CC1(CO)C=CCN1C(c1conc1CNC(=O)COC1CC1)=O 73583,C(=O)(C(C)C(=O)N1CC(NC(c2cc(OC)no2)=O)C1)OCC 73584,C(CC(C)(C)C(=O)NCC1(CCO)CCC1)NC(C(CCSC)O)=O 73585,CN1CCN(C(C2(CNC(=O)CCCN3CCCC3)CC=CC2)=O)CC1 73586,C1(CNC(CN(C)C)=O)(CNC(C2(Cc3nc[nH]n3)CC2)=O)CCCC1 73587,c1(C(N2CCC(NC(CCc3cccc(OC)n3)=O)C2C)=O)cc(C)c(O)nn1 73588,N1(C(CC2OCC(C)(C)C2)=O)CCC2CN(C(C3CS(=O)(=O)C3)=O)CCC12 73589,c1(SC)c(NC(c2ncccc2Cl)c2nnnn2CCCF)cncc1F 73590,c1(CC)ccc(C(c2nnnn2CCCF)NCCc2cccc(C)n2)cc1 73591,c1(CC)cccc(C(N2CCC(OCc3cn(CC(C)C)nn3)C2)=O)c1O 73592,N1(C(N2CCC(NC(=O)OCC)CC2)=O)CCC2OCCCC2C1 73593,Cc1cc(COCC(=O)NCC(C)CN(C(=O)CC2CC(=O)C2)C)no1 73594,c1(C(=O)NCCC(=C)CNC(c2cccn2C(C)C)=O)oc(CCC)cc1C 73595,C1(O)(CN(C(C2C(C#C)C2)=O)C)CCN(C(=O)CCC=C=C)CC1 73596,Cc1cc(C(N2CC3C(CNC(C4(C)CCN(C)C4=O)=O)C3C2)=O)cc(C)c1 73597,C1(OC)CN(c2ccncn2)CC1NC(N1CCC(CN2CCCC2)C1)=O 73598,CC(=O)CCCC(C)C(=O)NC1(C(N2CCC2C2CCCCC2)=O)CC(F)(F)C1 73599,C1(C(N(C2CCN(C(C3(C)CC=CC3)=O)C2)CC)=O)COCC1(C)C 73600,c1(C(=O)NC2C3CCC2N(C(c2occc2F)=O)C3)cc2ccc(F)cc2o1 73601,Cc1cc(CC(=O)NCCC2(O)CN(C(=O)CCc3ccc(C)s3)C2)on1 73602,N1(C(C(c2ncc(C)s2)C2CCNCC2)=O)CC(O)CC1C(=O)O 73603,c1(C(N2C(CNC(CN(C(=O)OC)C)=O)CCC2)=O)cc(Cl)cc(F)c1F 73604,c1(C(=O)NCC2CCN(C(C(CC=C)CC)=O)C23CC3)cc2ccccc2cn1 73605,C1(CNC(=O)Cc2ccns2)CN(C(=O)C=Cc2cc[nH]n2)CC12CC2 73606,C1(C(=O)NCCN(C(=O)CN(C)CCO)CCOC)CCCSC1 73607,c1(C(=O)NC2C3(CC(NC(c4c(C(C)C)noc4)=O)C3)C2)cnc2[nH]ncc2c1 73608,N1(C(C2C(=C)C2)=O)CCN(C(=O)CCc2ccc(Cl)cc2)CC1CF 73609,c1(CC)cc(N2CC3C(CNC(=O)C(C)Cn4ccnc4)C3C2)ncn1 73610,c1(CC(C(=O)NCCC2(O)CN(C(C3(OC)CC3)=O)C2)O)cc(Cl)sc1Cl 73611,C1(C(N(CCNC(=O)C(c2cccc(C)c2)O)CC)=O)CC12CCC(F)(F)CC2 73612,O=C1CC(C(=O)OC(C(=O)OC(F)(F)C(F)(F)F)C(F)(F)F)C2(CCC2)C1 73613,c1(C(=O)NCC(CO)NC(c2ccc(CO)o2)=O)cc2ccc(Cl)cc2[nH]1 73614,C(=O)(C(F)CC(C)C)N(C1CCCN(C(c2n(CC)ccc2)=O)C1)C 73615,C1(C(N(CC(=O)OCC)CC)=O)CCC(CNC(=O)Cn2cc(C#N)cn2)CC1 73616,C1(C)(CC)CCN(C(C2(CO)CCN(C(=O)C(CO)NC(=O)OC)C2)=O)CC1 73617,C(=O)(CCCCCCCC(=O)NC1CC(C)CN(C(c2cn(C)cn2)=O)C1)OC 73618,c1(C2CC2)cccs1.C(=O)(CCc1cccs1)NC1(C(N(CC)C)=O)CC1 73619,C12(C(N(C)CCNC(=O)C(=O)NC3CC3)=O)CCC(C(F)F)(CC1)CC2 73620,N1(C(C(F)=CC)=O)CCOC2(CCN(C(c3cscn3)=O)C2)C1 73621,C1(NC(C(CCC)N(C)C)=O)CC12CCN(C(c1ccc(CC)s1)=O)CC2 73622,C12CCCN(C1C)CC(=O)N2.c1(C(=O)OC)cc(F)cnc1Oc1ccccc1 73623,N#CC1(C(=O)NCCCNC(=O)CC2CCC23CCC3)CCOC1 73624,c1(OC)c(C(=O)NC2CC(CNC(=O)C(C)n3ccnc3)C2)csc1C 73625,CN1CC(O)CC1(C)C(=O)NCC1(CCNC(C2CNC(=O)C2)=O)CC1 73626,C#CC1(O)CCN(C(=O)CC2N(C(c3ccsn3)=O)CCC2(C)C)C1 73627,C1(OC)CC(F)CN(C(c2cnn(C3CCOCC3)c2)C(=O)NC(C)(C)C)C1 73628,CCCCC(C(=O)N1CCC(CNC(=O)C2=C(Cl)CCCC2)C(C)C1)C(C)C 73629,N1(C(c2c(C)noc2C)=O)CC(C)(C)OC2(C1)CN(C(=O)CCN1CCCC1)C2 73630,N1(C(C(CCC)N(C)C)=O)CCN(C(=O)C=Cc2cccc(F)c2Cl)C2CCC12 73631,CCC(C)C(C)N=c1[nH]c(=NCC2(c3cnccn3)CC2)[nH]c2c1COCC2 73632,C=CCC(C(=O)NCCCN(C(c1cccc(C)c1[N+](=O)[O-])=O)CC)C(C)(C)C 73633,C(=O)(CS(=O)(=O)CCOC)N1CC(CN(C(C2C(OC)CCC2)=O)C)OCC1 73634,c1(C(=O)OC(C(c2n(C)ncc2)=O)C#N)cnn2c(SC(F)(F)F)ccnc12 73635,c1(C(=O)NC(CCOC)CNC(=O)C(C)NS(C)(=O)=O)c[nH]c(=S)cn1 73636,c1(CC)nc2ccccc2c(C(N2CC3CN(C(=O)C(C)O)CC3(C)C2)=O)c1C 73637,C1(NC(CSCCCC)=O)C=CCN(C(=O)COC(C)=O)C1 73638,N1(C(C(CC(=C)C)NC(=O)Cc2ccon2)=O)CCN2C(=O)OCC2C1 73639,c1(CCCC(=O)NC2CC2NC(=O)Cc2ccccc2Br)ccccc1Cl 73640,c1(OCC)ccc(Cl)nc1C(=O)NC1CCN(Cc2cn(C)nc2CC)CC1O 73641,C=C1CC2(C1)CC(C(=O)NC1(CF)CCN(C(c3cc(N)cc(F)c3)=O)C1)C2 73642,C1(NC(c2ccc(C)cc2)=O)CCCC12CN(C(C1(C)CSC1)=O)C2 73643,c1(C(=O)NC(C2CCCC2)CNC(C2CC(OC)C2)=O)sc(SC)cc1C 73644,c1(C(=O)NCCCCN(C(C(CC)CC)=O)C)cccc(C(F)(F)F)c1O 73645,c1(CC(=O)NCC(C)(CO)NC(C(=Cc2cccnc2)C)=O)c(C)ncnc1O 73646,Cc1cnc(Cl)c(S(=O)(=O)Nc2ccc(C(=O)Nc3nccc(Br)c3O)nc2)c1 73647,c1(C(=O)NCCOC2CN(C(Cc3c(C)cccc3)=O)C2)cc(F)c(F)cc1F 73648,Cc1ccc(C(O)C(N2CCC(CCC(=O)N(CCC(C)C)CC(C)C)C2)=O)cc1 73649,c1(C(=O)NC2CC(C)CN(C(=O)C3=CCOCC3)C2)ccc2nc(O)sc2c1 73650,c1(NCC(C)CCCO)ccc(S(=O)(=O)Nc2ccc3c(c2)CN(C)C3)c(Br)c1 73651,C1(CC(C)NC(C2CC(OC)(OC)C2)=O)CCN(C(=O)CC2CC=CCC2)CC1 73652,N1(C(C2C(C=CC)C2)=O)CCN(C)CC1CNC(=O)CCc1nc[nH]n1 73653,N1(C(c2c(OC)scc2)=O)CCC(C(=O)N(C(CCO)CF)C)C(C)C1 73654,Cc1[nH]cnc1C(=O)NCc1ncoc1C1CN(C(C2CC(CF)C2)=O)C1 73655,CCCCC(CNC(c1cncc(OC)n1)=O)NC(=O)C(CC)n1ccnc1 73656,C1(NC(C(C=CCCC)O)=O)CCN(C(c2ccncc2)=O)C12CCC2 73657,n1(C)cc(CC(=O)NC2(C=O)CC2)cn1.C1(C(C)C2CC2)CCN(C(N)=O)C1 73658,CCCCCC(C)(C)C(=O)N1CCC1N1CCOCC(O)(C(F)(F)F)C1 73659,Cc1cc(C#N)ccc1S(=O)(=O)NC(C1(S(C)(=N)=O)CC1)=O 73660,N1(C(C2(C#N)CC=CC2)=O)CC2CCN(C(=O)CC3CC3c3ccccc3)C2C1 73661,C(=O)(CC(C)CC(C)(C)C)N1CC(NC(Cc2cc(OC)c(O)c(OC)c2)=O)C1 73662,c1(C(N2C3C(C(N(C4(CCO)CC4)C)=O)C(C3)C2)=O)cc(O)nc(O)n1 73663,C=CC(C)CCN=c1nc(-c2ccccc2)[nH]c(=NCC(C)(C)n2ccnc2)[nH]1 73664,c1(C(N(C2CCN(C(C3CC34CCOC4)=O)CC2)C)=O)ccnc2c1CCC2 73665,N1(c2cc(NC(COC)CCO)ncn2)CCN2C(CCS2(=O)=O)C1 73666,C12(C(=O)NCCC(CNC(C(COC)NC(C)=O)=O)OC)CC(C)(CO1)C2 73667,FC(F)=C1CCC(c2nnnn2CCCF)(NCC2CCC2CO)CC1 73668,c1(NCCNC(C)=O)ccc(S(=O)(=O)Nc2nc(Br)co2)cc1Cl 73669,CC(C)(CCC(=O)N1C2CCC1CC(C(=O)NCc1cnccn1)C2)[N+](=O)[O-] 73670,CC(C)C(C#N)C(=O)N(CCCC(=O)NCCCCCC)C 73671,C(=O)(C1Cc2ccc(F)cc21)N1CCCC(CSC)(NC(=O)CC(C)(C)CC)C1 73672,C1(O)(CCNC(C2CC(C)(O)C2)=O)CCN(C(=O)C2=CCCCO2)CC1 73673,C(CC(C)C)(C(=O)N1CC(C)CCC1CO)NC(CCCNC(C)=O)=O 73674,C1(CNC(Cc2cc(C)no2)=O)CN(C(C2CCCC(=O)CC2)=O)CCCO1 73675,c1(C(=O)NC2CCCC(OCC)CC2)ncc2cc(Cl)ccn12 73676,CON=CC(=O)NC(C)C(=O)NCC(=O)OC(C)C 73677,Cc1nn(C)c(C)c1CC(N1CCC(F)(C(F)(F)F)CC1)=O 73678,C(=O)(C(C)(C)C(C)C)NCCCC1OCCN(C(c2c(C)[nH][nH]c2=N)=O)C1 73679,N1(C(Cc2ccc(OCC)nc2)=O)CC2CC1CN(C(C1CC(=O)N(C)C1)=O)C2 73680,N1(C(CCC)=O)CCC(NC(c2ccnc(N3CCCC3)c2)=O)C(F)C1 73681,N1(c2nccc(SC)n2)CC2CN(C(c3cccc(OC)c3OC)=O)CC2C1 73682,c1(C(=O)NC(c2n(C)ncc2)C(=O)NCCn2ccnc2)ncnc(O)c1F 73683,CCCCCCC(C)C(=O)NC1CC(C(F)F)(NC(=O)CCCN=[N+]=[N-])C1 73684,c1(C(=O)NCCN2CCN(C(C(C)CC(N)=O)=O)CC2)cnn2c(N)ccnc12 73685,C1(NC(CN(C)C(c2ccsc2)=O)=O)CC2CC(NC(=O)Cn3nccn3)C1C2 73686,N1(C(Cn2ccc(C)n2)=O)CCC(F)(C(=O)NCC(OO)C2CC2)C1 73687,N1(NC(Cn2cc(-c3c(OC)c(C#N)ccc3)nn2)=O)CCOC(C2(C)N=N2)C1 73688,N1(C(c2c(OC)scc2)=O)CC2(CCN(C(=O)C(F)C(C)C)CC2)CC1C 73689,c1(C(=O)NC(CSC)CO)coc2cc(O)ccc12 73690,c1(NCC23CC(NC(=O)Cc4ccc(F)cc4)(C2)C3)noc2ccc(O)cc12 73691,N1(C(=O)Nc2c(OC)nsc2)CCC(NC(=O)CCCOC(C)=O)CC1 73692,C(C(C(=O)NCCN1CCC1)C(C)C)NC(c1c(C)ccn1C)=O 73693,CS(=O)(=O)c1ccc(C(O)CNC(=O)NCc2c(O)cccc2Cl)cc1 73694,CC12CCC(CNC(N3CCCOC(CCO)C3)=O)(CO1)C2 73695,c1(C(=O)NCC2C(C)(C)C(NC(=O)Cc3ccoc3)C2)cnn2c1OCC2 73696,c1(CCNC(C(C)(C)OC(C)C)=O)ccc(CNC(C2CCC(=O)NC2)=O)cc1 73697,C=CCC(C)C(=O)NCC1(C)CCCN1C(=O)C(C)OCCC(C)C 73698,c1(CC(=O)NCCCN(C(=O)Cc2ccsn2)CCC)nnc(C)o1 73699,C1(NC(COCCSC)=O)CCCC(NC(=O)C2=C(C)OCC2)CC1 73700,C1(C(=O)NC2CC(CNC(C34CC5CC3C4C5)=O)C2)CCCC2(CCCCC2)C1 73701,c1(OC)cccc(C(CNC(=O)C(Cl)=CCl)NC(c2c[nH]nc2F)=O)c1 73702,c1(CC(N2CC(CC)N(C(c3ccc(=O)n(C)n3)=O)CC2)=O)ccc(C)c(F)c1F 73703,N1(C(C2CCN(C(CC)=O)C2)=O)CCC(F)(CNC(c2coc(CC)n2)=O)C1 73704,c1(C(=O)NCC(C)(CC(C)C)NC(CCOCCC)=O)ccn2ccnc2n1 73705,c1(OC)cc(OC)cc(C(N2CC3CC(C2)N3C(c2sccc2F)=O)=O)c1 73706,c1(C(N(CC(CC)NC(CC(=O)OCC)=O)C)=O)cc(SC)cc(Cl)c1 73707,c1(CN2C3C(C(=O)Nc4ccc(Cl)c(Br)c4)C(C3)C2)ccc2c[nH]nc2c1 73708,N=c1[nH]c2c(s1)CCCC2C(=O)NCC1CC(O)CN1C(C1CCSCC1)=O 73709,C#CCCCCCC(=O)N(CCCCC(=O)N(C)Cc1ncnn1C)C 73710,CC1(C)COC(C(=O)NCCC2CN(C(=O)COC3CCCCCC3)C2)C1 73711,c1(CNC(=O)NCC(=O)NCC(O)CNC(c2ncc[nH]2)=O)ccccc1 73712,c1(OC)cnc(C(=O)N(C(C)C(=O)NCc2sccc2C)C)cn1 73713,C1(NC(C2C(C(=O)OC)CCO2)=O)C2CC1CN(C(C1CCCCO1)=O)C2 73714,Cc1cc(Cl)ccc1OCC(N1CCC(NC(c2ccsc2C#N)=O)C1)=O 73715,C1(NC(CCCC)=O)(CF)CCN(C(c2cnn(-c3ccccn3)c2C)=O)C1 73716,C1(CNC(CCc2n(C)ncc2)=O)C2CC1N(C(C1C(F)(F)C13CC3)=O)C2 73717,c1(CC(N2CCC(C(CNC(C(C=C)OC)=O)O)CC2)=O)ccc(C#N)cc1 73718,c1(CS(=O)(=O)NCC(=O)NCCCc2ccccc2)cncc(Br)c1 73719,C(=O)(C(C)=NOCC#N)N1C(C(=O)NCC(=O)OCC=C)CC1C 73720,C(CNC(c1cnoc1C)=O)(CC)(CC)NC(C1CCC(COC)C1)=O 73721,N1(C2CC2)CCCOC(CCCNC(c2ccc(COC)o2)=O)C1.C1(=O)CO1.CCO 73722,N#Cc1cc(Cl)c(C(=O)NC2(CNC(C3CN(C(N)=O)C3)=O)CCOCC2)s1 73723,CC1(C(=O)N(CC(F)F)C2CC2)CC12CCN(Cc1n[nH]c3ccccc13)CC2 73724,C1(CCC)CC1N=c1[nH]c(N(C)CC2(N(C)C)CCCC2)nc2c1COC2 73725,c1(C(=O)Nc2ncc(CC)cn2)ccnc(Cl)c1C.c12nc(cs1)CC(=O)N2 73726,N1(C(C(C)C2(O)CCC2)=O)CCC2(CC1)CC(NC(=O)CCSC(F)(F)F)CO2 73727,N1(C(COCCC(C)C)=O)CCS(=O)(=O)C(CCNC(C2CC3(CC3)CO2)=O)C1 73728,c1(C(N2CCCCC2CCOC)C(=O)NCCCC)cc(Cl)c(Br)cn1 73729,CC(O)CCCN=c1ccc(Br)c(S(=O)(=O)NC2CS(=O)(=O)CC2C)[nH]1 73730,N1(C(c2ncn(CC)n2)=O)CCC2C(C(=O)NCC3CCN(C4CC4)C3)C2C1 73731,N1(C(C2CC(=O)NC(=O)N2)=O)CCC2C(C1)CN2C(C12CSCC1C2)=O 73732,c1(C(=O)NCC2CN(C(C(CO)N(C)C)=O)CC2(C)C)csc2c1CCCC2 73733,c1(C(N2CC(CC(=O)N(C(C#C)C3CCC3)C)OCC2)=O)cnn2c1OCC2 73734,c1(CC(C(=O)N2CC(OC(=N)O)C2)N)cnn(C)c1O.CC(CN(C)C)C(=O)NCCO 73735,c1(NCCC2(CC(=O)OC)CCOC2)ccc(C(C)(C)C)cc1F 73736,C(c1cccc(F)c1F)=CC(=O)NC(C1(CNC(C2CCC(=C)CC2)=O)CC1)C 73737,n1(CCC(=O)N(CC(=O)NC2CCN(C(N)=O)C2)C)nnc2ccccc2c1=O 73738,CC(C)CC(CNC(=O)CC1(O)CCCCC1)NC(=O)CCc1cn[nH]c1 73739,C1(NC(=O)Cn2ncnn2)CCN(C(C2CCC([N+](=O)[O-])CC2)=O)C12CCCC2 73740,c1(C(=O)NCC(C(C)(C)C)NC(CCSCC)=O)ccc2c(=O)n(C)cnc2c1 73741,C1(NC(=O)CSc2cccc(F)c2)CN(C(C2CCC3(CC3)C2)=O)CC2CC12 73742,c1(C(=O)NCC(N(C(C2(CC)CCOC2)=O)C)C2CC2)cc2ccc(C)cn2c1 73743,C12(N(C(CCNC(CN3C(C)CCC3C)=O)C)C)CCC(CC1)CC2 73744,N1(C(CCCOC(C)=O)=O)CCCC1(C)CNC(C1CC1(c1ccccc1)C)=O 73745,C1(C(N2CCC(C)(NC(c3ccc(CO)nc3)=O)C2)=O)(OCC)CCOCC1 73746,C1(NC(c2cc(OC)ncn2)=O)CCN(C(c2cnc(Cl)s2)=O)CCC1CO 73747,N1(C(C2(C)CCCCO2)=O)CCC(F)(CC#N)CC1.n12cc(nn1)CNCC2C 73748,c1(C(=O)NCC(C(C)(C)C)NC(=O)CCc2ccco2)nnn2c1CCCC2 73749,C(=O)(CCCCCN(C)C)NC(CCNC(C(C)NC(c1ccoc1)=O)=O)C 73750,c1(OCC)nc(C)ccc1C(=O)NC(C1CCOC1)CNC(=O)CCC(C)C 73751,c1(C(N(C2CCC(NC(=O)CC34CCCC3C4)CC2)C)=O)ccc(CCO)cc1 73752,C1(C(CNC(C(c2scc(C)n2)(F)F)=O)F)CCN(C(c2ccoc2)=O)CC1 73753,c1(C(N2C(CNC(c3ccoc3)=O)CC(OC)C2)=O)ccc(N)cc1O 73754,C1(C)(CNC(C(c2n(C)ccc2)=O)=O)CCCN(C(c2cnncc2O)=O)C1 73755,N1(C(c2cn(CCC=C)nn2)=O)CCC(CNC(=O)CN(C)CCO)CC1C 73756,C1(CCNC(CN2C(C)CCC2)=O)CC(F)CN1C(=O)CCCN(C)C 73757,N1(C(CCOCC(C)C)=O)CCCCC(C(=O)NC2CC(CCC(N)=O)C2)C1 73758,N1(CC)CC(C(N2CCOC(CNC(C3CC4CC(=O)C3C4)=O)C2)=O)CCC1=O 73759,c1(CCNC(C(=C)F)=O)nc2ccc(Br)cc2s1 73760,c1(C(=O)NCCC2(NC(C(CC)SC)=O)CC2)cc([N+](=O)[O-])cc2c1OCCO2 73761,C1(C(N2C(C(=O)NC)CC2)=O)CCCCCCN1C(=O)C=CC(=O)N(C)C 73762,N1(C(CC2C(C)(C)OCC2)=O)C2CCC(C(=O)NCC3CC(CF)C3)C1CC2 73763,N1(C(c2c(CC)nccn2)=O)CC(O)CC1(C)C(=O)NC(c1nncs1)C 73764,C=CCC(C)(C)CC(=O)N1CCCCCC1C(=O)NC1(CO)CC(F)C1 73765,N1(C(C(C)(C)c2cncs2)=O)CCCCC1CNC(=O)Cc1n[nH]cc1Br 73766,C1(C2CCC(=O)NC2)(C(=O)NC2C(C)CN(C(=O)C(F)(F)C(C)(C)O)C2)CCC1 73767,N1(C(C23C(=O)C4CC2C3C4)=O)CC(NC(C2(Cl)CC2(F)F)=O)CC12CCCCC2 73768,Cc1cc(C#N)nc(=NC(C)CC(C)NC(=O)CCNS(C)(=O)=O)[nH]1 73769,N1(C(CN(c2ccc(F)cc2)C)=O)CC2CC(NC(=O)Cn3cccn3)C(C2)C1 73770,c1(NC(C(c2ccco2)NC(C(C)OCC)=O)=O)cccc2c1CCC2 73771,C1(NC(c2cncc(OC)c2)=O)CC2CN(C(c3cc(C)ccc3Cl)=O)CC2C1 73772,N1(C(Cc2c(C)n[nH]c2C)=O)CCC2CCCC12C(N1CC(CO)C(C)(C)C1)=O 73773,c1(C(=O)NC2C(NC(CNC(C(CC)C)=O)=O)CCCC2)n[nH]c2c1COCC2 73774,c1(C(=O)O)cccc(S(=O)(=O)NC2CCN(c3ccc(F)cc3)C2=O)c1 73775,S(=O)(=O)(c1cccnc1NC1CCOCC1F)NCC1CCCN(CCOC)C1 73776,C(CCC)(CCNC(=O)COCCOCCO)NC(COCC#C)=O 73777,N1(C(C)C)CCc2onc(C(N3CCC(N(C(=O)CC(C)CF)C)C3)=O)c2C1.C1(C)CCC1 73778,C(=O)(CCCCCCNC(=O)C(O)C1CCCC1)NCC(C(C)(F)F)Cl 73779,C(CCC)(C(=O)N1CCC(C(C)(C)NC(C23CC(C#N)(C2)C3)=O)C1)=CCC 73780,C(=O)(C(C)(C)C(=O)NC1CC1CNC(=O)CNC(c1ccccn1)=O)NC 73781,N1(C(C(C(C)C)OCC)=O)CCN(Cc2sccc2Br)CC1C#N 73782,N1(C(C(=O)NCCOC)c2cocn2)CCc2nn(C)c(=O)cc2C1 73783,CCCC(C)CCCNC(C1CCCCC1)CN 73784,CN=c1nc(N2Cc3cnn(C)c3C2)[nH]c(=NCCC2CC2C(=O)O)[nH]1 73785,Cc1ncc(C(=O)N(CC(C)(C)CNC(=O)CC2CCCC2O)C)cc1N 73786,C=C(Br)CCC(=O)NC1CCN(C(c2cc(C(N)=O)ccn2)=O)C1 73787,C12(NC(CC3N(C)CCC3)=O)CCCCC1CN(C(=O)COC(F)F)C2 73788,c1(CC(=O)NCCC(C)CCNC(C2(C)C=CCC2)=O)cc(Cl)cc(Cl)c1 73789,C1(C2(O)CCOC2)(C(N(CCCNC(C(N2CCCC2=O)C)=O)C)=O)CC1 73790,C(C(C)(O)C(=O)NCC1(C)CCCN1C(C1CCC(C)C1)=O)OC 73791,c1(C(CC(=O)NC2C(NC(CCCC)=O)CC2)C)c[nH]c2ccccc12 73792,C1(N(C)C(c2cccc(O)n2)=O)CC2CCC(C1)N2C(c1ccc(CO)cc1)=O 73793,N(S(=O)(=O)NC(C)C(C)C)(CC)CC1OCCC1c1cnn(C)c1 73794,N1(C(CNC(=O)OC)=O)CC(N(C)C(c2cnc(C(C)C)s2)=O)C(F)C1 73795,c1(C(=O)NCC(=C2CN(C(c3c(CC)n(CC)nc3)=O)C2)F)cc(C)cnc1Cl 73796,C1(C)(CC)CCCN(C(=O)C(C2CC2)N(C)C(c2cc(C(C)=O)c[nH]2)=O)C1 73797,N1(C(C(CO)OC)=O)CC(NC(=O)C(C)Cn2ccnc2)CC12CCCCC2 73798,N1(CC)CCOC(C(=O)NC2CC2CNC(C2(COC)CCCC2)=O)C1 73799,C1(CNC(CCOCCC)=O)C2CN(C(=O)Cc3ccnc(Br)c3)CC12 73800,Cc1ccc(C(F)(F)F)cc1C(N1CCCC(CNC(=O)C2=CCSC2)CC1)=O 73801,C(CCCS(=O)(=O)CCO)CCNC(=O)NC1CN(C(C)C)CC1C 73802,C1(NC(C(C(C)(C)C)SC)=O)CN(C(=O)CC2(O)CCCC2)CC(C)(C)C1 73803,C1(NC(c2ccc(CN(c3[nH]ncc3C#N)OC)cc2)=O)CC2(CCCO2)C1 73804,Cc1ncc(N)cc1C(=O)NCC1(C)CCCN1C(c1csc(S)n1)=O 73805,C(N=c1[nH]c(=NC2CCSCC2)c2[nH]ccc2[nH]1)c1c(Br)cn(CC)n1 73806,c1(OC)cccc(CC(=O)NCC(CO)NC(=O)Cc2cccc(Cl)c2F)c1F 73807,N1(C(C(CC)OC)=O)CC(C(=O)NCc2cn(C)nc2C)C(C)(C)C1 73808,N1(C(c2nccc(C(F)F)n2)C)CCC2(CCOCC2)C1 73809,c1(CC)cccc(C(N2CCN(C(=O)CCc3nncn3C)CC2)=O)c1N 73810,C1(C(N(C2CC3CC3C2)C)=O)CC2(CC(NC(c3c(F)cncc3F)=O)C2)C1 73811,Cc1ccn2nc(C(N3CCCC(NC(=O)CC(C)n4ccnc4)C3)=O)nc2n1 73812,c1(C(N(C2CCOC2)C(C)C)=O)n[nH]c2ccc([N+](=O)[O-])cc12 73813,C1(NC(c2ccc(CCC)s2)=O)C(C)CN(C(C23CC(F)(C2)C3)=O)CC1C 73814,C1(COC)(NC(=O)CSc2cccnc2)CCN(C(=O)CC2CCCOC2)C1 73815,C1(CC(=O)NC(CC)CN(C(c2[nH]cc(C)c2C)=O)CC)CCCC(C)(C)O1 73816,c1(C(C)C)cc(C(N2CC(CNC(=O)C(O)CC(F)F)C(C)C2)=O)cc(O)n1 73817,c1(C(=O)NC(C)C(C)NC(c2cccc(CF)c2)=O)cccc(N2CC=CC2)c1 73818,C(=O)(C1=CCCCCC1)NCC(CNC(C(C(C)C)NS(C)(=O)=O)=O)F 73819,O=C(CCCC(CC(=O)OC)NC(C1CC2(CCC2)CO1)=O)Oc1ccccc1 73820,c1(C(N2CC(O)(CCNC(CC(C=C)C)=O)C2)=O)nc(C)ncc1Br 73821,N1(C(C)=O)CCc2cc(CNC(C3CC3c3cncc(Br)c3)=O)ccc2C1 73822,c1(C(=O)NC2C(C(=O)NCCCC(=O)NC3CC3)COC2)ccc(O)cn1 73823,Cc1c(C(=O)NCC=CC(N2CCCC3CC23)=O)cnn1C 73824,c1(CC)c(C(=O)NCCOC)nnn1CC.C12CCCN1N1CCC2C1.C(=O)COC 73825,Cc1noc(CNC(c2c[nH]nc2CCNC(=O)C(O)C2CCC2)=O)n1 73826,N1(C(c2ccc(C)nc2C)=O)CCN(C(C2CCCN2C2CC2)=O)CC(C)(C)C1 73827,Fc1cccc(Cl)c1CN1CCC(C2OCCO2)C1 73828,CC(CN(C)C)C(=O)NCCCN(C(=O)CCc1nncs1)C 73829,C1(C(N2CC(CNC(c3c(C(C)(C)C)ocn3)=O)C3C2C3)=O)CCC(C)(C)CC1 73830,c1(C(N2C3(CNC(c4cccc(F)c4F)=O)CC(C2)C3)=O)nccn2ccnc12 73831,c1(C(CC(=O)O)NC(=O)CCNCCCO)ccccc1F 73832,c1(CN2CCC(C)(C(N3CCCC(F)(F)CC3)=O)C2)cnc2c(Br)cc(Cl)cn12 73833,C(C(C)C(C)C(=O)NCCN(C(=O)CN1CCOCC1)C1CC1)OC 73834,N1(C(C(=O)NCC(=C)C)C(C)C2CCCCC2)CCOC(C)(CC)C1 73835,c12cncc(c1)OC2=O.N1(CCCCCC)CCSCC1c1cnn(C)c1 73836,C1(C(=O)OCC(CO)OCC)CC2(CCO1)CC(F)(F)C2 73837,C1(F)(CO)CN(N2CCN(C(c3ccccc3)c3ccccc3)CC2)C1 73838,N1(C(C(CO)n2cc(C(C)(C)CC)nn2)=O)CCN(CC)C(C)C1.N(C)(C)C 73839,c1(OC)ccc(CN(C)Cc2nnn(C)n2)cc1-c1ccncc1F 73840,C1(NC(=O)C=CCC2CC2)CCCCC1NC(C1CCOCC1)=O 73841,CC1COc2ccccc2C1C(=O)N(C1CN(C(c2cnn(C)c2Br)=O)C1)C 73842,C1(NC(C(COC)(F)F)=O)CC2CCC1N(C(=O)Cn1ccc(O)nc1=O)C2 73843,c1(CNCC(=O)N(C2CCOC2)C)ccc(C(C)(C)C)s1 73844,Cc1c(F)ccc(Cl)c1C(N1CCN(C(=O)C=Cc2ccco2)C(C2CC2)C1)=O 73845,C(=O)(CS(=O)(=O)C(C)(C)C)NCCCC(C)(C)NC(c1n(CCC)ncc1)=O 73846,Cc1ncc(S(N)(=O)=O)cc1CNC1(c2nnnn2C)CCN(C2CC2)C1 73847,C1(CO)CCC(NC(c2cc(Br)c(Br)o2)c2nnnn2C2CC2)CC1 73848,C1(NC(CC(=O)NC2CC2)=O)COC2(CCN(C(=O)CCSC3CC3)C2)C1 73849,c1(OCC)ccccc1-c1cc(NCCN2CCCCC2c2cnn(C)c2)on1 73850,c1(C(N2CCC(N(C)CCO)C2)C(=O)NCc2ccco2)cccc(Cl)n1 73851,CCC(CC(=O)NC(CNC(C1(C)CCC1)=O)CCOC)C(C)C 73852,CCCCC(CC(=O)NC1C=C(C)CCC1)NC(=O)Cc1cc[nH]n1 73853,C#Cc1cc(C(=O)NCC#CCNC(=O)C(C)(CCC)OC)cc(N)c1 73854,Cc1cc(C(N2CCCCC23CC3)C(=O)NC2CCCC2)cnc1C 73855,c1(OC)cncc(C(=O)N(C(C)(C(=O)NCC(c2ccncc2)C)C2CC2)C)n1 73856,c1(OC)ccnc(NC2(c3ccc(-c4ccccc4)cc3)CCCC2)n1 73857,C1(NC(Cc2n(C)ccn2)=O)CC1C1CCCN(N2CCCC2C=O)C1 73858,c1(C(=O)NC(C(C)C)CNC(=O)C(c2ccccc2)O)cnc2ccsc2c1 73859,C1(C(N2CC3(C2)CN(C(=O)CC2CCC=CCC2)C3)=O)(OCC)CCCCCC1 73860,C1(CNC(CN(CC#C)C(C2(C)CCCC2)=O)=O)(CN(C)C)CCCC1 73861,N1(C(COCCCC(C)C)=O)CCC(NC(=O)Cn2cnc(Br)n2)C1C 73862,C1(C)(NC(C2C(C)C2)=O)CCN(C(c2ncccn2)=O)C1 73863,c1(C(=O)NC2CC3(CN(C(C4(CC#C)CC4)=O)C3)C2)cc(S(N)(=O)=O)cnc1C 73864,C(=O)(CC1=NNC(=O)C1)OC(=O)NCCCCC(C)(C)C.C12CN(C1)C(=O)N2 73865,C1(CNC(C=CCC)=O)CC2CN(C(c3nc(C)ccc3OCCOC)=O)CC12 73866,CCCCC(C)C(=O)N1CCOC(CN(C(=O)C(Br)=C(C)C)C)C1 73867,N1(C(C=NOC)=O)CCC(NC(c2cn3c(n2)CCC3)=O)C(CO)CC1 73868,N1(c2ncnc(NC3CCCC(n4c(C)ncc4)C3)c2C)CCC2(CCC2)CC1 73869,C1(C)(C(=O)NC2CN(C)C(CO)C2)CCCN(C(c2c[nH]c(=N)o2)=O)C1 73870,C1(COC)(NC(=O)C(C)=CC2CC2)CCN(C(=O)CS(=O)(=O)N(C)C)C1 73871,N1(C(CC(CC)C)=O)CC2CCN(C(c3cccn3C3CCCC3)=O)CC(C2)C1 73872,c1(C(=O)NC2COCCN(C(C3(CCOC)CC3)=O)C2)c(Br)ccc(C)c1F 73873,Cn1c(Cl)c(CNCc2cc3cccc(Cl)c3o2)c2ccccc12 73874,c1(-n2c(C(C3CC3)NC(C)(C)COc3ccccc3F)nnn2)ccc(Cl)cc1F 73875,C1(C(N(CCNC(C(CCC)OC)=O)CC)=O)CCn2cnnc2C1 73876,N1(C(C2ON=C(CC)C2)=O)CCC(C(N2CC(CC)(CO)C2)=O)C1(C)C 73877,c1(C(=O)NC(CNC(CN(C(C)C)C)=O)C2CC2)cc(F)ccc1C(F)F 73878,c1(NC(c2c(CC)cccc2)CC)ccc(S(=O)(=O)NC(C)C)cc1C#N 73879,N(C(=NCCCF)NC1CCCC1C#N)CC(c1ccccc1)(C)OCC 73880,C(c1cc[nH]n1)=CC(=O)NC1(CCNC(c2ccoc2Cl)=O)CCC1 73881,C=CC(C)(O)CC(=O)N(C1CCN(C(=O)C(=O)NCC2CC2)CC1)CC 73882,C1(NC(C(COC)OC)=O)CN(C(=O)CNS(=O)(=O)N(C)C)CCC1C 73883,c1(C(=O)NC(C2CCN2C(=O)Cc2csc(Br)n2)C)cn(C(C)(C)C)nn1 73884,c1(-c2ccc(C(=O)NC(CCC)CO)cc2)[nH]nc2c(C(=O)O)cccc12 73885,N1(c2nnn(C)n2)CCC2(CCCCC2NC(=O)CC2CCCCO2)CC1 73886,c1(C(=O)NC(CNC(CC(C)(C)OC)=O)C)ccc2cccc(Br)c2n1 73887,C1(C(N2CCC(CN(C(c3c(C)ncs3)=O)C)C2)=O)COC(=O)N1C 73888,c1(CC(=O)N(CCCCCNC(C2(C)CC(C)C2)=O)C)ccc(Cl)nc1 73889,O=C(CCCC(F)(F)CO)NC1CCOCC1NC(C1OCC2CCCC12)=O 73890,c1(CC(C)(C)NCC2(O)CCCNC2)nc2ccccc2s1 73891,c1(C(=O)NC(CNC(c2c(C(C)C)nns2)=O)(C)C(C)C)ccc(S(C)=O)cc1 73892,C1(C(N(C2CCN(C(CCSC)=O)CC2)C)=O)CCCCC(=O)N1 73893,C1(O)(CN(C(CC2C(C)CCO2)=O)C)CCN(C(=O)Cn2cnnn2)CC1 73894,C1(NC(C(C)(C2CCC2)NC(c2cc(OCC)n[nH]2)=O)=O)CCCC(O)C1O 73895,C(CCCCC(=O)NCc1ccc(CN(C(=O)C(C)(CC)CO)C)cc1)OCC 73896,C1(CNC(c2cccc(C)n2)=O)CC(C)(C)CN1C(C1SCCCS1)=O 73897,N1(C(CCC(=C)C)=O)CC(C)(C)OCC1CNC(c1scc(Cl)c1Cl)=O 73898,C1(CC=C)(C(=O)Nc2cnn(C(F)F)c2)CCN(C(=O)CCC2CC2(F)F)C1 73899,Cc1cc(CC(N2CCC(O)(C(C)CNC(c3cncc(Cl)c3)=O)C2)=O)n(C)n1 73900,CC1CCN(C(=O)C(=O)NCC2CN(C(=O)COCC(F)F)CC2C)CC1 73901,N1(C(=O)Nc2nc(C(=O)OCC)on2)CCC2C(C1)C(C)(C)O2.C1(CO)CC1 73902,CCCC(O)(CCC)CC(=O)N1CC2C(CNC(C3(C(=O)OCC)CCO3)=O)C2C1 73903,n1(C(C)C)cnc(CCNC(=O)C(=O)NCCCC2CCNC2=O)c1 73904,C12(C(N3CC(CC(=O)NCCC4CCCOC4)(OC)C3)=O)CC1CNC2=O 73905,CCCCC(CC)CC(C(=O)NC1CCOCC1)N(C)CC1CC(O)C1 73906,c1(CC(=O)NC(CNC(=O)CN2CCCC2)C2CC2)ccsc1Br 73907,c1(CNC(c2cc(CNC(c3cnc(CC)s3)=O)ncc2)=O)nnc2n1CCC2 73908,CC#CCCC(=O)NC1C2CC1N(C(=O)CCCN1CCOC1=O)C2 73909,c1(C(=O)NC2CC(C)(NC(CC3C(C(=O)OC)CC3)=O)C2)ccc(C#N)cc1C 73910,N1(C(C(c2ccc(C)s2)C)=O)CCN(c2cc(CNC(=O)C(N)=O)ccn2)CC1 73911,N1(C(c2occ(C)c2)=O)CCC(NC(c2ccc(C(F)F)cc2)=O)C(C)(C)C1 73912,N1(C(CC2(OC)CCOCC2)=O)CCOC2CN(C(=O)CCN(C)CCO)CC12 73913,c1(-c2scc(N(CCN(C(=O)COC3CCCCC3)C)C)n2)cccc(Cl)c1 73914,C(=O)(CCCC(C)(F)F)N1CC(NC(CC2CC(OCC)C2)=O)C(C)(C)C1 73915,N1(C(=O)Cc2ccc(Cl)nc2)CC2CN(C(=O)C(CO)c3ccccc3)CC2C1 73916,CC1COCCN1CCNC(=O)C(C1CCCO1)NC(c1coc(C(C)C)n1)=O 73917,N1(C(CCC=C)C(=O)Nc2ccc3c(c2)OCO3)CCCCCCCCC1 73918,Cn1ccc2c(-c3cncc(F)c3C(N3CCC(C)(C#N)CC3)=O)cccc12 73919,C#CCCC(=O)N(CCNC(c1ccccn1)=O)CCNC(C)=O 73920,O(NC(=O)CC(C(F)F)NC(C1CCCN1C)=O)CCN(C)C 73921,C1(CNC(C2CC(C)OC2C)=O)CN(C(=O)CCS(C)(=O)=O)CC(C)(C)O1 73922,C1(NC(c2n(CCCC)nnn2)(C)CCN2CCSCC2)CC(C)N(C)CC1C 73923,N1(C(C=CC)=O)CCC(NC(=O)Cn2ccc(NC(=O)OC(C)(C)C)n2)C(C)C1 73924,c1(NC(C2C(OCC)CN(C(C3CCNC(=O)C3)=O)C2)=O)cccc(C)c1C 73925,c1(CC(=O)N(CC(CNC(c2ccnc(C)n2)=O)O)C)ccc(Cl)c([N+](=O)[O-])c1 73926,C1(OCC)CC2CN(C(=O)NC(c3cccc(Br)c3C)C)CC12.OCC 73927,c1(NC(c2cc(CNC(C(C)N(C)C)=O)oc2)=O)cccc2c1OCC2 73928,C1(NC(CCC)=O)CCCC12CCN(C(=O)C=CC(=O)OCC)CC2 73929,N1(C(COC(C)C)=O)CC(C(N2CCC(CCCO)C2)=O)C(C2CC2)C1 73930,C(=O)(C1=CC2CCCC12)NCC1C(C)(C)CCN1C(=O)CC1=CCCC1 73931,Cc1cc(F)ccc1NC(C1(C)CCCN1C(=O)COCCN(C)C)=O 73932,C1(C(=O)NCC(=O)N(C)CC)CN(C(C2(N(C)C)CC2)=O)CC1C1CC1 73933,Cc1cc(C(N2CC3CC3C2C(=O)NCC(O)C(C)O)=O)nc(C)n1 73934,C1(C2CC2)(C(=O)O)CCN(C(C2CCC23CCCC3)=O)C1 73935,c1(NC(c2ccc(NC(C3(O)CC3)=O)nc2)=O)ccc2ccncc2c1 73936,Cc1ccc2nc(C)cc(C(=O)NC(C)CN(C)C(c3ccc(F)cc3)=O)c2c1 73937,C1(NC(C=NOC)=O)CCCC2CN(CCON=C3CCCCCC3)CC12 73938,N1(C(c2n[nH]c(C)c2C(F)(F)F)=O)CCC(NC(c2nncs2)=O)C(C)C1 73939,C(=O)(C(F)(F)C(C)O)NCC1N(C(C(C)Cc2ccc(N)cc2)=O)CCC1 73940,N#Cc1ccccc1CCCC(=O)NC1CCCCN(C(c2ccncc2)=O)C1 73941,N1(C(C(CCC)F)=O)CCN(C(c2cc(CC(C)C)on2)=O)C(C2CC2)C1 73942,S(=O)(=O)(CCC(=O)NC(C)(C)CCNC(c1c[nH]nc1-c1ccncc1)=O)NC 73943,C1(CNC(COCCCOC)=O)CN(C)CCN1C(=O)Cn1cccnc1=O 73944,N1(C(C(C(C)C)=O)=O)CC(NC(c2c[nH]nc2C(F)F)=O)CCC1C 73945,N1(C(=O)Nc2cnn(CCF)c2)CCCC(N2CCCC2)C1.C12CC(C1)C2 73946,C1(NC(C2CC(OC)(OC)C2)=O)CC(C(=O)N(C)Cc2nc(C)no2)C12CCC2 73947,c1(N2CCCN(c3c(N)c(Cl)ccn3)CC2)ccc2nncn2n1 73948,c1(C(N(CC(C)NC(C2CCCN(CCC)C2)=O)C)=O)c(Cl)ccc(C)c1O 73949,c1(C(N2CC(CNC(=O)CSCc3cscn3)C2)=O)cc2c(cc1Cl)NCC2 73950,C(CC)(CCC(=O)NCC1CCCC(C)(C)C1)NC(c1c(OCC)cccc1)=O 73951,C1(NC(C=C(CC)C)=O)C2COCC1CC(NC(=O)CCCn1ccnc1)C2 73952,N1(C(c2c(CCCC)ocn2)=O)CCOCC1CN(C)C(c1cc[n+]([O-])cc1)=O 73953,c1(C(N2CC(C(C)NC(C3CCC(OC)C3)=O)C2)=O)cc2sccc2n1C 73954,CCC(O)C(C)(C)C(=O)N1CC(NC(c2c(Cl)n[nH]c2C)=O)C(O)C1 73955,c1(C(=O)NC(CNC(c2n(CCC)ccc2)=O)CCOC)ccc(=O)n(C)n1 73956,Cc1nc(-c2ccc(Cl)cc2)oc1C(N1CCSC(C(N)=O)C1)=O 73957,C1(COC)CC(C2CCOC2)C1.c12nnc(s1)CN2C(CC)CC 73958,CC(C)C(C)C(=O)NC(C1CN(C(C2CN(C)C2)=O)C1)C 73959,C1(C(N(CC)CC)=O)CCCCC1NC(c1cc(C)nn1-c1ccncc1)=O 73960,C1(C(=O)N(CCCCNC(c2ccc(Cl)cc2)=O)C)(CC)CCCCO1 73961,N1(C(C2(F)C(C)OCC2)=O)CC2(C1)C(NC(=O)C(O)C1CCCC1)CCS2(=O)=O 73962,C#CC1(N(C)C)CN(C(C2CC=CCN2C(=O)CC2COCC(C)O2)=O)C1 73963,N#CC1(C(=O)NCC2CC(NC(c3ccc(CO)nc3)=O)C2)CCOC1 73964,c1(C(=O)NC(CNC(C2CC=CCC2)=O)CO)ccc(-c2cnc[nH]2)cc1 73965,CC1Cc2cc(C3(NC(=O)C(N4CCNC(=O)CC4)=O)CC3)ccc2O1 73966,Cc1[nH]nc(C(N2CC(O)CC2C(=O)NC(CO)C2(C)CC2)=O)c1O 73967,CON1CCC(CC(=O)N(CC(O)CNC(c2c[nH]ccc2=O)=O)C)CC1 73968,CC1(C)CCCCC1C(N1CCC(F)(CNC(=O)CCCC(F)F)C1)=O 73969,c1(C(N(CCNC(C(C(C)C)F)=O)C2CC2)=O)c(F)ccc2nc[nH]c12 73970,CC1CCN(C(C2(N(C)C(c3ccc(O)nc3)=O)CC2)=O)C(C)C1 73971,C1(O)(CC)CN(C(C2CCC2(OC)OC)=O)C1.c12ncoc1CNC2=O 73972,CCC(C)(C)C(C)CC(=O)NC1CCC(NC(=O)CCOC2CCOCC2)C1 73973,CCC(CC(=O)NC1CN(C(=O)C2=C(Cl)CC2)CCC1C(F)(F)F)C(C)(C)C 73974,CC1CN(C(C2(N(C)C(C3CC34CCOCC4)=O)CC2)=O)Cc2c[nH]nc21 73975,n1(CCCCNC(c2ccc(C#C)o2)=O)c(C)cc(C(=O)O)c1C 73976,c1(C(=O)NC2CC(C(C)NC(=O)C(F)C3CCOC3)C2)ccc(F)c(F)c1 73977,CCC(O)(CNCCCCCOC(C)(C)C)C(F)(F)F 73978,CCC(CCC(=O)NC1CC(N(C(=O)CN(C)CC2CC2)C)C1)OC 73979,C(=O)(C1Cc2c(Cl)cccc21)N1CCC(C)(NC(C(COC)C)=O)C1 73980,c1(SC)cnc(C=CC(=O)NC2CCC2)nc1.C1(C2CC2)C(=O)N1CCC 73981,N1(C(c2c(C)n(C)cc2)=O)CCC(NC(C2CC(O)C2)=O)CC(C)(C)C1 73982,Cc1c(Br)cc(C(=O)NCC2(O)CN(C(C3CC(=C4CC4)C3)=O)C2)c(=O)n1C 73983,C1(NC(c2csc(Cl)c2Cl)c2n(CCSC)nnn2)CC12CCCCC2 73984,CC(CC(F)(F)F)C(=O)NC12COC(C1)C(NC(c1nccn3ccnc13)=O)C2 73985,N1(C(C2C(CCC)CCC2)=O)CCCC2(C1)CN(C(C1(SC)CC(=O)C1)=O)C2 73986,CCC(C)C(O)C(C)C(=O)N1CC(C)(NC(c2cncc(NC)n2)=O)C1 73987,c1(C(N2CCN(C(Cc3scc(C)n3)=O)CC2C(F)F)=O)c(C)cc(F)cc1C 73988,Cc1cc(C)c(CNc2ccccc2N(C)CCN(C)C)cc1C 73989,c1(C(N(C(c2ccncc2)CC)CC)=O)nc(C)ccc1F 73990,C1(C(=O)NCc2c(C)ocn2)N(C(=O)COc2cnn(C)c2)CC12CCCC2 73991,c1(N(C)C)ccc(NC(=O)CCc2ccc(C(=O)Nc3cccnc3I)[nH]2)cc1 73992,C1(NC(C2(C)C(C)(C)C2)=O)C=CCC(C(N2CC=CCC2)=O)C1 73993,CCCCCC(O)C(C)C(=O)N1CCN(C(c2ccc(Cl)s2)=O)CC(C)C1 73994,c1(OC)cnc(F)c(C(=O)NCC2(CCNC(c3nccs3)=O)CC2)c1 73995,c1(CNCc2ccc(-c3c(CO)cncn3)nc2)cccc2nonc12 73996,C1(C(=O)NC2C(NC(Cc3cn(C)nc3C(F)(F)F)=O)C2)CCCS(=O)(=O)C1 73997,c1(SCC)cnccc1C(=O)NCC1CN(C(=O)C(O)c2ccsc2)CCO1 73998,C1(C(=O)NCC23CCC(CC2)C3)CC(O)CCN1C(C1CC12CCOCC2)=O 73999,CCCCCC(C(=O)NCC1=CCN(C(C2CCC(C)O2)=O)CC1)C(C)C 74000,CCC(CC(F)F)C(=O)N1CCN(C(=O)C=Cc2ccc(C(F)F)o2)C(C2CC2)C1 74001,c1(C(=O)NC2CCCN(C(C(C)OC)=O)C2C)c(F)cc(C)cc1Cl 74002,N1(CCNC(c2c(C)cccn2)=O)CCCN(C(C2(C)CCOCC2)=O)CC1 74003,Cc1nc(C(=O)NC(C)(C)CNC(=O)C(O)Cn2cncn2)c(C)n1C1CC1 74004,C(C(F)(F)CC(O)CO)NC(N(C)Cc1cccc(Cl)c1Br)=O 74005,c1(C(=O)NCCN(C(=O)C(C)(F)C(F)(F)F)C)cc2ccc(Cl)cc2s1 74006,CC1(C)CN(c2nc(=N)[nH]c(=NCc3ccc4nncn4c3)[nH]2)CCS1(=O)=O 74007,n1(CC)ccc(C(N2CCCN(C(=O)C3=CCCCC3)CC2)=O)cc1=O 74008,c1(OC)ccc(C(=O)NCC(C)(O)CNC(=O)CCc2ccc(F)nc2)nc1N 74009,N1(C(c2c(C)cc[nH]c2=N)=O)Cc2ccccc2C(CNC(c2ccns2)=O)C1 74010,c1(OC)ccc(C(C)C)c(C(=O)NC2CN(C(C3C4CCCC34)=O)C2)c1 74011,Cc1cc(C)n2ncc(C(=O)NCC3CN(C)CCN3C(=O)C3CC3)c2n1 74012,c1(C(C(=O)NCCSC)N(C2CCNC(C)C2)C)c(Cl)nc2sccn12 74013,CS(=O)C=CC(=O)NCC1CN(C(c2cc(CN(C)C)on2)=O)CC1O 74014,C1(NC(CCN(C)CCO)=O)CC(O)CN(C(c2cncc(C(N)=O)c2)=O)C1 74015,c1(C(N(C(CC)C)CC)=O)n[nH]cc1CNC(=O)CSC 74016,c1(C(N2CCC3(NC(CCCN(C(C)C)C)=O)C(C2)C3)=O)c(F)ccc(N)c1F 74017,N1(C(=O)CC2(c3ccccc3)CC2)CCN(C(C23CC2C3)=O)CC(CO)C1 74018,c1(OC)ccc2c(c1)CCN(C(=O)C(=O)N(CC1CCCCN1C(C)=O)CC)C2 74019,C(=O)(CC(C)(C)COC)NCC(CC)NC(=O)C(c1cccc(O)c1)OC 74020,Cc1ncccc1C(=O)NC1C=CCN(C(=O)CC2CCNC(=O)C2)C1 74021,c1(N(C(c2cc(O)c(O)c(O)c2)=O)CCC2CCCNC2)ncnc2n[nH]cc12 74022,CC1CC2CC(C(=O)NCC3CN(C(c4c(Br)nnn4C)=O)C3)(C2)O1 74023,N1(C(c2ncn(C(C)C)n2)=O)CCOC2(C1)CN(C(C1COCC(C)(C)O1)=O)C2 74024,C1(CNC(c2nc(CCC)sc2)=O)CN(C(c2cnsc2)=O)C2CC12 74025,C1(C(=O)NCC(C(C)C)NC(c2ccncc2F)=O)CCC2(CCOCC2)O1 74026,CC(C)C(C)C(CNC(=O)C(C)CF)Nc1ncc(O)cn1 74027,Cc1c(C(=O)NCC2CC3CCC(C2)C3)c[nH]c1C#N 74028,C1(C(N2CC(CNC(c3c(CC)c(C)sc3)=O)C2)=O)COc2ccc(Cl)cc2O1 74029,CN1CCCN(C(=O)CC(C(F)F)NC(C2(C)CCN(C)C2)=O)CC1=O 74030,N1(C(c2c(C)cn(C)n2)=O)CCN(C(=O)CCCc2ccc(Cl)cc2)CCC1C 74031,c1(N2CC3(CCN(C(CC(=O)N(C)C)=O)C3)C2)nc(Cl)nc2[nH]cnc12 74032,c1(NC(C(=O)NC2CCC(=C)CC2)=O)ccc2ncsc2c1Br 74033,C(CC1CC1)(C(=O)NOCCF)NC(C(C(C)O)N(C)C)=O 74034,C1(NC(c2n(CCSC)nnn2)c2cnc(C(F)F)s2)CNC(=O)OC1 74035,C1(C(N(CCCNC(CNC(C)=O)=O)C)=O)CN(C)C2(CCC2)C1 74036,Cc1ccc(F)cc1C(N1CC=CC(C(=O)NC2CCC(ON)CC2)C1)=O 74037,Cc1ccc(C=CC(N2CC(F)CC2CNC(C2(C3CC3)CCCO2)=O)=O)o1 74038,C1(C(=O)NCCN(C(CCOCC#C)=O)CCOCCO)CNC(=O)CC1(C)C 74039,c1(CN2CCC(N3CC(=O)NCC3)CC2)nc2ccc(Br)nc2[nH]1 74040,c1(CC)cc(C(=O)NCC2CN(C(c3csnc3C)=O)C(C)(C)C2)cn(C)c1=O 74041,n1(CC(=O)NC2CCC(NC(c3ncn(CC)c3)=O)C2)cnc2sccc2c1=O 74042,C1(C(C)(C)NC(Cn2c(C)cnc2)=O)CCN(C(c2[nH]ncc2C#N)=O)CC1 74043,CC(=O)C(C)CC(C)C(=O)NCc1nocc1C(=O)NCC(F)CO 74044,c1(NC(C)=O)ccc(C(=O)NCC2CCN2C(C2CCCCC2F)=O)cc1 74045,C1(C(=O)NC2CN(C(CC3CCC(C)(C)C3)=O)CC2O)CCS(=O)(=O)CC1 74046,c1(CC(=O)NC2CCC(N(C(=O)CCF)C)CC2)c[nH]c2ccc(Cl)cc12 74047,C1(C(C)NC(=O)CCc2ccnn2C)CCN(C(=O)C(C2CC2)N(C)C)CC1 74048,Cc1nc(C(C)C)[nH]c(=NC2CC(NC(=O)C3=NOC(C)(C)C3)C2)c1Br 74049,C1(NC(C(=O)NCC(C(=O)OC)C)=O)CC2(CCCC2)C1 74050,c1(C(CNC(CCC)CO)C)cccc(F)c1 74051,C1(CC)CCN(N(C)CCCCc2ccc(Cl)cc2Cl)CC1 74052,N1(C(C=CSC)=O)C2CCC1CC(N(C)C(c1ccc(C3CCC3)cc1)=O)C2 74053,c1(CC)nc(C(=O)N(C)CC2CCCN2C(=O)C=C(C)C(C)(C)C)cs1 74054,C1(C)(CNC(COCC#C)=O)CCC(NC(=O)COCc2nc[nH]n2)C1 74055,C1(C)(OCC(=O)NCCN(C(c2cc(C(=O)OC)oc2C)=O)CC)CCOCC1 74056,N1(C(CC2N(CC)CCC2)=O)CCC(O)(CCNC(=O)C=CC(F)F)CC1 74057,c1(CN(C)C(=O)Nc2[nH]ccc2C2CCC2)cc(C(F)(F)F)c(Cl)cn1 74058,Cn1nc(C(=O)NCCC2CCCN2C(=O)CN2CCOC2=O)cc1O 74059,NC(=O)CCC(=O)NC1CCCC(CNC(=O)Cc2coc(-c3cccs3)n2)C1 74060,N1(C(c2nc(C)n(C(F)F)c2)=O)CCC(C)(NC(=O)C(C)C(F)(F)F)CC1 74061,C1(=CC(=O)N(CC(C)NC(=O)C2=CC(O)CCC2)C)CCCCCC1(F)F 74062,c1(C(N2CC(C(C=O)OC)C2)=O)nnc(S)n1C.N1CC(F)(CF)C1 74063,CC(CC(C)(F)F)C(=O)N1CC(F)(F)CC1CCNC(=O)C(C)(C)c1cccs1 74064,C#Cc1cnncc1C(=O)NCC1(C)CCN(C(=O)C(C(C)C)SCC)CC1 74065,N1(C(c2n(CC)nc(C)c2)=O)CCN(C(=O)Cc2ccno2)CC2(CC2)C1 74066,C1(NC(c2c(OC)nn(C)c2)=O)CC(C)(C)C12CCC2 74067,C(=O)(C(O)CC(C)(C)C)N(C(C(=O)NCCC=CCCC)C)C1CC1 74068,N#CC1CCCN(C(c2cccc(C(F)F)c2F)C(=O)Nc2ccccc2Cl)C1 74069,S(=O)(=O)(c1ccc(S(N)(=O)=O)cc1)N1C(C)CCCC1C 74070,CC(C(=O)NCC1CCN(C(=O)CSc2ccc(Cl)cc2)C1)C(C)(F)F 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75017,Cc1nn(-c2ccc(Cl)cc2)cc1C(=O)NC1CC1CNC(=O)C=CS(C)=O 75018,C1(C2(O)CCOCC2)(C(=O)NCC2CC(NC(CC(C(F)(F)F)OC)=O)C2)CC1 75019,c1(N(C2(CC)CC2)C)ncccc1S(=O)(=O)NCCC=CBr 75020,c1(C(=O)NCC2CCCC(NC(C(C)C3(O)CCC3)=O)C2)ccsc1S(C)(=O)=O 75021,C1(C(N(CCCCNC(C(N2CC(C)C2)C)=O)C)=O)CCOC(C)(C)C1 75022,C1(CC)CN(C(C2CC3C(C2)C3(C)C)=O)CCN1C(c1cnc(C(C)(C)C)s1)=O 75023,C(=O)(CCCC(C)(C)NC(=O)CNc1ccccn1)NC1C(CCC)CCCC1 75024,C1(C(F)(F)F)(C(=O)NCC(CCOC)NC(c2cn(CC)nn2)=O)CCN(C)C1 75025,c1(C(N2CC(NC(C(C)n3cncn3)=O)C(C)C2)=O)cccc(O)c1Cl 75026,N1(C(c2c(C)ccs2)=O)CCCN(C(C2CC3(CCOC3)C2)=O)CC1 75027,C(=O)(C(F)(F)C(F)F)NCc1c(Cn2cc(-c3cccc(OC)n3)nn2)nco1 75028,CC(C)C(C)C(CNC(C1CC=CC1)=O)NC(c1nscc1Br)=O 75029,C#CCCCC(=O)NCCCN(C(=O)CC1CCN(CC(F)(F)F)C1)CCO 75030,C(CCN=C(NCc1cccn1C)NCC1(CO)CCCC1)OC(C)C 75031,C1(CC#C)(CNCCCc2n[nH]c(=N)s2)CC1(C)C 75032,c1(C(=O)NCC2C(NC(CCC(C)C)=O)CCCC2)ccc([N+](=O)[O-])c(C#N)c1 75033,N1(C(CNC(=O)NC)=O)CCCC2(CCN(c3cc(C)nc(C(C)(C)C)n3)C2)C1 75034,C(=O)(C(F)CCC(C)(C)C)N1CC(C(=O)NCC2(N(C)C)CC2)(CC)C1 75035,CC(F)(F)C(=O)NC1CCN(C(c2cc(C3CC3)no2)=O)C1 75036,C1(CC)CCC(C)N(C(c2c[nH]nc2CNC(c2ocnc2C(C)C)=O)=O)C1 75037,C1(C(=O)NC(c2cccnc2)CO)(NC(=O)C(F)C2CCC2)CC(F)C1 75038,C1(CC=C)(C(=O)NCCCCCOC)CCN(C(=O)C(C)OCCOC)CC1 75039,CCCCCCC(=O)N1CCC(C(C)C(N2CC(N3CCC3)C(F)C2)=O)C1 75040,Cc1c[nH]c(C(=O)NC(CNC(=O)C=Cc2cccs2)CO)c1 75041,N1(C(C2CN(C(C)=O)C2)=O)CCC(C)(C)C1CNC(c1nnc(O)cc1O)=O 75042,c1(C(N2C(CN(C(=O)CC(C)(C)C3CC3)C)CCC2)=O)nc(Cl)ccc1N 75043,N1(C(CC(C(C)C)OCC)=O)CC2CCCN(C(=O)CC(O)CC(C)C)C2C1 75044,CC1(C#CC(=O)NCC(C2CC2)NC(C2(OCC(CCl)OC)CCOC2)=O)COC1 75045,Cc1ccnc(O)c1C(=O)NCCOCCCN(C(=O)C(F)=C1CC1)C 75046,c1(C(=O)NCC2CC(F)(CNC(C3(N(C)C)CCC3)=O)C2)cc2c(s1)CCC2=O 75047,C=CCC(C(=O)Nc1ccsc1)NC(=O)CC1CCCC(=O)N1 75048,c1(C(N(CCCCN(C(=O)Cc2cncc(F)c2)C)C)=O)cnccc1Cl 75049,c1(C(c2nnnn2CC=C)NCCCC(=C)C)cccc2c1CCO2 75050,C1(NC(CN(C)C)=O)CN(C(=O)OC(C)(C)C)CC1C#N.c12csc(n1)CNC2=O 75051,C(C(C)C(C)C(=O)NC(C)(C)CN(C(=O)COC1(C)CCCC1)C)OC 75052,N(C(=NCCc1ccccc1Cl)NCC1CCCCO1)C(C)Cc1ccccc1 75053,N1(C(C(CC)n2ccnc2)=O)CCC(NC(c2sc(C)cc2C)=O)C(F)C1 75054,c1(SC(C(=O)N(C2CCN(C(c3nc(C)nn3C)=O)C2)CC)C)ccccc1C 75055,c1(C(N2CCN(C(=O)C=CC3CCOCC3)C3CC23)=O)cc2nccn2c(O)n1 75056,N1(C(c2oc(CC)c(C)c2)=O)CCC(C)(C)C1C(=O)NC1CCOC(C)(CC)C1 75057,N1(C(C(CC#C)C2CC2)=O)CCC(C)N(C(c2ccc3ncccn23)=O)CC1 75058,c1(OC)n[nH]c(C(N2CCOC(CN(C(=O)CSCc3ncc[nH]3)C)C2)=O)c1Cl 75059,C1(CNC(C2CCCO2)=O)CC(NC(c2cc(C3CCOCC3)no2)=O)CC1O 75060,N1(C(CSCC(C)C)=O)CCC2(CC1)CN(C(=O)CC1CCOC(C)(C)C1)C2 75061,C(=O)(C(C)C(C)(C)C)N(CC(=O)NC1CN(C)NC1=O)C(C)C 75062,c1(C(N(CC(CC)NC(=O)C2=C(C)CC2)C)=O)cc(C)c(=O)n(C)c1 75063,Cc1cc(C(=O)NC2CCC(NC(C3CC(F)C3)=O)C2)ccn1 75064,C(CN=C(NCc1cc(C(F)(F)F)n[nH]1)NC(C)CC(F)(F)F)OCC=C 75065,C(=O)(C(C)(C)c1ncco1)N(CCNC(=O)CCSCC(N)=O)CC 75066,n1(CC(=O)N(C(CNC(Cc2ncc(C)[nH]2)=O)C)C)cc(C#N)cn1 75067,C1(NC(Cc2c(C)n(C)cn2)=O)CCN(C(c2cc(Cl)ccc2N)=O)CC1F 75068,c1(OC)ccc2cnc(C(N3CCCC(CO)(NC(=O)C(F)OC)C3)=O)cc2c1 75069,C(CC1=CCCCC1)N(CCC(N1CC2C(C(N(CC(N)=O)C)=O)C2C1)=O)C 75070,C12(NC(C(c3ccc(F)cc3)CC)=O)CCCC(NC(C3CCN(C)C3)=O)(C1)C2 75071,C1(C)(C(=O)NC23CC(NCc4ncc(NC)nc4)(C2)C3)COc2ccccc2O1 75072,C(c1cccc(C)c1)=CC(=O)NC1CCC(C(=O)NC(C#C)COC)C1 75073,C1(CCNC(C(c2ccc(Cl)cc2)(C)C)=O)CSCCN1C(C1CCCC1)=O 75074,N1(C(C(CO)OC)=O)CC(C(=O)Nc2cnc(C3CC3)nc2)CCC1(C)C 75075,C(C(CC(F)(F)F)NC(=O)CC(C)n1cccn1)NC(CC=CCC)=O 75076,c1(CC)cccnc1C(N1CCCC(C(C)NC(C2(CF)CCC2)=O)C1)=O 75077,Cc1nc(O)nc(C)c1CCC(N1CCC(O)C(NC(c2n[nH]cc2F)=O)C1)=O 75078,CN1Cc2ccccc2CC1C(=O)NC1CCCN(Cc2scnc2C2CC2)C1 75079,C1(CNC(=O)COC(F)(F)F)CC(O)CN1C(=O)CNC(=O)C1CC1 75080,CC(C)CC(C)(C)C(=O)NC1CCC1NC(c1ccc2cc[nH]c2n1)=O 75081,c1(CNC(C2C(=C)CC2)=O)nc(CNC(C2(CO)CC(F)(F)C2)=O)cc(O)n1 75082,C1(C(N2CCC(O)(C(=O)NC3C(OC)(OC)CC3)C2)=O)CCc2c[nH]nc2C1 75083,c1(C(N2CC(CC=C)(NC(C3CC(C)CO3)=O)C2)=O)cc(NC(C)=O)ccc1F 75084,N1(C(C=CC(C)(C)NC(c2cc(OC)ns2)=O)=O)CCCCCC1CCO 75085,c1(C(C)=O)cc(C(=O)NC2CCN(C(C3CCCN3CCC(C)C)=O)C2)n(C)c1 75086,c1(CC)ccc(C(N2CCC(NC(c3cn(C)nc3C)=O)C(F)C2)=O)cc1F 75087,N1(C(C(C)C(C)O)=O)CC(C)(C)OC2(C1)CN(C(c1ccsc1Br)=O)C2 75088,Cc1nc(C(=O)N(C(C)CNC(c2cnc(C(N)=O)s2)=O)C)cn1C(F)F 75089,C1(CNC(C(C(CC)C)C)=O)CC2CCC(C1)N2C(=O)C(C)C1CCCO1 75090,C(=O)(C(CC(=O)NC1(CNC(c2cc3oc(C)cc3[nH]2)=O)CC1)C(C)=O)OCC 75091,N1(C(Cn2c(C)nnn2)=O)CCC2(C1)CN(C(C1(O)CC(C)(C)C1)=O)C2 75092,c1(CNC(C(CCC#C)O)=O)nn(C)c2c1CN(C(=O)C(C)N(C)C(C)=O)CC2 75093,Cc1nc(Br)c(Br)n1CC(=O)NC(c1ccnn1C)CO 75094,C1(C(=O)NCC(CNC(CC2(NC(C)=O)CC2)=O)O)CN2CCCN1CC2 75095,c1(NC(N2C(CC(=O)OC)COCC2)=O)cc(C)cnc1N1CCOCC1 75096,c1(C(N(C(c2ccccc2)CNC(C=C(CCC)C)=O)C)=O)sc(C)c(C)c1C 75097,CCC(C)C(O)C(C)C(=O)NC(C(=O)NCCc1ccncc1C)c1cccs1 75098,C(C(=O)NCc1cncs1)(C(C)(C)C)NC(C(N1CC(C)C1)C)=O 75099,c1(C(C(=O)NCC(C)(C)CN(C)C(C2CCS(=O)(=O)C2)=O)OC)ccccc1C 75100,N1(C(c2cc(C)ncn2)=O)CCC(CNC(C2COC(=O)N2)=O)C1(C)C 75101,C(CCC(C(=O)N(CC(C)(C)C)C)NC(=O)CC1CCCC(=O)N1)OC 75102,C1(NC(c2c(C)cn(C)c2)=O)C(C)CCN(c2ncc(Br)cn2)C1C 75103,N1(C(c2cc(C)cc(F)c2)=O)CCCN(C(C2CC=CCC2)=O)CC1C(C)C 75104,N1(C(c2cn(CC=C)nn2)=O)CCC2CN(C(=O)Cc3ccc(Cl)s3)C(C)C12 75105,C(=O)(C1CCCc2sccc21)NC(=O)COC(c1cc2ccccc2c(O)n1)=O 75106,N1(C(c2nc(Br)cs2)C(=O)NCC2CCCO2)CCN(CC2CCOC2)CC1 75107,C(C(COC)C(=O)NC1(O)CC(C(N2CCC(CCCO)C2)=O)C1)OC 75108,N1(C(C(C=C)OC)=O)CC2(CC(CNC(=O)CSC3CCOC3=O)CO2)C1 75109,c1(C(=O)NCC(CNC(=O)C2=NOCC2)O)cnc2[nH]c(O)nc2c1 75110,C1(C(=O)NC(C)C(=O)NCC2CC3(CC3)CO2)CCC(O)CN1C 75111,N1(C(C2C(C)(C)C2CO)=O)CCC(CNC(C2(C(O)C(F)(F)F)CC2)=O)CC1 75112,C1(S(N)(=O)=O)(C(=O)NCC2CN(C(C(C)(O)C3CC3)=O)C2)CCC1 75113,C1(OC)CN(C(=O)CNc2cnn(C)c2)C(C)(C(=O)NC2CN(C)C2)C1 75114,C1(C(COC)N(C(c2ccccc2)C(=O)NCCN(C)C)C(C)C)CCCCO1 75115,N1(C(CN(CC)CC)=O)CC2CCCC2(NC(=O)C(C)Cc2ccc(C)cc2)C1 75116,C(=O)(C1CCc2c[nH]nc21)NCCCN(C(=O)CCn1cncn1)CCC 75117,Cc1ncc(CNC(=O)CC=CCNC(=O)Cc2cc(C)on2)s1 75118,C(=O)(C(C)CCC(C)(C)C)N1CC(O)CCC(NC(C=CCCC(C)C)=O)C1 75119,c1(CC(=O)NC2CCCC(CNC(C)=O)C2)ccc(F)cc1[N+](=O)[O-] 75120,N1(C(c2c(CC)c[nH]c2)=O)CCCC(CO)(CNC(C2CCC2C)=O)C1 75121,N1(C(c2ccc(F)s2)C(=O)NCC)CCc2c(cc(F)c(F)c2F)C1 75122,c1(OC)ccncc1C(N1CCCC(N(C(=O)C(=O)N(C)C)CC2CC2)C1)=O 75123,Cc1ccc(C#N)cc1C(N1CC(CNC(=O)CC(O)CN(C)C)CC(C)C1)=O 75124,c1(C(N2CCC(O)(CN(C(C3CCC(=C)CC3)=O)C)C2)=O)cc2ccsc2n1C 75125,C1(C)(CC)CC(NC(c2cccc(OCCF)n2)=O)CN1C(C1(O)CC1)=O 75126,C12(NC(C)(C)C)C(NC(N(CCCOC)Cc3cccs3)=O)C3CC1C2C3 75127,Cc1cc(C(=O)NCc2occc2C(=O)NOCc2noc(C)n2)ccc1F 75128,c1(C(=O)NCCC(CNC(c2c(C)n(C)nn2)=O)O)cc(C(F)(F)F)ccc1F 75129,c1(N(CC(=C)Br)C)nc(N2CC=C(CN(C)C)CC2)nc2ccccc12 75130,n1(C(C)C)cnc2c(NCC3(C)CS(=O)(=O)C3)[nH]c(=NC3CCCCC3C)nc12 75131,C1(S(C)(=O)=O)(C(=O)NCC2N(C(C3C(CC)N(C)CC3)=O)CC2)CCOCC1 75132,Cn1c(=O)n(CCC(=O)NC2CCCCN(c3ncns3)C2)c2ccccc12 75133,C(CNC(c1coc(O)n1)=O)(CC(F)(F)F)NC(CN1CCCC(CC)C1)=O 75134,c1(CC)c(C(=O)NC2CC(NC(=O)C(F)(F)CC)C(O)C2)csc1C 75135,c1(SC)nc(Cl)cc(=NC(C)CNC(c2cc(C)n(C3CC3)c2C)=O)[nH]1 75136,C1(NC(C(CC)=CC)=O)CCCN(C(=O)CCCC(C)N(C)C)C1C 75137,O=C(C#CC1CCOC1)NCCn1cnc(C(=O)NCC(O)CO)c1 75138,c1(C(N2C(CNC(CC(C(=C)C)O)=O)CC2)=O)ccsc1S(N)(=O)=O 75139,N1(C(C23CN(C(c4cn5cccnc5n4)=O)C(C2)CO3)=O)CCCC(F)C(F)(F)C1 75140,c1(C=O)cc(C(=O)OC)cc(CN2CC3CCC2C3)c1.C1(COC)(COC)CCO1 75141,C1(C(N2CC(OCCCCC)C2)=O)C=CCN1C(=O)C(n1ccc(C)n1)C 75142,C1(NC(c2ccc(C(CC)(C)C)cc2)=O)CCN(C(=O)C(C)C(C)C)C12CCC2 75143,C1(OC)CN(C(=O)CC2(O)CCCC2)CC1NC(=O)C(C)Sc1ccccc1 75144,CCC(C(=O)NCC(C1CC1)NC(C1CN(S(C)(=O)=O)C1)=O)n1nccc1C 75145,N1(C(c2c(CC)ccs2)=O)CCC(C(N2CCCCCC2)=O)C1C(C)C 75146,c1(NC(C23C(CN(c4nc(SC)c(F)cn4)C2)C3)=O)cc(F)c(C#N)cc1F 75147,C=C(Cl)C(C)(C)C(=O)NCCC1(NC(c2cnc(C3CCOCC3)s2)=O)CCC1 75148,c1(C(=O)NC2CN(C(CCOC)=O)C3C2C3)ccc2ncn(C)c(=O)c2c1 75149,C1(CC)CN(C(=O)CCCN(C)C)CCC1NC(C1(F)CCCC1)=O 75150,C1(CCNC(COCC(=C)C)=O)CN(C(c2cnc(N(C)C)s2)=O)CCO1 75151,N1(C(=O)COC2CC=CC2)CCC2CCC(C1)N2C(c1cc2cc(Cl)sc2[nH]1)=O 75152,N1(C(c2cc(OC)cc(F)c2)C(=O)NCCC#N)CCCc2c(C)cccc21 75153,C(C(C)N=c1[nH]c(=NCCOC2CC(F)(F)C2)[nH]c2cc[nH]c12)(C1CC1)OC 75154,n1(C(CC)C)ncc(C(=O)NC2C3CC(NC(c4cn(C)cc4C)=O)CC23)c1C 75155,C1(CC)(NC(c2ccc(C(C)C)nc2)=O)CCN(C(C2CCC2(F)F)=O)CC1 75156,C(=O)(CC(F)(F)C(F)F)NC1C(NC(Cc2c(C)nc(C3CC3)s2)=O)COC1 75157,C1(C(=O)NC(C)Cc2nc[nH]n2)(CNC(c2nonc2N)=O)CCCCC1 75158,C(=O)(CC(C(F)F)n1cccn1)N1CC(C)C(CNC(c2cnsn2)=O)C1 75159,n1(CCC(=O)NCC(CC)NC(c2cncc(C(C)C)c2)=O)nc(C)cc1C 75160,C(c1ccc(OC)c(F)c1)=CC(=O)NCc1cc(CC)cc(Br)c1 75161,N1(C(C(CC)CC2CCCCC2)=O)CC(C)(CNC(C2(O)CC2)=O)CC1(C)C 75162,C1(C(=O)NCC2CC(C(=O)OC)C2)CC12CCN(C(=O)C1=CCN(C)C1)C2 75163,N1(C(CCS(=O)(=O)NC)=O)CC(C)(C)OCC1CNC(C1CCC(C)=C(C)C1)=O 75164,C1(F)(C(=O)NCCNC(CC(C)OC)=O)CCS(=O)(=O)C1 75165,C1(CNC(C(C=C)O)=O)CCN(C(c2nc(OC)c(C)s2)=O)C1(C)C 75166,N1(CC)CC(C(N2CCCC2C(=O)NCCCCCCC2CC2)=O)CC1=O 75167,CCCC(C(C)(C)C)NC(C1CCN(C(=O)CN2CCOCC2)CCO1)=O 75168,N1(C(C)C)CC(C(=O)N(C)CC2(NC(C3CC(CF)C3)=O)CC2)CCC1=O 75169,C1(C(=O)NC2C(NC(C3CC4CCC3C4)=O)CCC2)CCC(F)(F)CC1 75170,c1(OC)ncc(Cl)cc1C(=O)NC1CN(C(C2(Cl)CC23CCC3)=O)CC1C 75171,N1(C(C(C=C)OC)=O)CC(O)CC1C(=O)NCCOC1CCOC1 75172,N1(C(c2ccoc2Cl)=O)CCCC1C1CCCCN1C(c1c[nH]nc1F)=O 75173,c1(C(N2CCC(OCCNC(C(C#N)CC3CC3)=O)C2)=O)c[nH]c(=S)cn1 75174,C=CCC(CC)C(=O)N1CC=C(CNC(c2cn(CC(=O)N(C)C)nn2)=O)CC1 75175,C(=O)(CC(c1ccccc1)SC)NC(=O)CC1CCCN1C(C1CC1C(=O)OC)=O 75176,c1(C(N2CCC(NC(C3N(C(C)=O)CCCC3)=O)(CF)C2)=O)cc(N)ccc1O 75177,c1(C(=O)NCC(C)N(C(=O)CCc2cncn2C)CC)cc(F)cnc1O 75178,Cc1cnc(C)c(NC(C2CC2c2ccccc2OC(F)F)=O)n1 75179,c1(CNC(C(CC=C)C)=O)ccc2c(c1)CN(C(=O)Cc1cc(COC)on1)C2 75180,C(=O)(CC1=NNC(=O)C1)NC1CCN(C(C(CC)C2CCOCC2)=O)CC1F 75181,C1(C(C(=O)NC(CC)C)N(CCCCO)C)C2CCOCC12 75182,N1(C(C=CCCC)=O)CC(O)CC1C(=O)NCC1(CC(C)C)CC1 75183,C(C(C)(C)S(C)(=O)=O)n1c(-c2cc[nH]n2)nc(C(C2CC2)OC)n1 75184,CC(C)(C#Cc1cn(Cc2ncccc2Br)nn1)NC(c1cnsc1Br)=O 75185,N1(C(c2c(OC)c[nH]n2)=O)CCN(C(c2ccc(F)cn2)=O)C(c2cn[nH]c2)C1 75186,C1(CC)(CC)CC(NC(=O)CCCCSC)CN1C(c1ccc(C)c(C)n1)=O 75187,c1(OC)nscc1CNC(=O)COCCNC(=O)Cc1ncoc1C 75188,C1(F)(CNC(C(CC(C)C)N(C)C)=O)CCCN(C(=O)OC(C)(C)C)CC1 75189,N1(C(c2cn(CC=C)nn2)=O)CCC(F)C(NC(c2cc(C3(C)CC3)n[nH]2)=O)C1 75190,c1(C(N2CCC(C(c3nn[nH]n3)C)CC2)=O)[nH]nc2c(=O)n(C)cnc12 75191,c1(OCC(N)=O)cccc(C(C)N(CC(c2ccncc2)O)CCO)c1 75192,c1(C(N2CC(CC(C)NC(c3cc(=O)n(C)cn3)=O)C2)=O)ccc(F)c(O)c1 75193,CCCCC(CNC(=O)CCCN(C)C(=O)OC)NC(C1C2COCC12)=O 75194,Cn1cc(C(C(=O)NCCC(C)(C)O)NC(=O)CNC(N)=O)nn1 75195,c1(NC)cc(Cl)ccc1C(N1CCCCCC1CNC(=O)CCCC(C)SC)=O 75196,N1(C(=O)CC2=CCCC2)CCOC2(CCN(Cc3cc4cnccc4[nH]3)CC2)C1 75197,CCC(CC)C(C)NC(C1OCCC1NC(=O)C(C)(C1(C)CC1)OC)=O 75198,Cn1ncc([N+](=O)[O-])c1C(=O)NC1CCCC(NC(=O)C=CCF)CC1 75199,c1(C(=O)NCCC(C(C)C)NC(c2c(CC)nc[nH]2)=O)cccc2oc(O)nc12 75200,c1(OCC(=O)NCC2CN(C(CCC(C)O)=O)CC2C)ccc(F)cc1Cl 75201,CCCC(O)C(=O)N1CCC(C2N(C(=O)C=CC3CC3)CC2(C)C)CC1 75202,C1(C(=O)NCc2scc(C(N(C(C3CCCO3)C)C)=O)c2)CCN(C)C1=O 75203,C1(C)(C(=O)NC(C2CCN(C(=O)C(C3CCCO3)C3CC3)C2)C)C=CCC1 75204,c1(CC)cc(C(N2CCOCC2CC(=O)NCc2cnc[nH]2)=O)ncn1 75205,C(C(C)C(C)C(=O)NCC1(NC(C2CCC(C)C2C)=O)CCOCC1)OC 75206,C1(NC(=O)CCN2CCCC2)CC2CC(NC(=O)Cc3ccc(Cl)s3)C2C1 75207,c1(C(N2CC(O)(CNC(c3cnc(CC)nc3C)=O)C2)=O)c(C)cc(C)nc1O 75208,Cc1cc(N)c(C(=O)NCCCC(C)NC(=O)CC2(C)CCCC2)cc1C 75209,O=C(C#CC1CC1)NCC12CC1CN(C(C1CC(=O)N(CC3CC3)C1)=O)C2 75210,N1(C(C2CC(CC)(CC)C2)=O)CC(CNCC2N(C(C)=O)CCC2)CC1(C)C 75211,c1(C(=O)NCC(C)N(C)C(c2ncncc2Cl)=O)c[nH]cc(Cl)c1=O 75212,CC1CC(=O)NCC1C(N1CCCC1(C)CNC(C1CC(O)C1)=O)=O 75213,Cc1cnoc1C(C)NCC(N1CCOCC1)CNC(=O)OC(C)(C)C 75214,C#CCC(C)(CC)C(=O)NC1C2CC3C1C3C2C(=O)NCC#CCOC 75215,CCCCCCCCC(=O)N(C1CCCN(C(=O)CC2CCCCC2O)C1)C 75216,CCCC(CCC)=CC(=O)NC(C(=O)NCc1cc(C)on1)C1CCCO1 75217,C1(C(N2C(C)CCC2C(=O)Nc2ccc(F)nc2)=O)CC2CCCC2C1 75218,c1(C(=O)NCCCN(C(C(CC)OC)=O)C2CCCC2)ccc(C)n1C 75219,c1(COC)ccsc1C(=O)N(C1CCN(C(=O)CCC=C(C)C)C1)CCO 75220,C12(CC(=O)N(C3CC3)Cc3c(C)noc3)CCC1CNC2 75221,CC1(C)C(C)(C(=O)NCC2(O)CN(C(c3ccccc3CC#N)=O)C2)C1(C)C 75222,c1(C(=O)NC(CNC(CC2N(C(C)C)CCC2)=O)(C)C)ccc(C(N)=O)cn1 75223,C(C(=O)NNC(=O)C1=COCCO1)(c1cccc(Cl)c1)OC 75224,Cc1cc(C(=O)NCC2CCCC(NC(C34C=CC(CC3)C4)=O)C2)cn1C(C)C 75225,C(=O)(CC(C)(C(F)F)N(C)C)NC1CC(NC(c2c(C)cc(F)s2)=O)CC1O 75226,N1(C(CC(=O)NCC#C)=O)CCN(CCCNC(c2cnns2)=O)CC1 75227,c1(C(N2CC(N(C(C(C)CC3CC3)=O)C)C(O)C2)=O)cc(C(F)F)ccc1Cl 75228,c1(C(=O)NC2CCC(NC(CC3(C)CC3F)=O)CC2)cc(O)cc(Cl)c1Cl 75229,c1(N(CC)CC)ccc(CCC(=O)NCC(CC)NC(C2CCC2(C)C)=O)cc1 75230,CC(C(=O)N1CCN(C2CCN(c3cncc(Cl)n3)CC2)C(=O)C1)S(C)(=O)=O 75231,C1(C(=O)OCC)(NC(c2ccc(Nc3cccc(F)c3)cc2)=O)CCSCC1 75232,C1(F)(C(=O)NCc2cnc(CC)[nH]2)CCN(C(C2CC(=O)N(OC)C2)=O)CC1 75233,Cc1cc2[nH]c(C(=O)NC3CC4(CCN(C(=O)C(=O)NC5CC5)C4)C3)cc2o1 75234,N1(C(C2(CNC(C(C)NC(N)=O)=O)CCCCC2)=O)CC(O)C(O)C12CCC2 75235,C(C)(C)(CC(=O)NCc1ccoc1C(=O)NCCCC(O)CO)N(C)C 75236,c12cc(c(Br)cc1F)NC(=O)C2N(C(C)CS(C)(=O)=O)C1CC1.CCOC 75237,N1(C(C2C3(CCN(C(c4cnn(C5CC5)c4)=O)C3)C2)=O)CC2CCCC2C12CC2 75238,CC1CCN(C(c2ccc3c[nH]nc3c2)=O)C(C)C1NC(c1ccc(F)nc1)=O 75239,C1(NC(c2cc(C)nc(C)n2)=O)CC2CCC(C1)N2C(=O)C(O)c1cnc[nH]1 75240,c1(C(=O)NC2CCC(F)(CNC(C)=O)C2)ccc(Nc2ccncc2)cc1Cl 75241,c1(OC)cccc2[nH]c(CN3CC(C(N4CC(F)C(F)C4)=O)CC(F)C3)cc12 75242,C(=O)(C(F)(F)C(C)(C)O)N1C(C(=O)NC2(C#C)CC2)CC1C 75243,CCC(O)C(F)(F)C(=O)NCCCC1CCN(C(=O)CC(C)C(C)(C)C)CC1 75244,N1(C(CN(C(C(C)C)=O)C)=O)CCC2CN(C(=O)C(O)CC3CCOCC3)CC2C1 75245,Cc1cc(C)c(C(=O)NCCN(C(=O)CC2CC2C)C)c(C)c1 75246,N1(C(C(CC)=CC)=O)CCC(C)(C)C(C(=O)NCC(c2cccs2)O)C1 75247,C#Cc1ccc(NC(C2CCOCC2NC(C2CC3(CCC3)C2)=O)=O)cc1 75248,O=C(C1CCc2cccc(Cl)c21)NC1CCCN(C(C2CC(O)C2)=O)C1 75249,CN=c1nc(N2CCOc3cccc(Cl)c3C2)[nH]c(=NC(C)C2CCN(C)C2)[nH]1 75250,C1(NC(c2ccncc2F)=O)CC2CC1N(C(=O)Cc1cnn(C(F)F)c1)C2 75251,C1(C(=O)NC(CNC(C2C(COC)C2)=O)CO)Cc2cccc(OC(F)F)c2O1 75252,C(=O)(CCCC(F)(F)C(F)(F)F)N1C(CNC(C(CC=CC)CC)=O)CCC1 75253,c1(C(N2CCN(C(CCOCC#C)=O)C(COC)C2)=O)cnc2n1CCC(C)C2 75254,C1(C)(C(=O)OC)COCCN1C(c1nn(C)cc1Cl)C(=O)NCC(F)F 75255,Cc1ccc(C(=O)NCC2(NC(C3CCCCN3C)=O)CCCCC2C)c(N)c1 75256,N1(Cc2scc(C#N)c2)CCc2cccc(C(N3CCNC(=O)CC3)=O)c2C1 75257,C1(C)(COC)CCN1C(=O)CCC1CC(NC(=O)CC2(C)OCCO2)C1 75258,C1(C(N2CCC(C(C)NC(c3cscn3)=O)C2)=O)CC1C1CC1C 75259,N1(C(c2ccccc2Cl)C(=O)NCC)CCn2c(CC)nnc2C1 75260,Cc1ccc(Cl)cc1-c1cn(C2CN(C(c3csc(CC(C)C)n3)=O)C2)nn1 75261,CC1(C)CCCCC1C(=O)NC1C=CC(C(=O)NCC2CC(O)C(O)C2)C1 75262,N1(C(c2cc(C)on2)=O)CCC(F)(C(=O)NC(C2CCCOC2)(C)C)CC1 75263,N1(C(C(N2CCOCC2)C)=O)CC(NC(c2sc(Cl)cc2Cl)=O)CC1(C)C 75264,N1(C(C2(S(N)(=O)=O)CC2)=O)CCC2(C1)CN(C(=O)CC1COC3(CCC3)CO1)C2 75265,C1(CC(=O)NCCN(C(c2cscc2Br)=O)CC)CC(C)(C)OC1=O 75266,C(C(C)(C)CC(=O)NCC(C1CC1)NC(C1CC(C)(C)CO1)=O)N(C)C 75267,c1(C(=O)NCC2CC(NC(C34CCC(CC3)OC4)=O)C2)cc2cc(Cl)ccc2o1 75268,C1(O)(CNC(C2(COC)CC2)=O)CCN(C(=O)Cc2ccc(O)cc2Cl)CC1 75269,N1(C(CN(C)C(N)=O)=O)CCCC2CN(C(=O)CCc3cnn(C)c3)CCCC12 75270,c1(C(N2CC(CNC(C=CCCC)=O)N3CCC2C3)=O)cc2nccc(Cl)c2s1 75271,C1(C(=O)NCC(CCC)C)CCC2(CC2)N1C(c1cc(C)c[nH]1)=O 75272,c1(CC)ncccc1C(N1CCCC1C(C)NC(c1ccnnc1)=O)=O 75273,N1(C(C)=O)CCc2cccc(C(=O)NC3(CO)CCS(=O)(=O)CC3)c21 75274,C1(C(=O)NCc2ccsn2)CN(C(=O)C(c2cccc(Br)c2)O)CCC1(F)F 75275,CC1CC(N(C(=O)CCC2CCCN2C(=O)C(C)C2(O)CCC2)C)CCO1 75276,CCCCC(O)CC(=O)NCC1(O)CC(NC(=O)COc2ccc(C)cc2)C1 75277,C1(C)(C(=O)NC(CCC=C(C)C)C)CCN(C(=O)Cn2cnccc2=O)CC1 75278,c1(C(=O)NC2CC3(CN(C(CCCCC)=O)C3)C2)c(Cl)ccc(OC)c1N 75279,Cc1cc(=NCC(CC2CC2)C(C)C)[nH]c(=NCC(C)Cc2cn[nH]c2)[nH]1 75280,N1(C(C(C(CC)C)O)=O)CCCC2(C1)CN(C(=O)C1=NNC(C(F)(F)F)C1)C2 75281,C1(C(=O)NCC(C)N(C(=O)CCC(=O)c2ccc(Cl)cc2)C)CCC2CCC1O2 75282,C1(C(N(C)CC2(c3ccccc3)CCCC2)=O)CC(=O)C12CC2 75283,N1(C(C2(F)CCN(C(c3cnc(N(C)C)o3)=O)C2)=O)C2CCC1COC2 75284,Cc1cc(NC2CCC(CNC(c3cc(Cl)nc(Cl)c3)=O)C2)nc(C2CC2)n1 75285,C1(CNC(C=C(C)C2CC2)=O)(CNC(=O)C(C)NC(=O)Cn2cnnn2)CCCC1 75286,C1(CNC(c2cnc(C)s2)=O)CCN(C(=O)CC2CC(CF)C2)C1(C)C 75287,c1(C(N(CCC)CC)=O)ccc(CO)cc1.C(C)(C)(C)N 75288,C12(C(N3CC(CNC(CC4N(C)CCC4)=O)CC3(C)C)=O)CCC3CC1C2C3(F)F 75289,N1(C(C(CC(C)C)F)=O)CC(CO)C2(CCN(C(c3ccccc3F)=O)CC2)C1 75290,C1(CC(=O)N(CCNC(C(COCC)C)=O)C(C)C)COC2(CCC2)CO1 75291,C1(C(N(C)Cc2ccoc2)=O)CNC(C)(C)C1 75292,CC1CC(NC(=O)NCc2ncccc2C2CC2)CN(C(=O)OC(C)(C)C)C1 75293,c1(C(C)C)cc(NC(=O)C(N2CCCC2C(c2ccccc2)C#N)=O)n(C)n1 75294,N1(C(c2nc(CNC(c3occ(C(N)=O)c3)=O)oc2)=O)CC(O)CC12CCC2 75295,N1(C(C(CC)n2ccnc2)=O)CCC2OCCN(C(c3nc(=O)n(C)[nH]3)=O)C2C1 75296,CC1(NC(=O)CC2CC(=O)NC2=O)CCCCC1C(=O)NC1(CC2CC2)CCC1 75297,c1(OC)cc(C)c(CNc2cc(C(=O)N=c3cc(Br)[nH][nH]3)n(C)c2)c(O)c1 75298,c1(C(N2CC(NC(C3(F)CCOCC3)=O)C(F)C2)=O)ccc(Br)c(Cl)c1Cl 75299,C1(S(C)(=O)=O)(C(=O)NCC2CCCN(C(CN(C)C)=O)C2)COC(=O)C1 75300,Cn1ncc(=NC(=O)C2CN(Cc3ccc4nccn4c3)CCC2O)[nH]1 75301,N1(C(c2n[nH]c(CC)c2C)=O)CCOCC(C(=O)NCC(C)C(=O)OC(C)C)C1 75302,C12(CNC(c3cn(CCOC)nc3)=O)CC1CN(C(c1ccn(CCF)n1)=O)C2 75303,C(=O)(CCC(C)(F)F)NC1(C)CC(NC(CN(C2CCC(=O)NC2)C)=O)C1 75304,C(CCOCCO)(C(=O)C1CC1)NC(c1c(CC)ocn1)=O.c1(NC)c[nH]nc1C 75305,CC1=C(C(=O)NC2CC(C(F)C(=O)N(C)CCOCCOC(C)=O)C2)CCC1 75306,Cc1ccn(CC(N2CC(CNC(c3c(C)nsc3N)=O)CC2C)=O)c(=O)c1 75307,C1(NC(C(CSCC(C(=O)OC)OC)C)=O)CC2C=CCC(C1)C2 75308,C1(C(=O)OCC(=O)NC2(CC(C)C)COC2)CC(=O)N(Cc2ccccc2)C1 75309,c1(C(=O)NC2CC3(C2)CC(C(N2CCc4n[nH]cc4C2)=O)C3)ccc2ncsc2c1 75310,Cc1c(F)ccc(Cl)c1C(N1CC2CC(NC(=O)CC3OCCO3)C2C1)=O 75311,Cc1c(CC(=O)N(C)CCN(C)C(c2cn(C)c(C)n2)=O)cccc1Br 75312,N1(C(C2(C)CC(C3CC3)=NO2)=O)CCC2(CC1)CN(C(c1cccnc1S)=O)C2 75313,N#Cc1ccc(OCc2cccc(NCc3c(Cl)c(Br)cn3C)c2)cc1Br 75314,C1(C(=O)NCc2cc(C(=O)NCC3(COC)CCCC3)n[nH]2)CCC(O)CN1C 75315,C(=O)(CC(C)C1CC1)NCCCCN(C(C1(CC)CCC1)=O)C 75316,C(=O)(C(=O)N=S(C)(C)=O)NCCC1(CNC(C(C)CC2CC2)=O)CC1 75317,Cn1nc(O)cc1C(=O)NCC(c1ccccc1)NC(c1nnsc1N)=O 75318,C12(NC(CCc3n(C)ccc3)=O)CCC(CC1)N(C(C1CC=CCC1)=O)C2 75319,CCCC(CC)C(=O)N1CC(F)CC1CNC(c1cc(N2CCCC2)cc(Cl)c1)=O 75320,N1(C(C2CC(CCC)C2)=O)CCC(C(C)NC(c2ncn(C)n2)=O)CC1 75321,c1(CNC(C(C)N(C)C(C2(C#N)CCCO2)=O)=O)ccccc1CO 75322,C#CC1CN(C(=O)C(C2CCCO2)NC(=O)CCN2CCOCC2)CCO1 75323,c1(SCC(=O)NC(CC2CN(C(CCC=C(C)C)=O)C2)C)nc2ccccc2[nH]1 75324,N1(C(C(C)OCCOC)=O)CCC2(CCCN(C(=O)CCCC3CC3)C2)CC1 75325,n1(CC(=O)NCC2CCN(C(CC(=O)N(C)C)=O)C2(C)C)cc2ncccc2n1 75326,Cc1cc(NC(C2CN(C(C3CCCS3)=O)CCS2)=O)nc(C)n1 75327,C1(C)(C(N(CC(C)(CO)CO)C)=O)CCCN(C(=O)CCOC2CCC2)C1 75328,c1(NC(C2CCC(NCc3cnn(CCC)c3C)CO2)=O)cc(F)c(Cl)cc1F 75329,c1(NC(C(C)(C)C2CCN(C(=O)CC3(C)CCC3)C2)=O)ccc2nccn2c1 75330,C(C)(C(=O)NCCC1(C(=O)N(CC(C)O)CCOC)CCC1)OCC(C)C 75331,C1(NC(C(C2CC2)OCC)=O)CN(C(=O)Cc2ccc3c(c2)CC3)CCC1(F)F 75332,C1(C(=O)NC2(C(N)=O)C(C)(C)C2)CCC=CC1NC(c1cnncc1O)=O 75333,c1(N2CCN(Cc3onc(C(C)OCC)n3)CC2)ncc(C(N)=O)cc1Cl 75334,N1(C(C=CCC(C)(C)NC(c2ccc(C#N)[nH]2)=O)=O)CCC(F)(F)C(O)C1 75335,C(CNC(=O)C=CC(=O)N(C)C)(CO)NC(C=CC(C)C)=O 75336,C1(NC(c2n(C)ncc2)=O)CN(C(c2cnccc2Cl)=O)C2(CCCC2)C1 75337,C1(CNC(c2cnc(C(C)=O)s2)=O)CC2CCC(C1)N2C(c1csc(Cl)c1)=O 75338,C1(CNC(C2(CC)COC2)=O)CN(C)CCN1C(C1CCC(=O)N1C)=O 75339,C1(O)(C(C)C)CCCN(C(=O)C(C2CCC2)NC(c2ccn(C)n2)=O)C1 75340,C(=O)(C1CCCn2cc(C)nc21)N(CC(CC)NC(=O)CCC(C)(C)[N+](=O)[O-])C 75341,Cc1cnc(NC(C2CC2C(=O)Nc2cccc(I)n2)=O)c(C)c1 75342,C1(N(C)C)Cc2ccccc2N(C(c2ccnc(Cl)c2N)=O)C1 75343,C1(C)(N(C(CCC2CCC(C)O2)=O)CC2(OC)CCCOC2)CCCCC1C(=O)O 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75519,c1(OC)cncc(C(N2CCC(C(N3CCC(F)(CO)C3)=O)(OC)C2)=O)c1 75520,Cc1nc(C(=O)NC2CCN(C(=O)CC3NC(=O)NC3=O)C2)ccc1[N+](=O)[O-] 75521,N1(C(C2(C#C)CC2)=O)CCCN(C(=O)C(C)C(C)C)C(C(C)C)C1 75522,Nc1cc(Cl)nc(C(=O)NCC2CC2CNC(c2cnn3c2CCC3)=O)c1Cl 75523,c1(COC)cc[nH]c1C(=O)NC(CN(C(=O)CC1(C)CC1(Cl)Cl)CC)CC 75524,CC1(NC(C2(CO)CCCO2)=O)CN(C(c2cn(C3COCC3F)nn2)=O)C1 75525,Cc1cc2ccc(C(=O)NC3CC(C)CN(C(c4sc(C)nc4C)=O)C3)cn2c1 75526,c1(C(=O)NCC2(CN(C(=O)C=C3CCCC3)C)CC2)cnc2ncccc2c1 75527,N1(C(C(C)(CO)NC(C2C(C=C)OCC2)=O)=O)Cc2ncsc2C1 75528,C1(OC)CN(C(c2nc(Cc3ccc(C)cc3)oc2C)=O)CC1C(=O)O 75529,N1(C(CC(C)(C)F)=O)CCCC(O)(CNC(c2ccc(C(C)(F)F)cc2)=O)CC1 75530,C123CCCC1(F)CN(C2)C3=O.C1(CC(=O)NC)CCCN1C(=O)Cn1cncn1 75531,N1(C(CCn2cc(C(C)=O)nn2)=O)CCCC(n2cc(C(C)N(C)C)nn2)C1 75532,CN1CCN(CCc2nc(-c3cc[nH]n3)n(CC3CCCC3(F)F)n2)CC1 75533,Cc1cccc(NNC(=O)C2(n3cc(CN4CCCCC4)nn3)CC2)c1Br 75534,c1(C(=O)NC2(C3N(C(C(C)OCC)=O)CCC3)CC2)ccc(CC)c(O)c1 75535,n1(CC(C)NC(C2C(F)(C(=O)OCC)C2)=O)cc(CCCn2cc(C)cn2)nn1 75536,N1(C(CC(C)F)=O)CCC(C)(CNC(c2c[nH]nc2F)=O)CC1 75537,C1(N(C(=O)CS(C)(=O)=O)C)CN(C(=O)C(=O)NCC(F)(F)F)CC12CC2 75538,N1(C(C=CCC)=O)CC2CC1CCC2NC(=O)Cc1ncc(C)s1 75539,N1(C(C2(COC)CCCCC2)=O)CC(C2CCCN(C(=O)C(C)S(N)(=O)=O)C2)C1 75540,C1(C(=O)NC2CCCN(C(C(CC)(C)C)=O)C2)(CF)CC2(CCC2)C1 75541,c1(C(=O)NC(CNC(=O)C(F)=CCCF)C2CC2)ccn(-c2ccncc2)n1 75542,C(=O)(CCC(C)NC(c1nscc1C)=O)NC(C1C(C(=O)OC)C1)C 75543,c1(N(C(CNC(C(C)CC(N)=O)=O)C)C)nc2c(cc1C#N)CCC2(C)C 75544,N1(C(CCC(C)OCC)=O)CC(NC(c2cc(OC)n[nH]2)=O)CC(C)C1 75545,CC1CCC(C)(C)N1C(=O)CC1CC(N(C(=O)CC2(CO)CCC2)C2CC2)C1 75546,C(=O)(CC1=NNC(=O)C1)NC1C(CNC(C(C)CC2CCC2)=O)CC1 75547,N1(C(C2C(C)CC2)=O)CCOC(C(N2CCCC2C(N)=O)=O)C1 75548,CC(C)CC(CNC(c1cccc(C(C)C)c1)=O)NC(c1cccnc1)=O 75549,CC(C)CCN=C(NCc1ccc(N(C)C)cc1)NC1CC(=C2CCC2)C1 75550,c1(C(N2CC3(CCN(C(C(C)OCCOC)=O)C3)C2)=O)nc2nccc(C)n2n1 75551,C(CN=c1[nH]c2c(c(=NCc3conc3C3CC3)[nH]1)CCCC2)c1nc(C)[nH]n1 75552,c1(OCC)cc(-c2cccnc2)nc(N2CCCCC2CC(=O)OC)n1 75553,Cc1cc(=NCC(CC(C)C)NC(=O)CSS(C)(=O)=O)[nH]c(Cl)n1 75554,C1(CNC(c2oc(CC)c(C)c2)=O)COC(C)(C)CN1C(=O)CN1CCCC1=O 75555,N1(C(C(=O)NC2C(C)(C)CN(S(C)(=O)=O)C2)=O)CCC23CCCCC2(C1)C3(F)F 75556,c1(C(=O)NC2C(O)(COC)COCC2)ccc(S(=O)(=O)CC)cc1 75557,C1(C(=O)NC(C)CCN(C)C(c2cnsc2)=O)C2CC2CN1C(=O)OC(C)(C)C 75558,C1(NC(c2n(OC)cnc2C)=O)CCC12CCN(C(=O)CNc1cccs1)CC2 75559,CC(CS(C)(=O)=O)C(=O)N1CCC(Cn2cc(CN3CCOCC3)nn2)C1 75560,C1(CNC(c2ccc(F)o2)=O)CN(C(c2ccoc2Cl)=O)C2CCCCC12 75561,Nc1cc(C(=O)NCC23CC(NC(=O)C(O)CN4CCCC4)(CO2)C3)ccc1F 75562,C(=O)(CC(C)C(C)(C)C)N1CC(O)(CN(C(C(n2cnc(C#N)n2)CC)=O)C)C1 75563,CC1CN(C(=O)C(C)CN(C)C(c2cnsn2)=O)CC(C)(C)C1 75564,C1(NC(CN(C2CC2)CC)=O)CC2(C1)CN(C(=O)Cc1ccc(Br)cc1)C2 75565,c1(C(=O)NCC2N(C(c3cccc(C)c3C)=O)CC(O)C2)cc2c[nH]cnc-2n1 75566,Cc1cccc(CNC(=O)CCCCN(C(C2C=CCCC2)=O)C2CC2)c1 75567,C(=O)(CC(O)CC(C)C)NC(CCCC(=O)Nc1ccc(CCC)nc1)C 75568,c1(CNC(c2nc(C(=O)O)sc2)=O)cc(I)ccc1F 75569,C12(NC(C(CC)NC(C)=O)=O)CC(C1)N(C(=O)Cc1ccns1)C2 75570,C1(C(=O)NCC(C)NC(=O)NC)C=CC(NC(C2CCSC2)=O)C1 75571,C(c1ccc(Br)o1)=C(C)C(=O)NCC(O)CNC(=O)C(C)(C)n1cccn1 75572,N1(C(C2=CCCCC2C)=O)CCN(C(=O)CCc2cncnc2)C2(CCC2)C1 75573,Nc1nc(C(=O)NCC2CC2CNC(c2cc(Cl)ns2)=O)ccc1[N+](=O)[O-] 75574,FC1CCCC(N=c2nc(-c3ccccc3)[nH]s2)C1 75575,Cc1nnc2n1C(C(=O)NC1(CCNC(=O)Cc3ccc(F)c(F)c3)CC1)CC2 75576,Brc1cccc(CCNCc2ccn(C3CCC3)n2)n1 75577,Cc1ccc(C(=O)N(C)CC2CCCC2NC(=O)C(Cl)=CCl)cc1C 75578,c1(OC)cc(=O)n(C)cc1C(N1CCC2CN(C(=O)C3=NOCC3)CC12)=O 75579,C1(NC(=O)CC2CC(F)(F)C2)CC2CC1CN(C(c1cccc(CO)c1)=O)C2 75580,N1(C(CC2N(C)CCCC2)=O)CC2CCCC1C2CNC(=O)CCCC1CCC1 75581,N1(C(COCCN(C)C)=O)CCC(CO)C(NC(=O)CCc2ncc(F)cn2)C1 75582,C1(C(N2CCC(C(C)NC(=O)C(C)(F)F)C2)=O)CC2(COC(=O)N2)C1 75583,C1(C(=O)NCC(C)(C2CC2)NC(C(n2ccc(C3CC3)n2)C)=O)CCCC1(F)F 75584,c1(CO)ncnc2c1CCCC2.C12CC3CC1N(C3)C(=O)c1ccc(o1)C(=O)N2 75585,CCCC(C)(C)CC(=O)N(C1CC2CC1N(C(=O)Cc1cc(F)cc(Cl)c1)C2)C 75586,N1(C(C2CC(CCC)C2)=O)CC(NC(=O)Cc2ccc(F)cc2Cl)CCC1C 75587,N(C1CCc2ccccc21)C(CC(C)CNC(c1nsnc1O)=O)=O 75588,C1(C(=O)NC(CNC(c2cnc(COC)s2)=O)(C)CO)CCc2n[nH]c(C)c2C1 75589,CS(=O)(=O)C1CC(CNC(=O)C(N)C2CSC2)C1 75590,c1(C(C)C)cccc(F)c1C(=O)NCCC(C)NC(c1cnc(Cl)[nH]1)=O 75591,C1(CNC(C2C(C)CCC2)=O)(NC(C2CCC=CCC2)=O)CCOCC1 75592,c1(C(=O)NCCCCCN=[N+]=[N-])coc2c1CN(C(=O)COCC1CC1)C2 75593,c1(N2CCC(C(C)O)CC2)nc(N2CCC(N3CC=CC3)CC2)c2c(n1)CCS2 75594,C(=O)(C(C)(C)COC(C12CC(Cl)(CO1)C2)=O)NCC 75595,C1(NC(c2cnn(CCN(C)C)c2)=O)CCCN(C(C2(CF)CC2)=O)CC1 75596,C1(CC(=O)NCCC2N(C(CCC(=O)N(C)C)=O)CCCC2)CCCCC(=O)N1 75597,N1(C(C2CCCN(C)C2)=O)CCC2(C=C(C(=O)NC(c3cscn3)CO)C2)C1 75598,Cc1c(C(=O)N(CCOC2CC(F)(F)C2)C)cc(Br)cc1C(F)(F)F 75599,N1(C(CC2N(CC)CCC2)=O)CCN(C(c2nnsc2C)=O)CC1C(C)C 75600,CC(CN=c1[nH]c2c(c(=NCCc3cc(Br)no3)[nH]1)CCC2)c1ccc(Br)cc1 75601,c1(CS(=O)(=O)NC)ccc(Cl)c(OC)c1F.C12CCC(C)N(C1)C2=O 75602,c1(CCC(=O)NC(C)(CNC(=O)C=Cc2cn[nH]c2)CO)cccc(O)n1 75603,Cc1sc(Cl)nc1C(N1CCC(O)(CNC(C2C3CCOCC23)=O)C1)=O 75604,C(CN=c1ncc(F)c[nH]1)NC(c1cccnc1C(F)(F)F)=O 75605,c1(-c2nc(C(C)Sc3ccc([N+](=O)[O-])cc3)on2)ccnc2ncnn12 75606,Cc1cncc([N+](=O)[O-])c1N1CCC2(CC(NC(=O)COc3ccon3)C2)C1 75607,CC(C)C(O)CC(=O)NCC1CCN(CCOc2c(Cl)cccc2Cl)CC1 75608,C12(C3CCN3)CCCN1C2=O.C(CCC)(CCC)C1CCC2(COCC)C1C2 75609,c1(N2CCCC(C3N(C(CS(C)(=O)=O)=O)CCCC3)C2)ncnc2[nH]cnc12 75610,C(N=C(NCC(C)(C)C)NC1CCOc2ccc(Cl)cc21)c1c(OC)nccc1 75611,C1(NC(c2cnc(CC(C)C)[nH]2)=O)CCCC12CN(C(c1cc(Cl)ccn1)=O)C2 75612,C12(NC(C(C)S(N)(=O)=O)=O)CCCN(C(c3cc(CC4CC4)on3)=O)CC1C2 75613,C1(C(N2CC(NC(c3ccc(OC)cc3)=O)C(C)(C)C2)=O)CCCCCS1(=O)=O 75614,N1(C(c2n(C(C)C)ccn2)=O)CCN(C(=O)CC2CCC(C)(C)CO2)C(C)C1 75615,N1(Cc2c(OC)nccc2)C2CCC1CC(NC(=O)C=Cc1ccoc1)C2 75616,c1(C(N(CCN(C(=O)CC(C)C2CCCO2)C(C)C)C)=O)nc2cnccc2s1 75617,c1(C(N(C)CC2N(C(C3CN(CC)C(=O)C3)=O)CCC2)=O)ccc(Cl)nc1OC 75618,C1(C(N(C)CC=CC(N2CC(N(C)CCO)C2)=O)=O)CC(=O)C12CCC2 75619,C(=O)(C1SCCc2sccc21)N(CC(C)(C)CNC(=O)CCc1nccs1)C 75620,c1(C(N2CCN(C(C(CC)SC)=O)CC2)=O)ccc2nc[nH]c2c1 75621,C1(C)(CNC(CC(C)CN(C)C)=O)CN(C(=O)CSc2ccccc2F)CCO1 75622,C=CCCCCC(=O)N1CC(CCNC(=O)CN2CCC(C)C2)C1 75623,C1(NC(CCCSC)=O)CC2CC(C1)CN(C(=O)C(c1ccc(C)nc1)(F)F)C2 75624,c1(CN2C(C(C(=O)OC)C)CCC2)ccc2ncsc2c1 75625,C(=O)(CC(C)C(=O)NC1CN(C(=O)C(C)(C)c2ccno2)CC1(C)C)OC 75626,C1(C(=O)NCCCOCCNC(C2C(C(C)(F)F)C2)=O)CCCNC1=O 75627,c1(N2CCC(CCC)(CO)C2)ccc(Br)c(S(=O)(=O)NC(C)C(C2CC2)OC)n1 75628,C1(C)(C(N2C(C3(NC(C4C(C=C)C4)=O)CC3)CCCC2)=O)CCN(C)C1=O 75629,N1(C(C(C(C)C)O)=O)CCN(C(C2CCC(O)CN2C)=O)C(CCO)C1 75630,c1(C(=O)NC2CN(Cc3cnc(Cl)cn3)CCC2(F)F)cc2ccc(Br)cc2s1 75631,C(N=c1[nH]c(N2CC=C(C)CC2)nc2c1CCCCC2)c1c(OC)c(Cl)ccc1 75632,C(C)(C)(CCN=c1[nH]c(N(C)Cc2nccn2C(C)C)nc2c1SCC2)OC 75633,C1(F)(CNC(=O)CCc2ccncc2)CCC(CO)C1.C12CC1C(=O)NC2C 75634,N1(C(c2c(OC)nccc2)=O)CCC2CN(C(=O)COC3CCCC3)C2C1 75635,C1(Cn2cc(C3CCCN(C(c4c(C)ccs4)=O)C3)nn2)CCCCC1(F)F 75636,N1(C(C(CSC)O)=O)CCCC(N(C(=O)C(F)=C2CCC2)C)C1 75637,c1(C(N2CC(O)(CNC(C(CSC)O)=O)C2)=O)ccc(Cl)cc1O 75638,C12(C(N3CC(C)N(C(c4c[nH]nc4S(N)(=O)=O)=O)CC3)=O)CCN(C1)S(=O)(=O)C2 75639,c1(C(=O)NCCC2CC(NC(=O)CC3=CCCC3)C2)c(F)cccc1[N+](=O)[O-] 75640,c1(C(=O)NCC(C)N(CC)CC)ccc(OC)nc1Br.C1C(=O)S1 75641,C(=O)(C(F)CC(C)(C)C)NCc1nn(C)c(C(N2CCC(C)(CC3CC3)C2)=O)c1 75642,N1(C(C(c2ccnn2C)NC(C(CC)O)=O)=O)CCCC(C2CC2)CC1 75643,C=C(C)CC(=O)NCCC(C)NC(C1CC(OC(F)(F)F)C1)=O 75644,C(CC(C)(C)C(=O)NC1CC(Cn2cc(CO)nn2)C1)NS(C)(=O)=O 75645,C1(C(=O)NCCCC(C)NC(C2CC(N(C)C)C2)=O)CCCCS1(=O)=O 75646,Cn1ncc2cc(C(=O)NCCC(O)CNC(C3(n4cncn4)CC3)=O)ccc12 75647,CCC(CC)CC(=O)NC(C)(CNC(=O)C(O)C(F)(F)c1ccccc1)CSC 75648,c1(CC)c(C(=O)NCC=CCNC(=O)C(c2cccc(F)c2)(C)C)ccn1C 75649,C(=O)(C1=CC2CCC(C1)C2)N1CCCN(C(C2C(C(C)(C)C)C(=O)C2)=O)CC1 75650,c1(CNCc2cccc(-c3c(C(=O)OC)ccnc3)c2)ccc(Br)cc1[N+](=O)[O-] 75651,C1(NC(Cn2cc(C(C)C)nn2)=O)CC(CNC(=O)Cn2ccnn2)C1(C)C 75652,C1(NC(C2CCCCO2)=O)CN(C(c2ccc(C(F)F)o2)=O)CC12CCC2 75653,CN1CCN(C(c2ccccc2C(C)(F)F)=O)C(CNC(c2ccccc2)=O)C1 75654,c1(NC(C(CC2CCC2)NC(c2cnc(OC)nc2)=O)=O)ccc(C#N)cc1O 75655,S(=O)(=O)(c1nc(N2CCC=C(Br)C2)ccc1Br)N1CCC(COCC)C1 75656,c1(CC(=O)N(C2CCN(C(c3[nH]c(=NC)sc3)=O)C2)C)ccc2c(c1)CCOC2 75657,c1(C(=O)NC23C(CN(C(C(CC)F)=O)C2)C3)c([N+](=O)[O-])cnn1CC 75658,c1(OC)nc(=NC(C)CCNC2CC2C(C)C)[nH]c2c(C)nn(C)c12 75659,CC(C)CC(CNC(=O)Cc1ccsc1)NC(C12CC(CC(F)F)(C1)C2)=O 75660,C(CN=c1nc(OC)c2nc[nH]c2[nH]1)C1CCN(Cc2c(CC)cncc2)C1 75661,c1(CCCC=C)ccc(C(=O)NC2(CF)CCN(C(=O)C(C)CCO)C2)cc1 75662,c1(C(N(CCC(C)NC(c2ccc(CCC)s2)=O)C)=O)ccn(C)c1C1CCC1 75663,C(=O)(C1=NN(CCO)C(=O)CC1)NC1CCN(C(C(CC#C)O)=O)C1CC 75664,C(=O)(C(C)(C)CF)NC1CCC(N(C(c2c(CC(C)C)onc2)=O)C)C1 75665,CCC(C)(CCC(C)C)C(=O)N1CCCC(NC(=O)C(F)F)C1 75666,N1(C(C2(C(C)=O)CC2)=O)CC(CNC(=O)Cn2cnc([N+](=O)[O-])c2)OC(C)(C)C1 75667,C(=O)(CCC(C)C)NCCn1c(SC(c2ccccc2)C(=O)OCC)nnc1 75668,c1(C(N(C)CC2OCCN(C(C=NOC)=O)C2)=O)cccc([N+](=O)[O-])c1NC 75669,C1(CC=C)(C(=O)NCC2(CC)CCCO2)CCCN1C(=O)C(C)CC#N 75670,c1(C(=O)NC(c2ccccc2Cl)C)nc2ccccn2c1-c1ccoc1 75671,Cc1cc(C(=O)NC2C3CC(NC(=O)C(C)(C)c4cnn(C)c4)CC23)nc(C)c1 75672,CC1Cc2ccc(F)cc2C1Nc1cc(I)ccc1F 75673,C1(NC(C(Cc2ccsc2)NC=O)=O)CCOC(CNC(c2cc(Cl)cs2)=O)C1 75674,N1(C(c2noc(C3CCC(OC(F)(F)F)C3)n2)=O)CCC(F)C(F)C1 75675,N1(C(c2c(OC)scc2)=O)CC(NC(=O)COC2CCC2)CCC1C 75676,C1(C(=O)Nc2cc(O)n[nH]2)CN(Cc2c(F)cncc2F)CCC1O 75677,c1(C(N2CCC(CNC(C3ON=C(CC)C3)=O)C2)=O)cccc2c1CCC(=O)N2 75678,S(=O)(=O)(c1cnc(NCCCOc2cncc(Cl)c2)cc1C)NCCC(=O)NC 75679,N1(C(C(CCN(C)C)O)=O)CC2CCN(C(=O)C3=C(C#N)CCC3)C2C1 75680,C(=O)(C(O)CC(C)C)NC1(CNC(=O)C(C)c2cc[nH]n2)CC(OC)C1 75681,c1(C(N2CCN(C(CC3(C=C)CC3)=O)CC2CCC)=O)ncn2c1COCC2 75682,c1(C(C)OC)noc(CS(=O)(=O)Sc2nncs2)n1 75683,C1(O)(C(C)NC(Cc2cnc(C)s2)=O)CCN(C(c2ccc(Cl)s2)=O)C1 75684,C(=O)(C1=CC2C=CC1C2)NC1COCCN(C(c2c(COC)nn[nH]2)=O)C1 75685,N1(C(C2ON=C(C)C2)=O)CC2(CCCC2NC(C2(c3ccccc3)CC2)=O)C1 75686,C1(CNC(CCC#C)=O)CC2CC1CN2C(c1ccnn1CCOC)=O 75687,Cc1ccc(C2CC2C(=O)NC2(C)CC(O)C2)c(Cl)n1.N12CCCC(C1)C2=O 75688,C(=O)(C(C)(O)CC(F)(F)F)NCC1OCCN(C(CCCCC(C)C)=O)C1 75689,C(=O)(C(C)(C)CC(C)(C)C)NCC1CN(C(CCn2c(C)csc2=O)=O)C1 75690,c1(C(N2CCC3(NC(c4cc(C)cc(F)c4)=O)C(C2)C3)=O)ccc2nc[nH]c2c1 75691,c1(C(CCN(CC(F)(F)F)CC)NC(=O)C(=O)NCC(C)OC)ccccc1 75692,Cn1cnc2c(C(N3CCC(CNC(C4CCC5CC45)=O)CC3)=O)[nH]nc2c1=O 75693,N1(C(C2CCC(CCC)CC2)=O)CCCC(CCNC(=O)CS(=O)(=O)CC)CC1 75694,Cc1c(N(C)CCN(c2ccccc2Cl)C)ncnc1N1CCCC1 75695,C1(C(=O)NCC2CCCC(OC)C2)N(C(c2n[nH]cc2C)=O)CCC1(C)C 75696,c1(C(=O)NC(CC)CNC(c2cc(CO)[nH]n2)=O)cnccc1C1OCCO1 75697,Cc1ccn(CC(=O)N(CCCCN(C(=O)CCN(C)CCO)C)C)n1 75698,N1(C(c2cc[nH]n2)=O)CC2CC1CCN2C(=O)C(O)CN1CCCC1 75699,c1(OCC)ncccc1C(=O)Nc1cccc(NC(C2CC(C)(F)C2)=O)c1 75700,Cc1ccc(-c2noc(C3CC4CC(=O)C3O4)n2)cc1Br 75701,c1(C(=O)NCC(C(C)C)NC(c2ccn(CC)n2)=O)nc2nc(C)ccn2n1 75702,Fc1ccc2c(c1)OCCN(c1ccnc(NCc3csnc3C3CC3)n1)C2 75703,Cc1cccc(C(C)(C)C(=O)NCCC(C)NC(=O)CCCc2ncco2)c1 75704,c1(C(=O)NCC2N(C(C(C)(C)OC)=O)CC2)cccnc1I 75705,C1(OC)CCCC1C(=O)N(CC(F)(F)COC)C 75706,c1(N(c2n(CC=C)c(-c3scnc3C)nn2)C)ccc(OCCCC)c(Cl)c1 75707,N1(C(C=CC)=O)CCN(C(=O)C=CC2CCC2)C2CCCCC12 75708,N1CC2CC1C2CNC(=O)CSc1ccccn1.c1(C2C(C)C2)ccccc1 75709,C1(C(N2CC(NC(=O)C(F)Cl)C(F)CC2)=O)CCc2ccccc2C1O 75710,C1(CNC(CN2CCCC(C)C2)C)COC2(CCCCC2)C1 75711,C1(CN(C(=O)CC2CCCSC2)C)CCN(C(c2nnsc2N)=O)CC1 75712,C1(C(=O)NCC(C(C)(C)C)OC)CCCCCCN1C(=O)C=C(C)c1ccco1 75713,c1(C(N(C)CC2CN(C(C3(C#N)CCCO3)=O)C2)=O)cc(Cl)c(C(F)F)cc1F 75714,c1(CC(=O)N(CC(C)(C)NC(=O)CC2CC2(Cl)Cl)C)ccccc1OC(F)F 75715,Cc1ccc(C(N2CCN(C(=O)C(C)Cc3ccccc3)CC2C)=O)cc1F 75716,c1(CCC(=O)NC(CC(C)NC(C(=O)NCC)=O)C)ccccc1CC(=O)OC 75717,N1(C(c2ccc(C)cc2O)=O)CC(F)(F)CC1(C)CNC(=O)C1=CCCS1 75718,Cc1ccccc1C(C)CC(=O)N1CC(NC(=O)C=Cc2csc(Br)c2)C1 75719,S(=O)(=O)(c1cncc(Br)c1)NC(C1C(C(N2CCN(CCC(C)C)CC2)=O)C1)=O 75720,c1(CC)cc(C(N2CC(CCn3cc(-c4ccc(Cl)s4)nn3)C2)=O)n[nH]1 75721,c1(NC(=O)Cc2ccns2)ncnc2c1CCC2.C12CCCCC1CNC2=O 75722,c1(C(=O)NCC23C(CN(C(CCNC(CC(C)C)=O)=O)C2)C3)cn(C)c(=O)n1C 75723,C1(CC(=O)N(CCN(C(=O)CC(C)n2cccc2)CC)CC)CCCC(F)(F)C1 75724,Cc1c(C(N2CC(C3(NC(=O)C=CCOCC(F)(F)F)CC3)C2)=O)cncc1Cl 75725,N1(C(CCSCC)=O)CCC2OCCN(C(c3cc(C)cc(O)c3)=O)C2C1 75726,Cc1ccc2cccc(NC(C3CCN(Cc4c(Br)cncc4Br)C3)=O)c2c1 75727,N1(C(CCCCNC(N)=O)=O)CC(C2CCCN(C(c3ccc(F)cn3)=O)C2)C1 75728,CC(CF)CC(=O)NCC1(NC(c2ccc(C(C)(C)C)s2)=O)CCC1 75729,Cc1nc(C)n(CCC(N2CCC(N(CCO)C(C3CC(C)(C)O3)=O)C2)=O)n1 75730,C1(NC(CCC(=O)NC)=O)CCCN(C(c2ncc(OC)cc2F)=O)C1C 75731,C1(C(N2CCC(NC(C3CN(C4CCOC4)C3)=O)(CO)C2)=O)CN2CCC1CC2 75732,C1(C(=O)NCC(c2ccncc2)(C)C)(OCC)CCN(C(=O)OC(C)(C)C)C1.CO 75733,C1(C(N2CC(C(C)C)OCC2)=O)CC(C)CN(C(=O)C(C)(C)CC#N)C1 75734,c1(C(=O)NC2C3CC4CN(C(CC)=O)C2C4C3)[nH]c2cc(Cl)cc(Cl)c2c1C 75735,N1(C(C2(SC)CCC2)=O)CCCN(C(C2CCN2S(C)(=O)=O)=O)C(C(C)C)C1 75736,N1(CCNC(c2cnc(Cl)s2)=O)CCCOC1=O.C12CCC1CNC2=O 75737,C#CCC(CC(=O)NCC1(CCO)CCCC1)NC(C1(C)C=CCCC1)=O 75738,Cc1n[nH]c2cnc(C(=O)NCC3(O)CCN(C(=O)C(F)CC4CC4)C3)cc12 75739,S(=O)(=O)(c1cc(C(F)(F)F)cc(Br)c1)Nc1ncc(-c2ccc(C)cc2)s1 75740,Cc1cc(Br)c(F)cc1C(N1CCC(CC(N2CCOCC2CCO)=O)C1)=O 75741,C1(CC)CN(C(=O)CC2CC3(CC3)CO2)CCC1NC(=O)CS(=O)(=O)NC 75742,c1(C(=O)NC(C)CCCNC(C2(O)CCSC2)=O)ccc(CCNC(N)=O)cc1 75743,Cc1ccc(C(=O)NCC(c2ccccc2)NC(=O)CC#N)cc1Br 75744,c1(OC)cc(C(=O)NCC2(C(N)=O)CN(C(=O)COCC3CCCOC3)C2)[nH]n1 75745,n1(C(CNC(C(c2ccccc2)N(C)CC)=O)C)cc(SCC)nn1 75746,CC1CCCC(N(C)C(c2ccc(CNC(=O)CCCC3CCC3)s2)=O)C1 75747,N1(C(c2cc(F)c[nH]2)=O)CC2(C1)CN(C(c1ccncn1)=O)C2 75748,N1(C(C(C)=CC2CC2)=O)CC(CNC(c2c(C)ncnc2C)=O)CC(C)(C)C1 75749,Cc1cnc(C(=O)NC2CCC(CC(=O)NC3(C(C)O)CC3)CC2)c[n+]1[O-] 75750,C=CC(C)(C)C(=O)NCCN(CCC)C(C1CC1Cl)=O 75751,c1(C(N(C(CCNC(c2nn(CC)c(=O)cc2)=O)C)C)=O)cc[nH]c2nccc1-2 75752,C1(NC(CCC2C(C)(C)C2)=O)CCC(NC(=O)CC2(CO)CC2)CC1 75753,C1(C(=O)NCC2N(C(C(C)OC3CCCC3)=O)CC2)CCCN1C 75754,c1(C(N2CCC(NC(CC=CCC)=O)C(F)C2)=O)c(C)cc(Br)cc1C 75755,c1(C(=O)NC(CC)CNC(C2(C)CCCC2)=O)ccc(C(=O)N(C)C(C)C)cc1 75756,Cc1cccc(-c2cn(CCCC(N3CCN(C)C4CCCC34)=O)nn2)c1C#N 75757,N1(C(C(C(C)C)SCC)=O)CC(C)(CNC(=O)COCCCF)CC1(C)C 75758,C1(C)(C(=O)NC2C(OC)CN(C(c3cc(C4CCC4)on3)=O)C2)CCCNC1=O 75759,N1(C(C2C(C)CC2)=O)CCN(C(C2CC(O)(c3ccccn3)C2)=O)CC1C(F)F 75760,C(=O)(CC(CNC(=O)CC1(C)CCOCC1)C1CCC1)NCCc1c(C)csc1 75761,CC1(NC(c2conc2-c2ccccc2)=O)CCN(C(c2csc(=N)[nH]2)=O)CC1 75762,S1(=O)(=O)c2ccc(cc2)N1.N1(C(C)C(=O)N(C)C)CC2(CCC2)C1c1ccsc1 75763,C(C(C(C)C(C)C)NC(c1cccnc1C(F)(F)F)=O)NC(CNC(C)=O)=O 75764,C1(C(=O)NCC2(CNC(c3cnoc3)=O)CC2)CCCN1c1ccccc1 75765,Cc1cc(C(=O)N(CCCCN(C(=O)CCOc2ccc(F)cc2)C)C)c(C)[nH]1 75766,CC(CCN(C)C(C1CCCO1)=O)NC(c1cnsc1)=O 75767,N1(C(c2c(C)cc(CC)o2)=O)CCCN(C(=O)C=Cc2cnccc2C)C(C)C1 75768,C1(C(=O)NC(C=C)C)CN(C(=O)CC(C)CCC)CC12CC2 75769,c1(SC)cc(C(=O)NCC(C)CNC(c2ccc(C(C)C)o2)=O)ccc1F 75770,c1(C(c2nnnn2C)NCc2cnc(C)s2)ccc(Cl)c(C(F)(F)F)c1 75771,Cc1n[nH]c(=NCC2CCN(C(=O)CCCOc3cccnc3)CC2C)o1 75772,C1(C(=O)NCc2c(C(=O)NCC3CCC=CO3)occ2)CC2(CCC2O)C1 75773,c1(C(=O)NCC(CC)NC(=O)CC2CCn3cncc3C2)cc(Cl)c(O)cc1C 75774,C1(O)(CCNC(CC2C(C)C2)=O)CCN(C(c2ccc(N)cn2)=O)CC1 75775,c1(NC(C(CCCCCO)N(C(C(C)C)CO)C)=O)ccc2c(c1)OCCO2 75776,C=C(Cl)C(C)(C)C(=O)N1CCCCC(NC(=O)C(C(C)C)NC(=O)COC)C1 75777,Cc1csc(C(=O)NCCn2ccc(C(=O)N(CC3=CCSC3)C)c2)c1 75778,N1(C(c2c(C)nn[nH]2)=O)CC(NC(C2CCCN2c2nccs2)=O)C2CC2C1 75779,c1(C(N(CC(CNC(c2nn(CC)c(C)c2)=O)C)C)=O)[nH]cc2c1CCS2(=O)=O 75780,c1(C(N2CCC(CC)C2CNC(C2CC2(C)CC)=O)=O)cc2cnn(C)c2s1 75781,C1(C(N(C(CC)C(=O)NCCCNC(C)=O)C)=O)CCC(C)(C)C1 75782,C1(NC(c2c(CC)nc[nH]2)=O)CC2CC1N(C(=O)CC(O)c1cnc(Cl)s1)C2 75783,c1(C(N(CC(C)NC(c2c(Cl)ccc(C)c2)=O)C)=O)cccc2cnnc(O)c12 75784,c1(-n2nc(C)c(C(C(=O)NC3CCC3)N(CCCF)C)c2)c(C)oc(C)c1C 75785,c1(C(=O)NCC(C)(C2CC2)NC(c2cc(CO)[nH]n2)=O)cc2n(n1)CCO2 75786,C(c1c(C)noc1C)=CC(=O)NCCC(CC)(C)NC(=O)CSC(F)F 75787,c1(C(N2C3C(NC(C(c4cnn(C)c4)C)=O)C(C3)C2)=O)cc(C)c(F)cc1F 75788,C1(CC(=O)NCCSC)CN(C(C2CC3C=CC2C3)=O)C(C)(C)C1 75789,c1(C(N2CCN(C(C3CC(C)C3)=O)C(C3CCC3)C2)=O)cnn2c1CN(C)CC2 75790,c1(C(N2CC(F)CC(NC(C(COCC)(C)C)=O)C2)=O)ccnc(S(N)(=O)=O)c1 75791,C(=O)(C(O)C1=CCCCC1)NCC1CCCN(C(C(C)(C2CC2)NC(C)=O)=O)C1 75792,c1(NC(=O)NC2CN(C3(n4ccc5cccnc45)CC3)C2)c(F)cc(I)cc1F 75793,N1(C(c2oc(CC)c(C)c2)=O)CCC2(CC1)CC2CNC(c1csnc1OC)=O 75794,N1(C(c2c(C)cc(C3CC3)nc2)=O)C2CCC1CN(C(C1CCCC(C)C1)=O)C2 75795,c1(NC(C(C(C)C)CNC(=O)C(C)(O)C2CCC2)=O)ccc2c(c1)COC2 75796,C1(N(C(c2cnc(C(C)C)[nH]2)=O)C)CCCCC1N(C(=O)CNc1nccs1)C 75797,C1(C(N(C2CCC2)CC)=O)CC(C)N1C(=O)CCc1cncnc1 75798,C1(CNC(Cn2c(C)ccn2)=O)CC(F)(F)CN1C(c1c[nH]cc1Br)=O 75799,C(c1cccc(F)c1F)=CC(N1CCC(CNC(CCCC=C)=O)C(C)C1)=O 75800,C(=O)(CCCCC(C)C)NCC1(F)CC(NC(c2cccc(CC)c2N)=O)C1 75801,c1(OC)cccc(C2CCCN2C(=O)Nc2nccn2C(c2ccccc2)C)c1 75802,c1(C(c2n(C(CC)C)nnn2)NCc2ncc(Br)s2)cc(C)c(OC)c(C)c1 75803,CC12CCC(C(=O)NCC3(O)CN(C(=O)CC4CCCC45CC5)C3)(CC1)C2 75804,C(CCC(C)C)(C(=O)NC1CC2CC2C(=O)C1)NC(C(C(CC)C)=O)=O 75805,CC1CC(NC(=O)Cc2cnoc2)CCN1C(C1OCCO1)=O 75806,CC(CNC(C1C(C)C1C)=O)C(=O)NC(C)C(C)F 75807,CCC(CC(=O)NC1CC1)N(C(=O)C(C)Oc1ccc(OC)cc1)C 75808,N1(C(C2C(C)N(C(=O)CN3CCC(F)CC3)CC2)=O)CC(=O)N(C)C(=O)C1 75809,c1(C(N2CC(C)C(NC(=O)COc3ccc(Cl)cn3)C2)=O)ccc2n[nH]cc2c1 75810,C(=O)(CCCC(C)(F)F)NC1(CNC(c2nn(C)c(=O)cc2)=O)CCOCC1 75811,c1(NC(C(c2ccccc2Br)NC(=O)OC(C)(C)C)=O)cc(Cl)nc(I)n1 75812,CC1(C)CC(CNC(c2cn3cnnc3cn2)=O)CN(C(=O)COC(C)(C)C)C1 75813,c1(C(=O)NCC(CCCC)NC(=O)CC2CSCCS2)cccc2scnc12 75814,c1(C(N2C(CNC(c3ncccc3F)=O)CCC2)=O)cc(F)c(F)cc1O 75815,N1(C(C(C)C2CC2)=O)CC(O)CC1C(=O)NC(c1ccccc1)C1CC1 75816,CC1CC(CNC(=O)CC2(C)CC2)CCN1C(C12CC(c3ccccc3)(C1)C2)=O 75817,CCC(C)C(O)C(C)C(=O)N(CCCn1cc(CSCCO)nn1)C 75818,c1(-n2c(C(CCSC)OC)nnn2)cccc(OCC(F)F)c1.c1(CN)ccncc1 75819,N1(C(CC(CCC)C)=O)CCC2(CC(NC(c3cncc(OC)c3C)=O)C2)C1 75820,C12(CN3CC(C(=O)NCC)OCC3)CCC(C1)C(C)O2 75821,c1(N(C(=O)COC2CN(C(C3C4CC5C(C4)C35)=O)C2)C)ccc2c(c1)OCO2 75822,C1(C(=O)NCCOCCCNC(C2C(C)C2)=O)COc2ccccc2O1.C1CO1 75823,N1(C(c2cncc(Br)c2)C(=O)NCC=C)CC(C)(C)c2ccccc21 75824,CC1C(NC(=O)CC2CC3(CC3)C2)CCCC1n1cc(-c2csnn2)nn1 75825,N1(C(C(CC(=C)Cl)NC(=O)CCC2CCC2)=O)CCNC(=O)CC1C 75826,c1(C(N2CC=CC(NC(c3c(C)onc3Br)=O)C2)=O)ccc(Cl)c(N)c1 75827,c1(NC(C2CN(S(=O)(=O)CCBr)CCO2)=O)c(F)cccc1I 75828,CC1C(C)N(C(c2ccc(N)c(Cl)c2O)=O)CCN1C(C1C2CCC1CC2)=O 75829,CC1=CCSC1C(=O)NCCC1CCCN1C(=O)CC1CNC(=O)O1 75830,C#Cc1cc(C(N2CC(NC(=O)C3=C(C)CCCC3)CC2(C)C)=O)cc(N)c1 75831,C1(NC(C(C(C)C)C2CCC2)=O)CC2CC1CC2C(N1CC(CO)C1)=O 75832,c1(-n2cc(CC(C)O)nn2)ccc(C(=O)NON2CCOCC2C2CC2)cc1F 75833,c1(OC)cc(C(=O)NCC2(O)CC(CNC(C3CC(OC)C3)=O)C2)cc(Cl)c1 75834,Cc1cc(Cl)c(C(=O)N(CC(O)CN(C)C(c2cnc(O)c(F)c2)=O)C)cc1F 75835,N1(C(=O)COC2CCCCC2)CC2CCN(C(c3c(F)ccc(O)c3F)=O)CC2C1 75836,C12(C(N3CC(NC(C4CN(C(=O)NCC)C4)=O)C3)=O)CCOC1CC(=O)NC2 75837,c1(C(C(=O)NCC(C)NC(=O)C=Cc2ccoc2)O)ccc(Cl)c(Br)c1 75838,C=CCCCCCN1CCN(C2CCCN(C(C3CCCC(O)C3)=O)C2)CC1 75839,c1(C(=O)NCC2N(C(COCCC)=O)CCN(C)C2)cc(Cl)c2c(c1)OCCO2 75840,c1(C(=O)NCC(C(C)C(C)C)NC(C(C)(C)SC)=O)ccc2c(c1)OCCCO2 75841,c1(CN(C)C)ccccc1CN1CCOCC1CNC(c1cc(Cl)c[nH]1)=O 75842,N1(C(CN(CC)CC)=O)CCCCC1C1CCCN1c1ncnc2c1cnn2C 75843,C(=O)(CC1=CCCCC1)NC1CC(CCNC(C(C)(F)c2ccon2)=O)C1 75844,CCCCC(CNC(=O)COCC1CCC1)NC(=O)CN1CCN(C2CC2)C1=O 75845,CC1CCc2[nH]c(=NCC(C)(C)CCCCO)[nH]c(=NC3CCN(C)CC3)c2C1 75846,C(CC(=O)N(C)CCNC(C12COCC1C2)=O)(C1=CCCC1)OCC 75847,N1(C(c2cc(C)[nH]n2)=O)CCC2(CC1)CC2NC(=O)C(C1CC(F)(F)C1)O 75848,Cn1cc(C(=O)NCC2(NC(=O)CC3CCC(C#N)C3)CCC2)c2ccccc12 75849,C1(C(=O)NCCN(C(c2cnc(C)cc2Cl)=O)CC)CCC2(CCOCC2)O1 75850,N1(C(C(C2CCOCC2)C)=O)CCC(C(C)CNC(C2(C)CS(=O)(=O)C2)=O)CC1 75851,c1(CC(N2CCN(C(C(C)OC3CCOCC3)=O)CC2)=O)c[nH]c2ccccc12 75852,N1(C(C(C(CC)O)C)=O)CCC2C(C1)NC(=O)CN2C(=O)CCCC1CC1 75853,C#Cc1ccc(C(N2CCOC(CN(C(=O)CC3CCCCC3)C)C2)=O)nc1 75854,c1(COC)ncc(C(=O)NC2(C)CC(NC(=O)C(C)(C)c3ccno3)C2)c(=N)[nH]1 75855,c1(C(c2nnnn2C(C)(C)C)NC(CCCC=C)C2CC2)cc(C)c(C)cc1C 75856,C(=O)(CCCC1CCNCC1)OCC(=O)NCC(C)C 75857,C1(NC(c2cnc[nH]2)=O)CC2CN(C(=O)CCc3ncc[nH]3)CCN2C1=O 75858,N1(C(CCCC(C)C)=O)CCCC2C(CCCN2C(c2ccnn2C2CC2)=O)C1 75859,C(=O)(CCC(C)N1CCOCC1)N1CC(C2CCCC2CNC(CCC=C)=O)C1 75860,c1(C(=O)NC2(C)CN(C(C3C(C)CC3)=O)C2)cc([N+](=O)[O-])ncc1Br 75861,C1(C)(CC)CC(NC(=O)CC2(N(C)C)CCC2)CN1C(=O)CCC(C)(C)OC 75862,Cn1ncc(C(=O)NCC2CC(CNC(=O)CCS(C)(=O)=O)CO2)c1C#N 75863,C(=O)(C(C)(C(C)C)NC(c1cc(Cl)cc(C(F)(F)F)n1)=O)OCC 75864,C1(CC(=O)N(C)CC2CCC(NC(c3cncs3)=O)CC2)CC2(CCC2)CO1 75865,N1(C(CCOc2c(C)cccc2)=O)CC2CC1CCN2C(C12CC(C1)C2)=O 75866,CCCS(=O)(=O)CC(=O)NCC1(CNC(C2CCCC2C)=O)CCCC1 75867,c1(NC(C2CCN(C(=O)CNS(=O)(=O)C3CC3)C2)=O)c[nH]c2cccnc12 75868,Cc1cc(C(=O)O)ccc1C(C)NCC1CCC(F)(F)C1O 75869,c1(OC)noc(C)c1C(=O)NC1CC(NC(=O)C=CC2CCCO2)C1 75870,N1(C(CS(=O)(=O)NC)=O)CCC(C)(C)C(NC(C2CNC(=O)C(C)(C)C2)=O)C1 75871,C(=O)(C#CC(C)C)NCC(CC)(C)NC(c1cscc1SC)=O 75872,C(=O)(C1=CCCCCC1)NC(C(C)NC(CCc1ccc(OC)cc1)=O)C 75873,C#Cc1ccc(C(=O)NC(C(=O)NOCC(C)(C)C(=O)OC)C2CC2)cc1 75874,C#CCC(CC(F)F)C(=O)NCC(C)(C)OCC(=O)NCC1(c2ccsc2)CC1 75875,c1(CSC)cc(C(=O)NC(C)CC2CN(C(=O)CCC3CCCCO3)C2)sc1C 75876,C12(CS(N3C(c4onc(C(C)(C)C)n4)CCCC3)(=O)=O)CCC(CC1)CC2 75877,C1(NC(=O)C=CC2CCC2)CCCCC1NC(C1C(F)(F)C12CC2)=O 75878,N#CC1(C(N2CCCC(NC(c3cccc4c3CCC4)=O)C2)=O)CC2(CCC2)C1 75879,c1(C(=O)NC2CCC(C)N(C(=O)CC3CCCCC3)C2)cc2cccnn2c1 75880,C1(OC)CCN(C(=O)CC(C(C)C)NC(C2CCCN2C2CC2)=O)CC1(C)C 75881,c1(CC(N2C(C)CC(NC(=O)Cc3cnc[nH]3)C2)=O)c[nH]c2ccc(F)cc12 75882,c1(C(=O)NCC2CN(C(C3COC(=O)O3)=O)C2)ccncc1Br 75883,Cn1cc(C(=O)NCC2(NC(C3CC4C=CC3C4)=O)CCC2)c(C2CCCO2)n1 75884,C12(CC)CN(C(c3cc(C)nc(O)c3)=O)C(CNC(=O)Cc3nonc3C)(C1)C2 75885,N1(C(C2ON=C(C)C2)=O)CCN(C(c2ncn3ccccc23)=O)C2(CCC2)C1 75886,c1(C(=O)NCC(CN(C)C(C2CCSCC2)=O)O)ccc2c(O)nnc(O)c2c1 75887,Cc1nccnc1C(=O)NC(CNC(=O)CC1CC(n2cnnc2)C1)C1CCC1 75888,C12(CC(N3C(CN(C(=O)Cc4cc[nH]c4)C)CCCC3)=O)CCCCC1C2(F)F 75889,CC(C)(C)CC(F)C(=O)NCC(=O)NCC(N1C(C)CCC1(C)C)=O 75890,C=Cn1nccc1C(N1CC(F)CC1CNC(c1ccccc1)=O)=O 75891,C(=O)(CCCS(=O)(=O)N1CCCC1)N1CC(N(C)C(c2cc(O)cs2)=O)C2C1C2 75892,CCC(C)(C)CC(=O)NCC1CC(NC(=O)Cc2cccnc2)C(O)C1 75893,C(C(COC)C(C)C)NC(c1c(C(C)NC(CN(CCOC)C)=O)noc1)=O 75894,n1(CC(=O)NC2C3(NC(CCCC)=O)CCC(C2)C3)nc(C)ccc1=O 75895,c1(CN2CC(NC(C(C)(C)O)=O)C(F)(F)CC2)c[nH]c2ccc(F)cc12 75896,N1(CCO)CC2CCC1C2.c1(C(C)C)ncc(C(=O)N(CCC=O)CCCO)o1 75897,CCCCC(O)C(C)C(=O)NC(CCC(=O)NCCn1cc(CO)nn1)C(C)C 75898,c1(C(=O)NCC2CN(C(CC(COC)(C)O)=O)C2)ccnc2c1CC(=O)N2 75899,C(CN=c1[nH]c2c(c(=NCCOc3ccncc3)[nH]1)CSC2)C1(C)CCCO1 75900,N1(C(c2c(C)n(C)nn2)=O)CCC2C(C1)CN2C(c1cc(C2CCC2)nn1C)=O 75901,C1(CC(=O)NCC2CCN(C(=O)CC3CCSC3)C2)CCCCC12CC2 75902,Cc1cc(O)ccc1C(=O)NC1CC(NC(=O)CSc2ccncc2)CC1O 75903,C(=O)(C1=CCCCC1C)N1CCN(C(CCCOCC=C)=O)CC1CC 75904,C(=O)(C(CCCC(=O)OC)N(C1CCOC(C)C1)CC1CC1)NCC=C 75905,c1(C(=O)NC2CN(C(C3CC3(Cl)Cl)=O)CC2C(F)F)cnc(O)c2ncccc12 75906,c1(C(=O)NCC(CC=C)NC(=O)CCCCOC)cc(O)cc(F)c1F 75907,N1(C(C(C)NC(CC)=O)=O)CC2(C1)CN(C(C13COC(CS(C)(=O)=O)(C1)C3)=O)C2 75908,N1(C(c2ccc(SC)o2)=O)CCC(F)(C(=O)NCC2(O)CSC2)CC1 75909,c1(CN(CCCN(C(CCC)CN2CCOCC2)C)C)ccc(C)c(C)c1 75910,[N-]=[N+]=NCCCC(=O)NCC1(C(N2CCC(N3CCC3)CC2)=O)CC12CCC2 75911,C1(CC(=O)NCC(c2ccccc2)CNC(=O)CC2CS(=O)(=O)C2)CCOC1=O 75912,C(=O)(C1CCC(=O)c2cccn21)N1CC(O)(CCNC(C2CCC(=O)NC2)=O)C1 75913,N1(C(C(=O)NCC2CC2)=O)CC2(CCCN(C(C34CCCN3CC(O)C4)=O)C2)C1 75914,C#Cc1ccc(OCC(N2CC(NC(c3cnc(C)cc3C)=O)CC2C)=O)cc1 75915,c1(C(N2CCC(NC(c3cn(CC=C)nc3)=O)CC2C)=O)cccn2ccnc12 75916,c1(C(=O)NC2CCC(CNC(c3c(C)oc(Cl)n3)=O)C2)cc(O)cc([N+](=O)[O-])c1 75917,c1(NCC(=O)N(CCNC(C)=O)C)cc([N+](=O)[O-])c(F)cc1SCCCF 75918,C(CCCCCCn1cc(COCCCO)nn1)NC(CCC1CCCN(C)C1)=O 75919,N(C(=NCC1CCN(S(C)(=O)=O)C1)NC(C1(O)CCOCC1)C)C(C)C 75920,c1(NC(C2CCC(C(CC)(C)C)CC2)=O)cc(C)cc(Br)c1C 75921,C1(C(=O)NC2CCN(CCNC(C=CCCCCC)=O)CC2)CC2CCCCC12 75922,c1(C(=O)NCCC(CNC(CCCC=C)=O)(C)C)ccn2c1CS(=O)(=O)CC2 75923,c1(N(CC(N)=O)CC2(C)CCN2)ccc2ccccc2c1 75924,c1(C(=O)NCCCNC(c2c(C)noc2C)=O)ccc2nc(O)oc2c1 75925,C1(CNC(C(C)NC(C)=O)=O)CCN(C(=O)Cc2ccccc2Br)CC1 75926,C12(C(=O)NCC3C(C)CN(C(c4cnn(C)c4Cl)=O)C3)CCOC(C)(C1)C2 75927,c1(C(N2CCN(C)CC2)=O)c(F)cc(F)cc1Br.C1(C(N)=O)CCCC(C(=O)O)C1 75928,C1(C(=O)NCCCCC(C)NC(=O)C=CC2CCC2)CCc2ccccc2N1 75929,c1(C(=O)Nc2cnc(Cl)c(C(F)F)n2)ccc(=O)n(-c2ccccc2F)c1 75930,c1(OC)nsc(C(=O)NC2(CNC(c3nnn(C)n3)=O)CCCC2)c1Br 75931,C#Cc1cc(C(=O)NC2COCC2NC(=O)C(C)CC(F)(F)F)ccc1C 75932,c1(NC(C2CC(CO)C2)=O)nc2n(c1Cl)CCNC2 75933,c1(OC)cccc2c(CCNC(C3(c4ccc(F)cc4)CC(C)(C)C3)=O)c[nH]c12 75934,N1(C(c2ccc(COC)cc2)=O)CCCC2C1CCN2C(c1cnccc1C)=O 75935,C(=O)(C(C)CS(C)=O)NCC1(CNC(c2c(C)n[nH]c2C)=O)CC1 75936,C(=O)(C(C)(C)CC)NCC1(NC(c2cn(CCC3CC3)nn2)=O)CC(OC)C1 75937,C1(C(=O)NCC(CC(C)C)(C)C)CCN(C(=O)CCC(C)(C)F)O1 75938,CCC(O)C(C)(C)C(=O)NCC1(CN(C)C(c2cc(O)nc(Cl)c2)=O)CC1 75939,C=Cc1cncc(C(=O)NC(CC2CC2)C(=O)NCCC2(SC)CCC2)c1 75940,CC(C)C(O)C(=O)N1CCC(C(C)(O)CNC(=O)C(F)=C2CCCC2)CC1 75941,C1(CC(=O)NCC2(OC)CCOC2)CC2CCC(C1)N2C(c1cocc1C(N)=O)=O 75942,C(CC(CNC(=O)CN1CCCCC1)NC(=O)C=C1CC(C(C)(C)C)C1)OC 75943,CC(C)(CC(F)(F)F)C(=O)NCc1cccc([N+](=O)[O-])c1 75944,N1(C(C2CCN(C)C2=O)=O)CCCN(C(=O)CCc2cccc(F)c2F)CCC1 75945,C1(C(=O)NCC(=C)C)CC(N(C(=O)CCC2CCC2)C)C1 75946,N1(C(C2CC2c2cccc(F)c2)=O)CC2CC1CN2C(C12CCC(CC1)C2)=O 75947,N1(C(C(c2cn(C)nc2)O)=O)CCCCCC1C(N1CC(n2ccnc2)C1)=O 75948,c1(C(=O)N(C(C)CO)CC)c(C)[nH]c(C)c1C(=O)C(C)OC 75949,CCCCC(CNC(=O)OC(C)(C)C)OC(=O)CC1CC(F)(F)C1 75950,N1(C(C(Cc2cn[nH]c2)NC(c2cc(=N)[nH][nH]2)=O)=O)CC2CC1CS2=O 75951,c1(C(=O)NC2C(SC)CN(C(C3(C#N)CCC3)=O)C2)nn2cccnc2c1Br 75952,C12(C(=O)NCC3(C#C)CC3)CCC(CC1)N(C(=O)C=C1CCC(C)CC1)C2 75953,C1(CCC(=O)N(C(CC)COC)C)CCCCN1C(c1ccncc1O)=O 75954,c1(CC(=O)N(CCN2CCN(C(C(C(C)O)C)=O)CC2)C)ccc2ccoc2c1 75955,c1(COC(CN(CC(C)(O)C2CC2)C(C2C(C)C2)=O)=O)ccco1 75956,c1(C(=O)NCC2C(NC(CC(CC)OC)=O)C2)cc(-n2ccnn2)ccc1F 75957,N1(c2cc(OC)nc(OC)n2)CCC2CN(C(c3cc(O)cc(O)c3)=O)CC2C1 75958,C1(C)(C(N2CC(OC)(CO)C2)=O)CC(O)CN1C(=O)C=C(C)C(C)C 75959,N1(C(c2c(C)nsc2)=O)CC(NC(=O)COCc2nc[nH]n2)CC1C 75960,C(C(C)C(=O)N(C)OC)N(CC(C(=O)N(C)C)=C(C)C)C 75961,C1(CNC(C2CCN(C(=O)NCC3CCC4(CC4)C3)CC2)=O)CC(C)OC(C)C1 75962,CC1CCN(C(=O)COC(=O)CO)C1CNC(=O)CCCC1CC1 75963,c1(CNC(C(=O)NC(c2cccc(C)c2)CC)=O)cn2cccnc2n1 75964,N1(C(CSCCC)=O)CCCC(C2CC2NC(=O)CC2(O)CCCN(C)C2)C1 75965,Cc1cccc2[nH]cc(C(=O)NCCN(C(=O)C(C)n3ccnc3)CC(C)O)c12 75966,C1(OC)CC(CNC(=O)C2=CCCS2)N(C(=O)CC2(C)CCC2)C1 75967,C1(NC(CC2CCN(C)C2)=O)CN(C(c2cncc(N)n2)=O)CCC1CO 75968,N1(C(CC)=O)CCC(N=c2nc(N3CCC=CC3)c3c([nH]2)CCC(C)C3)C1 75969,N1(C(C2(C)COCCO2)=O)CC2CC(NC(c3ccn(CCF)n3)=O)C1C2 75970,c1(CCC(=O)N(CCC(C)NC(C(CC)(C)O)=O)C)nnc(O)nc1O 75971,Cc1cc(Cl)c(Br)cc1S(=O)(=O)N1CCc2scnc2C1 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75990,[N-]=[N+]=Nc1ccccc1NC(C1(NC(=O)C(O)CC2CCCC2)CCSC1)=O 75991,C1(NC(C(CC)OCC)=O)CCC2CN(C(=O)C(C)Sc3ncccn3)CC2C1 75992,C1(NC(CCC(=C)C)=O)CCN(C(=O)CCC2CCC(=O)C2)CC(O)C1 75993,c1(C(N(CC(CNC(c2ccn(C(C)C)n2)=O)C)C)=O)ccc2c(n1)CCCC2 75994,c1(C2(NC(CC3C(CC)C3)=O)CCC2)ccc(Br)nc1 75995,C#CCC(C)(C)C(=O)NCC(C1(O)CCN(C(c2ncncc2N)=O)C1)C 75996,C1(n2cc(-c3c(C)ncnc3)nn2)CCCCCCCCC1 75997,C1(COC)N(C(=O)CC2CCCC(NC(c3cccnn3)=O)C2)CC1(C)C 75998,N1(C(C2(S(N)(=O)=O)CCCC2)=O)CCC2(CC1)OCCC2NC(C1CCCC1)=O 75999,c1(N2CC(NC(C(c3cscn3)N(C(C)=O)C)=O)C2)cc(O)ncn1 76000,C1(CNC(c2cc(C)sn2)=O)CCCCN1C(c1cocc1C(N)=O)=O 76001,N1(C(Cc2nc(C)[nH]n2)=O)CCCCC1CCCNC(=O)C(F)CC1CC1 76002,C(=O)(CS(=O)(=O)C(C)C)N1CC(OC)CC1(C)CNC(=O)C=Cc1ccoc1 76003,N#CC12CCCCCC1CN(c1ccn3c(Br)cnc3n1)C2 76004,N1(C(c2c(CC)nnc(C)c2)=O)CC(NC(C2CN(CC)C2)=O)CC12CCOC2 76005,C12CCCCN1C(=O)O2.N1(C(=O)COCc2ccccc2)CCCC(F)C1 76006,c1(CC(=O)NCc2nc(CNC(C(COC)C)=O)sc2)ccc2c(c1)CCO2 76007,CC1(C)NC(=O)CCC1NC(C1CCN1C(c1ccn2ccnc2c1)=O)=O 76008,CC(CNC(=O)C(C)(C1CC1)N(C(=O)CC1NC(=O)NC1=O)C)C(C)(C)C 76009,Cc1cc(C(=O)NC2CN(C(c3csc(C(F)F)c3)=O)CCC2CO)cnc1O 76010,Cc1c(C(=O)NCC(CNC(=O)Cc2nc[nH]n2)CO)sc2nnc(S)n12 76011,C1(NC(C(C)OCc2ccccc2)=O)CN(C(c2cc(Br)cs2)=O)CC12COC2 76012,N#CC1CCC(C(=O)NC2CC(CNC(=O)Cc3cnn(C(F)F)c3)C2)CC1 76013,C1(C(N2CCC(CC#C)CC2)=O)CN(C)CCN1C(C1C2COCC12)=O 76014,c1(CN(C(C(c2cn(C)nn2)NC(Cn2c(C)nnn2)=O)=O)C)ccccc1F 76015,C12(CC)CN(C(=O)CC(C)OC)C(CNC(=O)CC3C(=O)NN=C3C)(C1)C2 76016,N1(C(CC=CCNC(CC=C(C)C)=O)=O)CCC(COC(C)C)CC1 76017,c1(CC)cscc1C(=O)NCc1n[nH]cc1C(=O)NC(c1cccnc1)C 76018,c1(CNC(=O)CC2CSCCO2)ccc(C(=O)Nc2n(CC)ccn2)nc1 76019,N1(C(C(C(CNC(c2ccnc(OC)n2)=O)C)F)=O)CCc2nc(O)[nH]c2C1 76020,C(N=c1cc(N2CCOC(C)C2)nc[nH]1)C1(Nc2c(SC)cccc2)CCC1 76021,C1(C)(C(=O)NCC2CC(O)(CNC(c3nc(C)oc3)=O)C2)CNC(=O)C1 76022,C(=O)(C(C)CS(C)(=O)=O)NCCC(C)CF 76023,CCCCCCOC.c1(C2C3(CC3)CN2)nnnn1CCOCOC.OC 76024,Cc1oc(CNC(=O)CC2CCCO2)nc1C(N1CCC(Cc2ccsc2)C1)=O 76025,Cc1ccnc(C(=O)N(C2CCC(NC(c3sc(Cl)cc3Cl)=O)C2)C)n1 76026,CC1C(C)N(C(c2ccc(OCF)cc2)=O)CCN1C(=O)CC(O)CCN(C)C 76027,Cc1cccc(C(=O)NCC)c1C.N12CCN(C(C)C1)C(=O)Cc1cc(cs1)C2=O 76028,N1(C(CN2C(=O)COCC2)=O)CCC2CCC(C1)N2C(=O)CN1CCCC1CO 76029,N1(C(CCOCC#C)=O)Cc2ncsc2C1.C12CC(CO1)C(=O)NC2 76030,Cc1cc2cc(C(=O)NCC3CC3CNC(C3CCC3)=O)oc2cc1C 76031,c1(C(N2C(C)CC(NC(c3nc(C)oc3)=O)C2)=O)ccc2c(c1)OCCC2 76032,c1(CNC2C(c3n(CCOCC)nnn3)CCCCC2)nc(OC)ccc1Cl 76033,N1(C(CSC(C)C)=O)CCCC1(C)C(=O)NCCC1OCCC1(C)C 76034,C12(CCNC(=O)C(=O)NC3(Cl)CCC3)CCCC(C1)C(=O)N2 76035,CN1CCOCC1C(=O)NCCC1CSCCN1C(=O)CN1CCSCC1 76036,C1(C(N2CCC(=CCNC(=O)C=Cc3ncc(C)[nH]3)CC2)=O)(CC)CCNC1=O 76037,C1(N(CCC)C(c2ccc(CSC)o2)=O)CCN(C(=O)CCSCCC)CC1 76038,CCCC(O)C(=O)N1CCC(NC(=O)CCCNC(C)=O)C1 76039,C1(CC(N2C(CNC(C3CCCC(OC)C3)=O)CC2)=O)CCn2cncc2C1 76040,N1(C(C#CC(C)C)=O)CC(NC(c2coc(Br)n2)=O)C(C2CC2)C1 76041,N1(C(c2cc3ccoc3cn2)=O)CCCC2C1CCN2c1ncc(Cl)cn1 76042,C(=O)(C1c2[nH]cnc2CCN1C(=O)C(COC)OCc1ccccc1)OC 76043,C1(Nc2ncnc(C)c2F)CN(C(C2CC(N=[N+]=[N-])C2)=O)CC12CCOCC2 76044,C1(=CC(=O)NCCC2(NC(C(C)OCC3CC3)=O)CCCC2)CN2CCC1CC2 76045,Cc1cc(NC(=O)CC2(C)CCN2C(C2(C)CC2)=O)c([N+](=O)[O-])cc1Br 76046,CC(O)C(C(=O)NCCNC(=O)CCC1CCCCCC1)NC(=O)C1CC1 76047,C1(CCNC(c2cc(C(=O)OC)[nH]c2)=O)CC(F)(F)CN1C(c1ccc(C)o1)=O 76048,C1(NC(C(CC(C)C)NC(N)=O)=O)CN(C(C2(C)CCCCO2)=O)CCC1(C)C 76049,C1(C(N(CCCn2cc(CCCS(N)(=O)=O)nn2)C)=O)CCOC2(CCCC2)C1 76050,C1(F)(CN(C(=O)Cn2nnc(C3CC3)n2)C(c2ccco2)=O)CCCOC1 76051,N1(C(=O)NCCOC(CC)CC)CCc2nc(I)[nH]c2C1 76052,C(=O)(CCN=c1nc2c(ncn2C(C)C)c(N(CC(C(C)C)NC)C)[nH]1)NCC 76053,C=C=C(C)CC(=O)NCC(C)NC(c1cccc(C(F)(F)F)c1)=O 76054,c1(NC(C2C3(CCN(C(c4ccc(C)c(O)c4)=O)C3)C2)=O)csc2nccnc12 76055,C(c1cncn1C)=CC(=O)NC1CC(C(C)NC(=O)CC2CCOC2)C1 76056,C1(NC(C2CC(N(C)C)C2)=O)CCCC(NC(c2ccc(=O)oc2)=O)C1 76057,C1(N(C(CCOCCN(C)C(C2CCCC2C#N)=O)=O)C)CCCCCC1 76058,C(C(C)(CC(C)C)NC(c1cc(C(N)=O)on1)=O)NC(C(C)=CC1CC1)=O 76059,c1(C(N2C(CC(=O)N(C(C=C)C)C)CC2)=O)cnn2ccccc12 76060,CN=c1[nH]cc(C(=O)N(CC(N2CCC(C)(O)C2)=O)C2CC2)o1 76061,c1(C(=O)NCC(Cn2cc(CC(CC)(C)O)nn2)(F)F)ccc(=O)n(C(C)C)c1 76062,CC#CC1CCN(C(c2coc(CNC(C3(COC)CCC3)=O)c2)=O)CC1 76063,N1(c2nccc(SC)n2)CCC(C2CN(c3cc(C)ncn3)C2)CC1 76064,N1(C(CCCCC=CC)=O)CCC(C2CCN(C(=O)CSC3CC3)CC2)C1 76065,N1(C(CC2(OC)CCC2)=O)CCC2C(C1)OCCN2C(c1ccccc1C#N)=O 76066,NC(=O)CCCNC(C1CCC(NCc2ncc(Cl)s2)C1)=O 76067,C=CCC(CC(C)C)C(=O)N1CCCOC(CNC(=O)C(=O)C(C)(C)C)C1 76068,Cc1c(C(=O)NCCCCN(C(=O)CC2CN(C)C2)C)cccc1Cl 76069,C=C(C)CCCC(=O)N1CCCCCC1CNC(=O)CC1CCCCN1C 76070,N1(C(c2cnc(C)nc2)=O)CCC2CN(C(c3cncnc3C3CC3)=O)CC2C1 76071,c1(C(=O)Nc2ccc(C(N3C(CCC=C)CCC3)=O)nc2)cnnc(C)c1C 76072,C(=O)(C1c2c[nH]nc2CN1C(C1CCCCN1C)=O)N(CCC(=O)NC)CC 76073,C1(n2cc(C(C)(C)CC3CC3)nn2)(OC)CCN(C(C2CC(F)(F)C2)=O)CC1 76074,C1(C(N2CCC(NC(=O)CC3CCCCC3)C23CC3)=O)CC2CCC(C1)C2O 76075,C1(C(=O)NOC(C)C(=O)OC)(CC=C)CCCN1C(c1ccc(C)cn1)=O 76076,C1(NC(Cc2scc(C#N)c2)=O)CC12CCN(C(C13CC(CO)(C1)C3)=O)CC2 76077,Cc1cnn(CCNC(=O)CC2(NC(C3CC(F)C3)=O)CC2)c1 76078,C1(C(=O)Nc2ccc(CCNC(=O)NC)cc2)CC2CCCC2C1 76079,C1(C)(C(N(CCOC)CCn2cc(C3(CCO)CC3)nn2)=O)CC(C#N)C1 76080,c1(C(N2CCN(C)CC2CNC(C2CC2(C)C)=O)=O)cc2c(cn1)OCO2 76081,C#CC1(C(=O)NCCC(=O)OC(C)(C)C)CN(C(=O)CCn2ccnc2)C1 76082,C(=O)(CC(F)(F)Cl)N(C(C)CNC(=O)C(C)Sc1nncn1C)CC 76083,C1(OC(=O)OCCSCCOC)CCCC1 76084,CCC(CC1CCCC1)C(=O)NC1CCCCC1NC(C1OCCCO1)=O 76085,N1(C(C)C)CCC(CC(=O)NCCC2CCN(C(C3C(C)C3(F)F)=O)C2)CC1 76086,C12(CNC(COC)=O)CCC(CC1NC(=O)Cc1ncn(C)n1)C2 76087,Cc1cc(C(=O)NCCN(C(=O)Cc2ccco2)C)n(C2CCC2)n1 76088,c1(CCC)cc(C(=O)NCC2C3CN(C(C4(CO)CCCO4)=O)CC23)nn1C 76089,C(=O)(C1=CCN(C(c2cscn2)=O)CC1)NCC1C(C)CCCC1 76090,c1(CCS(CC2OCC(C)(C)OC2)=O)ncc(Br)cc1[N+](=O)[O-] 76091,C(c1cn(C)nn1)=CC(=O)NC(C(=O)NC(CC=C)CC)CC1CCC1 76092,c1(C(=O)NCC2C(CC(=O)NCc3ncsn3)C2)cc(Cl)n[nH]1 76093,N1(C(C(CC(C)C)NC(=O)CC2CC=CCC2)=O)CCCCCCC1C 76094,c1(CCCC(=O)N(CC(C)NC(=O)Cc2ccon2)C)ccc(Br)cn1 76095,N1(C(C(C)N(C)C)=O)CC2CC(NC(c3ccsn3)=O)CC1C2 76096,N1(C(C(=O)Nc2ccc(C)cc2)=O)CCCN(C(c2cc(C)c(C)cn2)=O)CC1 76097,C(=O)(CCCC(=O)N1CC(C(C)NC(=O)CCC(=O)c2cccc(Cl)c2)C1)OC 76098,Cc1cnc2cccc(C(=O)N(C(C)CNC(=O)CSCC(C)C)C)n12 76099,N1(C(c2cn(CC=C)nc2)=O)CCC2(CC2C(N2CC(C(C)OC)C2)=O)C1 76100,N1(C(C2C(=C)CC2)=O)CC(C)OC2(CCN(c3nc4cc(C)ccc4o3)CC2)C1 76101,C1(NC(Cc2n[nH]c(=NC)s2)=O)CC2CC(C1)N(C(C1(O)CCC1)=O)C2 76102,C=CCC(C)C(=O)N1CCC(C(F)F)(CNC(=O)CN(c2ccnc(Cl)n2)C)C1 76103,c1(C(=O)Nc2cc(C)c3c(c2)NC(=O)CO3)cc2c3ccccc3n(C)c2s1 76104,C(CC(C)(C)C(=O)N(C)Cc1cncn1C)NC(C(C=C)CC)=O 76105,C1(CNC(C(CNC(C(CC)C#N)=O)(C)C)=O)CCOCC1(C)C 76106,c1(CC(=O)NCCCCNC(c2cnn(C)c2C2CC2)=O)ccc(S(N)(=O)=O)s1 76107,N1(C(C(CC)(C)O)=O)CCOCC(CNC(=O)CCc2ccn(C)n2)C1 76108,CCC(CN(C)C)CC(=O)N1CCCCC1CN(C)C(C1CCCC2(CC2)C1)=O 76109,c1(CC)cccc(C(N2CCCC(NC(C3CCC4(CCC4)C3)=O)CC2)=O)c1O 76110,CN=c1[nH]cc(-c2ccc(C(N3CC4CC(C(=O)OC)C4C3)=O)cc2)cc1C#N 76111,c1(NC(=O)NC(c2ccc(SCC)cc2)CC(F)(F)F)ccc(Br)cc1OCC 76112,C1(NC(C2C(NC(CCNC(CCc3cn(C)nc3)=O)=O)C2)=O)CCC(C2CC2)C1 76113,O(NC(=O)C(F)C1(O)CN(C(c2cn(C)c(C)n2)=O)C1)CC(=C)Cl 76114,C1(CNC(C(CC)CC)=O)CCCCCN1C(c1cc(-c2ccoc2)on1)=O 76115,Cc1cc(-c2ccc(C(N)=O)cc2)nc(C(F)(F)F)n1 76116,c1(C(=O)NC2CCN(C(C(C(C)C)OC)=O)C2C)cc([N+](=O)[O-])c(C)cc1C 76117,c1(-c2nc(C(C3CC3)OC)nn2C2CCCSC2)cnc(C(C)C)c(Cl)c1 76118,c1(CC)ccc(C=CC(=O)NC(CNC(C2CC(O)CN2C)=O)C(C)C)o1 76119,C1(CNC(C(c2ccccc2)N(C)CC)=O)CC2CC2N1C(C1CC(O)C1)=O 76120,c1(C(N(C2CCCN(C(C(CC)O)=O)CC2)C)=O)cc(=O)c2cc(F)ccc2o1 76121,c1(N(C)Cc2cccc(OC)n2)ncccc1S(=O)(=O)NC12CCN(CC1)CC2 76122,C12(C(=O)NCC(C)(CNC(=O)C(C)(C)OC(C)=O)OC)CCC(F)(CC1)CC2 76123,Cc1c(C(N2CCC(C)C2CNC(C2(CO)CC2)=O)=O)cc(C(C)(C)C)n1C 76124,c1(C(=O)NC(C(C)(C)C)CNC(C2C3CCCC23)=O)cnn2ccccc12 76125,c1(OC)noc(C2CC2)c1C(N1CCCC(Cc2cn(C(C)C)nn2)C1)=O 76126,c1(C(N(CC(=O)NCCN(C)C(C2CC2F)=O)C)=O)cccnc1 76127,N1(C(Cc2c(C)noc2)=O)CC(O)CCC1C(=O)NCC(C)(O)C1CCCC1 76128,CCC(C)(C(=O)NCCCOCCNC(=O)C(C1CCCC1)OC)N(C)C 76129,N1(C(C(C(C)C)N2CCCC2=O)=O)CCCN(C(C2CC3(F)CC2C3)=O)CC1 76130,C1(C(=O)NC2CCC(CNC(C(C=C)(C)O)=O)C2)CCc2cncn2C1 76131,N1(C(=O)Cc2cnn(C(F)F)c2)CC2CCCC(C1)N2C(C1CCC2CC12)=O 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76168,CCCCC(CC(=O)N(C1COC(C)(C)C1)C)NC(C1CCCC(C#N)C1)=O 76169,Cc1sc(Cl)nc1C(N1CCN(C2COCC2NC(=O)Cc2ccoc2)CC1)=O 76170,N1(C(CCCSC)=O)CCCC1C1CCCN1C(c1nc(OC)ccc1Cl)=O 76171,N1(C(CCCCOCC)=O)CCC2CN(C(=O)CC(O)CN(C)C)CC12 76172,N1(C(C2(C#N)CC3CC3C2)=O)C2CCC1CC(NC(=O)Cc1cc[nH]n1)C2 76173,C1(C(N(C)CC2CCCN2C(C2(CO)CCCCC2)=O)=O)CCC2(CCC2)O1 76174,C1(NC(CCC=C)=O)CC(C(=O)NCCC2CCN(C)C2=O)=CC1O 76175,C1(C(N2CCC(O)C2)=O)(CC)CCCN1C(=O)C=CCN(C)C 76176,C1(C(C)NC(Cn2c(C)nnn2)=O)CCN(C(C2C(F)(F)C23CC3)=O)CC1 76177,C1(CNC(=O)CCc2ccccc2)CN(C(=O)CCC2OCCO2)CCCO1 76178,C1(C(=O)NCC(=O)NOC)(OC)CCN(C(=O)C(F)C2CCC2)C1 76179,C(=O)(C#CC1CCCO1)N(C)C(N1CCCC(c2nnc(O)o2)C1)=O 76180,N1(C(c2c(Cl)cc(C)c(C)c2)=O)CCC2CN(C(=O)Cc3cnco3)CC2CC1 76181,c1(C(C(=O)NCC2(NC(CCOCC)=O)CC2)C)ccn(C)c1 76182,CCCCC(C(=O)N(C)CCOCCN(C(=O)C(n1cc(Cl)cn1)C)C)C(C)C 76183,C1(CNC(C(CC)CCOC)=O)CCC2(CN(C(=O)Cc3ccccc3F)C2)O1 76184,c1(C(=O)NC2(CC=C)CCN(C(c3cn(CC)cn3)=O)C2)cccc2cnsc12 76185,C1(C(N2CCC(NC(C3Cc4cscc4C3)=O)C2)=O)CC2(CCC2O)C1 76186,[N-]=[N+]=NCC(F)CC(C(=O)O)NC(=O)C=Cc1cn(CCF)nn1 76187,C=CC1CN(C(=O)CNC(C2CCC2)=O)CC1NC(=O)Cn1cc(C2CC2)cn1 76188,C1(C)(C(N2CCC(C(C)(C)NC(CC(C(=C)C)O)=O)CC2)=O)CCC(C)=C(C)C1 76189,c1(C(=O)NC(CC(C)NC(Cc2nnc(C)o2)=O)C)ccc2nc[nH]c2c1 76190,C1(CNC(c2cc(CF)on2)=O)CC2CC1CN2C(c1cc(Br)c[nH]1)=O 76191,c1(C(N2CCC(NC(C(C3CC3)OC)=O)CC2C)=O)cc(S(N)(=O)=O)oc1C 76192,C(CC(C)(C)C(=O)N1CCC(O)(CCNC(=O)C(F)C2CCOC2)CC1)OC 76193,C(=O)(CC1CCc2ccccc21)N1CC2C(NC(CSc3cn(C)nc3)=O)(C2)C1 76194,C(N=c1cccc(S(=O)(=O)NCC2CN(C)C2)[nH]1)C1CC(OC)C1(C)C 76195,n1(CCC=C)nc(COC2CCCCC2)nc1-c1cc(CO)on1 76196,c1(C(=O)NCC(C)NC(Cc2c(C)cc(Cl)cc2)=O)cc(C)n(C)c(=O)c1 76197,C(=O)(C(C)(C)CC(C)C)NCCN(C(=O)CCCSc1ccc(Cl)cc1)CCC 76198,C=CCC(F)(F)C(=O)NCC1CCCN1C(c1cc(OC)n(C)n1)=O 76199,c1(C(=O)NCC(C)CNC(c2c[nH]nc2C2CCCO2)=O)cnn(C)c1C(F)F 76200,N1(C(C(C2CC2)OC)=O)CCC(C)N(C(c2cc3ccsc3s2)=O)CC1 76201,C(C1c2ccsc2CCN1C(=O)C(C)OCCN(C)C)NC(C(C)OCC#C)=O 76202,c1(N)cc(C#N)cs1.C1(C(=O)NCCNS(CC)(=O)=O)CCCN1C(C1CC1C)=O 76203,c1(OC)ccc(Cl)c(C(=O)NC2CC(CCNC(C3CCOC3)=O)C2)c1 76204,c1(CNC(=O)NCC(C2CCC(F)(F)CC2)O)cccc([N+](=O)[O-])c1 76205,c1(OC(C)C(=O)NCC(c2ccccc2)C)ccc(C#N)c(Cl)c1 76206,N(C(=NCCOCC(C)(C)O)NC(c1cccs1)C)Cc1cn(C)nc1 76207,c1(C(N2CC3CC2C3)C(=O)NC(C)(C)C)nncn1C.C(CN(C)C(N)=O)SC 76208,C12(CNC(c3csnc3C3CC3)=O)CCC(F)(F)CC1CNC2 76209,N1(C(c2cscc2C(F)F)=O)CCc2[nH]nc(CNC(C3(F)CCOC3)=O)c2C1 76210,C(C(F)(F)C(=O)N(CC(O)CN(C(=O)C(c1cccc(OC)c1)C)C)C)OC 76211,N1(C(C(C=C)O)=O)CC2(CC(CC(N3CCC(C)(F)C3)=O)C2)C1 76212,c1(C(=O)NC2C(NC(C(CC)N(C)C)=O)CCCC2)cccn2ccnc12 76213,CN1CCN(C(=O)C(CCO)N(C)C)C(CNC(=O)CC23CCC(CC2)C3)C1 76214,N1(C(C2(CC#C)CCC2)=O)CCC(NC(c2coc(N(C)C)n2)=O)C(F)C1 76215,N1(C(CS(CC)=O)=O)CCC(NC(=O)CCCOCC)C1(C)C 76216,C1(CC(N2CC=CC(NC(=O)Cc3ccc(CO)cc3)C2)=O)CCC2(CCC2)O1 76217,c1(OC)ccc(NC2CCN(c3ccnc(SC)n3)CC2C)c(O)c1 76218,Cc1[nH]c2ccccc2c1C(=O)NCCC1CCCN1C(=O)CC1C=CCCC1 76219,N1(C(C2(C(F)(F)F)CC(=C)C2)=O)C2CCC1CN(C(c1ccoc1Cl)=O)CC2 76220,C1(CNC(c2c(C)nsc2Cl)=O)CC2CCC(C1)N2C(=O)CC1CSC1 76221,N1(C(c2c(C)scn2)=O)CC(CNC(C2(C)CC3(CCC3)C2)=O)CC12CCC2 76222,N1(C(C(=O)NCCC(C)N(C(CCN(C(C)=O)C)=O)C)C)CCCCCC1 76223,C1(OC)CC(CNC(=O)CC23CCC(CC2)C3)N(C(C2CCS(=O)(=O)N2)=O)C1 76224,C=CC(CCC)CC(=O)NCCC1CC(C(=O)NCC(F)(F)C(F)F)C1 76225,c1(C(N(CCOCCN(C(C(CC)(C)F)=O)C)C)=O)ncnc2c1cnn2C 76226,c1(C(=O)NC2CCC(NC(=O)CCc3cnc(O)[nH]3)C2)cc2cc(Cl)ccn2n1 76227,c1(C(=O)NC2CC(CNC(C3CC3(F)F)=O)C(O)C2)nc2ccccn2c1F 76228,c1(C(=O)NC(C)CCCNC(=O)CN2CCS(=O)CC2)cnn2c1OCC(F)C2 76229,O=C1CCC(CN=C(NC2CC2)NCC(C2CCCCC2)(F)F)C(=O)N1 76230,c1(CCC)sc(C(=O)NCC2(NC(C3CC=CCC3)=O)CCOC2)cc1CC 76231,c1(C(N2CCC(CC#C)CC2)C(=O)NCCC#N)cncc(C=C)c1 76232,O(N(CC)C(=O)C1(NC(C2CC=CCO2)=O)CCC1)CC 76233,N1(c2nnc(C(C)C)o2)CCCC2C(NC(C3CC(=O)CO3)=O)C(C)(C)C12 76234,C1(NC(=O)C(c2ccccc2)O)CC2(CCN(C(C3CC=CCC3)=O)C2)C1 76235,N1(C(=O)COCCc2nc(-c3ccncc3)no2)CC=C(CO)CC1 76236,Nc1cc(C(N2CC(F)CC2C(=O)NC2CC(C3CCC3)C2)=O)cc(F)c1 76237,C1(CNC(CN2C(C)CCCC2)=O)CCCCCN1C(=O)CC1(C)CC1 76238,C(=O)(C1=CCCN(C(C23CCCC2C3(F)F)=O)C1)NCC1C(N(C)C)COC1 76239,Cc1cc(C(=O)NCC2(CN(C)C(C3CCCC3C)=O)CC2)cc(C)c1C 76240,c1(CNC(C=CC=CC)=O)nc2c(s1)CN(C(C1C(C)(C)C1(C)C)=O)CC2 76241,c1(C(=O)NCCC(=C)CNC(C23CC(CCO2)C3)=O)c(Cl)cncc1Br 76242,CC1CC(C(=O)N(C)CC2(NC(=O)C(F)C(F)(F)F)CC2)=NO1 76243,N1(C(c2c(CC)c[nH]c2)=O)CC(C)CN(C(=O)Cc2csc(C3CC3)n2)C(C)C1 76244,C1(C(=O)NCC2CC(NC(CCn3ccc(C)n3)=O)C2)CCN(C(N)=O)CC1 76245,c1(C(=O)NCC(CCC)NC(=O)COCC2CCCOC2)cccn2cncc12 76246,N1(C(C2(C)C(CC)CCC2)=O)CC2CCC(C1)N2C(C1(CC2CC2)CCCC1)=O 76247,C(C)(C)(CCCCNC(C(c1ccc(C)cc1)F)=O)NC(C1CCN1C)=O 76248,CCCCC(CC)CC(=O)N1CCC(N=[N+]=[N-])(C(=O)NCCC(C)O)C1 76249,c1(C(=O)NCC2(O)CN(C(C(C)NC(CC)(C)C)=O)C2)cnc2cnn(C)c2c1 76250,c1(CC(N2CC(C)(NC(C3CCC4C3C4(F)F)=O)C2)=O)noc2ccc(F)cc12 76251,C1(NC(Cc2c(C)cc(Cl)nc2)=O)CN(C(=O)CCOC(C)C)CCC12CCC2 76252,N1(C(C(=O)NCCOC)=O)CC(NC(=O)Cc2nc(C)sc2Cl)C2(CC2)C1 76253,C1(OC(=N)O)CN(C(=O)CCOCCNC(C2CSC2)=O)C1 76254,N1(C(CCOC)=O)CCC2CCCC12C(=O)N(C)CCSC 76255,Cc1sc(=O)n(CC(=O)NCCN(C(=O)C(Cl)=CCl)C2CC2)c1-c1ccccc1 76256,N1(C(CN(C)CC)=O)CC2CC(C1)N2C(C1CC1Cl)=O 76257,N1(C(CC(C)N(C)C)=O)CC(NC(c2ccc(SC(F)(F)F)o2)=O)CC12CCC2 76258,N1(C(C(c2cccc(Cl)c2)SC)=O)CCC(F)(C(N)=O)C1 76259,O=C1CCC(C(=O)NCC23CCC(NC(=O)Cc4ccccc4Cl)(CO2)C3)=NN1 76260,N1(C(C(C)O)=O)CCC2CCN(C(=O)COc3ccc(Cl)nc3)CC2C1 76261,S(=O)(=O)(CCC(F)(F)C(C)(F)F)NC(=O)CN(CC(F)(F)F)CC#C 76262,c1(C(N2C(C(CNC(CC=CC)=O)(C)C)CCC2)=O)cc2occc2n1C 76263,C1(CNC(C(C)(O)c2ccccn2)=O)C2CN(C(=O)Cc3ccc(Cl)s3)CC12 76264,C1(NC(=O)C2=CCOC2)COC2(C1)CN(C(=O)Cc1ccc(O)cc1Cl)C2 76265,C(=O)(C(CC(C)C)C(C)C)N(C(C(=O)OCC)C)C 76266,C(C1CCCCC1)=CC(=O)NCC(=O)NC(c1cn(C2CCOCC2)cn1)C 76267,c1(C(=O)NCC2N(C(=O)Cn3ccnn3)CCN(C)C2)ccc2oncc2c1 76268,N1(C(CC=C=C)=O)CCC2(CCCN2C(=O)Cc2cncc(O)c2)C1 76269,N1(C(C(C)N(C(=O)C#CC2CC2)C)=O)CC2(CNC(=O)N2)C1 76270,CCC(CC)(CC)C(=O)NC1CC2CN(C(=O)Cn3ccc(C)n3)CC2C1 76271,c1(NCC(N2C(C)C(N3CCCCC3)CC2)=O)ccc(S(N)(=O)=O)cc1[N+](=O)[O-] 76272,CC1CC(NC(=O)CCCc2ccc(N)cc2)CN1C(c1cc(Cl)no1)=O 76273,C12(NC(c3c(C)cc(C)nc3)=O)CCCCCC1N(C(c1cn[nH]c1)=O)CC2 76274,c1(NC2(CNC(c3cccc4[nH]ccc34)=O)CCCC2)ncc2c(n1)COC2 76275,C#Cc1ccc(CC(N2CC(NC(=O)C=CC)CC2(CC)CC)=O)c(F)c1 76276,C1(C(=O)Nc2cnn(C(C)C)n2)CCCC2(CN(C(=O)CN3CCCC3=O)C2)O1 76277,c1(C(C)NC(=O)N(C)CC2CCCN2C)c(F)cccc1I 76278,C(CC(CCC)CCC)NC(C(CCCNC(C(C=C=C)C)=O)O)=O 76279,C1(C(N2CCC(Cc3cn(C4CCC4)nn3)C2)=O)(OC)CCCC1 76280,c1(N2CCC(CC=C)(NC(=O)CCc3ncc(C)[nH]3)C2)ncnc(C)c1C#N 76281,C(=O)(C(O)C(F)(F)c1ccccc1)N(C1CCN(C(c2c(C)nncc2)=O)C1)C 76282,C(=O)(C1=CNC2=NCCCN12)NC(C)CN(C(=O)CN1CCCCC1=O)C 76283,Cc1c(N)ccc(C(=O)NCCC2CCN(C(=O)OC(C)(C)C)C2)c1Cl 76284,c1(NC(CCN(C(=O)C=C(C2CC2)C2CC2)CC=C)=O)cc(CO)cc(C)c1 76285,c1(OC)c(Cl)cc(C(N2CC3(CC3)CC2CNC(=O)C(C)C)=O)nc1Cl 76286,c1(C(=O)OC)ccc(CC(=O)N(CCNC(=O)CC(C)CF)C)c(C)c1 76287,C(C)(C)(C(C)CC(=O)N(C)OC1CCCC1)NC(C(C(CC)C)c1ccon1)=O 76288,CCCCC(CCCC)C(=O)N(C1CCCC1)CCNC(=O)CC1CCCN1C 76289,C(=O)(C1=CCCCC1)N1CC2C(CNC(c3cc(C)sn3)=O)C2C1 76290,c1(CC)ccccc1C(CNC(=O)C(O)CCC1CC1)NC(=O)C(O)CCSC 76291,C1(C2CCN(C(=O)NCCC(C)n3ccnc3)C2)OC(C)(C)C(C)(C)O1 76292,c1(C(N(C(CNC(c2cn(CCCC)nn2)=O)C)C)=O)cc(S(=O)(=O)NC)cs1 76293,c1(CNC(CC2CC(=C)C2)=O)cc(C(=O)NCC2CC(COC)C2)cs1 76294,c1(C(=O)NCC2C=CCN2C(=O)C(O)C2CC2)ccc2nc[nH]c2c1F 76295,c1(OC)ccc(OC)c(C(=O)NC2CCCCCC2NC(=O)C2CC2)c1N 76296,Cn1c(O)nc2cc(C(=O)NC3(CNC(c4n[nH]c5c4COCC5)=O)CC3)sc12 76297,c1(C(=O)NCC2CCC2NC(C2(Br)CC2)=O)ccc2ncnn2c1 76298,C(=O)(C(CC)C(=O)N1CC(CO)(NC(c2cc(C(N)=O)ccc2C)=O)C1)OCC 76299,N1(C(c2n(CC)cnn2)=O)CC2CC2(CNC(=O)C(C)Cc2ccco2)C1 76300,C1(OC)CC(C(=O)N(C)CC=C(C)C)N(C(=O)CC=CC(C)(C)C)C1 76301,N(C(=NCC1CN(C2CC2)C(=O)O1)N1CCN(CC2CCC2)CC1)C(C=C)C 76302,c1(NC(=O)NCC2CCN(C(=O)C(N3CCOCC3)=O)CC2)nccc(Cl)c1I 76303,C1(CNC(C2CC3CCC3C2)=O)CN(C(=O)CC2(CO)CC2)C2(CCC2)C1 76304,C=C1CN2C(=O)CCC2(C(N2CC(NC(=O)CS(=O)(=O)C3CC3)C3(CC3)C2)=O)C1 76305,C12(CNC(C3C(C)(C)CCO3)=O)CCCC1CN(C(C1CC1C1CCC1)=O)C2 76306,N1(C(c2cc(F)ccc2Br)=O)CC2CC(NC(C3(F)CC3)=O)C(C2)C1 76307,C1(C(=O)OC)CC(C)N(C(C)CC2(c3ncn(C(C=C)CBr)n3)CC2)C1 76308,S(=O)(=O)(c1ccc2oc(O)nc2c1)Nc1c(C(N2CCOC(O)C2)=O)nccc1 76309,n1(CC)nc(C(=O)NC2C=CCN(C(C3CC(O)CN3C)=O)C2)ccc1=O 76310,c1(OC)ccc(C(=O)NCC(CO)NC(C2CCOC(=O)CC2)=O)cc1N 76311,C1(CN(CC(N2CC(NC(C)=O)C2)=O)C)CCCN1C(=O)CC(C)c1ccco1 76312,C#CCC(C)(CC)C(=O)N(CC(C)(C)CNC(=O)C(O)Cn1cncn1)CC 76313,C=CCCCC(=O)N1CCC(CN(C)C(C2CC2c2ccc(C)cc2)=O)C1 76314,CC1(C)OC2(C(=O)NC3CC(CNC(=O)Cn4cccn4)C3)CCC1C2 76315,N1(Cc2cccc(C(=O)OC)c2)CCC(C#N)(NC(C2CCCS2)=O)C1 76316,C1(CNCCC2CCN(Cc3cccc(C)c3)C2)CCCC(C)(C)C1 76317,C(=O)(N=c1[nH][nH]c2cc(Cl)ncc12)C1C2CN(Cc3c(OC)nc(Br)cc3)CC21 76318,c1(OC)ccccc1CNC(=O)NNC(=O)Nc1nc(C2CCCCC2)sc1C 76319,C1(COC)(CNC(=O)C(O)C2CC2)CCN(C(=O)CN2CC=CC2)CC1 76320,C1(C(=O)NCC(CN(C(=O)Cn2ncc(Br)n2)C)O)CC2CC2C1 76321,C1(CNC(CC(C)n2ccnc2)=O)CC2CCCCC2N1C(C1CC(=O)C1)=O 76322,N1(CCCNC(C2CCCSC2)=O)CCN(C(C2CCC(=O)NC2)=O)CC1 76323,S(=O)(=O)(c1cccc(=NC2C=CCC2)[nH]1)NCCc1c(C)nn(C)c1C 76324,c1(C(=O)NCC2CCN(C(c3ccc(C(C)=O)o3)=O)C2)ccc([N+](=O)[O-])n1C 76325,c1(NCC2N(C)CCOC2)ccc(S(=O)(=O)NCC2CC3(C2)CC(O)C3)cc1Br 76326,CC1CN(C(C2(CF)CC2)=O)CCN1C(c1cc(C2(Cl)CC2)n(C)n1)=O 76327,c1(NC(=O)C(N2CCCC2c2nc3ncccn3n2)=O)cc(Cl)cc(Cl)c1F 76328,C(C1CCOCC1)=CC(NCP(C)(C)=O)=O.C1(=O)C(Cc2cc[nH]n2)CN1 76329,Cc1cc(F)ccc1CC(=O)NCC1CCCC1NC(C1C2COCC12)=O 76330,c1(CS(Cc2onc(CC)n2)=O)cscc1C#N 76331,c1(C(N2CCC(C)C2CC)C(=O)NCC(=C)C)ccc(C(C)C)cc1 76332,C1(C2CN(C(C(N3CCOCC3)C)=O)C2)CN(C(=O)CC2(CO)CC2)CCO1 76333,Cc1ccccc1C=CC(=O)NCC12CC(NCS(=O)(=O)C3CC3)(C1)C(C)O2 76334,N#Cc1cccc([N+](=O)[O-])c1C(F)(F)F.c12cccc(Cl)c1CS(=O)C2 76335,Cc1csc2c(C(N3CCN(C(=O)CS(N)(=O)=O)CC4(CC4)C3)=O)ncnc12 76336,CC(CS(C)=O)N=c1ccc(Br)c(S(=O)(=O)NCCc2c(F)cccc2F)[nH]1 76337,N1(C(C(C)=C2CCC2)=O)CCC2(C1)CN(C(C1(Br)CC1(F)F)=O)C2 76338,C1(C)(C(N2CC(CNC(c3ccc(OC)o3)=O)C(F)(F)C2)=O)CCC(C)C1(C)C 76339,c1(CN(S(C)(=O)=O)CC)nnc(N(C)CCOCC)n1CCC1CCCCC1C 76340,C(C1(C)CCOCC1)=CC(=O)N(C)CC1CCCN1C(=O)CC1CC1(C)C 76341,C=C1CCN(C(=O)COCC)C(CC(=O)NOCC(O)C(C)C)C1 76342,C(CCC(CC)CC)N(C(C1C(CC)N(C(=O)C(C)OCCSC)CC1)=O)C 76343,C(=O)(CC(C)(C)CC(F)F)N1CCC(N(C(C(C)SC)=O)C)C2(C1)CC2 76344,N1(C(CC)=O)CCc2cc(N3CCCC(NC(N4CCCC(O)C4)=O)C3)ccc21 76345,c1(CC)cccc(NC(=O)CCCCCNC(=O)CN2CSCC2=O)c1C 76346,c1(CCC(=O)N(C2CCCN(C(C3(C)CC3C(F)(F)F)=O)C2)C)ccccc1F 76347,c1(C(=O)O)cc(Cl)c(S(=O)(=O)N2CCC3CC(O)CCC3C2)c(Br)c1 76348,c1(-c2ccc(CNCc3ccc(OC)nc3OC)cn2)cnn2cccnc12 76349,c1(C(=O)NC(C(=O)NCC2CC(OC)C2)C2CCOC2)[nH]ccc1C1CC1 76350,C(=O)(C1=CCN(C(=O)Cn2ccccc2=O)C1)NCCN1CCC(OC)C1 76351,C(CCCC(=O)N(C1CCN(C)C1)C)N(C(C(C)=CCC)=O)C 76352,c1(C(=O)NCCC2CCC(NC(C=CCOCCOC)=O)C2)nccc(Cl)c1C 76353,S(=O)(=O)(c1cc(C)cnc1N(C1CC1)C1CC1)N(CCN(CC(CC)C)CCO)C 76354,C1(C(N2CCC(CC)C2CNC(=O)C(F)(F)C(C)(C)O)=O)CCn2ncnc2C1 76355,c1(C(C)NC(CCCCC)c2ccccc2)ccc(S(=O)(=O)N(C)C)cc1 76356,Cc1nn(C)cc1CC(N1CCC(NC(=O)C=Cc2ccccc2)C1C(C)C)=O 76357,N1(S(CCC)(=O)=O)CC2CCC(C1)C2Nc1ncncc1C 76358,C#CCCCCCC(=O)NCC1CCN(C(=O)C2=CCOCC2)CC1C 76359,c1(CC)ccc(C(=O)NC(C)(CNC(=O)C(O)Cc2cnc[nH]2)CO)c(C)n1 76360,c1(NC(C2(SCC)CN(C(C3CCN(C)C3)=O)C2)=O)cccc(CCO)c1 76361,C1(NC(C(CC)C(C)C)=O)C2CC3CN(C(C4CN(C)CC4C)=O)C1C3C2 76362,c1(OCC(N2CC(NC(C3CC(SC)C3)=O)C(C)C2)=O)c(C)occc1=O 76363,c1(C(N2CC=C(CNC(C(CC)C)=O)CC2)=O)cccc2c1CNC2=O 76364,Cc1[nH]c(C)c(C(=O)NC2CCC(NC(c3ccc(C(F)F)cc3F)=O)C2)c1C 76365,CCCCCC(F)C(=O)N1CCC(C)C1C(N1CC(C(C)OC)C1)=O 76366,C12(NC(c3occ4c3CCC4)=O)CCCCCC1N(C(C1COC1)=O)CC2 76367,N1(C(c2cc(C(F)F)cs2)C(=O)NCC(=C)C)CCSCC(CO)C1 76368,C1(C(=O)NCC2(CN(C)C(C3CC(O)(C(F)F)C3)=O)CC2)CCCC2(CC2)C1 76369,N1(C(C2(CCN(C)C)CC2)=O)CCC(CN(C(=O)CCCC2CCCCC2)C)C1 76370,C(=O)(CCCCCCCCCO)NCC(CN(C)CCn1ccc(O)nc1=O)O 76371,C(=O)(CC1=CCN(C)CC1)NCC(CN(C(CSc1ccc(OC)cc1)=O)C)C 76372,N1(Cc2cc(C)sc2C)CCn2c(C(N3CCC4(CC3)COC4)=O)cnc2C1 76373,c1(C(=O)NCC2CC3CCC2N3C(=O)CCc2ccoc2)cnc2[nH]cncc1-2 76374,N1(C(c2cc(-c3ccco3)c[nH]2)=O)CCN(C(=O)C(c2ccccc2)F)C2CC12 76375,c1(NC(C2(CC(C)C)CCC2)=O)ccc2oc(CC3CC3)nc2c1 76376,C1(C(C)C)CN(C(=O)C(C)(O)C2CCC2)CCCN1C(=O)CCCC(N)=O 76377,N1(C(c2cccc(C)c2O)=O)CC2CC(C)N(C(C3CCNC(=O)C3)=O)C2C1 76378,CCC(CNC(=O)CC1C=CS(=O)(=O)C1)(CC)NC(=O)C(C)C(C)C 76379,C1(NC(c2cn(C)nc2-c2ccco2)=O)CCCC(NC(=O)C2=CSCS2)CC1 76380,CC(N=c1nc(N(CCCN2CCCC2)C)c2sccc2[nH]1)C(F)F 76381,c1(CC)cccc2c1OCCC2NC(=O)C(N1CCOCC1C1CCCC1)=O 76382,c1(CSCC)ccc(C(=O)NC2(CF)CC(NC(=O)Cc3cnn(C)c3)C2)cc1 76383,O=C(C1COc2ccc(Cl)cc21)NCC1CN(C(c2coc(CO)c2)=O)CC1O 76384,CC(C)CC(C)(C)C(=O)N1CCC1CNC(=O)C=Cc1ccc(F)cc1 76385,C(=O)(CC(C)(CN(C)C)C(F)(F)F)N1CC(F)(CNC(CC=C)=O)C1 76386,CC(C(F)C(=O)N1CCC(CCNC(=O)CCc2nncn2C)CC1)C(F)(F)F 76387,c1(C(c2ccccc2)N(C(N2CCCC2COC)=O)CC)ncccn1 76388,N1(C(c2cc(CC)nn2C)=O)CCC2(CCC(NC(C3(CC(C)C)CC3)=O)C2)C1 76389,C1(N=[N+]=[N-])(C(N(C(C)C)CCF)=O)CCN(C(=O)OC(C)(C)C)C1 76390,C1(F)(CNC(c2c(OC)cccc2)=O)CC2CCC(C1)N2C(C1CCC2CC12)=O 76391,C1(n2cc(NS(C)(=O)=O)nn2)CN(C(=O)C(C)NC(c2ccoc2)=O)CC1O 76392,N1(CC)CCN(CC(N2CCCC2CCCNC(C2(OC)CCSC2)=O)=O)CC1 76393,c1(C(=O)NC(C)CNC(=O)Cn2cc(C3CC3)nn2)cc(Cl)cc(Cl)c1F 76394,C1(C)(CCOC)CCN(C(=O)C(N2CCN(C(C#N)C(C)C)CC2)=O)C1 76395,N#Cc1c(NC(C2CCCN(C(=O)CNc3ccccn3)C2)=O)cc(Br)cc1F 76396,CC1(CNc2cn(CC3CC3)nn2)CCCN(C(C2CC23CCOC3)=O)C1 76397,C1(C(=O)NCCN(C(C)C)C(C2CC2c2ccccc2)=O)CC(S(C)(=O)=O)C1 76398,c1(CN2CC(C(=O)NCCCOC=C)SCC2)c(F)cc(O)cc1F 76399,c1(C(=O)NC2CCN(C(Cc3cccc(C)c3)=O)C23CC3)ccn2ncccc12 76400,Cn1nc(C(=O)NC2(C)CCN(C(C3CC4(C3)CC(C)(C)C4)=O)C2)c2c1CCC2 76401,C1(CNC(c2c(CC)ccs2)=O)CCN(c2ncc(Cl)c(C(C)=O)n2)CC1C 76402,C1(C(N2CCC(C(CC)CC)C2)=O)C=CCN(C(=O)CN(C)C(C)C)C1 76403,c1(CC)onc(-c2cccnc2)c1C(=O)NCC#CCNC(=O)C(C)C#N 76404,C1(NC(=O)CSC(F)(F)F)CCC2(CCN(C(C3CN4CCCN3CC4)=O)C2)C1 76405,C1(CNC(C2N(CC)CC2)=O)CN(C(C2CC2(C)C)=O)CC1C(F)(F)F 76406,N1(C(C2(OC(C)=O)CC2)=O)CCN(C(=O)Cc2csc(CC(C)C)n2)C(C)C1 76407,C1(SCC2CCN(CC=CC(=O)OC)C2)OCCOC1(C)C 76408,CCC(C)(CNC(C1OC2CCC1C2)=O)C(=O)NCc1cscc1C 76409,N1(C(CC2C(C)(C)OCC2)=O)CCC(C(=O)N2CCSCC2)=C(F)C1 76410,C1(NC(C(C)n2cccn2)=O)CCC2(C1)CN(C(C1(C#N)CCCC1)=O)C2 76411,N1(CC)CCOC(C(=O)N(CCCNC(C2(C3CCCO3)CC2)=O)CCO)C1 76412,N1(C(c2cc(OC(F)F)nn2C)=O)CCN(C(c2cccc(OOC)c2)=O)C2CC12.O 76413,c1(N2CCC(NC(c3c(C)n(C)nc3)=O)(CF)C2)ncc2c(c1C#N)CCC2 76414,C(N=c1[nH]c(=NCCC2COCC2O)[nH]c2c1SCC2)c1ccn(CCC)n1 76415,CP(C)(=O)CC(=O)NC1CC(CC(=O)NCc2cc(C(N)=O)co2)C1 76416,CC(=O)C1=C(c2ccc(F)cc2)N(Cc2ncnn2C)C(=S)NC1 76417,C1(NC(Cc2c(C)ccs2)=O)CCN(C(=O)CN2CCC(F)(F)C2)C(C2CC2)C1 76418,Cc1ccccc1CC(CNC(=O)C(C)(C)C1(O)CCNC1)CO 76419,c1(C(=O)NC(C(C(C)C)NC(c2cc(O)cs2)=O)C)ccc2ccn(C)c2c1 76420,C1(NC(C2CCCCC2)=O)CCN(C(C23CCCC2C3)=O)CC1O 76421,C1(C(C)C)CN(C(c2csnn2)=O)CCN1C(=O)C=C1CCC1 76422,Cc1cc(C(=O)NC2(CCNC(=O)C=Cc3cn(C)nn3)CC2)cc(=O)n1C 76423,Cc1noc2nc(C(=O)N(C3CCN(C(=O)C(F)=C4CCC4)C3)CCO)ccc12 76424,C(C(CC(=O)N1CC(C)(C)CC1CNC(c1ncccc1O)=O)C(F)F)N(C)C 76425,C#CCC(O)C(=O)N1CC(F)(CNC(c2ccc(-c3ccccn3)s2)=O)C1 76426,CC1(N2CCCC2)CCCN(C(=NCC(O)Cn2ccnn2)NCC(F)F)C1 76427,CN1CCCC(C)(C(=O)NC2COCCC2NC(=O)CCOCC2CC2)C1 76428,N1(C(C(c2ccccc2)NC(C2=C(C)CC2)=O)=O)CC2CCC2(C)C1 76429,C1(NC(C(Cc2cn[nH]c2)NC(c2n[nH]cc2Cl)=O)=O)C=CCCCC1 76430,c1(C(=O)NCC(CNC(CC=CC=C)=O)O)ccc2cc(CC)ccc2c1 76431,N1(CC)C(=O)COC(C(=O)Nc2ccnc(F)c2OC)C1c1nccn1C 76432,N1(C(COCCOC)=O)CC2(CC(NC(=O)CCSC3CC3)c3nccn32)C1 76433,C1(O)(CC(=O)NC2CCN(C(CCc3scc(C)c3)=O)C2)CCCCCC1 76434,c1(C(C)(C)CC(=O)OCC2OCCCO2)cc(C(F)(F)F)ccn1 76435,CCC(C(=O)NC1CC(F)CN(C(c2cc(C(F)F)cs2)=O)C1)C(C)C 76436,S(=O)(=O)(c1cc(C(N)=O)c(Br)cc1F)N1CCCC(c2nc(C)c(C(=O)O)s2)C1 76437,N1(C(C(CC)(O)c2ccsc2)=O)CCC(NC(=O)CCOC2CCC2)C(F)C1 76438,n1(-c2scc(CC(N3CC(COC(C)=O)C3)=O)n2)nnc2ccccc12 76439,CN1CCCC1C1CCCCN1C(C1CC1C1CC1)C(=O)NCc1cccs1 76440,Cc1ccc(CC(=O)N(C(C)CCNC(c2csc(Br)n2)=O)C)s1 76441,C(=O)(CC(C(F)(F)F)NC(c1cn(C2CC2)nn1)=O)NC(C)Cn1cnnc1 76442,C1(C(=O)NCCC(=C)CNC(c2ccncc2F)=O)C2CCC1(c1cscn1)C2 76443,c1(C(=O)NCC2CN(S(=O)(=O)c3nccs3)CCCO2)ccc2c(c1)CCO2 76444,C(=O)(CC(=O)N1CCC1CC(=O)N(C)CC1CCCCO1)OC 76445,c1(-n2c(C(C3CCC3)O)nc(CCCC)n2)ccc(Br)cc1OC 76446,N1(C(c2ccc(-c3ncc[nH]3)cc2)=O)CC2(CCCN2C(c2coc(Cl)n2)=O)C1 76447,CC(C)CC(O)C(=O)N1CC(=O)CC1C(=O)NCC1(C)CCCS1 76448,N1(CC(=O)NCc2c(C(N3CCC(CCOC)C3)=O)nco2)CCN(C)CC1 76449,c1(C(C)NC(C2C(CNC(C3(SC)CC(=O)C3)=O)CCC2)=O)ccc(C)nc1 76450,N1(C(=O)Cn2cncn2)CCC2(CC1)CC2NC(C1(C2OCCO2)CC1)=O 76451,C12(COC)CC(NC(=O)CCC(F)(F)F)(CN1C(=O)CC(C)NC(N)=O)C2 76452,C1(NC(C2N(CC)CC2)=O)CCCN(c2nccc(-c3ccc(F)cc3)n2)C1C 76453,C1(NC(C2N(CC)CC2)=O)CCC(F)(CNC(c2sccc2SC(F)F)=O)C1 76454,c1(C(=O)NCC(CC)(CC)NC(c2ccnc(C)n2)=O)ccc2nc(S)[nH]c2c1 76455,N1(C(CCC(=O)OC)C)CCCC(C)(C(=O)NCc2ccco2)C1 76456,c1(CC)nocc1C(=O)N(C(C)CN(C(=O)Cc1ccnn1C)C)C 76457,c1(OC)ccc(Br)c(C)c1C(N1CC(C)(CNC(c2oncc2C)=O)C1)=O 76458,C(C)(c1cnn(C)c1)=CC(=O)NCC(CNC(c1ccc(SCC)nc1)=O)C 76459,CC(C)C(O)C(C)C(=O)NCCC(C)(C)NC(c1ccncc1Br)=O 76460,CC1(C)COC(=O)C1NC(=O)CNC(=O)CCC(N)=O 76461,C(=O)(C1=C(Cl)CC1)NCC1(C(N)=O)CN(C(=O)Cc2ccc(F)cn2)C1 76462,Cc1ncc(CCC(=O)NCCC2CC(NC(c3ccccc3C)=O)C2)c(O)n1 76463,Cc1cc(CC(=O)N(CC(C)(C)CNC(C2CCC(C)O2)=O)C)ccc1Cl 76464,c1(C(C)(C)C)nccn2cnnc12.C12C3CN(CC13)C(=O)C=CCSCC(=O)N2 76465,c1(C(=O)NC(CC)CNC(=O)CC2(C)CC2(Cl)Cl)cnn2c(=N)[nH]cnc12 76466,C1(CN(C2CCN(Cc3ccccc3)C2)C)CCCCN1C(=O)CCCC1CC1 76467,C1(O)(CN(C(C2C(C=C)CC2)=O)C)CCCN(C(c2ccc(C)c(OC)c2)=O)C1 76468,N1(C(CC2(C=C)CCC2)=O)CCN(C(=O)C(F)(F)C2CCCC2)CC1COC 76469,N1(C(c2nccc(C)c2O)=O)CCN(C(c2ccc(Cl)o2)=O)C(C)C1C 76470,c1(NC(C(C2CCCO2)NC(C(C)OCC=C)=O)=O)cscc1OC 76471,c1(SC)cccc(C(=O)NCCCNC(=O)Cc2cnn(C)c2C)c1[N+](=O)[O-] 76472,c1(C(N2C3CCC(NC(C(CCC)C)=O)(C3)C2)=O)cc2cc(C(=O)OC)sc2s1 76473,N1(C(CC(CC)C(C)C)=O)CC2CN(C(=O)C(C)(C)NS(C)(=O)=O)CC2(C)C1 76474,C(=O)(CCC(CF)CF)NC1CC2CC(NC(=O)C=CCF)C2C1 76475,c1(C(c2ccc(CC(N3CCN(CCN)CC3)=O)cc2)=O)c[nH]c2ccccc12 76476,c1(C(C(=O)NCC2(O)CN(C(C(CC)N(C)C)=O)C2)CC)ccc(F)cc1 76477,CCN=c1[nH]c(C(N2CC(NC(=O)CCN3CCOCC3)C3CC23)=O)cs1 76478,C(=O)(CCC(N)=O)N1C(C(C)NC(c2cnoc2C2CC2)=O)CCC1 76479,c1(C(=O)NC2(CO)CCCN(C(CN(CCOC)C)=O)C2)ccn2cccc2c1 76480,N1(C(c2cc(OC)c(F)cc2)=O)CCc2sc(-c3ccc(C(C)N)cc3)cc2C1 76481,C1(NC(c2ccc(SC)o2)=O)C(C)CN(C(C2CC3C=CC2CC3)=O)CC1C 76482,N1(C(c2nc(C(=O)OC)oc2)=O)CCCCC(NC(=O)Cc2nocc2C)C1 76483,c1(C(N2CC(F)(CNC(C3CCCCO3)=O)C2)=O)cnc(C2CC2)nc1O 76484,CC1(C)CCCC1C(=O)NCC#CCNC(=O)CSc1nnc(S)s1 76485,N1(c2nccc(CC(=O)OC)n2)CCC2(CCOC2)C(CNC(C2CC2(C)C)=O)C1 76486,C#CCCCCCC(=O)NCc1nc(C(N2CCOC(CC)C2)=O)c(C)o1 76487,C1(C(N(CC(C)NC(C2(C)CC(C)(C)C2)=O)C)=O)CC2(CCOC2)C1 76488,N1(C(C2(C(F)(F)F)CCN(C)C2)=O)CCC(NC(=O)Cc2ccco2)C(C)(C)C1 76489,c1(NC)snc(C)c1C(=O)NCC1(C)CCCN1C(C1CC1COC)=O 76490,c1(C(=O)NC2CC(C)(CNC(c3csc(Cl)n3)=O)C2)ncn2c1CCC2 76491,C(=O)(C(CN=[N+]=[N-])NC(=O)C(C)N1CCCC1)NCCc1nc(C)[nH]n1 76492,C=CCCC(C(=O)N1CCC(C(N)=O)CC1)NC(C1CN(C)CCN1C)=O 76493,c1(C(N2C(CCNC(Cc3c(C)nsc3)=O)CCC2)=O)cnc2c(c1)OCCN2 76494,CCC(O)(CNC(=O)C(c1cccnc1)NC(=O)Cn1ccnc1C)CC 76495,CC(CC(=O)N1CCC(NC(=O)CC2CC3(CCC3)C2)C(F)C1)CC(F)(F)F 76496,N1(C(C(C)(C)OC)=O)CCC(NC(C2(C)CC2(Br)Br)=O)C(CO)CC1 76497,C(=O)(C(C)C(O)C(C)C)NC12CC(NC(c3cc(C(C)C)on3)=O)C(OC1)C2 76498,C(=O)(C(C)(O)C(F)(F)F)N1C(CN(C)C(C2(C(F)F)CCC2)=O)CCC1 76499,C(C)(CCCC(=O)NCCCc1nccs1)NC(C(C)NC(CC)(C)C)=O 76500,C1(C(N(CCNC(CCSC)=O)C)=O)CC(Br)(Br)C1 76501,CCC(C)C(O)C(=O)N(C1CCN(C(c2cccnc2OC(C)C)=O)C1)C 76502,C1(NC(c2c(C)nccn2)=O)CCC2(CCCN2C(=O)C2=CCOCC2)CC1 76503,c1(CCC(=O)NCCN2CCC(NC(C3CC4CCC34)=O)CC2)ccccc1O 76504,c1(C(=O)NC2CCC(C)N(C(C3CCCOCC3)=O)C2)cnc2c(c1)COC2 76505,C=C1CCCN(C(=O)CC=CCNC(c2coc(CCC)n2)=O)C1 76506,C12(C(=O)NCc3ccc(CNC(C(C)C)=O)cc3F)CCOC1CCOC2 76507,C(CCN(C)C(c1cccc(N(C)C)c1)=O)(C(C)C)NC(C(COC)N(C)C)=O 76508,c1nnn(C)n1.CCS(=O)(=O)N1CCCC1.C1(=O)C(=O)NCC(C2CC2)N1C 76509,C(CCSC)(CN=c1[nH]c(C)cc(=NCCN(c2ccc(Cl)cn2)C)[nH]1)OCC 76510,NC(=O)CCCCC(=O)N1CCCC(CCNC(c2c[nH]nc2C2CC2)=O)CC1 76511,C1(C(=O)NCCCC2(NC(CCC=C)=O)CC2)CCC(OCCN(C)C)CC1 76512,CC(C)CC(CN=c1[nH]c(C2CC2)nc2[nH]ccc12)NC(C1CC2(CC2)CO1)=O 76513,N#Cc1cc(S(=O)(=O)NC(C2CN(Cc3cnn[nH]3)C2)=O)ccc1Br 76514,C1(O)(CCNC(C(c2cnn(C)c2)OC)=O)CCCN(C(C2CCCN2C)=O)C1 76515,CC1CCC(C(=O)NCCCN(C(=O)CC2CC3CCC2CC3)C)CC1C 76516,C12(C(=O)NCC(CN(C(C=CCC)=O)C)(C)C)CCCC1C2(F)F 76517,C(=O)(C(C)(C)CCCOC)N(CCNC(c1nn(CC)nc1C)=O)C1CC1 76518,C1(CC(=O)N(CCCC(C)C)C)CC2(C1)CN(C(=O)C(O)C1CCC1)C2 76519,Cc1noc(C)c1S(=O)(=O)N(c1c(N)ccc(F)c1C)CC(=O)NCCC1=CCCCC1 76520,c1(C(=O)NCC(=O)NCC(=O)NCC(=O)NC2CC2C)ccccc1F 76521,c1(CCC(=O)NCC(n2cc(CCN(C)CC)nn2)C)nnc(C)n1C 76522,c1(C(=O)NC2CN(C(c3scc(C)c3)=O)C3C2C3)c(F)ccc2n[nH]cc12 76523,C#CCC(C)(CC)C(=O)NC1CN(C(=O)C=Cc2c[nH]c(=N)c(C)c2)CC1O 76524,C(=O)(C1=CNS(=O)(=O)N=C1C)NC1C(CNC(C2(COC)CCCCO2)=O)CC1 76525,N1(C(C(C2CCCC2)OC)=O)CCCC(C)(C)C1CNC(c1cc(CO)on1)=O 76526,N#Cc1cccc(C(N2CC3CC(NC(=O)Cc4cccnc4O)C3C2)=O)c1 76527,c1(C(=O)NC2CN(C(Cc3cn(C)nn3)=O)CC2F)cc(N=S(C)(C)=O)ccn1 76528,Cc1ccc(C(=O)NCC2CC(NC(=O)C(C)Cn3ccnc3)C2)cc1Br 76529,C1(CNC(CC2C(C)CCC2)=O)CC2(CC2)CN1C(=O)Cn1ncc(O)nc1=O 76530,c1(CC(=O)NCC#CCNC(C2C(C(=O)NCC#C)C2)=O)ccncc1C 76531,C1(CNC(c2[nH]c(=N)sc2)c2nnnn2CC2CCCO2)CCCC2(CCC2)O1 76532,C1(C(=O)NC(CCSC)C)CN(C(c2ccnnc2)=O)CC1(F)F 76533,c1(C(=O)NCC(C)CN(C)C(c2nccn2C)=O)ccc(F)c2c1CCC2 76534,c1(C(c2nnnn2CCCSC)NC(CC)CC)ccc(CSC)s1 76535,Cc1n[nH]c2cnc(C(=O)NC(C(C)NC(=O)C(C)(C)C(C)(F)F)C(C)C)cc12 76536,N1(C(C(CC)(C)C)=O)CCC2(C=C(C(=O)N3CC(N4CCCC4)C3)C2)C1 76537,c1(C(N2CCC3(CC3C(N3CC(O)(CO)C3)=O)C2)=O)cccc2c1CCC2 76538,C#CCC(C(=O)OC)NC(=O)CCC1CCCN1C(c1cnn(CC2CC2)c1)=O 76539,C1(NC(C2CC(OC)C(OC)C2)=O)CC2CCC1N2C(=O)CCSC 76540,C(=O)(C(CNC(c1ncccc1N)=O)C(C)(C)C)N(C)Cc1ccco1 76541,C1(CCNC(c2ncn(CC)c2)=O)CSCCN1C(=O)C(C)CCO 76542,c1(C(N(CCCCN(C(CC(C)c2ccccc2)=O)C)C)=O)ccncc1Cl 76543,Cc1cc(CCC(=O)NCCCCNC(=O)C(C)c2ccsc2)ccc1Cl 76544,O(P(C)(=O)CCCOC(=O)C(C)CCN(C)C)CC 76545,c1(C(N2CC3=C(CN(C(=O)C=C4CCC4)C3)C2)=O)csc2c(Cl)cccc12 76546,CC(CNC(=O)CCC(C)O)C(C)C(=O)O 76547,Cc1ccc(COC(F)(F)F)cc1.C12CN(CCN1)C(=O)NCCCNC2=O 76548,C1(C)(C(=O)NC(C)(C)CF)C=CCN1C(=O)CC1OCCO1 76549,S(=O)(=O)(CC(=O)N1CCCC1CCCNC(C1CC2(CSC2)C1)=O)N(CC)CC 76550,O=C(N=c1[nH]nc2ccc(Br)cn12)N1CCc2cc([N+](=O)[O-])ccc21 76551,C1(CNC(c2cccc(C(N)=O)n2)=O)CCCCN(C(c2cc[nH]n2)=O)C1 76552,C1(CNC(COCC(=O)OC)=O)C(C)CCCN1C(c1cccc(OC)c1Cl)=O 76553,C1(NC(C(CC)N(CC)CC)=O)CN(C(=O)CC2COCCOC2)CCC1F 76554,C1(C(N(C2CCN(C(=O)CC3CCCCC3O)CC2)CC)=O)CCNC(=O)C1 76555,c1(OC)ccc(C=CC(=O)NC2CC2CNC(=O)Cn2cc(CO)nn2)cc1Cl 76556,c1(C(=O)NC2C3(CC(NC(CC(COC)C)=O)C3)C2)cncc(P(C)(C)=O)c1 76557,c1(C(=O)NCC2CCCCC2F)c[nH]cc(Br)c1=O 76558,N#Cc1ccc(F)c(C(N2CC(NC(c3cnn4c3OCC4)=O)C3CC23)=O)c1 76559,C(CC)(C(=O)N1CCC(c2ccon2)C1)=CCCC.C(C1=NOCC1)CC=O 76560,C1(NC(C(C)C2CCCO2)=O)C2CC(NC(=O)CP(C)(C)=O)CC12 76561,N1(C(C2CC(C#N)(O)C2)=O)CC2CC(NC(=O)C(c3ccc(F)cc3)F)CC2C1 76562,C1(NC(C2(C)ON=C(C)C2)=O)CN(C(C2CCS2(=O)=O)=O)C2CCCCC12 76563,c1(C(N2CC(NC(C#CC(C)(C)C)=O)CC2(C)C)=O)cc2ccc(F)cc2s1 76564,c1(C(N2C(C)CCC(NC(COCC)=O)C2)=O)ccc2c(c1)NC(=O)CC2 76565,N1(CC)CCC(O)C(C(=O)Nc2n(Cc3ccc(F)c(C(=O)OC)c3)ncc2)C1 76566,C=CC(C)(CCOC)C(=O)N1CCOC(CN(C)C(C2CC(O)(C#N)C2)=O)C1 76567,C1(NC(c2c(OCC)scc2)=O)CC(C)N(C(C2CC3(CCC3)C2)=O)C1 76568,c1(C(N2CC(NC(C(C3CCCOC3)OC)=O)(CF)C2)=O)ccc(N(C)C)cn1 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76727,C1(CNC(C2(CC)CC2)=O)(CNC(=O)CC2CCC(C)C2)CCCC1.CCO 76728,c1(CC)cc(C(=O)NCC(C)(C)OCCNC(=O)C(C)CC2CCCC2)c(C)o1 76729,C1(C(=O)NC2CN(C(=O)NC(C)C(C)N)C2)Cc2ccccc2S1.C(C)(C)(C)O 76730,N1(C(C(C)=C(C)C)=O)C(C(=O)NCc2ccc(O)nc2)CCC1C(C)C 76731,N1(C(C2CCN(S(C)(=O)=O)C2)=O)CCOCC(C)(C(C2CC2)NC(=O)CSC)C1 76732,Cc1ccc(F)cc1C(=O)NCC1(CNC(=O)C2CC2)CCCC1 76733,c1(C(=O)NC(C2CCOC2)C2CC2)cc(C2CC2)ncn1 76734,N1(C(CSc2c(NC(C)=O)nc(C)nc2Cl)=O)CC2(CC(C(F)(F)F)CO2)C1 76735,CC1CC=C(C(=O)NC(C(=O)NCCc2ncon2)c2cccs2)CC1 76736,C(=O)(CCC[N+](=O)[O-])N1CC(N2CCN(C(C3C(=C)CC3)=O)CC2)C1 76737,C1(CNC(CC(CN(C)C)O)=O)C2CCCC1N(C(c1csc3nnsc13)=O)C2 76738,C(=O)(CCCCc1cnc[nH]1)NC(C)CC(C)NC(C1CCC(F)C1)=O 76739,C(=O)(C1=NNC(=O)CC1)N1CCC(C2C(NC(CC(CCC)C)=O)CCO2)CC1 76740,C(C(C)C(=O)NC(c1cn(C)nn1)C(=O)NCCC1(O)CCOC1)SC 76741,Cc1cccc(OC(C)C(=O)NCCCNC(C2(C3CCCO3)CCCC2)=O)c1 76742,C1(O)(c2nc(Cn3cc(CCCC(C)O)nn3)[nH]n2)CCNCC1 76743,CC1CN(C(=O)CC2(NC(c3ccc(F)s3)=O)CCCCC2)CC1F 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76762,C(=O)(C1=CC(O)C(NC(C2(CCF)CCC2)=O)C1)Nc1c(CC)noc1 76763,N1(C(CC(C)CNC(c2ccc3c(c2)CC3)=O)=O)CCC2(C=CCO2)C1 76764,C1(C2N(C(c3c(C)noc3)=O)CCC2)CCCN(C(=O)CC(=O)N(C)C)C1 76765,N1(C(c2c(CC)con2)=O)CC2CCC1C(CNC(C13CC(OC)C1C3)=O)C2 76766,C#Cc1ccc(C)c(NC(C2CCN(C(C3CCS(=O)(=O)N3)=O)CC2O)=O)c1 76767,c1(C(N2CC3(CCCN3C(C3CC34CCCC4)=O)C2)=O)ccc2cnoc2c1 76768,c1(C(N(CC(C)N(C(c2c(CC)noc2)=O)C)C)=O)nc(C)c(C)nc1O 76769,N1(C(CNS(C)(=O)=O)=O)CC2CC1CN2C(=O)CSc1ccccc1 76770,N1(C2CCN(C(CCCC)=O)C2)CCC(NC(c2nccc(C)n2)=O)CC1 76771,C1(CC)CN(C(=O)C(N2CCC(C(=O)NCCN(C)C)CC2)=O)C(C)CO1 76772,c1(C(N2C(C(=O)NC(C)C(=O)NCC(C)C)(CC)CCC2)=O)cn(C)c(=O)cn1 76773,C=CCCCCCCC(=O)NCc1nnn(C)c1C(=O)NCC(O)CN(C)C 76774,Cc1cc(C(N2CCC(CO)(Nc3ccncn3)CC2)=O)c(C)cc1Br 76775,C(=O)(C(O)CCCNC(=O)CC12CCCC1C2)NC1CCC(C)(C)C1 76776,c1(C(=O)NCC2(CCNC(C3(F)CC3(Cl)Cl)=O)CC2)ccc2c(O)ncnc2c1 76777,c1(C(=O)NC2CCC(N(C(c3c(C)snc3)=O)C)C2)ccn(C)c(=O)c1 76778,C1(CNC(=O)Cc2ccccc2O)CCC(CNC(C2CC23CC(O)C3)=O)CC1 76779,C1(O)(CN(C(c2cnc(C(C)C)[nH]2)=O)C)CCCN(C(C2CC23CC(O)C3)=O)C1 76780,C1(C(N(C(C)CNC(c2ccc(CN(C)C)o2)=O)CC)=O)CC2(C)CC1CO2 76781,CCCC(C(=O)NCC1CC(C)N(C(C2CCC(C(N)=O)C2)=O)C1)NC(N)=O 76782,c1(C(N2CCCC(NC(c3nccc(C)c3)=O)C2C)=O)cnc2c(F)cccn12 76783,C=CCCC(C)(c1nnnn1C(C)(C)C)NCC1(C=C)CCC1 76784,N1(C(c2c(CC)nccn2)=O)CC(NC(C2CCSC2)=O)C(C)(C)C1 76785,N1(C(C(CC)c2ccccc2)=O)CC2C(NC(c3noc(C)c3Br)=O)C2C1 76786,Cc1cc(Br)ccc1C(=O)NCCC1CN(C(=O)C(C)NC(N)=O)C1 76787,c1(C(N2CC(C(F)(F)F)C2)=O)csc(C2CCCN2C(=O)CCl)n1 76788,C1(NC(COCCOCC)=O)CCC2(CC1)CCN(C(c1cn(C3CC3)nn1)=O)C2 76789,C1(CC(=O)NCCCN(C)C(C23CC(O)C2C3)=O)CCC=CCC1 76790,c12c(ccc(C)c1C)[nH]c(=O)c(=O)[nH]2.c1(OCCC)ccc(C(=O)OC)c(C)c1 76791,CCC(C)(COC)C(=O)NCC(C)N(C(=O)Cc1cccc(C(N)=O)c1)C 76792,c1(CC(=O)NCC(CN(C(C2COCCN2C)=O)CC)(C)C)cccc(Cl)c1 76793,C12(NC(C3CCCC(F)C3)=O)CC1CN(C(=O)CNC(c1cccnc1)=O)C2 76794,c1(N(CCCN(C(=O)C(F)(F)c2ccccn2)C)C)cc(C(N)=O)ncn1 76795,C(=O)(C1CCCc2ncccc21)NCC1OCCN(C(C2(C(N)=O)CCC2)=O)C1 76796,c1(OC)c(CNC(CCC=C(C)C)c2nnnn2C)ccc2ccccc12 76797,C(=O)(CC1=NNC(=O)C1)N(CC(C)NC(C1(c2ccccc2)CC=CC1)=O)C 76798,c1(CNC(c2ccc(Cl)c(C)c2)c2n(C(CC)(C)C)nnn2)ccc(F)c(Cl)c1 76799,C1(C(C)CC(=O)NC(C2CCCCC2)CCO)CCCN(C(=O)OC(C)(C)C)C1 76800,C(CCC(=O)NC(C)CN(C(c1csc(CNC(C)=O)n1)=O)CC)OCC 76801,C#CC1(C(=O)NCC2CC(=C)C2)CN(C(=O)Cn2cnc(C(N)=O)n2)C1 76802,Cc1oc(C#N)cc1C(N1CCC(NC(c2ccn(C)c2)=O)C(CO)C1)=O 76803,[N-]=[N+]=NC1CC(C(=O)NCCc2cccs2)N(C(=O)CC2CCC2)C1 76804,C(=O)(CC(C)CC(C)(C)C)N1CCC(N(C(CCC#CC)=O)CC2CC2)C1 76805,C(=O)(C1CCCc2scnc21)N(CC(O)Cc1cnc[nH]1)CCOC 76806,C1(OCC(=O)N(CC(CC)NC(=O)CC2CCN(C)CC2)C)CCN(C)CC1 76807,c1(NC(COc2cccc(C)c2Br)=O)cccc(S(C)(=O)=O)c1 76808,N1(C(CCOCCN(C)C)=O)CC2CC(C1)N(C(c1ccc(N(C)C)nn1)=O)C2 76809,C(=O)(N=c1cc2n([nH]1)CCOC2)C1CC2N(C(c3ccc(C)cc3)=O)C(CC2)C1 76810,c1(N2CCC(NC(C3C(=C)C3)=O)C2(C)C)nc(C(=O)NC)nc(Cl)c1C 76811,Cn1nnc2cc(NC(C3CC3NCc3cccc(C(=O)O)c3)=O)ccc12 76812,C1(CC(=O)NC(c2cscn2)C)CC2(CC2)CN1C(c1cccc(F)c1N)=O 76813,c1(C(=O)NC2CCC(CNC(c3csnn3)=O)C2)c(F)ccc2n[nH]cc12 76814,CCC(C)CCCCC(=O)N1CCN(C(=O)C2=CC(C)C2)CC(C)(F)C1 76815,c1(C(=O)NC2(CF)CCN(C(CCC(=O)OC)=O)C2)cc(C)cc(Br)c1F 76816,c1(C(N2CC(NC(=O)CC3CC3)(Cc3ccncc3)C2)=O)ncccc1Cl 76817,C(CC)(C(C)(F)F)NC(C1N(C(C2N(CC)CC2)=O)CC=C1)=O 76818,CC1=NOC(C(N2CC(NC(=O)C(C)COc3ccccc3)C2)=O)C1 76819,N1(C(c2c(OC)scc2)=O)CC2CC2C1.C(=O)CC(F)(F)F.C12CC1NC2=O 76820,C1(NC(CCc2cc(C)no2)=O)COCCC1NC(c1cn(C(C)C)cn1)=O 76821,C1(C)(C(=O)NCC(CN(C(c2c(C)n[nH]c2C)=O)C)C)CC(C2CC2)=NO1 76822,C12N(CCCC1(C)C)C2=O.C(=O)(C(O)Cn1cc(-c2nccs2)nn1)OCC 76823,c1(OC(C)C(=O)NC(C)(C)CNC(=O)CS(C)(=O)=O)ccc(F)cc1Cl 76824,c1(C(N2CCC(NC(CC(C)F)=O)C(O)C2)=O)ccc(Br)c(F)c1N 76825,c1(C(=O)NCC(CC(C)C)NC(CNS(CC)(=O)=O)=O)ccc(O)c2ccccc12 76826,N1(C(Cc2nc(NC(=O)Nc3ccnc(O)c3)sc2)=O)CCCC(F)(CO)C1 76827,C1(CCC)CN(C(c2c(N)sc(C)c2C)=O)CCN1C(c1cnn2c1OCC2)=O 76828,N1(C(C(=Cc2cccs2)C)=O)CCC(C2CC2)C1CNC(c1ccoc1C)=O 76829,C1(C(N2CC3C(CO)C3C2)=O)C(O)CCN1C(c1cccnn1)=O 76830,Cc1nc2nccc(N(C(C)CNC(c3cc(F)cnc3O)=O)C)n2n1 76831,c1(OC)cc(C)cnc1C(=O)NCC1(OC)CN(C(C2CCC2)=O)C1 76832,CCC(C#N)C(=O)NCC(C)C(=O)NCCc1cnco1 76833,n1(C2(OC)CCOCC2)cc(C#N)c(=NC(=O)c2cc3c(cc2Br)OCO3)[nH]1 76834,C12(C(=O)NC3(CNC(c4ccc(OC)c(N)n4)=O)CCC3)C3CC(CC13)C2(F)F 76835,c1(C(N2CC(C(C)NC(C(C=CC)O)=O)C2)=O)coc2cc(C)c(C)cc12 76836,N1(C(CC2(OCC)CCC2)=O)CC(C(=O)NC2(CO)CCCCCC2)C2(CC2)C1 76837,c1(NCc2c(C)noc2)cccc(N2CCN(C(=O)Cc3cnn(C)c3)CC2)c1 76838,N1(C(c2ncccc2Br)=O)CCC2CCN(C(C3(F)CCOC3)=O)C2C1 76839,Cc1ncccc1CN1CCOCC1CNC(c1cn(C)cn1)=O 76840,c1(-c2ccc(OC)cc2)ccc(NC(=O)Nc2cnccc2Br)cc1F 76841,CC(C)C(C)C(=O)NN(S(N)(=O)=O)C1CC1.C12CCC1OC1CN(C1)C(=O)C2 76842,C12CCN(C1)C(=O)C(C)N(C)C2.N1(C(=O)NCC=O)CCOCC1.CO 76843,C1(C(=O)N(C)CC2CCN(C)C2)(COC)CC(C)(C)C1.C12CC(C1)CC(=O)N2 76844,N1(C(c2ccccn2)=O)CCN(C(=O)CCc2ccc(F)cc2F)C(C2CC2)C1 76845,CC1(C(N2CC(NC(C3CCCN3C(N)=O)=O)C(CO)C2)=O)CC2C=CC1C2 76846,CCC(C(=O)NC1(C)CCN(C(=O)CCN2CCC(C)CC2)CC1)C(C)C 76847,c1(C(N2CCC(C(C)NC(CSCC)=O)CC2)=O)cccc(I)c1F 76848,CC(O)C(CO)NC(=O)COC1CN(C(=O)C(O)c2ccco2)C1 76849,N1(C(CCC(CC)C)=O)CC=C(CC(=O)N2CCN3CCCC3C2)CC1 76850,CC1CC(=O)NCC1C(N1CC2(CCN2C(c2nscc2Br)=O)C1)=O 76851,C(=O)(C(CCOC)OC)NCC(C(=O)N(CC#C)CC1CC1)N(C)C 76852,Cn1ccc2c(C3(C(=O)NC4CC(c5cc(CF)on5)C4)CC3)cccc12 76853,Cn1cncc1C(=O)NC1(C)CC(NC(=O)CC2CCCOC2)C1 76854,c1(C(=O)NCC2N(C(C(C3CCOC3)OCC)=O)CC2)csc(C(N)=O)n1 76855,c1(OC)csc(C(=O)NCCCC(C)NC(=O)CC2(C)CC2)c1 76856,C1(C)(CCNC(CC2(OC)CCC2)=O)CCN(C(C2CC3C=CC2O3)=O)C1 76857,N1(C(c2c(C)ncc(Br)c2)=O)CCC2CN(C(c3cc(Cl)cc(Cl)c3)=O)CC2C1 76858,C1(NC(c2[nH]n(C)c(=O)n2)=O)C(CNC(c2cc(CF)on2)=O)CCC12CCC2 76859,CCC(C)C(C(=O)NC(CC(N)=O)C(=O)NCC(C1CC1)SC)N(C)C 76860,c1(CN(C(CC)CC)C)cn(CC(O)Cc2ccccc2)nn1 76861,n1(CC)cc(C(N2CCCCC2C(C(C)C)NC(=O)CCCNC(C)=O)=O)c(C)n1 76862,CC(C)CC(CNc1ccnn1C1CCCCO1)C(=O)OC(C)(C)C 76863,c12nc(Cl)ccc1CN2.c1(NC(Cc2cccc(CC)c2)=O)cc(C)nc(F)c1 76864,Cc1cc(C)c(C(=O)NCCC(O)CNC(=O)Cc2ncccc2C)c(S)n1 76865,c1(N(C2CCN(C(C3CCCCC3O)=O)C2)C)ncccc1S(C)(=O)=O 76866,N1(C(C(CC)C)=O)CCC2(CC2C(N2CCCC2(C)C(=O)OCC)=O)C1 76867,c1(C(=O)NC2(CNC(=O)C(N3CC4CCC3C4)=O)CCC2)cccc2c1CCC2=O 76868,N1(C(c2ccc(CC)s2)=O)CC(NC(=O)C(C)(O)C2CC2)C(SC)C1 76869,N1(C(=O)NC(C)C(C)(C)O)CC2CC(N)C(C2)C1 76870,CCCCC(CC)C(=O)N(CCNC(=O)Cn1cc(C2CC2)cn1)CCOCC 76871,N1(C(C2C(NC(=O)CCc3ccncc3)C=CCC2)=O)CCCC2(CCCO2)C1 76872,c1(CC)cc(C(N2CCC(C(F)F)(CNC(C3CCCC(O)C3)=O)C2)=O)ncn1 76873,C1(C(N2CCC(OCC=C)CC2)=O)CN(C(c2cccc(C)c2N)=O)C(C)(C)C1 76874,c1(COCCC2C(C)CC2)cncc(NC(c2cocn2)=O)c1 76875,N1(C(=O)CN2CC=CC2)CC2CC(C(N3CCC34CC(COC)C4)=O)(C2)C1 76876,C(=O)(C(C)C(O)C(C)C)N1CCN(C(C(CCC)(C)C)=O)CC1CF 76877,C1(CN(C(C2(NC(CN(C(=O)OC)C)=O)CCC2)=O)C)CCOC1C 76878,C(=O)(C#CC1CCOCC1)N(C)CC1(NC(C2C(CC)OCC2)=O)CC1 76879,N1(C(C(CC)CC)=O)CC2OCCN(C(=O)CC3CCCC34CC4)C2C1 76880,CCCCCCCc1cn(C(C)C(=O)N(C)CCOCCO)nn1 76881,CN1CCN(N(CC2CC2)CCCCN(C)C)CC1c1cccs1 76882,CC(C)CC(C(=O)N1CC2CC2C1C(N1CCCC(C)C1)=O)N(C)C 76883,c1(CC)noc(C)c1C(=O)NC1CCN(C(C23CC(C)C2C3)=O)C1C 76884,O=C1CCN(c2csc([N+](=O)[O-])c2)C(=O)N1Cc1nnnn1C1CC1 76885,c1(OC)ccc(C(N2C3CN(C(C4(C#N)CC4)=O)CC23)=O)c(Br)n1 76886,C=CCC(C)C(=O)NCC1CCN1C(=O)C=Cc1nc[nH]n1 76887,c1(OC)cccc(C(N2CCOC(CC(=O)NC3CCCC(OC)C3)C2)=O)n1 76888,C(=O)(CCCCC(=O)NCC1(OC)CN(C(C2CC2c2ccccc2)=O)C1)NC 76889,c1(C(=O)NCC(CCNC(=O)CCc2ccoc2)OC)cc(F)c(F)cc1O 76890,c1(OC)ccc(CN(C)C(c2ccc(I)cn2)=O)cc1OC 76891,c1(C(=O)NCC2N(c3ncc(COC)nc3)CCC2)ccc(OC)c(OC)c1Cl 76892,c1(C(=O)NC2C(CNC(c3c[nH]c(C(F)(F)F)c3)=O)COC2)ccc(O)cn1 76893,c1(C(=O)NC2CN(C(C(COC)(F)F)=O)CC(C)C2)ccc2nc[nH]c2n1 76894,C1(O)(CNC(C)=O)CCCN(C(=O)C(C)(C(C)C)OC2(C(=O)OCC)CCC2)C1 76895,C1(C(=O)NCc2c(C(=O)NC3(CC(C)C)CC3)cco2)CC(=O)CCO1 76896,N1(C(CC2C(C)C2(F)F)=O)CC2CC2(NC(c2ocnc2C(F)(F)F)=O)C1 76897,C1(NC(=O)C=Cc2cc[nH]c2)CN(C(=O)C#CC2CCCCC2)C2(CCOC2)C1 76898,c1(C(N2C(C3CCCN(C(C(=O)N(C)C)=O)C3)CCCC2)=O)cc([N+](=O)[O-])n[nH]1 76899,c1(C(CC(=O)NC(c2cnccn2)C)NC(C2(F)CCCC2)=O)ccc(F)cc1 76900,c1(CC(N2CC3C(CNC(C4C5COCC45)=O)(C3)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 76901,c1(N(C(C(=O)N(C)C(c2c(C)ncs2)c2ccccc2)C)C(C)C)ccc(F)cc1 76902,C(=O)(CCCCCOC)N1CCC(CC)C1C(=O)N(C1CCC1C)C 76903,CN1CC(NC(=O)C#CCNC(c2cc[nH]c2C2CC2)=O)C(C)(C)C1 76904,CCC(C)(CCC(C)C)C(=O)N1CC2CC(C1)N2C(=O)OC(C(=O)C(Cl)(Cl)Cl)=O 76905,N1(C(CSCC)=O)CCCC(CC)(NC(=O)C(C)NC(=O)C(C)(C)C)C1 76906,c1(C(N2CC(COCCOC)(NC(c3ccoc3C)=O)C2)=O)ccc(OC)cc1 76907,C1(CNC(=O)Cc2ccoc2)CCCN(C(c2ccccc2-n2cncn2)=O)C1 76908,C1(NC(c2c(OCC)oc(C)n2)=O)(CO)CCCN(C(c2cc(C)ns2)=O)C1 76909,c1(OC)nc(C)ccc1OC(c1cnn(C2CC2)c1)=O.C12CCC(C1)C(=O)NCC2 76910,C1(C(N(CCCn2cc(CCC3CCCO3)nn2)C)=O)CCC(=O)N1C1CC1 76911,C(=O)(CC(C)CC(C)C)N(C(CNC(C(CC)N1CCCC1=O)=O)C1CC1)C 76912,c1(N(C)Cc2c(C)nc[nH]2)nnc(CC2CCCOC2)n1Cc1cccnc1 76913,C1(NC(CC2(CSC)CC2)=O)CC(CO)N(C(c2nc(O)sc2C)=O)C1 76914,c1(C(=O)NCCCCN(C(C2C(OC)CCCC2)=O)C)cnc2cc(C)[nH]c2c1 76915,N1(C(C(C)NC(=O)C(C)(C)C)=O)CC(C2(NC(C3CN4CCN3CC4)=O)CC2)C1 76916,N1(C(COCC(C)C)=O)CCCC(C2CN(C(c3cccnc3Br)=O)C2)C1 76917,c1(CC(=O)NCC(CC)NC(c2cc3nccnc3[nH]2)=O)ccc2ncsc2c1 76918,c1(CC(=O)NC2CCCN(C(CC=C)=O)C2)coc2cc(O)ccc12 76919,Cc1nnc(=NCC(CC(C)C)NC(=O)CC(C(F)F)n2cccn2)[nH]c1C 76920,c1(CC(=O)NC2CC(F)(CNC(C(C)N3CCC3)=O)C2)cncc2ccccc12 76921,C1(C(N2C(CNC(C(C)(C)C3CCCC3)=O)CC(O)C2)=O)CC2(C1)CC2(F)F 76922,C(=O)(C(C1=CCCSC1)N1CCC(NC(=O)OCC)C1C)NCC=C 76923,N1(C(CCCSC)=O)CCC(C(F)CNC(=O)CN2CC(=O)NC2=O)CC1 76924,C(C(C)(O)CC(=O)N1CC(C2CCCCN2C(C2(C3CCCO3)CC2)=O)C1)OC 76925,C(CC)(C(C)(F)F)NC(C(CC1CCC1)NC(CNC(CC)=O)=O)=O 76926,c1(CNC(C2(F)CN(C(C(CC)=CC)=O)C2)=O)c(F)cccc1F 76927,C1(C(=O)NC(C2(C(N3CCOC4CC34)=O)CC2)C)CC(C)(C)CN1C 76928,CCCCC(CNC(c1ccsc1C(F)(F)F)=O)NC(c1cnsc1C)=O 76929,CC(CN(C)C)CC(=O)NC1(C(=O)NC(C)CCc2cn[nH]c2)CCC1 76930,N1(C(Cc2c(OC)cccc2)=O)CC(OCc2ccccc2)C(C)(C)C1 76931,N1(C(c2n[nH]c(C)c2O)=O)CCC(CO)(NC(C2CC(=O)CO2)=O)CC1 76932,C(C(CC(C)C)C(=O)Nc1ccc(C)cc1CC)NC(C1C(OCC)CC1)=O 76933,CCC(C(=O)N(CCC(N1CCC(CO)C(O)C1)=O)C1CC1)C(C)C 76934,c1(C(=O)NCC(c2ccc(O)cc2)NC(c2ccsc2)=O)ccn2nncc2c1 76935,N1(C(CCN(CCC)C)=O)CCCCC1CCC(=O)NCCCc1cccnc1 76936,C12(C(N3C(CC(=O)NC)CC3)=O)CC(CCO1)N(C(=O)CCn1cccn1)C2 76937,c1(C(N2CCC(C)(CCNC(c3c(C)occ3)=O)C2)=O)cc(F)ccc1N 76938,C1(C(=O)NC(CC)Cn2cncn2)CCOCCN1C(=O)CC1COCC(C)O1 76939,N1(C(Cc2c(C)ccs2)=O)CC2(CCCN(C(C3CCOC3C(F)(F)F)=O)C2)C1 76940,C1(CC(=O)NCc2cn(CC#C)nc2)CCCN(C(c2cc(Cl)cn2C)=O)C1 76941,C1(OC)CC(CNC(=O)CC(C)(C)N(C(=O)CC23CCCC2C3)C)C1(C)C 76942,C1(CC=C)(NC(c2cc(OCC)ccn2)=O)CCN(C(C2CCC(F)(F)C2)=O)C1 76943,Cc1noc(C(F)F)c1C(=O)NCCC1CCN(C(=O)C=Cc2cc[nH]n2)C1 76944,C(CC(C)(C)CC(=O)NCC(C1CCN(C(=O)CCCCCF)CC1)F)OC 76945,c1(C(=O)NCC(CNC(=O)CSCC(=O)N(C)C)OC)ccc(C2CCCO2)s1 76946,c1(OC)cnc(C(=O)NC2CCC2NC(C2(C)CC3CC3C2)=O)c(F)c1 76947,S(=O)(=O)(c1ccc(NCCCc2ccccn2)cc1Br)N(C)CC1CCN(C)C1 76948,CCCCC(O)CC(=O)NC(Cn1ccnn1)C(=O)NC1CC(N(C)C)C1 76949,C=CC(C)C(=O)NCC(c1ccccc1)NC(c1nn[nH]c1C1CC1)=O 76950,C1(C(=O)NCCCC(=O)OC)Cc2ccccc2CN1C(C1CC1C1CC1)=O 76951,C12(NC(C(COC)C)=O)CCCC1N(c1ncnc(O)c1Br)CC2 76952,C(=O)(C#CC(C)(C)CNC(C1C2CCC(F)C12)=O)N(C1COC(C)(C)C1)C 76953,c1(C(=O)NCc2cc3c(cc2)NC(C)CC3)cncc(C2=CCNCC2)n1 76954,Cc1nc(=N)[nH]cc1C(N1CCC(CNC(c2ccc(F)o2)=O)C1(C)C)=O 76955,C(=O)(C1COc2cc(C)c(C)cc21)N1CC(c2cn(C(CC)C)nn2)C1 76956,C=CC1(C(=O)NC2C(C)CCC2C)CCN(C(=O)CCn2ccc(C)n2)C1 76957,c1(OCC(C)C)cccc(C(=O)NC2CN(C(=O)C(=O)NCC(F)F)C3CC23)c1 76958,CC1(C)CN(C(=O)Cc2cccc(Cl)c2)CC1NC(c1c[nH]c(Br)c1)=O 76959,c1(COCCNC(=O)CC2CCC(Nc3ccccn3)CC2)cccc(F)c1I 76960,c1(CN(C(c2ccc(C#N)nc2)C(=O)NCCOC)C)ccc(S(C)(=O)=O)cc1 76961,C1(C)(NC(CC(CC)C2CCC2)=O)CCCN(C(=O)CC(C)(C)O)C1 76962,C1(C#N)(COC)CN(C(=O)C(C)CNC(=O)C(c2cccnc2)O)C1 76963,c1(NCC(CC)(C)NC2CC(C(N)=O)C2)cc(NC)ncn1 76964,CCC(C)(NC(Cc1nccs1)CO)CO.C(C)(C)(C)OC=O 76965,c1(CN2CC(NC(C3CCCO3)=O)C(F)(F)CC2)ccc(F)c2ccoc12 76966,CCC(C)C(O)CC(=O)NC1(CCC(N2CCC(F)(C#N)C2)=O)CCC1 76967,N1(C(C(C(C)NC(C(CCC)N(C)C)=O)C)=O)CCC(C2(C)CC2)CC1 76968,C(=O)(C1COc2ccccc21)N1CCC(N2CCN(C(c3cn[nH]c3)=O)CC2)C1 76969,C1(O)(CNC(CC2N(C)CCOC2)=O)CCN(C(=O)C=Cc2nnn(C)n2)CC1 76970,n1(C(C)(C)C)nc(C(=O)NCC2CC(NC(C3CCCSC3)=O)C2)cc1C1CC1 76971,C1(NC(C(c2cccs2)NC(c2ccsc2C(F)(F)F)=O)=O)CCN(CCF)C1 76972,N1(C(C2C(C(=O)OC)C2)=O)CCC(NC(=O)Nc2cccnc2I)CC1 76973,C1(NC(c2ccc(COC)cc2)=O)CCCCN(CCCSc2ccc(C)cc2Cl)C1 76974,CCCCCCCCCC(=O)N1CCCC12CN(c1cc(C)nc(C)n1)C2 76975,CC1CN(C(=O)Cc2cccc([N+](=O)[O-])c2)c2ncc(Br)cc2O1 76976,C(C(C)(O)CC(=O)N1CCC(NC(C2(c3cccc(OC)c3)CC2)=O)C1)OC 76977,C1(CS(C)(=O)=O)CN(C(c2c(F)cccc2Cl)=O)CCN1C(=O)C(O)C1CCC1 76978,c1(C(=O)OC)ccc(C(=O)NC2CC2NC(=O)C=C2CCC2)cc1 76979,C1(CC)(NC(=O)C(C(C)C)NC(N)=O)CCCN(C(C2CC3(CCOC3)C2)=O)C1 76980,c1(C(=O)NC23CC(NC(Cn4c(=O)ccc(C)n4)=O)(C2)C3)ccn2ccccc12 76981,N1(C(C2N(C(C)=O)CCCC2)=O)CC2CCC1C2NC(=O)C=Cc1cccnc1 76982,c1(C(C(=O)N(CCSCC(C)C)C)N(C(=O)OC(C)(C)C)C2CC2)ccc(Br)s1 76983,Cc1ccc(Cl)c(NC(N2CCC(n3nccn3)CC2)=O)c1Cl 76984,C1(OC)CC(CNC(c2cc(N3CCCCC3)ncn2)=O)N(C(=O)C(C)CO)C1 76985,c1(Oc2ccc(C(C(=O)NC3CCC3)N(C)CC#N)cc2)ccc(Cl)cc1F 76986,c1(CC(=O)NCCN(C(c2c(CC)con2)=O)C)cc(Br)cnc1F 76987,c1(NC(=O)NCC2CC(NC(=O)OC(C)(C)C)C2)cc[nH]c1CCO 76988,N1(C(c2cc(C)oc2)=O)CCC(NC(c2cc(O)no2)=O)C1(C)C 76989,C(CCCCCNC(c1cccc(-c2ccco2)c1)=O)NC(C1(C)CC1)=O 76990,C(=O)(C(COC)OC)N(CC(N1CC(CC=C)C1)=O)CCC 76991,c1(NC(c2c(-c3c(C)cccc3)cccn2)=O)cc(Br)ccc1Cl 76992,N1(C(C=CC(C)NC(c2cnc(CC)o2)=O)=O)Cc2ccc(C#N)cc2C1 76993,N1(C(C(CN(C)C)NC(C(C(CC)CC)OC)=O)=O)CCC2(CCC2)C(O)C1 76994,C(C)(CNC(c1cc(F)c[nH]1)=O)(C(C)C)NC(Cc1nc(C(C)OCC)sc1)=O 76995,C1(C(=O)NCC2C(C(=O)NC(c3c(C)nccc3)C)CC2)CCCC(C#N)C1 76996,c1(C(=O)NCCN2CC(C)N(C(=O)OC(C)(C)C)CC2)cccn2nncc12 76997,c1(C(N2C(CN(C(C(C)n3cncn3)=O)C)COCC2)=O)ncc2[nH]ncc2n1 76998,N1(C(c2cccc(OC)c2N)=O)CCN(C(=O)CCc2cncnc2)CC(O)C1 76999,c1(CC)ncc2c(n1)COC2.N12CCCN(CC1)CC2 77000,C1(C(N2CC(CCOC)C2)=O)CC2CC1CN(C(=O)C(F)C(C)C)C2 77001,c1(C(N2CCC(CCNC(C3OCCN(C)C3)=O)C2)=O)ccc(N)c(Cl)n1 77002,Cc1cc(C(=O)NCC2CCN2C(C2(C)CC2(Cl)Cl)=O)ccc1C(C)C 77003,CC(CC1CCCCC1)C(c1nnnn1C)NCC(C1CC(F)(F)C1)(C)C 77004,N1(C(C2C(CCOC)C2)=O)CC(NC(=O)Cn2ncc(Cl)c2C)C(C)(C)C1 77005,c1(SCC(N2Cc3c(cc(C(=O)OC)s3)C2)=O)cc2ccccc2c(O)n1 77006,C(=O)(C1=NOC(C)C1)N1CC(O)(CNC(COCCCCCC)=O)C1 77007,c1(C(C)(C(=O)NCC(F)CO)NC(C)C2CC2)c(F)cc(Br)cc1F 77008,CCCC(C(=O)N1CCCC1C1(CNC(=O)Cc2ccsc2Cl)CC1)N(C)C 77009,C(=O)(C(F)(F)C(O)C1CC1)NC1CCC(CNC(=O)CC2(O)CCCC2)C1 77010,C1(NC(C2CC3(CCC3)CO2)=O)CCCCC1N=c1[nH]c(Cl)nc(C2CC2)c1F 77011,C(=O)(C(O)C(F)(F)F)NC(CCCCNC(c1c(C)[nH]nc1Cl)=O)C 77012,N1(CC)CCCC2C1CCCN2Cc1ccc(-c2ccccc2C=O)s1 77013,C12(CC1(C)C)C(=O)N2.c1(CNC(C2(CC)CC2)=O)ccc(CO)o1 77014,C#CCC(C(=O)N1CCC(CCC)C1)NC(=O)CCc1cccnc1 77015,C(C(=O)NC1CC(CCNC(C2CC2(Cl)Cl)=O)C1)(C(C)(C)C)NC(C)=O 77016,CCCCCC(=O)N(CCCNC(=O)CN1CCN(C)CC1)CCO 77017,C1(CNC(CC(C=C)(C)C)=O)CN(C(c2ccc(C)nc2N)=O)C2CCN1C2 77018,Cc1cc(C(=O)NC2CCC2CNC(=O)C#CC(OC(C)C)OC(C)C)ncn1 77019,C(=O)(C1=NNC(=O)CC1)N1CC2C(CNC(c3c(C)ncnc3)=O)(C2)C1 77020,N1(C(C2CC(C(F)F)(OC)C2)=O)CCC2(CC1)CC(C)N(C(=O)C(C)SC)C2 77021,N1(C(c2nc(C)oc2C)=O)CCn2c(CNC(c3cc(C#N)c[nH]3)=O)nnc2C1 77022,C1(CC)C(C(=O)NCC(C)(CNC(C2CCC(=O)N2C)=O)OC)CCN1C 77023,c1(CN2C(CNC(c3ccc(OC)c(I)c3)=O)CCC2)ccc2c(c1)OCCO2 77024,CC1CC(CCNC(c2nocc2Cl)=O)CCN1C(c1ccn(C2CC2)n1)=O 77025,C1(NC(C2(N(C)C)CC2)=O)CCCC1NC(=O)CCOCC(F)F 77026,C#CC(CC)(CC)NC(C1(CC=C)CCN(C(C2CCS(=O)CC2)=O)C1)=O 77027,C(=O)(C#CC1CCCC(CC)C1)N1CCCC1=O.C(C)(C)(C)N(C)C(C)=O.CCO 77028,N1(C(C2(NC(c3cc(C)sc3)=O)CCSC2)=O)CCCC2(CC(O)C2)C1 77029,C1(C2(N)CCC2)(C(=O)NCC(c2cnn(C3CC3)c2)(C)C)CCC1 77030,n1(CC(=O)NCC(CCOC)NC(c2cncc(N)n2)=O)nnc2c1CCCC2 77031,CCCS(=O)(=O)NC(C)C(=O)N(CCCNC(=O)C(F)CC1CC1)C1CC1 77032,c1(C(C)(C)NC(c2c(C)[nH]nc2Cl)c2nnnn2C(C)C)n[nH]c2c(F)cccc12 77033,c1(N(CC(CNC(C)=O)(C)C)C)[nH]c(=NC2CSC2)nc2c1ncn2C 77034,C1(OC)CN(C(c2ccc(O)c(Cl)n2)=O)C(C)(CNC(c2cccc(N)c2)=O)C1 77035,c1(NC2C(O)CN(Cc3cccc(F)c3Cl)C2)ncnc2c(F)cccc12 77036,CCCCC(C)C(=O)N1CCN(C(C2CC(C)(C)C2C(F)(F)F)=O)CC1C 77037,O=C(CCCC(=O)NC(=O)CNC(C1CCCCC1)=O)NC1CNC(=O)O1 77038,C1(C(=O)NCC(C(=O)NC2CC(C=C)C2)OC)CC2CCCC2C1 77039,O=NN1CCCCC1C(N1CCC(NC(=O)COC2CCC2)C1)=O 77040,C1(C(=O)NCC(C)C(C)(F)F)CC12CCN(C(C1COCC1C(N)=O)=O)C2 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77128,C1(CC(=O)N(C(CNC(C2COC(=O)N2C)=O)C2CC2)C)CCCCC1(C)C 77129,C1(CNC(C2CN(CCOC)C(=O)C2)=O)(CO)CCN(C(=O)CSC)CC1 77130,C=CC(C)C(C)C(=O)N1CC(OCCNC(c2ccc(N(C)CCC)nc2)=O)C1 77131,C1(C(NOC(C(=O)OC)(C)C)=O)COCCN(C(C2CC3C=CC2CC3)=O)C1 77132,C1(C)(CNC(C2(OCC)CC2)=O)COCCN(C(c2cc(C(C)=O)on2)=O)C1 77133,CCC(CC)CC(F)C(=O)NC1CC=C(C(=O)N(C2CCNC2=O)C)C1 77134,C1(CNC(COCCC)=O)CN(C(=O)C=Cc2cccc(O)c2)CC(C)(C)O1 77135,C(=O)(CCC(=O)C(C)(C)C)N1C(C(=O)NCCN(C(C)C)C(C)C)CNC(=O)C1 77136,c1(CNC(C(C)Oc2ccc(-c3ncco3)cc2)=O)cc(Br)c2ccccc2c1 77137,C(=O)(C(C(=O)NC1CCCN(C(=O)C(N2CCSCC2)C)CC1)C(C)C)OCC 77138,C1(O)(CNC(C2(COCC)CCC2)=O)CCCN(C(=O)C=CCF)CC1 77139,N1(CC(C)(N(CCCC)CC=C)C2CC2)CCCC(C)C1C 77140,C1(CSC)CCN(CC(=O)N(CCN2CCOCC2)CC2CCCC2(C)C)CC1 77141,CC(C)C(F)(F)CC(=O)NC1CN(C(c2c(F)cncc2Cl)=O)CC1(C)C 77142,CC(C(C)C(=O)N1CC2(CC2)C1)NC(=O)C=CC(=O)NC1CC1 77143,Cc1ccc(COCC(=O)NCC2(F)CC(NC(=O)CSc3nc[nH]n3)C2)cc1 77144,Cn1[nH]c(C(=O)NC(C)(C)CNC(C2CCN(CC(F)F)CC2)=O)nc1=O 77145,C1(C(=O)NCC2(CC(=O)Nc3cn(CC#C)nc3)CC2)CC(=O)OC1(C)C 77146,c1(C(=O)NC(C)CN(C)C(C2CCC3CC3C2)=O)c[nH]c2cccc(F)c12 77147,c1(COC2CC(NC(C3CCC(C(=O)OC)C3)=O)C2)nc(O)ccc1C.C1CO1 77148,c1(OC(c2[nH]c(C)nc2C)=O)cccc(C2CC2NC2CCN(C(C)=O)CC2)c1 77149,c1(OC)ccc(CN(c2ccccc2)C(=O)CNc2ncc(F)cn2)cc1 77150,c1(C(N2CCN(C(=O)CSc3ccccn3)C3CC23)=O)cc2c(cn1)OCCO2 77151,C1(NC(=O)CCCF)CN(C(C23CCCC2CCC3)=O)CC2(CCC2)C1 77152,N1(C(C(CC)n2cncn2)=O)CC2(CCCN(C(=O)C(F)CC(C)(C)C)C2)C1 77153,C1(NC(=O)COCc2ccccc2)CCC(NC(c2sccc2Br)=O)CC1 77154,C1(F)(C(N2CC(F)(CNC(Cc3cc(C)[nH]n3)=O)C2)=O)CCN(C)CC1 77155,c1(C(N2CCCC(C(C)NC(=O)C(F)=CC3CC3)C2)=O)[nH]nc([N+](=O)[O-])c1Cl 77156,c1(C(=O)NCCCCN(C(C=C(C)C(F)F)=O)C)cnc2ccccc2c1C 77157,c1(C(N(C2CCN(C(c3nccn3C)=O)CC2)CC)=O)nc[nH]c2ncc(Br)c1-2 77158,N1(C(C=C(C)C)=O)CCC2CN(C(=O)CCc3cnccc3C)CC2CC1 77159,c1(C(=O)NC)ccc(C(N2CCC(NC3CC3(F)C(=O)OC)C2(C)C)=O)c(C)c1 77160,c1(NC(C2CC(CNC(=O)OCc3ccccc3)C2)=O)ncc([N+](=O)[O-])cc1F 77161,CC1CN(C(C23CC4CC2C3C4)=O)CC(C)CN1C(=O)CC(=O)OC(C)(C)C 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77356,c1(NC(c2ccc(C3(O)C(C)(C)COCC3)cc2F)=O)cccc(P(C)(C)=O)c1 77357,C(=O)(CCCC(C)(C)C#N)N1C2(C(N(CC(CC)O)C)=O)CC(C1)C2 77358,C(C1(C)OCCc2ccccc21)NC(NC(C1CN(C)CCO1)C)=NC 77359,N1(C(c2cc(C)on2)=O)CCCC(N(C(=O)CCCOc2ccccc2F)C)C1 77360,c1(C2(C#N)CC2)ccc(Cl)c(C(N2CCCC(c3nc(C4CC4)no3)C2)=O)c1 77361,N1(C(C(CC)CO)=O)CCN(C(c2cccc(Cl)c2N)=O)CC1C(C)C 77362,CC(C)CCC(C(=O)NCC1(O)CC(CO)C1)NC(=O)CCc1csnn1 77363,C(=O)(C1=CC2C=CC(C1)C2)N1CC(NC(C(C=C)C)=O)C(OC)C1 77364,c1(C(N(CCC(C)=O)C)=O)ccc(-c2cn(CCCCCO)nn2)o1 77365,c1(C(=O)OC)cc(C(N2CC(NC(=O)CN=S(C)(C)=O)CC(F)C2)=O)cc(C)c1 77366,S(=O)(=O)(c1ccc2nc(N3CC4CC=CCC4C3)sc2c1)N1CC2C(C)(CC2)C1 77367,N1(C(C2(NC(c3c(C)n(C)nn3)=O)CC2C)=O)CCOCC(O)C1 77368,Cc1c(N)ccc(C(N2CCC(=CCNC(C3CCCC3(F)F)=O)CC2)=O)c1C 77369,Cc1nc(C(=O)NCC(N2CCN(C(=O)C(C(C)C)NC=O)CC2)=O)ccc1C#N 77370,C1(CCC(N2CCC(CN(C)C(C3(F)CC3)=O)C2)=O)CC(C)(C)CO1 77371,N1(C(C(C(=O)OC)OC)=O)CCCC2(CNC(=O)CC(C)CC(C)C)CCCC12 77372,CC1(C)CC(NC(N2CCOCC2c2nc[nH]n2)=O)c2cccc(Br)c2O1 77373,c1(C(N2CCC(NC(C3(C)CCC(OC)CC3)=O)C2)=O)cc(C)n(C)c(=O)c1 77374,CCCC(CC(=O)NCc1c[nH]nc1C1CCC1)NC(=O)OC(C)(C)C 77375,c1(C(N(C2(CNC(C(CC(C)C)(C)O)=O)CC2)C)=O)ccc2c(c1)C=CS2(=O)=O 77376,N1(C(C(C(C)C)NC(N)=O)=O)CCOCC1(C)C 77377,c1(C(N(CCC)CCNC(=O)C(CC)C(F)(F)F)=O)ccc([N+](=O)[O-])c(C)c1 77378,c1(-c2c(SC(F)F)cccc2)nc(-c2cncc(Br)c2)nn1CCn1cccn1 77379,C12(NC(CCN(CCCO)C(C)=O)=O)CCC(C1)OC2C 77380,C1(NC(C(CC)C(C)C)=O)C2CCCN(c3cc(Cl)ncn3)C2C1(C)C 77381,CC(O)C(C)(C)C(=O)N1CC2CC1(C(=O)NCCCn1cnnc1)C2 77382,c1(COC)ccc(C(=O)NC2CC(CNC(C3CCC(=O)C3)=O)C2)cc1F 77383,C1(CNC(Cc2nc(C)oc2)=O)CCC(C)CN1C(c1cnc(C(F)(F)F)s1)=O 77384,C=CC(C)(O)CC(=O)N(CCC(=O)N1CCC(CSC)C1)OC 77385,c1(C(=O)NC2CCC(CNC(C3C=CCC3)=O)CC2)c[nH]c2nc(Br)ccc12 77386,c1(C(N(CCCCCNC(C2CCC(C)CC2)=O)C(C)C)=O)cc([N+](=O)[O-])ccn1 77387,c1(OC(C(N2C(CCC(=O)OC)CCCC2)=O)C)cnc2[nH]cnc2c1 77388,C(=O)(C(C(CC)CC)OC)N1C(C)(C(N2C(CC)CCCC2)=O)CCC1 77389,C1(NCC2(COC)CCCCC2)CCC12CCCO2 77390,c1(C(=O)NC2(CF)CCN(C(CCC(=O)OC)=O)C2)coc2c(F)cc(F)cc12 77391,CCCS(=O)(=O)N1CCCC1C(=O)NC12CC(C(C)C)(C1)C2.C12CC1CNC2=O 77392,c1(CNC(C2C=CCC2)=O)nc(CNC(C2(CC3CCC3)CCC2)=O)cc(O)n1 77393,CCS(=O)(=O)c1ccccc1CCNC(CC1CC(NC(C2CC2F)=O)C1)=O 77394,C1(C(=O)NC2(CCCCNC(c3n(CC)cnn3)=O)CC2)CCC(=O)CC1C 77395,N1(C(CNC(=O)NC)=O)CCC(C2CC2)C1CNC(c1n[nH]c2c1CCOC2)=O 77396,C1(C)(CC)C=C(C(=O)NC2(CCNC(=O)C(N3CCOCC3)C)CC2)C1 77397,n1(C(C)C)nccc1C(C(=O)NCc1ccco1)N(C)C(C1CCCO1)C 77398,c1(C(=O)NCC(CC=C)NC(c2cc(C#N)c[nH]2)=O)nc2sccn2c1C 77399,N1(C(c2cc(COC)oc2C)=O)CC2(CC2)CC1CNC(C1CC1OC)=O 77400,N1(C(C(C=C)O)=O)CCC2CCCN(C(=O)C=CCOc3ccc(F)cc3)C2C1 77401,CC1CC(=O)NC(C(=O)NCC(O)CNC(=O)C(=O)NCCC(N)=O)C1 77402,c1(CNC(=O)CC2CCCO2)cccnc1CNC(C1CCC(F)(F)C1)=O 77403,CCCC(CN1CCN(c2cc(C(=O)OC(C)(C)C)cc(F)c2)CC1)C(=O)OC 77404,CCC(C)(C)C(O)C(=O)NCC1CN(C(C2(C(N)=O)CC2)=O)CC1(C)C 77405,CN1CCn2nc(C(NC3CCc4ccc(CC(=O)O)cc43)=O)cc2S1(=O)=O 77406,c1(C(N(CC(CC)NC(C2CC2C(C)(F)F)=O)CC)=O)ncc(Br)cc1F 77407,CC1CC(CC(=O)NCCCn2cnnc2)CN1C(c1ccnc(CO)c1)=O 77408,c1(C(=O)NC2CC(CCNC(C3CC=CCC3)=O)C2)cc2c(nc1O)CCC2 77409,c1(C(=O)NCCN(CCC)C(C2(C)CC2C)=O)ccc(-n2ccnc2)c(C)c1 77410,Cc1n[nH]c(=NCC2(CCC(c3ccco3)=O)CC2)o1 77411,C(=O)(C1OCCn2ccnc21)N1CCC(CN(C)C(c2ccc3c(c2)CC3)=O)C1 77412,CCCCC(CNC(=O)CCC(C)=O)NC(c1csc(C)c1)=O 77413,c1(N(c2ccc(C)cc2)Cc2nc(CC)sc2)nc2ccccn2c1[N+](=O)[O-] 77414,N=c1nc(C2CC2)[nH]c(=NC2CCN(C(=O)CCNc3ncccn3)CC2)[nH]1 77415,C1(C(=O)NCCN(C)C(c2c[nH]cc(F)c2=O)=O)CC2CCCC2C1 77416,C1(C(=O)NCCn2cc(CNC(C(C(C)C)C)=O)nn2)CCCCNC1=O 77417,Cc1cc(Cl)cc(Cl)c1OCC(N1CCC(C(C)NC(C2CC(C)C2)=O)C1)=O 77418,C1(C)(CNC(=O)OC(C)(C)C)CCN(C(c2cc(N)c(O)nn2)=O)CC1 77419,C(=O)(CCC(C)(C)F)N1CCC(OC2CCN(C(c3ccn(C)c3)=O)CC2)C1 77420,c1(C(=O)NC2(C)CN(C(c3ccc(CO)cc3)=O)C2)ccc(N)c(O)c1 77421,c1(OC)ccc(-c2nncn2C(C)(C)C)c(F)c1.N12CCOC(C1)NC2=O 77422,CCC(CC)C(c1nnnn1Cc1cccs1)NCC1COCCC1C 77423,N1(C(C(=O)NC2C(C(=O)OC)CN(C(C)C)C2)=O)CCCCC(C)C1 77424,Cc1cc(C(N2CC(NC(c3cc(Cl)ccc3N)=O)CC(F)C2)=O)c(Cl)cc1F 77425,CCCC(C(=O)N1CCC(NC(=O)COC2CN(C(C)=O)C2)C1)NC(C)=O 77426,C1(CC=C)(C(=O)N(C(C(N)=O)C2CC2)C)CN(C(=O)CCc2cccnc2)C1 77427,C1(=O)C(N(C)C)CN1.C1(CC(=O)N(CCO)CC)OCCCOC1 77428,C1(=CC(=O)NCCN(C(C(c2c(F)cccc2F)OC)=O)C)CCC(C)(C)CC1 77429,c1(COCCCCCC)ccc(C)c(NC(CCC(=O)OC)=O)c1 77430,C1(CCC=C)(C(=O)NC(CCCC)c2ccccc2)CN(C(=O)C2CC2)C1 77431,c1(OCC)cc(C(=O)NC2(CNC(C3CCC3(C)C)=O)CC2)on1 77432,c1(NC)ccccc1NC(=O)C(CC1CC1)NC(c1cn(C(C)C)cn1)=O 77433,N1(C(C(C)SCC)=O)CCC2CN(C(c3cnc4cccnc4c3)=O)CC2CC1 77434,CC(C(F)F)=CC(N1CCC1CNC(=O)COCCOCCO)=O 77435,c1(CNC(c2cnn(C)c2C)c2n(C(CC)C)nnn2)cc(F)ncc1C 77436,C(=O)(C(C)S(C)(=O)=O)NC(CN(C(C=C(CCC)C)=O)C)C 77437,c1(OC)ccc(CN(C)C(C2CCCN2Cc2ccccc2)=O)cc1O 77438,CN1CCN(C(=O)CC2CC2(C)C)CC1C(=O)NCC1(C)NC(=O)NC1=O 77439,c1(OCCC(=O)NCCCCN(C(=O)CC2CCCN2C)C)ccccc1F 77440,N1(C(C(C)CC2CCCC2)=O)CCC(N(C(=O)CC(C2CC2)C2CC2)CCO)CC1 77441,N1(C(C(C=C)(F)F)=O)CC(CN(C)C(c2ccc(CC(C)C)nc2)=O)C2(CC2)C1 77442,C(=O)(CCC(=O)NCC(=O)NCC1CCCCC1OC)NCCC 77443,C1(CC#C)(C(=O)NCCC(O)CNC(=O)Cn2cc(Cl)c(C)n2)CC=CCC1 77444,c1(C(=O)NC2CC(N(C(c3cc(C(CC)C)no3)=O)C)C2)cc(C#N)c[nH]1 77445,c1(C(=O)NC(CNC(c2ccc(C)o2)=O)C2CCC2)cc(N)ccc1[N+](=O)[O-] 77446,C(=O)(CC(C)(C)CNC(=O)C(CC(C)C)OC)NC1(C(=O)OC)CC1C 77447,c1(C(C(=O)NCCCOC)N(CC=C)CC=C)cccc(Cl)c1 77448,CC1C(NC(C2CCCCCC2)=O)CCN1C(=O)C(c1cccc(Cl)c1)C 77449,N1(C(C2(SC)CCOCC2)=O)CCC2(CC1)CCN(C(=O)Cc1n[nH]c(C)n1)C2 77450,N1(C(=O)OC(C)(C)C)CCC(CNC(C(F)(F)F)C2CCCO2)C1 77451,CC(C)CC(C)C(=O)OCCC1(CCCNCc2ccc(Cl)cc2Cl)CCCC1 77452,N1(C(COc2ccn(C)n2)=O)CC2CC1(C(N1CCOCC1C1CC1)=O)C2 77453,c1(CCC(=O)NCC2(CF)CCNC2)cc(Br)sc1Br 77454,c1(C(=O)NCCOCCNC(C2C(SC)CCC2)=O)c(C)nc(C)n1O 77455,C1(CNC(C(C)SC)=O)N(C(=O)CCn2cccn2)CCC1(C)C 77456,c1(N(C(C2C(NC(CCC(=O)OCC)=O)C2)=O)C)cccc(O)c1.COC 77457,c1(C(=O)NCC(CN(C(C2CC2F)=O)CC)(C)C)ncccc1Br 77458,C1(C(N2CC(CNC(=O)Cc3csnn3)C2)=O)(CN2CCC2)CC(F)(F)C1 77459,c1(C(=O)NC(c2ccc(F)cc2)C)cc(F)cc(F)c1 77460,C1(CNC(=O)COCC2CCOC2)CC2CCC(C1)N2C(=O)C1=CCCC1 77461,Cc1ccc(O)c(C(=O)N(CCCOCCNC(=O)CNC=O)C)c1 77462,c1(CC)nn(C)c(Cl)c1C(=O)NCCCC1(NC(c2cccc(C#N)c2)=O)CC1 77463,N1(C(c2c(C)n(C)nn2)=O)CC(CNC(c2nccn2C)=O)CC(C)(C)C1 77464,C1(NC(c2ccc(C(C)=O)[nH]2)=O)CCN(C(=O)Cc2cccc(C)c2Cl)C(C)C1 77465,c1(C(N2CC(C)N(C(C3CCc4n[nH]cc4C3)=O)CC2)=O)cc2n(n1)CCCO2 77466,NS(=O)(=O)c1ccc(C(=O)NC2CCCC23CN(C(=O)Cc2cnns2)C3)o1 77467,Cc1nn(CCO)cc1C(N1CCOC(C2CN(C(=O)CCC3CCC3)C2)C1)=O 77468,c1(C(N(CCn2cc(CCc3nn[nH]n3)nn2)CC)=O)ccc(F)c(Cl)c1F 77469,n1(CCC(N2CC(CNC(c3ccc(OC)s3)=O)C2)=O)ccc(O)nc1=O 77470,C1(CN(C(=O)Cc2cn(C)nc2Cl)C)CCN(C(=O)CN2CC(C)(C)C2)CC1 77471,c1(C(N2C(C)CNCCC2)=O)nc(=O)c2c(Br)c[nH]c2[nH]1 77472,C(=O)(CCC(=O)NC1COCC1NC(c1cnc(C(N)=O)s1)=O)N(C(C)C)C 77473,C1(CNC(CSCC#C)=O)CN(C(c2cccc(F)c2CC)=O)CCC1(C)C 77474,c1(N2CCC(CCOC)(NC(c3cc(C#N)c[nH]3)=O)C2)ncnc(C)c1F 77475,N1(C(CN2CCCC(CC)C2)=O)CC=C(CNC(=O)CSN2CCCC2=O)CC1 77476,CCC(CNC(c1ncccc1F)=O)(CC)C(=O)NC1CC1C(C)C 77477,N1(C(CC)=O)CCOC2(CCC(NC(c3cc(C#N)ccc3C)=O)CC2)C1 77478,CC1CN(CCCNC(=O)CCC(=O)NC)CC(C)O1.C(c1ncc[nH]1)=CC=O 77479,C1(CC)CN(C(c2cn(CC)nn2)=O)CCC1NC(C1(C)CCN(C)CC1)=O 77480,N(C(=NCCF)NC1CC2(C1)CC(C(N)=O)C2)CC(C)(C)O 77481,c1(NC(C)=O)cccc(C(N2CC3CC3(CNS(=O)(=O)CCCl)C2)=O)c1 77482,c1(N2CCC(CC=C)(NC(=O)CN3CCOCC3)C2)ncnc2c1CCC2 77483,N1(C(C=Cc2ccc(C)c(Cl)c2)=O)CCCC12CCN(C(c1ccc(C)s1)=O)C2 77484,C1(C(=O)NCCOC)CC(=O)NC(C)C1.C=C1CC2(C1)C(=O)N2C 77485,c1(OC)ccc(C(=O)OCC2=CCCOC2)cc1[N+](=O)[O-] 77486,C(=O)(C1CCCn2c(Br)cnc21)N1CC(CNC(=O)NC2CC(CC)C2)C1 77487,Cc1cc(N2CCN(C(C3CCCC4(CC4)C3)=O)CCC2C)n2ncc(C)c2n1 77488,C1(O)(COC)CCN(C(=O)C(C2CN(C(=O)C(C)(F)c3ccon3)C2)OCC)C1 77489,N1(C(C2C(CNC(CCOC(C)=O)=O)CC2)=O)C2CCC1CC(CO)C2 77490,C1(OC)CC(NC(=O)C2=CSCS2)C12CCN(C(=O)C(C)(C)C(F)F)CC2 77491,c1(CC(=O)N(CCCNC(c2nc(C)sc2C)=O)C(C)C)cc(F)ccc1Cl 77492,C(=O)(C(C)(O)C(C)C)NCCSCC(=O)NC(c1nn[nH]n1)CC 77493,c1(OC)ccccc1C(CNC(C=CC=O)=O)N.C1(C(=O)NC2CC2)CC1C 77494,O=C(CC(=O)c1ccccc1)NC1CC1NC(=O)C(c1ccccc1)O 77495,C1(N(C(=O)Cn2ccsc2=N)C)CCCN(C(=O)CC2CCCCCO2)CC1 77496,C1(OC)CCCN(C(C2CC(O)CN2C(c2ncncc2N)=O)=O)CC1 77497,c1(C(N2CCCC(CNC(C34CCOCC3C4)=O)C2)=O)nc(O)nc(O)c1F 77498,C1(C(=O)NC2CC(CCNC(C(C)C3CCOC3)=O)C2)CC2C=CC1CC2 77499,Cc1ccc(C(=O)NC(C)(C)CC2CCN(C(C3(O)CC3(C)C)=O)CC2)nc1 77500,n1(CC)cnc2[nH]c(=NCC3CCCC3O)nc(N3CCCC(COC)C3)c12 77501,N1(C(C2CCC(C(F)(F)F)O2)=O)CCOC(c2n[nH]c(-c3ccccc3)n2)C1 77502,C1(NC(c2ccc(C(C)=O)cn2)=O)CCC(C)N(C(C2CCOC2)=O)C1 77503,C1(C(=O)NCCn2ncc(C)c2)CCCN(C(c2scnc2C)=O)C1 77504,N1(C(C(=O)Nc2cc(OC)cc(OCC)c2)=O)CC2CCCN2CC1C(C)C 77505,C1(C(N2CCC(CF)(NC(c3cnco3)=O)C2)=O)(CC)CCNC1=O 77506,c1(CN(C(c2nc(C)sc2)=O)C(C)C)cccc(NC(=O)C(C)C2CC2)c1 77507,c1(SC(C)COC(C)(C)C)cccc([N+](=O)[O-])c1.C1(C)CCC(=O)N1 77508,c1(OCC(=O)NCC(c2c(C)noc2C)N(C)C)cc(Cl)cc(Cl)c1 77509,N1(C(COCCCCC)=O)CCN(C(C2CNC(=O)N2)=O)C(C2CCC2)C1 77510,c1(CNC(C(CO)NC(CC2CCC(=O)NC2)=O)=O)cc(O)ccc1F 77511,CCCC(CCCNC(=O)Cc1csc(C)n1)NC(=O)COCc1cc(C)on1 77512,C#CCC(C(=O)NN1CCCC1C(=O)NCCc1cn[nH]c1)C1CC1 77513,c1(C(N2C(C(=O)NCCCN(C)C)CC(F)(F)C2)=O)cc(O)c(O)c(O)c1 77514,C1(NC(c2c(C)scc2)=O)C2CCN(C(c3ccc(N4CCC4)nc3)=O)CCC12 77515,C12(CNC(c3ccccc3F)=O)CCC(CC1)N(C(C1NC(=O)C3CC13)=O)C2 77516,c1(C(=O)NCC2C=CCN2C(=O)C=CBr)c[nH]c2ccc([N+](=O)[O-])cc12 77517,N1(C(C(CC)(F)F)=O)CCCC2(CCCN2C(C2CN(C)CC2C(F)(F)F)=O)C1 77518,C1(NC(CCCCOC)=O)CC2CCC1N2C(=O)C(C)Cc1cccc(Cl)c1 77519,C#CC1(OCC(=O)N(C)CC2CCN(C(=O)CC3(C(F)(F)F)CC3)C2)COC1 77520,C(N=c1cccc(S(=O)(=O)NC2CCC=C2Br)[nH]1)C1CC(C)(C)OC1 77521,C=CC1(C(=O)NOCC2CCC2)CCN(C(=O)CC2CCCNC2=O)C1 77522,c1(CC(=O)NCC2CCN2C(c2cc(C(F)F)no2)=O)ccccc1Br 77523,c1(C(=O)NC2CCCCN(C(CCC=C)=O)C2)cc(S(N)(=O)=O)c(F)cc1OC 77524,C(=O)(C1=CS(=O)CCC1)NC1CC(N(C)C(C2CC2c2ccccc2)=O)C1 77525,c1(C(=O)NC(C(C)NC(C2C(CCC)C2)=O)(C)C)c[nH]c(C)c(Br)c1=O 77526,N1(C(c2cnc(C)[nH]2)=O)CCN(c2ccc(CNC(C3CCC3)=O)cc2)CC1 77527,c1(N(c2c(CC)n(C(C)(C)C)nc2)C2(CC)CCCC2CC)ccc(F)cc1F 77528,N1(C(c2c(CNC(CCc3ncn(C)c3)=O)c[nH]n2)=O)CCCC(N=[N+]=[N-])CC1 77529,CC1CN(C(C2C3CCC(C3)C2NC(=O)Cc2cccn2C)=O)C(C)(C)C1 77530,C1(C(=O)NCCN(C(C)C)C(c2ccoc2Cl)=O)CCn2c(O)nnc2C1 77531,C1(NC(CC2(N(C)C)CC2)=O)C=CC(CNC(=O)CC2CC(F)C2)C1 77532,C1(CNC(c2n(CC)cnn2)=O)CCCCN1C(C1OCCOC1C(F)(F)F)=O 77533,c1(C(C)N(C(=O)OC(C)(C)C)C)ccc(OC(F)F)nc1.C12CC(C)(C1)NC2=O 77534,C(=O)(C(C)N=c1cnc2c([nH]1)CCN(C(C)=O)C2)N1CCCC(CCOCC)C1 77535,CC(C)(C)C(CC(=O)OCCn1cc(C#N)cn1)NC(C1COCCN1C1CC1)=O 77536,Cc1cc(C(C)(C)C(=O)N2CC(NC(c3cccc(CC#N)c3)=O)C2)ccc1F 77537,CN1CC(C(N2CC(F)(CNC(c3csc(CS(C)(=O)=O)n3)=O)C2)=O)CC1=O 77538,C1(CC(=O)NCC(CC)NC(=O)CCN2CCC(O)CC2)Cc2ccccc2O1 77539,N(C1CCCn2nccc21)C(C1CC2CCCC2N1C(C1CC(O)C1)=O)=O 77540,C1(CNC(COCCC=C)=O)CCC2CN(C(=O)CC3CCSC3)CC12 77541,c1(C(=O)NCCCN(C(CC2(OC)CC2)=O)CCO)cc2cc(Cl)ccc2s1 77542,C1(C(N(CCCNC(CNS(CC)(=O)=O)=O)C)=O)CC(F)(F)C1(F)F 77543,Cc1ccc(OCC(=O)NCC=CCNC(=O)CC2(C(F)(F)F)CNC(=O)C2)cc1 77544,C(N=c1[nH]cc(Br)c2ccc(Br)cc12)C1C(O)COC1 77545,c1(C(=O)NC(c2cccnc2)C(=O)NCc2[nH]nc(C(C)C)n2)ncncc1Cl 77546,C1(CNC(C(N2CCC(O)CC2)C)=O)CCCCC1NC(=O)C(O)C1CCC1 77547,Cc1cc2c(C(N3CC(NC(C4CC4(C)C)=O)C4(CCC4)C3)=O)nccn2n1 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77653,N1(C(c2cc(CNC(c3c(C)ccnc3O)=O)no2)=O)CCC(C2CCOC2)C1 77654,C12(C(=O)NC(C3CCN(C(=O)CC4CCOC4=O)CC3)C)CCOC(C)(C1)C2 77655,c1(N2CCC(OC(C)(C)C)CC2)nc(N2CCC(C3(C)CC3)C2)c2[nH]ccc2n1 77656,C(=O)(C(C)CCC(C)(C)C)N1C(C(=O)NC(CC#C)CC#C)CCOCC1 77657,c1(NC(C)=O)ccc2nccc(N=c3ccc4ccc(Cl)cc4[nH]3)c2c1 77658,C1(C)(CNC(C(CCC)C)=O)CCCN(C(=O)C(CC)C2CCC(=O)N2)C1 77659,c1(NC)ncccc1C(=O)NCC(C1CCCCC1)NC(=O)CSCC(=O)NC 77660,c1(C(N2C(CNC(CCCOC(C)C)=O)CC(O)C2)=O)nccn2ccnc12 77661,n1(CC)ncc2c(NC(=O)C(=O)NCC3CC4COCC34)cc(C3CC3)nc12 77662,c1(C(=O)NCC2N(C(C(C)OC)=O)CCN(C)C2)cccc2ccccc12 77663,Cc1ccc(CC(=O)NC2C=CCN(C(=O)CCOC3COC3)C2)c(F)c1 77664,N1(C(C2(CC)CCN(C(c3nc(C)ncc3Cl)=O)C2)=O)CC(CO)OC(C)C1 77665,CC(C)(F)C(C)(F)C(=O)NCC1(O)CC(CNC(c2cc(O)nc(Cl)c2)=O)C1 77666,c1(CCC)n[nH]cc1C(=O)NC(COC)C(=O)N(CCC(C)(C)O)C 77667,n1(CC)c2nc3cc(ccc13)N(C(Cc1ccc(Cl)cc1)C(C)(C)C)C2.NCC 77668,c1(-n2cc(C3C(OC)CN(C(c4cnncc4N)=O)C3)nn2)ccc(C)c(F)c1 77669,c1(CNC(CCC2CCC(NC(C3CCC(CC)O3)=O)C2)=O)cc(C)nc(O)c1 77670,N1(C(C(C)(C)C2CCN(C(=O)NC3CC3)C2)=O)CCC(C)(CCO)C1 77671,c1(C(=O)NC2CN(C(CC(C)F)=O)CC2(C)C)c2ccccc2nn1C 77672,c1(CC(=O)Nc2cc(C)c(O)cn2)c[nH]c2ccc(C3=CCOC3)cc12 77673,N1(C(C(C(C)SC)O)=O)CCC(C)(CNC(=O)CCN(C2CCCCC2)C)CC1 77674,c1(C(C(=O)NCCOCC)N(C)CCC2CCCCC2)c(Br)cnn1C 77675,Cc1cc(C)n(CC(=O)NC2C=CCN(C(=O)CC3CC(N(C)C)C3)C2)n1 77676,Cn1nc([N+](=O)[O-])cc1C(=O)NCC1CN(C(C2CCS(=O)(=O)CC2)=O)C2CC12 77677,C1(OC)C(NC(=O)C(c2cc(C)cc(Br)c2)N)CC12CCC2 77678,S(=O)(=O)(c1ccc(F)c(C2CC2)c1)N1CCC(c2noc(C)n2)(C(=O)OC)C1 77679,c1(CC(=O)OC)cccc(C(=O)NCCCNC(=O)C(c2ccc(Cl)s2)C)c1 77680,C(=O)(CC(CC(C)C)NC(=O)C(F)(F)CCCC)NCC(CC#C)(C)C 77681,Cc1cc(C)n(CCNC(=O)C(CC2CC2)NC(=O)COc2cnn(C)c2)n1 77682,c1(NC(C2CCN(C(CC)=O)CC2)=O)cc(OC)c(OC)cc1F 77683,Cc1cnc(C(N2CCC(C)(CNC(c3cncc(N)n3)=O)C2)=O)cn1 77684,N12CC3CN(CCC13)C(=O)Cn1cc(cn1)CC2=O.CC(=O)O.C1CC1 77685,N1(C(C(CC)OC)=O)CCCC(C2CCN(C(=O)CC(C)C)CC2)CCC1 77686,c1(C(=O)NCSCCCOCCCC)conc1CC(C)(C)C 77687,C1(CNC(C)=O)CC2(CO1)CN(C(=O)Cc1ccc(NCC(F)F)s1)C2 77688,N1(CC(=O)NC)CCCC1C1CCCCN1C(c1nccnc1SC)=O 77689,C1(CC(=O)NC(C)CCNC(=O)COCCN(C)C)CCC12CCC2 77690,Cc1ncnc(C)c1OCC(=O)NC1CCC(NC(C2CS(=O)(=O)CCO2)=O)C1 77691,N1(C(CC2C(C)CCO2)=O)CCCC(C)(C)C1C(N1CCC2(CC1)N=N2)=O 77692,O=C1C2CC3C1C3C2C(N1CCC1C(=O)NCC1(C2CCC2)CC1)=O.C1CC1 77693,c1(OC)oc(C)nc1C(=O)NC(C)CC(C)NC(c1c[nH]nc1C(C)(C)C)=O 77694,CCC(C)(C#N)C(=O)N(C)CC=CC(N1CCC(C)CC1C)=O 77695,C1(C2CN(C)C2)(N)CC1.c1(CC(=O)C(c2cc(C)no2)=O)ccccc1C1CC1 77696,Cn1cc(Cl)c(C(=O)NC2CC(CNC(=O)Cc3ccc(C4CCC4)cc3)C2)n1 77697,C1(CC(=O)NCC2C(CNC(C(C)CC3CCC3)=O)C2(F)F)CC(O)C12CCC2 77698,C1(C(=O)O)CC(NC2CCN(CC3CCN(c4n(C)nnn4)C3)CC2)CCC1O 77699,Cc1ccc(CN2CCSC(C(=O)Nc3ccc(OCCO)nc3)C2)nc1 77700,N1(C(c2c(OC)csc2)=O)CCC(CO)(CNC(c2cncnc2C2CC2)=O)C1 77701,Cc1[nH]c(-c2ccco2)nc(=O)c1C(=O)NCCN(C(=O)CCCF)C1CC1 77702,c1(C(N(C2CN(C(c3ccc(OC)nc3F)=O)C2)C)=O)c[nH]c2nc(F)ccc12 77703,C(=O)(CCCC(C)CC)N1C(C)CC(NC(C2(CC(=O)OCC)CC2)=O)C1 77704,N(C(=NCCCCC)N1Cc2cnn(CCO)c2C1)C(C#C)(COC)CC 77705,CCCCC(CC)CC(=O)N1CC(C(N2CC3(CCC(=O)O3)C2)=O)C(C2CC2)C1 77706,N1(C(C(C)c2cncs2)=O)CCCC12CCN(C(=O)CC(C)(C)N(C)C)CC2 77707,n1(CC)nc(C)c(C(=O)N)c1C.c1(N(C(COC(F)F)C)C)ncnc(Cl)c1CO 77708,c1(C2(C(=O)NC3CN(C(C=COCC)=O)CC3F)CC2)cn(C)nc1C(F)(F)F 77709,CCC(C)(C)CC(=O)NCC1COC(C(F)(F)F)C1.c12ccc(F)c(c1)CN2 77710,c1(CC(=O)NCC(C2CC2)NC(=O)CCn2ccnc2)ccc(Cl)nc1F 77711,c1(C(=O)NCC(C)N(C(=O)C(C)CC(F)F)CC)ccnc2[nH]c(C)nc12 77712,Cc1cc(N(C2CC3(CNC3)C2)C(=O)CN(C)C)n(CC2CC3CCC2O3)n1 77713,n1(CC)ccnc1C(C)NC(C1CSCN1C(=O)COCC(=O)OCC)=O 77714,c1(CC(=O)NCCC2(CNC(CN(C(C)=O)C)=O)CC2)csc(C)n1 77715,c1(C(N(CCOC(C(=O)OC)C)CC)C)ccccc1.C(C)(C)O 77716,n1(CCC)ccnc1C(F)(F)C(=O)N(C)CCN(C(=O)CC(C)C1CC1)C 77717,CCC(C)CC(C)NC(C(=O)O)c1cccs1 77718,C1(C(=O)NCC(C2CC2)NC(=O)CNC(=O)C(F)(F)F)CCN(C2CCC2)CC1 77719,CC(O)(CNC(=O)CCNC(c1ncc(F)cc1N)=O)C(F)(F)F 77720,N1(C(C2CCC(SCC)CC2)=O)CCCCC(NC(c2cn(C)cn2)=O)CC1 77721,CCS(=O)(=O)C=CC(=O)N1CCN(C(c2nnn(C(C)(C)C)n2)=O)C(C)C1 77722,c1(C(=O)NCC2CN(C(c3cnn(CCC)c3C)=O)CC2C)cnc(C)c(N)c1 77723,c1(COC)cccc(C(=O)NCC2(C)CCCN2C(=O)CCc2cnn[nH]2)c1C 77724,N1(C(=O)OC(C)(C)C)CCC2CC1CN(CC(=O)Nc1ccncc1)C2 77725,c1(C2(CNC(=O)NC3CCCC=C3Br)CC2)cccc(F)c1 77726,N1(C(C(c2cscn2)N(C)C)=O)CCN(C(c2cnn(C3CC3)c2)=O)CC(O)C1 77727,C1(CNC(c2nc(C(C)=O)sc2)=O)C2CN(C(=O)CC=C(C)C)CC12 77728,n1(CCC(N2CCC(N(C(C(CC)OC)=O)C)C2)=O)ccc2cc(C)ccc12 77729,CC1CN(C(=O)CCc2cn[nH]c2)CC2(CCN(Cc3ccc(F)cc3)CC2)O1 77730,c1(C(=O)NC(C2N(C(C(CC#C)O)=O)CCC2)(C)C)cc(C)nc(C)c1 77731,N1(C(c2c(C)nsc2)=O)CCCCC1CCCNC(C1CC1C)=O 77732,S(=O)(=O)(c1nc(C)cs1)Nc1cc(OC)c(OC(F)F)cc1 77733,N1(C(CC2(CC)CCC2)=O)CCCC2CCN(C(=O)CC3CC3)CC12 77734,N1(C(CC2C(NC(=O)CCc3ccccc3)CCCC2)=O)CC(CO)C2(CC2)C1 77735,N(C1COc2cc(Br)cnc21)C=O.c12nn(C)cc1S(C)(=O)=NC2=O.CO 77736,C(CC(C(=O)NOC(C)(C)C)NC(c1ccc(C)c(O)c1)=O)OCC 77737,c1(C(C)C)c(C(=O)N(CC(C)NC(=O)CC2COC(=O)N2)C)cnc2ncnn12 77738,C1(C(=O)OC(C)(C)C)COCCN1C(C1(C)CCN1C(c1cnccc1Cl)=O)=O 77739,Cc1cc(C(=O)NC(CNC(C2CC3C=CC2C3)=O)CO)cc(S(C)(=O)=O)c1F 77740,CC1(C)CC(C(=O)N2CC(C(C)(C)O)(CNC(C3(Cl)CC3(F)F)=O)C2)=NO1 77741,CCCC(CCC)C(=O)N1CCOCC1CCNC(=O)CSCCN(C)C 77742,CCC(C)C(O)CC(=O)NC1(CNC(=O)Cc2ccc(F)c(Cl)c2)CC1 77743,C1(CC(=O)NC2CCCN(C(C)C)C2=O)(OC)CC2(CCOCC2)C1 77744,C(C)(C)(CCC(=O)NC1CCC(N(C)C(c2cnsc2C)=O)CC1)OC 77745,c1(C(=O)NCC(=C)CCNC(=O)CSc2ccncc2)[nH]nc(C(F)(F)F)c1C 77746,C(C(C)(C)C(=O)NCC1CC(CF)C1)NC(C1CCC(C)C1)=O 77747,N1(C(C(C2CCN(C(CC3C(C)OCC3)=O)CC2)C)=O)CC2CCC2(C)C1 77748,C(c1csc(C)n1)=CC(=O)N(C(CN(C(C1CCN(C(C)=O)C1)=O)C)C)C 77749,Cc1[nH]c(=N)sc1C(N1CCOC(CN(C(=O)CC2C=NN(C)C2=O)C)C1)=O 77750,N1(C(C(F)OC)=O)CCC(C)(CNC(=O)CN2C(=O)CNC2=O)CC1 77751,N1(C(C2CC(OC)C2)=O)CC2CC(O)C1C2NC(c1cccnc1N)=O 77752,Cc1ncc(C(=O)NCC2(N(C)C)CCC2)o1.c12nc(no1)C(C)NC(=O)CC2 77753,N12CC(CCC1(C)C)C(=O)NC1(CCC1)C2=O.C(C(C)CC(C)C)OCC 77754,c1(C(C)(C(=O)O)NC(=O)C(Br)Cc2ccccc2)cccc(O)c1 77755,c1(CNC(C(=O)N(CCCC(C)C)C)=O)nnc2c(Cl)cccn12 77756,C1(n2cc(-c3cccc(C)c3)nn2)CON(C(=O)c2c(C)cnn2C)C1 77757,c1(C(C)OCC)ncc(C(C(=O)NCC(F)F)N(C)C(C2CCCO2)C)s1.COC 77758,C1(=O)N2CCC(O2)C(=O)N2CCCC12.C1(OC(C)=O)CC1C(C(C)(C)C)=O 77759,C1(C(=O)NC(C)CNC(c2ccc(-c3ccncc3)s2)=O)CCC2(CCC2)OC1 77760,c1(C(=O)NCC(C)N(C(C2CC3CC3C2)=O)CC)ccc(Cl)c2c1OCCO2 77761,CC(CCC(F)(F)F)NC(C1C2CCC1(c1ccco1)C2)=O 77762,C1(NC(CCCSC)=O)(CO)CCN(C(=O)CC2CC(F)C2)CC1 77763,Cc1nc(O)sc1C(=O)NCC=CCC(=O)NCC1(C(O)C(C)C)CC1 77764,N1(C(C(CCCC)O)=O)CCC2(CCC(NC(c3coc(C(F)F)n3)=O)CC2)C1 77765,C1(CN(C(C2(OC)CCCC2)C(=O)NCC2CCCO2)C)COC(C)(C)O1 77766,c1(C(=O)OC)ccc(Br)c(C(=O)NC2(C)CN(C(=O)C(C)C(C)O)C2)c1 77767,C1(C(=O)Nc2cccc(CC)c2F)CC(C)(C)CCN1C(=O)C(C)c1cc[nH]n1 77768,c1(C(=O)NC2CC3CC(NC(=O)Cc4ccco4)C2C3)cnc2[nH]cncc1-2 77769,N1(C(Cc2cc(C)no2)=O)CC(NC(c2cc(=O)c(Br)c[nH]2)=O)CC12CCC2 77770,Cc1cc2c(Br)ccc(C(=O)NC(C3CCN(C(C4(C)CC4)=O)CC3)C)c2o1 77771,c1(C(=O)NCC23CC2CN(C(c2ccc(O)cn2)=O)C3)ccc2oc(O)nc2n1 77772,c1(C(=O)NCCCCC(C)(C)N)cc2nc(Cl)ccc2s1 77773,N1(C(CC2(OC)CN(C(C34CCCCC3C4)=O)C2)=O)CCC2(CC1)CSC2 77774,C(=O)(C(O)CCCNC(=O)CCc1cccnc1)NC(CCC)c1nn[nH]n1 77775,C=C=CC(C)C(=O)N1CCCC1C(C)(C)C(=O)Nc1cnc(N(C)C)nc1 77776,C1(C(=O)NC(C(C)C)CCN(C)C(c2cnnn2C)=O)OCCN(C)C1=O 77777,C1(CNC(c2csc(C)c2C)=O)CN(C(C2CCOC2)=O)CC(C)(C)C1 77778,C1(NC(C2(C=C)CCC2)=O)CC(O)CN(C(c2ccc(OC)c(C)c2)=O)C1 77779,c1(C(=O)NC(CN(C(CNS(CCOCC)(=O)=O)=O)C)C)ccc(C)cc1CC 77780,c1(C(=O)NC2CC(NC(=O)COC3CC=CC3)C2)c(Cl)ccc(F)c1F 77781,c1(C(=O)NC2CN(C(CCCOCC)=O)C2)nccc(Br)c1O 77782,c1(OC)cc(C(N2CCC2CNC(=O)CCCC2CC2)=O)c(N)cc1F 77783,c1(C(N2C(CC(=O)N(C)CCO)CCC2)=O)cccnc1O 77784,N1(C(c2n[nH]c(C)c2C)=O)CCC(C)(CNC(C2CC2C(=O)NCCO)=O)CC1 77785,N1(C(Cn2ncc(CC)c2)=O)CC=C(CNC(C2CCN(C(N)=O)CC2)=O)CC1 77786,C1(CNC(C(C)C)=O)CN(C(=O)C(O)C2=CCCCC2)C2CCCC2O1 77787,C(=O)(C(F)(F)CCn1ccnn1)N(CC1C(c2cnn(C)c2C(=O)O)C1)C1CC1 77788,C1(C(=O)OC)(C(=O)OC)CN(N2CCC(c3nc(C4CC4)no3)C2)C1 77789,Cc1[nH]c2ccccc2c1CCNC(=O)C(C)SCC1CCCO1 77790,c1(CNC(c2ccoc2C2CC2)=O)cccc2c1CN(C(C1CCCO1)=O)C2 77791,c1(C(N(C)CC2COC(C)(C)C2O)=O)ccc(Cl)cc1N=[N+]=[N-] 77792,C1(C#N)(C(N(CCNC(CC(C)C)=O)C2CC2)=O)CCCO1 77793,C=CCCCCC(=O)NC(C)CCCCNC(C1CCCN1c1cnccn1)=O 77794,NC1CC2(CC(C(=O)NC3(CO)CC4CCCC34)C2)C1 77795,C1(C)(CNC(Cn2nnc(C(C)(C)C)n2)=O)CN(C(=O)CC2CC(F)C2)CC1C 77796,C(=O)(C1=C(Cl)CCC1)N1CCC(CNC(=O)CCC(=O)c2ccc(O)cc2)C1 77797,Cc1cc(C(N2CC(CNC(C3COC3)=O)CC2C)=O)c2nc(C)n(C)c2n1 77798,CCC(C)(O)C(=O)NC(C1CCCN1C(c1cc(CO)ccn1)=O)(C)C 77799,c1(C(C)=O)ccsc1C(N1CCC(OCCNC(=O)CCN2CCC(F)C2)C1)=O 77800,c1(C(=O)NCCC(C)NC(=O)C#CC2CC2)c(C2CC2)cccc1F 77801,c1(NC(COC(C2C(C)(NC)C2)=O)=O)ccc(Br)cc1Br 77802,C(=O)(CC(C)CC(C)(C)C)NCC(=C)CCNC(C1CCC(C(C)C)CC1)=O 77803,c1(-n2cc(COC3CCN(C(CC(C(C)C)O)=O)C3)nn2)cc(Cl)c(F)cc1F 77804,CC1CC(C)(C)CN1C(=O)COC1(C)CN(C(=O)C=Cc2cc[nH]n2)C1 77805,c1(CC(=O)NCCC2CCC(NC(CC(C=C)C)=O)C2)cn2cccc(C)c2n1 77806,Cc1cc(N2Cc3nn(C)c(N)c3C2)nc(=NCCn2ncc(Br)n2)[nH]1 77807,C(C(O)C(C)C)Nc1c[nH]nc1Cl.CC1=CC(=O)N(C2CC2)C1 77808,N1(C(c2cc(SC)oc2)=O)CC(C2CCN(C(C3CCOC(C)(C)C3)=O)CC2)C1 77809,C(CC(=O)OCC)N(C(COCC(=O)NC1CCC1)=O)CCC 77810,C1(C(N2C(CC)CCCC2)=O)CC1C1CN(C(=O)C(C)(C)CSC)C1 77811,CC(CC(=O)NCCCC1CCCN1C(=O)CCN1CCCC1)P(C)(C)=O 77812,C(CC(N)C(F)F)N(C)CC1ON=C(C)C1 77813,c1(C(CNC(CCCC#C)=O)NC(c2cn(C)c(C)n2)=O)ccc(F)cc1F 77814,N1(C(c2ncc(OCC)nc2)=O)CCC2(NC(=O)CCc3c[nH]c(=N)[nH]3)CC2C1 77815,C(C(N=[N+]=[N-])C(=O)Nc1nc(OCC)ccc1C)OCC 77816,C#CCC(CC(=O)N(C)CC1(N(C)C)CCC1)NC(=O)CC(C)C(F)F 77817,C#CC1(C(=O)NCC2CCC(NC(C3CC4(CCO3)CC4)=O)CC2)CCOCC1 77818,c1(C(=O)NCCC(CNC(C2N(C)CCC2)=O)O)cc(N)c(O)c(F)c1 77819,C1(NC(C2CCCC2)=O)CC2CCC1CN2C(c1cc(O)ncc1F)=O 77820,N1(C(CN(C)C(N)=O)=O)CCC(CO)(NC(c2coc(C(N)=O)c2)=O)C1 77821,C1(C(=O)NCC2C(NC(=O)C=Cc3nccs3)CCCC2)CCC2(CCC2)C1 77822,Cn1nc(C(=O)NC2CC(F)(CNC(C3COCCO3)=O)C2)cc1C(F)F 77823,C(=O)(C(C)(C)C(C)(F)F)N1CCC(F)(CNC(C2(C)CCCCCC2)=O)C1 77824,C1(C)(CC)CCCC1NC(c1c(C2CC2)cno1)=O.C12CC(C1)CNC2=O 77825,C1(C(C(=O)NCCC=C=C)C)CCN(C(c2noc(C)c2C)=O)CC1 77826,N1(Cc2ccc(OCC)nn2)CC(C(N2CCC(SC)CC2)=O)CC(C)C1 77827,C1(C(N2CCN(C(CSCCCC)=O)CC2CF)=O)COC2CCCCC12 77828,c1(C(N(CCOC)C(C)C2CC2)=O)coc(CNC(=O)CCC2CCC(C)O2)n1 77829,c1(NCCC(=O)NC(C2(C)CCC2)C)ncnc2sccc12 77830,c1(C(N2CCC(OCCNC(C3(CC#C)CC3)=O)C2)=O)cc2cc(Cl)cnc2o1 77831,CN1CCC2(CCN(C(=O)COCCNC(c3cccn3C)=O)C2)C1 77832,C1(NC(C)=O)CC(CC(N2CCC2C(=O)NC2(C3CC3)CC2)=O)C1(C)C 77833,N1(C(=O)Cc2ccccc2)CCC(F)(C(=O)Nc2cnc(-c3ccccc3)s2)C1 77834,c1(C(N2CCC(N(C(=O)C(c3ccc(C)s3)C)CCC)C2)=O)nc(CC)oc1C 77835,Cc1cc(N)cnc1C(=O)NCC1CCN(C(C2CCC3CCC2O3)=O)C1(C)C 77836,C(=O)(CC(CC)C(C)(C)C)NC(c1cccnc1)C(=O)N(C)CC1CC(=C)C1 77837,C(=O)(C(C)(C)C(=O)NCCCCCCNC(C1CCN(C)S1(=O)=O)=O)OC 77838,N1(C(c2c(NC)nccc2)=O)CC(C(N2CCC(CCO)CC2)=O)CC12CCC2 77839,C(C)(CN=c1[nH]c(N2CC(c3ccc4ccccc4c3)C2)nc(=N)[nH]1)OC 77840,c1(CC)nc(C)cc(=NC(CNC(=O)C(F)C(C)C)C2(c3ccccn3)CC2)[nH]1 77841,C1(CNC(C(n2ccc(C)n2)(C)C)=O)CCCCN1C(=O)C(c1cnccn1)C 77842,c1(C(=O)NC2C(CNC(c3c(CCC)onc3C)=O)CC2)cc(F)c(Cl)cc1Cl 77843,C1(CCC(=O)NCC)(CC2CCN(C(CCC)=O)C2)CCC(=O)N1 77844,c1(C(N(C)C)=O)cccc(CN2CCCCC2CNC(=O)CC2CC(=O)N2)c1 77845,c1(CC(C)C(=O)N(C)CCOCCNC(C2CCC(=O)N2)=O)cccc(F)c1 77846,C1(F)(C(N(CC(CCC)C)C)=O)CCN(C(c2cc(C)co2)=O)C1 77847,N1(C(CC(C)Nc2ccccc2)=O)CCCCC(CN=[N+]=[N-])C1 77848,c1(NC2C(CC)C2)ncccc1S(=O)(=O)NCc1nc2ncccn2n1 77849,C(CCCC(C)(C)NC(=O)C(CSC)OC)NC(CC1CC(OC)C1)=O 77850,c1(C(=O)OC)ccc(NC2CC(F)CN(Cc3ccc(Br)o3)C2)c([N+](=O)[O-])c1 77851,c1(C(=O)NC(CNC(C(CC=C)C)=O)C(C)C)c[nH]c2cccc(Cl)c12 77852,CC1(C)CNCCC1N1CCN(Cc2cc(Cl)ncc2Cl)CC1 77853,c1(C(N2CC(C(C)NC(c3cc(CF)on3)=O)OCC2)=O)cc(Cl)c(O)c(Cl)c1 77854,C1(O)(CNC(CC(C)F)=O)CCCN(C(c2ccc(C(F)F)cc2F)=O)CC1 77855,CCC(CC)C(C)(F)F.C1(=O)C(C2CCCC2)CN1CC 77856,CC1CN(C(=O)C(C)N(C)C(C2CC(=O)OC2(C)C)=O)C(C)C1C 77857,CC(CC(=O)N1CC(O)(C2CCCN2C(c2cnc3n2CCC3)=O)C1)C(F)F 77858,c1(C(N2C3C(NC(=O)C=CC4CCC4)CC(C3)C2)=O)ccc2ccncc2n1 77859,c1(N2CCN(C(=O)Nc3cc(C)ncc3Cl)CC2)cccc2nsnc12 77860,C=Cc1cncc(C(=O)NC2(CO)CCCN(C(=O)CN(C)C)C2)c1 77861,N1(C(C=CC=CCCCCC)=O)CC2C(CNC(C3CCC(=O)N3C)=O)C2C1 77862,N1(C(C2CCN(CC)C2)=O)CCOC(CCCNC(=O)CSC2CC2)C1 77863,N1(C(CCc2c(C)noc2Cl)=O)CCC2(CCN(C(=O)CCc3cncs3)C2)C1 77864,N1(C(c2c(C)ncnc2)=O)CC2CCC(C1)C2NC(C1(C)CC2CCC(C1)S2)=O 77865,c1(NC(c2n(CCC)nnn2)CC(C)OC)ccc2c(c1)OC(F)(F)O2 77866,c1(SC(=N)N)cccc(C(=O)NC2CC(C(=O)NCCC3NC(=O)NC3=O)C2)c1 77867,N1(C(c2ccc(C)s2)=O)CCCC(O)(CN(C)C(c2ccc(C(C)C)nc2)=O)C1 77868,C(=O)(C(C(=O)c1ccc(OC2CCOC2)cc1)NC(=O)C1CC1)OC(C)(C)C 77869,C(=O)(C1=CC2C=CC1C2)NC(C1CCCN1C(c1cc2ccccn2n1)=O)C 77870,c1(OCC(=O)NCCN(C(c2[nH]c(C)cc2C)=O)CC)ccc(Cl)nc1 77871,C(=O)(CC(O)CC(C)C)NC(C(=O)NC(CC(=O)OC)C)COC(C)C 77872,c1(C(=O)NCC(C)(C)NC(C(COCC)C)=O)cccc(C(=O)OC(C)(C)C)n1 77873,CCC(C)C(O)C(C)C(=O)NCC(C)(C)CC(=O)N(CC(N)=O)C 77874,CCC(CC(F)(F)F)NC(=O)CC(C)N(C(=O)Cc1cncnc1)C 77875,c1(CNC(CN(C)C(C2CC=CCC2)=O)=O)cccc(F)c1O 77876,C(=O)(C(C)CC(C)CC)N1CCC(OCC(=O)N(C(C=C)C2CC2)C)C1 77877,CC1CC2(CCN(C(=O)C(N3CCCC(N4CCC4)C3)=O)C2)CO1 77878,Cc1cc(O)c(Cl)cc1C(=O)NCCCCNC(=O)C(C)CC1CCC1 77879,N1(C(C2CCCN2C(C23CCCC2C3)=O)=O)CCc2nnnn2CC1 77880,C1(CNC(C23OC(C)C(C2)C3)=O)CC2(CO1)CN(C(=O)Cn1ncnn1)C2 77881,C#CC1CCN1C(C1CC(CCNC(=O)CC2(NC(C)=O)CC2)C1)=O 77882,c1(SC)sccc1C(N1CCCC1CNC(c1ncoc1C(F)(F)F)=O)=O 77883,c1(C(=O)OCCn2c(C)nnn2)ccc2c(c1)CCN2Cc1ccco1 77884,C1(C(C)C)CC(CC(=O)NC2(C)CCN(C(=O)C(F)=CCCF)C2)CCO1 77885,c1(CC(N2CCCC(NC(C(CC)O)=O)C2)=O)ccc(Cl)c(Cl)c1 77886,C=C(C)C1CN(C(=O)CCNC(C2CC2(C)C(C)C)=O)CCO1 77887,N1(C(c2ccc(N)cc2Br)=O)CCC2(CC(NC(=O)Cc3cnoc3)C2)C1 77888,CCCCCC(CC)C(=O)NCC1CN(C(C23CC(C2)C3)=O)CCCO1 77889,c1(C(=O)NC(c2ccncc2)CC)ccn(CCNC(=O)CCc2ccsc2)c1 77890,Cc1n[nH]cc1C1CC1C(=O)NCC1(F)CC(CNC(c2ccsn2)=O)C1 77891,N1(C(CN(C(=O)C(C)n2ccnc2)CC)=O)CCOC(C)C1C.C(C)(=O)O 77892,N1(C(CCC#C)=O)CCC(C=C)(C(=O)NCCCS(C)(=O)=O)CC1 77893,c1(OCC)cc(C)c(C(N2CCCC(NC(=O)NC3CC3)CC2)=O)cc1Cl 77894,C1(NC(CC(C)OC)=O)CN(C(=O)CCCc2cnccn2)CC12CCC2 77895,C1(C(=O)OC)CCC2(CC1)CC(S(=O)(=O)N1CC(NC(C)=O)C(C)(C)C1)C2 77896,CC(CC(=O)NCC1CCCN1C(=O)CCCc1cnccn1)C1CC1 77897,C1(CC)(CC)CC(O)CN1C(C1CC(CNC(c2c[nH]c(=S)cn2)=O)C1)=O 77898,N1(C(CC2(CNC(C3C(CC)OCC3)=O)CC2)=O)CCC(N=[N+]=[N-])C1 77899,C1(CC)CN(C(=O)C(CCOC)OC)CCN1C(c1ccc(O)c(Br)c1)=O 77900,C1(NC(C(CO)NC(C(CCC)NC(N)=O)=O)=O)CCCC(O)CC1 77901,C1(C(C)C)CCC(C(=O)NC2COCC2NC(=O)CC2COCCO2)CC1 77902,C1(C(N2C3CN(C(c4c(C)ocn4)=O)CC2CC3)=O)C(C)(C)CCCC1(C)C 77903,c1(C(=O)NC2C(CNC(c3cnc(O)s3)=O)CCC2)ccncc1Br 77904,c1(SC)cc(N2CC3(CCN3C(c3cncc(C(F)(F)F)c3)=O)C2)nc(C)n1 77905,S(=O)(=O)(c1cccc(=NCC2(C)CC3CC3C2)[nH]1)N(C(C)(C)C)C 77906,Cc1cc(Cl)ncc1CC(=O)NCC(C1CCCCC1)NC(=O)C1=COCC1 77907,N1(C(C2CCN(CC#C)CC2)=O)CC2CC(NC(C3CC(C)C3)=O)CC2C1 77908,C1(OC)Cc2ccccc2C1NC(=O)NC(C1(CO)CCOCC1)C 77909,N1(C(C=NOC)=O)CCN(c2ccccc2CNC(C2(N(C)C)CCC2)=O)CC1 77910,c1(C(N2CCC(CO)C(O)C2)=O)cccc2[nH]nc(C3=COCC3)c12 77911,C(=O)(C(C)(C)C1=CCN(C(=O)C2=CC3(CCOC3)C2)C1)NCC(C(CC)C)CO 77912,C=CCC(CC=C)C(=O)NCC(CNC(=O)Cc1c(C)nc(O)nc1O)OC 77913,C#CC1C(C(=O)NCC2(NC(=O)COc3ccc(C)cc3)CCCC2)C1(C)C 77914,c1(C(CC)(C)C)n[nH]c(=NC2CC23CC(NC(=O)Cc2nnc(C)o2)C3)s1 77915,c1(OCC)cc(Br)ccc1NC(C(COc1ccccc1)C(=O)NC(C)(C)C)=O 77916,C(=O)(C(CO)NC(=O)C(CC1CC1)NC(c1cc(C(C)=O)[nH]n1)=O)OC 77917,N1(C(C(C)CS(C)(=O)=O)=O)CCN(C(c2ccc3cnsc3c2)=O)CC12CCC2 77918,Cc1cc(-c2csc(NC(c3ccnc(Cl)c3Cl)=O)n2)cnc1O 77919,C1(CCNC(=O)Cc2ccsn2)CN(C(c2cocn2)=O)CCO1 77920,c1(C(N2CC3CN(C(C4N(CC)CCC4)=O)C3CC2)=O)cnn2cc[nH]c(=O)c12 77921,c1(C(N2CC3(C(NC(c4cnc[nH]4)=O)CC3)C2)=O)noc2ccc(Cl)cc12 77922,Cc1cc(=NC(=O)C(=O)N(C)Cc2cc(Cl)cc(Cl)c2)[nH]n1C(C)C 77923,CS(=O)(=O)CCCCNC(N1CCCCC1C1CCC1)=O 77924,C1(C(N(CC(N)=O)C)=O)CN(C(c2n[nH]c3ccccc23)=O)CC1C1CC1 77925,c1(C(=O)NCC2C(NC(CCn3ccc(C)n3)=O)C2)ccccc1N(C)C 77926,N1(C(CN(C(=O)CCC2CCC(C)O2)CC)=O)CCC2=C(CCCC2)C1 77927,CC1(C)CCN(C(=O)C(F)C2CCCC2)CC1NC(c1cc(C2CCC2)no1)=O 77928,C#CCCCC(C)C(=O)NCCOCC(=O)NC(C1CCCCC1)C 77929,c1(CNCC2(C)COC2)c[nH]c2c(F)cc(C(=O)O)cc12 77930,C1(C(=O)NC(CNC(C2COC(=O)N2C)=O)C(C)C)(CC)CNC(=O)C1 77931,c1(NCC2(C)CCCCC2)cc(=NC2CCCc3sccc32)[nH]c(C(F)(F)F)n1 77932,C1(CNC(C(C)OCC)=O)(Cn2cc(C3(O)CCOC3)nn2)CC12CCC2 77933,C1(CC)CC(C)CN(C(=O)CC2CC(F)CN2)C1 77934,c1(CC)c(C(c2nnnn2C2CC2)NCCCc2ccccc2I)cccc1F 77935,S(=O)(=O)(c1ccc(=NCC2CC2C)[nH]c1)NC(c1ncc(C)cn1)C 77936,C(=O)(C1=C(Cl)CCOC1)N1C(C(=O)NCC(CC)(C)OC(C)=O)CCCC1 77937,C1(NC(c2ccc(F)c(CO)c2)=O)CCS(=O)(=O)C12CN(C(C1C=CCC1)=O)C2 77938,N1(C(CCC2CCN(C(C3(C)C(C)CCC3)=O)C2)=O)CCC(O)(C2CC2)CC1 77939,CC1CCC(NC(=O)CCC(=O)c2ccc[nH]2)CN1C(c1cc(F)ccc1O)=O 77940,c1(C(N2CCC3(CCN(C(=O)C(F)(F)C(F)F)C3)C2)=O)ccc2[nH]ccc2c1 77941,N1(CC2C3(CCC(C)(C)CC3)C2)CCc2c(Br)ccc(C#N)c2C1 77942,C(C1=CCCOC1)N(C)C(C1CCC(NC(c2cnc(C3CC3)o2)=O)CC1)=O 77943,N1(C(C(C)=C(CC)C)=O)CCC2CCCC12CNC(=O)COc1cccc(C)c1 77944,C(CCNC(C1CC1c1cccs1)=O)(C(C)C)NC(Cc1ccn(CC)n1)=O 77945,C(C)(C)(CC(F)C(=O)NCc1occc1C)NC(CCOCCOC)=O 77946,N1(C(C2(SC)CC2)=O)CC2CCC1CN2C(C1(CO)CC1)=O 77947,c1(C(CC)(C)C)nnc2c(N3CCC(O)(Cc4ccccc4)C3)nccn12 77948,c1(OC(C)C(=O)NCCCCN(C(=O)CC2COC(=O)C2)C)cc(Cl)cc(Cl)c1 77949,n1(CC(=O)N(CCC)CCN2CCC2C)cc(-c2ccnn2CC)nn1 77950,CC(C)(F)CCC(=O)NCC1CCCC1C(N1CCC(CC(N)=O)CC1)=O 77951,c1(C(=O)NCC2C(NC(C=NOC)=O)CCC2)cnc2c(c1)CCCC2 77952,c1(C(=O)NC2C(C)CN(C(=O)CC3SC(=N)NC3=O)C2)nc2ccccc2[nH]1 77953,N1(C(C(CC=C)C)=O)CCC2(CC1)CN(C(C1CCCN1C1CC1)=O)C2C(C)C 77954,c1(C(=O)NC2CC(NC(CCC(C)(C)OC)=O)C2)ccc2ncnn2c1 77955,C1(C(N(C2CC(C(N)=O)C2)C)=O)CC=CCC1NC(=O)Cc1cccnc1O 77956,c1(C(N(CC(C)N(C(C(C)OCCN(C)C)=O)C)C)=O)cccn1C 77957,C1(NC(C(CCC)N(C)C)=O)CC12CCC(NC(=O)C(=O)NCCOC)CC2 77958,n1(CCC)cc(C(=O)NCCSCCC(=O)NC2(CCCF)CC2)cn1 77959,C#CCC(C)(C)C(=O)NCc1ncccc1C(=O)Nc1ccc(C(C)C)cc1 77960,O=C(C1=Cc2ccc(Cl)cc2OC1)NCC(C1CC1)NC(c1cscn1)=O 77961,c1(C(=O)Nc2ccc(C(=O)O)nc2)cc2c(o1)=CCC(c1sccc1CO)=CC=2 77962,C(=O)(CCC(C)CC)N1CC(CCNC(C2CC(=C)C2)=O)OCC1 77963,N1(C(COCCOCC)=O)CCN(C(c2cscc2F)=O)CC1.C12CCC(C1)N2 77964,c1(C(N2CCCC(CC(N3C(CC)CCC3)=O)C2)=O)cnn2ccc(Cl)c(F)c12 77965,C(CNC(=O)CCCOC1CCCC1)(CC(=O)NC1CN(C)C1)OC 77966,CCC(CCCC(=O)N1CC2(COC(C)C2)C1)NC(=O)C=CC(C)(C)C 77967,N1(C(c2c(C)nc(CC)o2)=O)CCC2CN(C(=O)C(C)(C)CSC)CCC2C1 77968,CC(C)(CC(=O)NC1(C2CCN(C(=O)C(F)CC3CC3)C2)CC1)C(F)F 77969,C1(O)(CNC(=O)Nc2c(-n3cc(C=CC)nn3)cccc2)CCC(F)(F)CC1 77970,C1(CC)CCCC1(C)C(N1CC(NC(=O)CSc2ccccc2OC)C1)=O 77971,c1(CC)nc(=N)[nH]cc1C(N1CCC1CNC(=O)CC1CC1(C)C)=O 77972,C1(C(=O)NCC(C)C)CC12CCN(C(=O)Cc1ccc(Br)cc1F)C2 77973,C(C(C(=O)N1CC(OC(C)=O)C1)NC(C1C=C(C)CS1)=O)OC 77974,N#Cc1ccc(NC(=O)C(N)=O)cc1C#N.C1(=O)CC(Cc2cccs2)N1 77975,Cc1ncnc(C)c1C(N1CC2C(CNC(=O)Cc3cccc(F)c3O)C2C1)=O 77976,C1(C(=O)NCC2(OCC)CC2)CC2(CCCN1C(=O)CCCC(=O)OC)CC2 77977,c1(C(=O)NCC2OCC(CNC(CC3CC(=C)C3)=O)C2)ccc[n+]([O-])c1 77978,c1(C(=O)NCCCNC(=O)CN2CCCCCC2)cc2c(Cl)cncc2o1 77979,C(=O)(C1=CC2C=CC1C2)N1CC2C(CC(=O)N(CCCO)C)(CC2)C1 77980,N1(CC(=O)NC2CCC(NC(c3c(C)nc[nH]3)=O)C2)CCN(S(C)(=O)=O)CC1 77981,Cc1cccc2c(C(=O)NC3CC4CCC(C3)N4C(=O)Cc3nc[nH]n3)csc12 77982,c1(OC)cc(=O)n(C)cc1C(=O)NCCOC1CN(C(=O)C2=CCSC2)C1 77983,N1(C(c2cc(C)on2)=O)CCC(NC(c2cc(C(F)F)cs2)=O)C(O)C1 77984,C1(NC(N2CC(N(C(CC3N(CC)CCOC3)=O)C)C2)=O)CC2C=CCC(C1)C2 77985,N1(C(C(C2CC2)SC)=O)CC=CC(C(N2CCC(N(C)C)C2C)=O)C1 77986,c1(C(=O)NCCC2(NC(CC3CC(=C)C3)=O)CC2)sc2ccccc2c1Cl 77987,n1(CC#C)ccnc1CN(C)C(=O)N.C1(C(=O)OC)(CC=C)CCOC1 77988,c1(CNC(=O)Cc2ccccc2F)ccccc1CNC(c1c[nH]c(Br)c1)=O 77989,c1(C(=O)NCC(CO)NC(C2C(=C)C2)=O)c[nH]nc1-c1cnn(C)c1 77990,n1(CC(C)C)c(N2CC=CCC2)nnc1Cc1cccs1 77991,c1(-n2ncc(C)c2)ccc(CNC(N2CCOC(C)(C3CC3)C2)=O)cc1F 77992,N#Cc1c[nH]c2ncnc(NC3CC(Nc4ccc(F)cc4C#N)C3)c12 77993,N1(C(C2CCC(COC)C2)=O)CCSCC1C(N1CCCOCC1)=O 77994,CC(C)CC(C)CNC(=O)CC1CCCCN1C(=O)C(C)SC(C)C 77995,C1(NC(C=C(C)C(F)F)=O)CN(C(=O)C(CCN(C)C)N(C)C)CCC1O 77996,CCC(=O)CCC(=O)NC(C)CCCC(=O)NC1CCN(CC)C1 77997,N1(C(CC2C(C(=O)OC)C2)=O)CCC2CCN(C(C3CCCCCCC3)=O)CC12 77998,c1(C(N2C(CNC(C(C)Cc3ccccc3)=O)CCC2)=O)nc[nH]c2ncnc1-2 77999,O=C(CC1=CCOCC1)NCCC1CCC(NC(=O)Cc2ccc(F)cn2)C1 78000,c1(C(=O)OC)ccc(NC(C2CCN(C(=O)C(=O)c3ccco3)C2)=O)c(Br)c1 78001,C1(CNC(C2(C(C)(C)OC)CC2)=O)CN(C(c2cc(C)c(C)o2)=O)CC1C 78002,Cc1noc(C(CO)NC(=O)CCNC(=O)CNC(c2ccco2)=O)n1 78003,C1(C)(C(=O)OC)CCCN1C(c1cc(Br)ncn1)c1nc(SC(C)(C)C)no1 78004,c1(OC2C(NC(N3C(C(=O)OC)CC(O)C3)=O)CCC2)cc(Cl)c(Cl)cc1O 78005,C1(C)(CNC(CCOC(C)=O)=O)CCN(C(=O)C=Cc2cnn(C)c2C)CC1 78006,Cc1ccc(C(N2CCOC(C(C)NC(C3CCS(=O)CC3)=O)C2)=O)c(N)c1 78007,c1(C(N2C(CCNC(C3C(C=C)C3)=O)CCC2)=O)ccc2c(c1)CCN2C(C)=O 78008,c1(C(N2CC(C(C)NC(C3CCC4CC4C3)=O)OCC2)=O)ccc(O)cc1O 78009,N1(C(C)=O)CCC2(CC1)CC(NC(=O)C(C)CS(C)(=O)=O)C2 78010,c1(C(=O)NCC2N(C(c3nccc(N)c3)=O)CCOC2)noc2ncccc12 78011,C(=O)(C1=Cc2ccccc2C1)OC(=O)CN(C(=O)NC(C)C)Cc1cccc(C)c1 78012,C1(CC)CN(C(=O)C(N2CCCC2)C2CC2)CCC1NC(c1ccncc1)=O 78013,N1(C(CCC(=O)N(CC)CC)=O)CCC(NC(=O)C(C)(C)CO)C(C)(C)C1 78014,C1(CNC(c2cnn(C3CCC3)c2)=O)CN(C(=O)C=CBr)CC1(F)F 78015,C(=O)(C(C)CS(C)=O)NCC1(NC(Cc2ccc(CC(=O)NC)cc2)=O)CC1 78016,O=C(C#CC1CCCCC1)NCC1CCN1C(=O)CCF 78017,C(C)(C)(CCCNC(=O)C(CSC)SC)NC(C(c1cccc(Cl)c1)OCC)=O 78018,CC1CCCCC1(CNC(=O)CC1CC=CC1)NC(C1OCCN(C)C1=O)=O 78019,c1(OC)ncc(C(N2CC(C(=O)NCCC3CCOCC3)CC(F)C2)=O)cc1F 78020,N1(C(C(CC)N2CCCC2=O)=O)CC(F)(F)CC1CNC(c1ncccc1C)=O 78021,C#CCC(C)(C)C(=O)NC1C2CN(C(c3ccc(C(O)CF)cc3)=O)CC12 78022,Cc1ccncc1CC(=O)NC1CCC1C(=O)NCc1occc1C 78023,C1(CNC(c2cncn2C2CC2)=O)CCCCCN1C(=O)CC1COCCO1 78024,C1(NC(c2ncc(NC)nc2)=O)CC(NC(C2CCS2(=O)=O)=O)C12CCOCC2 78025,C(=O)(C(CC)C(=O)N1CCC(NC(=O)CNC(c2cccc(C)c2)=O)C1)OCC 78026,C(=O)(CCC(C)NC(=O)Cn1nc(C)cc1C)NC1(C(=O)OC)CC=CC1 78027,N1(C(c2cnc(Cl)s2)=O)CCC2CN(C(c3cccc4sccc34)=O)CC2C1 78028,c1(CC(=O)OC)cccc2c1CN(C(C1(c3ccccc3)CCCC1O)=O)CC2 78029,N1(C(=O)C(Cl)=CCl)CC(NC(C2(c3cccnc3)CC2)=O)C(F)C1 78030,N1(C(c2cc(C)c(C)nc2)=O)CCCC(NC(=O)C(O)CCC(C)C)CCC1 78031,N1(C(C=C(COC)C)=O)CCCC1C(C)NC(=O)COc1ccccc1 78032,N1(C(Cc2c(C)cc(C)s2)=O)CC2CCN(C(=O)CCN(C)CCO)C2C1 78033,C1(C(OC)OC)CN(C(C2CCCN(c3cccnn3)C2)=O)CCO1.CO 78034,n1(CCC)nc(C)cc1C(=O)NC1CCCCC1NC(c1n[nH]c(C)c1C)=O 78035,C1(SC(C2(C(=O)OC)C(C(=O)OC)C2)=O)C2CC3C(C2=O)C13 78036,Cn1ncc2c1CCC(C(N1CCC(CO)(NC(=O)Cc3c[nH]nc3O)C1)=O)C2 78037,C1(C)(NC(C(c2ccccc2F)C)=O)CC2(CC2)C1 78038,N1(C(CCCCC)=O)CCN(C(c2ccn(CCC(F)(F)F)n2)=O)C(C)C1C 78039,C#CCCCCCC(=O)NCCCC(C)NC(=O)C(C)c1ccsc1 78040,c1(N(C(CNC(=O)CNC(C2CCCC(O)C2)=O)=O)C2CC2)cc2ccccn2n1 78041,CCN=C(NCc1noc(-c2ccccc2)n1)NC(c1cccs1)C 78042,C1(C(=O)NCCCC(O)CO)CCN(C(=O)Nc2ccccc2)CC1 78043,C(=O)(C1=CC(C)CC1)NCCC(C)NC(c1c(C)occ1C(F)(F)F)=O 78044,C(=O)(C(F)C(C)C(F)(F)F)NC1(C)CN(C(CCOc2cccc(C)c2C)=O)C1 78045,C1(CN(C(C2C(C)C(=O)C2)=O)C)CCCN(C(=O)C=CC(C2CCCCC2)=O)C1 78046,C#Cc1ccc(Cl)c(C(=O)NC2(C)CC(NC(C3(C)CCC3)=O)C2)c1 78047,C1(CC(N2CC(c3cn(-c4nccs4)nn3)C2)=O)CCC2CC12 78048,CN1CC(CC(=O)NOc2ccc(N)c(Cl)c2)CCC1C(F)(F)F 78049,N1(C(c2cnn(C(C)C)n2)=O)CCN(C(=O)CNC(=O)CN2CCCC2)CC1 78050,C(=O)(C1=C(C)OCCS1)NC1C(OC)CN(C(=O)CN2CCC(C)(C)C2)C1 78051,C=CC(C)N=C(NC1CCc2ccccc21)N1CCC(NC(=O)C(C)(C)C)CC1 78052,C(=O)(C1CCCOc2ccccc21)N1CC(F)(CNC(C2(C)ON=C(C)C2)=O)C1 78053,C12(NC(C=C(C)C(C)C)=O)CCC(F)(F)CC1CN(C(=O)CC1CNC(=O)C1)C2 78054,C1(O)(CC(=O)NCc2csc(Cl)n2)CCCN(C(=O)CC2CCCC23CC3)C1 78055,N1(C(c2cnn(C3CCOCC3)c2)=O)CC2(C1)CN(C(C1(Cl)CC1)=O)CCO2 78056,c1(C(N2CCC(O)(CCNC(CC(C=C)C)=O)C2)=O)cc(F)c(C(F)F)cc1F 78057,C1(NC(c2coc(Cl)c2)=O)C2CC3CN(C(c4ccc5n[nH]cc5c4)=O)C1C3C2 78058,CCC(CC(=O)NC(CNC(c1csc(-c2ccc(Cl)cc2)c1)=O)CO)C(C)C 78059,c1(NC)nc(N(C)C(c2ccc3c(c2)C(C)CO3)=O)[nH]c2ncnc1-2 78060,c1(N(C2(CCO)CCC2)C)ncccc1S(=O)(=O)NCc1n(CC)ccn1 78061,C#Cc1cn(C)nc1C(=O)NCC1CN(C(C2CS(=O)(=O)C2)=O)C1 78062,CC1CC(NC(c2cc(-c3cn(C)nn3)on2)=O)CN1C(c1ccc(N)cc1)=O 78063,C12(CC(=O)NCCC(CC)C)CCC1CN(C(c1cc(CO)on1)=O)C2 78064,N1(C(C2Cc3ccccc3C2)=O)CC2(CCCCN2C(C2CCCS2)=O)C1 78065,c1(OC)cccc(-n2nnc(C(=O)N(CC(C)NC(=O)C(C)C(C)O)C)c2C)c1 78066,N1(C(CC(c2ccc(F)c(F)c2)C)=O)CC2CCC(C1)N2C(=O)CNS(N)(=O)=O 78067,CCC(C)CCCCC(=O)NC(CN(C(=O)CN1CC2CC2C1)CC)CC 78068,c1(C(=O)NC2(C)CN(C(C3N(CC(C)C)CCC3)=O)C2)cc2ncccn2n1 78069,N1(C(c2c(C)ncs2)=O)C2CCC1C(CNC(c1cnn(C)n1)=O)C2 78070,N1(C(c2cnc(C)o2)=O)CC(NC(c2ccnc(N(C)C)c2)=O)CCC1C 78071,c1(-c2c(-n3cc(CO)nn3)cccc2)nnc2ccccn12.C1CCN(Br)CC1 78072,C(=O)(CC(Cc1ccccc1)NC(c1c[nH]cc1C(C)C)=O)OC 78073,C1(NC(CN(CCCCCC)C)=O)(CNC(c2ccsc2Cl)=O)CCCCCC1 78074,C=CCC(CC=C)C(=O)NCc1ccc(C(=O)NC2CCCCCC2F)nc1 78075,C(=O)(C(C)(C)C1CCCCO1)N1CC(CCNC(C(c2ccc(Cl)o2)C)=O)C1 78076,C(C)(C)(CCCCC(=O)NC1CC2CCC1C(NC(C1CCC(C)O1)=O)C2)OC 78077,c1(C(=O)OCC)[nH]c(C)c(C(=O)NC2(CNC(C3CC(O)CN3C)=O)CC2)c1C 78078,c1(C(N(CCNC(Cn2cccc(N)c2=O)=O)C2CC2)=O)cnc2ccnn2c1 78079,c1(NC(N2CCC(C(=O)O)C2)=O)ccc(S(=O)(=O)NC2CCCC2)cc1 78080,C1(N(CC(CCCC)CC)C=O)COc2ccccc2C1 78081,c1(CNC(C2(C)CCCO2)=O)ccc(-c2ccccc2)c(F)c1.C12CCN1C2=O 78082,c1(C(=O)NC(CN(C(C2(C#C)CCOCC2)=O)C)C)ccc(C)c2c1CCC2 78083,C(=O)(CC(CNC(=O)Cc1cccnc1F)OC)NCc1cc(C(=O)OC)no1 78084,C1(CNC(C2CC=CCO2)=O)CCCCN1C(=O)Cc1ccccc1 78085,c1(C(N2CC(NC(c3c(C)ocn3)=O)C(C#N)C2)=O)c(F)c(F)nc(F)c1F 78086,c1(CNC(C(c2ccc(F)cc2)OC)C)cc(S(C)(=O)=O)ccc1F 78087,c1(C(=O)NC(c2cn(CCCC)nn2)C)c(C)nn2ccccc12 78088,CCCCC(CC)CC(=O)NCC(C)=CC(=O)NCc1ccccc1Cl 78089,Cc1cc(CC(N2CCC(CCC(=O)NCC(n3ccnn3)C)C2)=O)no1 78090,N1(C(c2cc(CCC)[nH]n2)=O)CCC(C(F)F)(CNC(C2C(F)(F)C23CC3)=O)C1 78091,c1(C(=O)NC(C(C)O)C2CCCC2)c[nH]nc1CNC(c1cccs1)=O 78092,c1(C(c2ccc(CS(=O)C(c3ccccn3)C)cn2)C)ccc(C#N)cc1 78093,c1(C(=O)NC2C(SC)CN(C(c3cccc(F)c3N)=O)C2)ccc(F)c(C)c1C 78094,CCCC(CCC)=CC(=O)NC1(CNC(C2CNC(=O)C2)=O)CCC1 78095,c1(C(=O)NC(CN(C(c2ccon2)=O)CC)C)cn(C)c2c(cnn2C)c1=O 78096,c1(C(=O)NC(CNC(C(=O)NC(C)(C)C)=O)CO)cccc(OC(F)F)c1 78097,C1(NC(c2n[nH]c(C)c2Cl)=O)CN(C(C2(C3CCC3)CC2)=O)CCC1CO 78098,C#CC(CC(C)C)NC(=O)CCC1CCN(C(C2CCC(=O)NC2)=O)C1 78099,C12(C(=O)NC3(C)CCN(C(C4CCCCCC4)=O)CC3)CCCN1CC(O)C2 78100,c1(C(N2CC(C)(NC(C=CSC)=O)C2)=O)ccnc(S(N)(=O)=O)c1 78101,c1(C(N2CC(CCNC(=O)CCF)(OC)C2)=O)nn(C)c(C)c1Br 78102,c1(C(N2CCC(OC)(CNC(c3oncc3C)=O)C2)=O)cc(C)[nH]c(=NC)n1 78103,C1(OC)(CNC(c2nc(Cl)cs2)=O)CCN(C(C2CCC(C)C2)=O)CC1 78104,N1(C(C(C)(C)N=[N+]=[N-])=O)CCC(C(=O)NCC(F)C(C)(C)O)=C(F)C1 78105,N1(C(C(CC=CC)C)=O)CCC2C(C1)CN2C(c1cc(C)cc(OC)c1N)=O 78106,C1(NC(CCC2(OC)CCCC2)=O)CC2(CCCCC2)C1.C1=CCNC1=O 78107,c1(CN2CCCC(CC(=O)NCCCn3cncn3)CC2)ccc(F)c(F)c1Br 78108,N1(C(CC(C)=C(C)C)=O)CCC(CF)(NC(=O)Cc2cc(C)no2)C1 78109,c1(CCC=C)ccccc1C(=O)NCC1COCC1NC(=O)CC1CC12CC2 78110,n1(CC(=O)NCC(CNC(c2c(C(C)(C)C)c[nH]c2)=O)(C)C)cccnc1=O 78111,C1(C(N(C2CCN(C(c3nc(OC)ccc3C)=O)C2)CC)=O)CC(=O)NC(C)C1 78112,C1(CNC(C=Cc2cn(C)nn2)=O)CC2CCC1N(C(=O)CC1(O)CCCC1)C2 78113,C(CC(C)(C)COC)NC(CNC(C(CC)SC)=O)=O 78114,N1(C(Cc2c(CC)nccc2)=O)CCCC(C)C1CCN 78115,c1(C(=O)NCC2C(NC(c3c(C)ncnc3)=O)C2)cc(C)c2[nH]cnc2c1 78116,c1(OC)ccc2c(c1)OC(C(=O)OC(=O)COC1CCCC(C)C1)C2 78117,C(=O)(CCCN=[N+]=[N-])NCC12CC(NC(CC3(C)CC3F)=O)(C1)C2 78118,N1(C(C(C)O)=O)CC(CNC(c2ccnn2CC(F)F)=O)CC(C)(C)C1 78119,C(=O)(N=c1[nH]onc1-c1ccc(Br)cc1)N(CC(C)C#N)C 78120,c1(N2CC(COC)OCCC2)[nH]c(=NCCCc2n[nH]c(=N)s2)nc2scnc12 78121,C1(C)(C(=O)NC(C(C(=O)NCc2c(C)cccc2)C)C)CC2CCC1C2 78122,Cc1c(Cl)ccc2c1CN(C(C1CC13CCOCC3)C(=O)NCCC#N)CC2 78123,c1(CC2CCN(C(c3cnc(C(C)C)s3)=O)C2)ccc(Cl)cc1 78124,C1(CNC(CCC=C)=O)CCN(C(C2(CC3CCCC3)CCCC2)=O)C1(C)C 78125,c1(CNC(c2cc(CC)c(C)cc2)=O)c(C)c2ccccc2n1C 78126,c1(CC(N2CCCC(C)(c3cn(CC(=O)OC)nn3)C2)=O)cnc2cc[nH]c2c1 78127,c1(Cn2c(C)c(NC(=O)C(C)OC3CCCC3)cn2)cccc(Cl)c1Cl 78128,C1(C(=O)NC2(C)CC(NC(C3(OCC)CCOC3)=O)C2)Cc2ccccc2C1C 78129,CC(CNC(=O)C(C)N(C(c1ncccc1Cl)=O)C1CC1)C(F)(F)F 78130,c1(NC(c2ncccc2NCc2c(F)cc(F)cc2F)=O)ncc2sccc2n1 78131,N1(C(c2cnc(C)[nH]2)C(=O)NC(C(=O)OC)C)CCC(CF)CC1 78132,C(=O)(NN=c1[nH]c2ccccc2[nH]c1=S)c1nc2ccc(NC(C)=O)cc2[nH]1 78133,C#CCCC(C(=O)NCc1ccc(OC)cn1)NC(=O)CC(C)(C)OC 78134,c1(OC)cccc(CC(=O)N(C2CCN(C(=O)CCc3c(C)c[nH]c3C)C2)C)c1 78135,C(=O)(CCC(=O)NC1(CC(=O)OC)CC(F)C1)N(CC)CC 78136,CCCCCC(C)(C)C(=O)N1CCCC(C2(NC(c3cn(CC)nn3)=O)CC2)C1 78137,C1(CNC(CCC)=O)CCCCC1NC(=O)C=CCN1CCCC1 78138,N1(C(CCN(C)CCN)=O)CCC2(CC1)C(=O)Nc1cc(Br)ccc12 78139,c1(C(=O)NCC2(C)CCC(NC(c3cn[nH]c3)=O)C2)ccc(N)c(Cl)c1 78140,C(=O)(C#CC1(C)CC1)Nc1ccc(OC(C)C)nc1 78141,c1(OC)c(C(=O)N(C(C)CNC(=O)CN(c2ncccn2)C)C)cccc1C 78142,N1(C(c2n(C)ncc2)=O)CCC(C2OCCC2C(N2CCCC2(C)C2CC2)=O)CC1 78143,C1(NC(C2(CCCC)CC2)=O)CCN(C(=O)CN2CCC(C)C2)CC(C)(C)C1 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78162,C1(C(=O)NCCC(CC)C)CCCC(NC(=O)Cc2cccnc2C)C1 78163,C(C)(CC(C)CC)NC(c1nc(CNC(C2(C(CC)=O)CC2)=O)oc1)=O 78164,C1(NC(c2c(OC)n(C)nc2)=O)CC(O)CN(C(C2(O)CCCCCC2)=O)C1 78165,c1(CC(=O)NCCN(C(c2cn[nH]c2F)=O)CC)n[nH]nc1C 78166,C(=O)(C(C)CC(N)=O)N1CCC(NC(c2c(C)nsc2C)=O)C1 78167,C(=O)(CCCC(C)(C)C)N1CCCN(C(C2N(CC)CCCC2)=O)CC1 78168,CCCC(CC(C)C)C(=O)NC1CC2CC(NC(=O)CSCc3ncc[nH]3)C1C2 78169,c1(N(CCCC)C)nc(-c2ccccc2)nc(=NC2CN(CCOC)C2)[nH]1 78170,N#Cc1ccc(F)cc1C(=O)N(C1CCC2(CC1)CNC2)c1cccnc1 78171,C(=O)(CC(O)CNC(=O)C(c1ccccc1)O)N(CCC)CCC 78172,O=S(=O)(CCO)CCCCCc1nc(C2CCCOC2)no1 78173,C1(C)(CNC(c2ccn(C)n2)=O)CCCN(C(C2CCC3(CC2)CC3)=O)C1 78174,S(=O)(=O)(CCC(=O)N1CCC12CN(C(C1(C)CCOC1)=O)C2)N(C)C 78175,c1(NC(CCN(CC#C)CC2CC=CCC2)=O)ccc(C)nc1 78176,N1(C(C(CC#C)NC(c2ccn3cncc3c2)=O)=O)CC(=O)N(C)C(C)C1 78177,N1(C(C=Cc2ccc(C)nc2)=O)CCC(C2CC2)(CNC(=O)CSC(F)(F)F)C1 78178,c1(CC)cc(C(N2CC=CC(NC(=O)C(C)SC(C)C)C2)=O)ccn1 78179,Cc1ccc(-c2ccc(C(F)(F)F)nc2)cc1NCC1CC(C)OC(C)C1 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78197,n1(-c2c(C(N3CC(CO)OCCC3)c3cccs3)cccc2)nnc2ccccc12 78198,c1(CCC(=O)NCC(CNC(C(COC)(C)C)=O)CO)ccc2ncsc2c1 78199,CN1CC(CNC(C2(C)CCN(C(C3CC(=O)CCO3)=O)C2)=O)CC1=O 78200,C(=O)(C(C)(CC)CCCCC)N1CCC(C(C)NC(C(CC=C)(C)C)=O)C1 78201,CC1CCOCC1C(N1CC(C(=O)N(CCN=[N+]=[N-])C)C1)=O 78202,Cc1ccsc1C(=O)N(C1CC1)Cc1cn(Cc2ncoc2C(F)F)nn1 78203,c1(NC(C2COCCN2C(=O)C=Cc2ccc(Cl)cc2)=O)ccc(Br)c(Cl)c1F 78204,C1(CNC(CCN(C(C)=O)C)=O)CN(C(=O)CN(C2CCCC2)C)CC12CCC2 78205,c1(C(=O)NC2CCC(CNC(c3cncc(SC)c3)=O)C2)cc(O)nc(O)n1 78206,c1(C(N2C(C(C)NC(=O)COC3(C)CCC3)CCC2)=O)ccc(F)cc1F 78207,C1(CCC)CN(C(=O)C(C)COC)CC1C(=O)N(CC(C)COC)C 78208,C1(C2CCN(C)CC2)(C(=O)NC2CCN(C(CCOCC#C)=O)C(C)C2)CC1 78209,c1(CN(C(c2ccc(Cl)nc2NS(=O)(=O)C2CC2)=O)CC)ccc(F)cc1F 78210,c1(CC)oncc1C(N1CCC(CNC(C2CC(C)(F)C2)=O)C1)=O 78211,c1(C(=O)NC2C(CNC(C(C)(F)F)=O)C2)cnc2cc(Br)ccn12 78212,C(=O)(C1CCCn2nccc21)NC(CCNC(C(F)=C(C)C)=O)C 78213,N1(C(C2N(C(=O)C(C#N)C(C)(C)C)CCC(=C)C2)=O)CC2(CCC2)C12CCC2 78214,c1(C(N2CC(COc3cccc4ccccc34)C2)=O)cc(=NC(=O)OC)[nH]n1C 78215,N1(C(C2(NC(=O)Cn3ccccc3=O)CC(O)C2)=O)Cc2c[nH]nc2C1 78216,CC1CS(=O)CCN1C(C1CN(C(C2CNC(=O)N2)=O)CCN1C)=O 78217,c1(C(=O)Nc2cccc(NC(C(CC)(C)COC)=O)c2)cc(F)c(O)c(Cl)c1 78218,Cc1cc(NCC(C)NC(c2cncc(C)c2Cl)=O)n2nc(C)cc2n1 78219,C1(NC(c2n(CCC)ccc2)=O)CCOCC1C(N1CCC1(C)C)=O 78220,N1(C(C2N(C)CCC2)=O)CC(C2CC2C(=O)NC2CC(n3ccnn3)C2)C1 78221,c1(C(=O)OC)cc(C(=O)NCC(O)CNC(c2cnc(C(C)(C)C)s2)=O)c[nH]1 78222,N1(C(CC(CC)C)=O)CCC2(CCC(NC(=O)CCCCc3ccccc3)C2)C1 78223,c1(CC)nc(C(N2CCC(C(C)N(C)CCCNC(=O)CCSC)C2)=O)n[nH]1 78224,C=C1CCC(C(=O)NC(CN(C)C)C(=O)NC2(COC)CC2)CC1 78225,CCC(CCC(=O)NCC(C(C)C)OC)NC(C1(C)CC1C)=O 78226,C(c1ccc([N+](=O)[O-])cc1)=C(C)C(=O)NCCN(C(=O)CCCC(N)=O)C(C)C 78227,Cc1ccnc2nc(-c3nc(-c4cc(Br)c(Cl)cc4[N+](=O)[O-])no3)nn12 78228,N1(C(C(C2CCN(C(c3ccoc3C(C)C)=O)CC2)C)=O)CC2(CCNC2=O)C1 78229,c1(C(N2CCC(NC(C(C#C)(C)C)=O)CC2)=O)c(F)ccc(C(=O)OC)c1C 78230,c1(C(N2CC(N3CCN(C(c4cc(C)oc4)=O)CC3)C2)=O)cc(S(N)(=O)=O)co1 78231,N1(C(C=CC=CC)=O)CC(O)(C2CCN(C(C3(C)CCCC3CC)=O)CC2)C1 78232,N(C(=NCC1CCCO1)NCc1cccnn1)C(C1CCCCC1)C 78233,C1(CNC(CCC=CC)=O)C2CCC(C2)N1C(c1ccc(F)c(F)c1)=O 78234,N1(CC(=O)Nc2ccccc2)CCC(NCCCC(=O)Nc2cnc(C)[nH]2)CC1 78235,N1(C(c2[nH]cc(C)c2)=O)CCC2(CCN(C(=O)CC(C)NC(N)=O)C2)C1 78236,c1(CC(C)C)cc(C(N2CCCC2C2(O)CN(C(C3CC3C(F)F)=O)C2)=O)n[nH]1 78237,C1(NC(C2(O)CC(C)(C)C2)=O)CN(C(C2CC23CCOC3)=O)C2CCCCC12 78238,C1(C#N)(C(N2C(CCOC)COCC2)=O)CC12CCC2 78239,CC(C)N(O)C(=O)C(=O)N1CC(C)(C)OCC1CNC(=O)C(C)N(C)C 78240,C1(NC(=O)CN2CC3CC3C2)CCCC(NC(C2CCC(F)(F)C2)=O)C1 78241,C1(NC(c2ccncc2F)=O)CCN(C(=O)C2CC2)C12CC2 78242,c1(NC(C2CCN(C(C3C(OC)(OC)CC3)=O)C2(C)C)=O)ccc2c(c1)OCC2 78243,CS(=O)(=O)c1cccc(-c2noc(-c3csc(-c4ncccn4)n3)n2)c1 78244,c1(OC)cc(C(C(=O)NC2CCC2)N(Cc2cncs2)CC2CC2)cc(C)c1 78245,c1(C(=O)NC2C=CC(CNC(C3ON=C(CC)C3)=O)C2)cc(F)c(Cl)cc1F 78246,C1(NC(C2COCCO2)=O)CN(c2ncnc3sccc23)C2CCCCC12 78247,N1(C(C2(CCC)CC2)=O)CCC(CNC(c2cn(C3CC3)cn2)=O)C(O)C1 78248,c1(C(N2CC(C)(NC(CCCC)=O)C2)=O)cnn(C2CCOCC2)c1C 78249,c1(SC(C)C(N2CC(NC(C3CCS(=O)CC3)=O)C(C)C2)=O)ccc(F)c(F)c1 78250,N1(C(C2CC(C#N)(OC)C2)=O)CC2CN(C(c3ncoc3C3CCC3)=O)CCC12 78251,CC(C)(C)C(=O)NCC1CC(NC(C2CCCSC2)=O)C1 78252,CC1CCN(C(=O)CC2N(C(=O)CC3CCCNC3=O)CCC2(C)C)CC(C)O1 78253,C1(NC(CC=C(C)C)=O)CC2CN(C(=O)C(C)(C)COC(C)C)CC2C1 78254,N1(C(C(C(CC)C)=O)=O)CC(C(=O)NCCC(=O)OC)C2(CCC2)C1 78255,N1(C(C2C=C(C)CS2)=O)CC(C2CC2C(=O)NCC2CNC(=O)C2)C1 78256,N(C1CCCn2ccnc21)C(C(CCC1CC1)NC(C1CCCCS1)=O)=O 78257,c1(C(=O)NCC2C(NC(=O)COc3cncc(Cl)n3)C2)cnc2n1CCC2 78258,n1(CC)cc(NC(=O)CC2(C)CCN2C(C2CN(C)C(=O)N2)=O)ccc1=O 78259,N1(C(CCC)=O)CCCC(CCNC(=O)Cc2nn(CC)cc2Br)C1 78260,c1(N2CCC(CC#N)C2)ccc(S(=O)(=O)N2CCN3CCC2CC3)cc1Cl 78261,c1(CC(=O)NCC2CCN(C(C(COCC)C)=O)C2)cc(Br)ccc1C 78262,N1(C(CCSCC)=O)CCC(C(F)CNC(=O)C(O)COC)CC1 78263,c1(NC(C2N(C(C=CC=CCC)=O)CC(O)CC2)=O)cncc([N+](=O)[O-])c1 78264,Cc1ccc(N(C(=O)CCC2NC(=O)NC2=O)C)cc1C 78265,c1(CC2(C(=O)NC34CC(NC(C5C(CC)C5)=O)(C3)C4)CC2)ccc(F)cc1 78266,c1(C(=O)NCC(CC)NC(c2cn(C(C)(C)C)nn2)=O)c[nH]c(C)c1 78267,C1(CC(=O)NCCc2ocnc2CNC(=O)C(O)CC2CC2)CC(O)C12CCC2 78268,C1(O)(C(C)NC(c2ccnn2C)=O)CCN(C(=O)C=Cc2cnn(C)c2)CC1 78269,C(=O)(C1CCc2ccc(Cl)nc21)NC1CN(C(C(N)=O)=O)CC1CC(F)(F)F 78270,CC(C)(C)CC(F)C(=O)N(C1(CNC(C2CC(C(C)(C)C)C2)=O)CCC1)C1CC1 78271,c1(C2C(C)C2)ccc(C(=O)N(C)CCN(C)C(c2csc(Cl)n2)=O)o1 78272,c1(NC(=O)CC2CN(Cc3cc(O)cc(Cl)c3)C2)cccc([N+](=O)[O-])c1Br 78273,C1(C(N(CC(=O)OCC)C)=O)CCCCN(C(=O)C(C)(C#N)CC)C1 78274,CC1=C(C(=O)N2CCC(CF)(NC(=O)CCc3cc(C)cc(C)c3)C2)SCCO1 78275,Cc1ncc(C(=O)NC2CN(C(C3C(C)C3C)=O)CC23CC3)cc1N 78276,CC1(C)CCc2ccccc2C(NCC2COC(=O)O2)C1 78277,C1(=CC(=O)N(C)CC2N(C(c3c(C)oc(CO)c3)=O)CCC2)CN2CCC1CC2 78278,Cc1ncc(C(N2CCC2CNC(C2CC23CCCC3)=O)=O)cc1C(F)(F)F 78279,C1(C(N(C(C)CCNC(C2(NC(N)=O)CC2)=O)C)=O)COC(c2ccsc2)C1 78280,n1(C(C)C)cc(Br)c(C(=O)NCC23CC(CN2C(=O)C(C)C#N)C3)n1 78281,c1(N2CCC(C)(CNC(c3cnc(Br)s3)=O)CC2)ccncc1[N+](=O)[O-] 78282,CC1(C)CC(NC(C2CCCS2(=O)=O)=O)CN1C(c1csc2nnsc12)=O 78283,CCCC(C(=O)NC(CN1CCCC1)CO)NC(=O)C(F)COC 78284,CC(C(=O)N(CCCCNC(=O)C1=NOCC1)C1CC1)C(C)(C)c1ccccc1 78285,CCCCC(C(=O)NC(C)CNC(C1CCCN(C(=O)OC)C1)=O)N(C)C 78286,CCCC(C)(CCC)C(=O)NC(C1CN(C(=O)Cc2ccc(C)nc2)CCO1)C 78287,N1(C(c2noc(C)c2[N+](=O)[O-])=O)CCCCC(C2CN(C(C3(F)CC3)=O)C2)C1 78288,C(CC(CC)C(=O)N(CC(=O)NCC(C)(C)O)CCOCCN(C)CCO)=CC 78289,N1(C(Cc2ccc(C(=O)OC)nc2)=O)CCCC(NC(=O)C(F)C(C)(C)O)C1C 78290,c1(OC)cc(OC)cc(C=CC(=O)NC2CC(CNC(c3ccncc3)=O)C2)c1 78291,c1(OC)ccc2c(c1)C(N(C)C(c1cc(C)c(Cl)s1)C(=O)NCCCF)CC2 78292,C1(C(=O)NCC2(OC)CN(C(C3CSCC(=O)N3)=O)C2)CCC2CCCCN12 78293,Cc1ccc(C(N2CC(O)CC2(C)C(=O)NCCCF)=O)nc1C 78294,c1(C(C(F)(F)F)NCc2cn(CC(=O)OCC)nn2)ccc(F)c(Cl)c1 78295,C12(C(N)=O)CCCC1(C(=O)NC1CCCC1NC(c1nncs1)=O)C2 78296,C1(C(=O)NCc2ncc[nH]2)COCCC12CN(C(c1ccnc(Cl)n1)=O)C2 78297,N1(C(c2cc(CC)ncn2)=O)CCCC(O)(CCNC(c2ccc(Cl)o2)=O)C1 78298,c1(C(=O)NC(CNC(C2N(CCC)C(=O)CC2)=O)CO)ccn2nnnc2c1 78299,N1(C(C=C(C)c2cccs2)=O)CCC(CO)(NC(=O)CCN2CCOC2=O)CC1 78300,C(=O)(C1CCCc2sccc21)N1CC(CNC(c2c(C)cno2)=O)OC(C)(C)C1 78301,C1(OC)CCC(C(N2CC(F)CC2CC(=O)NCC(C2CCCC2)O)=O)CC1 78302,c1(C(=O)NC(n2cccc2)(C)C)cn(C2CCOC2)nn1 78303,C(CC(=O)N(C(C)CN(C(=O)C(C)n1cncn1)C)C)OCCC 78304,c1(OC)ccc(C(=O)CCC(=O)N(CCNC(=O)C(O)C(C)C)C2CC2)cc1 78305,c1(C(N2CCCC(n3nccn3)C2)C(=O)NC2CC2)csc([N+](=O)[O-])c1 78306,c1(C(C)C)cnn(C)c1C(=O)NCC1CCN(C(=O)CCCCc2cnc[nH]2)C1 78307,C(=O)(C(C)(C)CCCF)N1CCC(C2N(C(C3=CC(C)(C)C3)=O)CCC2)CC1 78308,C(=O)(C1CCCn2cnnc21)NCC(CO)NC(Cc1ccc(OC)cc1)=O 78309,c1(OC)cc(C(C)NC(=O)NCCCCN2CCC2)sn1 78310,c1(C(N2CC(NC(c3ccc(OC)c(C)n3)=O)C(C)C2)=O)c(C)cc(Br)cc1C 78311,CC1(C)C2CCC(C2)C1C(N1CC(NC(C2CC(O)C2)=O)C1)=O 78312,c1(OC)cc(C(N2CC(CNC(=O)C3=CC4CCCC34)CC2C)=O)cc(N)c1N 78313,c1(OC)ccn2cc(C(N3CC=CC3CNC(c3cc(Cl)c[nH]3)=O)=O)nc2c1 78314,c1(C(N2CCC(NC(c3nn(CC)c(O)c3)=O)C(C)C2)=O)c(N)cc(F)cc1Cl 78315,CC(C)C1=NOC(C(=O)NCc2nnn(C)c2C(=O)N(CCC(C)(C)O)C)C1 78316,C1(NC(c2cnn(C)n2)=O)CCCCC12CCCN(N1CCC1C(=O)N(C)C)C2 78317,c1(C(N2C3C(NC(=O)C(F)n4ccnc4)C(C3)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 78318,c1(C(=O)NC2CCC(CNC(C3C(C)(C)C3(F)F)=O)C2)cc(F)ccc1F 78319,c1(NC(C2C(C)C2)=O)cncc(NC(=O)CNC(=O)Nc2ccccc2F)c1 78320,C(=O)(C1=CNC2=NCCCC2=C1)N(CC(CO)(CO)NC(CSC(C)C)=O)C 78321,CC1CCC(CNc2ccccc2)CN1 78322,N1(C(c2cc(Cl)ncc2O)=O)CC2CC(C1)N(C(c1coc(O)n1)=O)C2 78323,C1(NC(c2ccc(C)cn2)=O)CCN(CCCNC(c2ccccc2)=O)CC1C 78324,C1(CNC(C(COC)(C)O)=O)CC2CCC1N(C(c1cnn3c1OCC3)=O)C2 78325,c1(C(C)NC(C(c2ccccc2C2CCC2)N(CC)CC)=O)cccc(C#N)c1 78326,C(=O)(C(F)(F)C(C)(C)O)NCC(=C)CCNC(=O)C(c1ccccc1)F 78327,N1(C(c2c(OC)csc2)=O)CCC2(NC(=O)CCCCC(C)C)CCCCCC12 78328,C1(NC(CCC(C)OC)=O)CN(C(c2cnc(O)c(C)c2)=O)CCC1(C)C 78329,Cn1cc(C2CC2NC(=O)CCCn2cc(CCC3CCCCC3)nn2)cn1 78330,C1(CC)CCN(C(C)=O)C1C(=O)N(CCNC(C1CCCN1C(N)=O)=O)CCOC 78331,c1(C(=O)NC2C(NC(c3sccc3C3CC3)=O)CC2)cn2c(n1)CCC2 78332,C#Cc1ccc(C2(C(=O)OCC(C)(C)C(=O)OC(C)C)CCCC2)cc1 78333,c1(C(=O)NCC2(C)CCN(C(c3c(C(C)C)cco3)=O)C2)ccc(N)c(Cl)c1O 78334,C(=O)(C(F)(CNC(C1(C)CCC(=O)C1)=O)C(C)C)N(C(C)C1CC1)CC 78335,N1(C(Cn2cc(CNC(=O)C=CC3CCCCC3)nn2)=O)CC2CCC(C1)O2 78336,C1(C(=O)NCC2C(C(=O)NCC(C3CC(C)(C)C3)O)C2)CCNC(=O)C1 78337,c1(C(N2CC(CNC(C3C(=C)C3)=O)CC23CCC3)=O)csc2cccc(F)c12 78338,CC(C)CCCC(C)CNC(=O)C(F)CC1CN(C(C2CC2[N+](=O)[O-])=O)C1 78339,c1(OC)cccc(CNC(C2CCCN(C(=O)COCC3CC3)C2)=O)c1C 78340,C(=O)(C#CC1CCCOC1)NC1(CNC(C(COC)CC(C)C)=O)CC1 78341,c1(OC)ccc(NC(=O)C(CNC(C2CN(C)CCO2)=O)N(C)C)cc1O 78342,C(=O)(CC(C)CC(=O)N(C(CC(F)F)C(=O)NCC1=C(C)CCC1)C)OC 78343,N1(C(c2ccc(COC)o2)=O)CCC2C1CCCN2C(=O)CCN(C)CCO 78344,C12(C(N(CC)Cc3cccc(Br)c3)=O)CCNC1CNCC2 78345,CC1CC(=O)NCCN1C(=O)CC(C1CC1)NC(C1(CO)CCCC1)=O 78346,N1(C(C23CC(CC(C)O2)C3)=O)CC2CCCC(C1)N2C(=O)CCc1ncc[nH]1 78347,c1(C(=O)NC(CNC(c2ccc(C)s2)=O)(C)CO)cc(C(C)(C)C)[nH]c1C 78348,C1(N(C)C(c2cnnn2C)=O)CC2CCC(C1)N2C(C1CC1F)=O 78349,C1(C(=O)Nc2ncco2)CC12CCN(C(c1cccc(-c3ncccn3)c1)=O)C2 78350,S(=O)(=O)(CCC(=O)NC1CC(NC(c2ccc(Cl)c(N)c2)=O)CC1O)NC 78351,C1(C(N(CCNC(C(F)=CCC)=O)C)=O)CC(CC)=NO1 78352,CCC(C)CC(C(=O)N(CC1=CCCOC1)C)NC(C12CCC(OC)C1C2)=O 78353,C1(NC(c2cc(OC)ncn2)=O)CCCN(C(=O)OC(C)(C)C)C1C 78354,c1(C(=O)NCC2CCCN2C(=O)CC2CCC(O)CC2)ccc2ccoc2c1 78355,C(=O)(CC(C)CC(C)(C)C)NCC(CC)(CC)NC(C1CC(O)CN1C)=O 78356,N1(C(C(CC)n2cccn2)=O)CCC(NC(=O)CCCn2ccnn2)CC1 78357,C12(NC(=O)C(C3CCOCC3)O)CCCC1N(C(=O)CCc1ccon1)CCC2 78358,N1(C(C23CC(COC)(OC2)C3)=O)CCC2CN(C(=O)C(O)P(C)(C)=O)CC2C1 78359,c1(C(=O)NCCNC(C(C(C)C)SCC)=O)ccc(C)c(C#N)c1 78360,c1(CC)cc(C(N2CCC(C)N(C(=O)COC(C)=O)CC2)=O)c2c(c1)CCO2 78361,CC1CCC(NC(=O)C=C2CCCC2)CN1C(c1cc(Br)n(C)c1)=O 78362,c1(C(CNC(=O)NC(CC)C(F)F)CC)ccc(F)c(F)c1 78363,N1(C(c2nc(CC)oc2)=O)CC2CN(C(C3CCOC3)=O)CC2C1 78364,N1(C(c2cc(C3(C)CC3)n[nH]2)=O)CC(CNC(=O)CC2CC2)C(C(F)F)C1 78365,c1(CC)nc(NC2(C(N)=O)CCCN(C(c3sccc3OC)=O)C2)cc(C)n1 78366,c1(OC)cc(CN2CCCC(C(=O)N(C)C)C2)ccc1S(C)(=O)=O 78367,C1(OCC)CCCN(C(=O)CCC2(CN)CCCCC2)C1 78368,C1(CC=C)(NC(=O)CCN2CCCC2)CCN(C(C2(CSC)CCC2)=O)C1 78369,C1(CNC(=O)C=CCN2CCCC2)(NC(C2COC(=O)N2)=O)CCOC1 78370,c1(CC)cccc(C(=O)NC2(CNC(=O)C(C3CCCC3)OC)CCOC2)c1O 78371,CC1CCN(C(c2coc(OCC(=O)OC(C)(C)C)n2)=O)CC1CN(C)C 78372,CC(C)CCCC(C)C(=O)NCC1(NC(C2COC(=O)C2)=O)CCCCC1 78373,CCC(C)(C(=O)NCc1cc(C(N2CCC(C(=O)OC)C2C)=O)ccn1)OC 78374,c1(N2C(CNC(C(C)C)=O)CC(F)C2)cc(-c2cccs2)ncn1 78375,c1(C(N2C(CNC(=O)C=CCN3CCCC3)CC(OC)C2)=O)cc2cnccc2o1 78376,c1(COC)cc(C(=O)NC(C2CCCN(Cc3cnc(Br)s3)C2)C)ccn1 78377,C(=O)(C1=CCCC1C)N(CC(C)O)CCNC(c1ccc(C2CC2)o1)=O 78378,Cc1cc(C)c(CCNC(=O)C(C)Oc2ccc(C(C)(C)C)cc2)s1 78379,CC1CN(C(c2cnc(Cl)s2)=O)CC(C)N(C(c2cc(F)ccc2O)=O)C1 78380,c1(-c2cnc(OCC)c(C)c2)cc(C(=O)NC(C)C(N)=O)cc2[nH]ccc12 78381,n1(CC)cc(C)c(C(N2CCC(C3CCCN3C(=O)CCC(C)C)C2)=O)n1 78382,Cc1ccc(=N)[nH]c1C(N1CC(NC(=O)C(C)(C)c2cnsc2)CC1C)=O 78383,N1(C(c2cnc(C)s2)=O)CCCN(C(c2coc(Cl)c2)=O)CC1CO 78384,Cc1nn(CC(F)F)cc1C(=O)NCC1CC1NC(=O)C(c1ccc(F)cc1)F 78385,C1(NC(C(C)(C)OC(C)C)=O)CCCC(NC(c2cncc(C(C)(C)C)c2)=O)C1 78386,C(CC(=O)N1CC2CN(C(c3ncccc3F)=O)CC2C1)(C(F)(F)F)OC 78387,CCC(O)C(C)C(=O)NC1CN(C(=O)CSc2cn[nH]c2)CC1C(F)F 78388,C1(N(C(C(c2ccnn2C)NC(CNC(CN(C)C)=O)=O)=O)C)CCC(F)(F)C1 78389,N1(C(C2C(NC(CC(COC)(C)C)=O)CCCC2)=O)CCc2ccncc21 78390,N1(C(C=CC=CCC)=O)CC2(CCC2)CC1CNC(c1cnccc1Br)=O 78391,C(CCC(C)CC(=O)NCCNC(c1cccc(O)c1F)=O)=C(C)C 78392,C(=O)(C1CCCc2nnn(C)c21)N1C(CN(C)C(c2n[nH]cc2Cl)=O)CCC1 78393,C1(F)(CNC(c2n(CC(C)C)ncc2)=O)CCN(C(c2nc(=O)n(C)[nH]2)=O)CC1 78394,N1(Cc2n(CC(F)(F)F)cnn2)CCC(S(=O)(=O)NC2=NCCCCN2)C1 78395,c1(CNC(C2C(C(=O)Nc3ccccc3CCO)C2)=O)c(Cl)cccc1[N+](=O)[O-] 78396,C1(O)(C(=O)NC2CCC(CNC(c3c(C)ccnc3C)=O)C2)CCC(C)(C)CC1 78397,N(C(=NCCC(C)C)N1CCC(C(=O)N(C)C)C1)Cc1onc(C)n1 78398,N1(C(C2CC(C3CN(C(CCCC4C(C)C4)=O)C3)C2)=O)CCC(O)C(F)C1 78399,CN1N=C(C(=O)NC2CC(F)(CNC(C3CCCCS3(=O)=O)=O)C2)CCC1=O 78400,N#Cc1ccc(CC(N2CC3CC2C3NC(c2cnccc2C(N)=O)=O)=O)cc1 78401,C(=O)(C1=CCCC1C)NCC1(COC)CCCN1C(=O)CCS(C)(=O)=O 78402,N1(C(c2ccc(CC=C)cc2)C(=O)NCC(=C)C)CCOCC1C=C 78403,c1(Cn2cc(C(=O)NCC3(NC(C4(C)CCCS4)=O)CC3)nn2)cccc(F)c1 78404,c12ccc(cc1)NC(=O)C(=O)N1CCC1C2.c1(C2(C)CC2)ccccc1 78405,c1(C(C)C)noc(CCCC(=O)N(C(CNC(c2nccn2C)=O)C2CC2)C)n1 78406,C123CC1CN(C2)C(=O)NC3.N1(Cc2c(CC)nco2)CC(=O)NC1=O.C1C(=O)O1 78407,c1(C(C)C)ncc(CNCCc2cnc[nH]2)s1 78408,N1(C(C2(OC)CC2)=O)CCC(NC(C2(C(F)(F)F)CC3(CCC3)C2)=O)C(O)C1 78409,CC1(C)OC2CC(C(N3CC(NC(=O)CCCS(C)(=O)=O)C(O)C3)=O)CC2O1 78410,c1(C(=O)NC23C(CN(C(C(C(C)C)F)=O)C2)C3)ccc2c(c1)OCCNC2=O 78411,N1(C(=O)Cc2cn[nH]c2)CC2CCN(C=O)CC(C2)C1.N1(OC(F)(F)F)CCOCC1 78412,C(=O)(C(C1(C)CC1)NC(=O)C(F)OC(F)(F)F)NCC(C1CCC1)OCC 78413,N1(C(N(c2c(C)cc(F)cc2)c2ccco2)=O)C2CCC1CC(CC(F)(F)F)C2 78414,N1(C(C2ON=C(C)C2)=O)CCC2(NC(C3(c4cccs4)CC3)=O)CCCCCC12 78415,CCCCC(CNC(=O)C(C)Cc1cnco1)NC(c1cc(C)nn1C(F)F)=O 78416,Cc1ncncc1C(=O)NCC1CN(C(c2ccnc(Br)c2)=O)CCO1 78417,c1(OC)cc(C(N2CCC(C(N3CC4CCC3C4)=O)C2)=O)cc(OC)c1C 78418,N1(C(C=C(CC)CC)=O)CCC2(CCCC2NC(C2CCS2(=O)=O)=O)CC1 78419,C1(CC)(NC(=O)C(C)OCC(C)C)CCCN(C(c2cc(N)nc(Cl)c2)=O)C1 78420,c1(C(=O)NC(c2ccnn2C)C(=O)NC(c2ccccc2)C)ccc(C#N)cn1 78421,CN1CC(C(N2CCCCC2C2CCN(C(=O)Cn3[nH]cnc3=N)C2)=O)NC1=O 78422,C1(C(=O)NC(c2nocc2C(=O)N(CCF)C2CC2)C)CC=CCC1 78423,C12(C(=O)OC(C(=O)C(F)(F)F)Cc3cccc(O)c3)CCCN1S(=O)(=O)CC2 78424,c1(CC)c(C)noc1CN(CCNC(c1nn[nH]c1C(F)(F)F)=O)CC 78425,Cc1nn(C)c(NC(C2CC2NCc2ccc(Cl)cc2Cl)=O)c1C(N)=O 78426,C1(O)(C(N2C3C(NC(=O)CC4CCCC4O)CC(C3)C2)=O)Cc2ccccc2C1 78427,c1(C(=O)NC(CNC(C2CCC(=C)CC2)=O)CO)cc(C(F)(F)F)ccc1F 78428,c1(OC)cc(C)cc(C(=O)NCC2(O)CN(C(=O)C3=COCCC3)C2)c1N 78429,c1(C(C(=O)NC(C)CC)N(CCCN(C)C)CCC)ncc(C)c(OC)c1C 78430,c1(CCNCCCC2(N)CC2)cc(Cl)c(F)cc1F 78431,C1(C)(NC(CCSCC)=O)CCCN(C(c2cc(Br)cnc2N)=O)C1 78432,C1(CNC(c2ccn(CC)n2)=O)CC2(CCC2)CN1C(=O)Cc1ccsc1 78433,C(c1csc(C(F)(F)F)c1)=CC(=O)NCCC1N(C(CCC#C)=O)CCC1 78434,C1(CNC(c2c(C)snn2)=O)CC(NC(c2cnc(C3CCCO3)s2)=O)C(O)C1 78435,N1(Cc2nc(CCC3(C)CC3(F)F)on2)C(=O)COCC1=O 78436,C1(C(=O)NC2CCN(CCNC(c3c(C)n[nH]c3)=O)CC2)CC(C)CC(C)C1 78437,C1(CC(=O)N(CC(C)NC(c2ccc(COC)s2)=O)C)Cc2ccccc2O1 78438,N1(C(c2cnc(-c3cccc(C#N)c3)s2)=O)CCC2(CC(=O)NC2=O)C1 78439,CC1(C)CCN(C(=O)CNC(=O)C2CC2)CC1C(=O)NCCCn1nccn1 78440,C(N=c1[nH]c(C)c(Br)cc1C(=O)OC)c1ccc(CC(=O)NC)cc1 78441,c1(C(N)=O)c[nH]c(=NC(=O)C2(F)CN(C(c3cccc4nccnc34)=O)C2)cn1 78442,N1(C(C(C)NC(C2CCCC2)=O)=O)CCCC(CNC(c2ccc(F)cc2)=O)C1 78443,C1(C(=O)NC(C2CCCN2C(C2CCCS2)=O)(C)C)CCC2C(C1)C2(F)F 78444,C(=O)(CCS(=O)(=O)N(C)C)NC1(C)CC(NC(c2cc(CC)nn2C)=O)C1 78445,C1(CNC(Cn2ncc(C)c2)=O)CC2(CO1)CN(C(=O)C(N1CCCCC1)C)C2 78446,CC1CN(C(=O)CCc2cccnc2)CC(C)N(C(c2ccc(CO)cc2)=O)C1 78447,C(CC(C)C(=O)NCC1(NC(=O)CCCc2n[nH]c(=N)s2)CCCC1)OC 78448,N1(C(=O)C(c2ccccc2Cl)O)CC(NC(C2(O)CCC2)=O)CC12CCOCC2 78449,CC(=Cn1ccnn1)C(=O)NCCC1(NC(C2CCCN2N=O)=O)CC1 78450,Cc1cc(C(N2C(C(N3CC(F)(CF)C3)=O)CCC2C2CC2)=O)[nH]c1C 78451,C1(NC(CC2N(C(C)=O)CCC2)=O)CC2(CCN(C(c3cc(O)cs3)=O)C2)C1 78452,C1(N(C(c2cccs2)=O)CC)CCCN(C(=O)CSc2ccccc2)C1 78453,C(=O)(C(C)(C)CCCOC)NCCN(C(=O)C(N1CCCCC1)C)CCC 78454,c1(C(N(C)CC2CN(C(=O)C=Cc3ccco3)C2)=O)ccnnc1Cl 78455,N1(C(C2N(C(C(CC3CC3)OC)=O)C(C(C)C)CC2)=O)C2CCC1CN(C)C2 78456,C(CCCCC(=O)NC1CCC1CNC(=O)CC12COC(C)(C1)C2)SC 78457,c1(C(=O)NCc2cn(CCNC3(C(=O)NC)CCCCC3)nn2)ccc(C)cc1F 78458,c1(C(C)C)ccc(OCC(=O)NCC(CC(C)C)NC(C2CCC2)=O)cc1 78459,c1(OC(C(c2ccccc2)C)=O)cccc(OCC(F)(F)F)c1 78460,c1(C(=O)NCC2(F)CC(NC(CCCCOC)=O)C2)cc2n[nH]cc2cc1C 78461,C(=O)(C(O)CCCC)N1CCC(CC=C)(C(N2CC(Cc3ccoc3)C2)=O)C1 78462,c1(CN2CCOCC(C(=O)NC(c3ccc(Br)cc3)C)C2)ccc(C#N)cc1O 78463,N1(C(c2ccc(C(=O)NCC(=O)OC)cc2)=O)CCCCCC2CCCC12 78464,N1(C(CSSC)=O)CC(CNC(c2cc(C(F)(F)F)ncn2)=O)C(O)C1 78465,c1(C(=O)NCC2CC(NC(=O)CC3CSCCS3)C2)ccc(F)c2ccoc12 78466,C1(C(=O)NCC(C)(C)NC(=O)CN2CCSCC2)CCc2nncn2CC1 78467,c1(C(N2C(COC)CN(C(=O)CCS(C)(=O)=O)CC2)=O)cccc(S(N)(=O)=O)c1 78468,CCC(CC(=O)NCCc1ccccc1C)NC(=O)Cc1coc(C)n1 78469,N1(C(C(C(C)C)C#N)=O)CC2CCC1CN2C(c1ccc(C(C)(C)C)cn1)=O 78470,Cc1ccc2c(NC(C3CC3NC(=O)CC(C)CC(C)(C)C)=O)cccc2c1 78471,S(=O)(=O)(c1ccc([N+](=O)[O-])cc1Cl)NCC1CCCN(C(C2(C)CC=CC2)=O)C1 78472,C1(N(C(C(C(C)C)F)=O)C)CCCCN(C(=O)Cc2cncc(Br)c2)C1 78473,c1(C(=O)OCC)cc(Br)cc2c1CCN2C(=O)Nc1nc(Cl)c(C(N)=O)s1 78474,C1(F)(CNC(=O)CSc2ccccn2)CCN(C(C2(O)CCCC2)=O)C1 78475,c1(C(=O)NC(CCNC(C(CCC)N(C)C)=O)C)cc([N+](=O)[O-])n(C)n1 78476,C1(CCF)(NC(COCCCNC(C2C(C)C2)=O)=O)CC(O)C1 78477,Cc1cc(C(=O)NC(CO)CCCCNC(=O)C(C)C(C)(C)C)cc(=O)n1C 78478,c1(C(N2CCN(C(C3CCS(=O)(=O)N3)=O)CC(O)C2)=O)csc2ncnc(O)c12 78479,Cc1nc(C(=O)NCC(C)N(C(=O)C(C)OCc2ccccc2)C)ccc1Br 78480,N1(C(c2cc(C(CC)CC)no2)=O)CC(C2CN(C(C3(CN(C)C)CC3)=O)C2)C1 78481,C1(C(=O)NCCC(C)NC(C=C(C)Cl)=O)CC2(C1)CC(C(=O)N(C)C)C2 78482,CC1(CO)CCCC1NCCn1cc(C)nn1.c1(C(=O)N)ccccc1 78483,N1(C(=O)Cc2ccc(Cl)cn2)CC2CCCN(C(C3COC4(CCC4)C3)=O)C2C1 78484,c1(CC)nc(NCC2CCCN2C(=O)C(O)CC(C)(C)C)c2ccsc2n1 78485,C1(F)(C(=O)NCC(C)CC2CC2)CCN(C(=O)C=CC2(C)COC2)C1 78486,C(=O)(CCCCC(C)(C)C)N1C(C(C)NC(c2cc(OC)ns2)=O)CCCC1 78487,C(=O)(C1CCc2snnc21)N1CCC(NC(C2CCC(=C)CC2)=O)C(C(N)=O)C1 78488,c1(C(=O)NC(C)CNC(C2OCCO2)=O)ccnc2ncsc12 78489,c1(N2CCC(C#CC)C2)ncccc1S(=O)(=O)NCC(C)CCOC 78490,C1(CC(=O)N(CCC(C)NC(C=CSC)=O)C)CCCCN1C(=O)OC(C)(C)C 78491,c1(C(N2C3(CNC(COC)=O)CCC2CC3)=O)cccc2c1OC(C)C(=O)N2 78492,Cc1ccc(C(N2CC(NC(C3(Br)CC3)=O)C(n3cccn3)C2)=O)nc1C 78493,N1(C(c2ccc(OC(C)C)nc2)=O)CCN(C(=O)Cc2ccc(Br)nc2)C(C)C1 78494,C1(C2C(CNC(CC#C)=O)C2)CCCN(C(=O)C(F)(F)c2cnc(CCC)s2)C1 78495,N1(C(c2c(C)nsc2)=O)CCCC2(C1)C(NC(c1cn(C)nc1Cl)=O)CCN2C 78496,N#Cc1ccc(CF)cc1.C(N=c1[nH]nc(C2CC2)s1)S 78497,N1(C(c2cn(CC=C)nn2)=O)CCC2C(C(=O)N(C3CCOC(C)(C)C3)C)C2C1 78498,Cc1cc(C(=O)NC2CCCN(C(=O)CSC3CC3)CC2)ccc1[N+](=O)[O-] 78499,c1(C(=O)NC2C(F)CCN(C(CSCC(N)=O)=O)C2)ccc2ccc(F)cc2n1 78500,C1(CNC(COC2CCN(C(CC=C(C)C)=O)C2)=O)CN2CC3CC2(CO1)C3 78501,C1(CN(C(C2CCS(=O)(=O)CC2)C(=O)NCCOC)C)(OC)CCCCCCC1 78502,c1(C(=O)NC2CCN(C(C3C(CC)C3)=O)CC2)ccc(C)c(NC(C)=O)c1 78503,C1(C)(CNC(C(C2CN(C(=O)CC3(C)CCOC3)C2)OC)=O)CCCC1 78504,c1(C(N2C3C(NC(C4(C)CC=CCC4)=O)CC(C3)C2)=O)ccc2sc(=N)[nH]c2c1 78505,C1(C(=O)OC)CCC(C(=O)NCC2COCCN2C(c2nc(O)sc2C)=O)CC1 78506,C(CCCC(C)NC(c1c(Cl)n[nH]c1C)=O)NC(CC1(CSC)CC1)=O 78507,c1(C(N(C2CCCC(NC(c3occc3F)=O)C2)C)=O)ccc(F)cn1 78508,Cc1nc(CNC(=O)C(C2(O)CCC2)NC(C2CC(C3CC3)C2)=O)sc1C 78509,C1(CNC(CNC(CCC)=O)=O)C(C(N2CCC(CC(C)C)C2)=O)C1(C)C 78510,Cc1cc2ncc(C(=O)N(CCCCCNC(c3ccc(C#N)[nH]3)=O)C)cn2n1 78511,CC(CC(=O)N1CC(NC(=O)Cc2cc(F)cc(Br)c2)C(O)C1)C(F)F 78512,N1(c2snc(C(=O)OC)n2)CC(CNC(=O)Cc2cnc[nH]2)OC(C)(C)C1 78513,N1(C(C2(OC)CS(=O)(=O)C2)=O)C2CCC1CN(C(=O)CCCNC(C)=O)CC2 78514,C1(C(N2C(C)C(NC(C3(C)CC(C)=NO3)=O)CC2)=O)CC2C(C1)C2(F)F 78515,CCC(C)(COC)C(=O)N1CCC(CNC(c2cnn(C3CCCC3)c2)=O)C1 78516,CCC(CC(C)C)C(=O)N1CC(O)(CNC(c2nc(Cl)sc2Cl)=O)C1 78517,c1(NC(N2CCCC(CCCO)C2)=O)cccc(-c2ccc[nH]2)c1 78518,c1(CC)cc(C(=O)NCCC2CC(NC(C3CC(OC)C3)=O)C2)oc1CC 78519,C(=O)(CCC1=CCCCC1)NCCCCCNC(c1nc(N)c(Br)cc1)=O 78520,CC1=NOC(CNC(=O)C(C)(C2CC2)N(C(=O)CN=[N+]=[N-])C)C1 78521,c1(C(=O)NCC(CC=C)NC(=O)Cc2cccnc2C)ccc([N+](=O)[O-])cc1O 78522,C1(C)(C(N2CC(Cn3cc(-c4cnc(C)nc4)nn3)C2)=O)Cc2ccccc2C1 78523,CCCC(CC)CCC(=O)NC1CC2(C(=O)NC(C)(CO)CO)COC1C2 78524,C12(C(=O)NC(C3(C)CC3)CO)CCCC1CCN2C(c1ccc(F)c(N)c1)=O 78525,C(CNC(=O)CCC(C)N(C)C)(CC(F)(F)F)NC(Cn1c(C)nnn1)=O 78526,C1(C(=O)OCC)CC(C(N2CCC2(C)NC(CCC)=O)=O)C1(C)C 78527,C(C(CN=c1[nH]cnc(Cl)c1Br)[N+](=O)[O-])NC(c1ccc(OCC=C)cc1)=O 78528,C(C(O)C(=O)NCCNC(C1CC12CC2)=O)SC.c1ccccc1 78529,C(CCC(=O)N(C(C)C)CC1CC1)(C(C)C)NC(=O)OC.C1(C)C(=O)N1 78530,N1(C(CC2C(C)C2)=O)CCOC2(CCN(C(c3cc(Br)sn3)=O)CC2)C1 78531,c1(C=O)ncc([N+](=O)[O-])cc1C.C(=O)(CCCN1CCCC1)N1C2CCN1C2.CS 78532,C1(C(N(CC(C)(C)C#N)C)=O)CN(C(=O)C(C)(C)n2cncn2)CCO1 78533,CC1C(C(=O)O)C(C(=O)N(c2nnc(C#N)s2)C)CC1C 78534,c1(CC(=O)NC2CC(C(=O)NCc3c(C)nns3)OCC2)c(F)cccc1F 78535,C1(O)(C(C)NC(=O)CC2CCC2)CCN(C(=O)CC2CC2(Cl)Cl)C1 78536,c1(OCCC(N2C(Cn3cc(CCS(C)(=O)=O)nn3)CC2)=O)ccc(F)c(F)c1 78537,c1(C(=O)NCC(C)NC(c2cc(C(C)(C)C)no2)=O)cn(CCC2CC2)nn1 78538,Cc1cc(C(=O)N(CC(C)CNC(=O)C=Cc2ccc(Cl)s2)C)ncc1C(F)F 78539,N1(C(c2c(C)noc2C)=O)CC2CC1CN2C(=O)CSCC(F)F 78540,C(C)(C(C)SC)(N1CC(Cn2cc(CCC(c3ccccn3)O)nn2)C1)C1CC1 78541,N1(C(c2c(C)cccc2Cl)=O)CC2(CCCC2NC(C2CCC3CC3CC2)=O)C1 78542,c1(COC)ccc(C(N2CC(O)(CNC(=O)C(C)(C)c3ccccn3)C2)=O)s1 78543,CCC(CNC(=O)CCCN(C(=O)C(C)NC(C)(C)CC)C)CO 78544,CC1(C)CC(C(=O)NCC2CC2(F)F)CN1C(=O)CCc1cccc(O)n1 78545,N1(C(CCN(C(C)C)C(C2(F)CCCCC2)=O)=O)CC(S(N)(=O)=O)C1 78546,c1(C(=O)NC(CC)CC(=O)NCC(F)Cl)ccnc(C)c1C 78547,c1(CC)ccc(C(=O)NC2CCC2NC(C2CNC2)=O)cn1 78548,Cc1ccc(CN2CCCC2CCC(=O)N(C)Cc2ccccc2)c(Cl)c1 78549,c1(NCC2(NC(=O)C(O)CN3CCCC3)COC2)nc2c(cc1Cl)C(=O)OC2 78550,C1(NC(C(CC)N(CC)CC)=O)CCN(C(=O)C2=CCCCCC2)CC12CCC2 78551,c1(CC)nc(C(=O)NC(C)C=CC(=O)NCCC2(C)N=N2)co1 78552,C1(C(C)N(C(=O)CC2CCC2NC(=O)C(C)CN2CCCC2)C)CCCOC1 78553,C=CCCCCC(=O)N(C)CC1(C)CCCC1NC(c1ccsn1)=O 78554,C1(CC(=O)N)CCCCC1.C1C(=O)NCC2(CC2)CC(=O)N1CCC.C(C)(C)(C)O 78555,N1(C(Cc2ccn(CC)n2)=O)CCCN(C(=O)C=CSC)C(C)C1 78556,c1(C(N2C(C)CC(NC(=O)C(C)(C)O)C2)=O)ccn2ccccc12 78557,CN=c1[nH]c(=NCc2cccnc2C)[nH]c(=NCC(=O)N2CCOCC2)[nH]1 78558,N1(C(C2CC(C(N)=O)C2)=O)CC2C(CC(=O)NCC3(n4cncn4)CC3)C2C1 78559,C1(C(N2C3CC(NC(c4ccn(C5CC5)n4)=O)C(C3)C2)=O)CN2CCCN1CC2 78560,C(=O)(C(COC(CC)COC)CC(C)C)OC(C(COC)NC(=O)CC1CCC(OC)CC1)=O 78561,C=CC1(CO)CCN(C(=O)C(CCC)NC(=O)CSCC(N)=O)C1 78562,C1(NC(c2cc(C(F)F)ccn2)=O)CC2(CCCCN2C(C2(C(F)F)CC2)=O)C1 78563,C(=O)(CC(O)C(=O)NCC1CCN1C(C12CC(C1)C(C)(C)O2)=O)OC(C)(C)C 78564,S(=O)(=O)(c1cccc(C)c1C#N)N1CCC(COCC#C)CC1 78565,N1(C(C)=O)CC(O)CC1C(=O)NCC1CCN(C(C2(C)CSC2)=O)C1 78566,C(=O)(CCCCCCCCCO)N1CCC(CN(C(=O)Cc2ccco2)C)CC1 78567,Cc1ccccc1C=CC(=O)NC(C(=O)NCC12CCN(CC1)C2)c1cccs1 78568,c1(C(=O)NCC2CC(C)N(C(C3(C)CCC(=O)NC3)=O)C2)cc(O)cc(F)c1 78569,c1(C(C)=O)cc(C(=O)NCc2cn(CC(C)NC(=O)CCF)nn2)oc1C 78570,N1(C(C2C(=C)C2)=O)CCCC2(C1)CN(C(c1ccc3nccnc3c1)=O)CCO2 78571,n1(CC)cnc2nc(N(C)CCc3nc(=N)[nH][nH]3)nc(N(C)Cc3ccns3)c12 78572,C1(C)(C(=O)NC2CCCC(CNC(CC(C)C)=O)C2)CCC(O)CC1 78573,c1(C(=O)NCC(C)CN(C)C(C2CNC(=O)N2C)=O)coc2c(F)cc(F)cc12 78574,O=C(CCCC1CCC1)N1CCC(CNC(C2CC(n3ccnn3)C2)=O)C1 78575,C1(C(=O)NCC2(OCC)CN(C(=O)C(C)=CCO)C2)CCNC(=O)C1 78576,c1(OC)ccc(=NC(=O)C23CC2CN(C(c2cc(Br)ncc2F)=O)C3)[nH]n1 78577,n1(CC(=O)N(C2CN(C(c3cnn(CCO)c3)=O)CC2F)C)nc(Cl)ccc1=O 78578,N1(C(C(C)c2ccon2)=O)CCC(F)(CNC(c2cc(Cl)cc(Cl)c2)=O)CC1 78579,N1(CC)CC2=C(C1=O)C(c1ccc(C(F)F)c(F)c1)NC(=O)N2CC(C)C 78580,c1(C(=O)NC(C)CCNC(=O)CC(C)(C)C)c(O)cnc2cc(F)ccc12 78581,C1(CNC(C=CC=CCC)=O)(OC)CCC(C)C1.C12(F)CN(C1)C2=O 78582,N1(C(C(CC)(C)O)=O)CC2(NC(c3ccc(Br)cc3N)=O)CCC1CC2 78583,C1(CNC(=O)COC2COC2)CCC2CN(C(c3ccc(O)cc3)=O)CCC2C1 78584,C1(NC(C(C)(C)SC)=O)CC12CCN(C(=O)Cc1ccoc1C)CC2 78585,C(c1cn(C)cn1)=C(C(=O)NC(C)C(CO)NC(=O)CCNC(C1CCC1)=O)F 78586,C(=O)(C(C)NC(=O)CC1CCC1NC(=O)CCc1nc[nH]n1)N(CC)CC 78587,c1(C(N(CC(CNC(c2n(C(C)C)ccc2)=O)C)C)=O)[nH]ncc1C#N 78588,CCCCS(=O)(=O)NCC(=O)N(C)CC1CCCCN1C(=O)CCCCSC 78589,c1(CCN2C(COC)C2=O)ccccc1.CCCC(c1ccco1)CC1(C)CC1 78590,c1(C(=O)NC(CCCNC(c2nnc(C)s2)=O)C)cccc(CO)c1C 78591,CC(C)CCN=C(NCc1cnn(CCF)c1)NCc1ccc(Cl)nc1 78592,c1(C(C(N2CC(NC(C3(OC)CCCC3)=O)C2)=O)N(C)C)c(F)cccc1F 78593,N1(C(Cc2ccc(OC)nc2)=O)CCC2C(C1)NC(=O)CN2C(C1CC1F)=O 78594,N1(C(C(CC)(F)F)=O)Cc2occ(C(N3CC(CO)CC3CO)=O)c2C1 78595,Cc1cc(C)n(CCNC(=O)CC(N)Cc2ccc(F)cc2)n1 78596,Cc1sc(Br)nc1C(=O)NCC1(C)CCN(C(C2CC(F)(F)C2)=O)C1 78597,c1(C(C(=O)NC2C(OC)CN(C(C3CN(C)C3)=O)C2)O)ccc(Cl)cc1Cl 78598,Cc1cc(C)c2c(=NC(=O)NC(c3ccnc(Cl)c3)C)[nH]sc2n1 78599,Cc1nc2ccccc2cc1C(=O)NCC(C)(C)NC(=O)C(C)CC(F)(F)F 78600,N(C(=NCCC)NCCC(C)(C)CO)CC1(CC=C)CCCC1 78601,N1(C(c2cn(CC)nn2)=O)CC2CCC2(CNC(c2oncc2C)=O)C1 78602,c1(CC(=O)NCCC2N(C(C(CC)C(C)C)=O)CCOC2)ccccc1[N+](=O)[O-] 78603,C1(N(C(C(CC)F)=O)C)CN(C(c2ccc(C(=O)NC(C)C)cc2)=O)CC1(C)C 78604,C1(=CC(=O)NCC2C3CN(C(c4c(C)nsc4N)=O)CC32)CCCCC1(C)C 78605,N1(C(c2nc(CC)oc2)=O)CC(NC(c2sc3cncn3c2C)=O)C(C2CC2)C1 78606,C(CCCCCC(=O)N1CC2CCC2(CNC(=O)C(O)C(C)(C)C)C1)SC 78607,C(=O)(CC(C)(C)C(F)F)N1C(CNC(C(CCC)CC)=O)CCC1 78608,c1(C(=O)NCC(C)CNC(=O)CCCC(C)(C)C)n[nH]c2c1CCCCC2 78609,Cc1cc(C(=O)NCC#CC(N2CCOC(C(N)=O)C2)=O)sc1C 78610,C(N=c1[nH]c(=NC(CCO)C2CCCC2)[nH]c2ccsc12)c1ccn(C)c1 78611,c1(NC(c2occ(C(C)=O)c2)=O)ccc(NC(C2(O)CCCCCC2)=O)cc1C 78612,C1(N=c2[nH]nc(CC(C)C)s2)(CNC(c2cccc(OCC)c2)=O)CCCC1 78613,C(=O)(N=c1cc(C)n(C)[nH]1)C1OCCC(NC(CCCOCC=C)=O)C1 78614,N1(C(C)=O)CCCC1CC(=O)NC1CC(C)(NC(c2cnnn2C)=O)C1 78615,c1(OCCOC)ccc(C(=O)NC2CCC(NC(=O)C(C)C(C)C)CC2)cc1 78616,C1(C(=O)NCC2CN(C(CN(C3CC3)CC)=O)CC2C)CCc2cnnn2C1 78617,N1(C(COCC)=O)CC2C3CCC(C2C1)N(C(c1ncccc1C(F)F)=O)C3 78618,Cc1cccc(C(=O)OC2CC2CNC(c2nn(C)cc2Cl)=O)c1.C1C(=O)N1 78619,C1(C(=O)NCC(n2cc(CCCC(C)O)nn2)C)CCc2ncccc2C1 78620,c1(NC(CSCC=C)=O)ccc(C(C)NC(=O)CS(=O)(=O)N(C)C)cc1 78621,Cc1nnc2n1CCC2(C)C(=O)N1CCC(C)(NC(=O)CC2COCCOC2)C1 78622,CCCC(C)C(=O)N1CC=CC1(C(=O)NC1CC(CF)C1)COC 78623,C(=O)(C1=NOC2COCC12)NC(CCC(=O)NC1(C#C)CCC(C)CC1)C 78624,Cc1nn(C)c(C)c1CN1CC(CNC(=O)CN(CC(C)C)C)C1 78625,C(N=c1ccnc(N2CCC(C(C)COC)CC2)[nH]1)c1c(CC)nco1 78626,c1(N(C)C)cc(NCC2CCCSC2)nc(C(F)(F)F)n1 78627,CC1CC=C(C(=O)NC2COCC2NC(c2cccc3nccn23)=O)CC1 78628,C1(C)(C(=O)NCCc2n(C)nnc2)CCN(C(c2csc(C#N)c2)=O)CC1 78629,CC1(C)CC=C(C(=O)NCC(=O)NCC(=O)Nc2cc(CO)ccn2)CC1 78630,c1(OC)cc(C)c(Cl)cc1S(=O)(=O)N1CCN(C(c2cnc[nH]2)=O)C(C)C1 78631,CC1=C(C(=O)NCC2(NC(=O)CC3CCCN3C(C)C)CCOCC2)CCC1 78632,Cc1c(C(=O)NC(CNC(=O)C(C)(O)C2CC2)CC(C)C)[nH]c2ccc(F)cc12 78633,c1(CCC(=O)OC)cccc(CN2CCCC(C(N3CCSCC3)=O)C2)c1 78634,N1(CCC2CC(C)C2)CC2CC1CN2C(=O)C(F)Cc1ccccc1 78635,C=CC1(CC(=O)NC(C)C(C)NC(=O)CC2CSC2)CCCCC1 78636,C1(NC(C(CCOC)OC)=O)CCN(C(=O)Cn2nnnc2C(C)C)C(C)C1 78637,N1(C(c2cc(OC)n[nH]2)=O)CCC2CN(C(=O)CC3CCC=CCC3)CC2CC1 78638,N1(C(COC(C)C)=O)CCC(C)(C)C(NC(=O)COCC2(F)CC2)C1 78639,C1(COC)(NC(c2ncccc2OC)=O)CCN(C(c2ccc(C3CC3)s2)=O)C1 78640,c1(C(=O)NC(CC)CNC(C2(F)CCOC2C)=O)c(C)nn(CC)c1C(F)F 78641,Cn1cnc(CNC(=O)CC2CC2CNC(=O)COCC2CCC2)n1 78642,CCC(C(=O)N1CC(OCC(=O)NC2CCOC2)C1)OC 78643,N1(C(C#CC2(CC)COC2)=O)CC=C(C(=O)N2CC3(CCC3)CC2C)CC1 78644,CC1(C)COCCC1C(N1CCC(CC(N)=O)(NC(C2(CO)CCC2)=O)CC1)=O 78645,C(CCC(F)(F)F)N(C(c1scc(C(C)=O)n1)=O)C 78646,C(=O)(CC(CC)C(C)(C)C)NCC(CC=C)NC(=O)Cc1n[nH]cc1Br 78647,c1(C(N(CC(C)NC(c2cc3ccnn3cn2)=O)C)=O)c(F)c(F)cc(F)c1F 78648,c1(-n2c(C(C=CC)O)nc(-c3ccncc3)n2)cccc2nc[nH]c12 78649,C(=O)(CC(C)(C)CNC(c1cc(O)ccc1C)=O)NCCC(C(C)C)OC 78650,C1(C(N2CC(C(=O)NCc3cc(=O)cc(Cl)[nH]3)OCC2)=O)CC2(CCC2O)C1 78651,CC(CCCC(=O)NCC#CC#CCO)NC(C1CCCN1C1CC1)=O 78652,c1(C(C(=O)NCCCC)N(C2CCC(C)(C)C2)C)ccc(OC)cc1Br 78653,c1(C(=O)NC2CCN(C(COC(C)C)=O)C(C3CC3)C2)ccc2n[nH]cc2n1 78654,c1(C(=O)NC(CCC(=O)OC)c2cccs2)ccc(C)c(F)c1.C1(C)C(=O)N1 78655,C#CCCCCCCCC(=O)NCCN(C1CCCCC1)C(C1(C)CCCO1)=O 78656,CCCCCCCC(=O)NC(C(=O)N1CC(c2nn[nH]n2)C1)C(C)(C)C 78657,C1(C(N(CCCCCNC(C2CC(C(C)C)C2)=O)C(C)C)=O)CCCS1(=O)=O 78658,c1(C(=O)NCC(n2cncn2)C)ccn(CCNC(=O)CCCc2ncco2)c1 78659,C1(C(=O)NC(C2(C(=O)NCC(C)(C)C)CC2)C)CCC2(CC2)C1 78660,N1(C(c2cc(C)c(Br)o2)=O)CC(NC(c2snnc2C)=O)CC(F)C1 78661,C(=O)(CCS(N)(=O)=O)NCC(N1CCC(C)(CO)C1)=O.C1CN1CCO 78662,c1(CN2CC(C)(CNC(c3cccc(OC)c3)=O)C2)cc([N+](=O)[O-])ccc1Cl 78663,C1(NC(=O)CC2COCC2O)C2CN(C(=O)CCCc3ccccn3)CC12 78664,C1(NC(=O)COCC2CC2)CC2CCC1(C(=O)N(C)CC1(F)CCC1)C2 78665,C1(N2C(=O)C2)CCN(C(C2CCOC2C(F)(F)F)=O)C1.C(C(C)C)SC 78666,C1(C(=O)NC2C=CC(C(=O)NCc3nc(C)on3)C2)CCCN1C=O 78667,C1(CNC(CC2C(C)CCO2)=O)CCCCCN1C(c1csc(=N)[nH]1)=O 78668,N1(C(Cc2c(C)occ2)=O)CCOC(CCNC(=O)CC2COCCOC2)C1 78669,Cc1ccc(F)c(C(=O)N(C)CC2(O)CCN(C(=O)CCC3CC3(C)C)C2)c1F 78670,C1(C)(C(N(CCCO)C)=O)CCN(C(c2cc(C(F)F)[nH]n2)=O)CC1 78671,C12(NC(CCC)=O)CCCC1CN(C(c1sc(C(C)C)nc1C)=O)C2 78672,C1(NCC(N2CCC(CC(=O)NCc3ccc(O)cc3)C2)=O)CCC2(CCC2)C1 78673,c1(C(N2CC(CC)N(C(C3CC4CC4C3)=O)CC2)=O)ccc2nccn2n1 78674,C1(NC(C(COC)OC)=O)CS(=O)(=O)C12CCN(C(c1ccoc1Cl)=O)CC2 78675,N1(C(c2cc(CSCC)on2)=O)CC2C(NC(C3CCCC(C(F)F)O3)=O)C2C1 78676,CCC(CC)(C(C)C)NC(=O)C=CCNC(c1cc(CCO)on1)=O 78677,c1(CC(C(=O)N(CCCNC(=O)CC2(C)CCCCC2)C)O)ccc(F)cc1 78678,N1(C(c2c(C)[nH]cc2)=O)CC2C3CCC(C2C1)N(C(C1CC(C)CO1)=O)C3 78679,C1(C(N2CCC(CC(C)(C)C)C2)=O)CC(N=[N+]=[N-])CN1C(C1CS(=O)C1)=O 78680,c1(OC)cc(F)c(C(N2CC(O)C(O)C2CNC(=O)CSC)=O)cc1OC 78681,C1(CC)CC2(CC(C(=O)OCC)C2)C1.C12(COC(C)C1)CS(=O)(=O)N2 78682,c1(C(=O)NC(C)CCN(C(=O)CC2(C)CCCO2)C)cc2c(nn1)CCCC2 78683,N1(C(C2(NC(=O)C=CCO)C(C)CCC2)=O)CCC(O)C(N=[N+]=[N-])C1 78684,c1(C(=O)NCCC2CN(C(C3C(C)CC(=O)N3)=O)C2)nnc(O)cc1O 78685,c1(CC)ccc(-c2nc(CNC3C=CS(=O)(=O)C3)c(C)o2)cc1 78686,c1(NC(=O)NCC2C(C)C2(F)F)ccnc2c(Br)cccc12 78687,C1(NC(COc2cccc(OCC)c2)=O)CCN(C(=O)CC2CC2)CC12CCC2 78688,c1(C(N2CCC(C)C2CNC(=O)C#CC(C)(C)C)=O)cc2n(n1)CCCO2 78689,N#CC1(C(N2CC(NC(=O)C(N)=O)C(n3cccn3)C2)=O)CCSCC1 78690,Cc1onc(C2CCCCC2)c1C(=O)NC(CNC(=O)CC(F)(F)F)C1CC1 78691,Cc1ccc(F)c(C(=O)NCC2(NC(c3cnc4n3CCCC4)=O)COC2)c1F 78692,N1(C(C=CC2(C)COC2)=O)CC(C(=O)NCC2C3CCCCCC23)C(C)(C)C1 78693,CC(C)(CC=CC(=O)NC1CCCC1C#N)NC(=O)CC1CNC(=O)O1 78694,c1(C(N2C(C(C)C)CN(C(=O)C=CCO)CC2)=O)cccc2cc(Cl)ccc12 78695,C1(CC)CNC(=O)CN1C(C1(NC(C2CCCCNC2=O)=O)CCCC1)=O 78696,C1(NC(C=CC)=O)CS(=O)(=O)C12CCN(C(c1ccn(C3CC3)n1)=O)CC2 78697,C1(C(=O)NC2CCC(CCNC(CCC3C(C)(C)C3)=O)C2)CCc2n[nH]cc2C1 78698,c1(C(=O)NCC(CC)NC(C2(CC)CC(F)(F)C2)=O)cnc(S)n1C 78699,N#CC1(C(=O)NC2CC2CNC(c2ccnn2C2CC2)=O)CCC(=O)CC1 78700,CCCC(O)C(=O)NCCCN(C(C1C2CC2C2CC12)=O)Cc1ccccc1 78701,C1(NC(COCC#C)=O)(CNC(C2(OC)CC2)=O)CCCC1 78702,c1(SCC(=O)NCC2CCCN2C(c2ncccc2Cl)=O)ccsc1[N+](=O)[O-] 78703,CC(CNC(C1(CCCF)CC1)=O)CC(=O)Nc1cccc(O)c1 78704,CN=c1[nH]c(=NCc2cc(C)c(C)s2)[nH]c(=NC2CCC3(CC4CCC3C4)C2)[nH]1 78705,Cc1cnc(C(=O)NCC2(CNC(=O)C(c3ccn(C)c3)C)CC2)cn1 78706,C(C(F)(F)C(F)(F)CO)NCC(=O)N(c1ccc(OCC)cc1)CC 78707,N1(C(c2ccccc2[N+](=O)[O-])=O)CC2CCN(C(C3CC3(Cl)Cl)=O)CC2C1 78708,C1(CNC(C(CC)F)=O)CCC(C)(C)CN1C(c1sc(C)cc1Cl)=O 78709,C1(COC)CCCN1N(C)C(C)C1CCN(CC(F)(F)F)C1 78710,C1(NC(CS(=O)(=O)NCC)=O)(CNC(c2ccoc2)=O)Cc2ccccc2C1 78711,C12(C(=O)NCCOCCNC(c3cc(Cl)no3)=O)CCCC1CC(F)(F)CC2 78712,c1(C(=O)NC2C(NC(C3(COC)CCC3)=O)CCC2)cc(F)c(F)cc1O 78713,c1(C(N2C(CNC(C(CC)C)=O)CC(C)(C)C2)=O)ccc(S(N)(=O)=O)cc1F 78714,c1(OC)ccc(CCN(C(CSCCC)=O)C2CC2)c(OC(F)F)c1 78715,CC1CCN(C(c2ccoc2Cl)=O)CC1NC(c1cnc(-c2ccccc2)o1)=O 78716,N1(C(C(C=C)C)=O)CCC2(C=C(C(=O)N3CCOCC3C(N)=O)C2)C1 78717,c1(C(C(N2CC(COC)(NC(c3nccnc3N)=O)C2)=O)O)ccc(F)c(Cl)c1 78718,C(CC(C)(C)CNC(=O)Cc1ncc(C)o1)NC(CC1C(CSC)C1)=O 78719,CC(C)(C)CC(O)CC(=O)NCC(C(N1CCCC2(CCC2)C1)=O)C(=O)O 78720,CC1CC2(CCCC2)CN1C(C1CCC(CNC(C2CC(C)(C)C2)=O)O1)=O 78721,CC1CC(NC(=O)CCc2ccsc2Br)CCS1(=O)=O 78722,N1(C(C(C)(C)c2nccs2)=O)CCN(C(=O)C(C)(C)N2CCCC2)CC1 78723,C(CS(=O)(=O)Cc1cn(C2COCC2O)nn1)C(N(C(c1onc(C)n1)C)C)=O 78724,C(C(C)C(F)C(=O)NCC1CN2CCC1C2)NC(c1c(C)cnn1C)=O 78725,C(=O)(C(C)(C)NC(=O)C=CC(C)(C)NC(c1cc[nH]c1)=O)OC 78726,c1(C(=O)OC)ccccc1C(=N)NOCC1CC12CCOCC2 78727,C(=O)(CCCCC(C)=O)N1C(C(N2CCC(CC#CC)CC2)=O)CCCC1 78728,N1(C(C(CC#CC)NC(=O)CC2=CCCC2)=O)CCCC(N=[N+]=[N-])C1 78729,c1(C(=O)NCC(CNC(=O)CCOC(C)C)OC)c(C)cc(Cl)cc1C 78730,C(CCC(=O)NCCC1CCCO1)NC(CC1CC(=C)C1)=O 78731,CC1CN(C(c2ocnc2C(F)F)=O)CC(C)C1NC(=O)Cn1nnnc1C1CC1 78732,c1(NC)ccc(C(=O)NCC2CCCN2C(c2snnc2C2CC2)=O)nc1 78733,Cc1ncc(CN(C)C(c2cn(CCNC(=O)CC34CCCC3C4)cn2)=O)s1 78734,c1(C(c2ccccc2)N)cc(NCC2CN(C(C3CCCC3)=O)C2)ccn1 78735,N1(C(c2c(CC)c[nH]c2)=O)CC(N=[N+]=[N-])CC1C(=O)N(C)CC1CCCCO1 78736,Cc1cc(NC(C2(NC(=O)CCn3cncn3)CCSC2)=O)cc(CO)c1 78737,N1(CC(C)(C)NC(C(C)=C(C)C)=O)CCN(C(=O)C(C)(C)N(C)C)CC1 78738,N1(C(CN(C(=O)C=CC2CCOC2)CCOC)=O)CC(CO)CC(C)(C)C1 78739,c1(N(C)Cc2nnc(C)s2)nc(N2CCn3cc(Br)cc3C2)c2c(n1)CSC2 78740,C1(NC(CC2N(C(c3c(OC)cnnc3)=O)CC(O)C2)=O)CCN(C)CC1C#N 78741,N1(C(c2c(Cl)ncc(N)c2)=O)CC2CCCC1C2CNC(C1CCS1(=O)=O)=O 78742,C1(F)(C(N2CCOCC(CNC(c3cnccc3Cl)=O)C2)=O)CC12CCCCC2 78743,CC1(C)CC(NC(=O)C=Cc2cncs2)CN(C(=O)COC(F)(F)F)C1 78744,Cc1cnc(CNC(=O)C(C)OCCNC(=O)CN2CCCC2=O)[nH]1 78745,Cc1cc(C(N2CC3(CC3C(=O)NCc3cc(F)cc(Br)c3)C2)=O)c(Br)cc1F 78746,c1(C(=O)NC2CC3CN(C(CSC(C)C)=O)C(C2)C3)nc2cc(O)ccc2[nH]1 78747,C1(CCC)COCCN1C(=O)CC(C1CC1)NC(C1OC2CCC1C2)=O 78748,N1(C(C2C(C=C)OCCC2)=O)CC2OCCN(C(c3oc(CC)cc3C)=O)C2C1 78749,Cc1csc2cc(C(=O)NCC(C)NC(c3csc4nccn34)=O)[nH]c12 78750,CC1(C)C(NC(=O)CC(O)C2CC2)CCN1C(=O)CCn1cnccc1=O 78751,C#Cc1cccc(C(N2CC3(CCN3C(=O)CCc3cc(OC)no3)C2)=O)c1 78752,c1(C(=O)NC23CC(NC(C4C(C)(CC)C4)=O)(C2)C3)cnc2ncc(Cl)cn12 78753,C12CC(F)CN(C1)C2.N1(C(c2c(SC)cccc2)=O)CCC(CO)C(O)C1 78754,c1(N(Cc2cc(OC(F)F)c(OCC)cc2)CC2CCCO2)ncc(N)cc1C 78755,c1(OCC)cc(CNC(=O)NCC(CC)(CC)SC)ccc1OC 78756,C1(O)(CNC(C2(CCC)CC2)=O)CCCN(C(C23CCC(C)(C2)OC3)=O)C1 78757,C(=O)(CCCC(F)(F)F)NCC=CCNCCOCCCCOC.C1C(=O)N1 78758,N1(C(CC2CCC(C)CO2)=O)CC(NC(c2nccc(C(F)F)n2)=O)CC(F)C1 78759,CCC(O)C(C)C(=O)N1CCC(O)(C(=O)NOC2CCCCC2)CC1 78760,c1(C(N(C(C)CNC(=O)Cn2[nH]cnc2=N)C)=O)ccnc(Cl)c1Cl 78761,c1(SC)cc(=NC(=O)C(C)C(C)NC(=O)C(C)OC(C)=O)[nH]n1C 78762,CC1(C)C2CCC(C(=O)NC3CCCC(NC(=O)C(C)(O)C4CCC4)C3)C1C2 78763,C1(c2ncc(C(=O)OC)o2)CN(N2CCCC3(COCCO3)C2)C1 78764,Cc1ncc2n1CCC(C(=O)NC1(C)CC(NC(=O)Cc3sc(O)nc3O)C1)C2 78765,C(=O)(CCCCC(F)(F)F)NCCCN(C)C(c1nnc2n1CCCC2)=O 78766,CC1CCCCC1(CNC(C1C2(CC2)C12CC2)=O)NC(=O)CN1CCSCC1 78767,C1(C(=O)NCCc2cc[nH]n2)COCCN(C(c2ocnc2C2CC2)=O)C1 78768,c1(C(=O)NC23CCN(C(c4c(CC)noc4)=O)CC2C3)ccc2nc(C)cn2c1 78769,CC1=CCC(C(=O)NCC(C)(C)NC(C2CCCN(C(=O)OC(C)C)C2)=O)CC1 78770,N1(C(C2C(C(=O)NCCCn3c(C)ncc3)C2)=O)Cc2ccc(Cl)nc2C1 78771,N1(C(C2C(=C)C2C(=O)OC)=O)CC2CN(C(c3cnn4ccsc34)=O)CC(C1)O2 78772,C1(C(N2CC(COCCNC(CCCOC)=O)C2)=O)CC2(C1)CC2(F)F 78773,c1(Cn2cc(CN(C(=O)C(F)(F)Cl)C)nn2)cccc(Cl)c1Cl 78774,C(=O)(C(CN(C(CCO)C(F)F)CCOCC)Cc1ccc(OC)cc1)OC 78775,Cc1c(N)cc(C(N2CCC(CCNC(=O)C(C)CC(C)(C)C)CC2)=O)cc1N 78776,Cc1cc(NC(c2ccccc2O)=O)sc1C(=O)NC1CONC1=O 78777,C1(CC)CN(C(=O)C(c2ccccc2)C)CCC1NC(C1(F)CC2(CCC2)C1)=O 78778,C(=O)(C(O)CCN(C)C)NC(C1CCCCC1)C(=O)NC(C)COC(F)(F)F 78779,C1(C(=O)O)CN(Cc2ccccc2OCF)CCN1Cc1ccccc1 78780,C(c1ccc(Br)cc1)=CCC(=O)NCC(CNC(C(C)C1CC1)=O)CO 78781,N1(C(C(CCCC)O)=O)CC2CCCC2(CNC(c2ncc(F)c(OC)n2)=O)C1 78782,C1(NC(c2c(CC)n(C)nn2)=O)CCCCCC1NC(=O)CCCn1ccnn1 78783,N1(C(CCCC#C)=O)CCCC(C(=O)NC(c2ccccc2F)CO)CC1 78784,c1(C(=O)NC(C(=O)NCCN(CCCC)C)CC(F)F)c[nH]c2ccccc12 78785,C(C)(CCC(C)(C)C)(NC1c2n(nnn2)C12CC2)SC.c1(OC)ncccc1Cl 78786,C1(CO)(CNC(c2cc(I)cs2)c2nnnn2C)CCCO1 78787,CC(C)C(N=[N+]=[N-])C(=O)NC1CC(C(=O)NC(C)(C)CO)C12CCC2 78788,C1(NC(=O)CC=C(Cl)Cl)CC2(C1)CN(C(=O)CN1C(=O)CCCC1=O)C2 78789,C1(C(N2C3CN(C(c4nnc(O)cc4O)=O)C(C3)C2)=O)CC2CCC(C1)S2(=O)=O 78790,Cc1ncc(Cl)cc1C(N1CCCC1CNCc1cc(Br)cnc1F)=O 78791,C1(C(=O)NC(C(=O)OC)C)CCCC1NC(C1(F)CCC1)=O 78792,C1(C(N2CCC(CCNC(c3cscn3)=O)CC2)=O)CC1C1CC(F)(F)C1 78793,C(=O)(C(F)C(C)CNC(=O)C(C)OCCC)NCCC=CC=C 78794,c1(C(C)C)ccc(C(N2CC(NC(=O)CC(C)c3cccnc3)C(O)C2)=O)nc1 78795,N1(C(c2c(C)snn2)=O)CC2ON=C(CNC(=O)Cc3ccsc3Cl)C2C1 78796,c1(CNC(C2(NC(CSCCOC)=O)CC(CO)C2)=O)cc(C)cnc1O 78797,C1(C(=O)N)CCN(C(=O)CCc2ccccc2)CC1O.c1(CC2CC2)cnoc1 78798,C1(C(=O)NC(c2nc(=O)o[nH]2)C)CC2(CCN1C(C1CC(=O)C1(C)C)=O)CC2 78799,Cc1nc(C=CC(=O)N(C)CC2CCCN2C(=O)C(C)SC(C)C)[nH]c1C 78800,C1(C(C)C)CN(C(=O)Cc2cn[nH]c2)CCN1C(c1cc(Cl)n(C)n1)=O 78801,c1(CC(N2CCC(n3cc(C4CCCC4)nn3)C2)=O)c[nH]c2ncccc12 78802,c1(-c2cn(C3CCC(NC(C4CCC(O)CC4)=O)C3)nn2)cc(Cl)c(Cl)c(Cl)c1 78803,N1(C(C(CC)C2CCC(=O)N2)=O)CCN(C(C2C(C)C2C)=O)C(C)C1 78804,c1(-c2ccc(CCC)nc2)n[nH]c2cccc(C(=O)Nc3cc(O)ncc3C)c12 78805,CCC1=NOC(C(=O)NC(C2CCCN2C(C2CC(Cl)(Cl)C2)=O)C)C1 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78824,N1(C(c2nc(C)n(C)c2)=O)CCC(C2CCN(C(=O)COCCC(C)C)C2)C1 78825,O=C(CC1CCCc2ccccc21)N1CCC2CN(CC3CC34CC4)CC2CC1 78826,C1(NC(c2cn3[nH]ccc3n2)=O)COC2(C1)CN(C(=O)C=Cc1cn[nH]c1)C2 78827,C12(C(=O)Nc3c(CC)ccnc3)COCC1CN(C(c1cn(C)cn1)=O)C2 78828,C1(C(=O)NCC(CC)NC(c2snc(C)c2N)=O)CC2CC1C1C2C1(F)F 78829,N1(C(COC)=O)CCN(C(C2CCCC2(F)F)=O)CC(C)(C)C1 78830,N1(C(=O)Nc2c(OC)ccc(-c3cnc[nH]3)c2)CC(F)(CO)C2(CCC2)C1 78831,c1(CC)cccc(C(=O)NCC(C)(C)NC(c2cc(C3CC3C)on2)=O)c1 78832,CC1CC(C)CN(C(=O)CN2CCCC2C(C)(C)CO)C1 78833,CN(C)NC(=O)CCC(=O)NC1CC2(C(=O)NC3CC3(C)C(F)F)COC1C2 78834,N1(C(CCc2ccc(C)cc2)=O)CCN(C(=O)C(C)c2ccsc2)C2CC12 78835,N1(C(C(C2CC2)OC)C(=O)NC2CCOCC2)CCn2c(C(F)(F)F)nnc2C1 78836,C1(CNC(c2c(CC)nco2)=O)C2CN(C(=O)CC(O)Cc3ccccc3)CC12 78837,C1(CNC(C2(SC)CC2)=O)CC2COCC2N1C(c1cncn1C)=O 78838,c1(C(=O)NC2CN(C(C(CC)COC)=O)CC2C2CC2)cc2cc(F)ccc2[nH]1 78839,N1(C(C2(CC)CCC2)=O)CCC2(CCN(c3ccc(C#N)nc3)C2)C1 78840,c1(NCc2ccc(C(N3CCCC3COCC)=O)cc2)cc(S(=O)(=O)NC)cs1 78841,N1(C(C2(C(=O)OCC)C=CCC2)=O)CCN(C(=O)CNc2ncccn2)CC1 78842,N1(C(c2c(C)cco2)=O)CC2CC2(CNC(c2sccc2-n2cccc2)=O)C1 78843,c1(C(C)=O)sc2cccc(C)c2c1Cl.C1(=O)C(C)OC(=O)COC(C2CC2)CN1 78844,n1(CC(=O)NCCC(C)NC(C2CC2(Cl)Cl)=O)c(O)nc2ccccc12 78845,CCCCC(F)C(=O)N1CCCC1C=CC(N1CCC(CN=[N+]=[N-])C1)=O 78846,C(CCF)(C(=O)NCC1(CO)CCCC1)NC(C1(OCC)CCC1)=O 78847,CC1(CCNC(c2cscn2)=O)CCN(C(=O)CC2(C)CCCO2)C1 78848,c1(CC)cc(CC(=O)N(CCC(=O)N(CC(C)OC)CC(C)C)C)on1 78849,C1(NC(C(CCC)C)=O)(CNC(c2cc(C)nc(OC)n2)=O)CCCCC1C 78850,C(=O)(CC(C)CC(F)(F)F)NC1CCC(C)N(C(C2(O)CCCC(C)(C)C2)=O)C1 78851,C(CC(C)C(=O)NCCC(O)CNC(C1(CCN2CCCCC2)CC1)=O)=CC 78852,S(=O)(=O)(c1ccccc1F)N1CCC(CN(C(CCCC=C)=O)C)CC1 78853,C1(C(C)C)CC(C(=O)NC(c2nccs2)CC2CC2)CCO1 78854,c1(C(=O)NCC(CNC(C2C(C#N)C2)=O)CO)ccc(OCC2CC2)nc1 78855,C1(CNC(CN(C(C)=O)C)=O)CCCC(NC(c2ccc(OCCO)cc2)=O)C1 78856,c1(OCC)ccc(Br)cc1CN1CCC(NC(c2cc(CC)[nH]n2)=O)C(O)C1 78857,N1(C(C2(CNC(C3C(CC(C)(C)C)C3)=O)CC=CC2)=O)CC2(CCCC2)C1 78858,C1(NC(C(CCSC)OC)=O)CN(C(=O)C2CC2)CC2(CC2)C1 78859,C12(NC(C(C)CC(N)=O)=O)CCC(CNC(c3cccnc3O)=O)(CC1)OC2 78860,c1(C(=O)NCCCCCNC(C2C(C=C)C2)=O)cc(=NS(C)(=O)=O)cc[nH]1 78861,c1(CNC(c2ccc[nH]2)=O)c[nH]nc1C(=O)NCCC1CCOC1 78862,Cc1ncccc1C(N1CC(NC(=O)COC2CCN(C)CC2)C(C(F)F)C1)=O 78863,c1(C(=O)NC2(CC=C)CN(C(c3ccccc3CC)=O)C2)nc(=O)n(C)[nH]1 78864,C(CCC(C)C(=O)NC(C)C(C)(C)C(=O)NCc1cc(C)sc1C)OC 78865,c1(OCC)ncc(C(=O)NCC2CCN(C(C3CC(O)CN3C)=O)C2)cc1Cl 78866,N1(C(C(CC=C)CC)=O)CC2CC(CNC(c3ccc(C)cc3C)=O)CC1C2 78867,C(C(C)(C)C1=CCCC1)N(C(=O)CONC(=O)CNC(=O)Nc1ccccn1)C 78868,N1(C(Cn2ncc(C)c2)=O)CC2CCC(NC(=O)CCS(C)=O)CC1C2 78869,c1(C(=O)OC)ccc2[nH]c(=NCC3CCN(C(=O)CNC(N)=O)C3)sc2c1 78870,C1(CC)(CC)CC(NC(=O)C(C(C)(C)C)OC)CN1C(c1cc(O)no1)=O 78871,c1(OC)cncc(C(=O)NCC2CC2NC(C2CC(n3cnnc3)C2)=O)c1 78872,n1(CC)nnc(C)c1C(=O)NCC1CCCN(C(=O)C(F)CC2CCC2)C1 78873,CC1CNc2ccc(C(=O)N(C(C)CCNC(=O)C(N)=O)C)cc21 78874,CC(=O)CCCC(C)C(=O)NC1(C(N2CC(C)C2)=O)CC(O)C1 78875,c1(CNC(CC(CC)N(C(C(CCC)OCC)=O)C)=O)cccc(F)c1F 78876,N1(C(CSc2n(C)cnn2)=O)CC(NC(=O)CCO)CC1CO.C1(CF)CCC1 78877,c1(CN(C(C(C2CCCC2)NC(C2CC(=C)C2)=O)=O)C)cccnn1 78878,C1(C(C(=O)N(CC)CC)(C)C)CCCN(C(=O)CC(=O)NCC2CC2)C1 78879,C1(CNC(c2cn(C)nc2)=O)CCC2(CO1)CC(NC(=O)C=Cc1ccco1)C2 78880,CC1CCc2nc(N3CCC(CO)C3)[nH]c(=NCc3ccc(S(N)(=O)=O)s3)c2C1 78881,N1(C(C(C(C)C)OCC)=O)Cc2occ(C(=O)NC(C)C(CC)CC)c2C1 78882,C=CCC(CNC(=O)C(CC)C(=O)OC)C(=O)NC(C)CSC 78883,C1(NC(c2c(CNC(CCC(C)N(C)C)=O)n[nH]c2)=O)CCC(O)C(O)C1 78884,C1(C(=O)NC(C(=O)OC)Cc2cn(CC(C)(C)C)nn2)CCn2cncc2C1 78885,Cc1cnccc1CCNC(N1CCCC1Cc1cnn(C)c1N)=O 78886,C1(NC(CS(CC)(=O)=O)=O)CN(C(=O)Cc2conc2C)Cc2ccnn2C1 78887,c1(OC)ccc2c(N3CCCN(C(c4cc(C)ccc4Cl)=O)CC3)ncnc2c1 78888,CC1(C(=O)NC2CC2NC(C2(CC3CC3)CCOCC2)=O)CCCCO1 78889,c1(CNC(CC2(C)CCCN2C(=O)Cc2cnoc2)=O)cc(F)cc(F)c1 78890,CC1(C)Oc2ccsc2C(NC(c2c[nH]c3ccc(Br)cc3c2=O)=O)C1O 78891,c1(CC(CCNC(=O)NCC(C)=O)N(C)C)c(Br)c(C(F)(F)F)nn1C 78892,c1(CC)c(C(=O)N(C2CCCN(C(=O)CC(C)(C)OC)C2)CCF)cccc1F 78893,C(=O)(C#CC1(C)COC1)NC(C(=O)NC(c1nc(=O)o[nH]1)C)Cc1cn[nH]c1 78894,N1(CC(C)(C)CCOCCOC)CCN(C(=O)C(C)(F)c2ccon2)CC1 78895,C1(CCCNC(C2CC(OC)C2)=O)CCN(C(=O)Cc2nnc(C)o2)CC1 78896,c1(OC)cnc(C(=O)NCC2(F)CC(CNC(=O)C=CC(F)(F)F)C2)nc1 78897,C(=O)(CC(C)(C)CNC(=O)CCCC1CC1C)NCC1(OC)CCOC1 78898,C=CCCCC(=O)NC(C1CCCCC1)C(C)NC(=O)CCc1ccoc1 78899,N1(C(C)C)CC2(CC2)CC1C(=O)N(CCCO)Cc1ccc(CO)cc1 78900,C1(N(C(c2c(CC)c[nH]n2)=O)C)CCN(C(=O)CCc2cn(C)nn2)CC12CC2 78901,CS(=O)(=O)c1ccc(F)c(C(N2CCCN(C(=O)C3=CCOC3)C(CO)C2)=O)c1 78902,C1(C)(C(N(CCCCN(C(C(CC)(C)C#N)=O)C)C)=O)CCCNS1(=O)=O 78903,c1(C(=O)NCCC(C)NC(c2ccnc(N(C)C)c2)=O)c(F)ccc2[nH]ccc12 78904,CN1CCOC(C(=O)NCC2CN(C(=O)CCc3ncc[nH]3)CC2(F)F)C1=O 78905,c1(CNC2C(C(=O)NCCCC(F)(F)F)CCCC2)ccc(O)cc1Cl 78906,C1(C)(CNC(C2CN(C(C)C)C2)=O)CCCN(C(C2C3CCCC23)=O)C1 78907,c1(NC(c2c(NCc3c(C)c(Cl)ccc3)cnc(Cl)c2)=O)c(Br)ccc(F)c1F 78908,CC1(CNC(=O)CNC(C2(C)CCCOC2)=O)CC2(CCC2)C1 78909,c1(SC)ncc(C(F)(F)F)c(N2CC(F)(C(=O)NCc3ncccc3Br)C2)n1 78910,N1(C(c2[nH]cc(CC)c2)=O)CCCC(NC(=O)Cn2cnc([N+](=O)[O-])c2)C(F)C1 78911,C(CCC)(C(=O)N1CC(CNC(c2cn(C(C)C)cn2)=O)(COC)C1)=CCC 78912,Nc1cc(Cl)ncc1C(=O)NC1CC2CCC1(CNC(=O)Cn1ncnn1)C2 78913,C1(CN(C)C(c2csc(Cl)n2)=O)COCCN1C(c1ccsc1Cl)=O 78914,CC(CS(C)(=O)=O)C(=O)NC1CC(CNC(c2ccc(-c3cc[nH]n3)s2)=O)C1 78915,Cc1[nH]nc2c1CN(C(C1CCCC1CNCc1ccco1)=O)CC2 78916,c1(C(N(C2CCN(C(=O)CN3CCOCC3)C2)CC)=O)ccnc(C(C)(C)C)n1 78917,O=C(C1=CS(=O)CCC1)NC1CC2CC1N(C(c1cncc3[nH]ccc13)=O)C2 78918,N1(C(c2sccc2Cl)C(=O)NCc2cccc(OC)c2)CCc2cccnc2C1 78919,CC1(O)CCN(C(C2CCCCC2NC(C2CCCC(C#N)C2)=O)=O)CC1O 78920,C1(OC)CC2CC(C(N3CC(NC(c4cccc(C)c4)=O)C3)=O)CC12 78921,C1(C#N)(C(=O)N(CC)CC)CCN(CC(CO)CO)CC1 78922,c1(CNC(CC2(CC(=O)OC)CC2)=O)ccoc1NC(C1CC1C(N)=O)=O 78923,N1(C(C2N(CC)CCC2)=O)CCC(O)CC1C(=O)NC1C2C=CC(C2)C1CO 78924,c1(C(=O)NC(C(=O)N(CCOCCOC)C)CC2CC2)ccc(=O)n(C)c1 78925,C(=O)(C1=CCCCCC1)N1C(C)(C(=O)NC(C)CN2CCCCC2)CC(O)C1 78926,C1(C)(C(N2C(CNC(c3ccc(CC)[nH]3)=O)CC2)=O)CCCCCC1 78927,C(c1ccc(C2CC2C)o1)=CC(=O)NC1C(CNC(COC2(C#C)COC2)=O)C1 78928,Cc1cc(C(N2CCC(O)(CNC(c3coc(C(C)C)n3)=O)CC2)=O)cc(O)c1 78929,c1(C(=O)NC2C=CC(CC(=O)NCCCN(C)C)C2)cc(O)cc(F)c1 78930,C1(C=C)(C(=O)NC2(CC=C)CN(C(c3cc(Cl)ccc3N)=O)C2)CCCCC1 78931,N1(C(C(C)C)=O)CC(NC2CN(C(=O)OC(C)(C)C)C2)C1(C)C 78932,C1(NC(C2C(C)(CO)C2)=O)C=CCC(C(=O)NCc2ncoc2C2CCC2)C1 78933,N1(C(C2(C)CCCCO2)=O)CCOCC(NC(c2c[nH]nc2-c2cccs2)=O)C1 78934,n1(C(C)C)ncc2c(N(CC(Cl)Cl)C)nc(N3CCCC(C)(C(C)C)CC3)nc12 78935,C#CC1(C(N2CCC(NCC)C2)=O)CCN(C(C2CN(C3CCC3)C2)=O)C1 78936,Cc1onc(Br)c1C(N1CCC(C(C)NC(c2cccnc2O)=O)C1)=O 78937,CC(C)C(F)(F)CC(=O)NCCN(C(=O)CC1CCC(C)C1)CCOCCO 78938,c1(OC)ccc(C(N2CC(C(C)NC(c3c(C)noc3C(C)C)=O)C2)=O)c(F)n1 78939,C(CC(O)CC(=O)NC1CC(NC(=O)CC(C)O)C1)SC 78940,c1(N2CCC(CC=C)(NC(C3CC4CCCC34)=O)C2)ncnc(Cl)c1C#N 78941,C1(NC(C2N(C(c3cn(CC)nc3C)=O)CC3CC32)=O)CC2(CCC2)C1OC 78942,CC(C)C(CCN(C)C(C1COCOC1)=O)NC(C1CCOC1(C)C)=O 78943,CCCN=C(NCC(c1cc(C)cc(Cl)c1)(C)O)N1CCN(C2CC2)C(=O)C1 78944,CC(C)(C(C#N)OC(c1cc(C2CCNCC2)no1)=O)c1ccc(F)cc1 78945,c1(C(N(CCCNC(C(C)OC)=O)C)=O)ccc(N(C)C)c([N+](=O)[O-])c1 78946,c1(OC)cccc(CNC(=O)NCC2CCN(C)CC2c2ccnn2C)c1O 78947,n1(CC(=O)NCCCN(C(CC(=O)NCC)=O)C2CCCC2)nc(C)ccc1=O 78948,C(=O)(C1=CCCCC1)N(CC(O)CNC(C1CC12CC2)=O)C 78949,C1(C(=O)NCC2C(NC(c3ccc(NC)cn3)=O)CCC2)CN2CCN1CC2C 78950,N1(C(C(C(CC)O)C)=O)CC2CCC(C1)N2C(=O)C(NS(=O)(=O)N(C)C)COC 78951,C1(C(N(C(c2ccco2)C)C)=O)CN(C(=O)C(F)CC(C)(C)C)CC1C1CC1 78952,CC(CC1CCCC1)C(C(=O)NC1(C)CC1)N1CCC(c2nc(O)n[nH]2)CC1 78953,CCCS(=O)(=O)CC(=O)N1CC2CC1CC2NC(=O)CSc1cc[n+]([O-])cc1 78954,N1(C(c2cc(OC)no2)=O)CC(NC(c2ccc(CCC#N)cc2)=O)C(C)(C)C1 78955,C(=O)(CC(C)n1cc(Br)cn1)NC(COC)CNC(=O)COCCF 78956,c1(C(=O)NCCCCCN(C(C2C(C(C)C)C2)=O)C)cc2cccc(Cl)c2s1 78957,c1(CC(=O)NC2C(NC(CC(C)(C)O)=O)CCCC2)c(Cl)cccc1Cl 78958,CC(CN(C(=O)C(N1CCC(c2cccc(Br)c2)CC1)=O)C)C(F)(F)F 78959,N1(C(c2c(C)onc2)=O)CCC2(CCC2)C(NC(C2CC3CC2C3)=O)C1 78960,C1(N(C(C(c2cnn(C)c2)OC)=O)C)CC2CC1N(C(c1ccc(F)cc1)=O)C2 78961,CC1(C)CCC2(CC1)CC2N(C)C(=O)NCC1CCc2nnnn2CC1 78962,c1(C(=O)NCC(C)CN(C)C(c2ccc(CO)c(F)c2)=O)cc2cn[nH]c2cn1 78963,C(CC(F)F)(C(=O)NC(C)C(=O)NCC1CC1)NC(CCC(=O)NC)=O 78964,C1(C#N)(C(N2CC(CNC(c3ccc(CSC)cc3)=O)C2)=O)C(C#N)C1(C)C 78965,C(C(C(=O)N1CCOC(COC)C1)C(C)(C)C)NC(C(C=C=C)C)=O 78966,c1(C(=O)NCCC(=C)CNC(c2sc(C)nc2C(C)C)=O)cccc(COC)c1 78967,C1(C)(CNC(C(C)(C2CCC2)NC(C2CCN(CC)CC2)=O)=O)CC2CCC1C2 78968,N1(C(c2n(CC)ncc2)=O)CC(CNC(=O)C(F)(F)C(O)C2CC2)CC1(C)C 78969,N1(C(c2nc(C)sc2)=O)CC2CCCC2(NC(=O)CN2CCC(=O)NC2=O)C1 78970,N1(C(Cc2c(C)ncs2)=O)CCC(C(N2CCN(C)CC2C)=O)C12CCC2 78971,N1(C(C)(C)C)CC(NC(=O)NCc2nc(CSc3ccccc3Cl)no2)CC1=O 78972,CCCC(CC(=O)NCCC(=O)NC1OCCCC1(C)C)OC 78973,Cc1c(C(N2CCC(O)(CCNC(c3cccc(=O)n3C)=O)C2)=O)cncc1N 78974,C1(CC(=O)NC2CN(C(c3c(C)oc(C(C)C)c3)=O)C(C)C2)CCCC(C#N)C1 78975,C(CC(C(=O)NC1CCOC1CC)NC(c1oc(C)nc1CC)=O)OCC 78976,Cc1cc(C(N2CC(CNC(=O)Cc3nccs3)C(C)C2)=O)c(C(F)(F)F)o1 78977,C(=O)(CC1OC(=O)c2ccccc21)NC(=O)NC1CC1c1c(C)ccc(F)c1 78978,CC(C)C(O)C(=O)NCC1CN(C(c2ccnc(-c3ccccc3)n2)=O)C1 78979,C(=O)(CC(CNC(c1ccccc1Cl)=O)C1CCC1)NCC1(CO)C(C=C)C1 78980,c1(CC(C(=O)O)NC(=O)NC2CCCC(C(N(C)C)=O)C2)cccc(Cl)c1F 78981,C1(NC(c2n(CC)cc(Cl)c2)=O)CCC(O)CN(C(=O)C=C(C)C(F)F)C1 78982,C1(CNC(Cc2ncc(C)s2)=O)CN(C(=O)Cc2cc(C3CC3)on2)C(C)(C)C1 78983,C1(C(=O)NCC(CNC(c2cnc(NC(C)=O)o2)=O)(C)O)CC12CCCCC2 78984,CON1CCC(C(=O)NCC2(O)CCCN(C(=O)CC3CCC3(C)C)C2)CC1 78985,N1(C(c2n(CC#C)cnn2)=O)CCOCCC1C(=O)NC1CCCCC1(C)C 78986,C(C(CNC(c1ncnc(C)c1C)=O)C(F)(F)F)NC(c1c(C)coc1C)=O 78987,N1(C(Cc2cccc(CC)c2)=O)CCN(C(=O)C(C)C(C)O)CC(C)(C)C1 78988,c1(CC)ccc(NC(C2(NC(=O)NCc3cnc(CN)o3)CC2)=O)cc1Cl 78989,Cc1cc(Br)ccc1C(N1CCC(CN(C)C(c2cccc(F)c2F)=O)CC1)=O 78990,c1(C(=O)NC2C(NC(=O)CC3C=CCCC3)CC2)cnc2ccccc2n1 78991,C1(C(=O)NC2CCCC(C(N(CCC)C3CC3)=O)C2)CC2(C1)CC(C)C2 78992,C1(CCC(=O)NCC(=C)CCNC(=O)C(C)c2cccs2)(CO)CCCCC1 78993,C=CCC(CC=C)NC(C1CCOCC1NC(=O)CC(C)F)=O 78994,c1(C(N2CCC(CCNC(CN(C(C)=O)C)=O)CC2)=O)cc(N)c(Cl)c(O)c1 78995,c1(C(N2CCC(NC(C3CC(O)(CC#C)C3)=O)C23CC3)=O)cc(N)cc(C#C)c1 78996,CC(=O)CCCCC(=O)N1CCC(C(=O)NCc2ncccc2F)(CF)C1 78997,N1(C(c2c(N)non2)=O)CCCC2(CCCN2C(C2C3CCCOC23)=O)C1 78998,C(N=c1[nH]c2ccc(Cl)cc2s1)C1C(C)CN(C(C2(C)CNC(=O)C2)=O)CC1 78999,c1(C(=O)NCC23CN(C(C(CC#C)C)=O)C(C2)CO3)cn2cc(Cl)cc(Cl)c2n1 79000,c1(CC)ccc(C)cc1NC1(c2nnnn2C(C)C(=O)OC)CC2(CSC2)C1 79001,CCCCCCCCC(=O)N(C1CCCN(C(c2ccc(N)c(O)c2)=O)C1)C 79002,CCC(C)(CC(=O)NCC1CC(NC(=O)CSC(F)(F)F)C1)C(=O)OC 79003,CC1(C)COCC1CNC(c1ccc(CNC(=O)CC2(N(C)C)CCC2)s1)=O 79004,C=CC1(c2cn(C3(C(N)=O)CC3)nn2)COCCN1C(C1CC(C)CO1)=O 79005,CC(C)(CC(=O)NCC12CCCC1CN(C(c1ccco1)=O)C2)CC(F)F 79006,C#CCC(CC(F)F)C(=O)N1CCC(CC)C1C(=O)NOCCC(C)O 79007,c1(C(=O)NC2(CNC(COC)=O)CCC2)nc(S(N)(=O)=O)c2ccccn12 79008,CN1CCN(C(=O)CCC2CCC(NC(c3ccsc3)=O)C2)C(C2CCC2)C1 79009,c1(OC)cccc(Cl)c1CN1CC(CO)(NC(c2cccnc2C(C)C)=O)C1 79010,CC1=C(C(=O)NC2CC(C)N(C(c3csnc3C)=O)C2)CCC(C)(C)C1 79011,C1(NC(=O)Cc2sc(O)nc2O)CCCC12CN(C(C1CCC(C(N)=O)O1)=O)C2 79012,C(CCc1ccco1)(C(=O)NCC1CC1)N(CCC#N)C 79013,Cc1cc(Br)c(NC(C2CC(F)CN2C(c2cccc(Br)c2Br)=O)=O)c(Br)c1 79014,C1(NC(C(c2cc(Br)no2)N(C)CC2CC2)=O)CCS(=O)(=O)C2(C1)CC(C(N)=O)C2 79015,c1(C(N2C(CNC(C(F)=CCC)=O)C=CC2)=O)cc2c(nc1O)CCCC2O 79016,CC(CC(F)(F)F)C(=O)NCCOCCCN(C)C(c1cc2ccccn2n1)=O 79017,C(CC(C)(C)C)(C(=O)NCC1(C)CCCS1)NC(C1=CCCC1C)=O 79018,c1(NCC(=O)N(CCCN(C(C(C)=C(C)C)=O)C)C)ncnc2sc(C)c(C)c12 79019,N1(C(C23C(NC(CCC(C)C)=O)CC(CC2)C3)=O)CC2CCC(C1)C2O 79020,c1(N2CCC(CCOC)(NC(C3CCC(C)C3)=O)C2)nccc(S(C)(=O)=O)n1 79021,n1(CCC(=O)NCCOC2CCN(C(C(C=C)O)=O)C2)c(C)csc1=O 79022,CON=Cc1ccc(C(=O)N(CCCn2cc(C(O)C(C)(C)C)nn2)C)cc1 79023,N1(C(CCN(C(CC(CC(C)C)C)=O)CC2CC2)=O)CCc2ccc(C#N)cc21 79024,N1(C(C(=O)NCCCSC)C2CCOC2)CCCC(c2nncn2C)C1 79025,C1(C2(CNC(C3(C)CC3)=O)CC2)CCCN1C(=O)CC(O)C1CCC1 79026,C(C(CC)CCCC)c1n(-c2c(COC)cccc2)nc(C2CSC2)n1 79027,c1(C(=O)NC(CC)CNC(=O)CC(C)N(C)C)ccc(N)c(Cl)n1 79028,C1(NC(CNC(C(CC)CC)=O)=O)CN(C(C2CCC2OC)=O)CC12CCC2 79029,N1(C(C23CN(C(C4C(C(C)C)C4)=O)C(C2)CO3)=O)CCN2C(=O)NCC2C1 79030,c1(CNC(C(CC=CC)C)=O)nc2ccc(C)cc2s1 79031,C1(CC)CCCCC1OCC(=O)NCC(C)(C)CN(C(=O)C=CC(C)CC)C 79032,N1(C(CN2C(=O)CNC2=O)=O)C2CCC1CC(NC(C1(F)CCOC1)=O)C2 79033,C(C)(CC(=O)NC12CC(NC(=O)C(C)CC3CC3)(C1)C2)SC 79034,C(=O)(CCCCCCCCCO)N(CCNC(c1cccc(CC#N)c1)=O)CC 79035,CC1CN(C(=O)C(C)Oc2cccc(F)c2)CCN1C(=O)C(C)(C)C#N 79036,Cc1nc(O)c(C(=O)NC(C)(C)C(C)NC(=O)C=CC(F)(F)F)cc1Br 79037,C(=O)(C(O)C(F)(F)F)NC(C1(CNC(=O)CCc2ccccc2Cl)CC1)C 79038,C(CCC(C)C)(C(=O)NOCCC(C)O)NC(CC)(C)C(=O)OC 79039,N1(C(C2C(C(N)=O)C2)=O)CC=C(C(=O)Nc2c(O)cccc2Cl)CC1 79040,CC(C)(C)C(CNC(c1cccc2nccn12)=O)C(=O)N1CC=CCC1 79041,N1(C(CC2CC(C)(C)OC2)=O)CCCC2(NC(=O)Cn3cccnc3=O)CC2C1 79042,c1(N2CCC(C)C(CO)C2)ncnc2cc(F)c(F)cc12 79043,C1(C)(C(N2CC(COC)(CNC(C3CCCOC3)=O)C2)=O)CC2CC2C1 79044,N1(CCC)CCCC(C(N2CCCC2C(C)NC(=O)CC(C)(C)O)=O)C1 79045,CCC(CN=c1nc2c(cnn2C)c(NC(c2ncc(Br)cn2)C)[nH]1)N(C)C 79046,C(=O)(CC(C(N)=O)N(C)CC)NCC(C1CCCC1)NC(CCCOCC=C)=O 79047,c1(C(=O)NCC(O)CCNC(C2COCCC2(F)F)=O)ccc2ccnn2c1 79048,N1(C(Cn2c(C)ncc2)=O)CCC2CN(C(C34CC(C#N)(C3)C4)=O)CC2CC1 79049,N1(C(Cc2c(C)cc(F)cc2)=O)CC(C2CN(C(c3n[nH]c(C)c3O)=O)C2)C1 79050,Cc1cc(C(=O)NC23CCOC(CNC(C4CCCCC4C)=O)(C2)C3)ccc1Cl 79051,c1(CN2CCN(C(c3c(C)nsc3)=O)C(C)C2)ccccc1[N+](=O)[O-] 79052,c1(CC)ccc(NC(C2CCCN2C(C2CCCN2C2CC2)=O)=O)cn1 79053,CC(C)C(CNC(C1CCN1C)=O)C(=O)N1CCC1c1ccccc1 79054,O=S(=O)(c1cccc(O)n1)N1CCN(C2CCC2)CC1 79055,Cc1ocnc1C(N1CC(CC(C)NC(=O)C=CC2CCCO2)C1)=O 79056,C1(C(=O)NC2C=C(C)CCC2)CC2CC1CN(C(c1cn(CCO)nn1)=O)C2 79057,CCC(CC(=O)NCC1(C)CCC(NC(c2ccc(CO)o2)=O)C1)CC(F)(F)F 79058,c1(C(=O)NCC2C(C)CCN2C(=O)CC2CN(C)C2)nccc2ncccc12 79059,N1(C(C(Cc2cn[nH]c2)NC(=O)CC2CCCCC2)=O)CCC(O)(C(F)F)C1 79060,C(=O)(C1SCCc2sccc21)N1CC(C)C(O)C1 79061,c1(NC(C(=O)NC2(C)CCN(C(c3c(CC)nn[nH]3)=O)C2)=O)ccc(Cl)c(F)c1 79062,C(=O)(CCCCCC(C)O)NC1C2CN(C(c3nn(CC)c(C4CC4)c3)=O)CC21 79063,c1(C(=O)NCC(CC)NC(c2cc(C)c(C)cc2Cl)=O)ccc2c(c1)nnn2C 79064,Cc1occc1C(=O)NCC(=O)NCC1(NC(C2CCC3CC23)=O)CCC1 79065,c1(CC(C(=O)O)NC(C2CCC(CC)C2)=O)c(F)cccc1Cl 79066,C(=O)(CC1CN(C)c2ccccc21)NCC1CC(NC(C2=CCCC2C)=O)C1 79067,N12CCOCC(C1)C(=O)N(C)C(C)C2=O.c1(OCCSCCCC)cccc(Cl)c1 79068,c1(CCC)cc(C(=O)NC2CC(CNC(C3CC34CCC4)=O)CC2O)nn1C 79069,c1(C(=O)NCC2(CN(C(C(CC)SC)=O)C)CC2)cnn(CCO)c1C 79070,Cc1ncc([N+](=O)[O-])n1CC(=O)NCCCCC(CO)NC(c1n[nH]cc1Cl)=O 79071,c1(NC(CCC(C)(C)C#N)=O)cccc2c1CNC2=O 79072,Cc1ccc(S(=O)(=O)NC2CCOCC2Cc2ccccc2)cc1[N+](=O)[O-] 79073,C(C(=O)NOCCNC(c1cnsc1)=O)OCCOCC 79074,N1(C(C2CC(C)(F)C2)=O)CCN(C(=O)C=CCO)CC2CCCCC12 79075,C1(NC(c2c(C)[nH]c(=N)s2)=O)CCN(C(=O)CN2CCC(C)C2)CCC1(F)F 79076,C1(C(=O)NCc2c(C)cccc2O)CCC2CCC1N2C(=O)CCNC(N)=O 79077,N1(C(c2c(OCC)cncc2)=O)CC2CC(NC(=O)C=CCF)CC1C2 79078,CC(C)CCCC(=O)N1CC2(CNC(=O)C(O)Cn3cncn3)CC1CO2 79079,N1(C(CCCSC)=O)CC=CCC1C(N1CCCC1CC(C)C)=O 79080,c1(C(N2CC(CCC)C(NC(=O)C(c3ccccc3)F)C2)=O)cc(C)cc(O)c1 79081,N1(C(C2C(=C)C2)=O)CCC2(COC(CNC(c3sc4cncn4c3C)=O)C2)C1 79082,c1(NC(C2CCS(=O)(=O)C2)CSC)ccc(S(=O)(=O)NCCC(F)(F)F)c(Br)c1 79083,C1(C(=O)NC2CCN(C(CCSCCC)=O)C2C)CCC2CC1CO2 79084,N1(C(C(CC)C#N)=O)CCN(C(c2n[nH]cc2F)=O)CC1c1cc(F)cc(F)c1 79085,C1(C(=O)NCC=CC(C)(C)C)CC2(CCN(C(=O)CCc3cncs3)C2)C1 79086,Cc1oc(CNC(C2CCCC(F)C2)=O)nc1C(=O)N(C1CSC1)C 79087,c1(C(=O)NCC2CC(NC(C3C(C)(CC)C3)=O)C2)cnc(C)n1C(F)F 79088,C1(C(=O)NC2(C(=O)NC(c3cccs3)CO)CSC2)(CC)CCOC1 79089,C1(NC(C=CCNC(C(C)NC(C)=O)=O)=O)CN(C)CC12CC2 79090,c1(CCC)cccc(C(=O)N(C)CC2CCN(C(C34CC(C)C3C4)=O)C2)c1 79091,N1(C(CCC(=O)NC)=O)CCn2nc(CNC(=O)CC(O)C3CCCC3)cc2C1 79092,c1(C(=O)NCCNC(C(C=C=C)C)=O)cc(Br)ccc1N1CCCC1 79093,c1(-c2scc(CC(=O)N(c3ccc(Cl)cn3)C)n2)ccccc1Cl 79094,N1(C(CCn2c(C)ncc2)=O)CCCCCCC1C(=O)N(C)CC1CCOC1C 79095,N1(C(C=CC=CCC)=O)CCC(C)(CCNC(C2(C)CC2(Cl)Cl)=O)CC1 79096,c1(C(=O)NCC2C=CC(NC(=O)Cc3cc[nH]n3)C2)cnc(C(F)(F)F)c(Cl)c1 79097,C1(NC(C(C2CCCC2)NC(C=C(C)C)=O)=O)CC(F)(F)C1(C)C 79098,C1(C(N(CC(O)CNC(c2cscc2Cl)=O)C)=O)Cc2nccnc2C1 79099,C1(C(=O)NC2CC(CC(=O)NCC(=C)CC)C2(C)C)CCCCC(=O)C1 79100,N1(C(C2CCCC(=O)CC2)=O)CCCC2(C1)CN(C(c1cnnc(Cl)c1)=O)C2 79101,N1(C(c2cc(C)sn2)=O)CCN(C(c2ccnc(C(C)C)n2)=O)C2CCCCC12 79102,C(=O)(CC(C(F)(F)F)NC(=O)CC1OCCCO1)NC(CC)C(=O)NC 79103,C12(CC(N3C(CN(C(=O)CC4CCNC4=O)C)CCC3)=O)COC(C)(C1)C2 79104,C(C1=CCN(C(=O)Cc2cccs2)CC1)NC(c1c(SC)n(C)nc1)=O 79105,CC1CCCN(C(=O)CCCCCN(C)C)C1CNC(=O)CCC1CCC1 79106,n1(C(CC)C)nnnc1C1(NCC(C)(C)n2cccn2)CCC1CC(F)(F)F 79107,c1(C(=O)NCCCCNC(C2C3CCC2(c2cncs2)C3)=O)cccc(Cl)c1F 79108,CC(C)CCCCCC(=O)NCC(C)CNC(=O)C=CC1CCOC1 79109,CCC(C)(C)C(O)C(=O)NCC1(O)CCN(C(=O)C(C)(C)C(C)C)C1 79110,CCCCC(CC)CC(=O)NC1CN(C(c2c[nH]nc2CCC)=O)CC1N=[N+]=[N-] 79111,C=CCCC(CC(C)C)C(=O)N(CCCCCNC(C1CC12CC(C)(C)C2)=O)C 79112,N1(C(COCCCC#C)=O)CCC2(CCCCN(C(=O)C#CC(=O)N(C)C)C2)C1 79113,CC1CCN(C(=O)COC2CC=CC2)CC1NC(C1CCOCC1(C)C)=O 79114,C1(CC)(NC(c2ccc(C#N)s2)=O)CCN(C(=O)CCC2CCC(C)O2)CC1 79115,C(c1ccccn1)=C(C)C(=O)NC(C1CCCC1)CNC(C1(C#N)CC=CC1)=O 79116,C(CNC(=O)CSCCC#N)(CCCC)NC(c1cc(CC)no1)=O 79117,C(c1cccnc1)=C(C)C(N1CCC(=CCNC(=O)CC2(C)CC2(F)F)CC1)=O 79118,CC1COC(CO)CN1C(=O)CCN(C(=O)CCc1cccs1)CCO 79119,C1(C)(NC(CN2C(C)CCCC2)=O)CCCN(C(=O)CC2CC3CC3C2)C1 79120,Cc1ccc(C2(C(=O)NCCC(C(C)C)NC(=O)C(O)C(C)C)CCC2)cc1 79121,c1(NC(C(N2C(C(C)N)CCCC2)=O)=O)coc(S(C)(=O)=O)c1 79122,C1(OC)CN(C(c2ccn(CCF)n2)=O)C(C)(CNC(C2CC3(CC3)C2)=O)C1 79123,c1(C(N(CC(C)C(=O)NC2CCN(CCF)C2)C)=O)cnn(C)c1Cl 79124,c1(C(=O)NC2(C(F)F)CC2)cnn(-c2ccccc2)c1I 79125,n1(CC(=O)NC(C2CCCN(C(c3cnco3)=O)C2)C)cc(Br)c(=N)[nH]1 79126,c1(CC(=O)NCCOCC=CCSC(C)C(=O)NC2CCCO2)ccc(O)cc1 79127,c1(NC(C(=O)NC(C)(C)C)=O)ccc(-c2ncn(C(F)F)n2)cc1 79128,Cc1nc[nH]c1CC(=O)NC1(c2ccccc2)CC(NC(=O)C(C)SC(C)C)C1 79129,c1(CC(N2CC(NC(C(C(CC)O)C)=O)C2)=O)ccc2cccnc2c1 79130,c1(C(N(C)CC2(CNC(C(C)OCCCC)=O)CC2)=O)nnn2c1CCCC2 79131,C(=O)(C1=COCCC1)N1CC(NC(C2CN(C)CC2C(F)(F)F)=O)C1 79132,C1(C(=O)NC(CNC(C=Cc2cncc(C)c2)=O)CO)CC2(C1)CC(C)(C)C2 79133,N1(C(c2ncc(C)s2)=O)CC2(CCC2)CC1CNC(C1COCCN1C)=O 79134,N1(C(c2ccc(C)nn2)=O)CC2CCCC1(CNC(=O)C(O)C1CCCC1)C2 79135,N1(C(CC=C=C)=O)CCC2CN(C(=O)CCSc3ccc(Cl)cc3)CCC2C1 79136,c1(C(N2CC(NC)C2)=O)ccc(S(=O)(=O)N(C)Cc2ccc(F)cc2)o1 79137,C(CC(=O)NC(c1ccc(C)nc1)C)(C(F)(F)F)NC(C=CCC)=O 79138,CC(C)(CNC(=O)C(F)CC1CN(C(=O)CC(C2CC2)C2CC2)C1)C(F)(F)F 79139,CC(CCC(=O)NCCN(C1(CO)CC1)C)N(C)C.C12(CCC1)CC(=O)N2 79140,C(N=c1[nH]c(=NCc2ccc(Cl)cc2C)[nH]c2c1CCC2)c1ncc(C)cn1 79141,N1(CC2CN(C(c3cc[nH]n3)=O)CC23CCC3)C(=O)c2ccccc2C1=O 79142,C1(N(C(CCOCC#C)=O)C)CCCCN(C(=O)CCC2CCCCO2)C1 79143,N1(C(c2ccco2)CN(CC(=O)NC(C)(C)C)C(=O)C2CC2)CC2CCCCC2C1 79144,C12(NC(Cc3ccn(C)n3)=O)CCCC1N(C(c1cc(F)cnc1O)=O)CC2 79145,C1(CC#C)(C(=O)N(CC)Cc2ccco2)CCN(C(=O)CN2CCCCC2=O)C1 79146,N1(C(c2c(OC)csc2)=O)CC2=C(C1)CN(C(C1(C(F)(F)F)CC3CC3C1)=O)C2 79147,CCCC(C)CC(=O)N1CC(CCNC(C2CC23CC(OCC)C3)=O)C1 79148,c1(C(N2CCN(C(C3CCSCC3)=O)C3C2C3)=O)cc2nc(=O)ccn2[nH]1 79149,N1(C(C2CN(CCC)C(=O)C2)=O)C2CCCC1CC(NC(c1cscc1C)=O)C2 79150,Cn1c(C(=O)NC2CCCC(CNC(C3CC4(CC4)C3)=O)C2)cnc1S 79151,c1(C(C)=O)ccc(C(N2CC(NC(=O)C(C)OCCC(C)C)CC2C)=O)cc1C 79152,C(C(F)(F)C(=O)NCC1(C)CCCC1NC(=O)CC1COCCN1C)N(C)C 79153,C1(NC(c2cc(COC)on2)=O)CN(C(C2CCOC2C)=O)CCC12CCC2 79154,c1(C(N2C(C(N(CC#C)C3CC3)=O)CC2C)=O)ccc(C#N)cc1C 79155,c1(C(=O)NCC2(NC(C(CC)SC)=O)CCC2)cc(NC)nc(Cl)c1 79156,C1(C)(CCNC(C(C)=CC2CC2)=O)CCN(C(=O)C=C2CCC2)C1 79157,c1(C(N2CCC(CCNC(c3c(CCC)nco3)=O)C2)=O)c(C)nnn1CC 79158,N1(C(CCOCC#C)=O)CCC2(NC(c3ccc(CSC)cc3)=O)CC2C1 79159,C1(C)(C(N(CCCCN(C(c2cnc(C)s2)=O)C)C)=O)CCCN(C)C1 79160,CC(C)(O)CC(=O)NCC(O)CCNC(C1CCCC(O)C1)=O 79161,N1(C(CCCNC(CC(=O)NCC#C)=O)=O)CC(C#N)C2(CCC2)C1 79162,C1(NC(C(c2cccc(F)c2)C)=O)CC(NC(c2cc(C(N)=O)c[nH]2)=O)C(O)C1 79163,C1(NC(c2c(Br)cn(C(C)C)n2)=O)CC(F)CN(C(=O)COCCF)C1 79164,N1(C(CCC(C)SC)=O)CCCC(NC(=O)C=Cc2cnn(C)c2)CC1 79165,C1(CC)(CC)CC(NC(C2CCCC2CNC(=O)CC(=O)OC)=O)C1 79166,c1(C(=O)OCCc2cccc(OC)c2)cccc2c1NC(C)CC(=O)N2 79167,c1(C(=O)NC2CCC(CNC(c3c(N)c(O)ccc3)=O)C2)ccc2ncnn2c1 79168,C1(NC(C=CC(C)C)=O)CN(C(C2CC2C2CC2)=O)CC1c1cccc(F)c1 79169,Cn1cc(S(=O)(=O)NC(C2CC(N)(C(F)F)C2)=O)nn1 79170,c1(C(=O)NCCOC2CN(C(=O)CCC3CC3(Cl)Cl)C2)ccc(O)nc1Cl 79171,C(CNC(=O)CC(C)Cc1ccc(Cl)cc1)(C(C)(C)C)NC(CSCC#C)=O.C 79172,N1(C(c2n[nH]c(=N)[nH]2)=O)CC2CC(NC(=O)CCc3cccs3)CC2C1 79173,N1(C(C2C(c3c(C)n(C)nc3)C2)=O)CC(NC(=O)C(C)C(C)C)CC(F)C1 79174,C(CCCCC(=O)NC1(C(=O)NCc2cccc(F)c2C)CCC(C)(C)C1)OC 79175,CC1CC(=O)CCC1C(=O)NC(C(=O)NCCC(=O)NC1CC1)C1CCC1 79176,N1(C(=O)C=CCBr)CC2(C1)CN(C(c1c(Cl)ccnc1Br)=O)C2 79177,N1(C(C(CCC)Cl)=O)C2CCC(C2)C1C(N1CCCC(C)C1)=O 79178,C(=O)(C(C(C)C)OCCNC(=O)C(C)C)N(CC(CC)OC)CC 79179,C1(NC(CC(C)C(F)F)=O)CC2CC(C1)N(C(=O)CCCc1ccc(N)cc1)C2 79180,C(=O)(C#CC(=O)N(C)C)NCC1C(NC(c2c(CCC)occ2)=O)CCC1 79181,Cc1nccc(C(N2CCC(O)(CNC(c3cc(Cl)cs3)=O)CC2)=O)c1C 79182,c12cn(nn1)CC(=O)NC2(C)C.c1(C(=O)OC(C)(C)C)csc(Cl)c1 79183,CC1(CC(N2CC3CC3C2C(=O)NCC2C3CCCC23)=O)CCCCC1 79184,Cc1nc(C)n(O)c1C(=O)NCC(CNC(=O)Cn1ccc([N+](=O)[O-])n1)CO 79185,N1(C(C(N2CCOC2=O)C)=O)C2CCC1CN(C(c1cncn1C)=O)CC2 79186,C1(C(=O)NCC2(F)CCN(C(C(C=C)O)=O)C2)(OC)CCCCCC1 79187,C(=O)(CCC(F)(F)F)N1C(C)(CC(=O)NC(C(=O)OCCCC)C)CC1 79188,N1(C(C2CCN(C(CCC)=O)CC2)=O)CCCC2(NC(C3CCC3)=O)CC2C1 79189,C1(NC(C2CC(F)(F)C2)=O)CC2CC(C1)N(C(=O)CCc1ccc(Cl)c(F)c1)C2 79190,CC1(C(=O)NCC2CCC(NC(=O)CC(=O)NCC3CC3)CC2)CC2C=CC1C2 79191,c1(C(=O)NCC2C(NC(COCCC)=O)CCC2)ccn2c1CCCC2 79192,C12(CNC(c3cnc4cc[nH]c4c3)=O)CN(C(=O)CCC(F)F)CC1CCO2 79193,c1(OC(C)C)ccc(C(=O)NCC2CC(C)(C)CN2C(=O)C(C)N(C)C)c(Cl)c1 79194,c1(SCC(=O)NCC2CC2CNC(=O)Cc2nc[nH]n2)ccccn1 79195,C1(C(=O)OC)CC(O)CN1C(C1CCN1C(c1ccc(F)cn1)=O)=O 79196,c1(C(C(=O)NCC(C)NC(C2(CC#C)CCCOC2)=O)OC)c(F)cccc1F 79197,CCC(C)CCC(=O)NCC1(O)CCCN(C(c2ccnc(NC3CCC3)c2)=O)C1 79198,c1(C(N2C(CNC(C(C)c3ccsn3)=O)CCC2)=O)cc(C(F)F)cc(Cl)c1 79199,Cc1cc(-c2ccnc(CC(=O)NCc3cccc([N+](=O)[O-])c3)c2)cc(O)c1F 79200,CC#CCCCC(=O)NC(c1ccccc1F)CNC(=O)C(C)Cc1cnc[nH]1 79201,Cc1nn(C)c(N2CCN(C)CC2)c1CNCC1CC12CCC2 79202,C(=O)(C(O)CC(F)(F)F)NC(c1nocc1C(=O)Nc1ccc(O)c(F)c1)C 79203,c1(CNC(C2C(C(C)C)(CC)C2)=O)nc(CNC(=O)C(O)C(C)(C)C)cc(O)n1 79204,C1(NC(c2c(CC)ccs2)=O)C2CC1N(C(=O)CC1CC3CCC1O3)C2 79205,C1(C(N(CCCNC(=O)C2=CCCCC2)CCO)=O)CCCC2CCCN12 79206,c1(CC)cc(C(=O)NC2CCCCC2NC(C2CC(C(F)(F)F)C2)=O)c(C)o1 79207,C1(COC)CN(C(=O)CCCc2ccccn2)CCN1C(C1COC(=O)N1)=O 79208,N1(C(c2n(CC)nnc2)=O)CC(NC(=O)C2=CCCC(C)(C)C2)CC12CCOC2 79209,N1(C(c2c(O)ccc(C)c2)=O)CCCC(C)(C)C1C(=O)NCCC(C)(C)C 79210,c1(C(=O)NCCN(C(C2C(C)(C(C)C)C2)=O)C)ccc2c(=N)[nH]cnc2c1 79211,c1(C(C(N2CCC(N(C(=O)CC3CC3)CCO)C2)=O)O)ccc(Cl)c(Cl)c1 79212,c1(C(C)C(=O)NC2C3CC(C(=O)O)CC23)n[nH]c2c1CCCC2 79213,C12(NC(CCCNC(c3c(C)nn[nH]3)=O)=O)CC1COC2(C)C 79214,c1(C(=O)NCC2(CNC(CCCOC)=O)CCC2)cccc(C(=O)OC)n1 79215,Cc1c(C(=O)NCC2CC2NC(c2ccn(CC#N)n2)=O)ccn1CCO 79216,c1(C(c2n(CCCC)nnn2)NCCCCC(C)(C)C)ccc2c(c1)OCCO2 79217,c1(CCC)cc(C(=O)NC2CC2CNC(=O)C=CCN2CCCCC2)nn1C 79218,c1(CC)c(C(N2CC(CCNC(C3C4CC4C4CC34)=O)C2)=O)oc2ccccc12 79219,C1(C(=O)NCc2cc(C)no2)(NC(=O)COc2ccsn2)CCCC1C 79220,C1(NC(c2cc(Cl)cc(F)c2F)=O)CN(C(C2(O)CCOC2)=O)CC2(CC2)C1 79221,c1(C(=O)NCC2CN(C(CN(C(=O)OC)C)=O)C3C2C3)ccnc2c1nnn2C 79222,N1(C(CC(C)(C)N(C)C(C2CC(=O)CC(=O)C2)=O)=O)CC2(CCC(=O)N2)C1 79223,N1(C(C(CC)COC)=O)Cc2ccc(CNC(C3CCCC3)=O)cc2C1 79224,c1(C(=O)NCC2C3CN(C(C(CC(N)=O)O)=O)CC32)cccc2nc(O)[nH]c12 79225,Cc1ccc(O)cc1C(N1CCC(CC(N2CCOC(C(N)=O)C2)=O)C1)=O 79226,N1(C(CN(C)C(N)=O)=O)C2CCCC1CC(CNC(C1(O)CCC1)=O)C2 79227,C1(O)(CNC(Cc2c(C)oc(-c3ccco3)n2)=O)CCCN(C(=O)C=CCO)C1 79228,C(C)(C)(CC(=O)NC1CCCN(C(C2CCCC2c2ccc(F)cc2)=O)C1)SC 79229,N1(C(C(COCC)n2cc(COC)nn2)=O)CCCC(OC2CC2)C1 79230,C1(NC(CC=CCC)=O)CCC2(CCCN(C(c3cncc(C4CC4)c3)=O)C2)C1 79231,c1(OC)ccc(CNC2CC2C(=O)NCc2ccncc2C)cc1Br 79232,c1(CN2CC(NC(CCc3scc(C)c3)=O)C(F)C2)ncc(Br)cc1[N+](=O)[O-] 79233,C12(CNC(=O)C(F)F)CCCC1CCN2C(c1ccc2nn[nH]c2n1)=O 79234,c1(C(=O)NC2CN(C(CCC(=O)NC)=O)CC(O)C2)cccn2cnnc12 79235,C#CC1(C(=O)NCC2CCN(C(C)C)C2)CN(C(=O)CC(C)=C=C)C1 79236,O=C1CC2(CCN(C(C3CN(C(=O)CCN4CCCCC4)CCS3)=O)CC2)C1 79237,CN1Cc2ccc(C(=O)NC(C)(CNC(=O)CC3CC3(C)C)CO)cc2C1 79238,N1(C(C2N(C)CC2)=O)CCC(C(=O)NCCC2C=CCC2)C1(C)C 79239,c12cnoc1C(=O)NCCN1CCC21.C1(CNC(=O)CCF)CC(CO)CO1 79240,N1(C(C2CCC(C)C2)=O)CC2(C=C(C(=O)O)CO2)C1 79241,C1(CC=C)(C(=O)NCC(c2ccccc2)F)CN(C(c2c[nH][nH]c2=N)=O)C1 79242,CC(C)(C(=O)NCCNC(C1SC2C=CC1C2)=O)C(N)=O 79243,c1(CCC(=O)NC2CN(C(C=C(C)Cl)=O)C2)c(C)nc(-c2ccccc2)nc1O 79244,N(C)(S(=O)(=O)N1CCC(C(=O)OC(N2CCNCC2)=O)CC1)C(C)C 79245,C(CC(C)C)(C(=O)NC1CC(C)CCC1O)NC(C(CC)COC)=O 79246,C(=O)(CCCC(c1nnnn1C(C)(C)C)NCCc1nncn1C)OCC 79247,CC1OCCC1NC(=O)NCC1(N(C)C)CC1c1ccccc1 79248,C(=O)(CCCN(C)N=O)N1CCC(C)C1CNC(=O)COCC1CCC1 79249,C1(CC)C(NC(=O)Cc2ccccc2O)CCCN1C(=O)Cc1cccs1 79250,c1(C(CNC(N2CCCC2CC(n2ccnn2)F)=O)OC)ccccc1Cl 79251,c1(C2C(C(N3C(CNC(C(CC)(C)O)=O)CCC3)=O)C2)c(Cl)cncc1Cl 79252,C1(NC(=O)COCC(C2CCN(C(=O)CSc3nccn3C)C2)C)CCOCC1 79253,C1(C(N2CC(N(C(c3c(OCC(=C)C)cccc3)=O)C)C2)=O)CC2C(C1)C2(C)C 79254,c1(CC)nc(=N)[nH]c(=NC2CC3CC(C2)N(C(C2CC(=O)N(C(C)C)C2)=O)C3)[nH]1 79255,C1(CNC(c2ccccc2OCc2cccs2)=O)CC2(C1)CC21CC1 79256,C12(COC)CC(NC(=O)C3=CCSC3)(CN1C(C1CC1C)=O)C2 79257,CC1=C(C(=O)NC2CC2NC(=O)CC(C)(C(F)F)N(C)C)Cn2nnnc2N1C 79258,c1(OC(C(=O)NCC(C(C)C)NC(c2cn(CC=C)nc2)=O)C)cccc(F)c1 79259,N1(CCC(=O)NCC2CC(CNC(CC(C)C)=O)C2)CCCCC1C 79260,C(=O)(CCC(C)(C)O)NC(C(C)C)CNC(C1CN(CC(F)(F)F)C1)=O 79261,N(C(=NCCCN(C)CCOc1cccc(Cl)c1)NC(C)CC)C(C=C)C 79262,c1(N2C3CN(C(c4ccc5nc[nH]c5c4)=O)CC2C3)ncnc2cccc(F)c12 79263,C(N=c1[nH]c(=NCC2CCCC3(CCC3)O2)[nH]c2c1SCC2)c1nccc(Cl)c1 79264,C=CCC(C(=O)NC(CCC)C(O)C(=O)NCC(C)(C)CC=C)C(C)C 79265,c1(CN(C(=O)C(=O)NCC(c2c[nH]c(=N)s2)N2CCCC2)C)cccnc1Cl 79266,C(N=c1ccnc(NCC(C)C(F)(F)F)[nH]1)C1(C=C)CCOCC1 79267,C1(NC(C(C)(C(=O)O)c2ccccc2)=O)CCOC2(CCC2)C1 79268,N1(C(c2c(C)cco2)=O)CCCC(C(C)NC(=O)C2=CCCC2)C1 79269,c1(C(=O)NC2CN(C(COCC)=O)C(C)C2)ccc([N+](=O)[O-])cc1 79270,N1(C(CC2(C)CCN(C(C3COCC3C(N)=O)=O)C2)=O)CCC2(CCC2)CC1 79271,C1(CNCC2CC(F)(CC)C2)CCN(C(=O)c2cc(O)ncn2)O1 79272,C1(C2CN(C(=O)C(C)(C)CF)C2)(NC(c2ccc(COC)o2)=O)CC1 79273,C1(C(=O)NC(C2CCN(C(c3ccncc3N)=O)CC2)C)Cc2ccncc2C1 79274,N1(C(CC2ON=C(C)C2)=O)CC(NC(c2c(N)cccc2Cl)=O)CC(F)C1 79275,CC1CN(C(c2cc(CN(C)C)on2)=O)CCC1NC(c1csc(C2CC2)n1)=O 79276,c1(NC(C2N(C(C3(C#N)CC3)=O)CC(O)C2)=O)ccc2c(c1)OC(F)(F)O2 79277,C1(OC)(CN)CCOCC1.C1(C2CN2)CC2CCC1C2 79278,CC(Cn1cccn1)C(=O)NCC1C(CNC(=O)C(F)CC2CCOC2)C1(F)F 79279,Cc1cn2cc(C(N3CCCC3CNC(C3(C)CCCN3C)=O)=O)cc(F)c2n1 79280,CC(CC(C)(F)F)C(=O)N(CCCCCNC(c1cc2n(n1)CC(F)C2)=O)C 79281,C1(C(N2CCCC(C(=O)NCC3N(CC)CCC3)C2)=O)CCCCC(C)O1 79282,S(=O)(=O)(c1[nH]c(=NCCC(F)F)ccc1Br)NCC1(C=C)CCOCC1 79283,C=C(C)CCC(=O)N1CCC(C(C)(C)NC(c2c[nH]cc2-c2ccc(C)s2)=O)C1 79284,c1(C(N(C(CC)CC)Cc2cccs2)=O)cc(CC)c[nH]1 79285,c1(C(=O)NC2CCCC(NC(c3c(CC)c[nH]c3)=O)C2)nncc2c1CCCC2 79286,N1(c2nc(CC)on2)CCC2(CC1)CC2C(N1CCC2OCC2C1)=O 79287,c1(OC)cc(CO)ccc1C(=O)NC1C2CC1CN(C(=O)C(C)(O)C1CCC1)C2 79288,N1(C(C=CCC)=O)CCCCC2(C1)CN(C(=O)Cn1ccnc1C(C)C)C2 79289,c1(C(=O)OC)cc(C(=O)N(C)CCNC(=O)C(C2CCOC2)SC)c(C)o1 79290,Cc1cc(=O)n(C)cc1C(=O)NCC1(F)CCCN(C(=O)C=C2CCC(C)C2)C1 79291,N1(C(Cc2c(OC)nccc2)=O)CCCC(C)(NC(=O)CC2CCCN2C)C1 79292,N1(C(C2C(=O)OCC2)=O)CCC2(CCCCN(C(c3ccc(O)nc3)=O)C2)C1 79293,c1(C(=O)NCCCC2N(C(C=NOC)=O)CCC2)ccc(C2CC2)nc1 79294,C1(CNC(c2nn[nH]c2Cl)=O)CCCCN1CC1(C(N)=O)CCCC1 79295,C1(C(=O)NC(CCCNC(CCCCN(C(C)=O)C)=O)C)CCC2CC2CC1 79296,c1(N2CCCCC2)nc2cc[nH]c2c(=NCC2CCCO2)[nH]1.N(C)CC 79297,N1(C(C(C=CCCC)O)=O)C2CCCC1CC(NC(=O)C=C1CCC(C)CC1)C2 79298,c1(C(=O)OC)c(NCC2CC(C3CC3)C2)cc(C(=O)OC)cc1Br 79299,C(C1CN(C(=O)COC2(C)CCCC2)Cc2ccccc21)NC(C(C)(C)CF)=O 79300,c1(NC(C2C3CN(C(c4cc(CC)c(C)s4)=O)CC32)=O)ccc(CO)cc1OC 79301,C1(CC=C)(C(N2CC(OCCNC(=O)CO)C2)=O)CC=CC1 79302,Cc1ccnc2sc(C(=O)NCC(C)NC(c3occ4c3CCC4)=O)c(C)c12 79303,C(=O)(C(O)C(C)(C)CC)NC1C(NC(c2cc(CC)[nH]n2)=O)C1 79304,CCC(O)C(C)(C)C(=O)NC1CC2(CCN(C(c3coc(SC)c3)=O)C2)C1 79305,Cc1cccc(C(C2CCOCC2)NC(N2CCC(C)(c3ccc(C)cc3)C2)=O)n1 79306,c1(C(N2CC3C(CNC(C4C(C)C4)=O)C3C2)=O)cc2ccccc2s1 79307,C(=O)(C(F)(F)CCC1CC1)N1CCC(CCCNC(C(N)=O)=O)CC1 79308,c1(NC(C(C)C)CNC(C2CCCNS2(=O)=O)=O)ncnn2cccc12 79309,Cn1cc([N+](=O)[O-])cc1C(=O)NC1COCCN(C(=O)CSC2CCOC2=O)C1 79310,C1(C(=O)NC2(CNC(C(C)n3ccnn3)=O)CCOC2)C2CC3C(C2=O)C13 79311,C(=O)(CCCCC(=O)Nc1nccn1C)NCCN(c1ccccc1)CC 79312,Cc1ccc2c(C(=O)NC(C3(O)CN(C(c4scc(C)c4Cl)=O)C3)C)n[nH]c2c1 79313,CC(CC(=O)N1OC2CCC1C2)NC(=O)Cn1cc(Cl)cn1 79314,c1(C(=O)NC2C(C(C)C)N(C(=O)CCC(C)C#N)CC2)cccc2ccncc12 79315,C#CCC(O)C(=O)NC(c1cn(C)nn1)C(=O)N(C)Cc1conc1CC 79316,c1(OC(C(N2CCC(NC(C=CSC)=O)C2)=O)C)ccc([N+](=O)[O-])cc1 79317,C(=O)(C1CCCc2nc[nH]c21)NCC1CC(OC)CN1C(C1CCC1(F)F)=O 79318,Cc1nn2cccnc2c1C(=O)NCCCCNC(=O)COC1CCCCC1C 79319,Cn1ncc(C(=O)NCC2(NC(C3CCC(F)CC3)=O)CCC2)c1Cl 79320,C(=O)(C(C)C(F)(F)F)N1CCC(NC(c2cc(OC)c(Cl)s2)=O)C1 79321,N1(C(c2c(C)cnn2C)=O)CCC(NC(C2CCCN2C(C)C)=O)C(F)C1 79322,c1(CC)cc(C(=O)NCC(C2CC2)NC(C2CCC(C(=O)OCC)O2)=O)ccn1 79323,Cc1cncc(CC(N2CC(NC(=O)Cn3nnc(C4CC4)n3)C2)=O)c1 79324,C1(C(=O)NCC)Cc2c([nH]c3ccccc23)CN1Cc1c(F)ccc(C)c1Cl 79325,Cc1cc(CCC(=O)NC(C(=O)NCC2CC2(Cl)Cl)C2CC2)n[nH]1 79326,S(=O)(=O)(c1cc(C(N2CCCN(C(=O)C=CCO)C(C)C2)=O)cc(C)c1C)NC 79327,CCCCC(O)C(=O)NCC(CC(F)(F)F)NC(c1cc(Cl)ccc1C(F)F)=O 79328,C1(C(=O)NCC2N(C(C(C)Cc3cnc[nH]3)=O)CC(O)C2)CC(C)(C)CCO1 79329,c1(C(=O)NC2CCC(NC(C3CCC(C)C3)=O)CC2)cnn2c1N(C)CC2 79330,C12(CNC(C)=O)CN(C(=O)Cc3cc[nH]c3)CC1CS(=O)(=O)C2 79331,C(=O)(CC(O)CCC)NCCC1N(C(C2N(CC#C)CCC2)=O)CCCC1 79332,c1(C(=O)NC2CC(C)N(C(c3cc4oc(Cl)cc4[nH]3)=O)C2)cn2ccccc2n1 79333,C(=O)(CCC(=O)C(C)(C)C)N1CC(C(=O)NCCc2onc(C)n2)OC(C)C1 79334,C(=O)(C(CCC1CC1)NC(=O)CCC=C(C)C)NC(CC)C1CCC1 79335,c1(OC)ccnc2ccccc12.c12cc(OC)ncc1CO2 79336,N1(C(c2cc(C)n(C)c2)=O)CC(NC(c2conc2C(C)(C)C)=O)CCC1C 79337,C1(CC)CN(C(C2CCOCC2(C)C)=O)CCN1C(=O)C=CSc1ccccc1 79338,C(=O)(C1=CC2C=CC(C1)C2)Nc1c(C)cccc1.C12CCCC(C1)NC2 79339,C=CC1CN(C(c2cn(C)ccc2=O)=O)CC1NC(c1conc1C(C)C)=O 79340,c1(C(=O)NCC2C(Cn3cc(CC(C)O)nn3)C2(F)F)[nH]c(=N)ccc1Br 79341,C1(C(=O)NC2CC(NC(c3ccccc3C(C)C)=O)C2)(OC)CCCC(C)C1 79342,N1(C(CSC)=O)CC2CC(C1)N(C(=O)CNc1ccccc1[N+](=O)[O-])C2 79343,C1(NC(c2c(C)ccs2)=O)C2CC3CN(C(c4cnc5sc(C)cn45)=O)C1C3C2 79344,N1(C(CC2CC(CC)OCC2)=O)CCCN(C(c2cnsn2)=O)CCC1 79345,C(C1c2ccsc2CCN1C(=O)C(O)CN1CCCC1)NC(CCC=C=C)=O 79346,c1(OC)ccc(S(=O)(=O)NC(c2csc(C(C)C)n2)C(=O)O)cc1C(N)=O 79347,Cc1cc(C(=O)NC23CCC(C(N4CCNC(=O)C4C)=O)(CC2)C3)nc(Cl)c1 79348,C1(CN(C(CSCC(C)C)=O)C)CN(C(=O)CC2COCCN2C)CCO1 79349,N1(C(CC)=O)CCC(C(=O)N(C)CC2CN(C(C3(CCF)CCC3)=O)C2)C1 79350,CC1(CNC(c2n[nH]c(C3CC3)n2)=O)CCCN1C(=O)CCC1CCC(=O)N1 79351,Cn1nnc2cc(C(=O)NC3(C)CC(NC(c4c[nH]c(=N)s4)=O)C3)ccc12 79352,C1(NC(Cc2ccc(C)cc2)=O)CCN(C(=O)C=CC(=O)NC2CC2)CC1CO 79353,C(=O)(CC1CCc2ccccc21)NCC(COC)NC(=O)CC12CCC(CC1)C2 79354,C1(C(=O)NC2C(NC(c3n(C)nc(C4CC4)c3)=O)CC2)CN2CCN1CC2.C1(C)CC1 79355,C(C(=O)NCCNC(=O)Cc1ccnc(Br)c1)(C(C)(C)C)N(C)C 79356,c1(NC(C=CC(C)NC(=O)C(C)(Cl)Cl)=O)ccc2ccoc2c1 79357,CCC(C#N)(CC)C(=O)NCn1cc(C(=O)NCC2CC(C(C)C)C2)nn1 79358,c1(C(=O)NCC=CCNC(c2n(CCSC)ccn2)=O)n[nH]c(C)c1[N+](=O)[O-] 79359,c1(N2CC(C=C)OCC2)nc2ccc(S(=O)(=O)N3CCSC(C)(C)CC3)cc2s1 79360,C1(CNC(C2(CC)CCCC2)=O)CCCCC1C(=O)NCc1ccc[n+]([O-])c1 79361,N1(C(c2cn(C)c(=O)cc2)=O)C2CCCC1CC(CNC(C1(C)CC1(F)F)=O)C2 79362,c1(C(N2CCN(C(COC)=O)CC(C)(C)C2)=O)cc2c(O)ccc(F)c2[nH]1 79363,c1(C(=O)NC(C)CN2CCCC2)c(I)ccc(Cl)c1Cl 79364,c1(-c2ccc(OC)cc2)n[nH]c(=NC2CCC2C)c2ccccc12 79365,C1(C(=O)NCC2(F)CCN(C(C=C(C)Cl)=O)CC2)CC(C)(C)OC(C)(C)C1 79366,C1(C(N2CCC(N(C(=O)Cn3nnc(C4CC4)n3)C)CC2)=O)OC2CCC1CC2 79367,c1(CC)ccc(C(C(=O)NC(C)(C)CC)N(C)CC2CC=CCC2)nc1 79368,N(C(=NCc1ccc(OCF)cc1)NCC12CC(CCO1)C2)C(c1cccs1)C 79369,c1(C(=O)NC(CCOC)CNC(=O)C(=O)NCC(F)F)ccnc(C)c1N 79370,CCC1(C)CNC(=O)CO1.C1(NC(C2CSC2)=O)(OC)CCOC1 79371,C1(NC(C(C)NC(CC)=O)=O)CCC(N(C)C(c2cc(C)c(C)[nH]2)=O)CC1 79372,N1(C(COCC=C)=O)CC(C)CCC1C(=O)Nc1ccc(OC)cc1C(F)(F)F 79373,Cc1cc(C(=O)N(C)CC2CN(C(=O)CC3CCC(C4CC4)O3)C2)nn1CCO 79374,C1(C(=O)Nc2cc(O)n[nH]2)CCCC12CCN(Cc1cscn1)C2 79375,Cc1cc(=NC(CCO)c2c(C)nn(C)c2C)[nH]c(=NCc2ccc(Cl)cc2)[nH]1 79376,C1(c2ccccc2)(NC(C(CC)NC(C)=O)=O)CCN(C(c2nocc2C)=O)C1 79377,c1(C(=O)NC(CNC(c2c(SC)ccs2)=O)C2CCC2)ccc(F)c(C)c1C 79378,C=CC(C)(CC)C(=O)NC(CC(=O)Nc1cnc(N(C)C)nc1)C1CC1 79379,n1(CC)ncc(Cl)c1C(=O)NCC1(COC)CN(C(C2CC(=O)N2)=O)C1 79380,C1(NC(CCOCC)=O)CCCCC1NC(c1ccc(C(C)=O)nn1)=O 79381,Cc1c(C(=O)OCC(=O)NC2CCN(Cc3ccccc3)C2)cccc1O 79382,c1(C(=O)NC(CNC(c2c(CC)[nH]nc2Cl)=O)CCOC)c([N+](=O)[O-])cnn1CC 79383,n1(CC(=O)NCC(N(C(C(CSC)C)=O)C)C2CC2)nc(C(F)F)cc1C(F)F 79384,c1(C(=O)NC2C(C)CN(C(c3ccc(C(N)=O)s3)=O)C2)cccc(S(N)(=O)=O)c1 79385,c1(CC(=O)NCC(n2cc(C3(CO)CCN(C)CC3)nn2)C)c(F)cncc1Cl 79386,c1(C(N2C(C(C)C)C(NC(c3ccnnc3S)=O)CC2)=O)cc(=O)cc(Cl)[nH]1 79387,C=C(C)CCCC(=O)N(C)CC1CCCN1C(=O)C(N1CCOCC1)C 79388,N1(C(CSCCC)=O)CC(CO)C2(C1)CN(C(=O)C(O)CN1CCOCC1)C2 79389,N1(c2cc(NCc3cn(CC(C)C)nn3)nc(C)n2)CC2CCCCC2(CO)C1 79390,c1(C(=O)NC2CCC(CCNC(C3(CC(C)C)CC3)=O)C2)cnn2ccsc12 79391,Cc1cc(C(N2CCC(CNC(=O)CN3CCCC3=O)C(C)C2)=O)c(N)c(Cl)c1 79392,c1(NC(C(=O)NC(c2nc(C)cs2)C)=O)cccc(N)c1.CCCCOC 79393,C(CC(O)C(=O)NCC(O)CCNC(=O)CCC(C)OC)SC 79394,Cc1c(C(=O)N(CC(=O)NOCCF)C2CC(C#N)C2)cco1 79395,C(=O)(CS(=O)C(F)(F)F)NCCC(C(C)C)NC(c1cnc2ccoc2c1)=O 79396,c1(C(C)CC(=O)NCC(O)CN(C)C(c2ncn(C)n2)=O)ccc(Br)cc1 79397,N1(C(c2cccc(OC)c2)=O)CCN(C(C2CC(C)(F)C2)=O)C2COCC12 79398,N1(C(C(C=C)(F)F)=O)CCN(CC)C(=O)C1.c12cc(on1)C(=O)NC2 79399,C12(CNC(CNC(=O)OCC=C)=O)CCC1CN(C(=O)CC1CC(F)(F)C1)C2 79400,c1(NC(=O)NCC2(O)CCOC2)ccccc1I 79401,N1(C(c2cnc(N3CCC(CC4CC4)CC3)cn2)=O)CCC(C2CCOC2)CC1 79402,N1(C(c2c[nH]c(=NC)s2)=O)C2CCC1CC(CNC(=O)Cc1csc(C)c1)C2 79403,c1(CC(=O)NC(CC)CNC(=O)C(C)n2cnnn2)ccc(C)c(C)c1 79404,N1(C(CSC(C)=O)=O)CCCC1COC(F)(F)F 79405,c1(C(CCO)NC(CC2(NC(=O)Cn3cccc3)C(C)C2)=O)ccc(Cl)cc1 79406,C1(C(=O)NCCC(=C)CNC(=O)CC2=CCOCC2)C2CC3CC(C2)CC1C3 79407,C(=O)(C(F)CCC(C)(C)C)NC(C)C(CO)NC(=O)C1=NOC2(CCC2)C1 79408,C(CCCN=C(NCC1(Cl)CCCCC1)NC1CCCC1)C1CCC1 79409,c1(CC)nc(C)[nH]c1C(N1CCOC(C(C)NC(=O)CCc2cscn2)C1)=O 79410,C1(C(C(=O)NC(CNC(c2c(OCC)ccs2)=O)(C)C)C)CCC(C)(O)CC1 79411,N1(C(C2CN(C)C2)=O)CC(C(C)(C)O)(CNC(c2cnoc2C2CCC2)=O)C1 79412,c1(CN2CCC(NC(C(c3ccccc3)SC)=O)C2)c(F)ccc(O)c1F 79413,Cc1nc(Br)cnc1NC(C1CCCN(C(c2cnnn2C)=O)CC1)=O 79414,C1(NC(C=C(C)C(F)F)=O)CCCC(CNC(=O)Cc2c(C)n[nH]c2C)C1 79415,C[Si]1(C)CCCCN(CC(N2CCC(CCS(N)(=O)=O)CC2)=O)C1 79416,N1(C(c2c(C)nc[nH]2)=O)CCC(F)(F)C(CNC(=O)Cc2ccnc(Br)c2)C1 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79641,C(CCF)(C(=O)NCC(O)CCC1CC1)NC(CC1ON=C(C)C1)=O 79642,c1(OC)cc(N)c(C(N2CC(NC(c3cnn(C)n3)=O)C2)=O)c(F)c1 79643,c1(NC(C)C)ccc(C(=O)NCC2(NC(C3C(C)CC3C)=O)CCC2)cc1 79644,c1(C(=O)NC(C2CCCC2)CNC(CCSCC(N)=O)=O)cc2cccnc2[nH]1 79645,C1(C(=O)NCCN(C(=O)CCCc2ccccn2)C2CC2)CCCC2(CC2)C1 79646,C(c1ccc(C(N(CC(C)C)CC(=O)Nc2cc(Cl)sc2Cl)=O)o1)=CCO 79647,C1(NC(c2c(OC)nsc2)=O)CCOC2(CCN(C(=O)C(C)C(F)(F)F)CC2)C1 79648,c1(OC)cc[n+]([O-])c(C(N2CCC(NC(c3ncc(C)cc3F)=O)CC2C)=O)c1 79649,c1(CNC(C2CCSC2)=O)ccc2c(c1)CN(C(C1CCCC(CF)C1)=O)C2 79650,C=CCC(C(=O)N(C1(NC(c2ccc(-n3cccn3)nc2)=O)CC1)C)C(C)C 79651,C(=O)(CC(C)(C(F)(F)F)NC(c1cc(N)cc(I)c1)=O)N(C)C 79652,c1(CC(C(=O)NC(c2ccc(F)cc2)CC)N)c[nH]c2cc(Cl)ccc12 79653,O=S(=O)(c1ccc(Br)c(Cl)c1)N1CC2CN(Cc3cnc4ccccn34)C2C1 79654,c1(C(c2n(C)nnn2)NCC2CC(C)(C)C2)cncc(C(C)(F)F)c1 79655,c1(C(=O)NCC2C(N(C)C)CN(C(C3N(CC)CC3)=O)C2)c(OC)cccc1O 79656,N1(C(C=CC=CCC)=O)CC(CNC(c2cc3ccsc3s2)=O)C2(CCC2)C1 79657,C(C(CC(=O)N(C1CC(F)(F)C1)C)NC(C1CCC(=O)CC1)=O)OC 79658,N(C1CN(C(=O)CC2CC3CC3C2)CCc2ccccc21)C(C=CC)=O 79659,c1(OC)ccc(CC2CCN(C(c3ccccc3)=O)CC2)cc1C(F)(F)F 79660,c1(C(=O)NCCCN(C(C(CC)SC)=O)CC)cccc2ncoc12 79661,C12(NC(C(CC)OCC)=O)CCCC1N(C(c1cc(C(C)C)ccc1C)=O)CC2 79662,C1(CC(=O)NCCC2CC(C(=O)NC(C(C)C)C3CC3)C2)COCC1O 79663,c1(N2CCC(C(=O)OC)CC23CC3)cn(C)c(=O)n(C)c1=O 79664,c1(C(N(CCNC(CCN(CCCCC)C)=O)C(C)C)=O)nccn1C 79665,C1(COC)(NC(=O)C=CCN2CCOCC2)CCN(C(=O)CS(N)(=O)=O)C1 79666,C1(OC)CC(CNC(C2(CNC(=O)C(F)(F)c3ncc[nH]3)CC2)=O)C(O)C1 79667,C1(CNC(=O)CC2CCC3CC23)(NC(=O)CSc2cccc(O)c2)CCOCC1 79668,CCC(C)C(C(=O)N1CC(CO)C1(C)C)NC(=O)CCc1cncs1 79669,c1(C(N2CC(C(C(=O)N(CC(O)CO)CC)O)C2)=O)cnc(C2CC2)o1 79670,C1(NC(C2CNC(=O)O2)=O)C2CC1N(C(C13CCCCC1C3)=O)C2 79671,C(=O)(C(C)CC(C)(C)C)N1C2CC(NC(C(C(CC)O)C)=O)C2CC1 79672,c1(N(C(=O)NCC(c2ccc(OC)cc2)OC)C)ccc(F)cc1Cl 79673,N1(C(C(CCCC)NC(c2ccc(C#C)cc2)=O)=O)CC(C)(C)CCC1C 79674,C1(C(=O)NCCN(C(c2cn(CC(F)(F)F)nn2)=O)CC)CCC2(CCC2)O1 79675,C12(C(=O)NCC3N(C(CC4C(CC)C4)=O)CC(F)C3)CCCN(CCC1)C2 79676,C1(NC(C2(CCCC)CCCC2)=O)CCCCN(C(c2cccn(C)c2=O)=O)C1 79677,Cc1ccncc1C(C)NC(c1nc(CNC(c2cc(C)c(C)[nH]2)=O)oc1C)=O 79678,N1(C(=O)NCCOCCCC)CCC(CO)C(F)(F)CC1 79679,C(=O)(C1CCCc2sccc21)N1C2C(NC(C3C(CCC)CCC3)=O)C(C2)C1 79680,C(=O)(C1=Cc2ccccc2C1)NCCC(C)CCC(=O)NCCCCCCSC 79681,c1(OC)ccc(Cl)c2[nH]c(C(=O)NC3(CNC(=O)C(C)NC(C)=O)CCC3)cc12 79682,Cc1n[nH]cc1C(=O)NC(C)CCN(C(=O)CC1(O)CCOC1)C 79683,C1(C(N(C2CCN(C(C(CN(C)C)(C)C)=O)C2)C)=O)CC2CCC(C1)N2C 79684,c1(CNC(C2CC2C(N2C(C(N)=O)CCCC2)=O)=O)cc(F)ccc1[N+](=O)[O-] 79685,c1(C(=O)NC(CNC(c2c(Cl)ccc(OC)n2)=O)CO)cccc2c1CCO2 79686,c1(-c2cc(C(=O)Nc3c(SC(C)(C)C)cccc3)no2)ccc(Br)cc1[N+](=O)[O-] 79687,C1(NC(C(CC)n2cccn2)=O)CCC(O)CN(C(=O)C2=CCCC2)C1 79688,C1(S(N)(=O)=O)(C(=O)NCCCCCNC(c2c(SC)cnn2C)=O)CCC1 79689,C(=O)(C(C)(CSC)NC(=O)CC1CCC(O)C1)N(CCCCC=C)C 79690,Cc1cc(C(=O)NC(C)(C)CCNC(=O)C(C)CS(C)(=O)=O)c2occc2c1 79691,c1(C(N2CC(NC(CCc3cc(OC)no3)=O)(CO)C2)=O)c(C)ncn1O 79692,c1(CC)nc(C(=O)NC2CCC(CC(=O)N(C)Cc3cc(=O)cc[nH]3)C2)c(C)o1 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79745,N1(C(CCN(CC=C)C(c2ccn(CC)c2C)=O)=O)CCOC2COCC12 79746,Cc1ncc(Cl)c(-c2nc(CP(C)(C)=O)no2)n1 79747,C1(C(=O)NCCN(C(=O)CC2CC(=O)C2)CC)CC(n2cnnc2)C1 79748,N1(C(C(=O)NC(=O)CNC(c2coc(O)n2)=O)=O)CCN(C(=O)C2CC2)CC1 79749,c1(C(=O)OC)cccc2c1cnn2COc1cccc(NC(C2CCCC2)=O)c1 79750,N1(C(C(CCOC)C)=O)CCC(NC(C2CCN2C)=O)C12CC2 79751,N1(C(C2(C)CSC2)=O)CCC(CNC(C2(C)CCC(=O)NC2)=O)C(F)(F)C1 79752,C1(C(=O)NC2(C(COC)O)CC2)CCN(C(=O)c2[nH]nnc2C)O1 79753,C12(NC(COCC)=O)CC(C)(C1)OC21CN(C(=O)Nc2cc(C)c(C)cc2C)C1 79754,C1(CNC(CCCCC#C)=O)CCC2(CCN(C(=O)CNC(=O)OCC)C2)C1 79755,C1(C)(CC(=O)NCC(COC)C)CCN1C(C1CC(C#N)C1)=O 79756,CCCC(C(=O)NCc1cc(C2CC2)on1)NC(c1cscc1OC)=O 79757,C1(OC)CCN(C(=O)C(c2cscn2)OCCNC(C2CC(N(C)C)C2)=O)CC1 79758,c1(CNC(C=CC2N(C(C(CC)CN(C)C)=O)CCC2)=O)ccc(F)cc1F 79759,C1(NC(C(CCSC)O)=O)CCOC12CCN(C(=O)CN(CC(C)(C)C)C)CC2 79760,Cn1cccc1-c1cn(CCCC(=O)NCC(O)Cn2cccn2)nn1 79761,Cc1nnc2cc(C(=O)NCC=CCNC(C3(C4CCCC4)CC3)=O)ncn12.C 79762,N1(C(C(CC)O)=O)CCC(n2cc(COc3ncccn3)nn2)CC1 79763,CCC(F)(F)C(C)(C)C(=O)N1CC2CCC1CN(C(c1[nH]cnc1C)=O)C2 79764,N1(C(COC(C)=O)=O)CCC2C1CCCN2C(=O)C=Cc1ccccc1[N+](=O)[O-] 79765,C12(C(=O)OC)COCC1CN(S(=O)(=O)c1csc(C(C)(C)C)n1)C2 79766,c1(C(C(=O)Nc2ccccc2)N(C(C(=O)NCC)CC)C)cc(C)nn1CC 79767,c1(C(=O)NC(CCOC)CNC(=O)CCC(C)N(C)C)cccc(C)c1O 79768,c1(C(N2CC(CNC(CC3(OC)CC3)=O)C3C2C3)=O)cc(C)nc(C)c1 79769,CON(C)CCCNC(C1C=CCCN1C(=O)CC1(C)OCCO1)=O 79770,C(CCCCC(=O)NC(C)C(C(C)C)NC(C1CCSCC1)=O)OC 79771,O=C(CC1COCc2ccccc21)NCCC1CCN(C(=O)Cn2cnnc2)C1 79772,C(CC(C)C)(C(=O)NC1CC(CNC(=O)Cc2c(C)noc2Cl)C1)NC(C)=O 79773,c1(C(=O)NCC2(COC)CN(C(C3C(C)(CC)C3)=O)C2)c(C)nc(C)n1O 79774,c1(C(=O)NCC2C(NC(C(n3cc(Cl)cn3)C)=O)CC2)c[nH]cc1C(F)(F)F 79775,C1(C)(CNC(C(c2ccc(C)o2)C)=O)CCCN(C(c2cn(C(C)C)nn2)=O)C1 79776,C1(C(=O)NCC2(CNC(C3(C#N)CCCO3)=O)CC2)CCC=CCCC1 79777,C1(C(c2ccc(-c3ccco3)nn2)Nc2n(CCC)nnn2)C2CCCOC12 79778,C1(C(=O)NCC(CC)(C)NC(=O)CCOCCCOC)CCCC(CF)C1 79779,C1(CC(=O)NCc2cccc(Cl)c2)CCCN(C(C2CC(F)(F)C2)=O)C1 79780,C=C(C)CCCN=c1c(Br)ccc(NC(=O)CNC(=O)C(C)(C)C)[nH]1 79781,C1(C(=O)NCC2CCCCN2c2ccnc(CO)n2)CCC(=C(F)F)CC1 79782,C1(NC(c2c(CNC(C3C(C)(C)C3)=O)occ2)=O)CC2CC1C(O)C2O 79783,C1(CNC(C(CCCC)O)=O)CCC12CCN(C(c1cnc(C)[nH]1)=O)CC2 79784,N1(C(C=CC2N(C)CCC2)=O)CCN(C(=O)CCc2cnn[nH]2)CC1CO 79785,C1(CN(C(=O)CNC(c2ncc[nH]2)=O)CC)CC1C1CC1 79786,C1(NC(CC(C)c2ccco2)=O)CN(C(c2cn(C)nc2O)=O)CCC12CCC2 79787,CC1CN(C(c2cn(C)c(=O)n2C)=O)CCC1NC(C1(CO)CCCC1)=O 79788,C1(CC=C)(C(=O)NCCC2CN(C(C3CC3c3ccoc3)=O)C2)CCC1 79789,CCC(O)C(C)C(=O)N1CC(CNC(c2cccc(Cl)c2F)=O)CC1(C)C 79790,C1(NC(C(CC2CCC2)OC)=O)CC2CC1CC2C(=O)NC1CC1C1CCC1 79791,CC(O)C(C(=O)NCCC1CCCN(C(c2csc(Cl)n2)=O)C1)N(C)C 79792,Cc1ccc2c(=NC(C)c3scnc3C)[nH]c(N(C)CCn3ccnc3)nc2c1 79793,c1(CCC)ncc(C(=O)NC2CCC(NC(=O)CSc3nncn3C(C)C)C2)s1 79794,C(=O)(C#CC1CCOC1)N1CCCC(C(=O)NCc2nc(C)c(C)s2)C1 79795,C12(NC(COC)=O)CCCCCC1N(C(=O)CNC(=O)CC1CCCCC1)CC2 79796,c1(NC(C(C(C)C)NC(=O)Cc2ccns2)=O)ccc(F)cc1CO 79797,c1(CN(C(c2c(N)ccc(CC)c2)=O)C(C)C)ccc2c(C)[nH]nc2c1 79798,C1(C(N(C)CC2(O)CCN(C(Cn3c(C)csc3=O)=O)C2)=O)C2CCC(F)(F)C12 79799,c1(CNC(=O)NC2CC(C(N)=O)OCC2)cc(O)cc(Br)c1 79800,CC1COc2ccc(C(=O)NC3CCC3NC(=O)CCCc3ccsc3)cc21 79801,c1(CNCC2(COC)CCC2)cc(C(=O)O)c(NC(=O)C=CC2CC2)cn1 79802,C1(CCC=C)(C(=O)NCC(C)OC(F)F)CN(C(=O)C(C)C2CCCC2)C1 79803,C1(CC(N2CC(O)(CN(C(=O)C(C)(C)C3CCOC3)C)C2)=O)OC(C)(C)OC1=O 79804,C(=O)(C(C)C(O)CC(C)C)NCC(C)(C)OCC(=O)NCC1CC(OC)C1(C)C 79805,C(=O)(C(CC(C)C)CC(C)C)NC1CC2CN(C(CC(C)SC)=O)C1C2 79806,C1(C(C)C)CN(C(C2C3COCC23)=O)CCN1C(=O)C(C1CCC(=O)N1)C 79807,C1(CC=C)(NC(=O)CC2CCCC2C)CCCN(C(c2cc(O)ccc2O)=O)C1 79808,n1(CC)ccc(C(=O)NCCN(C2CCCCC2)C(=O)CN(C2CCSC2)C)n1 79809,C1(CCC)COCCN1C(=O)C(C)C(C)NC(=O)C=C(C)C 79810,C1(NC(C=C(CCC)C)=O)CN(C(=O)CC2CN3CCC2CC3)CC12CCCC2 79811,C1(CNC(CC(C)C)=O)CN(C(C2CCN(C)CC2)=O)CC(C(F)(F)F)O1 79812,C1(C(=O)NC(C(=O)N(C)C)CO)COC(=O)N1C.C1(=O)C(C)(C)n2cc(nn2)CN1 79813,C1(NC(C2(F)CCN(C(=O)C3=NOCC3)C2)=O)CC12CCOCC2 79814,N1(C(C(C)n2cncn2)=O)CCCC12CCN(C(C1(C#N)CC1)=O)C2 79815,C1(NC(Cc2ccc(C)nc2)=O)CC2CC(C1)N(C(=O)CCc1ccco1)C2 79816,c1(C(=O)N(C2(C=C)CC2)C2CC2)noc2c1CCC2 79817,c1(NCC(C2CC2)NC(=O)CCc2cccs2)nccc(-c2cncs2)n1 79818,N1(C(CCCCCC)=O)CCN(C(=O)CCc2cccc(C#N)c2)C(C)CC1C 79819,Cc1[nH]nc2cc(NC(=O)C(C(C)C)n3ccnc3)ccc12.C12(CC1)CC(=O)N2 79820,C1(CCNC(C2CCC(CC)O2)=O)COCCN1C(c1cccc(SC)c1)=O 79821,c1(C(=O)NC(C(CCC)O)CO)cc2[nH]nnc2cc1OC 79822,C1(C(=O)NC(C#C)C2CCC2)CC(=O)CN1C(c1cc(OC)nn1C)=O 79823,N1(C(CC(=O)NCC)=O)CCCC(F)(CNC(c2cc(C(=O)OC)n[nH]2)=O)C1 79824,CCCCCCC(O)CCC(=O)NC1(C)CCCN(C(C2OCCC2(C)C)=O)C1 79825,N1(C(CCCNC(=O)OC)=O)CC2CN(C(C3CCC3OC)=O)CC(C1)O2 79826,C(=O)(C1SCc2cccnc21)NC1CN(C(c2c(C)n(C)cc2)=O)CC1O 79827,C1(N(CC)CC)CCN(CC(c2ccccc2Cl)OC(=O)C(C)C2CCC2)CC1 79828,CN=c1ccc(C(=O)N(C(C)CNC(c2csc(C3CCCO3)n2)=O)C)c[nH]1 79829,C(=O)(C(C)S(N)(=O)=O)NCCOC(CNC(CSC)=O)(C)C 79830,N1(C(C(CCO)N(C)C)=O)CC(C2CCN(C(C3CC3(C)C)=O)CC2)C1 79831,N(C(=NCc1cc(C)on1)N(C)Cc1cccc(Cl)c1)CC(=O)NC(C)C 79832,CC1(NC(c2cc(-c3ccoc3)[nH]n2)=O)CCCN(C(=O)CC2CCC(=O)N2)C1 79833,CCS(=O)(=O)CC(=O)NCC1C(C(=O)Nc2ccc(O)c(C(N)=O)c2)C1(C)C 79834,Cc1cnc(NCCC2CCC(NC(=O)C(C)C(C)(C)C)C2)nc1S(C)(=O)=O 79835,c1(C(=O)NC2CN(Cc3ccc(Br)nc3)CC2F)ccnc(Cl)c1Cl 79836,c1(C(=O)NCC(CC=C)NC(=O)Cc2cc(C)cc(C)c2)cc(OC)ccc1C 79837,C(=O)(C1=CCC(C)(C)CC1)NCC1CCN(C(c2ccc(C#C)cn2)=O)CC1C 79838,c1(C(=O)NCCC(C)NC(CCc2c(C)cccc2)=O)c(C)cc(O)nc1C 79839,Cc1cc(F)ccc1NC(C1(NC(c2csc(-c3ccccc3)n2)=O)CC1)=O 79840,N1(C(C(C2CCCC2)NC(CC)=O)=O)CCC(CO)C(C)C1.C1C(=O)N1 79841,C1(NC(C=CC(=O)OCC)=O)CCCC1(C)CN(C(=O)CCCN(C)C(C)C)C 79842,C1(C(N(C)CC2CN(C(c3cc(Cl)ccc3F)=O)C2)=O)Cc2ccccc2N1 79843,c1(C(N2C(C(=O)NC3C(CC=C)COC3)C3CC3C2)=O)ccc(C#N)cn1 79844,C12(CNC(Cc3cccc(C)c3F)=O)CCCC(CN1C(=O)C(F)F)C2 79845,C(=O)(C(F)CCC(C)C)N1CCN(C(C2C(CC)CCO2)=O)C(CC)C1 79846,C=CC1(C(=O)NC(C2CCCCC2)CNC(=O)Cc2n[nH]c(C)n2)CCCC1 79847,C1(CNC(c2cc(C)nn2C2CC2)=O)CCCN(C(C2CC3(CC3)CO2)=O)CC1 79848,c1(C(N(CCN(C(C(C(=O)OC)C)=O)C)C(C)C)=O)ccc2nccn2n1 79849,c1(CCCOCCOC)c[nH]c2ccc(C(N3CC(C)C(C)(CO)C3)=O)cc12 79850,C(=O)(C(C(C)C)n1cncn1)NC1C(NC(CC(OCC)OCC)=O)CC1 79851,N(C1CCCc2c(F)cc(F)cc21)CCCCc1c(C)ccc(Br)c1 79852,c1(C(=O)NC2C(C)CN(C(C3CCO3)=O)C2)cc2cccc(Br)c2[nH]1 79853,C1(C)(CC)C=C(C(=O)N2CCN(C3CCCN(C(=O)C(O)C(C)(C)C)C3)CC2)C1 79854,C1(OC)CC(CF)N(CC(=O)NCC(c2ccccc2)Oc2ccccn2)C1 79855,Cc1ncncc1C(=O)NC1CN(C(c2occc2CN(C)C)=O)CC1F 79856,C(CC1=CCN(C(C2CC23CCCC3)=O)CC1)NC(C(C=C=C)C)=O 79857,N1(C(C(C)CC(F)F)=O)C2CCC1CN(C(=O)C(C)(C)C1CCCO1)C2 79858,c1(CNC(CC2OCC(CN)C2)=O)ccc2cc(C(=O)O)[nH]c2c1 79859,c1(C(=O)NCC2N(C(C3CCCC(OC)C3)=O)CCC2C)cccn(C)c1=O 79860,CCC(CC)C(C(=O)N1CCCC1C(C)NC(c1nncn1CC)=O)OC 79861,C1(NC(c2ccc(CCC)[nH]2)=O)CCCC(NC(=O)CCCc2cccs2)C1 79862,n1(CC(C)C)cc(NC(c2ccn(C)n2)c2nnnn2Cc2ccco2)cn1 79863,c1(NC(C2CCCC2C(=O)NC2(c3cc[nH]n3)CC2)=O)cccc(F)c1F 79864,c1(OCC)ccncc1C(=O)NC1CC(C(C)NC(=O)CC(C)(C)OC)C1 79865,C1(C(C)C)CCc2[nH]nc(C(=O)NC3(CNC(=O)C(O)CCN(C)C)CC3)c2C1 79866,CC1(C)CN(C(C2(Cl)CC23CCC3)=O)C(CNC(c2cc(C(F)F)no2)=O)CO1 79867,C(C(CO)(CO)NC(=O)CN(C1CCSC1)C)N(C(c1nc(C(C)C)sc1)=O)C 79868,C12(NC(COCCSC)=O)CCCC1CN(C(=O)C(=O)NCC1CC1)C2 79869,N1(C(c2cccc(CC)c2)=O)CCC(CO)C(NC(=O)CCC(N)=O)C1 79870,N1(C(C(C)SC(=N)O)=O)CC2CCC2(CNC(=O)C(F)(F)Nc2ccccn2)C1 79871,N1(C(=O)C=Cc2ccncn2)CCN(C(C2(O)CC2)=O)CC(O)C1 79872,C(=O)(CCCCCCCCC1CCCC1)NCCn1cc(CN(S(C)(=O)=O)C)nn1 79873,C1(C(NOCCCCC)=O)CC(C)CN1C(=O)C(=O)NOC 79874,Nc1cc2[nH]cnc2cc1C(N1CCC(NC(=O)Cc2csc3cncn23)C1)=O 79875,C(C(O)CC(=O)NCC1(C)CCOCC1)NC(C(C)OCCC=C)=O 79876,C(=O)(C(C)(O)CCC)N(C1CCCN(C(c2c(CC)nccc2)=O)C1)CCF 79877,C1(CNC(CCCC(N)=O)=O)CN(C(c2cc3ncccc3[nH]2)=O)CCC1(F)F 79878,C(=O)(C1=CS(=O)CCC1)N1CCC(NC(c2cn(C(F)(F)CO)nn2)=O)C1 79879,N1(C(CN2CC(C)(OC)C2)=O)CC(CNC(=O)C=CC2CCCC2)CC1C 79880,C12(NC(Cc3scc(C)c3)=O)CCCC1N(C(c1cnc(F)cc1C)=O)CCC2 79881,C(=O)(C1CCc2cc(Br)ccc21)N1CCN(C2CCCN(C)C2)CC1 79882,Cc1scc(CNC(c2ccccc2CC(N2CC3C(C2)C3(C)C)=O)=O)c1N 79883,c1(C(=O)NC(CCC)CC)ccc(=N)[nH]c1Cl 79884,c1(CNC(c2csc(C)c2C)c2n(CC)nnn2)cccc(F)c1 79885,Cc1cc(C(N2CCC3(CC3C(=O)Nc3[nH]cnc3C#N)C2)=O)ccc1O 79886,C(C(=O)NN1CCCC1C(N1C(C)CC1(C)C)=O)SC(C)C 79887,C(=O)(C1CCCc2ccccc21)NC(C1N(C(Cc2cnc(C)[nH]2)=O)CCC1)C 79888,c1(C(N2CC(O)(C(C)NC(C3CCCN3C)=O)C2)=O)ccccc1Br 79889,C1(OC)CC2CCC1N(C(C1(O)Cc3ccccc3C1)=O)C2 79890,c1(C(=O)N(CCc2nn[nH]n2)CC2CCOCC2)cc([N+](=O)[O-])c(Cl)cc1Cl 79891,Cc1cc(C(=O)C=CC(=O)N(CCC(C)NC(c2ccc[n+]([O-])c2)=O)C)ccc1F 79892,N1(C(Cn2c(C)ccn2)=O)Cc2nccn2CC(NC(=O)OC(C)(C)C)C1 79893,c1(OC)cc(Br)c(C(=O)NC2CCN(C(=O)CO)CC2(C)C)cc1OC 79894,N1(C(c2ccn3cncc3c2)=O)CCCC2(CCCN2C(=O)C2=NOCC2)C1 79895,C1(NC(C2CC=C(C)CC2)=O)CCN(C(c2ccncc2Cl)=O)C(C)C1 79896,c1(C(=O)NCC(C)NC(C2(OC)CCOC2)=O)cccc2cc(F)ccc12 79897,N1(C(C(C)=C(CC)C)=O)CC(F)CC1CNC(=O)COc1ccccc1Cl 79898,CC(C)C(C)(C)C(=O)NC(C1CCCN1C(C1CCCOC1)=O)C 79899,c1(C2(F)CC(N(C)Cc3cn(CC(C(=O)OC)O)nn3)C2)ccccc1F 79900,CC1CCN(C(=O)CCCn2cncn2)C1CNC(=O)CCc1cnn[nH]1 79901,c1(CNC(=O)COC2CCN(C(=O)CC3CC4CC3C4)C2)nc2ccccc2[nH]1 79902,c1(C(N(C2CCN(C(=O)CSCc3cccs3)C2)C)=O)cnncc1O 79903,C1(CSC)CC2CN(C(=O)CC3(NC(=O)OC(C)(C)C)CCCC3)CC12 79904,Cn1nc(Br)c2c(NC3CC(=CC(C)(C)C)C3)ncnc12 79905,c1(NC(=O)NC2CCN(CC(F)(F)F)C2=O)ncccc1OCOCC(F)F 79906,N1(C(CN2C(C(N(C)C3CC3)=O)CC(F)(F)C2)=O)CCC2(CC1)OCCO2 79907,N1(C(CCc2onc(C)n2)=O)CC2(C1)C(NC(=O)CC(C)C(F)F)CCS2(=O)=O 79908,c1(C(=O)NCC)ccc(OC)c(-c2cccc(F)c2O)c1 79909,n1(CC)c(N)c(C(=O)CN(C)C(c2ccc3ccccc3c2)C)c(O)nc1=O 79910,c1(C(=O)NCc2cc(C)c(C(=O)NC(C)CS(N)(=O)=O)o2)cc2ccncc2[nH]1 79911,O=C(C1=CC2CCC(C1)C2)N1CCC2(CC1)CN(C(c1cnc(O)s1)=O)C2 79912,c1(OCC(=O)NC(C2N(C(CC(C=C)CC)=O)CCC2)C)cccc([N+](=O)[O-])c1 79913,CC(O)C(C(N)=O)NC(=O)COC1CCN(C(C2CCCN2C2CC2)=O)C1 79914,C1(C(=O)NC2(CN(C)C(C3CC(c4ccccc4)O3)=O)CC2)CC2C(C1)C2(F)F 79915,C1(C(N2CC(CC)C(NC(=O)COCCOC)C2)=O)CC2C(C1)C2(C)C 79916,O=S(=O)(c1cccnc1NCC(C1CCCCC1)F)NCCN1CCC(CF)C1 79917,c1(C(C(=O)NCC(C2CC2)NC(C(CC)F)=O)O)ccc(F)c(F)c1 79918,Cc1cc(C(N2CC(NC(=O)C(C)(C)C#N)C3CC23)=O)nc(O)n1 79919,N1(C(=O)Cc2nnc(S)s2)CCS(=O)(=O)CC1C1CC1 79920,c1(OC)ccccc1C1CC1NC(c1n[nH]cc1NC(c1ncc(Br)cn1)=O)=O 79921,C1(NC(CC(C=C)C)=O)CCCCC12CCN(C(=O)C=Cc1cncn1C)CC2 79922,Cc1nc2ncnn2c(C)c1C(=O)N(CC(C)(C)NC(=O)CC1CC(F)(F)C1)C 79923,C(c1cccc(Cl)c1)=CC(=O)NC(C)CC1CN(C(C2CC=CCC2)=O)C1 79924,N1(c2ccnc(C(=O)OC)n2)CCC(C)(NC(=O)NC(C)C)CC1 79925,c1(N2C3CC(CNC(C4CCS(=O)(=O)N4)=O)CC2CC3)nc2ccc(Br)cc2s1 79926,CCN=C(NCc1nccn1CCC)N1CCCC1.S(C)(=O)(=O)N 79927,CC(c1cccc(Cl)c1)=CC(=O)NCC(C)NC(c1cn(C)nc1Cl)=O 79928,C1(NC(C2(NC(=O)CC3CCC(O)C3)CCC2)=O)CCCC2(CCC2)C1 79929,N1(C(Cc2n(C)ncc2Cl)=O)CCCCC2C1CCCN2C(=O)C(F)CC1CC1 79930,O=NN1CCCC1C(=O)NCCC1CCN(C(C2CC(CF)C2)=O)CC1 79931,n1(-c2ccc(C)cc2)nc(C)c(CNCC2(C#N)CCCN2)c1Cl 79932,c1(NCc2c(C)nc(CC)o2)nccc(=NCC2(OC)CCCC2)[nH]1 79933,c1(C(=O)NCC(CNC(C(CC)F)=O)O)ccc(Nc2ncccn2)cc1 79934,Cc1c(C(=O)NCC2(NC(=O)CCSCC(C)C)CCCC2)c(C(F)F)nn1C 79935,C#Cc1ccc(C(=O)N(C(C)C(=O)NCCN2CCCC2)C)c(C)c1 79936,N1(C(C2CC(=O)NC2)=O)CCCC(C2(NC(c3c(F)cc(F)cc3Cl)=O)CC2)C1 79937,CC1CC(CNS(=O)(=O)Cc2ccccc2F)C(=O)N1c1ccccc1 79938,[nH]1cnnc1CC.C1(C(=O)NC(C)CN2CCCC2)CN(CCN)C1 79939,c1(CC(N2C3CC(NC(c4cc(Br)co4)=O)(C3)C2)=O)ccc2c(c1)OCO2 79940,c1(-c2nc(C(=O)NC(c3cccc(Br)c3)C(C)C)on2)cccc(OCC#N)c1 79941,CC(C)S(=O)(=O)CC(=O)N(CC(O)CNC(=O)CNC(c1cccc(O)c1)=O)C 79942,Cc1ccc(C(C)C)c(C(N2CC(C(=O)O)C(C(F)(F)F)C2)=O)c1 79943,CCC(C)C(O)C(=O)NCc1nc(CNC(c2ncccc2F)=O)cc(O)n1 79944,CCC(C)(CO)C(=O)NCC#CC(=O)N1CCC(CCC(C)C)C1 79945,c1(C(=O)NC2CC(C)(Nc3cccc(F)c3C#N)C2)cccn2ccnc12 79946,Cc1cnc(C(N2CCC(C(=O)NCCCC3CCCC3)C(C)C2)=O)c(F)c1 79947,N1(C(c2ccc(SC)s2)=O)CCC(F)(C(=O)Nc2ccc(F)c(C)n2)CC1 79948,CCC(CC(=O)N1CC(CO)(NC(=O)C=Cc2ccco2)C1)C(F)F 79949,c1(C(=O)NC23CC(NC(CC4CC(C)OC4)=O)(C2)C3)cccc2ccn(C)c12 79950,CC(CC(C)NC(=O)C=C1CC1)NC(C1CC1OC)=O.c1(C)ccccc1 79951,N1(C(c2ccc(C)cc2)=O)CCC(C(N2CCC(OC3CC3)CC2)=O)CC1C 79952,c1(C(=O)NC2CC(C)(NC(C3C(OC)C3)=O)C2)nc(C(F)(F)F)cn1C 79953,c1(C(c2n(CCCCCC)nnn2)NC2CC(CSC)C2)cnn(CC)c1CC 79954,c1(COC)nc(C(=O)NC(C)CCN(C)C(C2CC23CCC3)=O)co1 79955,c1(CNC(CC2(NC(Cn3c(C)nnn3)=O)CCC2)=O)cc(Cl)ccc1F 79956,C(CN1C(=O)Cc2ccccc21)NC1(c2n(CC=C)nnn2)CCNC(=O)C1 79957,C#Cc1cncc(C(=O)NCC2C3CN(C(c4cnc(OC(C)=O)s4)=O)CC23)c1 79958,N1(C(CC(=C)Br)=O)CC(CNC(=O)CCCN(C)C)CC1C 79959,C(=O)(C(O)C(C)(C)CC)N1CC(CCNC(=O)CN2CCC(C)(O)C2)(OC)C1 79960,C(=O)(N=c1cc(C(=O)OC)n(C)[nH]1)C1(NC(C(C)=CCC)=O)CCCC1C 79961,c1(C(C(=O)NC)N(C2CCC(C(F)(F)F)CC2)C)cc2n(n1)CCCCO2 79962,C1(NC(C)=O)CCN(C(=NCCCC2CCCCO2)NCCc2cccs2)C1 79963,c1(CN(C(C(=O)NCCc2ccc(Cl)cc2)=O)CC2CC2)ccccc1C#N 79964,C1(NC(CC2CCN(C)C2)=O)CCN(C2CCN(C(C3CC3F)=O)CC2)CC1 79965,C(CCCC(=O)NCCC(C)NC(c1n[nH]c(C2CC2)c1Br)=O)OCCC=C 79966,O=C(C#CC1CCOCC1)NC1CN(C(c2cccc(CO)c2)=O)CC1F 79967,c1(C(=O)NC(C)CNC(=O)Cc2cc[nH]n2)cc(C(N)=O)n(C)n1 79968,CN1CCN(c2nc(Cl)ncc2Cl)C(CNC(C2CC3CCC(C2)C3)=O)C1 79969,C1(F)(CNC(c2ncc(C)s2)=O)CCCN(C(C2(C(F)(F)F)CC2)=O)C1 79970,S(=O)(=O)(c1ccc(NCC2(N(C)C)CC2)nc1)N1C(C)CCc2ccccc21 79971,c1(C(N2CC(CN(C)C(C3CCC4CC4CC3)=O)C2)=O)cnn2c(N)ccnc12 79972,C1(F)(C(N2CCC(c3cnc(Cl)s3)C2)=O)CS(=O)(=O)CC12CCC2 79973,C1(NC(CC(COC)C)=O)CCN(C(=O)CSCC(=O)Nc2ccco2)C12CC2 79974,c1(C(N2CC3(C2)CN(C(C2(CF)CC2)=O)C3)=O)ccc([N+](=O)[O-])cc1 79975,c1(C(=O)NCC23C(CN(C(C(C(=C)Cl)(C)C)=O)C2)C3)cccc2c1ncn2C 79976,C1(C(=O)NC2CN(C(C(C)NS(CC)(=O)=O)=O)C2)(SC)CC(C(F)F)C1 79977,c1(NCC2CCCCN(C(Cc3ccc(C)s3)=O)C2)nc(Cl)nc2ncn(C)c12 79978,Cc1c(NCCCOCCC(C)C)ncnc1N1CCC(C)(F)C1 79979,c1(CN(C(=O)C=CC2(C)CCOCC2)C)cc2ccccc2[nH]1 79980,c1(C(=O)NC(CC=C)CNC(C2CC(F)(CO)C2)=O)cc2ccccc2nc1C 79981,c1(C(=O)NCC2N(C(C(F)=CCC)=O)CCC2)cc2ccc(OC)cc2s1 79982,O=C(CCCCc1ccc(F)cc1)NCCC1CN(C(C2C3CC3C3CC23)=O)C1 79983,C1(NC(c2cc(F)cs2)=O)CCCN(C(=O)Cc2cnccn2)CC1 79984,C1(NC(c2cc(O)cc(Cl)c2)=O)CCN(C(c2ccccc2)=O)CC1CO 79985,c1(C(=O)NC(CNC(C2C(C)C2)=O)C)nc(C2CC2)ncc1Br 79986,c1(C(C)OC)ncc(C(=O)NCCN(C)C(C2CC2C2CC2)=O)s1 79987,c1(NC(=O)Cc2cccc(Cl)c2Br)cc(Cl)cc2nc(O)oc12 79988,C1(C(C)C)C(NC(=O)CCC2CCOC2)CCN1C(=O)CCCN(C)C 79989,c1(C(N2CCN(C(C(CC)C)=O)C(C)C2)=O)oc2ccccc2c1CO 79990,n1(CC)cc(Br)c(C(=O)NC(C)CC(C)NC(c2cc(C)[nH]n2)=O)n1 79991,N1(C(=O)NCc2c(C)nc[nH]2)CC(CNC(C)(C)C)C2(CCOCC2)C1 79992,C1(C(N2CC(N(C)C(c3ccnc(S)c3)=O)C(O)C2)=O)CCC2CCC1O2 79993,N1(C(c2n(CC)ncc2)=O)CCCCC(N(C(=O)COCc2ccccc2)C)C1 79994,C1(C(=O)NC2CC(n3cc(C(C)(C)C4CC4)nn3)C2)CCC(C2CC2)C1 79995,C(C)(C)(CN(C(=O)C(C1(C)CC1)NC(=O)C(=O)NCC(F)F)C)OC 79996,c1(OCCOC)cncc(C(=O)NC2CCC(NC(C3CC=CC3)=O)C2)c1 79997,N1(C(CC2(COC)CC2)=O)CCOC2CN(C(C3CCSCC3)=O)CC12 79998,N1(C(c2cnc(OC)nc2)=O)C(CNC(c2cc(Br)c[nH]2)=O)CC2COCC12 79999,c1(C(N2C(CCNC(CCOCCOC)=O)CSCC2)=O)cnc2ccoc2c1 80000,c1(C(=O)OC)sc(NCC2CCCCC2NC(c2nccn2C)=O)c(CN)c1C 80001,CC(C)CCC(=O)C(=O)NCC(O)CNC(C1CCOCC1(C)C)=O 80002,C1(OC)CC(C)CN(C(=O)C(CCC2CCC2)NC(C2CCC(O)CC2)=O)C1 80003,C=CC(C)(CC)C(=O)NC1CCN(C(c2c(C)ccnc2OCC)=O)CC1 80004,C12(CNC(C(CSC)(C)C)=O)CCC(CNC(=O)C3=COCC3)(CC1)CO2 80005,N1(C(C(C)(C)NC(=O)OC)=O)CCN(C(C)CNC(=O)Cn2ccnc2C)CC1 80006,C#CCCC(O)C(=O)N1CC(C2(NC(=O)Cc3ccc(CO)cc3)CC2)C1 80007,CC1CN2CCN1C(C(=O)NC1CC(CNC(C3CCCC(O)C3)=O)C1(C)C)C2 80008,C(=O)(CC(CC(C)C)NC(=O)COCC1CCC1)N1C(CC)C(O)CC1 80009,CCCCCCC(=O)NCC1CN(C(C2CC3(CC3)CN2C)=O)CC1C 80010,N12CCC(C)(C1)OC1CCN2C1.C1(C#N)(C=O)CCCO1.C(C=O)SC(C)C 80011,CC(C(CO)NC(=O)CCc1nncs1)NC(=O)C=CCO 80012,Cc1ccc(OC(F)(F)F)c(CN2CCN(C)C(C(=O)N(C)C)C2)c1F 80013,C(CCOCCO)(C(=O)N(CC(F)F)C)NC(Cc1c(C)scc1)=O 80014,CCCN=C(NCCC(=O)Nc1nnnn1C1CCC1)NC(c1ccnn1C)C 80015,C1(C(N(C2CC(=C)C2)C)=O)CCCCC1NC(=O)CCOCC(F)F 80016,C1(C2CN(C(=O)Cc3cn(CC4CCCCNC4=O)nn3)C2)(C(=O)OC)CC1 80017,N1(C(CC(C)SC)=O)CCC2(CCC2)C(CNC(=O)CC=CC(C)(C)C)C1 80018,n1(CC(N2C(CNC(C(CC=C)C)=O)C=CC2)=O)cccc(C)c1=O 80019,C=Cn1ncc(C(=O)NCC2CCCN2C(=O)CCc2ccc(C)o2)c1N 80020,CC1(CC(=O)NCC(F)CNC(=O)CCCNS(C)(=O)=O)CC1(Cl)Cl.C1=CC=C1 80021,N1(C(C2CCC2)=O)CCCOCC1.C(=O)(CCCC#N)NCc1cc(C(N)=O)[nH]c1 80022,N1(C(C2C(C)N(C)C(=O)C2O)=O)Cc2ccnn2CC(NC(=O)OC(C)(C)C)C1 80023,c1(C(=O)NCC(CNC(C2CC(C(C)=O)C2(C)C)=O)F)ccc(F)cc1F 80024,N1(C(c2cc(C)c(Br)cc2)=O)CC(CNC(c2cncnc2)=O)C2(CCC2)C1 80025,C1(C)(N(C(=O)C2CC2)CC)CCN(C(c2sncc2C)C(=O)NC(C)(C)C)C1 80026,N1(c2n(CCOC)c(-c3cnn(C)c3)nn2)CCOC2(CCOC2C)C1 80027,Cn1nc(C2CCOCC2)cc1C(N1CCOCC1CCNC(=O)C(C)(Cl)Cl)=O 80028,C(=O)(C(C)(C)CCSC)N(CCN(C(C(CSC)O)=O)C)C 80029,C(=O)(C1=CCCN(C(C2CC2OC(C)=O)=O)C1)N1C(C)CC1(C)C 80030,c1(NC(C=C2CCN(Cc3ccc(OC)cc3O)CC2)=O)nc(Cl)c(C)c(Cl)n1 80031,C1(C(=O)NC2CC3(C(NC(c4ncn(C)n4)=O)C3)C2)Cc2ccccc2NC1=O 80032,Cc1ncnc(C)c1C(=O)N(CC(C)N(C(=O)C(CC(C)C)n1ccnc1)C)C 80033,Cc1cc(C(=O)NC2CC(CC(=O)Nc3nccnc3Cl)C2)ncc1[N+](=O)[O-] 80034,CC1CCN(C(=O)C(C)CC(N)=O)C(CNC(=O)Cc2cccc(O)c2)C1 80035,N1(C(C2C(C)C2)=O)CC2CC2(NC(c2coc(Cc3ccccc3)n2)=O)C1 80036,C1(C(=O)NCC2(CNC(C3C(C(N)=O)C3)=O)CCC2)CCCCNC1=O 80037,n1(C(C(=O)NCC2CCN(C(C(C=C)O)=O)CC2)C)nc([N+](=O)[O-])cc1C 80038,N1(C(c2cn(C)nc2)=O)CCCC2CCN(C(c3cc(C(N)=O)cs3)=O)CC12 80039,C1(NC(COCCCCC)=O)CCCC(NC(C2CC(N(C)C)C2)=O)C1 80040,N#Cc1cc(NC(C2CN(C(=O)CC3CCCCO3)CCS2)=O)cnc1Cl 80041,C1(NC(CNC(CC(C)C)=O)=O)CC2CC1CC2C(N1CC(C)C(O)C1)=O 80042,Cc1cc(C)c(CC(=O)NCC2CCCCC2NC(=O)CCc2cnc[nH]2)c(C)c1 80043,C1(CC(=O)NCc2[nH]nc(C3CCN(C(CC)=O)CC3)n2)CCCC(C#N)C1 80044,C(=O)(C(CC1CCCC1)NC(c1ccncn1)=O)NC(C(=O)N(CC)CC)C 80045,C1(O)(CNC(CCC(C)SC)=O)CCCN(C(=O)C(F)=CC2CC2)C1 80046,N1(Cc2nn(CC)nc2C)CCCC1C1CCCCN1C(=O)Cc1ccsc1 80047,N1(C(c2ccc(Cl)cn2)=O)CCN(C(c2ccc([N+](=O)[O-])o2)=O)C(CC(F)F)C1 80048,N1(CC(=O)N(CC=C)CC(C2CCCCS2)=O)CCC(OC)C1 80049,c1(C(=O)NC(C2CN(C(c3cnc(O)n3C)=O)CCO2)C)cc([N+](=O)[O-])cn1C 80050,N1(C(c2nnn(CC)c2C)=O)CC2(CNC(C3CN(S(C)(=O)=O)C3)=O)CC1CO2 80051,Cc1cc(NC(c2nncn2C2CC2)=O)ccc1N1CCOCC1 80052,c1(C(=O)NC(C2CCCO2)CC)ccc(CNC(C2CC(C)(O)C2)=O)o1 80053,CC(Cc1ccccc1Br)N=c1cccc(S(=O)(=O)NCCC2CC2)[nH]1 80054,N1(C(CC(C=C)CC)=O)CCC(CNC(=O)C2=CCCC2(C)C)C(F)(F)CC1 80055,N(C1CCC(NC(C)C)c2ccccc21)C(CN(C(C)C(C1CC2CC1C2)=O)C)=O 80056,c12cccc(c1)C(=O)N2.N1(CC2N(C(c3c(C)cco3)=O)CCC2)CC(C)C(O)C1 80057,c1(OC)cccc2cnc(N3CCC4(CC3)CC(NC(C3(Br)CC3)=O)C4)nc12 80058,c1(C(=O)NC2C(n3cc(C(C)(C)SC)nn3)COC2)cc(Cl)ncc1Br 80059,CC(C)C(CNC(=O)CN1CCCCCC1)C(=O)NCc1ccc(CO)cc1 80060,c1(SC)cccc(C(N)C(N2CCCC2Cc2nccn2C)=O)c1 80061,C1(C(=O)NOC2CCC2)(C(C)C)CCCN1C(C1CC(C)(C)CO1)=O 80062,CN(C)S(=O)(=O)NCC(=O)NCCC1CCN(C(C2C=CCCC2)=O)CC1 80063,C1(CNC(C(CC)NC(N)=O)=O)CCCCC1NC(=O)CCNc1ccc(C)cc1 80064,C1(C)(CCNC(C2(N(C)C(c3nc(Cl)cs3)=O)CC2)=O)CCOCC1 80065,c1(C(=O)NCC2C3CN(C(C(C)OC4CCCC4)=O)CC32)nnn2ccccc12 80066,C1(C(N(CC#C)CCO)=O)CCOCC1NC(=O)C1=NOCC1 80067,N1(C(CC=C(C)C)=O)CCC(CCNC(=O)C=Cc2cscn2)CC1C 80068,Cc1ccc(C)c(C(=O)NC2CC(C)N(C(C3CCC(N(C)C)CC3)=O)C2)c1 80069,CCCC(F)C(=O)NCCCOCCC(N1CC(OCC)C(F)C1)=O 80070,n12nnnc1C(c1cnc(C(F)(F)F)s1)NCC2.C1(CCCSC)CCCCO1 80071,S(=O)(=O)(c1ccc(C(=O)N(C)CCNC(=O)CC2CCC(OC)CC2)o1)NC 80072,Cc1ccc2nc(C(N3CCCCC(NC(c4ccc(Cl)o4)=O)C3)=O)c(N)n2c1 80073,N1(C(c2cncc(OC(C)C)c2)=O)CC(C)(C)CCC1CNC(C1CCSC1)=O 80074,N1(C(C2C=CCN(C(C(CC#C)O)=O)C2)=O)CCOCC(O)C1 80075,N1(C(C(C)=C2CC2)=O)CCC2(CC1)CN(C(c1cccc(C#N)c1C)=O)C2 80076,c1(OCCC(=O)OC2(C(=O)NCC(C)(C)CN(C)C)CCC2)ccccc1F 80077,O=C(C1CCCc2n[nH]cc21)NC1(CF)CCN(C(=O)C(F)(F)C2(O)CCC2)C1 80078,c1(C(=O)NC(C(C(C)C)NC(C2(C)CCC(=O)N2)=O)C)cncc2nc(O)[nH]c12 80079,NS(=O)(=O)c1n[nH]cc1C(N1CCCC(NC(=O)CC2CCCCC2O)CC1)=O 80080,Cc1cnc2cc(C(N3CCOCC3CNC(=O)CCc3csnn3)=O)ccn12 80081,C(=O)(C1=CC2(CN(C(=O)C(C(CC)CC)OC)C2)OC1)N1C(C#C)CCC1 80082,C(=O)(C(CNC(=O)C(OC)OC)C(C)C)Nc1c(CC)noc1C 80083,C1(C(=O)NCc2cc(COC)n[nH]2)CCCN(C(=O)COCCC(C)C)C1 80084,c1(C2(C(=O)OC)CC2)cn(CC2CCN(C(=O)CSc3cccs3)C2)nn1 80085,Cc1cc(C#N)ccc1NCC(C1CCN(c2ncc(Br)cn2)C1)C 80086,C12(C(N(CCN(C)C(c3cnc(O)s3)=O)C)=O)CCC(CC1)C2(C)C 80087,c1(C2OCCN(C(C(CC(=O)NC(CC(C)C)=O)F)=O)C2)ccc2ccccc2c1 80088,C1(C(=O)NC)CCC2(CCN(C(C3CC(F)(F)C3)=O)CC2)O1 80089,Cc1cccc(NC(=O)Nc2cccnc2C(N)=O)c1.c12ccc(cc1)c(=O)[nH]2 80090,c1(C(=O)NC2CC2C(=O)N=c2ccn(CCNO)[nH]2)cccc2c(O)nccc12 80091,CC1(C)OCCC1C(=O)NC1CCC(NC(C2CC(F)(CO)C2)=O)CC1 80092,C(CCCCCNC(C1(C)CC(C#N)C1)=O)N(C(=O)C(C)(C)n1cccn1)C 80093,c1(C(C)C)ccc(F)c(C(N2CC(NC(c3ccnc(C(C)C)n3)=O)C2)=O)c1 80094,C(=O)(C1=CC2(CCN(C(c3ccoc3)=O)C2)C1)NCC(N1CCOCC1)C 80095,C(=O)(CC(CC)C(C)(C)C)N.CCCCCCc1cccnc1.c12n[nH]c(n1)CC2=O 80096,C(C(=O)NCC1(NC(=O)CCc2cncs2)CCC1)(c1cccs1)SC(C)(C)C 80097,C=CC(C)(C)CC(=O)NC(C1CCCCN1C(c1ncccc1NC(C)=O)=O)C 80098,c1(C(=O)NC2CCC(CNC(C3(SCC)CC3)=O)C2)cncc2c[nH]nc12 80099,C1(NC(C(C(C)C)O)=O)C2CC1CN(C(c1cc(C#N)on1)=O)C2 80100,N1(CC)CC2CC1CN2C(C1CC(CNC(C2CC=C(C)CC2)=O)C1)=O 80101,N1(C(C(C(C)C)SC)=O)CCCC2(C1)CN(C(c1cccc(O)c1F)=O)CCO2 80102,C12(C(=O)NC3CCN(C(c4n[nH]c(C)c4Cl)=O)C3)CCCN(CC1)C2 80103,CC1(CNC(c2cc(N)ccc2O)=O)CCCN(C(c2c(F)ccnc2Cl)=O)C1 80104,CC1(C)CN(C(c2ccc3sncc3c2)=O)C(CNC(=O)C=CCO)CO1 80105,c1(C(=O)NCC(C)(C2CC2)NC(=O)CCCC#N)cc2cncn2c(O)n1 80106,c1(C(N(C2CCN(C(CC(C=C)C)=O)C2)CC)=O)cc2nc(Cl)ccc2s1 80107,c1(NCCC)nccc(N2CCC(Cn3ccnc3)CC2)n1 80108,C1(NC(C(C(CC)CC)C)=O)CCOC12CCN(C(=O)CC(=O)N(C)C)CC2 80109,C1(NC(C2C(OC)C2)=O)CC1C1CCN(C(c2cnc3ccnn3c2C)=O)CC1 80110,c1(C(CNC(NNC(c2cccc(OC)c2)=O)=O)C)ccc(S(C)(=O)=O)cc1 80111,C1(C(=O)NCCCN(C(c2cncc(NC)n2)=O)CC)CCCCC1C1CC1 80112,N1(C(CC(CC)N(C(=O)CN2CCOC2=O)C)=O)CCC(O)C(CO)C1 80113,Cc1nc(C(C)C)ccc1C(=O)NC1CN(C(=O)CN2CCC(C)CC2)CC1F 80114,C(=O)(C(C)(C)CS(N)(=O)=O)NCCC1CC(C)(C)OC1 80115,Cc1ccc(O)c(NC(=O)CC2(N(C(=O)CC=Cc3ccccc3)C)CC2)c1 80116,c1(OCC)ccc(C(=O)NCC2CC(NC(C3(n4cccn4)CC3)=O)CCO2)cc1 80117,C1(COC)COCCN(C(=O)CC(C)NC(c2cc(Br)cs2)=O)C1 80118,C(=O)(C1CCc2cc(C)ccc21)N1CC(CNC(COCC#C)=O)(COC)C1 80119,C(CC(=O)NOCC=C(C)C)C1CC(NC(C2(C(=O)OCC)CC(F)C2)=O)C1 80120,c1(CC(=O)NC2C3CC(NC(C=CC=CC)=O)CC32)c[nH]c2ncccc12 80121,O(NC(=O)C(CCF)NC(c1cccc(O)c1F)=O)CCCC=C 80122,c1(C(N2CCCN(C(C3CCC(=C)CC3)=O)CC2)=O)cc(C)cc(OC)c1C 80123,N1(C(c2[nH]cc(C)c2)=O)CCC2(C1)CN(C(=O)CCCNS(C)(=O)=O)C2 80124,c1(OC)ccc(C(=O)NC(C2(O)CN(C(C3CCCSS3)=O)C2)C)cn1 80125,c1(C(=O)NC(CN(C)C(C2CC3CC2CC3O)=O)(C)C)ccn2ncccc12 80126,Cc1nc(N2CCCCC(CNC(=O)CC(C)C)C2)c2c[nH]nc2n1 80127,CC(N=c1cc[nH]cc1S(=O)(=O)NCCc1cncn1C)c1ccccn1 80128,c1(C(N(CCNC(C2(SC)CC2)=O)CCOC)=O)c(C)cc(Br)cc1F 80129,c1(C(=O)NC2CCC(CCNC(c3cscc3F)=O)C2)cn2c(n1)SCC2 80130,C(C(=O)NCC1CC(C(=O)N(CC(O)CF)C)CO1)(C(C)C)SC 80131,N1(C(c2cc(CCC)on2)=O)CC(NC(=O)C(C)=C2CC2)CC12CCC2 80132,N1(C(C2C(CC)NCC2)=O)CCC(N)c2c(Br)cccc21 80133,CC(C)C(C)CC(=O)NCC1CC(O)(CNC(c2cc(Br)sn2)=O)C1 80134,N1(C(c2nc(C)sc2)=O)CC2(CCC(NC(c3c(C)cncc3C)=O)CC2)C1 80135,c1(CCC(=O)N2CC(CC(CC(=O)OC)NC(C)C)C2)ccc2c(c1)CCO2 80136,C1(C(=O)NCC(CNC(C(C(=C)C)(C)C)=O)(C)C)CCc2nncn2CC1 80137,C(c1ccc([N+](=O)[O-])s1)=CC(=O)NCCN(C)C(C1COC(=O)N1C)=O 80138,N1(C(c2cccc(N3CCCC3=O)c2)=O)CC2CCC(C1)N2C(C1CCC1F)=O 80139,CC1CCN(C(c2cnn(C)c2Cl)=O)CC1CC(N1CC(n2ccnn2)C1)=O 80140,C1(C(=O)NCCc2cccnc2O)CC2CC1CC2O 80141,n1(CC)ncc([N+](=O)[O-])c1C(=O)NCC(C)CNC(c1ncn(C(C)(C)C)n1)=O 80142,c1(C(=O)NCCc2cc(C(=O)NCC3CC3(Cl)Cl)no2)n[nH]c(C2CC2)n1 80143,N1(C(CC2(OC)CCCC2)=O)CCC(NC(=O)Cc2cncn2C2CC2)C1C 80144,c1(C(=O)NC2CCCCN(C(C(CC)C#N)=O)C2)cc2cc(OC)ccc2cn1 80145,n1(C(C)C(N2CC=CC(NC(=O)CCC3CC3C)C2)=O)cnc2ccccc12 80146,c12ccc3c(ncn3c1)C(=O)N2.N1(C(C2CCCN(C)C2)=O)CCOCC1(C)C 80147,C1(C(=O)NCCCN(C(C(C)=C(C)C)=O)C2CC2)CC12CCS(=O)(=O)CC2 80148,c1(N2CC(NC(C(c3ccc(Cl)cc3)C)=O)C(C#N)C2)ncnc2cnccc12 80149,N1(C(c2c(CC)nc[nH]2)=O)CC2(CCN(C(=O)CSC(C)C)C2)C1 80150,c1(CC)nc(C2CC23CC3)n(-c2ccn(C)n2)n1 80151,C#CC1(C(=O)NC2CCC(C)(CC)CC2)CCN(C(=O)Cc2cncnc2)CC1 80152,C1(C(=O)NC(c2ccc(F)c(F)c2)CC(F)(F)F)(COC)COC(C)(C)OC1 80153,N1(C(Cc2cnc(C)s2)=O)CCC(CNC(c2c[nH]nc2C)=O)C(C)C1 80154,C1(NC(C2CCn3nccc3C2)=O)CCC2(CCNC2)C1 80155,c1(CCCNC(c2cn(C)nn2)C)nc2c(s1)CCCC2 80156,c1(C(N2C(CNC(CC(=O)NCC)=O)CC(C(F)(F)F)C2)=O)coc2c1CCCC2 80157,C(=O)(C1Cc2ccccc21)N1C(CCNC(C2N(C)CCOC2)=O)CCC1 80158,N1(CCNC(CNC(=O)OCC)=O)CCN(C(C2CCOC2C2CC2)=O)CC1 80159,c1(NC(C=CC(C)(C)NC(C2CCCCCC2)=O)=O)ccc(O)cc1O 80160,C1(COC)(NC(=O)CCCC2CCCCC2)CCN(C(=O)C2=NOC(C)C2)CC1 80161,CCCCCC(O)CC(=O)NC12CC(C1)N(C(=O)COC1CCC1)C2 80162,C12(C(N3CCC(N(C(=O)C(C)N(C)C)CCC)C3)=O)CCC(O)(CC1)CC2 80163,c1(C(N2CCCC(F)(C(=O)NCCC(O)C3CCC3)C2)=O)cc2occc2[nH]1 80164,CC(C)(C)C=CC(=O)N(C1(CNC(=O)C(=O)NC2CC2)CC1)C1CC1 80165,c1(CC)cnc(O)c(C(=O)NC(C)(CNC(C2CC2(Cl)Cl)=O)C2CCC2)c1 80166,S(=O)(=O)(c1ccc(Cl)s1)N1CCN(C(c2ccn(C3CC3)n2)C(=O)NCC)CC1 80167,C1(NC(C(CSC)O)=O)CCN(C(=O)Cc2c(F)cncc2Cl)CC(O)C1 80168,C=CCC(CC=C)C(=O)N1CCC(F)(F)C(CNC(c2ncc(C)cc2F)=O)C1 80169,c1(C(N2C(CC(C)O)CCCC2)=O)cccc2c1COC2 80170,c1(CNC(=O)Nc2ccc(Oc3ccc(Cl)cc3Cl)cc2)cc(F)c(Br)cc1F 80171,C1(NC(C=CC=CC)=O)CCCC1(C)CNC(=O)CC(c1ccccc1F)NC 80172,CCCCS(=O)(=O)CC(=O)NC1(CC)CCN(C(=O)C(C)=C2CCCC2)CC1 80173,c1(CCC(=O)N(C(CNC(CC(=C)C)=O)C)C)ncccc1C 80174,c1(C(N2CCC(C)(OCC(C)C)C2)=O)cnc(O)c2ccccc12 80175,c1(C2(CNC(CC)CSc3nc(C4CC4)ns3)CCC2)nnnn1C 80176,N1(C(CC(CC)(F)F)=O)CCC2CCN(C(C3C(C=C(C)C)C3(C)C)=O)C2C1 80177,C1(CNCC(CN(C(=O)OC)C)O)CC2CCCC2C1 80178,CCCC(CCO)NC(c1n[nH]cc1NCc1cnc(-c2ccccc2)[nH]1)=O 80179,C(=O)(CCN(OC)C(=O)CC(C)n1cccn1)N(C)Cc1cccc(OC)c1 80180,C1(OC)(CN(C)C(C2CSCN2C(C2CC(C(C)C)C2)=O)=O)CCOC1 80181,C1(CC(=O)OC)CCN(N2CCC(CCOc3ccccn3)CC2)CC1 80182,C1(F)(CNC(C(C)C2CC2)=O)CC(NC(C2(c3ccccc3)CC2(Cl)Cl)=O)C1 80183,C=CCC(CC)C(=O)NCC(C)NC(C1(C)COC1)=O 80184,N1(C(c2cncc(C(C)(C)C)c2)C(=O)NC2CC2)CCc2ccc(Br)cc2C1C 80185,N1(C(c2c(CC)nc(C)o2)=O)CC(C(=O)N(CCCO)C2CC2)C(C)(C)C1 80186,c1(NC(C(=O)NCCc2cc(C)oc2C)=O)ccc(S(C)(=O)=O)cc1 80187,C1(NC(COCCCCCC)=O)CCCC(CN(C(=O)C2=CCSC2)C)C1 80188,c1(NC(C)=O)ccc(C(N2CCC(CC(=O)Nc3cc(O)n(C)n3)C2)=O)cn1 80189,C1(CC(N2CCCC(NC(CCc3n(C)cnn3)=O)C2)=O)OCCOC1(C)C 80190,C1(C(N2CC(COC)C2)=O)CCCC12CCN(C(c1cc[nH]c(=NC)c1)=O)C2 80191,C1(CCC)(NC(C2CCCN2C=O)=O)CCN(C(c2[nH]cnc2C)=O)CC1 80192,N#Cc1ccc(COc2ccnc(N3CCC(C4CCC5(CC5)CO4)C3)n2)cc1 80193,n1(CC(=O)NCC(C(C)C)NC(C2CN(C)CCO2)=O)cc2ccccc2n1 80194,c1(OCCN2CCCC(C(=O)NC3CC(C)(NC(C)=O)C3)C2)c(C)cc(C)cc1C 80195,C1(CNC(CC(C)OC)=O)(CO)CCN(C(c2ncoc2-c2cnn(C)c2)=O)C1 80196,C(CC(O)CNC(C1C2CCCC12)=O)NC(c1sccc1C(F)F)=O 80197,Cc1ncc(C(N2CC(C)CNC(C)C2)=O)c(Cl)c1Cl 80198,CC(C)(N=[N+]=[N-])C(=O)NCC(CNC(=O)C(O)C(F)(F)F)CO 80199,CC1(C(=O)NC2C3CN(C(=O)CC4CC4(Cl)Cl)CC23)CC2(C1)CC(F)(F)C2 80200,c1(NC(CC2N(C(CCSC)=O)CCOC2)=O)ccc2nc(C)oc2c1 80201,c1(OC)cccc(NC(C2(CF)CCN(C(c3cnn(CCSC)c3)=O)C2)=O)c1 80202,C1(C(N2CCN(C(COC(C)C)=O)CC2)=O)CCc2n[nH]cc2C1 80203,c1(C(=O)NC2C(C)(C)CN(C(C3CC(F)(F)C3)=O)CC2)cc2cc(O)ccc2[nH]1 80204,C(=O)(C(C(C)O)NC(=O)C(=O)N(CCCOC(C)(C)C)C)OCC 80205,C1(CNC(c2c(C)n[nH]c2)=O)CN(C(c2c(C)ncn2C)=O)CC12CC2 80206,n1(CC(=O)NCCN(C(C(=Cc2cccc(Cl)c2)C)=O)C)cc(S(C)(=O)=O)cn1 80207,CC1=NNC(=O)C1CCC(=O)NCC1(CNC(C2CCC2(C)C)=O)CCC1 80208,Cc1ccc(CC2CC3CCC2N3CC(=O)NCc2ccccc2)c(O)c1 80209,C(=O)(CCCCCN=[N+]=[N-])N1CC(C)C(CC(=O)N(C2CC2)Cc2ncnn2C)C1 80210,c1(C(=O)NC2CC(CNC(CN(C)CC)=O)OCC2)sc(Cl)c(Cl)c1OC 80211,C1(NC(CC=CCC)=O)CN(C(c2cc(OC)c(O)c(N)c2)=O)CC2(CC2)C1 80212,c1(OC)cccc(C2(C(=O)NCC(CC(C)C)NC(=O)CN3CCC3C)CC2)n1 80213,N1(C(C(N2CC(Cc3c(C)noc3C)C2)=O)=O)CCOC(C)(C)C1 80214,c1ccc2nc(NCC3CCCS3)c(=NCC3CC34CCC4)[nH]c2c1 80215,c1(C(=O)NC(C)CNC(C2C(C)(C)C2(F)F)=O)ncn2cc(Br)sc12 80216,C1(C(N2C(CCCNC(c3cn(CC=C)nc3)=O)CCC2)=O)COCCC1(F)F 80217,CCC(CC)CCCC(=O)N1C2CCC1C(C(N1CC3CC=CCC3C1)=O)C2 80218,C12(C(=O)NC3CC(C#C)C3)CCCC1CCN2C(c1cn(C)cc1C)=O 80219,c1(C(N(CCN(C(CCC(=C)C)=O)C(C)C)C)=O)ccc(OC)c(OC)c1C 80220,CCC(C)(O)CCNC(=O)C(C1CCN(C(c2sc(C)nc2C)=O)C1)C 80221,N1(C(C2CN(c3n(C)nnn3)C2)=O)CCC(NC(c2nccn2C)=O)C12CC2 80222,N1(C(c2[nH]cc(OC)c(=O)c2)=O)CCC2C1CCCN2C(=O)Cc1cn[nH]c1 80223,C1(C(=O)NCC(C2CCCC2)O)CC2CN(C(=O)C=Cc3ccncc3)CC2C1 80224,C1(C(=O)NCCNC(=O)CCOC(=O)COCc2ccccc2)CCC(F)CC1 80225,C(C)(CO)(CS(C)(=O)=O)NC(C(n1cc(Cc2n[nH]c(C)c2C)nn1)C)=O 80226,N1(C(c2cnc(OC)s2)=O)CCC2CCCC12C(=O)NCC1CC2CCCC2C1 80227,c1(C(=O)NCC(CC)NC(=O)C(C)OC(C)=O)cc2c(s1)CCC(C)(C)C2 80228,c1(C(=O)NCC(CNC(c2c(C)c(N)ccc2)=O)O)ccccc1S(C)=O 80229,C1(CC)OCCC1C(=O)N(CC(C)(C)CNC(=O)CC1CN(C)C1)C 80230,c1(OC)cc(C(N2CC3C(C2)N3C(C2(C)CCCN2)=O)=O)cc(C(F)(F)F)n1 80231,Cc1cc(Cl)ncc1NC(C1CCC(C)N1C(c1cccs1)=O)=O 80232,CC(C)CC(C)(O)C(=O)N1CCN(CC(=O)NCCCOCC(F)F)CC1 80233,C1(C(=O)NCC(CNC(C(C)(CO)OC)=O)(C)O)CC2(C1)CC(CO)C2 80234,C(C1c2ccccc2CCN1C(c1cnsn1)=O)NC(c1cccc(OC)n1)=O 80235,Cc1noc(NC(C2C3CN(C(=O)CCCN4CCCC4)CC23)=O)c1C 80236,C1(NC(CCNC(=O)OC)=O)CCCCC1.C(=O)(C(C)n1ccnc1)NCC1CC1 80237,C1(Cn2c(C(N3CCC(F)(CF)C3)C(C)(C)C)nnn2)COc2ccccc2O1 80238,N1(C(=O)Nc2ccccc2Cl)CCC2CN(Cc3c(OC)cc(OC)nc3)CC12 80239,N1(CCNC(c2cc(CCCCC)[nH]n2)=O)CCN(C(=O)COCCCC)CC1 80240,C(=O)(C1=NN(C)C(=O)CC1)N1CCCCCC(NC(c2nccc(CC)c2)=O)C1 80241,N1(C(C(C2(O)CCCCC2)NC(c2cc(C)[nH]n2)=O)=O)CC(C)OCCC1C 80242,C1(NC(C2CCC23CCOCC3)=O)CN(C(c2ccc(Cl)o2)=O)CC2CCCC12 80243,N1(C(=O)NC2(C)CN(S(=O)(=O)CCCCCl)C2)Cc2ccccc2CC1CO 80244,N1(C(C(C)NC=O)=O)CCC(C)C(CNC(c2cc(O)nn2C)=O)C1 80245,Cc1nc(Cl)ccc1CC(N1CCN(C(=O)Cn2cnnc2O)CC1C)=O 80246,CC1CCCCC1C(=O)NCC(C)(C)CCNC(=O)Cn1ncnn1 80247,CS(=O)CCC(=O)N1CCCC(CCNC(C2(c3ccncc3)CC2)=O)C1 80248,CN1CC(O)(CN(C(=O)C(Cc2cc[nH]n2)NC(=O)CCC2(C)CC2)C)C1 80249,N1(C(C2C(C)(C)C2)=O)CCCC2(CC(NC(=O)Cn3ncc4ncccc34)C2)C1 80250,C12(CC3(CCC3)C1)NC2.C(C)(CCC(=O)NC1CC(=O)N(c2cn[nH]c2)C1)OC 80251,c1(NC)ncccc1C(=O)NC1CC(C)N(C(=O)CCc2nc(C)c(C)o2)C1 80252,C(=O)(C(C(C)O)N(C)C)NCC(CC)NC(c1ccccc1OC(F)F)=O 80253,CN=c1[nH]cc(C(=O)NC2CC(C)(NC(=O)C(C)C3CC3)C2)o1 80254,c1(C(N2CCC(N(C)C(C3CCCCS3)=O)C2)=O)ccnc2nccnc12 80255,Cc1nc(C=CC(=O)NC2CCC2CNC(c2cc(C(F)(F)F)cs2)=O)cs1 80256,N1(C(C2(SC)CN(C(=O)CCn3ccnc3)C2)=O)CCCOC(C(C)C)C1 80257,c1(OC)ccc(CNC(C2C3CN(C(=O)CNC(=O)N(C)C)CC23)=O)c(Br)c1 80258,CC(C)C(C(C)NC(c1cncc(C2CC2)c1)=O)NC(=O)C(F)(F)CO 80259,C=CCCCC(C(=O)N1CCSC(C)CC1)NC(c1cccnc1O)=O 80260,c1(NCCc2c(F)c(Cl)ccc2)[nH]c(=NC2CCC(C3CC3)C2)nc2scnc12 80261,c1(C(N2CC(C)C(NC(=O)C3=C(Cl)CCCC3)C2)=O)ccc2c(=O)cc[nH]c2c1 80262,Cc1csc2c(NC3CCC(NC(=O)CCCC(=O)NC(C)C)CC3)ncnc12 80263,c1(C(N2CC(NC(c3cncc(C(F)(F)F)n3)=O)(CO)C2)=O)ccnc(Cl)c1F 80264,c1(CC=C)cccc(C(=O)NC2CCC2NC(=O)CS(=O)(=O)N2CCOCC2)c1 80265,c1(C(N2CC(CCC)C(NC(=O)CS(=O)CC)C2)=O)ccc(OC)cc1OC 80266,C1(CC)C(NC(C2C3CC(=O)CC23)=O)CCN1C(C1CCCCS1)=O 80267,N1(C(c2[nH]cc(C)c2C)=O)CCC2CN(C(C3CN(C)CC(C)O3)=O)CC2C1 80268,N1(C(COC(C)=O)=O)Cc2ccccc2C1CNC(C1CCC1(F)F)=O 80269,c1(N2CCCC(NC(C(C)OC3CCCC3)=O)(CO)C2)ncnc2ccccc12 80270,C1(CNC(C2CCC(C(=O)NCC3C4CC5C(C4)C35)CC2)=O)C2CCCCCC12 80271,c1(NCCC2(COC)CC2)cc(S(=O)(=O)NC(C2CCC2)C)ccc1C#N 80272,c1(C(N2CC(COC)C2)=O)ccc(CNC(C2C(C(C)C)CCC2)=O)cc1 80273,c1(C(=O)NCCN(C(C(C)OCCC#C)=O)C2CC2)cc(F)c(F)c(OC)c1F 80274,c1(CC)cccc(NC(C2CCN(C(=O)C(N3CCC(CC)C3)=O)C2C)=O)c1C 80275,c1(C(N(C2CCCCC2NC(=O)C(O)C(F)F)C)=O)cccc(O)c1 80276,O=C(C#CC1CCCO1)NC1CN(C(C2CCc3nn[nH]c3C2)=O)C1 80277,CC(CCC(F)(F)F)NC(=O)CC(C)NC(=O)CC1OCCCO1 80278,c1(-c2cn(C3CCN(C(CC)C(N)=O)CC3)nn2)ccc(CSC)cc1[N+](=O)[O-] 80279,c1(OC)ccc(CC(=O)N(CC(C)CNC(C2(CC(F)F)CCC2)=O)C)cc1F 80280,c1(NC(C)=O)cccc(C(=O)NC2CC2CNC(=O)C(CCOC)N(C)C)c1 80281,Cc1csc(CCNC(C2C(CNC(c3csc(=N)[nH]3)=O)C2(C)C)=O)n1 80282,c1(C(=O)NC2CN(C(=O)CC3CCOC3)CC2C(F)F)ccc(C(F)(F)F)cn1 80283,N1(C(c2ccc(O)nn2)=O)CC2(C1)CN(C(c1ncoc1C(F)(F)F)=O)C2 80284,C#CC(Cc1ccc(F)cc1)N(C)N(C)Cc1nccn1C(C)C 80285,c1(OC)ccc(OCC(O)CN2CCC(C(C)C)C2)cc1C.C12CCNC(C1)N2 80286,c1(C(N2CC3CN(C(C4(Br)CC4)=O)CCC23)=O)n[nH]c2c1CCSC2 80287,N(C(=NCc1ccsc1Cl)NC1(CF)CCC1)C(c1cccs1)C 80288,C1(CCCC)CN(C(=O)CC(C)OC)CCN1C(c1coc(C(F)F)n1)=O 80289,CCS(=O)(=O)c1ccc(C(N2CC=CC(NC(=O)CC3CCCOC3)C2)=O)cc1 80290,C1(CC#C)(C(=O)NCCCCNC(=O)CC(c2c(C)n[nH]c2C)C)CC=CCC1 80291,c1(CC=C(C)C)ccc(CN2CCN(C(=O)NC3(C)COCCO3)CC2)cc1 80292,C1(c2cn(CC(F)(F)CO)nn2)(C(=O)OC)CN(c2ccncn2)C1 80293,C(CCCC(=O)N1CC(CC(C)(C)CNC(C2(Cl)CC2(C)C)=O)C1)N(C(C)=O)C 80294,c1(C(=O)NC2(CO)CCN(C(=O)C3=CCSC3)CC2)nc2ncccn2n1 80295,CCCCC(C(=O)NCC1(C)CCCN(C(c2ccc(F)cc2Cl)=O)C1)C(C)C 80296,Cc1nscc1C1CCCN1C(=O)NCCOCCNC.c1ccccn1 80297,C(=O)(C1=CC2CCCC12)Nc1ccc(NC(c2cc(C(C)=O)oc2)=O)cc1C 80298,C1(C)(NC(C(CCOC)C)=O)CCN(C(C2(C)CCC(C)C2)=O)CC1 80299,CC(C)CC(O)CC(=O)N1CC(C2CN(C(C3CC(O)CN3C)=O)C2)C1 80300,C1(C(=O)NCC2CC(F)C2)CC2CC1CN(C(=O)CCCC1CCC1)C2 80301,N1(C(C2(CC)CCCCC2)=O)CCC2CN(C(C3CC(C)CO3)=O)CC2CC1 80302,C1(F)(C(=O)NC(C)CO)CN(C(=O)CCc2cn(C)nn2)C1 80303,c1(C(N2C(CNC(C(C3CCOC3)OCC)=O)CCC2)=O)cncc(C(N)=O)c1 80304,C1(F)(CNC(C2C(C)OCC2)=O)CCN(C(=O)C(C)(C)Nc2ccccc2)CC1 80305,c1(OC)cccc(C(N2CC(CNC(c3cncc(N)c3)=O)CC2C)=O)c1 80306,C(=O)(C1(C)CCc2ccccc21)NC1CCN(C(CC=CCC)=O)CC1(C)C 80307,CC1COC2(C1)CN(C(C13CC1CCN3C(C13CCC(C1)C3)=O)=O)C2 80308,c1(CN(C(c2cncc(F)c2)C(=O)NCCCSCC)C)cccc(F)c1Cl 80309,C12(C(N3CCCC(NC(=O)CN4CCC(F)CC4)C3)=O)CCCC1C2(F)F 80310,c1(CC)c(C(=O)NCC(C2CCCC2)NC(=O)CNc2nccs2)cnn1C 80311,c1(NC(CNC(c2[nH]cc(CC)c2)=O)C2CCC2)cc(C(C)=O)c([N+](=O)[O-])cn1 80312,C1(NC2(c3n(CC(=C)C)c(-c4ccco4)nn3)CC2)CCC(C)(C)CC1CN 80313,C(=O)(C1=NOC2COCC12)N(CCCCCNC(c1cccn2cncc12)=O)C 80314,c1(OC)ncccc1C(N1CC(CN(C)C(=O)CC2CCCN2C(=O)CC)C1)=O 80315,C12(C(N3CC(CC=C)(NC(C4CC5(CC5)CO4)=O)C3)=O)CCC(CC)(C1)OC2 80316,N1(C(C(CC)=CCCC)=O)CCN(C(=O)C(N2CCOCC2)C)CC1C 80317,c1(C(=O)NC2CC(CNC(=O)C=Cc3cccs3)CC2O)csc2nccn12 80318,CC1CCC(NC(=O)COCc2nccn2C)CN1C(c1ccn(C)c1)=O 80319,C(=O)(C1=C(C)OCCC1)N1CCCC(C(C(NOC(CC)C)=O)(C)C)C1 80320,C(=O)(CCCCN(C)C)N(C1(C(=O)NC(C(=O)OC)C2CC2)CCC1)C1CC1 80321,c1(C(=O)NC2CC(CNC(C=Cc3n(C)cnc3)=O)C2)ccc2nccn2c1 80322,CCC(CC)(CO)CN=C(NCC1CC1(Cl)Cl)NC1CCC1 80323,C1(C(=O)NC2CC(NC(c3ccc(OC)o3)=O)C2)(OC)CCCOC1 80324,C(=O)(CC(CC)C(C)(C)C)N1CC(C(C)NC(c2cncc(C#C)c2)=O)C1 80325,C1(CC(=O)NCCC2CC(NC(c3cnc(CC)s3)=O)C2)CCC(=O)NC1 80326,C=C=CC(C)C(=O)N1CCC(CN(C)C(c2cc(CO)n(C)n2)=O)C1 80327,c1(C(C)C)cccc(F)c1C(=O)N(CCCNC(c1nncs1)=O)C1CC1 80328,C(C(C)(C)CC(=O)NC1CCN(C(c2ccnn2C2CC2(F)F)=O)C1)OC 80329,C1(C(=O)NCC2(OC)CCN(C(CCC=C)=O)C2)CC2(C1)CC(F)C2 80330,C(=O)(C(O)CC(F)(F)F)N(C(CC)C(=O)N1CC(NC(=O)OC)C1)C 80331,c1(OC)cc(N)ccc1C(=O)NC1CN(C(=O)CC2CCCC2O)C1 80332,c1(C(=O)NCC2CN(C(c3cc(C4CC4)cs3)=O)C2)ncn2cc(Cl)ccc12 80333,CCCCCS(=O)(=O)CC(=O)N1CCCC2(C1)CN(C(C1(CF)COC1)=O)C2 80334,CCC(C(O)C(=O)OC)NCCc1cc(C#N)c(Br)s1 80335,c1(C(=O)NCC(CC=C)NC(C2(Cl)CC2C(C)=O)=O)cc(C)nc(C)c1 80336,CC1(C)CC(NC(c2ccncn2)=O)CN1C(c1cn(C2CC2)nn1)=O 80337,C1(NC(C(C)(C)OC)=O)CCN(C(=O)C2=CCOC2)CC1O 80338,c1(CN2CCCC(C)(C(=O)Nc3cc(F)ccc3O)C2)cccc2nonc12 80339,c1(C(N2CC(C(C)NC(CC(CC)C)=O)C2)=O)cc2c(C)c(F)ccc2[nH]1 80340,C1(CC(=O)NC(C)CCNC(c2ccc(CC3CCCC3)o2)=O)CC2(CCC2)C1 80341,CC(C)(C(=O)N1CCCCC(CNC(=O)CC2(O)CCC2)C1)S(=O)(=O)C1CC1 80342,Cc1cc(C(=O)NC(C2CCN(C(C3CC3(C)C)=O)CC2)C)cc2nn[nH]c12 80343,c1(C(N2CCC(C)(NC(CCC(C)O)=O)C2)=O)cc2c(cn1)CCCC2 80344,Cc1ncnc(C(=O)NC2CCOCC2C(=O)NC2(C)CCSC2)c1C 80345,c1(C(=O)NCC2OCCN(C(C3CC(OCC)C3)=O)C2)cc2ccc(F)cc2[nH]1 80346,CC1C(NC(c2c[nH]cc2Br)=O)CCCN1C(=O)C=Cc1ccc(=N)[nH]c1 80347,c1(C(N(CCOCCCNC(CCSCC(C)C)=O)C)=O)cc(=O)cc(Cl)[nH]1 80348,n1(CC(=O)NCCN(C(=O)C(C)N(C)Cc2ccccc2)CC)ccccc1=O 80349,c1(C(N2CCC(C(C)NC(c3cc(C)nn3C)=O)C2)=O)cc2c(nn1)CCC2 80350,c1(OC)ccc2c(C(=O)NC3(C#N)CC4CCC3C4)coc2c1 80351,C1(NC(c2cc(C)nc(O)c2)=O)CC2CC1CN(C(=O)C=Cc1ccn(C)c1)C2 80352,Cc1nc(CN2CCC2(C)C(=O)NC(c2ccno2)C)co1 80353,c1(C(N2CC(NC(C(CC)(F)F)=O)C(SC)C2)=O)cccc2scnc12 80354,C(CS(=O)(=O)c1ccccc1[N+](=O)[O-])NC(c1ccc(F)cc1)CC 80355,c1(NC(CCSC)C(=O)OC)cc2c(cc1[N+](=O)[O-])CCC(=O)N2 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80859,CC1(C(N2CCOC(CNC(=O)Cn3cc(C4CC4)cn3)C2)=O)CC2CC2C1 80860,CCCC(CNC(=O)C(C(C)CC)N(C)C)C(=O)NCC(F)(F)C(C)(C)O 80861,Cc1ccc(-c2cc(F)ccc2CO)c2nc(C(=O)NCCc3ccc[nH]3)cn12 80862,N1(C(CNC(C2C(C)=CCS2)=O)=O)CC2CCCCCC2C1 80863,Cc1ccc(C(N2CCCC2(C)CNC(=O)CCNc2cncnc2)=O)cc1Cl 80864,c1(COC)nn(C)c(Cl)c1C(N1CCCCC(N(C(=O)C=CCO)C)C1)=O 80865,c1(C(N2CCCC(NC(COC(CC)(C)C)=O)C2C)=O)cnc(S(C)(=O)=O)s1 80866,c1(CNC2CN(C(c3cnc(SC)nc3)=O)CC(C)C2)cc(C)c(F)c(C)c1 80867,CC1CN(C(=O)COC2CCCC(C)C2)CC1CC(=O)NN1CC(CO)C1(C)C 80868,c1(NC(C(CC=CC)NC(C2CCCN2C=O)=O)=O)cnc(C)nc1C 80869,C1(OC)(CNC(C2SCCS2)=O)CCN(C(=O)Cc2cccc(Cl)c2)C1 80870,N1(C(C(C)OCC)=O)CC(CO)C2(C1)CN(C(=O)C(c1cnn(C)c1)O)C2 80871,N1(C(Cc2c(C)cccn2)=O)CC2CCC1C(NC(c1cc(N)ccc1F)=O)C2 80872,C1(NC(CC2(NC(CC3(C)CC3)=O)CCSC2)=O)CC2(CCOC2)C1 80873,Cc1noc(C)c1CSCC(=O)N(CC(C)NC(C1(O)CCOCC1)=O)C 80874,C=CCCC(C(=O)N1CC(c2nncs2)C1)NC(=O)C(C)CCCC 80875,C(=O)(CCCC(=O)N1CC(C2CC2)(C(=O)NC2(C)CCSC2)C1)OC 80876,C12(CO)CC(c3ccccc3)(C1)C2(F)F.N12CCN(CC1)C(=O)N1C(CCC1)C2=O 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80894,c1(C(N(C2CN(C(Cc3c(C)occ3)=O)C2)C)=O)ccn(C(C)C)c(=O)c1 80895,C12(C(=O)NCC3C(CNC(C4(CC#C)CCCC4)=O)C3)CCCC(CO1)C2 80896,C(=O)(C(CC1CCOCC1)NC(C1CNC(=O)N1)=O)NCC1C(CC)C1 80897,C(c1cc2ccccc2o1)=CC(N1C(C(=O)Nc2c(CC)cc(Cl)cc2)CC1)=O 80898,c1(CCC(=O)NC(C2CCC2CNC2CCN2c2ccccc2)=O)ccccc1F 80899,C1(CC(=O)NC(c2cccnc2)CNC2CC2c2ccco2)COCCO1 80900,C(=O)(C(O)C(C)C)NC1C(NC(c2ccc(CSC)o2)=O)CCC1 80901,C1(NC(C(=O)NCC(c2ccccc2O)OC)=O)CN2CCC1(C)CC2 80902,C(CO)(C(O)CCC)NC(C(CC1CCCC1)NC(CC=C)=O)=O 80903,CC#CCC(C(=O)N1CC=CC1CF)NC(c1ccc(CO)nc1)=O 80904,c1(C(NOCC(N2CCC(C(C)O)CC2)=O)=O)ccc(N)cc1[N+](=O)[O-] 80905,Cc1ncn(C)c(=O)c1C(=O)NCCC1CC(NC(=O)Cc2ccsc2Cl)C1 80906,C1(C(N(C(C)CCNC(C2CC2(C)C)=O)C)=O)CCOC2(CCCC2)C1 80907,C1(C(=O)NCC2(N(C)C)CCC2)CNC(=O)CN1C(=O)CC1(C)CCCCC1 80908,c1(C(=O)NCC2CCC(NC(C(=O)NCC)=O)C2)cc(C)ccc1N1CCCC1 80909,c1(CC(=O)NCC(CNC(c2ccc(CC)o2)=O)F)ccc(F)c(Cl)c1 80910,C1(CC#C)(C(=O)NC(CO)C(C)NC(c2cc(Cl)cs2)=O)CCCC1 80911,Cc1cncc(N(C2CC3CNC2C3)C(c2c[nH]cc(Br)c2=N)=O)n1 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81051,N1(C(c2c(C)n(C)nc2)=O)CC2CCCC2(NC(C2CC=CC(O)C2)=O)C1 81052,c1(C(N2CC(C3CC3)(C(=O)NOC3CCOC3)C2)=O)cccc2ccoc12 81053,CC(CC(=O)N(CCCCCNC(C1(O)COC1)=O)C)c1cccnc1 81054,C#CC1(O)CCCN(C(=O)C(C)(C)CNC(=O)CC2NC(=O)NC2=O)C1 81055,n1(CCNC(C(N2CC(C)(OCC)C2)=O)=O)c(C)cc2cc(F)ccc12 81056,C1(OC)CN(c2cc(NCc3ccc(F)cc3C)nc(C)n2)CCC1F 81057,C1(C(=O)NCC2CN(C(C3(C4CCCO4)CCC3)=O)C2)CCCOC1 81058,N1(C(c2ccc(C#N)s2)=O)CC2(C1)SCCC2NC(C1CC2CCCC(C1)C2)=O 81059,C1(NC(c2c(OC)nccn2)=O)CC12CCN(C(c1ccccc1I)=O)CC2 81060,N1(C(C(C)n2cccn2)=O)CCCC2(C1)CN(C(=O)CC1COCCO1)C2 81061,CC(C)C(C)(CNC(=O)CC1C2CCC(C2)N1C(C1CCCOC1)=O)C(C)C 81062,C(=O)(C(C)CCCC(C)=O)NC(CC#C)(C)C(=O)NC(C1(O)CCCCC1)C 81063,N1(CCNC(=O)CC2(F)CN(C(c3cc(CCO)on3)=O)C2)CCNC(=O)C1 81064,C12(CNC(C=CC)=O)C(NC(=O)COCCCOC)C3CC1C2C3 81065,c1(COC)nc(=N)[nH]cc1C(=O)NCCCNC(=O)C(c1ccccc1Cl)OC 81066,c1(COC)nc(NCCCNCC2CCCO2)cc(=NC2CCC(=O)NC2)[nH]1 81067,N1(C(c2c(CNC(C3(CC#C)CCCC3)=O)occ2)=O)CC(F)(F)C(F)(F)C1 81068,C1(CNC(c2scnc2C(F)F)=O)CCCCN(C(=O)CC2CCOCC2)C1 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81087,N1(C(CC2CCC(C)CO2)=O)CCC2(CC(C(=O)NC(C3CCCC3)C)C2)C1 81088,c1(C(=O)NCC2C(OCC)CN(C(=O)C(C)(C)C)C2)cc(C)c(C)cc1N 81089,C1(CNC(c2nnnn2-c2ccc(F)cc2)C(C)C2CC2)CCC(C(F)F)CC1 81090,N(C1CC2(CCOCC2)Oc2ccccc21)C(c1cccc(NC(N)=O)c1)=O 81091,N(C1CC2(CCN(C(=O)C(C)=C(C)C)CC2)Oc2ccccc21)C(C(CC)F)=O 81092,N1(C(=O)CC2CCC2)CCCC1C1CCCN1C(C1(c2ccccc2)CC1)=O 81093,N1(C(C2CCCC(=O)O2)=O)CCCC2(CCCN2C(C23CSCC2C3)=O)C1 81094,C(=O)(CC(C)(O)CCC)NC(CCCC)C(=O)NC1CC(C)N(C)CC1C 81095,N(C1CCc2ccc(C)cc21)NC1COCCN(C(C2CCC(CC)CC2)=O)C1 81096,Fc1cc(-c2ncc(CN3CCCC(CN4CCOCC4)C3)s2)cc(Br)c1 81097,N1(C(CCN(CC)CC)=O)CCCN(C(c2cc(F)cc(Cl)c2N)=O)C(C)C1 81098,c1(C(N(CCNC(Cn2c(=O)ccc(C)c2)=O)C)=O)cc(F)c(Cl)cc1F 81099,C1(CNC(COCCCC#C)=O)CN(C(C2CC(Cl)(Cl)C2)=O)CCC12CCC2 81100,C1(CC=C)(NC(C2CC2C(C)C)=O)CCCN(C(=O)C(C)(C)n2cnc(C)c2)C1 81101,c1(OC)cc(C)c(Cl)cc1S(=O)(=O)NC1C2CN(C(=O)Cc3cc(C)on3)CC12 81102,N1(C(c2cnc(C)[nH]c2=N)=O)CC2(CCN(C(c3cn(C)c(C)n3)=O)CC2)C1 81103,c1(OC)nc(C)ccc1C(=O)NC1(CO)CCN(C(=O)C(C)S(C)(=O)=O)C1 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81645,c1(OC)cccc(OC)c1C(N1C(C)C2CC1C2NC(c1cn(C)cn1)=O)=O 81646,CCC(CNC(C1CC2(C1)CC(O)C2)=O)(CC)C(=O)N(C)CCn1cncn1 81647,C(CCN=c1cc(Cl)nc(S(C)(=O)=O)[nH]1)N(C(=O)C(=O)NC1CCCC1)C 81648,Cc1ccc(Cl)c(C(N2CCC3(CC2)CC3NC(=O)C=CCO)=O)c1O 81649,c1(NC)ccc(C(=O)NCC(CC2CC2)C(=O)NC(C)(C)CC2CCCC2)nc1 81650,C1(C(N(CCN=[N+]=[N-])C)=O)CCN(C(=O)C2CC2(F)Cl)O1 81651,CC(C)S(=O)(=O)C(C)C(=O)NCC1(C(C)(C)O)CN(C(c2cn(C)cn2)=O)C1 81652,Cc1nc(C)c(C(=O)NC2CC(NCc3ccccc3OC(C)C)C2)[nH]1 81653,Cc1ccn(CC(=O)N(CCNC(=O)CN2CCCCC2)C(C)C)n1 81654,Cc1cc(=NC2CN(C(C3(C)CC3(F)Cl)=O)C2)[nH]cc1C#N 81655,C(=O)(C(C(C)C)NC(=O)CC(C)C)NCC1(NC(CC(=C)C)=O)CCOC1 81656,C#Cc1ccc(NC(c2nc(-c3ccnc(C(C)C)c3)cs2)=O)cc1 81657,C(=O)(CCCCCC(=O)OCCC)N(CC(C)NC(=O)C(C)=C1CCC1)CC 81658,CC1CCCCC1(CNC(c1ncc(F)cc1N)=O)NC(C1(F)CC1)=O 81659,C1(NC(CC(=O)OC)=O)CCN(C(=O)COCC(F)(F)F)C(C2CC2)C1 81660,c1(C(=O)NC(CNC(=O)CSC2CC2)C2CC2)cc(=O)c2ccccc2o1 81661,c1(NC(C(C2(C)CC2)NC(C2CC(c3ncc[nH]3)C2)=O)=O)cnc(C2CC2)cn1 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81679,C12(C(N3CCCC(NC(c4onc(CC)c4C)=O)C3)=O)CCCC1OCC2 81680,C1(NC(CCc2cc(C)on2)=O)C2CC3CN(C(c4nocc4C)=O)C1C3C2 81681,C1(NC(C(C(COC)C)C)=O)CC2CC(C1)N(C(=O)CCNC(c1cccs1)=O)C2 81682,N1(C(C2CC(C)C2)=O)CCCC2(CNC(=O)CCc3nccs3)CCCCC12 81683,c1(C(C)=O)cncc(C(N2CCCC(C3CCCCN3C(=O)C(C)C)C2)=O)c1 81684,CCCCC(O)C(C)C(=O)NCCCNC(=O)C(C)=CC(C)(C)C 81685,c1(NC(C23CN(C(=O)C(F)F)CC2CCO3)=O)ccc2ccccc2c1 81686,C1(C(C)(C)C)CN(C(c2cccc(Cl)c2N)=O)CCN1C(c1sccc1Cl)=O 81687,C12(OC)CC(CN(C(=O)C(O)C3CN(C(=O)C(C)C)C3)C1)C2 81688,C(=O)(CC(C(F)(F)F)OC)N(CCCCNC(C(CC)(CC)N(C(C)C)C(C)C)=O)C 81689,C1(CN(C(CC2(OC)CCCC2)=O)C)CCCN(C(=O)Cc2cnn(CC)c2)C1 81690,N1(C(C(C)SCCCC)=O)CCC(CCNC(=O)C(C)P(C)(C)=O)(OC)CC1 81691,N1(C(CCC(=C)C)=O)CCCC(C)(CNC(=O)C(C)Cc2ccccc2Cl)C1 81692,C1(CC(=O)OCC)CCC(C(=O)NCCc2cnn(CC)c2F)CC1 81693,CCC(C)(C)CCCC(=O)N(CCNC(c1c(C)nc(O)nc1C)=O)C(C)C 81694,CC(CC(=O)N1CCC(C(N2CCC(O)CC2(C)C)=O)C1)CC(C)(C)C 81695,n1(NC(c2n(CC)nnn2)(C)CNC2CCN(CC)C2=O)cnc2sccc2c1=O 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81785,C(C(C)C(F)C(=O)NOCC(=O)NC1CC2CC(=O)C1O2)NC(C)=O 81786,c1(N2CCC(CC)C2)ccc(S(=O)(=O)NC(C(C)(C)CO)C2CC2)cc1Br 81787,c1(CC(=O)NCC(C)(C)NC(C(CC)Oc2ccccc2)=O)nn(C)cc1Cl 81788,N1(C(c2c(C(C)C)ncnc2)=O)CCN(C(=O)C(O)C2CCC2)C(C)C1 81789,C1(NC(c2cc(C)nc(O)n2)=O)CC2CCC1N(C(c1cc(Br)n(C)n1)=O)C2 81790,C(CN=c1ccnc(C(C)C)[nH]1)OCCNC(C(CC(C)C)C)=O 81791,N1(C(CC(C=C)C)=O)CC(C)C(C)(CNC(=O)Cn2ncn(C)c2=O)C1 81792,c1(C(CNC(=O)C2CC2)NC(CNC(C)(C)C)=O)cc(C(N2CCCC2)=O)no1 81793,c1(SCC)cncc(C(=O)NCC(CNC(c2[nH]ccc2C2CC2)=O)CO)n1 81794,C(=O)(C(C)CCCC(C)C)N1CC(C(C(N2CCC(C(=O)OCC)CC2)=O)OC)C1 81795,c1(C(N2C(C(C)C)CNC(=O)C2)C(=O)NC2CC2)cccc2nc[nH]c12 81796,C(=O)(CCC(=O)N1CC2C(C(=O)O)C2C1)N(C)CCn1cncn1 81797,C(=O)(C(C(C)C)(C(C)C)NC(C)=O)NCCCN(C(C(C=C)O)=O)C 81798,N1(C(c2c(C)cn(C)c2)=O)CC2(C1)CN(C(=O)C(F)C(C)C)CC2CO 81799,c1(C(N(C(C)C(=O)NC(CCO)C(F)F)CCC)=O)ccc2[nH]ccc2c1 81800,c1(C(=O)OC)ccncc1NC(C1CCC(NC(=O)Cc2cc(C)no2)C1)=O 81801,C(=O)(C(C)(C)C(=O)NC1CCCN(C(=O)C(c2cnn(C)c2)C)C1)OC 81802,C#CCC(C)C(=O)NC1(CNC(=O)COc2cc(C)on2)CCCC1 81803,C1(NC(C2N(C)CCC2)=O)CN(C(c2cn(CC(F)(F)F)cn2)=O)C(C)(C)C1 81804,C1(C(=O)NCC2(C)CCCO2)CC12CCN(C(=O)C(C)(C)C(C)(C)O)CC2 81805,C1(COC)COCCN1C(=O)CN(C)C[Si](C)(C)C 81806,c1(C(N2CCCCC(Nc3cnc(C)[nH]3)C2)=O)ccccc1S(=O)(=O)N(C)C 81807,c1(N2CCC(NC(C(C)O)=O)(CF)C2)nc2c(cc1C#N)CCC2(C)C 81808,C1(C(=O)NC(C)C(CO)NC(c2cc(C(F)F)nn2C)=O)CCC(C)(C)C1 81809,C1(=O)C(C(F)(F)F)OC(=O)N(CC)CCN1.C=CCC(C)COC 81810,CC1CN(C(=O)CCS(=O)(=O)N(C)C)CCCN1C(=O)C1=NSC(C)C1 81811,c1(C(C)C)cc(C(=O)NCc2cn(C3CCN(C)C3)nn2)c(C(C)C)[nH]1 81812,N1(C(C(CC)CC)=O)CC(C2CCCN(C(C3CCCC3C)=O)C2)C1 81813,C1(OCCN(C)C)CCN(C(=O)C(=O)NCC2(C)CC2(C)C)CC1 81814,CC1CCC=C1C(=O)NC(C)CNC(=O)CSc1ncc[nH]1 81815,C1(CNC(c2cn(CCC)nc2)=O)CCC2(CN(C(=O)COC(F)F)C2)O1 81816,c1(OC)ccc(C(c2nnnn2C)NCC(c2ccncc2)N(C)C)c(Cl)c1 81817,c1(CC(C)NC(=O)CN2C(=O)NC3(CCCC3)C2=O)ccc(O)c2ccccc12 81818,C(=O)(C1=CCOC1)N(CCC(C)NC(Cc1n(C(C)C)cnn1)=O)C 81819,CCCCCCCCNC(=O)NC1CCCN(C(=O)C(=O)NCC(F)F)CC1 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81838,C1(CC=C)(NC(c2cn(C)nc2C)=O)CCCN(C(=O)C(=O)NCC(F)F)C1 81839,C1(CNC(c2cc(C)[nH]n2)=O)CC(F)CN1C(c1ccoc1Br)=O 81840,CCC(CC)C(=O)N(CC(C)(C)NC(c1cn(C(C)(C)C)nc1C)=O)C 81841,C1(NC(CCNC(C)=O)=O)CC2COCC(C1)N2C(c1cc(C)nc(O)n1)=O 81842,c1(C(=O)NCC=CCNC(=O)CN2CCNCC2)c(C(F)(F)F)cccc1Cl 81843,C1(OC)CCC2(C(N3CC(O)(C(C)NC(=O)C(n4nccc4C)C)C3)=O)CC12 81844,N1(C(c2n(C(C)C)cnc2)=O)CCC2(CCCCC2NC(=O)C2=CCC2)C1 81845,N1(C(C2CCC(=O)O2)=O)CC2(CCC2)CC1CNC(=O)C(F)n1cccn1 81846,C1(C(=O)NC(CC)CNC(=O)Cc2cc(F)ccc2Cl)CNC(=O)CC1(C)C 81847,CC1CN(C(=O)CCC2CC2)CC1CNC(c1cc(-c2cnn(C)c2)no1)=O 81848,C(=O)(CC(C)(C)CC(F)(F)F)N(CCOCCN(C(c1cc(C)sc1C)=O)C)C 81849,C(=O)(C(C)CC(C)C)N1CC(C(C)NC(c2ccc(SCC)nc2)=O)C1 81850,c1(COC)nc(C)c(C(=O)NC(CO)C(C)NC(C2CC2c2ccsc2)=O)s1 81851,c1(C(N2CCC(CCN(CC(=O)NCCCC)C)CC2)=O)cc(C)cc(Cl)c1 81852,CN1CCCC(F)(C(N2CCCOC(CNC(=O)CC3(O)CCC3)C2)=O)C1 81853,CN1CC(O)CCC1C(N1CCC(C)(C)C1CNC(=O)CCP(C)(C)=O)=O 81854,c1(C(N2CCCCC2Cc2c(-n3cc(CN)nn3)cccc2)=O)c(F)cncc1Br 81855,C1(NC(COCCOC)=O)CCCCN(C(C2CCOC2=O)=O)CC1 81856,N1(C(Cc2cn(CC)nc2)=O)CCN(C(c2cc(C)nnc2O)=O)CC(O)C1 81857,N1(CCOc2ccc(OC)cc2)CCOC(C)(NC(=O)C(C)OC)C1 81858,c1(OC)ccc(O)cc1C(=O)NC1CN(C(C2CC3C=CC2CC3)=O)CC1(C)C 81859,C(=O)(C1CCOc2ccccc21)NCC1N(C(c2cc(N)c(Cl)cc2)=O)CCC1 81860,c1(CC)cc([N+](=O)[O-])ccc1N(C(C)CNC(=O)C=C1CC2CCC(C1)N2C)C 81861,C(CCCCCNC(=O)CC1COC(=O)C1)N(C(=O)CSCc1ccccc1)C 81862,c1(OC)ccc(C(=O)N(C)C(C2CCOCC2)C)c(C(F)F)c1 81863,c1(CCC(=O)NCC(C(C)(C)C)NC(=O)CCc2ncc[nH]2)cccc(C#N)c1 81864,c1(C(=O)NC(Cn2cc(C3(COC)CCC3)nn2)C)ccc(Br)cc1 81865,c1(C(N2CCN(Cc3cncs3)C(C(F)(F)F)C2)=O)cnc2cc(Br)ccc2c1 81866,C1(CNC(C(C)(C)C(F)F)=O)CCC2(CN(C(C3CC4(C3)CS(=O)(=O)C4)=O)C2)O1 81867,CCCCC(C(=O)N1CCCC(CN(C(c2cn(C)nc2C)=O)CC)C1)C(C)C 81868,c1(CC)c(C(N2CCC(CC(=O)NCC3CC(C(C)(C)C)C3)C2)=O)ccn1C 81869,C1(O)(CNC(C2(CC=C)CN(C(=O)CCC3(C)CC3)C2)=O)CCOC1C 81870,c1(NC(C(=O)NC2(C)CCN(C(C3C(C)CC3)=O)C2)=O)ccc(Cl)c(F)c1 81871,CC1(NCc2cccc(C(=O)NCC(=O)NCC3CCCCC3)c2)CCCCO1 81872,C(=O)(CC(C)(C)Nc1cccnc1C)N(CCCC(=O)NCCC)C 81873,C1(N(C)C(C2CCC(c3ccccc3)C2)=O)CCN(Cc2cnccc2Cl)CC1 81874,C1(NC(c2nccc(C)n2)=O)CC2(CCN(C(C3COC(C)(C)C3)=O)C2)C1 81875,N1(C(CC2N(C(C(C)NC=O)=O)CC2)=O)CCC(C)C(C(N)=O)C1 81876,C1(CC(=O)NC(c2ccccc2C2CC2)C)CC2(CC2)CN1C(=O)C(=O)C(C)C 81877,N(C1CN(C(=O)CC(C)(C)NC(C)=O)CCc2ccccc21)C(CSC)=O 81878,N1(C(c2cnc(CC)[nH]2)=O)CC(CNC(=O)C(c2cncnc2)C)C(C)C1 81879,c1(C(C(=O)NC(CC)(C)C)N(C)C(c2cc(C)on2)C)ccc2c(c1Cl)OCO2 81880,c1(OC)c(N(C)C(c2nc(NC(=O)C#CC3CC3)sc2)=O)ccc2c1CCC2 81881,c1(OCC)cccc(C=Cc2nc(CN3CCCOC3=O)no2)c1OC 81882,c1(C(=O)NCCCCN(C(C(C)NC(c2cccs2)=O)=O)C)cccn(C)c1=O 81883,C(=O)(C(C)(C)CCSC1(F)CCCN(C)C1)NCCN1CC(c2ccccc2)(OC)C1 81884,C1(NC(C(C)N(CC(F)(F)F)C)=O)CC(C)CN(C(c2cc(Cl)c[nH]2)=O)C1 81885,c1(C(=O)NCCCN(C(C)=O)C)cnc2ccccn2c1=O 81886,C1(CNC(C2(C)CCCO2)=O)COC2(C1)CN(C(=O)Cc1cn[nH]c1)C2 81887,c1(NC)ccc(C(N2CCC(NC(=O)CC3C=CS(=O)(=O)C3)CC2C)=O)cc1F 81888,C1(CNC(CCCN(C)C)=O)COCCN(C(=O)C=CCNC(=O)OC(C)(C)C)C1 81889,c1(COC)cccc(C(=O)NCC#CCNC(=O)CSc2ccccn2)c1 81890,c1(-c2n(C(C3CCCCC3)C)nc(-c3cccnc3)n2)cnn2c1CN(C)CC2 81891,c1(C(N2CCCC(C)(NC(=O)C=CC3CCOCC3)C2)=O)cnc2sccc2c1 81892,C1(NC(=O)Nc2scc(C)c2)CCC(C)N(C(=O)C(C(C)C)c2ccccc2)C1 81893,CC(C(C)C(=O)N1CC(C)(F)C1)NC(c1ccc[nH]1)=O 81894,C(c1cncnc1O)=CC(=O)NC12CC(NC(c3c(C)oc(C(C)C)c3)=O)(C1)C2 81895,c1(C(=O)NCC(CC)NC(=O)C(F)(F)CN(C)C)cc(F)c(Br)c(C)c1N 81896,N#CCCCCCC(=O)N1CCN(C(=O)CCF)C(CCO)C1 81897,CC(C)(C(=O)N1CCC(O)(CCNC(C23CC(CCO2)C3)=O)CC1)C(F)F 81898,CCC(C)(CCC(C)C)C(=O)N1CCCC(CCNC(=O)C(OC)OC)CC1 81899,N1(C(C23CC2C3)=O)CCOC2(CCC(Nc3ncnc4[nH]ccc34)CC2)C1 81900,C1(NC(c2c(C)sc(O)n2)=O)CN(C(c2cc(F)cnc2O)=O)CCC1C 81901,C#Cc1cccc(C(=O)NCCC(C)(C)NC(=O)NC(c2ccccc2)=O)c1C 81902,c1(CN(C(=O)CC=CCNC(C2CC2C(=O)N(C)C)=O)CC)cncn1C 81903,N1(CC(C)(C)NC(C2N(CC)CCC2)=O)CCN(C(=O)Cc2scnc2C)CC1 81904,c1(C(c2nnnn2C)(C)NC(Cc2c(C)noc2C)C)ccc(Cl)cc1F 81905,CC(F)(C(=O)N(CCNC(C1CCCOC1)=O)C1CC1)c1ccon1 81906,C(=O)(C(C(C)O)NC(c1ccc(O)cn1)=O)N1CCC(CCC(=O)NC)C1 81907,Cc1nnc2n1CCN(C(C1CC(O)CN1C(=O)Cc1nccn1C)=O)C2 81908,S(=O)(=O)(C1CC1)N(CC(=O)N(C(C)C)CCN(C)C(C1C=CCC1)=O)C(C)C 81909,C1(CC)CN(C(C2CCS(=O)(=O)C2)=O)CCN1C(=O)Cc1cn(C(C)C)nn1 81910,N1(C(C2(CC#C)CC=CCC2)=O)CCC2(CCCCN(C(=O)CNC=O)C2)C1 81911,C(C(C)C(F)C(=O)NC(C)(C)C(C)C)NC(C1CC(C(=O)OC)C1)=O 81912,Cc1noc(C)c1C(C)C(=O)NCC(CNC(=O)Cc1cccnc1)CO 81913,c1(CC)nn(C)c(C(=O)NCCN(C(=O)C(CC)C(C)O)C2CC2)c1Cl 81914,C=CC(C)(C)C(=O)NCc1cccc(CN(C(=O)C(C)Cc2ccnn2C)C)c1 81915,c1(C(=O)NCC2CN(C(C=C3CCN(C)C3)=O)C(C)(C)C2)csc(S(C)(=O)=O)c1 81916,C(=O)(CC1=CCCCC1)NC1C(C(N2CC(C(C)(C)C)OCC2)=O)OCC1 81917,C1(NC(C=CC)=O)CC2CCC1CC2NCC1CCC(c2ccccc2)CC1 81918,S(=O)(=O)(CC(=O)NCCC1CN(C(=O)Cc2cc[nH]n2)C1)NC(C)(C)C 81919,C1(C)(CC(=O)NC2CN(C(C=C(COC)C)=O)C2)CC1(Cl)Cl 81920,N1(C(Cc2n(C)cnc2)=O)CCOCC(CNC(C2(C3CCCO3)CCC2)=O)C1 81921,Cc1noc(Cl)c1CCC(=O)NCC(O)CN(C)C(c1c(C)nnn1C(F)F)=O 81922,c1(N2CC(CC)OCC2)ncc(C)cc1S(=O)(=O)NCC(C)(C)n1cccn1 81923,Cc1oc(-c2ccco2)nc1CC(=O)NCC(C)(C)NC(=O)CNC=O 81924,c1(-n2c(COc3ccccc3F)nc(CC)n2)ccc(F)cc1OCC 81925,c1(C(N(CCNC(c2ccnc(CO)c2)=O)CC2CC2)=O)cccc(O)n1 81926,c1(C(=O)NCC2CN(C(=O)Cc3ccc(F)cc3)CCO2)cccc(Cl)c1Br 81927,C1(NC(C(=O)NC2(C)CN(C(=O)OC(C)(C)C)C2)=O)CCCCCC1C 81928,c1(CNCCCCC)ccc([N+](=O)[O-])cc1Cc1nc(OC)ccc1Cl 81929,N1(C(c2cnn(C)c2Cl)=O)CC2CCC(C(=O)NCC3=NOC4CCCC34)(C2)C1 81930,CCCC(C(=O)NC1CCCCC1CNC(c1cn(CCCF)nn1)=O)OCC 81931,C1(C(=O)NCCCC(C)NC(c2scc(C)c2Cl)=O)CCC(=O)C(C)C1 81932,N1(C(CC=CC)=O)CCCC2C1CCCN2C(c1cc(Br)cs1)=O 81933,c1(CN2CCC(CC(=O)NC3CS(=O)(=O)C3)C2)ccc(Cl)c(Br)c1 81934,C1(C(C)NC(C2CCCS2)=O)CCCCN1C(c1ccnc(O)c1)=O 81935,c1(C(=O)NC2(C#N)CCN(C(c3cc(O)no3)=O)C2)cccc2ncsc12 81936,C1(CC=C)(NC(=O)C(F)=C2CCC2)CCN(C(C2CC(=O)N(CCN(C)C)C2)=O)C1 81937,C1(NC(=O)Cn2nnc(C3CC3)n2)CCN(C(=O)C(c2ccccc2)F)CC1O 81938,C=CCC(CC(=O)NCCc1cnc(C)c(C)c1)NC(=O)COCC(=O)NC 81939,c1cnn(C)c1.C(CCCN1CCC1)N(C)C(=O)NCCOCCN(C)C 81940,Cc1cccc(NC(CN(C2(NC(=O)C(C)C3CC3)CC2)C(C2CCCC2)=O)=O)c1 81941,C(C(C)(C)CC(=O)N1CCCC1CN(C)C(c1c(C(F)(F)F)n[nH]c1C)=O)OC 81942,N1(C(c2c(C)scc2)=O)CCCC(O)(CNC(=O)C(C)OCC2CC2)C1 81943,FC(F)CCN=c1[nH]c2c(c(=NCc3ccnc(C(F)(F)F)c3)[nH]1)CSC2 81944,Cc1ccc(=NCCC(=O)NCCNC(c2cc3n(n2)CCN(C)C3=O)=O)[nH]c1 81945,n1(CC)ccc(C(=O)NCCCN(C(=O)C=C(C)C(F)F)C(C)C)c1C 81946,c1(C(CNC(C(CC)NC(C)=O)=O)NC(=O)CCN(C)C)cccc(C)c1 81947,C(C(=O)NCCCN(C(=O)C(F)CC)CCO)(C(C)C)N(CC)CC 81948,C(=O)(CCCC(C)CC)NCC1CN(C(c2c(C)cc(CC)o2)=O)CC12CC2 81949,C(CC(C)C(=O)NC(C)CC1CN(C(C2(CC)CC(C)(C)C2)=O)C1)=CC 81950,Nc1c(F)cc(-c2ccc(-c3nccn3C3CNC(CCO)C3)c(F)c2)cc1F 81951,c1(OCC)cnc(C(N2CCC(C)C2CNC(C2CCN(CC)C2)=O)=O)cn1 81952,C1(NC(CCCOC(C)C)=O)CCN(C(=O)CCSc2ccccc2Cl)CC1C 81953,C1(C(N(CC(C)NC(C2C(C)OCCC2)=O)C)=O)CCCC2C1C2(F)F 81954,O(NC(=O)C(C1(O)CCCCC1)NC(=O)CCC(C)C)C(C=C)C 81955,c1(OC)ccc(F)c(C(=O)NCCC2CCCCN2C(c2csnn2)=O)c1Cl 81956,C1(CC(=O)N(CCC)C)CCCNC(=O)C1.C1CC(=O)N2CC(C2)CNS1 81957,c1(CNC(=O)NC2C(c3ccc(C)o3)C2)cccnc1N1CCCC1 81958,n1(CC)c(C)cc(C(N2CCCC(NC(=O)CCCCCF)CC2)=O)c1C 81959,c1(CNC(C2(CCCC)CC2)=O)cccc(CO)n1 81960,C12(CNC(c3cc(CCC)nc(O)c3)=O)CCC(CC1)N(C(=O)C(F)=C(C)C)C2 81961,C1(CC(N2CC(COC)(NC(=O)C=CCO)C2)=O)CCOCC1(C)C 81962,N1(C(c2cc(CC)no2)=O)CCN(C(c2ccn(CC(C)C)n2)=O)C(CCO)C1 81963,Cc1cccc2c1ccn2CC(=O)N(C1CN(C(=O)C(F)C(F)(F)F)CC1O)C 81964,N1(C(=O)Cc2cnsc2)CCN(C(C2C3CNC(=O)C23)=O)C(c2ccccn2)C1 81965,Cc1c(C(=O)NC2CCC2CNC(=O)CCS(C)(=O)=O)sc2cncn12 81966,c1(OC)ccnc(C(=O)NCC(O)CN(C(=O)C=Cc2ccnn2CC)C)c1N 81967,CCC(CCC(=O)NC1CCN(CCCNC(=O)Cc2cncn2C)C1)OC 81968,c1(C(=O)NCC(C)N(C(c2cc(C)cs2)=O)CC)cc(O)n(C)n1 81969,N1(C(c2c(COC)cccc2)=O)CCN(Cc2cc(C)sc2C)C2CC12 81970,N1(c2nnc(CC)s2)CC(F)(F)CC1(C)C(=O)NCC1C(C(F)(F)F)C1[N+](=O)[O-] 81971,CC1CCC(C)(C=CC(=O)NC2CC3(CCN(C(C4(C)CC4)=O)C3)C2)C1(C)C 81972,c1(C(=O)OC)cc(Cl)ccc1NC(C)C(=O)OC(c1ccc(C(C)(C)C)cc1)C 81973,c1(CC)cccc(C(N2CCCC2CCCNC(=O)C(O)C(C)(C)C)=O)c1N 81974,c1(C(C)NC2CCCN(C(=O)Nc3ccco3)C2)ccc(F)c(Cl)c1F 81975,c1(CC(=O)NC23CCN(C(C4(F)CC4)=O)CC2C3)cnc2ncccn12 81976,C1(CNC(c2n(C=C)ncc2)=O)CN(C(C2(C#N)CC3CC3C2)=O)CCN1C 81977,C(CCCC(C)(C)C(=O)NNC(=O)CC1CCC(O)C1)CNC(CC(C)(C)C)=O 81978,c1(CNC(C(C2CCOC2)NC(C(F)=CCC)=O)=O)ncnn1C 81979,C12(NC(C(C)n3cccn3)=O)CCC(C(N3CCCC(O)C3)=O)(CC1)C2 81980,C(=O)(CC(O)C1CCCC1)N1C(CNC(=O)Cc2csc(Br)c2)CC1 81981,c1(NCC(c2ccc(C)cc2)NC(C2C(C(C)=O)C2)=O)nc[nH]c2ncnc1-2 81982,N1(C(c2ccc(N)cc2Cl)=O)CCN(C(C2CC3CC3C2)=O)C2CS(=O)(=O)CC12 81983,C1(CC(=O)N(C)CC2CN(C(=O)C(C)(C)n3cccn3)C2)(OC)CCCCC1 81984,C(=O)(C(C)CC(N)=O)N1C(CC(=O)NCc2n[nH]c(C)c2C)CCCC1 81985,N1(C(Cc2c(C)ccc(F)c2)=O)CC(=O)N(C)CC1Cc1ccc(Cl)cc1 81986,CC(C)(C)CCCC(=O)NC1(C)CCN(C(C2(C)CCCO2)=O)C1 81987,N1(C(C(OC)OC)=O)CC(=O)NCC1C(=O)NCCOCCCF 81988,c1(C(N2CC3CN(C(C(CCC)O)=O)CC32)=O)ccc2cnn(C)c2c1 81989,c1(CNC(c2nccc(OC)n2)=O)ccc2c(c1O)CCC2 81990,C1(NC(c2cnc(CC)o2)=O)CC(NC(=O)CCc2nc(C)c(C)[nH]2)C12CCC2 81991,C(=O)(C1CCCc2nn[nH]c21)N(C)CC1CCN(C(CCNC(=O)NC)=O)C1 81992,N1(C(CCSC)=O)CC2C(CNC(=O)Cc3scnc3C)C2C1 81993,Cc1c(F)ccc(C(N2CCOC(CNC(C3(C)C=CCC3)=O)C2)=O)c1Cl 81994,CCC(CC)CCC(=O)NC1CCOC(CNC(=O)Cc2ccc(Cl)nc2)C1 81995,N1(C(CCCCC)=O)CCN(C(C2CC(=O)N2)=O)C2(CCC2)C1 81996,c1(N(C)C)ccc(C(=O)NC2CCC2NC(c2ccncc2F)=O)cc1[N+](=O)[O-] 81997,O=C(NNc1nc[nH]n1)c1ccc2n[nH]cc2n1 81998,C1(NC(c2cnc(CC(C)C)[nH]2)=O)CCSC12CN(C(=O)CCc1nc[nH]n1)C2 81999,C1(C(N2CCCC(OC)C2)=O)COCCN(C2CCCC(C)C2)C1 82000,c1(CC)ccc(CCCC(=O)NC2CCN(C(C3CC34CCC4)=O)C2)cc1 82001,c1(N2CC3C(NC(C(CC)CCOC)=O)C3C2)c(Br)cccc1[N+](=O)[O-] 82002,C1(CC)CCC(O)(C(=O)NCCN(C(=O)CS(C)(=O)=O)C2CC2)C1 82003,n1(CC)nc(-c2ccc(OCc3ccccc3Cl)cc2)nc1C1CCCCC1C 82004,C(N=c1[nH]c(C)ncc1F)C1C(NC(Cc2c(C)cccn2)=O)C2(CC1)CCC2 82005,N1(C(Cc2cnc(C)o2)=O)CCCC2(CCC(NC(C3(C)CC(F)(F)C3)=O)C2)C1 82006,C1(C(=O)NC2CC(C(=O)NC(C(C)C)C)C2)(CF)CCOCC1 82007,Cc1cc(N)ccc1C(N1CCC(O)(CCNC(c2ccnc(CO)c2)=O)C1)=O 82008,c1(C(=O)NC(CCSC)C(=O)N2C3CSCC2C3)cc(C)c(F)cn1 82009,C1(C(=O)NC2(C)CN(C(=O)CCC3CCOC3)C2)CC(O)CN1c1ccncn1 82010,N1(C(C2CCC(CNC(CC(C)F)=O)C2)=O)CCOC2(CCCC2)C1 82011,C1(CCNC(N2CC(c3ccc(Cl)nc3)C2)=O)CCC2(CCC2)O1 82012,C(=O)(CC(C)(C)CC(=O)NCC=CCNC(C1CCC1(F)F)=O)OCC 82013,c1(COC)nc(C)c(C(=O)NCC2(CC(N3CC(F)CC3CO)=O)CC2)o1 82014,N1(C(COC(CC)C)=O)C(CNC(c2ccc(C)nn2)=O)CC2COCC12 82015,N1(C(c2cc(OC)no2)=O)CCCCC1C1(NC(=O)CCc2cncnc2)CC1 82016,N1(C(c2c(N)ccc(CC)c2)=O)CCOC2CCN(C(=O)CC(F)F)CC12 82017,CC(CC(F)F)C(=O)NCC1CCCCN1C(=O)CCCNC(N)=O 82018,c1(OC)cccc(C)c1C(=O)NCC1CC(OC)CN1C(c1cc(N)ccn1)=O 82019,c1(OC)cc(F)c(S(=O)(=O)Nc2ccc(F)cc2OC(C)C)cc1F 82020,n1(CCOC)cccc(C(N2CCOC(C3CCCCC3)C2)=O)c1=O 82021,C1(CC#C)CCN(C(C2CCC(NC(=O)CCC3CC3C)CC2)=O)CC1 82022,C1(C(N(CCNC(CC2C(C)CCC2)=O)C)=O)COCCN1C=O 82023,N1(C(C2CCN(Cc3ccc(C#N)s3)CC2)=O)CC2CCC(C1)O2 82024,c1(N(C)CC2CCN(C(Cc3cccc(SC)c3)=O)CC2)ncc(Br)cc1C#N 82025,C12(C(=O)NC3(C)CC(NC(C(C)Cc4ccncc4)=O)C3)CCC(C1)OC2 82026,N1(C(C2(CCC=C)CN(C(C3C4C5CCC(C5)C34)=O)C2)=O)CC(O)C(C)(C)C1 82027,c1(OCC)ccc(CC(=O)NCC2CN(C(C3CN(C)C(=O)N3)=O)CC2C)nc1 82028,c1(C(C)C(=O)NCC2(NC(=O)C(C)SC(F)(F)F)CCC2)ccc(N)cn1 82029,C1(C(=O)NCC(CNC(=O)CCc2ccc(Cl)cc2)O)NC(=O)C2CCC12 82030,N1(C(c2cnc(OCC)nc2)=O)CC2CC(NC(C3CN4CCC3C4)=O)C2C1 82031,c1(SCC(=O)NC(C)C(C)NC(=O)CCn2ccnn2)ccc(F)cc1 82032,c1(C(=O)NC(CCC)CO)cc(F)ncc1NCc1ccnc(Cl)c1Br 82033,C1(C(=O)NCCC(CCC)O)C2CCC(C2)N1C(c1coc(N(C)C)n1)=O 82034,C(=O)(CC(C)(C=C)CC)NCC(CC=C)NC(=O)CCCCCOCC 82035,N1(C(COC(C)C)=O)CCC(O)(CNC(=O)CCc2cnn(C)n2)C1 82036,Cn1cc(C(=O)NCC2(F)CCN(C(c3cc(N)ccn3)=O)C2)nc1O 82037,C1(OC(c2cncc(OC(C)(C)C)n2)=O)CCC=CCCC1 82038,C(c1cccc(Cl)c1)=CC(=O)NCCCOCCCNC(C1(C)CC1)=O 82039,C1(NC(C(C)C)=O)CN(C(=O)C(c2ccccn2)O)C2(CCOCC2)C1 82040,N1(C(Cc2ccc(OC)nc2)=O)CC(NC(=O)Cn2cccn2)CC12CCOC2 82041,c1(CC(=O)NC2CCCC(CNC(C=CC=CC)=O)C2)ccc(C#N)nc1 82042,CC1CCOCC1C(=O)NCC1(C(=O)NC2CC(=O)N(O)C2)CCCCC1 82043,c1(CC(N2CC(CCCC)N(C(=O)C(C)CCC)CC2)=O)cnn2c1CCCC2 82044,O=S(=O)(c1ccc(Br)cc1NC1CCSC1)NCCCCCOC1CCOCC1 82045,c1(C(CNC(C2CCCC2)C)O)ccc2c(c1)CCCC2 82046,C1(CC(=O)NC(Cc2cn[nH]c2)C(=O)NCCN2CCOC2=O)CCCNC1=O 82047,C1(C(=O)NC2CC(NC(c3ccc(C(N)=O)cn3)=O)C2)C(F)(F)C12CCC2 82048,c1(C(C(=O)NC(C)CC)N(CC(=O)NCC)C)ccc(CC)o1 82049,C1(CC(N2CCC(O)(CNC(=O)COc3ccsn3)C2)=O)CC2(CCCC2)CO1 82050,c1(CC(N)=O)cccc(NC(=O)CC(=O)NCC2(C(O)C(F)(F)F)CCC2)c1 82051,c1(C(=O)NCc2ccc(C(C)NC(C(C)(C)SC)=O)cc2)ccc2nn[nH]c2n1 82052,N1(C(c2cc(C)no2)=O)CC(C)N(C(=O)CN(C(=O)C(C)C)C)C(C)C1 82053,C(N=c1cccc(S(=O)(=O)NC2CCCc3occc32)[nH]1)C1C(C)(C)C1 82054,c1(-c2ccn(C)n2)cc(C(=O)Nc2cc(Cl)nc(Cl)c2)cc2cc[nH]c12 82055,Cc1cc(C(=O)NCc2n[nH]cc2C(=O)N(C)Cc2cnn(C)c2C)c(C)nn1 82056,N1(C(c2c(OC)cc(Br)c(C)c2)=O)CCC2(CCCC2C(=O)N(C)C)C1 82057,N1(C(c2cn(CC=C)nc2)=O)CCC(C)C(NC(=O)CC(C)(O)C2CC2)C1 82058,c1(NC2C(C(=O)OCC)CNCC2)ccc(-n2cccc2)c(Cl)c1 82059,c1(OC)nc(C)c(C(C)OC(C2CC(C)(C)C2)=O)s1 82060,C(=O)(CCC(=O)NCCC1(C(=O)N(C)Cc2ccn(C)n2)CC1)NCCC 82061,c1(C(N2CC(O)CC2C)C(=O)NC(CC)C)cc(C)c(Br)s1 82062,c1(NC(C2CC(C(=O)Nc3cc(C(C)(C)C)[nH]c3)C2)=O)c(O)cccc1Cl 82063,c1(C(=O)NC(C(=O)NC2(CO)CC(C)C2)c2cccs2)cc(C#N)cs1 82064,CC(Cn1cnnc1)N=c1[nH]c(=NC2CCn3c(O)nnc3C2)[nH]c2cc[nH]c12 82065,c1(C2(C(=O)NCC3C(CCC)CN(C(=O)C(C)O)C3)CC2)ccc(F)cc1F 82066,C1(NC(c2ccnc(C)n2)=O)CCCN(C(c2cc(C(C)(C)C)on2)=O)C1C 82067,C1(NC(C2CC(OC)C2)=O)CCN(C(c2cc3n(n2)CCC3)=O)C(C)C1 82068,C1(NC(C(COC)C)=O)CC2(CCCCN2C(C2CCCN2c2nccs2)=O)C1 82069,C1(CNC(Cc2ccc(SCC)cc2)=O)CCCCN(C(C2OCCCO2)=O)C1 82070,CC1(C)C=C(C(=O)NC(=O)Nc2cncc(Cl)c2Br)C1.C(C)(C)(C)O 82071,C1(CNC(c2c(C)cnn2C(C)C)=O)CN(C(=O)CCCC2CC2C)CC1(F)F 82072,c1(C(N(CC(C)NC(C2COC3(CCC3)C2)=O)C)=O)ccc(N)c(CC(C)C)c1 82073,C1(=Cc2n(CCC)ncc2)SC(=S)N(CC(c2c(C)cccc2C)=O)C1=O 82074,C1(C)(NC(CN(C)C)=O)CCC(NC(=O)CCC2CC(C)(C)CO2)CC1 82075,COn1cnc(C)c1C(N1CC(NC(C2CCC2(C)C)=O)C(O)C1)=O 82076,CC1(NC(=O)Cc2csc(S)n2)CCCN(C(C2CCCC2(F)F)=O)C1 82077,N1(C(COCC=C)=O)CC(CNC(c2cc(OCC)n[nH]2)=O)CC1C 82078,CN1CC(C)(C(=O)NCCCCC(CO)NC(c2ccc(F)cc2F)=O)CC1=O 82079,C(CNC(=O)Cc1cccs1)(CC(=O)NCCC1CC(F)C1)OC 82080,n1(CCCCC)cc(COC2CCN(C(C3(CF)CC(=O)C3)=O)C2)nn1 82081,C1(OC)CC2CCC1CC2C(=O)O.c1(CC2CN(C(=O)C=C(Cl)Cl)C2)ccc(F)cc1 82082,c1(CSC)cccc(OCC(=O)NCC2(CC(=O)OC)CC2)c1 82083,c1(C(N2CC3CCN(C(C4CC(C)(O)C4)=O)CC32)=O)cnc2ccc(F)cc2c1 82084,C1(CNC(C2(OC)CCCCC2)=O)CC2CN(C(C3CCN(OC)CC3)=O)CC12 82085,c1(CN(C(C(COC)O)=O)CCNC(=O)Cn2ccnc2C)ccc(F)cc1 82086,C12(CNC(c3c(OC)nn(C)c3)=O)CCC(CC1NC(=O)CC1CC(F)(F)C1)C2 82087,c1(C(C)OC(c2cnn(C)c2)C(=O)NC)cc(Cl)c(N=[N+]=[N-])cc1OC 82088,C(=O)(C(CO)C(F)(F)F)NCC(C1(O)CCCCC1)(CC)C 82089,c1(C(N2C(CC(=O)NCCCc3cc[nH]n3)COCC2)=O)occ2c1CCC2 82090,C1(CNC(CN(C)C2CC2)=O)CN(C(=O)CC2NC(=O)NC2=O)CCC1(C)C 82091,C1(C(C)NC(=O)C(C)(C)C2CCCC2)CN(C(C2COCCO2)=O)CCO1 82092,Cn1cc(C(N2CCN(C(=O)COC3(C)CCCC3)C(C3CC3)C2)=O)ccc1=O 82093,C1(C(N2CCC(=C)C2)=O)C=CCCN1C(=O)CN(CC(C)(C)C)C 82094,C1(CC(=O)N(C)CC2CCCCN2C(C2CCCS2(=O)=O)=O)CCC2(CC1)CC2 82095,c1(SC)nc(N2CCC(NC(=O)CSCCN(C)C)C(F)C2)c(C)c(Cl)n1 82096,Cc1sncc1C(=O)NCC(C)C(=O)NCCNS(N)(=O)=O 82097,c1(C(=O)NC(C2CN(C(=O)COC(C)(C)C)CCO2)C)noc2cc(F)ccc12 82098,C1(C)(NC(C(n2cc(CCN3CCCCC3)nn2)C)=O)CCC(=O)NC1.N(C)C 82099,N1(C(C(C(C)(C)C)CO)=O)CCC2C(CCN2C(c2cc(C#N)c[nH]2)=O)C1 82100,c1(C(N(C)CC2CCCN(C(c3csc(O)n3)=O)C2)=O)nn(C)c(Cl)c1Cl 82101,C(C1CCCN1C(=O)C(C)n1ccnn1)=CC(=O)NC1(C(COC)O)CC1 82102,CN=c1[nH]cc(C(N2CCC(OCCNC(c3cc(C(N)=O)co3)=O)C2)=O)s1 82103,C1(C(=O)NC(CN(C(CCOCC#C)=O)C)CC)CCOC1(C)C 82104,C(CC(=O)N1CC2=C(C1)CN(C(c1nccn1C)=O)C2)(C1=CCCC1)OCC 82105,C(C(C(=O)NCc1cscn1)NC(=O)C(n1ccc(C)n1)C)OC 82106,C12(C(=O)NCCOCCCC)CCC(CC1NC(=O)C(C)CCOC)C2 82107,C1(NCC(=O)NCC2(CNC(C=CC(=O)N(C)C)=O)CC2)CC1 82108,C1(C(C)NCC(=O)Nc2ccc(Cl)cc2Cl)CC(=O)N(C)C1c1ccccc1 82109,C(N=c1nc2c(cnn2C)c(NCCc2cc(C)no2)[nH]1)C1(OC)CCCSC1 82110,C1(CC(=O)NC)CN(C(c2ccc(C)nc2OC)=O)CCN1C(=O)C1CC1 82111,N1(C(CCCNC(=O)OCC)=O)CC=CC(NC(C2C=CC2C(N)=O)=O)C1 82112,c1(CC)nscc1NC(=O)C(=O)N(C)CCSc1ccccc1 82113,CC(C)C(C(=O)NCCCNC(=O)Cc1cccn1C)c1cccc(Cl)c1 82114,C1(C(N(CCC=C)CC)=O)CCN(C(=O)C(C)CC=CC=C)C1C(C)C 82115,C12(CC)CN(C(c3ccnn3CC(F)F)=O)C(CNC(C3CC(C)=NO3)=O)(C1)C2 82116,N1(C(Cc2cn(C)nc2)=O)CC(CNC(=O)CCNS(C)(=O)=O)C(C)(C)C1 82117,N1(C(C(c2cnn(C)c2)OC)=O)CC2(CCN2C(c2ccc(Cl)c(C)c2)=O)C1 82118,c1(C(=O)NCC2N(C(C(C=CC)O)=O)CC2)ccc2c(c1)B(O)OC2 82119,C(=O)(CCCCCNC(c1cc(Cl)n[nH]1)=O)NCCCS(C)(=O)=O 82120,CC1C(C(N2CCC(C(CO)NC(C3CCS3(=O)=O)=O)CC2)=O)CCN1C 82121,c1(CC)conc1CC(=O)NC1C(C(=O)NCC2CCCC2CF)C1(C)C 82122,S(=O)(=O)(c1ccc(Br)c(C)c1C)NSc1c(C)n(C)nc1C(c1ccccc1)C 82123,c1(C(=O)NC(C)CCN(C)C(C2CC2F)=O)cn(C)c2c(Cl)cccc12 82124,C1(CCOC)(NC(c2ccc(CC(C)(C)O)s2)=O)CCN(C(c2ccc[nH]2)=O)C1 82125,CC1C(C)N(C(=O)Cn2cc(C3CC3)nn2)CCN1C(C1CC(C)(C)CCO1)=O 82126,c1(N(C)C)cccc(C(=O)NC2CCN(C(=O)Cc3csc(Cl)c3)C2C2CC2)n1 82127,N1(C(Cc2c(OC)nccc2)=O)CC(N=c2[nH]c(Cl)ncc2OC)CC1C 82128,c1(NC(C(=O)NCCC(C)(C)OC)=O)cnc(OCc2nccs2)cc1C 82129,c1(C(=O)NC(CCNC(C(C(=O)OCC)(C)F)=O)C)cc2cnccc2o1 82130,CC1(C(=O)NCCC2CN(C(=O)CNC(c3cccs3)=O)C2)CC=CCO1 82131,C1(CNC(c2cnc(C)s2)=O)CC(C)(C)CN1C(C1CCCC(O)C1)=O 82132,c1(C(=O)NC2C=CC(CNC(=O)CN3CSCC3=O)C2)cc2cc(F)ccc2o1 82133,c1(C(=O)NCC2CCN(C(C(CN(C)C)(F)F)=O)C2)cnc2c(cnn2C)c1O 82134,c1(C(N2C(C)(CNC(c3nc(C(C)OC)sc3)=O)CCC2)=O)cnc(C)c(C)c1 82135,N1(C(c2ccc(F)cc2F)C)CC2CN(C(=O)C(C)(C)CC(F)F)CC2C1 82136,C1(CNC(CCNC(C)=O)=O)C2CCCC1N(C(c1ccc(C)s1)=O)C2 82137,Cc1c(C(=O)NC2CN(C(=O)CO)C3(CCC3)C2)ccc(Br)c1Cl 82138,C(=O)(C1=CC2(CCN(C(c3cc(C)c(C)o3)=O)C2)C1)NCc1cc(C)sc1 82139,CC1(C(N2CCN(Cc3cnc(-c4ccccc4)[nH]3)CC2)=O)CCOCC1 82140,n1(CC)nc(-c2ccc(Br)cc2)nc1C.C1(S(C)=O)(CN2CCC2)CC1 82141,N1(C(C2(CC)CC2)=O)CCC2(CC1)OCCC2NC(=O)CNC(c1cccs1)=O 82142,c1(C(=O)NCC(C)NC(=O)C(C(C)O)NC(=O)C(C)(C)C)cc(F)c(F)cc1O 82143,N1(C(C)C(N)=O)CCCC(CCNC(C2(C)CCC2)=O)C1 82144,C12CN(C(c3cc(C(C)=O)c(C)o3)=O)CC1C(=O)NOC2=O.C1(CCC)CC1CC 82145,C1(C(=O)NCC2CCCOC2)(CNC(=O)CCc2cnoc2)CCCCC1 82146,c1(-c2c(C)n[nH]c2C)ccc(=NCc2cc(Cl)cnc2Cl)[nH]c1 82147,c1(C(=O)NC(C(C)NC(c2nc(COC)sc2)=O)C(C)C)cc(=N)[nH]c(Cl)n1 82148,C1(CNC(CS(CC)=O)=O)CCC2CN(C(c3cn4ccccc4n3)=O)CC12 82149,c1(C(N2CCCC(CN(C(C(C)C3CC3)=O)C)C2)=O)coc2c1CSC2 82150,n1(CCCN(C(C)=O)C)cc(CNC(C2CCC(ON(C)C)C2)=O)nn1 82151,C(C1CCN(C(C2CN(C)C(=O)N2)=O)CC1)=CC(=O)NC1C(OC)C(O)C1 82152,c1(NC(C2CC(C)(NC(=O)CCC3NC(=O)NC3=O)C2)=O)ccc(O)nc1 82153,O=C(N=c1[nH]nc(-c2cccnc2)s1)NC1CCC(OC(F)(F)F)CC1 82154,C(=O)(NNC(=O)CC(C)(C)C)OC1CCCC1.C(=O)(NOC1CN1)OC(C)(C)C 82155,N1(C(C(=O)NCCOCCOC)=O)CC(CNC(c2scnc2Cl)=O)C2CC12 82156,C(CCC(O)C(=O)NC1(c2ncc(C)o2)CC1)NC(CCn1ncc(C)c1)=O 82157,c1(C(N2C(C(=O)NCCCc3ccsc3)CC(OC)C2)=O)ccc(C)cc1O 82158,C1(OC)(CNC(=O)CSC2CCOC2=O)CCN(C(c2nccn2C)=O)C1 82159,c1(C(=O)NC2CCN(C(=O)Cc3cnn(CC(F)F)c3)C2)ccc(F)c(F)c1 82160,C1(NC(C)=O)CC2CC(NC(c3cnc(C)[nH]3)=O)C1C2 82161,c1(C(=O)NCCCCNC(C2C(SC)CCC2)=O)cc(C(F)(F)F)ncc1Cl 82162,C12(CC(=O)NC3C(CNC(=O)CCN4CCOC4=O)C3)CCC(CC1)C2 82163,CCC1=NOC(C(N2CC(NC(=O)COCc3cc(C)no3)C(C)C2)=O)C1 82164,C1(C(=O)NCC23C(CN(C(c4cccc(C)c4Cl)=O)C2)C3)CCn2nccc2C1 82165,N1(C(C(COC)OC)=O)CCN(C(c2cc(=O)n(C)cn2)=O)CC1C1CCC1 82166,c1(C(N(C)CC)=O)ccc(SCCC(C)N)cc1 82167,Cn1c(C(N2CCCN(C(=O)CN3CCCCC3)CC2)=O)cc2c1CCOC2 82168,Cn1nnc2c1C(C(=O)NCC(C1CCC1)NC(C1(C(F)(F)F)CC1)=O)CCC2 82169,CCCC(CC(C)C)C(=O)N1CC2CC(C)N(C(=O)CCC(C)CN(C)C)C2C1 82170,C(=O)(CC(C)CC(C)(C)C)N1C(CNC(C2=C(C)OCCC2)=O)CC(C)(C)C1 82171,C1(NC(=O)C(C2CCCCCC2)O)COCCN(C(C2CC3C(C2)C3(F)F)=O)C1 82172,c1(C(N2C3CC(CC(NC(CC)=O)C3)C2)=O)cnc2snc(C)c2c1 82173,c1(-c2cn(CCN(C(C3CN(C)CCO3)=O)CC)nn2)cc(Cl)cc(Cl)c1 82174,O=C(C1CCc2cccc(Cl)c21)NCC1(F)CC1 82175,N1(C(C(Br)=C(C)C)=O)CC(C2CCCN(C(c3cnc4sccn34)=O)C2)C1 82176,c1(C(C(=O)NCc2cccs2)N(C(CCSC)C)C)nnc2n1CCN(C)C2=O 82177,C1(CNC(C2CC(OC)C(OC)C2)=O)CCCCN(C(c2c(N)cnn2C)=O)C1 82178,N#Cc1ccc(=NC(=O)OCCNC2CCC(Oc3ccc(F)cc3)CC2)[nH]c1 82179,c1(C(=O)NC(CCCC)CNC(c2cn[nH]c2)=O)ccc(C(F)(F)F)nc1OC 82180,C1(C(=O)NCCS(CC)(=O)=O)COCCN(c2ccc(Cl)c(NC(C)=O)n2)C1 82181,C1(CC(=O)N(C)Cc2cn(CC)nc2)CCCN(C(c2cccnc2C)=O)C1 82182,Cc1cc2ncc(C(N3CCC(O)(CN(C(=O)C(C)CO)C)CC3)=O)cn2n1 82183,N1(C(c2nc(OC)c(F)cn2)=O)CC2CCC(C1)N(C(=O)Cc1ncc(C)o1)C2 82184,C(=O)(CCCCNC(N)=O)NC1CCC(CNC(CC2(C=C)CCC2)=O)C1 82185,c1(OC)ccc(S(=O)(=O)N2CCCCC2c2nc(=O)o[nH]2)cc1C(=O)O 82186,c1(-n2cc(C3(C)CCCN3C(=O)Cc3csnn3)nn2)cc(Cl)ccc1CO 82187,c1(CN2C(C(=O)Nc3cn(CC)nc3C(N)=O)CCC2)cccc2c1OC(F)(F)O2 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82330,C(C(C)(C)CNC(=O)N(C)C(c1ccc(Cl)s1)C)SC 82331,C1(C(=O)NC2CC(N(C(=O)C=CBr)C)C2)CN(C)CCN(C)C1 82332,Cc1c(C(=O)NCC(C)(C)NC(C2CCCS2)=O)ccc(F)c1F 82333,C12(NC(=O)CC3(O)CCCCC3)CCN(C(=O)Cn3cc(CO)nn3)CC1C2 82334,C1(CNC(=O)CNC(C2CCC2)=O)CCC(NC(=O)Cc2ccccc2)C1 82335,c1(NC(CC)CNC(c2cc(O)nc(Cl)c2)=O)nc2c(cc1C#N)COCC2 82336,C(N=c1[nH]c(O)nc(=O)n1CCC(=O)N(C)C)c1c(C)c2c(o1)cccc2 82337,Cc1cnc(C(=O)NCC2CCN(C(=O)C=CC3CCCC3)CC2)cc1C#N 82338,c1(NC(=O)NC(CC)C(=O)N2CCC2C(=O)NC)cc(CO)cc(F)c1 82339,c1(NC(=O)NCC2(NC(=O)OC(C)(C)C)CCCCC2)cnc2[nH]c(=N)sc2c1 82340,C#CC1(NC(=O)C(=O)NCC(C)(C)CO)CCCC(C)(C)C1 82341,C1(CNC(CCC#C)=O)CCCCN1C(c1cnc(COC)s1)=O 82342,C1(C(N2CC(CCCCNC(c3cc(C(C)C)[nH]n3)=O)C2)=O)COCC(C)O1 82343,C1(CC(C)NC(C2CCSC(C)C2)=O)CCN(C(c2nncs2)=O)CC1 82344,Cc1ccc(F)cc1C(=O)COC(C1(C#N)CC1(C)C)=O 82345,C1(COC)CN(C(=O)C(C)CN(C)C)CCN1C(=O)C=C(C)c1cccnc1 82346,c1(OC)ccc(C)c(C(=O)NC2CC2CNC(=O)CC2CCC(C(N)=O)CC2)c1 82347,Cc1nonc1CNC(=O)CCn1cc(CC2(c3ccccc3)CC2)nn1 82348,c1(C(=O)NC(C(C)NC(Cc2c(C)scc2)=O)C)cccc(-c2nc(O)n[nH]2)c1 82349,Cc1cc(C(=O)NCCC2(O)CCN(C(=O)Cc3cnn(C)n3)CC2)ccc1Cl 82350,N(C1CCCn2nccc21)c1cc(N2CCCC(CC(N)=O)C2)nc(C)n1 82351,CC1(C)CN(C(=O)C2=COCCC2)CCN(C(=O)C2=CCCOC2)C1 82352,c1(NCC=CCNC(c2c(C)nc(-n3cccc3)s2)=O)ncccc1[N+](=O)[O-] 82353,c1(C(=O)NC2(CO)CCN(C(C(COCC)C)=O)C2)cc(C#N)c(N)cc1O 82354,c1(C(=O)NCCCNC(CC2C=NN(C)C2=O)=O)cc2cc(Cl)cnc2o1 82355,C(=O)(CC(C(F)(F)F)n1cccn1)NCC1(F)CC(NC(C(C)N(C)C)=O)C1 82356,c1(CCN2CC(C(=O)OC)CC(C(=O)OC)C2)nc2ccccc2[nH]1 82357,c1(CC(=O)NCC2CC2NC(C2(CF)CC2)=O)coc(-c2ccccc2)n1 82358,C1(=O)CCCCCN1.C1(C(N(C(C=C)C2CCC2)C)=O)CC1(F)Cl 82359,N1(C(c2cnsc2)=O)CCC2(CCCN(C(C3CC34CC(O)C4)=O)C2)C1 82360,c1(C(=O)NCC(C2CC2)NC(c2cc(Cl)n[nH]2)=O)occ2c1CCC2 82361,CC(C(C)(C)C(=O)NC1C=CCC1)NC(=O)Cn1cccn1 82362,C1(NC(CNS(CCCC)(=O)=O)=O)CCN(C(c2ccc(O)nn2)=O)CC1CC 82363,N1(C(CCC(C)N(C2CCCC2)C)=O)CCC2CCC(C1)N2CC(n1cncn1)Br 82364,C(=O)(C1=CCC(C)(C)CC1)NC(C1CN(C(C2CC2(F)F)=O)CCO1)C 82365,c1(C(=O)NC2C(NC(c3nn(C)c(Cl)c3)=O)C2)cccc2c1OCCN2 82366,N1(C(N(CC#C)CC2CC2)=O)CCCC1(C(C)C)CO 82367,c1(NC(CN(CCNC(c2csc(C3CCCO3)n2)=O)CC)=O)ccccc1 82368,CCCCCCCCC(C)C(=O)N1CC=C(CCNC(C2CCCSC2)=O)CC1 82369,C(CC(F)F)(C(=O)N1CC=CCO1)NC(c1ccc(CC#N)cc1)=O 82370,C(=O)(N1OC2CCC1CC2)c1c(C)oc(CNC(c2cccc(O)c2F)=O)n1 82371,c1(C(N2CC(CNC(c3c(OC)cccc3)=O)C(O)C2)=O)nc(O)nc(O)c1N 82372,N1(C(C2N(C)CCC2)=O)CCOC(C(=O)NC2CCN(CC3CC3)C2)CC1 82373,C1(N(CC#C)C(C2CC(CC)C2)=O)CCN(C(C2CC(N=[N+]=[N-])C2)=O)CC1 82374,CC1(C)CC(C)(C(N2CCN(C(N)=O)CC2)=O)CN1C(c1cscc1Cl)=O 82375,C(=O)(C1SCCc2ccccc21)N1CCN(C(C=C=C(C)C)=O)C(CCO)C1 82376,C(C)(CC(C)C(F)F)NC(CCCCNC(C1(CC)CC(C)(C)C1)=O)=O 82377,c1(NC(C2N(Cc3ccc(C(=O)OC)[nH]3)CCCC2)=O)c(F)c(F)nc(F)c1F 82378,Cc1ccc2[nH]c(C(=O)NC3(C)CCC(NC(=O)C4=CCC4)CC3)cc2c1C 82379,CCCC(CC(=O)NCCC(C(C)C)N(C)C)NC(c1ocnc1C1CC1)=O 82380,N1(C(C2C(CC)N(C(=O)C(C)OCC3CC3)CC2)=O)CCC(C)CC1C 82381,N1(C(COC2(C)CCCC2)=O)C(CNC(C2CCC2(C)C)=O)CC2CC12 82382,C1(NC(C2(C)CCC2)=O)COC2(CCN(C(c3cc(Cl)c4n[nH]cc4c3)=O)C2)C1 82383,N1(C(CCC(=O)N(C)C)=O)CCN(C(C2CCC(C(C)(C)O)CC2)=O)CC(O)C1 82384,Cc1ccc(NC(C)(C)CCN2CCSCC2)c([N+](=O)[O-])c1Br 82385,Cc1ccc(C=CC(=O)NCC2C(C)CCCN2C(=O)C(C)NC=O)c(C)c1 82386,C(C(C)NC(=O)CC1(C(F)F)CC1)(C(C)C)NC(CCn1ccc(C)n1)=O 82387,c1(OC)nccc(C(=O)NCC2C(O)CCN2c2nc(C)cc(C)n2)c1F 82388,C1(C(N2C(CC(=O)NC)CC2)=O)CCCN1C(=O)Cc1cncs1 82389,N#Cc1ncccc1NC(c1ccc(NC(=O)Cc2ccsc2)cn1)=O 82390,c1(C(=O)NC(C2CCCN2C(N)=O)C)ccccc1Nc1ccc(F)nc1 82391,c1(C(=O)NC2CC(NC(C(CC(N)=O)O)=O)C2)n[nH]c2c1CCSC2 82392,O=C1NCC2(CO1)CN(C(c1ccc(Br)c(F)c1)=O)C2 82393,N1(C(CC#N)=O)CCC(C2CN(C(c3cccc4nn[nH]c34)=O)C2)C1 82394,C1(NC(CCC#C)=O)CN(C(=O)CCc2nnc(C(C)OC)o2)CC1C 82395,c1(CC)ccc(C(=O)N(C2CCN(C(C3CCCC(CF)C3)=O)C2)C)cn1 82396,n1(CCCC)ncc(C(=O)NCC(CC(C)C)NC(c2cnnc(Cl)c2)=O)c1C 82397,C(CO)(CCC(C)C)NC(CONC(C1(SC)CC1(C)C)=O)=O 82398,C(CN=c1ccnc(N(CC2CCC(C)(C)CO2)CC2CCCO2)[nH]1)NS(NC)(=O)=O 82399,C(c1cn(C)cn1)=CC(=O)NC1CCN(C(c2nc(CC)oc2)=O)C1 82400,C1(NC(C)=O)CCCN(C(C2CC(O)(CNC(c3ccn(C(C)C)n3)=O)C2)=O)C1 82401,CC1(CCC(=O)NC2CC(C)(NC(c3csc(C4CC4)n3)=O)C2)CC1(F)F 82402,Cc1cc(Cl)cc(CN(CC(C)C(N2CCC2c2ccc(F)c(Cl)c2)=O)C)c1N 82403,C1(=CCNC(CN(C(=O)CC2CC=CC2)C)=O)CCCC1 82404,C1(NC(C=CCN(CC)CC)=O)CC2CN(C(=O)CS(N)(=O)=O)CCN2C1=O 82405,c1(C(=O)OCC(c2ccc(Br)s2)C)ccc(C2CCCC2)c(F)c1 82406,c1(CC(N2CC(C3N(c4ncc(C)c(C)n4)CCC3)C2)=O)ccn2cncc2c1 82407,N1(CCNC(C2CCCN2C(=O)CCN2CCCC2)=O)CCCC1=O 82408,N1(C(CC2CC(=O)NC2)=O)CCCCCC1CNC(C1CC1c1ccccc1)=O 82409,C1(c2onc(C3(COCC)CC3(F)F)n2)C2CN(C(=O)C(C)(C)C)CC12 82410,C12(CNC(C(C)SC)=O)CN(C(=O)Cn3ncn4cccc4c3=O)CC1CCO2 82411,c1(C(N2CC3(CC(NC(=O)Cc4c[nH]nc4O)C3)C2)=O)cnn2c1OCC(O)C2 82412,Cc1cccn2cc(C(=O)NC3CC3NC(=O)CC(C)(C(F)F)N(C)C)cc12 82413,O=C1CC2(CCN(C(c3cc4ccccc4s3)C(=O)NC3CCOCC3)C2)C(=O)N1 82414,C1(CNC(C2(OC)CCOC2)=O)CCC(CNC(c2ccoc2)=O)CC1 82415,N1(C(CCc2ccc(C)s2)=O)CC2CN(C(=O)CN3CCCNS3(=O)=O)CCC12 82416,C1(N(C(c2cccc(OCCC)c2)=O)C)CCN(C(=O)CCC2CC2)CC12CC2 82417,C1(C(=O)NC(C2(C)CC2)CO)COC2(C1)CN(C(=O)C=C1CCC1)C2 82418,C(C(C)(O)C(F)(F)F)NC(C1N(C(COCCOC)=O)CCOC1)=O 82419,CC1COCCC1N=c1[nH]c2c(c(=NCc3nc(C4CC4)cs3)[nH]1)COC2 82420,C(=O)(C(C)(C)CNS(C)(=O)=O)N1C(CNC(C(C)NC(=O)C(C)(C)C)=O)CCC1 82421,C12(NC(C(C)N(C)C)=O)CN(C(=O)C(Cl)=CCl)CC1CS(=O)(=O)C2 82422,C1(CN(C(c2ccc(C)n2C)=O)C)CN(C(=O)CC2CC=CCN2C)CC12CC2 82423,c1(OC)cc(CCNC(=NC)NC2CCCC(C)C2)cc([N+](=O)[O-])c1O.C(C)(C)S 82424,c1(C(N(CC(CC)NC(c2cnn(C3CCCC3)c2)=O)CC)=O)cnnn1C 82425,C=CCC(CC(=O)NCC(O)(COC)CO)NC(c1nc[nH]n1)=O 82426,Cc1[nH]c(C)c(C(=O)NC2CCCC2NC(c2c(C)n[nH]c2C)=O)c1C 82427,C1(C(N2CCC=C(C)C2)=O)CN(C(C2CC(CC3CC3)C2)=O)CCN1C 82428,c1(CNC(C(c2ccccc2F)C)=O)cnn2c1CN(C(=O)CCS(C)=O)CC2 82429,C1(N(S(C)(=O)=O)C)CN(C(c2cccc(CN3CCOCC3=O)c2)=O)CC1O 82430,CC(=Cn1ccnn1)C(=O)N1CCCC(NC(c2coc3c2CSC3)=O)C1C 82431,c1(C(=O)NC2C(NC(c3c(C)nncc3)=O)COC2)cc2ccccc2[nH]1 82432,N1(S(C)(=O)=O)CCCC(C(=O)NCC(C)(C)NC(C2CCC(C(N)=O)CC2)=O)C1 82433,C(C1CN(C(=O)CC(C)=C(C)C)CC1C(=O)NCCC)=CC 82434,C1(C(=O)OC)CC2C(CC1C(=O)NC1(CO)CCOC1)C2(F)F.C(C)C 82435,CCCC(O)CC(=O)NCC1CCC1NC(C1(C2CCC2)CC1)=O 82436,C1(COC(=O)Oc2n(CCC)ncc2C)COCCN1C=O 82437,c1(C(=O)NCc2cc(C(=O)OC)ncc2)cc(OC)ncc1-c1c(C)nn(C)c1C 82438,N1(C(C2N(S(C)(=O)=O)CCC2)=O)CC(NC(c2cc(N)ccn2)=O)C(C)(C)C1 82439,c1(C(=O)NC(CCCNC(CC(CC)CC)=O)(C)C)ccn2ncccc12 82440,C1(CNC(=O)C(O)c2cnc[nH]2)CCCN1CC(F)F 82441,N1(C(c2cc(OC)ncn2)=O)CCCC2(NC(c3cnsc3C)=O)CCCC12 82442,C1(SCC)CN(C(=O)C=NOC)CC1NC(=O)C=CCn1cncn1 82443,C1(N(C(C(c2scc(C)n2)C)=O)C)CCCCC1N(C)C(c1ccc(O)cn1)=O 82444,C(=O)(C1Cc2ccccc21)N(C1CN(C(CC2CCN(C)CC2)=O)C1)C 82445,Cc1nc(C(C)N(C)C)ccc1-c1ccc(-c2cc[nH]n2)cc1 82446,C(=O)(C1=CC2(CCOC2)C1)NCc1occ(C(N2C(CCC(C)C)CCC2)=O)n1 82447,C1(NC(CCCC=C)=O)CN(C(=O)CCCc2ccc(F)cc2)CC1C=C 82448,C1(NC(CC(C)O)=O)CCC(C(=O)Nc2cccc(CS(C)(=O)=O)c2)OC1 82449,c1(OC)cc([N+](=O)[O-])ccc1CNC(=O)CNC(=O)OCc1ccccc1 82450,C1(C2C(=O)N2c2ccc(F)cc2)CCC(C(F)F)CC1.C1(N)CCCCC1 82451,C(=O)(CCC(=O)N1CCCCC1CNC(=O)CC1(O)CCCCC1)N(CC)CC 82452,c1(C(N2CCC(NC(c3c(C)cno3)=O)CC2)=O)cc([N+](=O)[O-])c(C)s1 82453,N1(C(c2c(C(C)C)cccc2)=O)CCCC(C2CC2NC(c2cncn2C)=O)C1 82454,C1(NC(c2cc(C(C)(C)C)no2)=O)CCC(O)CN(C(C2CCCN2C=O)=O)C1 82455,Cc1cc(Br)c(S(=O)(=O)N2CCOCC2c2cccc(F)c2)s1 82456,c1(C(N2CCC3CC23)C(=O)NCC2CC2c2ccccc2)ccc(F)cn1 82457,C12(CC(F)C1)C(=O)NOCC=CCN2.N1(CC(=O)OC)CCCC1=O 82458,C(C(C)(C)CN=[N+]=[N-])NC(C(c1ccoc1)NC(c1ccc(C)cn1)=O)=O 82459,C1(OC)CN(C(C2CC2C)=O)CC1NC(c1ccn(C)c1C)=O 82460,c1(NC(C#C)=O)cccc(C(N2CCC(C3CC(N)CCO3)CC2)=O)n1 82461,c1(C(N(CCNC(C(CC(C)C)NC(C)=O)=O)C2CC2)=O)ccn(C)c(=O)c1O 82462,Cn1c(C(=O)NCCC2CN(C(C3CCCCC3C(F)(F)F)=O)C2)cccc1=O 82463,C1(C(N(CCN(C(CCN(CCC)C)=O)C)C)=O)CCCN1C1CC1 82464,c1(CC(=O)NC(C2(O)CN(C(c3c(C)nc(CO)o3)=O)C2)C)nc([N+](=O)[O-])n[nH]1 82465,C(c1cncs1)=CC(=O)N(CCC(=O)NN(CC(C)CSC)C)CC#C 82466,CC1CN(C(=O)CC2CC2)CC1NC(C1CC1c1cccs1)=O 82467,N1(C(c2n(C)nc3c2CCC3)=O)CCOC2(CCN(Cc3ncco3)CC2)C1 82468,C(=O)(C(C#N)C(C)C)NCCN(C(CC1C(CC)C1(F)F)=O)CC1CC1 82469,c1(C(N2C(C(C)C)CC(F)C2)C(=O)Nc2ccccc2)cncc2ccccc12 82470,Cc1cc(C(=O)NC2CCC(CC(=O)NC(C3C=CC(CO)C3)=O)C2)ccc1F 82471,C1(NC(=O)NCCC2CCCCO2)CCCN(c2ncccn2)C1 82472,C1(C)(N(C(C=C)COC(=O)COCC(C)C)C(C)=O)CCCC1CC 82473,CC1CN(C(=O)CCC2CC2)CC1NC(=O)CC1CC(=O)NC1=O 82474,n1(CC(N2CC(NC(C(COC)(C)OC)=O)C(O)C2)=O)cc(P(C)(C)=O)cn1 82475,C(C(C)(C)C1=CCCC1)NC(C=C(CNC(C1(NC(C)=O)CCCCC1)=O)C)=O 82476,C(=O)(CP(=O)(C(C)C)C(C)C)N1C2CC(NC(C(F)=CC)=O)CC1CC2 82477,c1(N2CCC(CC(C)NC(c3cscn3)=O)CC2)ccn2nccc2n1 82478,C12(CNC(C(CC)(F)F)=O)CC(C1)C(NC(=O)Cc1ccccc1C(C)C)CO2 82479,n1(C(C)C)ncc2c(N3CCC(NC(c4csc(S)n4)=O)C3(C)C)nc(Cl)nc12 82480,c1(COC)cc(C(N2CCCC2CN(C)C(c2ccsc2C#N)=O)=O)c(C)o1 82481,N1(C(C(c2ccccc2)NC(CCCCC=CC)=O)=O)CCOC(C)(C)CC1 82482,N1(C(C(C)Cc2ccc(Cl)cc2)=O)CC(NC(C23CC4CC2C3C4)=O)CC(C)C1 82483,CC(CC(N)=O)N=c1[nH]c(C(=O)N(C)C)c(CC(F)(F)F)s1 82484,N1(C(CC2(C)CC2)=O)CCOC2(CCN(C(c3cccn(O)c3=O)=O)CC2)C1 82485,N1(Cc2c(C)ccnc2)CCC(NC(c2ccc(C(F)F)o2)=O)CC(C)(C)C1 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82659,c1(C(N(CCN(C(c2ccc(C3CC3C)o2)=O)CC)CC)=O)cc(C#N)on1 82660,N1(C(C(C(C)O)(F)F)=O)CCC(C2(NC(=O)CC(O)CC(C)(C)C)CCC2)CC1 82661,N1(C(CC(C)OC)=O)C2CCC1CC(NC(c1coc(C(F)F)n1)=O)C2 82662,CC1SCCCC1C(N1CCC(CC(=O)NC2(N3CCCC3)CC2)C1)=O 82663,c12nccc(n1)NC(=O)C(c1ccc(C(F)(F)F)cc1)N2CC.C(CCOC)SC 82664,C1(C(C)O)CCN(C(C2CC(O)(CNC(=O)CCN3CCCC3=O)C2)=O)C1 82665,c1(NCC2CCN(C(c3c(COC)scc3)=O)C2(C)C)ncc2c(n1)COC2 82666,CC1(C)COCCC1C(=O)NCCCC1CCCN1C(c1ccc(CO)cc1)=O 82667,c1(CN(CC(=O)NC2COCC2n2cc(C(=O)O)nn2)C)ccccc1 82668,C1(C(=O)NCCN(CCC)C(C2CC(C)(C(C)(C)C)C2)=O)CCC(C)(C)OC1 82669,C1(CNC(c2c(C)ccn2C)=O)CN(C(=O)C(C)(O)CCN(C)C)CCCO1 82670,N1(C(CCCC(=O)OC(C)(C)C)=O)CC2CCN(C(C3CCNC3=O)=O)C2C1 82671,CC1=NS(=O)(=O)NC(C)=C1CC(=O)N1CC(NC(=O)CCCN(C)C)CCC1C 82672,c1(C(=O)NCCCOCCOC)ccc(NCCCC(C)NC(C)=O)cc1O 82673,CN1CCC(c2nnnn2CCCF)(NCC2OCCCC2(C)C)CC1 82674,C1(CNC(c2cc(C)sc2)=O)CN(C(C2CCSC2)=O)CC2(CCC2)O1 82675,CC1(C)CCC(C)(Cc2cn(CCNC(c3c(F)cc(F)cc3F)=O)nn2)CC1 82676,CC1CC(=O)NCCN1C(=O)CC(C)CNC(c1ccn(C)n1)=O 82677,C(=O)(C(F)C(C)C(F)(F)F)NCCC(C)NC(CC(CC)c1ccc(C)cc1)=O 82678,C(CC(=O)N1CCCN(C)CCC1)(C(C)CC)N(C(CC=CC=C)=O)C1CC1 82679,c1(OC)cc(F)c(C(=O)NCC(CNC(=O)C(C)(C)OC)C(F)(F)F)c(F)c1 82680,O=C1CN=C(NC2CC2)N2CCC(C2)O1.c1(Cc2ccccc2)ccccc1 82681,c1(-c2scc(C)n2)nc(C2CC23CC3)n(CCF)n1 82682,c1(C(C(=O)NCc2nc(Cl)sc2Cl)NCC)cccc(-c2nn[nH]n2)c1 82683,C(CCCCCN)N(C)C(c1cc(C(N)=O)c[nH]1)=O.C(=O)(CC(C)c1ccco1)C(C)=O 82684,c1(N2CCC(C(C)NC(=O)CCN3CCC(F)C3)C2)nc(C2CC2)nc(=N)[nH]1 82685,Cc1[nH]c2ccc(C(=O)NC3CC(NC(C4(O)CC(C)(C)C4)=O)C3)cc2c1C 82686,C1(NC(C(CCSC)OC)=O)CN(C(c2ccc(N)cn2)=O)C2(CCC2)C1 82687,C=C(Cl)CC(C(=O)NCC1(O)CC(C)(C)C1)NC(c1ccc(OC)cn1)=O 82688,N1(C(C2(C(=O)O)CC2c2ccccc2)=O)CC(O)C(O)C(O)C1C=O 82689,CCS(=O)(=O)C1CN(C(C2CCC(CCC(=O)O)O2)=O)C1 82690,C(=O)(C(C(=O)N1CC(O)(CNC(c2cc(=O)cc[nH]2)=O)C1)OC)OCC 82691,Cc1ccc(OC(C)C(=O)NC(c2ccccc2)CN(C(=O)CC(C)C)C(C)C)cc1 82692,C(c1ccc([N+](=O)[O-])s1)=CC(=O)NCC(C)CNC(C1(F)CCCN(C)C1)=O 82693,c1(C(=O)NCC(C)CN(C(=O)C=CS(C)=O)C)ccnc(C(C)(C)C)c1 82694,c1(C(=O)NCC2C(C)CCN2C(c2ccns2)=O)ccc2c(c1)CCC2 82695,N1(CC2CN(OC(C)(C)C)C2)CCC(N=c2[nH]ccc(CO)c2F)C(C)(C)C1 82696,Cc1nnn(CC(=O)N(CCC(C)NC(=O)CC(C)c2ccncc2)C)n1 82697,C(CCCC(CO)NC(=O)C(F)=C(C)C)NC(C=C(C)c1ccsc1)=O 82698,C(=O)(CS(=O)(=O)C1CC1)N(CCOC)CCNC(c1cc(OC)nn1C)=O 82699,C1(C(N2CCC(C)(C(=O)NCC(C)OCC#C)C2)=O)CCOC(=O)CC1 82700,C1(C(=O)NCCN(C(=O)CCc2ccncc2)CCCN(C)C)CCOCC1 82701,CC(CCNCCCCCC1CCNCC1)CC(C)(C)C 82702,Cn1ncc(C(=O)NCc2nocc2C(N2CC(CO)(CO)C2)=O)c1N 82703,Cc1cnc(Cl)c(C(=O)N(C)CC2CN(C(C3(C)CCCC3)=O)CCO2)c1 82704,N1(C(C(CC)(C)CC)=O)CCCCC(CNC(c2cnc(SC)cc2C)=O)CC1 82705,C1(C(=O)NCC2C(NC(C3CC4(CCOC4)C3)=O)CC2)CN2CCC1CC2 82706,C1(C2CC2)(C(=O)NC(c2onc(C)n2)C)CN(C(=O)CC2CCCN2C)C1 82707,c1(CC(N2CCCCC2Cn2cc(CCCO)nn2)=O)cccnc1Cl 82708,N1(C(c2ccsn2)=O)CCC(C(=O)NC2(c3nc[nH]n3)CC2)C(O)C1 82709,c1(C(=O)NCCCC(C)(C)NC(C(C)n2ccnc2)=O)ncc(F)cc1F 82710,CC(C)CCC(C)NC(=O)C(C)(C1CCC1)NC(=O)CCN=[N+]=[N-] 82711,c1(C(=O)NC2CN(C(C3(C)CC3Br)=O)C2)cnc(Cl)c(N)c1 82712,N1(C(C(c2scc(C)n2)C)=O)CCOCC1c1nccn1C 82713,Cc1nn(C)c2c(NCC3CCCCO3)nc(=NCCC(O)C3CC3)[nH]c12 82714,CC1CN(c2cc(CNC3CCNCC3C)ccn2)CCO1 82715,c1(C(=O)OC)cc(C)n(CC(=O)NCC(C)(O)CNC(=O)Cc2c[nH]nc2O)n1 82716,C12(NC(C3C(=C)CC3)=O)CCC(C1)N(C(c1ccnc(-c3ccco3)c1)=O)C2 82717,N1(C(C(CNC(C)=O)(C)C)=O)CCC2(CC1)CN(C(c1cnn3c1CCC3)=O)C2 82718,Cc1nc(CC(=O)NC(C(=O)NCC2CCCSC2)c2cccs2)n[nH]1 82719,N1(CC(C)O)CCN(CC(C2CCCN(C(C)C(C)(C)C)C2)=O)CC1.C(C(C)(C)C)CC=O 82720,C1(NC(C2N(C(C)=O)CCC2)c2cnccn2)CN(c2nnco2)CCC1C 82721,c1(CN(C)C)ccoc1C(=O)N(CCCCNC(=O)C=CC(F)F)C 82722,CCCC(C)(C)CC(=O)N1CC2CC(NC(=O)CCC3CCOCC3)CC1C2 82723,C1(NC(c2ccnnc2O)=O)C=CCN(C(c2ccc(CF)cc2)=O)C1 82724,C1(C#N)(C(N(C2CCCN(C(COCC(C)C)=O)C2)C)=O)CCOCC1 82725,C(=O)(CCCCCCCCCO)N1C2C(NC(CCOCC)=O)CC(C2)C1 82726,N1(C(C(C)SC)=O)CCCCC1C(=O)NCC1CC1(C)C 82727,C#Cc1ccc(C(=O)NC2(C)CC(NC(C3CCOC3)=O)C2)nc1 82728,S(=O)(=O)(c1cccnc1)NCC(=O)NC1N(C(C2N(CC)CC2)=O)CCCCC1 82729,CN1CC(NC(C2CN(C(c3ccccn3)=O)CCO2)=O)CC1CO 82730,C1(N(C(C(C2CCC(C)CC2)CC)=O)C)CCCN(C(=O)CN2CC=CC2)CC1 82731,N1(C(CN(C)CC)=O)C2CCC1CN(C(=O)C(C)Cc1cnc[nH]1)C2 82732,CC1=NNC(=O)C1CC(=O)NC(CO)C(C)NC(=O)Cn1c(C)csc1=O 82733,C12(C(CNC(=O)CC3CCCC3C)NC(CC=C(C)C)=O)CCC(CC1)C2 82734,C1(=Cc2c(COC)cccc2)CCc2ccccc2C1=O.C1(=O)C(C(=O)OC)O1 82735,C(CC(=O)Nc1cc(O)cc(F)c1)(C(F)F)NC(c1n(CC)nc(C)c1)=O 82736,C1(NC(CC#N)=O)CCC12CCN(C(c1ccc(SCCC3CC3)cc1)=O)CC2 82737,C=CC(C)(CC)C(=O)N1CCN(c2ccnc(OC)c2)C(=O)C1 82738,c1(NC(=O)CC(O)n2ccnc2)ccc(C2(CC3CC3)CCCC2)cc1 82739,C(=O)(C1CCCc2ccccc21)NC(C)CNC(=O)C(C1CCC(=O)N1)C 82740,c1(CC(=O)NCC(n2cc(CC(C=C)O)nn2)C)cccc(COC)c1 82741,C(=O)(CC(C(F)(F)F)NC(c1ccc2c[nH]nc2c1)=O)NCCC 82742,C1(NC(C(C)(C2CC2)OC)=O)CCN(C(=O)CN2CCOCC2)CC1C 82743,C12(CNC(C3(CC#C)CCOC3)=O)CC(CO1)N(C(c1cc3n(n1)CCC3)=O)C2 82744,C=C1CC(C(=O)NC(C)CC2CCCCC2)(CNC(=O)CN2CCCC2SC)C1 82745,C1(C(N2C(C)(CNC(=O)COc3ccc(F)nc3)CCC2)=O)CCCCNC1=O 82746,c1(NC(CCC)=O)c(OC)cccc1O.C(=O)(CCC(=O)NCCCC1CC1)OC 82747,C1(C)(C(N2CC(CCCCC)C2)=O)CCN(C(=O)C(C)(CC)OC)C1 82748,O(N=C1CCCCCC1)CC(=O)NCC(N(C(C(C)OCC)=O)C)C1CC1 82749,N1(C(CNC(C(N)=O)=O)=O)CCN(C(C2(c3ccccc3)CC2(F)Cl)=O)CC1 82750,N1(C(c2ccc(C(C)=O)c(F)c2)=O)CCN(C(=O)Cn2cnnc2O)C(C)C1C 82751,C(=O)(CCCS(C)(=O)=O)NC(C1CCCN(C(c2cccc(C)c2N)=O)C1)C 82752,CC(C)S(=O)(=O)CC(=O)NC1(CNC(=O)C(=O)Nc2ncc[nH]2)CCCCC1C 82753,N1(C(C2(COC)CCOCC2)=O)CCCC(CNC(c2cc(OC)cs2)=O)CC1 82754,Cc1oc(C(=O)NC(C)(C)CN(C)C(c2csnc2Cl)=O)cc1CO 82755,C1(COC)CN(C(c2csc(-c3ccncc3)n2)=O)CCN1C(=O)C(N)=O 82756,N1(C(C2C(OC)(OC)CC2)=O)CCC(F)(CNC(c2cnn(C(F)F)c2)=O)C1 82757,c1(C(=O)NC2C(NC(c3ccc(CF)cc3)=O)CCC2)ncc(F)cc1F 82758,Cc1nccc(C(N2CCCCC2CCC(=O)NC2(C)CC2)=O)n1 82759,C(C)(C(=O)NC1CC(F)(CNC(C2(N(C)C)CCCOC2)=O)C1)(C(C)C)OC 82760,C1(C(=O)NC2C(C)CN(c3nnc(C#N)s3)CC2)CN2CCN1C(C)C2 82761,C1(C(=O)NCCN(CC(F)F)C)CC2(CCC2)CN1C(=O)CC1CCCO1 82762,c1(C(=O)NCC(C)(C)NC(C(COC(C)(C)C)N(C)C)=O)cc(Br)ccc1O 82763,C(c1cn(C)cn1)=CC(=O)NC(CCOC)CNC(C1CCCN1C1CC1)=O 82764,CC1CN(C(c2cc[nH]n2)=O)CCC1NC(=O)CC1CCN(OC)CC1 82765,C1(CNC(CCC(=C)C)=O)CCCN(C(c2cc(NC(C)=O)cnc2C)=O)CC1 82766,N1(C(CNS(N(C)C)(=O)=O)=O)CCN(C(=O)C(C)(O)C2CC2)CC(CO)C1 82767,S(=O)(=O)(c1cc(C(F)(F)F)ccc1NCC(F)Br)N(C)Cc1cc2c(s1)CCC2 82768,c1(CNC(c2c(CNC(CS(CC)=O)=O)ccs2)=O)ccnc(C#N)c1 82769,C(CCC(C)CO)NC(C1(NC(CC)=O)CCSC1)=O 82770,C=C1CC(C(=O)Nc2cc(C(=O)OC)no2)N(C(=O)Cc2ccc(Br)cc2)C1 82771,Cc1nnc2n1CC(C(N1CCOCC(NC(=O)Cc3ccoc3)C1)=O)CC2 82772,Cc1cc(NC(c2cnn(C(C)C)c2C(F)(F)F)=O)ccc1NC(=O)C(C)O 82773,C(=O)(C1COc2ccc(Cl)cc21)N1CC(NC(C(C)(C)C2CC2)=O)C(C(F)F)C1 82774,C1(CC(=O)N(CC(c2nn[nH]n2)C)C2CC2)CCCN1C(=O)CCc1ccoc1 82775,n1(CC)nccc1C=CC(=O)NCC(C1CC1)N(C)C(c1snnc1C)=O 82776,c1(C(N(CC(C2CC(F)(F)C2)O)C)=O)ccc(N)c(Cl)c1 82777,c1(C(=O)NC2CC2C(=O)Nc2ncc(F)cc2Br)cc(Cl)c(Cl)cc1F 82778,C(=O)(CC(F)(F)C(F)F)N1C(C(=O)NC2(Cc3ccc(Cl)nc3)CCC2)CCC1 82779,N1(C(CC2CCC(=O)NC2)=O)CCN(C(C2CCCCC2)=O)C(CC(F)F)C1 82780,Cc1nc(-c2cccs2)sc1C(=O)NCCN(C(=O)CC(F)(F)F)CC1CC1 82781,CC(C)C(O)C(=O)N1CCC(CNC(=O)C(n2cnc(C#N)n2)C)C1 82782,c1(C(N2CCC(C)CC2)CNC(=O)CCC2CC2(C)C)cc(F)ccc1F 82783,c1(C(N2C(CN(C(C3(CC(C)C)CC3)=O)C)COCC2)=O)nccc2cc[nH]c12 82784,c1(C(N(C)CC2C(C)OCC2)=O)c(CNC(C2SCCS2)=O)nnn1C 82785,C1(CNC(c2ncc(C)nc2)=O)CN(C2CCc3ccccc32)C1 82786,C1(C(=O)NCC(C2CCCCC2)NC(=O)C2=CCCC2)CCC(F)(F)CC1 82787,c1(CC)ccc(CNC(=O)CCC(C)NC(C2CCOC2C(C)C)=O)cc1 82788,CC1(C(N2CC3(CC(NC(=O)C4=NNC(=O)CC4)C3)C2)=O)CCCCC1(F)F 82789,CC1CC=C(C(=O)NCc2cc(C(=O)NCC(C)C(C)(F)F)n[nH]2)CC1 82790,c1(-n2cc(CCCNC(c3c(C)nsc3C)C)nn2)ccc(F)cc1C(F)(F)F 82791,C1(NC(CCC(=O)OCC)=O)CCCC12CCN(C(C1CCC1(C)C)=O)CC2 82792,Nc1cc([N+](=O)[O-])ccc1C(=O)NCC1CCCN1C(=O)CC1CCC(=O)N1 82793,N1(C(c2nn(CC)c(O)c2)=O)CC(CO)C2(C1)CN(C(=O)C(O)C(F)(F)F)C2 82794,c1(NC(C2CCCC2)CC)nc2cc[nH]c2c(=NC(C)Cc2cccnc2)[nH]1 82795,C1(CC)CN(C(c2ccnc(F)c2F)=O)CCN1C(=O)Cc1ccccc1OC 82796,c1(N2CC(C)C(NC(C3(F)CCOC3)=O)CC2)ccc(Br)cc1[N+](=O)[O-] 82797,N1(C(c2sccc2Br)C(=O)NC)CC2CC(OC)C(C2)C1 82798,N1(C(CSCCC#N)=O)C2CCC(C2)C1C(N1CC(N(C)C)C2(CC2)C1)=O 82799,N1(C(CC2CCCC(OC)C2)=O)CCCC(CN(C)C(C2(OC(C)C)CC2)=O)CC1 82800,c1(CC(=O)NCC(C2CCOC2)NC(CC2(OC)CCCC2)=O)ccncc1F 82801,CC1CN(C(C2CC(C)(F)C2)=O)CC2(CCN(Cc3ccon3)C2)O1 82802,c1(COC)ccc(C(=O)NCC(O)CN(C(=O)CC(C)(C)C)C)n(C)c1=O 82803,C1(NC(C=CS(C)=O)=O)C2CC(O)C1N(C(=O)CCCn1cccn1)C2 82804,Cc1cc(=NCC2CCCC(C)CC2)[nH]c(=NCCc2cccc(N)c2)[nH]1 82805,CCCC(CC)CCC(=O)NC1CCC(C(=O)NC(C)Cn2cnnc2)CC1 82806,N1(C(C2C(C(=O)OC)CCO2)=O)CCC(NC(=O)C(C)NS(C)(=O)=O)C(CO)C1 82807,CC1(C)CC(CNC(C2CC23CC(O)C3)=O)CN1C(=O)CCC1CCC1 82808,c1(C(N(C2CC(NC(=O)CCC(N)=O)C2)C)=O)cnc(O)c2cccnc12 82809,Cc1cc(C)c(CC(N2CCOC(CNC(=O)C=CC3CCCO3)C2)=O)c(C)c1 82810,C1(CC(=O)NCc2[nH]nnc2C)(OC)CN(C(c2cnn(C)c2)=O)C1 82811,CC1CCCC(C(=O)NCCn2ccc(C(=O)NCCC(C)(C)O)c2)C1 82812,c1(C(N(C(=O)C(C)NC(N)=O)CCNC(c2c(C)occ2)=O)C)cccc(Cl)c1 82813,C1(C(=O)NCc2cncc(C)c2)CCN(C(=O)COCCN(C)C)CC1(C)C 82814,C1(CC=C)(NC(=O)C(N2CCCC(O)C2)C)CCN(c2nc(C)cc(C)n2)CC1 82815,C(=O)(C(C(C)=Cc1ccccc1)N1CCCC1COCc1csc(C)n1)NCC 82816,CCC(CC(=O)NC(CNC(c1ncoc1-c1cnn(C)c1)=O)CO)C(C)C 82817,C1(NC(CC2C(NC(CNC(CCC)=O)=O)CC2O)=O)(COC)CCC(C)C1 82818,c1(CC(=O)NC2(CNC(c3cc(CCC)oc3)=O)CC2)ccc(OCC#N)cc1 82819,N(C(=NCCSCNC(C1CCC1)=O)NCCN1CCCC1)C1C(C)CSC1 82820,C1(CNC(CCN(C(=O)CCOC2COC2)C)=O)(CO)CCCO1 82821,C1(C(=O)NC(CCCNC(C2(OCC)CCCC2)=O)C)CS(=O)(=O)CC12CCC2 82822,C1(C)(NC(C2CN(CC)C(=O)C2)=O)CCN(C(C2CC(CC(C)(C)C)C2)=O)CC1 82823,N1(CC)CC(NC(=O)CN2CCN(C(=O)C(C)c3ccsc3)CC2=O)C(C)(C)C1 82824,C12(C(=O)NC3C(NC(=O)Cn4cnc(Br)n4)C3)CC(C1)C(C(F)(F)F)O2 82825,C=CC(O)C(=O)N(CCNC(=O)CN1CCC(C)C1)CC 82826,c1(N2CCN(CC)C(C)(C)C2)nc(N(CC(F)(F)Br)C)c2ncn(CC)c2n1 82827,c1(C(N2C(C)(C(N3CC4(CC4)C3)=O)C=CC2)=O)n[nH]c2c1COC2 82828,C1(N(c2nn[nH]n2)C(c2c(C)occ2)=O)COCC1C1CC1(C)C 82829,C1(NC(c2c(CC)nco2)=O)CCC2CCN(C(C3(C)CC(C)C3)=O)C1C2 82830,c1(CNC(=O)CNC(c2ccsc2C)=O)nccc(=NCCCCC(C)OC)[nH]1 82831,c1(C(C)C(N2CCC(CNC(C3(O)CCSCC3)=O)C2)=O)c(F)cccc1F 82832,C(=O)(C1=Cc2ccccc2C1)N1CC(NC(C2C3CC3C3CC23)=O)(CF)C1 82833,N1(C(C(C2CCC2)OCC)=O)CC2(CCCCN2C(c2ccnc(S)c2)=O)C1 82834,CC(C)(C)CC(F)C(=O)NC(C(=O)NCC(O)C1(Cl)CC1)C(C)(C)C 82835,CCCC(C(=O)N1CCC(C)N(C(c2cc(C)c(F)c(C)c2)=O)CC1)S(N)(=O)=O 82836,N1(C(C(CC)OC)=O)CCN(C(C)CNC(=O)CN2CCCCC2)CC1 82837,Cc1coc(C)c1CNC(=O)C(=O)NCC1CCCC1CC(C)C 82838,Cc1cc(=NC(=O)c2ccc(F)c(C(=O)O)c2F)[nH]n1-c1ccccc1Br 82839,Nc1sc2ccccc2c1C(N1CCOCC(NC(c2nccnc2N)=O)C1)=O 82840,CCC(CC(C)C)C(=O)NCC1CCCCN(C(=O)CS(=O)CC)C1 82841,CCC(CC)(C(=O)N1CCC(NC(=O)CCC(C)(C)F)C(C)C1)OC 82842,c1(OC)cc(C)cnc1C(=O)N(C)CC1C2CN(C(C3CC3C)=O)CC12 82843,c1(C(=O)NCCN(C(c2ncoc2C(C)C)=O)CC)cnc(CC(C)C)cn1 82844,CCCC(O)CC(=O)N1CCOCC1CNC(c1sc(C)nc1CC(C)C)=O 82845,C1(CNC(C(C)CN(C)CN2C(=O)CNC2=O)=O)CN(C)CCN1C 82846,CC1CN(C(C2CC2F)=O)CCCN1Cc1c(Br)ccnc1Br 82847,Cc1cccc(C)c1C(c1nnnn1CC(F)F)NCC1(C)CC=CC1 82848,Cc1nc(-c2nccs2)ncc1C(N1CC(O)(CCNC(=O)C=CBr)C1)=O 82849,c1(OC)ccc2[nH]nc(C(=O)NCC3(NC(=O)CSc4ccncc4)CC3)c2c1 82850,C(=O)(C(F)C(=O)NCC(CC)NC(=O)CCCc1cc(C)no1)OCC 82851,CCC(C(=O)NC1CC(C)(C(=O)NCc2cccs2)C1)OC 82852,C(CCCC1CC1)(c1nnnn1CCCOCC1CC1)NC1(C(C)C)CC1 82853,CCS(=O)(=O)C=CC(=O)NC1CCCC(N(CC2CC2C)CC)C1 82854,C12(C(N3CC(CCNC(Cc4c(C)n[nH]c4)=O)C(C)C3)=O)CCC(CC1)CC2 82855,c1(C(=O)NCC(CNC(=O)C(C)(C)n2ccc(C(N)=O)n2)OC)ccc(C)n1C 82856,C1(CNC(c2[nH]cc(C(C)=O)c2)=O)CCCCN1C(C1(n2nccn2)CC1)=O 82857,C1(NC(C2C(C(C)(C)C)C2)=O)CS(=O)(=O)CC1NC(=O)C=Cc1cnccn1 82858,C1(CCNC(C2C(C)CCC2)=O)CSCCN1C(=O)COc1cccnc1 82859,C1(C(N2CCC(CCN(C(=O)COCP(C)(C)=O)C)CC2)=O)CC12CCOCC2 82860,Cn1cnc2nc(=NCc3cnccn3)[nH]c(NCC3C(F)(F)C34CCCC4)c12 82861,C=C(Cl)C(C)(C)C(=O)N1CC(C(N)=O)C2(CC2)C1.c12cc(c(C)o1)NC(=O)CC2 82862,CC(C)CC(C(=O)NC1C2CC3C1C3C2C(N1CC(C)C1(C)C)=O)C(N)=O 82863,C12(C(=O)Nc3cccc(-n4ccnc4O)c3)CCCC1C2(F)F 82864,C(=O)(N=c1[nH]onc1C1CC1)OC(=O)Cc1cn(C(CCC)C(=O)NCC)nn1 82865,C(CCCCCNC(c1ccc[n+]([O-])c1)=O)NC(c1ccsc1)=O 82866,C1(CC(=O)N(C(C)CO)CCO)CC(OC(=O)C(C)n2cncn2)C1 82867,C1(N(C(C(C)N=[N+]=[N-])=O)C)CCCN(C(=O)C(c2cncnc2)C)CC1 82868,C12(CC(N3CC(C#C)C3)=O)COCCC1CN(Cc1ccccc1)C2 82869,C(CCCCC(=O)N1CC2(CC(NC(=O)C(n3cc(C)cn3)C)C2)C1)SC 82870,C1(CC)CN(C)CCN1C(=O)C(=O)N(c1ccccn1)CC1CCCCC1 82871,C1(OC)CC(NC(C2(C)CCN(C)C2=O)=O)CN(C(=O)C=CC2CC2)C1 82872,c1(OC)cc(OC2CC2)ccc1C(=O)N(C)CC1(NC(=O)CC(C)C)CC1 82873,C(CC1CC1)(C(=O)NC(CC1CC1)C(=O)N1CCC(CC2CC2)C1)OC 82874,Cc1cc(C(N2CC3CCC3(CCNC(c3cnc(S)n3C)=O)C2)=O)cc(C)c1 82875,C1(C(=O)OC)CN(C(c2ccnc(Br)c2F)C(=O)NCc2cccs2)CC(=O)N1 82876,CC(CC(=O)c1ccc(F)cc1)C(=O)NCCCCCNC(=O)C(C)(F)F 82877,c1(CC(=O)NC2CN(C(c3occ(C)c3)=O)CC2C)c[nH]c2cccnc12 82878,c1(NC(C2CC(C)CN2C(c2cc3sccc3[nH]2)=O)=O)nc2ccccc2s1 82879,C1(NC(c2c(C)cc(SC)s2)=O)CN(C(c2n[nH]c(C)n2)=O)CC(C)(C)C1 82880,c1(OCC)cc(C(=O)NCC(O)CCNC(=O)CCSc2ccoc2)cc(F)c1 82881,c1(OC)c(Br)ccc(F)c1CN1CCCC1CCC(N1CCC(F)CC1)=O 82882,C12(C(=O)NCC3(C)CN(C(C45CCCC4CCC5)=O)C3)CCCC1CC(=O)C2 82883,C1(C)(CC)CC(NC(c2cc(F)ccc2F)COC)CCO1 82884,n1(CC)ncc(Cl)c1C(=O)Nc1cccc(C(C)N)c1 82885,Cc1ccc(C(=O)NC2CCC(C)N(C(C3CC4(C3)CC(O)C4)=O)C2)cc1C#N 82886,C1(C(N2CCC(C(C)NC(Cc3c(C)nc[nH]3)=O)CC2)=O)OCCOC12CCC2 82887,N1(C(c2c(C)c[nH]n2)=O)CCC2(CCC2)C(NC(=O)CSCCN(C)C)C1 82888,c1(C(=O)NCC2(C)CCC(NC(c3cc[n+]([O-])cc3)=O)C2)cnc2n1CCC2 82889,c1(C(C)OCC)nc(C)c(C(=O)NC(C)(C)CNC(=O)C=Cc2nccs2)s1 82890,CC1C(=O)N(C)CCN1C(=O)C(C)(C1CC1)N(C(=O)CCCC1CCCO1)C 82891,Cc1cc(N2CCCCC2CCNC(=O)Cn2nccn2)cc(C#N)c1[N+](=O)[O-] 82892,CCCC(C(=O)NCc1ccccn1)N1CCCC1C(c1ccccc1)O 82893,c1(-c2cc(OC)c(F)nc2)cc(C(=O)NCCCSC)cc(Cl)c1OC 82894,c1(OS(CC2CCCC(C)C2)(=O)=O)ccc2cccnc2c1 82895,C1(NC(C=CCOC)=O)C=CCCC1C(N1CC(c2cc(O)no2)C1)=O 82896,N1(C(C(CC)N(C)C)=O)CCN(C(c2ncoc2C2CCCO2)=O)CC(C)(C)C1 82897,c1(C(N(CCC(=O)NC(C2CC(C)C2)CC)C(C)C)=O)cccnn1 82898,CC#CC1CCN(C(c2cc(CNC(C3CC3C(C)C)=O)nn2C)=O)C1 82899,Cc1cc(O)ncc1NC(C1(C)CC(O)CN1C(=O)C(C)C)=O 82900,c1(OC)ccc(C(=O)NC(C2CCCN2CCc2ccccc2)C)cc1 82901,C1(CNC(=O)CCc2nc[nH]n2)CCCCC1NC(=O)CCc1cn[nH]c1 82902,N1(C(C2CCSCC2)C(=O)NCc2nnn(C)n2)CCCc2occc2C1 82903,N1(C(=O)CC2CC2)CCCCC1C1CCCN1C(=O)Cc1ccccc1 82904,C1(CCNC(C(C(C)C)OC)=O)CCCN(C(c2c(C)noc2N)=O)CC1 82905,CN1C2CCCC1CN(C(=O)C1=NOC(CNC(=O)C3=CCCCCC3)C1)C2 82906,N1(C(C2(C)N(C(CCn3ccc(C)n3)=O)CC=C2)=O)CC2CSCC(C2)C1 82907,C1(F)(C(N(CCN(C(c2c(C)cc(C)s2)=O)C(C)C)C)=O)CCCCCC1 82908,C(=O)(CC(C)(C)C=C)NC1CN(C(C=CC=CC)=O)CC1c1ccccc1F 82909,C(=O)(C(C)CC(F)F)NC1CN(C(c2n(CC#C)ccc2)=O)CC1O 82910,Cc1ccc(C(N2CC3CCC2C3NC(C2(C)CC2(F)F)=O)=O)cc1OC(F)F 82911,N#Cc1ccc(S(=O)(=O)NC2(C3CCC3)CC2)cc1N1CCc2sc(Cl)cc2C1 82912,c1(C(N2C(C)CC(NC(C3(OC(C)=O)CC3)=O)C2)=O)cc2cccnc2s1 82913,N1(C(c2ccc(COC)o2)=O)CC(OC)CC1C(N1CC(C)(OC(C)=O)C1)=O 82914,C1(C(N(C2CCN(C(c3c(F)cncc3Cl)=O)C2)C)=O)COCCC1(F)F 82915,N1(C(CC2C(C)CCO2)=O)CCCCC2(CCN(C(C3CS(=O)(=O)C3)=O)C2)C1 82916,N1(C(c2c(CC)nn[nH]2)=O)CCOC(C(=O)NCC(=O)OC)CC1 82917,C(CC(CC)C(=O)NC(CN(C(=O)CSCC(N)=O)CC)CC)=CC 82918,C1(OC)CC2CC1CN(C(=O)CC1C3CCC(C3)N1C(C1CC(=O)N(C)C1)=O)C2 82919,C1(NC(CC=CC=C)=O)CC2(C1)CC2NC(=O)C(c1ccc(Cl)s1)=O 82920,C1(C(=O)NCCCCC2C(C)C2)CN(C(=O)CC2CCCC(=O)C2)CC(C)(C)C1 82921,N1(C(CC2(N(C)C)COC2)=O)CCN(C(=O)CNC(=O)C(F)(F)F)C2(CCC2)C1 82922,N#Cc1cccc(I)c1NC(C1CCCCC1NC(c1ccc(CO)cc1)=O)=O 82923,c1(NC(CCNC(C(CCC)NC(N)=O)=O)(C)C)ncnc2cccnc12 82924,c12ccc(I)cc1N(c1c(OC)cncn1)C2=O.C1(SC)CCNCC1F 82925,c1(C(=O)NCC(C)CN(C(=O)CN2CCSCC2)C)conc1C1CCCO1 82926,c1(OCC=C)c(OC)cc(-c2nn[nH]n2)cc1NC(c1cccc(C)c1CC)=O 82927,Cc1c(F)ccc(C(=O)NC(CO)C(C)NC(=O)CC2OCCC2(C)C)c1C#N 82928,Nc1ccc(CCC(=O)NCCCCCCNC(C2COCCOC2)=O)nc1 82929,C1(CC)CC(N=c2[nH]c3c(c(=NCC4(C(C)(F)F)CC4)[nH]2)COCC3)CCO1 82930,Cc1ccnc(C(=O)NCCN(CC(C)O)C(=O)CC2CCC(=O)N2)n1 82931,C1(CCCCNC(CN(C)CC)=O)CCN(C(C23CCCC2C3)=O)CC1 82932,N1(C(C(C)CF)=O)CCOCC2(COCCN2C(=O)C2CCCc3sccc32)C1 82933,C(=O)(C(C)(C1CC(F)(F)C1)NC(=O)C(C)N(C)C)OC 82934,CC1C(C)N(C(=O)Cc2cc(F)ccc2O)CCN1C(=O)CCc1ncc[nH]1 82935,c1(C(=O)NCCC2N(C(c3c(=N)[nH][nH]c3)=O)CCC2)cc(O)nc2ncccc12 82936,c1(C(=O)OC)ccc(CN2CCNC(C(=O)NCc3ccn(C)n3)C2)c(O)c1 82937,C1(CNC(C)Cc2ccc(N(C)C)cc2)COCCC1c1ccccc1 82938,c1(OC)cc(O)c(C(N2CC(C3CN(C(=O)C(C)(CO)OC)C3)C2)=O)cc1OC 82939,C(=O)(C(F)(F)C(O)CC)N(CC(CC)NC(=O)Cc1sc(C)nc1C)C 82940,C12(CNC(c3c(OC)cccc3Cl)=O)CCCC1CN(C(=O)CC1CC=CC1)C2 82941,N1(C(=O)COCC2CCCCO2)CC2CC(C1)CN(C(c1cocn1)=O)C2 82942,Cc1cc(N)c(C(=O)NC(CO)C(C)NC(C2C3CC4C(C3)C24)=O)c(F)c1 82943,C(=O)(C1CCCc2cncn21)NC(C(C)C)CCNC(c1c(O)cccc1Cl)=O 82944,c1(C=O)sc(C(N)=O)cc1C.n1(CC)ccnc1C1OCCC1c1ccccc1 82945,c1(C(=O)NCC(CC=C)NC(C2CS(=O)(=O)C2)=O)cnc2c(F)cc(C)cc2c1 82946,CCCC(C(=O)N1CC(N2CC(F)C2)C1)NC(=O)C(C)c1cccs1 82947,C1(CCCN(C(C2C(NC(CCNC(N)=O)=O)CCC2)=O)CCO)NC(=O)NC1=O 82948,C1(F)(CNC(C(C)(C)OC(C)C)c2nnnn2CCC2CC2)COCCOC1 82949,C#Cc1cc(C(=O)NCC(C)CNC(c2ccc(Cl)nc2O)=O)ccc1C 82950,CC(=O)CCCC(C)C(=O)N1CCC(C)C1C(N1CC(C)(C)C1)=O 82951,C1(C(=O)NC2C(NC(c3cccc(OC)n3)=O)CCC2)CC12CCC(F)(F)CC2 82952,C1(N(C)C(C2CCCOC2)=O)CCCN(C(=O)C(C)(C)c2ccno2)CC1 82953,c1(C(=O)NCCC(C)(C)NC(=O)C=CC2CCCCC2)cccc(N)c1 82954,Cc1cc(C#N)ccc1CC(=O)NC(C1CN(C(C23CCCC2C3(F)F)=O)C1)C 82955,C1(NC(CSCC)=O)COC2C(NC(=O)CN(C3CCC3)CC)COC12 82956,C(=O)(C(C)CC(C)(F)F)NCCC1N(C(C2(C)CCN(C(C)=O)CC2)=O)CCC1 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83170,C1(NC(CCN(c2ccccc2)C)=O)CC2(C1)CC2NC(=O)CCS(C)=O 83171,c1(SC)nc2ncnc(NCC3(NC(=O)CN4CCCCCC4)CC3)c2s1 83172,c1(C(N(C(C)C)CCNC(C2CCC3(CCC3)O2)=O)=O)ccnc2c1CCC2 83173,c1(C(=O)NC(C2CCN(C(c3cccc(NC(C)C)c3)=O)C2)C)cc(Cl)nnc1O 83174,C=C=C(C)CC(=O)N(C1CCN(C(=O)CNC(=O)C2CC2)C1)CC 83175,C1(C)(CNC(C2CC(CC)(CC)C2)=O)CCC(NC(=O)C=Cc2cnccn2)C1 83176,CC(C)(CNC(=O)CCCn1ccnc1)CC(=O)NC(C1CCOC1)CO 83177,c1(C(N2CCC3CCC(C2)S3)C(=O)NC2CCCC2)csc2ccccc2c1=O 83178,c1(C(C(=O)NC)N(C)CC2CCCO2)cc(Br)c(F)cc1F 83179,C=CC1(O)CCN(C(=O)C(C)N(C(=O)Cc2nncn2CC)CCC)C1 83180,c1(C(=O)NC(C(N2CC(CC)C2)=O)C2CCCO2)ccc(C)c(C#N)c1 83181,N1(C(=O)Cc2ccsc2)CCC2C1CCN2C(c1cc(F)cc(Br)c1)=O 83182,Cn1cc(C(=O)NCCCCCCNC(=O)CCC(C)(C)F)ncc1=O 83183,c1(NC(C2N(C(Cc3cccc(SC)c3)=O)C3C(C2)C3)=O)ccc(F)cc1Cl 83184,c1(CN2CCCC(C(=O)NCc3ncc(Cl)cn3)CC2)cc(Cl)c(Cl)cc1Cl 83185,N1(C(C2C(C)CC2)=O)CC2CC(C1)C2NC(=O)CCC(C)(C)C 83186,c1(C(=O)NCC2N(C)CCN(C(C3COCCO3)=O)C2)cc2c(nn1)CCOC2 83187,C1(NC(CNC(CC)=O)=O)CC2CCC(C1)N2C(C1(CC)CCCNS1(=O)=O)=O 83188,c1(C(N2CCCC(CCNC(c3c(COC)ncs3)=O)C2)=O)ccc(C)c(O)n1 83189,C1(NC(C=CC(C)NC(C2CS(=O)(=O)C2)=O)=O)CCCC(O)CC1 83190,Cc1ccc(C(=O)NC2CN(C(c3coc(CN(C)C)n3)=O)C2)cc1 83191,c1(C(=O)OCC)ccc(NC(=O)N(C2CC3(C2)CC3F)CCN(C)C)cc1 83192,C(CC(C)C(=O)NC1COCC1CNC(=O)CC1(C)CCOCC1)=CC 83193,c1(NC(CC2(C)CN(C(C3N(C)CCC3)=O)C2)=O)cc(F)c(F)cc1F 83194,c1(CC(=O)NC2CC3CC2N(C(C2CS(=O)(=O)C2)=O)C3)ncc(F)cc1F 83195,C1(CCNC(=O)CN=[N+]=[N-])(OC)CN(C(=O)CCSC)C1 83196,c1(C(N2CC(C3(NC(=O)Cc4ccsc4)CC3)C2)=O)cc2c(=O)[nH]ccn2c1 83197,C1(NC(C(C)OCCOCC)=O)CC(NC(=O)Cc2ccc(F)nc2)C(O)C1 83198,C1CCN=C(NC(C2(O)CCC(C)(C)CC2)C)NCCNS(=O)(=O)N1.CS 83199,C1(C(=O)NC(CNC(=O)C(C2CC2)C2CC2)C2CCC2)CC12CCCC2 83200,Cc1ccc(CNC2CCN(C(c3ccc(C4CC4)cn3)=O)CC2C)c(O)n1 83201,c1(C(N2CCN(Cc3ccc(C)cn3)CC2)C(=O)NCC)cnc2ccsc2c1 83202,c1(CC(N2C(CNC(C3OCC(C)C3)=O)CC2)=O)cc(OCC(F)(F)F)ccn1 83203,N1(C(C(CCF)NC(c2c(C)nns2)=O)=O)CCC2(CCCO2)C1 83204,N1(C(c2cc(C)oc2C)=O)CCC2(COC(CNC(C3(C)CCC(C)C3)=O)C2)C1 83205,c1(C(N(CCN(C(CC(=O)OC)=O)C)C)=O)cccc2c3c([nH]c12)CCCC3 83206,c1(C(N2CC(NC(=O)C=Cc3cncs3)C2)=O)ccc2c(c1)C(=O)NC2 83207,c1(C(=O)NCC(C)NC(=O)CC2CCCN(C)C2)cccc2c1CCCCC2 83208,C12(CC(=O)NC(C=C)C3CC3)CCC1CN(C(c1cc(O)cc(=O)o1)=O)C2 83209,C#Cc1ccc(CCC(=O)NCC2CCCN2C(=O)C(C(=O)OC)OC)cc1 83210,c1(COC)cc[nH]c1C(=O)NCCC1CCN(C(=O)CC2CC2C(F)(F)F)C1 83211,C1(CN(C(CC2C(C)C2)=O)C)COCCN1C(c1ccc(N(C)C)cn1)=O 83212,C(C)(C(F)(F)C(F)(F)F)=CC(N1C2(CN(C(C3CCC(=C)CC3)=O)C2)CC1)=O 83213,C1(NC(c2ccc(CNC(C(=O)NCC)=O)o2)=O)CCCC(C(N)=O)CC1 83214,C1(C(C(=O)N(CC(C)NC(c2cc(C)oc2)=O)C)C)CCCCCC1 83215,c1(CNC(c2n(CC=C)nnn2)(CCC)C2CC2)nc2c(n1C)CCCC2 83216,c1(C(=O)OC)cnc(N2CCN(C(C3CC3C)=O)C(C)C2)nc1C 83217,C1(C(F)(F)F)(OC)CC(C(=O)NCCNC(=O)CCCOC2CCOCC2)C1 83218,C(=O)(CCCC(F)(F)CO)NC1CCC(N(C(c2c(SC)ccc(F)c2)=O)C)C1 83219,Cn1cc(CC(=O)NCC2CCC(NC(=O)CC3CCCOC3)C2)cn1 83220,c1(C(=O)NCC2N(C(CC3N(C(C)=O)CCC3)=O)CCC2)ncc(C#N)cc1Cl 83221,c1(CC)c(NC(=O)C(c2ccoc2)NC(=O)CCCCN(C)C)cnn1C 83222,C(CCC(C)C(=O)NCC(C)(C)CCNC(c1sccc1OC)=O)OC 83223,N1(C(c2nc(COC)sc2)=O)CCC2(CCCC2NC(c2[nH]c(C)nc2C)=O)C1 83224,C#CCCCCCCC(=O)NCC(C)(C1CC1)NC(c1ccc(F)cc1CC)=O 83225,C1(C(=O)NCC(CN(C(=O)CC(=O)N(C)C)CC)(C)C)CCCC12CCOCC2 83226,C(CC1CC1)(C(=O)N1CCCC1C(C)CC)NC(C(C)=C(CC)C)=O 83227,C1(C(=O)NCC2=C(C)CCC2)CC2CCC(C1)N2C(=O)C(O)c1ccsc1 83228,Cc1oc(C(=O)NC2CCN(C(c3cc(O)nn3C)=O)C2C)cc1Br 83229,C1(NC(CC2(C)CC2)=O)CCCCC1CNC(=O)CC1OCCCO1 83230,C(=O)(C(CC(C)C)ONC(c1sccc1C#N)=O)NCC1(CC)CCC1 83231,N1(C(C(CC)C(C)C)=O)CCC(C2CC2)C1C(N1CCC(C)(C(=O)OC)C1)=O 83232,C1(NC(=O)Nc2cn(CC(C)(C)CO)nc2)(Cc2cccnc2)CCCCC1 83233,c1(OC)cc(C(N2CC(F)CC2CN(C(=O)Cc2cnn(C)c2)C)=O)n(C)n1 83234,c1(C(=O)NC(CCSC(C)C)C)cc(Cl)ncc1F 83235,c1(CC)ccccc1CC(=O)NCCCCCCNC(=O)CC1CCCC(=O)N1 83236,C(=O)(CC1=NN(C)C(=O)C1)NC(c1nocc1C(=O)NCC1(CC(N)=O)CC1)C 83237,c1(C(=O)NC2CN(C(CC(CC)SC)=O)CC(O)C2)cncc2sccc12 83238,c1(NC(c2n(C(C(=O)OC)C)nnn2)C2(CC#N)CC2)cc(C)cc(Br)c1 83239,c1(NC(CN(C(c2ccccc2)C(=O)OC)OCC)=O)cccc(F)c1C 83240,CC(C)CC(CO)NC(C1(N(C(=O)CC2CC3CC3C2)C2CC2)CCC1)=O 83241,C1(CNC(C(CCC)(C)CCC)=O)CC2(CCOCC2)CN1C(c1csnn1)=O 83242,N1(C(C2(C)CN(C(c3cccc(COC(C)C)c3)=O)C2)=O)CCC(O)C(F)C1 83243,N1(C(C=C(C)C)=O)CC2CC(NC(c3cc(C)on3)=O)C2C1 83244,C12(C(=O)NCCCN(CCCNC(C)=O)C)CCC(C1)c1ccccc12 83245,N1(C(C)=O)CCC(NC(=O)CC2CCC(C3CC3)O2)C2(CCC2)C1 83246,c1(C(N(C)CC2CCN(C(COCCCC#C)=O)CC2)=O)ccc(CO)c(Cl)c1 83247,N1(C(c2n(C)ncc2)=O)CCC(NC(=O)CC2(C)CC2(Cl)Cl)C(F)(F)CC1 83248,C1(C(C)(C)CO)CCN(C(c2cc(-n3cccn3)ccn2)=O)CC1 83249,Cn1c(C(=O)NCC2COC(CNC(=O)CCCCC#N)C2)cc2occc12 83250,CN=c1[nH]c(=NCc2cc(Br)ccc2C)[nH]c(=NC(C)c2cnn(C)c2OC)[nH]1 83251,c1(CC)nn(C)cc1C1C(=O)Nc2cccc(c2)N1C.C(C(=O)OC)OC(C)C 83252,c1(CCNC(=O)COc2cc(F)cc(F)c2)c(F)cccc1Br 83253,C1(C(N2C(C3(C(=O)NC(c4ccc(O)cc4)C)CC3)CCC2)=O)CC1C1CCC1 83254,C1(O)(CN(C)C(C2CCC(F)(F)C2)=O)CCCN(C(c2ccc(C3CC3)o2)=O)C1 83255,C1(NC(C(CC)c2ccccc2)=O)CC(F)(F)CC1NC(c1ccc(Cl)cc1)=O 83256,c1(CN(C2CCC23CCNCC3)C(C2CCCCO2)=O)cccc([N+](=O)[O-])c1F 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83379,C1(NC(C2C(C)CCO2)=O)CC(F)CN(C(=O)CNS(=O)(=O)C2CC2)C1 83380,c1(C(=O)NCC2OCCCN(C(C3N(C)CSC3)=O)C2)cccc([N+](=O)[O-])c1 83381,C1(CC)CNCCN(N2CCCC2(C)C(N)=O)C1 83382,c1(CC(=O)NCC(C2CCC2)NC(=O)COCC2CC2)ccsc1Br 83383,C(=O)(C(C)(F)C(C)(C)F)N(C)CCNC(C1(F)CCCOC1)=O 83384,CC(C)CC(C)C(=O)NCCCCC(=O)NC12CCN(CC1)C2 83385,c1(C(C(C)C)C(N2CC3C(C2)C3(C)C)=O)cc2ccc(-c3cncc(O)c3)cn2n1 83386,N1(C(COCC=C)=O)CCC(C2CCN(C(c3cc(CSCC)on3)=O)CC2)C1 83387,CC1CNc2ccc(C(=O)NCCCOCCNC(C3CCCCO3)=O)cc21 83388,c1(CCC(N2CCC(Cn3cc(CC(C(C)C)O)nn3)C2)=O)ccc(F)cc1F 83389,C(=O)(C(F)C(C)(C)O)N(C(CC)C(=O)NCC(C)C)C 83390,C1(COCC)CCCN1C(C1CCC(n2cc(C(O)C(C)(C)C)nn2)C1)=O 83391,c1(OC)cccc2c(C(=O)NCCNC(c3cc(OC)nn3C)=O)c(C)[nH]c12 83392,CC1CC(CNC(C2(F)CCC2)=O)CN1C(c1ccncc1)=O 83393,c1(C(=O)NC2CC(C(=O)NCC(C3CCCC3)OC)CC2O)ncc(F)cc1F 83394,CC1(CC(F)(F)F)CN(CC(=O)N(Cc2cn(C3CC3)cn2)Cc2ccccc2)C1 83395,Cc1cc(Br)cc(C)c1CN1CCN(C(c2cc(O)n(C)n2)=O)C(C(F)(F)F)C1 83396,N1(c2nnn(C)n2)CCCC(C2CC2NC(c2cccs2)=O)C1 83397,N1(c2cc(C)[nH]c(=NCc3ccc(F)c(Br)c3)n2)CCN2C(CNS2(=O)=O)C1 83398,c1(C(N(CC(C)O)CCNC(C2(CC=C)CCCC2)=O)=O)ccccc1C1CC1 83399,C1(C(N(C(CC)CO)CC)=O)CN(C(=O)Cc2cccc(O)c2)CC12CCC2 83400,c1(OC)ccc(CC(=O)NC(C)C(CO)SC(C)C)cc1[N+](=O)[O-] 83401,C1(C(N(C)CC2N(C(c3ccc(CC)cn3)=O)CCOC2)=O)CC(C)(C)CCO1 83402,C#CCCCC(C)C(=O)NC1(CNC(=O)Cc2nocc2CC)CCCCCC1 83403,N1(C(C(C(=O)OCC)C2CC2)=O)CCOC2(C1)CN(C(C1CCCCO1)=O)C2 83404,C#CC1CCC(CN2CC(C)CC(C(=O)NCc3c(C)cccc3F)C2)CC1 83405,C1(NCC2C(CF)CCC2)CCC12CCCCC2 83406,CC(CC(=O)NC1CN(C(=O)C2=CCC2)CC1N(C)C)C(=O)c1ccc(Cl)cc1 83407,CC1(CNC(C2(F)CN(C(=O)Cc3cscn3)C2)=O)NC(=O)NC1=O 83408,c1(C(=O)NCCNC(CCN(CCC)C)=O)ccc(N)c(C)c1F 83409,N1(C(c2cnc(C)[nH]2)=O)CCC(CO)(CNC(=O)CCN2CCNC(=O)C2)CC1 83410,c1(C(N2CC(NC(CCCN=[N+]=[N-])=O)C3(C2)CC3)=O)cc2scc(Cl)c2[nH]1 83411,C#CC1CN(C(=O)C(C=C)CC)CCN1C(C1CCN1C1CCCC1)=O 83412,C1(CN(C(C(C)SCC)=O)C)CCN(C(=O)C(O)CC2CCOCC2)CC1 83413,C#CCC(CC(F)F)C(=O)N1CC(CNC(=O)C2=C(Cl)CCCCC2)(OC)C1 83414,Cc1c(CCC(=O)NC(C)CC2CN(C(=O)C(CCO)N(C)C)C2)cnn1C 83415,c1(C(=O)NC2CN(C(CCCCC#C)=O)CC(O)C2)cncc2n[nH]cc12 83416,C1(CNC)C2CCC(C2)N1Cc1ccc(-c2cccc(C(=O)O)c2)s1 83417,c1(CC(=O)N(CC(C)(C)NC(C(C)O)=O)C)cnnn1C 83418,c1(NCC(C2CC2)SC)cc(Br)ccc1S(=O)(=O)N(C)NCc1ccc(Cl)nc1 83419,CCC(CC(=O)N(C)CCOCCN(C)C(c1ccc(COC)s1)=O)OC 83420,C1(C(=O)NC(C=C)C)CCCN1NC(=O)c1scnc1C 83421,c1(CC(=O)NCCNC(C(CCC)(C)C)=O)ccc2scc(C)c2c1 83422,c1(NC(=O)NC2(CCNC(CC)=O)COC2)cc(C(F)(F)F)nn1CC 83423,CC1CCCCN1S(=O)(=O)NCc1ncc(F)cc1F 83424,Cn1cccc(C(N2CCC(C(=O)Nc3cnc(Cl)cc3I)C(O)C2)=O)c1=O 83425,C(C(CC1CC1)C(=O)NCC1C2CCCCC12)NC(c1ccc(CC)o1)=O 83426,c1(C(=O)NC2C(CNC(c3c(=N)cc[nH]c3)=O)C2)cccn2nccc12 83427,CC1CCN(Cc2ccc(Cl)cc2Cl)CC1NC(c1cnn(CCF)c1)=O 83428,CCCC(CNC(C1CCCCCN1C)=O)C(=O)NC1CCCCC1CCO 83429,N=c1[nH]cc2c(c1C(N1CC3(CCN(C(=O)CNC=O)CC3)C1)=O)CCC2 83430,N1(C(CCCC(C)O)=O)CCCC12CCN(C(c1cc(Cl)c(Cl)[nH]1)=O)C2 83431,C1(C(=O)NC2(C)C(C)CCC2)C2CCC(C2)N1C(c1ccc(F)s1)=O 83432,C12(C(=O)NCC3(NC(c4ncc(NC)nc4)=O)CC3)CCCCC(=O)N1CCC2 83433,CCCCCC(C)(C)C(=O)NCC(C)NC(c1nnn(C(C)(C)C)n1)=O 83434,c1(CC(N2CCC(CNC(c3cccc(C)c3)=O)CC2)=O)cccc2nsnc12 83435,N1(CC)CCCC2(CCCN2C(c2cccc3c2OCCN3)=O)C1=O 83436,c1(C(N2CCC3(CCC(=O)N3)CC2)C(=O)NC)ccc2c(c1)C(=O)N(C)C2 83437,C=CCCCC=CC(=O)NCCC1(NC(=O)C(F)n2ccnc2)CCCC1 83438,C12(C(=O)OCCN3C(=O)CCC3=O)CCOC1CCOC2.C12CC1CNC2 83439,c12ccc-1cc2[N+](=O)[O-].Cc1cc(O)cc(O)c1C(=O)NCc1csc(CO)n1 83440,N1(C(C(CC=CC)C)=O)CCc2cc(CNC(c3ccco3)=O)ccc2C1 83441,c1(C(N(C)CC)=O)cc(NC(c2ccc(-c3cccnc3)cc2)=O)cn1C 83442,c1(CC(N2CC(F)(C(=O)NCC3COCC(C)O3)C2)=O)cccc2ccoc12 83443,N1(C(CNS(N)(=O)=O)=O)CCOCC(CNC(c2ccc(-c3ccco3)o2)=O)C1 83444,C(=O)(CCCCC(C)(C)C)NC(CC)CNC(c1ccc(C2CC2)nc1C)=O 83445,CN1C(=O)C(NC(c2cccc(C#N)c2Cl)=O)c2cc(Br)ccc21 83446,N1(CC(=O)NC(C2(O)CCN(C(C3(C=C)CC3)=O)C2)C)OC(C)(C)CC1=O 83447,C(=O)(CC(C)C(=O)NCC=CCC(=O)NCC1(CC(N)=O)CC1)OC 83448,N1(C(C(C)C(F)F)=O)CCN(C(C2(C#N)CCSCC2)=O)CC1CF 83449,N1(C(C2C3CN(C(C4N(C)CC(O)CC4)=O)CC32)=O)CCC12CCOCC2 83450,N1(CN2CCN(c3ccc(-c4ccc(SC)cc4)cc3)CC2)CCC12CCOC2 83451,C=C1CC(NC(=O)COc2ccccc2C)N(c2ccnc(C3CC3)n2)C1 83452,CC(C)S(=O)(=O)C(C)C(=O)NCC(C)(C)NC(=O)Cn1cc([N+](=O)[O-])ccc1=O 83453,c1(C(=O)NC(C2CCCCC2)C(=O)NCCC)oc(C)nc1C 83454,C#CC1CN(C(C2(NC(C3CC3(F)Cl)=O)CCSC2)=O)CCO1 83455,C1(C)(OC)CN(CC(=O)NC(CCOC)CNC(=O)C(F)CN(C)C)C1 83456,C1(CC(=O)N(C2CCN(C(=O)CC3(O)CCC3)C2)C)CC2(CCC2)C1 83457,c1(C(=O)NCC2CC3(CC3)CN2C(C23CC=CC(C2)OC3)=O)ccc2c(n1)CCC2 83458,C1(CNC(C(CCC)F)=O)N(C(=O)CN2CC(C)(OC)C2)CCCC1(C)C 83459,N1(C(C(c2n(C)ncc2)O)=O)CC2(C1)CN(C(=O)C(F)C(C)(F)F)C2 83460,C1(C(=O)NC(Cc2ccc(C)s2)C)CCCN1S(=N)(=O)N(C)C 83461,N1(C(C2(CC)CC2(F)F)=O)CCC(CCNC(=O)CCCNS(C)(=O)=O)CC1 83462,CC(C)C(F)C(=O)NC1(CNC(c2cscc2C#N)=O)CCOC1 83463,C(c1ccc(S(N)(=O)=O)cc1)=CC(=O)NC(CCNC(C(CC(C)C)C)=O)C 83464,CC1C(=O)NC(=O)CN1C(=O)C(CN=[N+]=[N-])NC(c1ccc(C(F)F)o1)=O 83465,N1(C(CC2N(C(CC3N(C)CC=CC3)=O)C3C(C2)C3)=O)CCCC12CCNC2=O 83466,c1(C(=O)NCC2CC(NC(CC(COC)(C)O)=O)C2)ccc(P(C)(C)=O)s1 83467,Cc1nnc(O)c(C(=O)NCC2CC3CN(C(c4ccccc4F)=O)CC23)c1C 83468,C(=O)(C1=CCCOCC1)NC(C(C(=O)NC1(CC)CCOCC1)C)C 83469,C(=O)(C(CO)C(F)(F)F)NC1CN(C(c2cccc(C(C)(C)C)c2)=O)CC1SC 83470,CC1OCCC1CC(=O)NCC1(CNC(c2cncc(NS(C)(=O)=O)c2)=O)CC1 83471,c1(OC)ccc(CC(=O)NC2CCC2NC(c2sc(N)nc2C)=O)cc1F 83472,C1(C)(C(N(CC(CNC(c2nn(CC)c(O)c2)=O)C)C)=O)COCC1(F)F 83473,C=CCC(C)C(=O)NCCOC1CN(C(=O)CC2COC(C)(C)C2)C1 83474,CCCC(CCC)C(=O)NCCNC(c1c[nH]nc1-c1ccccc1Br)=O 83475,Cc1cnc(CC(=O)N(C(CNC(=O)CCCN2CCCCC2)C2CC2)C)s1 83476,N1(C(CCOCC(C)C)=O)CC(NC(C2C3CCCCCC23)=O)CC(F)C1 83477,CC(C)CCCCN(C(=O)C(n1cc(-c2cnc(C3CC3)s2)nn1)C)C 83478,C1(C(=O)NCC(CC)(CC)NC(=O)Cc2ccc(C)c(O)c2)CC12CCSCC2 83479,C(=O)(C(C)(F)C(F)(F)F)NCC(CC)NC(c1ncoc1-c1cc(C)no1)=O 83480,c1(C(=O)NC2CCN(C(CCSCC)=O)CC2C)cc(Cl)c(F)c(Cl)c1 83481,N(C(=NCCc1ccns1)NCC(C)(C)C(F)(F)F)CC(C)C 83482,C1(C(=O)NC2CC(NC(c3ncn(C)n3)=O)CC2O)CCc2ncncc2C1 83483,c1(C(=O)NCC(C)CN(C)C(c2cncn2C2CC2)=O)cc2ccccn2n1 83484,N1(C(=O)Nc2ccc(C)cc2)CC(NC(=O)C(C)n2cncn2)CC(C)C1 83485,Cc1ccccc1NC(=O)NC1CC(C(=O)N(CC(C)CO)C(C)C)C1 83486,C1(C)(CNC(COC(CC)C)=O)CCCN(C(c2cc(C(C)(C)C)n[nH]2)=O)C1 83487,N12CCCC(C3(CC3)CC1=O)C2.CCCCCN(C(=O)CCc1cnn[nH]1)C(C)C 83488,O=C(CCCCn1ccnn1)NC1(NC(=O)C(N2CC3(CCC3)C2)=O)CCCCC1 83489,N1(C(CC2COCC(C)(C)O2)=O)CCCC(N=c2cc[nH]cc2C#N)CC1 83490,C(=O)(C(=O)N=S(C)(C)=O)N1CCC(C)(NC(C2C(=C)CC2)=O)C1 83491,C1(CNC(C2(CC(C)C)COC2)=O)CN(C(=O)CC2CC(O)C2(C)C)CC1C 83492,C(=O)(C#CC1CCCCO1)N1CC(CNC(C(C)NC(CC)=O)=O)C1 83493,CC(C)CC(CC(=O)NC(C)COC(F)(F)F)NC(c1cncc(Cl)c1)=O 83494,N1(C(C=CCN(CC)CC)=O)CC2(NC(=O)C(CCSC)OC)CCCC2(F)C1 83495,CCC(C)C(C(=O)NC1CCN(C(=O)CCCF)CC1)N(C)C 83496,c1(CC)nnc(C(=O)NCCCN2CCC(OCCF)C2)s1 83497,c1(C(C)NC(C2CCN(C(=O)CCCC3CC3C)C2)=O)nn(C)cc1O 83498,C1(NC(Cn2c(C)cnc2)=O)CN(C(c2cncc(N)c2)=O)CCC1CO 83499,C1(NC(C(CCC)OC)=O)CN(C(C2CCC(=O)O2)=O)C2CCCCC12 83500,c1(NC(C(CC2CCC2)NC(CNC(C2C(C)C2)=O)=O)=O)cc(CO)ccc1C 83501,C1(CC(N2CC(NC(=O)C(c3ccc(Cl)cc3)=O)C3C2C3)=O)CN2CCC1CC2 83502,C12(C(N(CCCNC(=O)C(=O)N(C)CC)CC)=O)CCC(CC)(CC1)OC2 83503,N1(C(CC2ON=C(C)C2)=O)CCCC(C)(NC(c2cncc(C3CC3)c2)=O)C1 83504,c1(C(=O)NC2(CN(C(=O)Cc3ccon3)C)CC2)cnnn1C 83505,c1(CCC(=O)OCC2(CCC3CCCCC3)CCOCC2)ccc(F)nc1 83506,C1(CCC=C)(C(N2CC(C(=O)NC)C2)=O)CN(C(=O)C(C2CC2)C2CC2)C1 83507,CCCCCC(C)CC(=O)NC(CCN(C(=O)CCS(C)(=O)=O)C)C(C)C 83508,C1(CNC(CCC(N)=O)=O)(NC(C2CC(=O)N(CCC)C2)=O)CC2CCC1CC2 83509,c1(C(C)COc2ccccc2)nc(-c2ccnc(Cl)c2)nn1CCC(F)(F)F 83510,CC1CN(C(C2C3CCC2(c2ccco2)C3)=O)CC1CNC(=O)CN(C)C 83511,C1(C2CN(C(=O)COc3cccc(Cl)c3Cl)C2)(NC(c2nc(C)nn2C)=O)CC1 83512,C1(C(=O)NC(C(C)C)c2nc[nH]n2)(CC)CCCN1C(c1ccncn1)=O 83513,c1(OC)cc(CNC(C2(CNC(c3oc(C)cc3C)=O)CCC2)=O)ncn1 83514,CC1CC(C(=O)NC(C)(C)CN(C(=O)COc2ccc(CC#N)cc2)C)C(=O)O1 83515,C#CC(C(C)OC)NC(=O)CC1CCN1C(c1cn(CC)nn1)=O 83516,CCC(Cc1cn(CC2CCCN2C(c2nscc2C)=O)nn1)C(=O)NC 83517,C(=O)(C#CC1CCC1)N1CCC(CNC(CSc2n(C(C)(C)C)cnn2)=O)C1 83518,C(=O)(C1=NNC(C(F)(F)F)C1)N(CC(C)NC(CCC(=O)c1ccc(C)s1)=O)C 83519,N1(C(CCC(C)OC)=O)C2CCC1CC(N(C(=O)CCc1cc(C)no1)C)C2 83520,Cc1noc(N)c1C(=O)NCc1cc(C(=O)NC(C)Cc2ccccn2)n(C)n1 83521,C1(NC(C(C(C)O)NC(C)=O)=O)CCSC12CN(c1nc(C)ns1)C2 83522,c1(C(N2CCC(CC=C)(NC(C(C=C=C)C)=O)C2)=O)cc(=O)c2ccncc2o1 83523,C1(OC)CN(C(c2ccc(CO)cc2)=O)CC1NC(c1scnc1C)=O 83524,c1(NCCNC(c2[nH]c(C)c(C(=O)OC)c2C)=O)ccc(C)nc1C(=O)NCC 83525,N#CC1CN(C(C2CCCN2Cc2cccc(F)c2OC(F)(F)F)=O)CCO1 83526,C(=O)(C1=CC2CCCCCCC12)NCCC(C)NC(=O)C(c1cccc(F)c1)O 83527,N1(C(C(N)=O)=O)C2CCC1C(F)C(NC(c1cc(Cl)n[nH]1)C1CCCCC1)C2 83528,C(C(=O)C(N)C(C)C)NCc1c(SC)cccc1 83529,c1(C(=O)OC)cc(F)c(F)cc1NC(c1ncncc1-c1c(F)cccc1Br)=O 83530,c1(CNC(c2n(C)cnc2Br)c2nnnn2CC(F)F)cccn2ccnc12 83531,c1(C(=O)NCC(c2ccccc2)NC(C2(CC)CCOC2)=O)cccc(C)c1Cl 83532,Cc1occc1C(=O)NC1C=CC(CNC(=O)CCN(CC(C)C(C)C)C)C1 83533,Cc1nc(C)c(C(N2CC3(NC(C4CCC(C)C4)=O)CC2C3)=O)c(C)n1 83534,CC1CN(C(=O)CS(=O)CC)CC1(C)C(=O)NCC(N1CCCC1)=O 83535,C=CC1OCCC1C(=O)NC1(C(=O)NCCSC(F)F)CC(O)C1 83536,N1(C(c2cc(C)c(C)nn2)=O)C2COCC1CC(O)C2 83537,C1(C(=O)NC2(CC#C)CCC2)(NC(=O)CC2CC(=O)NC2=O)CCN(C)C1 83538,C(=O)(C1CCOc2ccccc21)Nc1c(C#N)ncc(Br)c1 83539,c1(C(=O)NC2(C)CN(C(C3CCCN(C)C3)=O)C2)cnn2ccn(C)c12 83540,c1(OC)cc(C)cc(C(=O)NC2(C)CC(NC(C34CC3CNC4=O)=O)C2)c1N 83541,N1(C(CC2(OC)CCC2)=O)CC(C)CN(C(c2cncc(C)c2Cl)=O)CC1C 83542,C(=O)(C(F)(F)CC(C)C)NC1CCN(C(C2C(c3n(CC)cnn3)C2)=O)CC1C 83543,N1(C(c2cc(OC(C)C)ncc2)=O)CC2(CCCC2NC(C2COC(=O)O2)=O)C1 83544,C1(C2CCC2)(CNC(C(C)(C)OCC)=O)CCN(C(c2cc(CO)on2)=O)CC1 83545,c1(C(N2CC(NC(c3n(C)cc(Cl)c3)=O)C(F)C2)=O)ccc2sncc2c1 83546,C(CC(CC)C(=O)N1CC(CC(=O)NC(CN(C)C)CCO)CC1C)=CC 83547,C1(NC(c2ccc(CNC(=O)C(F)F)nc2)=O)CC2(C1)CC(O)C2 83548,N1(C(CCCCCNS(NCC)(=O)=O)=O)CCN2C(=O)N(CC(C)C)CC2C1 83549,C(c1ccc(O)cc1)=CC(=O)N(CCCNC(c1csc(C(C)C)n1)=O)CC 83550,Cc1cc(C)c(C(=O)NCC2C3CC2N(C(=O)C(CCN(C)C)N(C)C)C3)c(C)n1 83551,S(=O)(=O)(c1cccc(=NCc2nnc(CCO)s2)[nH]1)NCC1CCCN(C)C1 83552,C1(CNC(C(C)C2(O)CCC2)=O)CC(C(=O)N2CCOCC2C(N)=O)=NO1 83553,N1(C(C2C(C=C)C2)=O)CCOC2(CCN(C(C3CN4CCC3CC4)=O)CC2)C1 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83677,Cc1csc2cc(C(N3CC(CO)N(C(=O)CSC(C)(C)C)CC3)=O)[nH]c12 83678,C1(COC)(NC(=O)C=CS(C)=O)CCN(C(=O)CN2CCC(C)C2)CC1 83679,CC(C)C(O)CNC(=O)CCOCCNC(=O)CCn1cncn1 83680,Cc1cc(N2CCC(NC(=O)CC3CCC3)C(F)C2)c(C#N)cn1 83681,c1(C2C(Nc3ncc(Cc4ccccc4)s3)CCC2)ccc2c(c1)OCCO2 83682,Cc1noc(C(C)(C)NC(C2CC(N(C(=O)CCn3cnnn3)C)C2)=O)n1 83683,C(=O)(C#CC1CCOC1)NC1CCC(C)(CNC(CCS(=O)(=O)N(C)C)=O)CC1 83684,C#CC1(C(N2CC(C)(CSC)C2)=O)CN(C(=O)CN2C(=O)CNC2=O)C1 83685,C1(NC(c2c(OC)n[nH]c2)=O)CCN(C(=O)CC(C)F)CCC1(F)F 83686,C(CC(=O)N1CCCCC1C1CC1)(C(C)C)NC(c1cc(C)on1)=O 83687,C(C(C)C)(C(O)C(=O)NC(C1CCCCC1)C(N1CC(C)(CF)C1)=O)OC 83688,C1(NC(C2CC(=O)NC(=O)C2)=O)CN(C(=O)CCCN2CCCC2)C2CCCC12 83689,C(=O)(C(C)CC(C)(C)C)NCC(CC=C)NC(c1c(C(F)F)n[nH]c1C)=O 83690,CC(c1ccccc1)=CC(=O)NC(C)(CO)C(=O)NCCc1[nH]cnc1C 83691,C1(C(N2C(CN(C(=O)C(C)(C)n3cccn3)CC)CCC2)=O)CCS(=O)(=O)N1C 83692,N1(C(C(=O)NC(C)C)c2ncco2)Cc2cccc(F)c2C1 83693,CC(C)CN=c1[nH]c(N2CCN3C(=O)OCC3C2)nc2c1CSC2 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83748,C=CC(C)(CCOC)C(=O)N(C)CCN(C(=O)C(c1ccc(C)cc1)C1CC1)C 83749,C1(C(=O)NC(C(C)C)C(=O)N(C2CCCC2C#N)C)CC2CC(=O)C1O2 83750,c1(NCc2ncc(C)nc2)nc2ccccc2nc1N1CCCC2(C=CCO2)C1 83751,C1(CNC(C(=O)N(C)C)=O)CCN(C(=O)CC(C)(C)Cc2ccccc2)C12CC2 83752,N1(C(CCCOCC)=O)CC(NC(C2(C)CCC(=O)NC2)=O)CC(F)C1 83753,C1(NC(=O)C=Cc2cnccn2)CN(c2ncc([N+](=O)[O-])cn2)CC2(CC2)C1 83754,c1(CC(=O)NCC2(O)CN(C(C34CCCC(C3)OC4)=O)C2)ccc(F)cc1F 83755,N1(C(CC(C#CC)c2ccc(O)cc2)=O)CCCC2(CCCN2C(=O)C=C(C)C)C1 83756,C1(O)(CNC(C2C=CCN(C(CCC3C(C)(C)C3)=O)C2)=O)CCCCCC1 83757,C#CC(C1CCc2ccccc21)NC(=O)Nc1ccnc(N2CCC(O)CC2)n1 83758,c1(CN(C(CN(C(=O)C2=CCCC2)CC#C)=O)C)ccc(C)nc1 83759,C1(NC(CCN(C(C)=O)C)=O)CN(C(=O)CCN(C)CCO)CCC1C 83760,N12CC(C3(CC3)C1)N(C)CC1(CC1)C2=O.C12(CC(=O)OC)COC(C(=O)OC)(C1)C2 83761,c1(N2CC3C(C)(C)C(C3)C2)nc2ccccc2nc1NCC1CCC(F)C1 83762,Cn1ncc([N+](=O)[O-])c1C(=O)NC1CCC2CC1CN2C(C1CC=CCO1)=O 83763,N1(C(C(C)(C)C2CCCO2)=O)C2CCC(C2)C1C(N1CCC(N2CCCC2)C1)=O 83764,C1(NC(C(C)(C)OC)=O)CC(NC(c2cc(N)ccc2SC)=O)C12CCC2 83765,C(CC(F)F)(C(=O)NC1CCC(O)CC1)N(C(=O)CC1OCCCO1)C 83766,c1(COC)nn(C)c(Cl)c1C(N1CCN(C(=O)CC2CC(C)=NO2)C(CF)C1)=O 83767,c1(CC)nnc(O)c(C(=O)N(C2CCCN(C(=O)C(C)(CC)OC)C2)C)c1CC 83768,C1(CC(=O)NC2CC(NC(=O)CC3CCNC3=O)C2)CCCC1(F)F 83769,c1(C(=O)NC(CN(c2nccc(CC(=O)OC)n2)C)C)coc2ccc(C)cc12 83770,c1(CCC(=O)NCCC(C)N(C)C(c2cccn2C2CC2)=O)cc(C2CC2)on1 83771,C(=O)(C(C)C(C)NC(c1ncoc1C1CC1)=O)N(CC=C)CCOC 83772,C1(C(=O)NC(C(=O)NCCC)CC)CC(NC(C2CC(F)CN2C)=O)C12CCC2 83773,Cc1cc(C(=O)NCC(CC2CC2)C(=O)NC2CC2C(C)(C)C)ccc1F 83774,C1(CNC(CNC(=O)OC)=O)CC2CCC1N(C(=O)C(C)Cc1cccnc1)C2 83775,n1(CC(N2CC(OC)(CNC(c3ocnc3C)=O)C2)=O)cc([N+](=O)[O-])nc1C 83776,C1(C(N2CCC3(C(CNC(C(CC)(F)F)=O)C3)CC2)=O)CCc2ncccc2C1 83777,C12(C(=O)NCCC(=C)CNC(C3CNC(=O)N3)=O)CCCCC1NC(=O)C2 83778,CCC(O)C(C)(C)C(=O)N1CCCNC(=O)C(C)C2(CCCC2)C1.C1(CC)CC1 83779,C(=O)(CC(C(F)(F)F)C1CCOCC1)N1CC(CC(CC)O)C1 83780,n1(CC(=O)NCCOCCN(C(CCC=C(C)C)=O)C)ncn(C)c1=O 83781,CCC(CC(F)(F)F)C(=O)NC1(CCNC(=O)COCc2nc[nH]n2)CC1 83782,c1(C(=O)NC2C(F)CCN(C(CN(C(C)=O)C)=O)C2)c(C)nn2c1CCCC2 83783,c1(C(=O)NC(c2cn(CC(N)=O)nn2)C)cc2cccc(C(F)(F)F)c2nc1O 83784,N1(C(c2ccc(C#C)c(C)c2)=O)CCC2CCC(C1)N2C(=O)Cn1ccnc1C 83785,N=c1nc(O)c(C(N2CCCCC2C(=O)NCCC2CCSC2)=O)c[nH]1 83786,c1(C(=O)NC2C(CNC(c3cccs3)=O)CCCC2)cc2ccccc2[nH]1 83787,N(C(=NCC(C1CC1)N(C)C)NC1CC1)CC(=O)Nc1ccc(SC)cc1C 83788,c1(C(=O)NC(C)(C(N2CC(O)C(F)C2)=O)C2CCC2)ccc(N)cn1 83789,C(=O)(C(O)CN(C)C)N(CC(C)N(C(=O)COC1CCCCC1)C)C 83790,c1(C(=O)NC2CCCC2NC(C2CCCC2(F)F)=O)cc(F)c(CO)c(F)c1 83791,c1(CC)cccc(C(N2CCC(C(=O)NCCc3cccc(O)n3)C2)=O)n1 83792,C(=O)(C#CC1CCOC1)NC(CC#C)C(=O)NC1(c2cc[nH]n2)CC1 83793,C1(C(=O)NC(C)C(=O)NCC(C)(C)CN(C(=O)CNC(=O)C2CC2)C)CCCCC1 83794,CC1C(NC(c2ccnc(N(C)C)c2)=O)CCN1C(C1CC(c2ccccc2)C1)=O 83795,Cc1cc(=NCC23CC(NC(c4ncc(Cl)cc4Cl)=O)(C2)C(C)O3)c(C#N)c[nH]1 83796,N1(C(CC(C(=C)C)O)=O)CCCc2nc(O)ccc2C1 83797,C1(C(=O)NC(=O)C(=O)NCC2CC3CCCCN3C2)CCC2(CCCC2)CC1 83798,C(=O)(C1=CC=CN2CCS(=O)(=O)N=C12)NC1CN(C(c2c(C=C)cnn2C)=O)C1 83799,N1(C(c2nn(C)cc2Br)C(=O)NC(CC)(C)C)CC(S(C)(=O)=O)CCC1C 83800,c1(C(=O)NC2CCCC(NC(CCc3cc(C)sc3C)=O)C2)ccnc(C)c1N 83801,[N-]=[N+]=Nc1cccc(C(=O)NCC2CCCC2NC(=O)CCc2cc(Cl)cs2)c1 83802,c1(CC(=O)NCC2N(C(C3C(C#N)C3)=O)CC(O)C2)cc2ccccc2s1 83803,c1(C(N(C(CN(C(Cc2cc(C(=O)OC)sc2)=O)C)C)C)=O)cc2n(n1)CCC2 83804,CC(C)CC(C)CC(=O)NCC1(F)CCN(C(=O)COc2ccc(Cl)c(F)c2)C1 83805,C1(NC(CN(C(C(CCCOC)C)=O)C)=O)CC1C1CCCCC1 83806,C(N=c1cc(Cl)nc(C2CCCO2)[nH]1)C1CN(C(C2CCC(C)(C)OC2)=O)C1 83807,N1(C(c2n(CCOC)ncc2)=O)CCC(CNC(c2ncc(Cl)n2C)=O)C(C)C1 83808,C1(CC)CN(C(c2c(Cl)noc2C)=O)CC1NC(=O)CCc1ccncc1 83809,C1(NC(CCCC)CCCC)Cc2cc(OC)ccc2O1 83810,Cc1ccccc1C=CC(N1CCC(C)(CNC(C2C3CCC(=O)C23)=O)C1)=O 83811,c1(CNC(C2CCN(C(C=CC(=O)OCC)=O)CC2)=O)cc(F)c(F)cc1F 83812,c1(OC)cccc(-n2nnnc2C2(NCC3CC4CCC3O4)COC(C)C2)c1 83813,C(CCCN=c1[nH]c(Cl)nc2c1SCC2)NC(C(CCCC)O)=O 83814,Cn1nc(CSc2nc(N3CCC(C)(C(N)=O)C3)cc(O)n2)ccc1=O 83815,Cc1cc(C)c(C(N2CC=CC(NC(=O)CCCc3ccncc3)C2)=O)c(N)c1 83816,Cn1c(C(=O)NCCCC2CCCN2C(=O)CC2(C)OCCO2)nnc1S 83817,c1(CCC(=O)NCC(C)NC(CCC=CC)=O)cccc(C#N)c1 83818,n1(C(C)C)cncc1C(=O)OCC1CC=CCO1 83819,c1(OCC(=O)NC2CC(NC(C3CC(CF)C3)=O)C2)ccccc1Br 83820,N1(C(c2cc(C)ns2)=O)CC2CC(C1)N(C(C1CCC(C)(C)O1)=O)C2 83821,CCCC(C)(O)CC(=O)NC(C)(CC)CCNC(=O)CC1CCCC(C)O1 83822,N1(C(C2OCCC(C)(C)C2)=O)CC(CNC(C2CCC2(F)F)=O)CC12CCC2 83823,C#CCC(C)(C(=O)NC(C(O)CO)C1CC1)NC(=O)C(C)C1(O)CCC1 83824,N1(C(C=Cc2ncc(C)[nH]2)=O)CC(NC(c2cc(C(F)F)n(C)n2)=O)CCC1C 83825,c1(C(=O)OCC(n2cc(CC(=O)OC)nn2)C)nc(OC)c(OC)c(Cl)n1 83826,Cc1cc(NCC2(F)CC(NC(C3(C)CCCOC3)=O)C2)ccc1[N+](=O)[O-] 83827,c1(C(N2CCC(SC(F)(F)F)CC2)C(=O)NCCCCCC)cc(C)nnc1C 83828,Cc1ccc(C2CC2C(=O)NCC2(NC(=O)CC(C)C(C)C)CCC2)c(Cl)n1 83829,Cc1c(C(=O)NC2CC2NC(=O)CC2CCCO2)cccc1C#N 83830,N1(C(c2c(F)ccc(C)c2)=O)CCCN(C(c2cc(Cl)cs2)=O)CC1C 83831,Cc1cnc2c(C(=O)NC3CN(C(c4cnsc4)=O)CC4(CCC4)C3)cccn12 83832,C1(CNC(CC2(N(C(C(COC)(C)O)=O)C)CC2)=O)CC(C(N)=O)=NO1 83833,N1(C(CCNC(N)=O)=O)C2CCC(C2)C1C(N1CC(O)(C(F)F)C1)=O 83834,c1(C(=O)NC2CC(NC(c3cc(Cl)c(Cl)cn3)=O)C2)cnc2cc(Cl)ccn12 83835,C12(C(N3CCCC(CC=C)(NC(=O)C=CC(C)C)C3)=O)CCC(C#N)(CC1)CC2 83836,CC(CC(=O)NC1CSC1)NC(=O)Cc1ccn(C)n1 83837,c1(CC)ccc(Br)cc1C(N1CCCCC1C1CCN(C(=O)COC)C1)=O 83838,C(CCCCCCC(=O)NC1CC2CN(C(c3onc(C)c3C)=O)CC2C1)SC 83839,O=C(N1CC(CN2CCOC2=O)CO1)C1CCCCN1n1cc(C2CC2)nn1 83840,C(=O)(C(CCC)C(C)C)NCCC1CCCN(C(C(CCC)F)=O)CC1 83841,C(=O)(CC(C)(C)OC)NCCC1CCN(C(C2N(S(C)(=O)=O)CCC2)=O)C1.CCO 83842,C1(C(=O)NCCCOC=C)(CC)CCCN(C(=O)C(c2cnn(C)c2)=O)C1 83843,C(=O)(C(C)(C)C(C)(F)F)N(C(C(N1CCCC(C#C)C1)=O)C)CC 83844,C(=O)(CCCCC(F)F)N1C(CCNC(C2CCN(C)C2=O)=O)CCC1 83845,c1(C(=O)NCCC2CC(NC(CSCC)=O)C2)ccc(Br)nc1N 83846,C1(C(N2CC(OC)CC(NC(CCC#C)=O)C2)=O)CC(C(C)(C)C)=NO1 83847,c1(CC(=O)NCC(CC=C)NC(=O)C(O)C=CCCC)ccc(Cl)cc1C 83848,c1(C2(C(N(CCN(C)C(N)=O)C)=O)CC2)ccc(OC(F)F)cc1 83849,N1(C(CCCN(C)C)=O)CCN(C(c2cccc(-n3ccnc3)c2)=O)CC1CF 83850,CC(C(=O)NC1C2CC1CN(C(c1ccnn1C1CCOCC1)=O)C2)C(C)(C)C 83851,CC1(C)CCCC(CC(N2CC(NC(=O)CC3SC(=N)NC3=O)CC(F)C2)=O)C1 83852,C=CCC(C)(C)CC(=O)N1C(C)C2CC1C2NC(c1cnc(O)n1C)=O 83853,C1(CN(C(=O)C=CC(C)(C)C)C)CCN(C(=O)CSc2nncn2C)CC1 83854,CN1CCN(CCN2CCN(C(C3CCCC(c4ccccc4)O3)=O)CC2)CC1 83855,c1(-c2n(CC(C)CO)nc(-c3cc(C(F)F)cs3)n2)cc2cnn(C)c2s1 83856,CC(CC(=O)NC1CCCC(NC(c2ccn(C)c(=O)c2)=O)C1)CC(F)(F)F 83857,N1(C(CC(C(C)C)O)=O)CCC2(CCCCN(C(c3cn(C)c(=O)cn3)=O)C2)C1 83858,C(C)(CNC(=O)C(C)C(C)(F)F)(CC(C)C)NC(CCNC(C(C)C)=O)=O 83859,c1(CC)n[nH]c(=NC(=O)NC2CCCCC2n2ccnc2)s1 83860,c1(-c2ncc(C(N(CCCNC(COC)=O)C)=O)s2)ccc(Br)cc1 83861,C=Cc1cc(C(N2CC(CNC(=O)COC3CCCCC3)C(C)C2)=O)cc(F)c1 83862,c1(C(N(CCOC)CCNC(=O)C(F)(F)CN(C)C)=O)sc(C)c(C)c1C 83863,C(=O)(C1CCCc2nncn21)NC(CNC(C(CCC(C)C)NC(C)=O)=O)C 83864,C1(NC(C(F)=CC)=O)CN(C(c2ccc(-c3cccnc3)cn2)=O)CC1(C)C 83865,C1(C(=O)NCCC(C)N(C)C)CC1C1CN(C(=O)C(C)(C)C2CCOC2)C1 83866,c1(CC(N2CCC(C)(CNC(c3c(C)ncnc3)=O)C2)=O)ccc2nn[nH]c2c1 83867,CC1(C)CCCCC1=CC(N1CC(CNC(C2C3CCCOC23)=O)C(O)C1)=O 83868,N1(CCC)CC(C(N2CC(O)(CNc3ncc(C(F)F)cn3)C2)=O)CC1=O 83869,C1(O)(C(=O)NC2C(NC(c3cc(OCC)n[nH]3)=O)CCC2)CC2(CCOCC2)C1 83870,C1(CNC(=O)Cc2ccsn2)CCN(C(=O)CCC2CCOCC2)CC1O 83871,Cc1noc2cc(C(N3CC(CCNC(=O)CN(C)CCO)C(C)C3)=O)ccc12 83872,CCCC(CC(C)C)C(=O)N1CCOCC(CNC(c2ocnc2C2CC2)=O)C1 83873,c1(C(=O)NCC2(F)CCN(C(C3(CCC)CC(=O)C3)=O)C2)c(C)cc(C)oc1=O 83874,CC1CCN(C(C2CC(=O)N(C)C2)=O)CCN1C(=O)CCN1CCCCC1=O 83875,N1(C(C2N(CCC)C(=O)CC2)=O)CCCC2(CCN(C(=O)CN3CCCC3)C2)C1 83876,C(CC(C(C)C)NC(c1nccnc1C(N)=O)=O)NC(C(C)=C(C)C)=O 83877,CC(C)CC(CNC(=O)CC1(C)CC1)NC(c1ccc(C2CC2)o1)=O 83878,c1(OCCCCC)ccc(-c2nc(C(C)OC)nn2-c2ccnn2C)cc1OC 83879,C(C)(N=c1ccnc(NCCCCNC(c2ncsc2C)=O)[nH]1)C1C(=C)C1 83880,CC(C)(C)[Si](C)(C)OCC1(F)CN(C(c2cnc(C#N)nc2)=O)C1 83881,N1(CC(N2CCC(O)(CN(C)C(c3cn(C)nn3)=O)C2)=O)CCCCCC1=O 83882,c1(NC2CCN(C(CC)C)CC2)[nH]c(=NCC(CC)C(C)(F)F)nc2sccc12 83883,c1(C)cc(COC(=O)C(C)C2CCOC2)no1.C1(NOC)CCCC1 83884,C(=O)(C(C)C(C)(C)C)NC(C1CCCN(C(COc2c(C)cccc2)=O)C1)C 83885,N1(C(C(C)OC)=O)CC2CCC(C1)C2C(N1CCCC1c1ccccc1)=O 83886,c1(C(N(CC(CNC(C(c2cccc(C)c2)=O)=O)O)C)=O)cc2sccc2n1C 83887,Cc1cc(C(=O)NCC2C3CCC(C3)N2C(=O)CCc2cnn(C)c2)c(C)cn1 83888,C(=O)(C(C)(C)CC(F)F)NC1CCN(C(c2cnn(C)c2F)=O)C1C1CC1 83889,C(C(N=c1nc(C2CC2)[nH]s1)C1CCC1)NC(C(C)Nc1ccccc1)=O 83890,C#CCCN=C(NCCOC1CCS(=O)(=O)C1)NCc1cnn(C)n1 83891,C1(C(=O)N(C2CCOCC2)C2(C3(CCO)CCC3)CC2)CC2CN(C(=O)C3CC3)CC2C1 83892,N1(C(COCC=C)=O)Cc2n[nH]cc2C1C(=O)N(C1CCCCCC1)C 83893,C(c1c(NC(=O)C=Cc2sccc2Br)cnn1-c1cc(C)ccn1)=CCCC 83894,c1(CCC(N2CCC(n3cc(CCSC)nn3)C2)=O)cccc(NC(C)=O)c1 83895,c1(CN2CCC(O)(Cc3ccccc3)C2)noc2c1COCC2 83896,CCC(C)CCCC(=O)NC(C1CCCN1C(=O)CSCc1ncc[nH]1)(C)C 83897,N1(C(C2C(=C)C2C(=O)OC)=O)CCN(C(C23CCOC(C)(C2)C3)=O)C(C)C1 83898,c1(C(=O)NC2CN(C(=O)C(C)C(C)O)C2)cc(C(=O)OC)cc(C(F)(F)F)c1 83899,O=C(C1=CCCOCC1)NCC1CN(C(=O)C=Cc2ccc(F)nc2)C1 83900,c12ccc(F)c(c1)C(c1nnnn1C1CC1)N2.C=CC1(OC)CCCC1 83901,N1(C(C(CC(=O)OC)C2CC2)=O)CCc2ccc(N=[N+]=[N-])cc2C1 83902,N1(C(c2c(CC)nn[nH]2)=O)CCC(CF)(NC(=O)CCCN(C)C)C1 83903,CC1CN(C(C2CCN(C)C2=O)=O)CCC1NC(=O)C(C)Cc1cccc(Cl)c1 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83921,N1(C(C(CC=C)C)=O)CCC2(CC1)CCN(C(c1ccc(O)c(Br)c1)=O)C2 83922,c1(CNC(=O)NC(CCCC(C)c2n(C)ncc2)=O)ccc2c(c1)CCNC2=O 83923,CC1CC(NC(=O)CNS(N)(=O)=O)CN(C(=O)Cn2ccc(O)nc2=O)C1 83924,C1(NC(c2c(C)coc2)=O)C2CCCN(C(C3OC4CCC3C4)=O)C2C1(C)C 83925,C1(NCCc2ccc(OC)c(C(F)(F)F)c2)C2CCCC(F)(F)C12 83926,n1(CCC(=O)NCC(CNC(CC2(C)CC2(Cl)Cl)=O)CO)ccccc1=O 83927,c1(C(=O)NC2CCC(N(C(c3c(C)ncnc3)=O)C)C2)cc([N+](=O)[O-])c[nH]1 83928,C1(CNC(=NC)NCc2ccc(N3CCC(O)C3)cc2)CC2C(C1)C2(F)F 83929,c1(CNC(C(CC)F)=O)cccc(NC(=O)CC(C)CN(S(=O)(=O)CCC)C)c1 83930,c1(-c2ccc(OCCC)cc2C)ccc2cc(C(=O)Nc3cnnn3C)[nH]c2n1 83931,N1(C(C2OCC(C)C2)=O)CCC2(CCN(C(c3ccc4cc[nH]c4n3)=O)C2)C1 83932,c1(C(=O)NC(CC)CN(C(C2CCC(CCO)CC2)=O)CC)cnc(O)c(F)c1 83933,Cc1cc(O)ccc1NC(=O)N(C1CC1)Cc1ccsc1 83934,C1(NC(C2(C)ON=C(C)C2)=O)CC2(CCN(C(c3sc(C)nc3C)=O)C2)C1 83935,N1(C(c2c(C)ccc(OC)c2)=O)CCCCC(CNC(=O)Cc2cnc[nH]2)CC1 83936,C1(C(=O)OC)CCCC(NC(=O)CCOCc2ccnc(O)c2)CC1 83937,C1(C(=O)NCC2CC23CC3)(NC(C2CC(O)(CC#C)C2)=O)CCCCC1 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83955,N1(C(CC2CCN(C)C2)=O)CCC2(CCN(C(C3CC4CC4C3)=O)CC2)C1 83956,c1(-n2ncc(NC(=O)CC3CC(NC(=O)C#CC4CC4)C3)c2)ccc(Br)cc1 83957,n1(CC(=O)NCC2OCCC(NC(C(COC)COC)=O)C2)nc(C)n(C)c1=O 83958,N1(C(c2c(C)cc(F)nc2)=O)CCC2(C1)CN(C(C1C(C)(C)C1(C)C)=O)C2 83959,C1(CCNC(CN(S(C)(=O)=O)C)=O)COCCN1C(c1ccc(CO)cn1)=O 83960,C(N=c1[nH]c(Cl)ncc1[N+](=O)[O-])C1CCN(C(c2cc3n(n2)CCCC3O)=O)C1 83961,N1(CC(=O)NC2CCC(NC(C3(CCOC)CC3)=O)C2)CCC(F)CC1 83962,C1(CC)CCN(C(=O)Cc2cnnn2C)C1NC(C=CC(=O)NC(C)(C)C)=O 83963,N1(C(c2c(Cl)ccc(C)c2)=O)CC2CC(C1)N(C(C1CN(C)CCO1)=O)C2 83964,N1(C(c2ccc(C)o2)=O)CCC2(CC1)CC2(C)C(=O)Nc1cccnc1 83965,Cc1nc2ccc(C(N3CC4CN(Cc5nccnc5Cl)C4C3)=O)cc2o1 83966,c1(OC)ccc(OC)c(CC(=O)NCC2CCN(C(c3oncc3C)=O)CC2)c1 83967,c1(C(N2CC3CCC(C2)N3C(=O)Cc2ccnc(O)c2)=O)cccc2nsnc12 83968,c1(C(N2CCCC(CNC(c3nc(C(C)OC)oc3)=O)C2)=O)ccc(Cl)cc1N 83969,CCCC(C(=O)OC(C)(C)C)C(=O)NCCCN(C(=O)C(C(C)O)SC)C1CC1 83970,CCCCC(O)CCC(=O)N1CCC(CNC(=O)CC2CC(C(F)F)C2)C1 83971,C1(CC(=O)NCC(c2cccc(C)c2)NC(=O)C(Cl)=CCl)CCn2cncc2C1 83972,C1(C(=O)NC(C#CC#C)(C)C)CC(C)CCN1C(C1CC1C#N)=O 83973,Cc1nc(C)c(C(=O)NC(C)CCCNC(=O)C(c2cccnc2)C)[nH]1 83974,c1(CCC(=O)N(C)CC2CCC(CNC(=O)C(F)F)CC2)ccc(CO)cc1 83975,C(=O)(C(C)CC(N)=O)NCC(CCCC)NC(=O)C(C)Cc1ccccc1C 83976,c1(CC)c(C(N2CCOCC2CNC(=O)C=C(C2CC2)C2CC2)=O)cnn1CC 83977,CC(CC(=O)N1CCCCC1C1(NC(=O)CCCC(F)(F)F)CC1)CC(C)(C)C 83978,N1(C(c2cc(C3CC3)no2)=O)CCC2(CCCN2C(=O)C2=CCCO2)C1 83979,CC1C(NC(c2nnc(O)nc2O)=O)C(C)CCN1C(=O)C=CC1CCCC1 83980,c1(OCC)ccc(NC(c2sc(Br)c(C)c2Br)c2nnnn2C)cc1Br 83981,c1(C(=O)NC2C(C)(CNC(=O)OC(C)(C)C)CCCC2)n[nH]c2cc(Cl)ccc12 83982,CC1CC(CO)CN(C(=O)CCCCCNC(c2coc(C(N)=O)c2)=O)C1 83983,Cn1cc2c(n1)CCC(C(=O)Nc1cc(NCc3ccc(Cl)c(O)c3)ncn1)C2 83984,C=C(CCN(C)C)C(=O)N(C1CC1)CC1CC1 83985,C1(C(N2CCCC2CNC(=O)CCOC2CCOC2)=O)(OCC)CCCC1 83986,N1(C(c2nn(C)c(CO)c2)=O)CCC(NC(=O)Cc2ccccc2)(CO)CC1 83987,C(=O)(CCCCC(=O)NC(=O)C=C(CCC)CCC)NC1CC(CCCCC)C1 83988,N1(C(C(N2C(=O)CCC2=O)CC)=O)CCOC(CNC(C2(O)CCC2)=O)C1 83989,C1(C(N2CC3CC3(CO)C2)=O)(NC(CN(CCOC)C)=O)CCN(C)C1 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84059,C1(CC)(CC)CC(NC(c2cc(O)nc(C)n2)=O)CN1C(=O)C(C)OC 84060,N1(C(C#CC2(C)COC2)=O)CCC2CCNC2C1.c1(C=O)nccnc1C(N)=O 84061,N1(C(C)C)CCCC(CCNC(C2CCCCN2C(=O)COC2CC=CC2)=O)C1 84062,c1(NC(c2ccc(C(C)(F)F)cc2)C)nc2ccccc2nc1NC1CCC1 84063,CC(CC(=O)N1CC2(NC(=O)C=Cc3nccs3)CCCC2(F)C1)CC(C)(C)C 84064,C=CC(C)(C)CC(=O)NCCCN(C(C1CC(O)CN1c1ccncn1)=O)CC 84065,C(=O)(CCCN(C)N=O)N1C(C)CC(CNC(=O)C(C)(C)N(C)C)C1 84066,c1(C(N2C3CN(C(c4c(OC)cccn4)=O)C(C3)C2)=O)oc2ccccc2c1C 84067,C1(C(N(CCOCCC(=O)NCc2nccc(C)c2)C)=O)C2CCC(C2)C1C 84068,C(C)(CNC(C1(c2ccno2)CC1)=O)(C(C)C)NC(c1c(SC)ccs1)=O 84069,N1(C(C2CCC(COCC)CC2)=O)CCC2CC2(NC(=O)CC(C)C(C)C)CC1 84070,CC1=CCC(C(N2CCC(C)(NC(C3CSC3)=O)C2)=O)CC1 84071,S(=O)(=O)(C1(CNC(=O)NC2CCC(c3cccc(Cl)c3)C2)CC1)N(C)C 84072,N1(C(C(C)n2ccnc2)=O)CCC(CNC(C2(c3cccs3)CC2)=O)CC1 84073,C1(NC(CN2CCC(C(N)=O)CC2)=O)CC2CCC(C1)N2C(c1ccnnc1)=O 84074,N1(c2nc(OC)c(F)c(C)n2)CCCC2(CCN(C(=O)C(C)(C)SC)C2)C1 84075,C1(C(NOCCCCCC)=O)CCCN(C(=O)Cc2cnccc2C)C1 84076,N1(C(Cc2cccc(C#C)c2)=O)CCCCCCC1C(=O)N(C(C)C=C)C 84077,C(=O)(C(C)(C)C(N)=O)N(CCC(C)NC(c1cnn(C(C)C)n1)=O)C 84078,N1(C(C(Cc2ncn(C)c2)O)=O)CCC(F)(CNC(=O)C(S(C)(=O)=O)C2CC2)CC1 84079,n1(C(C)(C)C)cnc(C(N(C2CCC(NC(=O)C(=O)N(C)C)C2)CCC)=O)c1 84080,C=CCC(CC(C)C)C(=O)N1CC(C2CC2)C1C(=O)NC(C)(C)C 84081,c1(NC(C)=O)ccc(C(N2CCCC(N(C)C(c3cccn3C)=O)C2)=O)cc1F 84082,N1(C(CC)C(=O)Nc2nccnc2C)CCc2ccccc21.C12CC1CNC2=O 84083,CN1CC(C(=O)NCCCN(C(C2CCCS2)=O)CC2CCCC2)CC1=O 84084,c1(C(N(CCNC(C2CC3CCC3C2)=O)CC2CC2)=O)cc(F)cc2nc[nH]c12 84085,c1(C(N2C(CNC(CCC=CCC=C)=O)COCC2)=O)cc(F)cc(C)c1N 84086,Cc1cc(C(C)NC(C2CCN(C(c3ccnnc3)=O)C2)=O)on1 84087,CCCC(CNC(=O)COCC(C)(C)C)C(=O)NCc1ncnn1C1CC1 84088,C(=O)(CCC(C)(F)F)NCCSCC(N1C(CCCCC)CCC1)=O 84089,C(=O)(CCCCC(=O)NCC(O)CN(C(=O)C(O)C1=CCCCC1)C)OC 84090,CN1CCC(=CC(N2CC3C(CNC(=O)CC(O)(C4CC4)C4CC4)C3C2)=O)CC1 84091,Cc1csc2c(CNC3CN(C(=O)CC4=CCCC4)CC34CCC4)ncnc12 84092,c1(COC)ccc(C(C(=O)NC2CC2)N(C)CCOC)nc1.C1(=O)C(C)ON1 84093,C(CC(O)C(=O)NCCC(C(=O)NCC(O)C(C)C)OC)SC 84094,c1(C2(C(=O)NCCCN(C(=O)COC(=O)CO)C)CCC2)c(F)cccc1F 84095,C(=O)(CC(C)(C)CN(C)C)NCC(C(N1CCC(CC)C1C)=O)(C)C 84096,C(CN=C(NC1CCC1)N1CCC(O)(C(F)(F)F)C1)=CCOC 84097,N1(C(c2cc(C3CCC3)[nH]n2)=O)CC2CCC(C1)N2C(C1(CC(F)(F)F)CC1)=O 84098,c1(C(N2CCCC2c2cccc(Cl)c2)=O)cc(Cl)c(F)cc1[N+](=O)[O-] 84099,c1(CC(=O)NC2CCN(C(c3c(C)ncnc3)=O)C2)cnn2c1OCCC2 84100,N1(C(C2(C#C)CCCC2)=O)CC2=C(C1)CN(C(c1cc(F)cc(Cl)c1O)=O)C2 84101,c1(OC(C(=O)NCCN(C(=O)C(O)C(C)C)CCC)C)cccc(C(C)=O)c1 84102,CC(C(F)(F)C(F)(F)Br)Oc1ccc(OCCc2ccccc2)cc1 84103,C(=O)(C(Cc1ccco1)NC(=O)CC1CCCOC1)N(CCC#C)C 84104,N1(C(CCCCC)=O)CCN(C(=O)CCCCCn2cnnn2)CC1COC 84105,c1(CC)cc(C(=O)N(C2CCN(C(=O)CCc3cnc(C)o3)CC2)C)c(C)o1 84106,c1(C(=O)NCC2CC(NC(c3ccnc(O)c3)=O)C2)cccc2c1CCC2 84107,C(CC(CNC(C1(C)CC(F)C1)=O)NC(=O)COCCF)OC 84108,c1(CC(N2CC3CC(CNC(C4(C)CC4)=O)C3C2)=O)ccc2ncsc2c1 84109,N1(C(CC2N(CC)CCOC2)=O)CCC2OCCN(C(=O)CCOC)C2C1 84110,C1(CC(=O)N(C2CCN(C(=O)C(C)CC3CC3)C2)CC#C)CSCCO1 84111,C12(CC)CCCC(CN1C(C1CCCC(F)C1)=O)C2.C(c1cn(C2CCCC2)nn1)=CC 84112,C1(C(=O)NC2CN(C(c3cc(SC)oc3C)=O)CC2C)(OC)CCOCC1 84113,S(=O)(=O)(c1cccc(C(F)(F)F)c1)N1C(C2CCN(C(C(=C)F)=O)CC2)CCC1 84114,c1(C(CC)=O)ccc(OCC(=O)NC(CNC(c2ccnnc2O)=O)CO)cc1 84115,c1(C(C)C)cc(F)ccc1C(=O)NCC(CNC(=O)C(C)OCC1CC1)CO 84116,C1(CNC(N(C2CCCN(C)C2)C)=O)CCCN2CCCCC12 84117,CC(C)CCCCC(=O)NC1(C)CC(NC(c2cnn(-c3ccccc3)c2)=O)C1 84118,c1(CC)c(C(=O)N(C2CCN(C(=O)C(C)Sc3ccccc3)C2)CC)nnn1C 84119,C1(=O)CC(CC(C)C)N1.Cc1noc(-c2noc(Cc3cccc(O)c3)n2)c1C 84120,C1(C(=O)NC2CC(C)(NC(=O)C3=CCOCC3)C2)CCc2ccccc2C1 84121,N1(C(CN2CCN(C(C=CC(CC)C)=O)CC2)=O)CC2CCCCC2C1C 84122,C(C)(CNC(c1c[nH]nc1C(F)F)=O)(C(C)C)NC(C(CO)OC)=O 84123,C1(OC)CCC(C(=O)NC2C3CC2N(C(C2(C)CC=CC2)=O)C3)CC1 84124,c1(NC(N2C3CCCC(O)C2CC3)=O)cnc2ccc(F)cc2c1 84125,N(C(=NCCF)N(C)CCS(=O)(=O)c1ccccc1)C1CCCC(C(N)=O)C1 84126,C1(C(=O)NC(C(C)C)CNC(c2cccc(O)n2)=O)CCCCC1(F)F 84127,c1(C(=O)NCC2CCN2Cc2ccc(C(=O)O)c(F)c2)ccc2c(c1)COC2=O 84128,C1(O)(CCNC(=O)C(C2CCCCC2)O)CCCN(C(=O)CC2CCC2)C1 84129,CCC(CNC(C1CCOC1)=O)(CC)C(=O)N1CCC(C(=O)OC)O1 84130,N1(C(c2c[nH]c(=NC)s2)=O)CCC2(CC1)CC2C(N1CCOC(C(C)(C)C)C1)=O 84131,c1(C(=O)NC2(CNC(=O)C(O)C3CCC3)CCOC2)cc2ccccc2cn1 84132,Cc1c(C(N2CCC(C(C)NC(c3cnc(N(C)C)nc3)=O)CC2)=O)nnn1C 84133,C1(COC)(NC(=O)CN)CCN(C(=O)CCC2(C)N=N2)C1.n1(C2CC2)cccn1 84134,C1(CC(=O)NC2(C)CN(C(c3cc(C)oc3)=O)C2)CCC(=O)NC1 84135,C(=O)(C(C)(C)C(N)=O)N(C)CCNC(c1cnc(Cl)n1C)=O 84136,N1(CC)CCCC(C(=O)NC2C=CCCC2C(=O)NCC2(CC3CC3)CCC2)C1 84137,CC(=O)CC(C)(C)C(=O)NCCC1CC(C(N2CCC23CCN(C)C3)=O)C1 84138,C1(C(N(CCCC=C)CC)=O)CCC(C2CC2)N1C(=O)C=Cc1cc[nH]n1 84139,c1(C(=O)NC2C(CNC(=O)CN3CCCC3)CCC2)ccncc1F 84140,c1(C(=O)NC2(COC)CCN(C(=O)CC3CCOCC3)C2)cnc2n1CCCC2 84141,C(CO)(CCCCNC(=O)CC(C)c1cccnc1)NC(c1nc(CC)sc1)=O 84142,c1(C(=O)NCCCNC(CC2COCC(C)O2)=O)cccc(F)c1F 84143,C(CCCCNC(=O)CCCF)NC(C(C)c1cccs1)=O 84144,C1(C(=O)NCC2(CCC)CC2)CCCCN(C(=O)C(C)(CO)OC)C1 84145,C(=O)(C1=CCOCC1)NC(C1(O)CCN(C(=O)CC2SC(=N)NC2=O)C1)C 84146,n1(C2(CC(N3CC(N4CCOC4=O)C3)=O)CC2)cc(-c2ccco2)nn1 84147,c1(C(N(C2CN(C(c3c(C)nc(C(C)OCC)s3)=O)C2)C)=O)occ2c1CCC2 84148,Cc1ccc(C(N2CCCOC(CNC(=O)CNC=O)C2)=O)c2c1CCC2 84149,N1(C(=O)NC(c2ccc(Cl)cc2F)C(C)C)CCN(C)CC1CN 84150,c1(C(N2CCC2CNC(=O)C=CSC)=O)ccc(C=O)cc1C.CO 84151,C(=O)(C(C(C)(C)C)C1CCCCC1)N(C)CCNC(c1cn(C)[nH]c1=N)=O 84152,CC1CN(C(=O)Oc2ccc(Br)cc2)CCN1C(=O)COc1ccccc1 84153,CCCC(C)C(=O)NC1CCCN(C(C2(C#N)CCC2)=O)C1 84154,Cc1cc(F)c(CNCC2CCCCN2C(c2csc3c2CCCO3)=O)cc1Br 84155,CCC(CNC(=O)C(c1cncnc1)C)(CC)C(=O)NCC(O)C1CC1 84156,Cc1scc(C(=O)NCCC2(O)CCN(C(=O)CCC3CCCOC3)C2)c1C 84157,CC1(C)COC(CCC(=O)NCCN(C(=O)CCOCC(F)F)C2CC2)C1 84158,c1(OC)cc(F)cc2[nH]c(C(=O)NCCCNC(C3(C(F)F)CCCC3)=O)cc12 84159,Cc1cc2[nH]c(COC(c3ccc(CNC(=O)OC(C)(C)C)s3)=O)cc(=O)n2n1 84160,C(CC(C(=O)N(C)Cc1nnnn1C)NC(C1CC(OC)C1)=O)OC 84161,C12(NC(c3ccc(F)cc3Cl)=O)CCCC1N(C(=O)C(O)C1CCC1)CC2 84162,N#Cc1ccc(C(c2cc(C#N)c[nH]2)OC(C2CCN(C3CCC3)C2)=O)cc1 84163,CC(O)C(C)(C)CNC(=O)C(F)CC1CN(C(C2CCC(N(C)C)C2)=O)C1 84164,Cc1cc(C(=O)NCC2(F)CN(C(=O)CCCCC(C)(C)C)C2)cc2c1CCC2 84165,C1(CC(=O)NC(C)CC2CCCCO2)CCCCN1C(=O)C=CCO 84166,C1(NC(CC)=O)C2CC3CN(C(c4ccc(F)c(Br)c4)=O)C1C3C2 84167,c1(C(N(CCN(C(=O)CC2CCC(O)C2)C)C)=O)cn2ccc(F)cc2n1 84168,C(CSC)(CC1CCC1)NC(CC)C 84169,C1(C)(C(N(CC(c2ccccc2)CC)CC)=O)CN(CC(Cl)=CCl)CCO1 84170,c1(C(CC)C(=O)N(C)CCN(C)C(C2CNC(=O)C2)=O)cccc(Cl)c1 84171,c1(C(=O)NCC(CC)(C)NC(C2C3CC4C(C3)C24)=O)cc(C(C)C)nn1C 84172,CCC(CC1CCCC1)C(=O)N(C)CCN(C)C(C1CC(C)(F)C1)=O 84173,C(=O)(C1=CC(C)(C)C1)N(C(C)CN(C)C(c1ccc(C2CCC(=O)N2)cc1)=O)C 84174,c1(C(N2CC(CNC(C(C=C)OC)=O)C(OCC)C2)=O)cccc2ccoc12 84175,C1(C(=O)NCc2ncccc2C)(CC)CCCN(C(c2cnn(C3CC3)c2)=O)C1 84176,N1(C(c2csc(C)c2C)C(=O)NC2(OC)CC2)CCC(F)(F)C(C)C1 84177,c1(CCCNC2CC3CC(C)CC3C2)nc(O)c2c(C(C)(C)C)csc2n1 84178,c1(CC(=O)N(C)CCNC(c2ccc(F)s2)=O)cnccc1C(F)(F)F 84179,CN1CCC(F)(C(N2CC3C(CN(C)C)C3C2)=O)CC1 84180,C1(CNC(c2cc(OC)ncn2)=O)CC2(CC(NC(=O)C(F)(F)CC3CC3)C2)C1 84181,C1(NC(C(CC)NC)=O)CCC2(C1)CN(C(c1cc3cn[nH]c3cn1)=O)C2 84182,N1(C(CC=CCC)=O)CC2CCC2(CCNC(=O)CCc2csc(=N)[nH]2)C1 84183,N1(C(CCC)=O)CCC2(CCCN(C(c3ccc(Br)c(Cl)n3)=O)C2)C1 84184,CC1CCC(C)(CNC(c2c(CNC(=O)C(O)C3CC3)nnn2C)=O)CC1 84185,C1(C(NOCC#C)=O)C2CN(C(=O)C(CO)OC)CC12 84186,N1(C(Cc2ccc(OC(C)C)cc2)=O)CCN(C(C2CCSC2)=O)CC1COC 84187,c1(C(=O)Nc2scc(C(=O)NC(C(C)C)CO)n2)cccc(OC(F)(F)F)c1 84188,C1(=O)CCCCCN1.C(=O)(CC(F)(F)F)OCC1CCN(C(C)C)C1 84189,C1(C(N(CC(C)(C)CNC(=O)Cc2nc[nH]n2)CC)=O)CCc2cnc(C)n2C1 84190,C(=O)(CC(CC)C(F)F)N(C1CC(C(N2C(CSC)C=CC2)=O)C1)C 84191,C(=O)(CCCCC(C)(C)C)N1C2CC(C(=O)NC(c3ccn(C)n3)C)(OC2)C1 84192,C(=O)(CCCCCCBr)N1CCC(C(C(=O)OC)c2nn[nH]n2)CC1 84193,C(CC(C)CCNC(c1c(Br)n[nH]c1C)=O)NC(C(C)=C(C)C)=O 84194,C=CCC(C)(C(=O)NC1CN(C(=O)CC2CCNC2=O)CC1(C)C)N(C)C 84195,c1(C(N2C(C(N3C(C)CCCC3)=O)C3CCC2C3)=O)ccc(S(N)(=O)=O)cc1 84196,c1(C(N2CC(OCCNC(C(Br)=C(C)C)=O)C2)=O)nc(C)oc1C 84197,C1(C)(Nc2cc(C)on2)CCN(CC(=O)NCCN2C(C)CCCC2C)CC1 84198,c1(OC)cccc(C(O)C(N2CC(C(C)(C)O)(CNC(C3CC3F)=O)C2)=O)c1 84199,c1(C(N2C(CO)CC(NC(C(C=C)O)=O)C2)=O)ccc2c(c1C)CCC2 84200,c1(C(=O)NC2CCCC2C(=O)Nc2onc(C)c2C#N)cccc([N+](=O)[O-])c1I 84201,Cc1cc(C)nc(CCNC(=O)NCC2CN(C)NC2=O)n1 84202,c1(C(=O)NCC(Cn2cc(-c3n(CC)ncc3)nn2)OC)ccc(F)cn1 84203,C1(CNC(C(CC)(C)C#N)=O)CC12CCN(C(c1cnccc1C)=O)CC2 84204,Cc1cc(Cl)cc(C(N2CCCC(NC(c3c[nH]nc3C)=O)CC2)=O)c1C 84205,CC(C)C(CNC(c1nnnn1CC1CC1)c1cncs1)C(C)C 84206,C1(C(C)NC(C(N2CCC(OCC)CC2)=O)=O)CCc2ccccc2O1 84207,N1(C(=O)Cc2nc[nH]n2)CCC(C2(O)CCN(C(=O)C(O)C3CCC3)CC2)CC1 84208,N1(C(CC=CC)=O)CCCC1CN(C)C(c1cscc1C1CC1)=O 84209,Cc1ncc(C#N)cc1NC(=O)C(CCC1CCC1)NC(=O)CC1CCOC1 84210,CC1C(=O)CCC1OC(C1CCCO1)=O.C1C(=O)O1 84211,C12(C(=O)NC(CCC)c3ccco3)C(NC(C3(O)CCOC3)=O)C3CC1C2C3 84212,N1(CCC(=O)NC2CC(C)(NC(C(CSC)C)=O)C2)C(=O)CCC1=O 84213,N1(C(=O)Cn2cnnc2O)CCN(C(c2n[nH]cc2[N+](=O)[O-])=O)CC1CC(F)(F)F 84214,c1(C(=O)NCCC2(NC(COC(C)=O)=O)CC2)ccc2nnn(O)c2c1 84215,CS(=O)(=O)CC(=O)N1CCCC1CCCNC(c1cncn1C1CC1)=O 84216,CCC(O)C(F)(F)C(=O)NC1CCN(C(c2cscc2C(F)F)=O)C1 84217,c1(C(=O)NCC(CNC(c2ccc(C(C)C)o2)=O)F)cc(Cl)nnc1O 84218,c1(C(=O)NC2C(NC(=O)Cc3cn[nH]c3)CCCC2)cnc(O)c2ccccc12 84219,C(=O)(C1=CC2CCCCCC12)N(C1CC2N(C(C3(C#C)CC3)=O)C(CC2)C1)C 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84274,c1(OCC(=O)N(CC(C)N(C)C(c2cnc(N)cn2)=O)C)ccccc1C(N)=O 84275,C1(O)(C(=O)NC2CC(C)(CC)N(C(=O)Cn3nnnc3C)C2)CCC(C)(C)CC1 84276,C(=O)(CC(C(C)C)NC(c1cnc(Cl)n1C)=O)NCC(C(=O)OC)(F)F 84277,CC1(C)OCCC1C(=O)NCC1CCN(C(c2cnc(S)[nH]2)=O)C1 84278,N1(C(CC(=C)Br)=O)CCN(C(=O)Cc2ccc(F)cc2)C2CCCCC12 84279,c1(CC)cccc(C(N2CC(NC(=O)C(=O)NC3(Cc4ncc[nH]4)CC3)C2)=O)c1 84280,C1(C(=O)NCCC2OCC(C)(C)C2)CC12CCN(C(=O)Cn1ccnc1O)CC2 84281,C(c1c(F)cccc1F)=CC(=O)NCC1(O)CCN(C(COCC)=O)C1 84282,C(=O)(C(C)(C(F)F)NC(=O)OC(C)(C)C)NCCCCN(C(C(CC=C)C)=O)C 84283,N1(C(C(CSC)C)=O)C2CC1CN(C(C1(F)CCN(C)CC1)=O)C2 84284,C(=O)(C#CC1CCOC1)N(C(C)CNC(C1(c2ccc(F)cc2)CCC1)=O)C 84285,c1(CNC(=O)CC2C3CN(C(=O)CCc4cccnc4)CC23)cnc2n1CCC2 84286,CCC(C)(CO)C(=O)NCC(C1CCCC1)NC(c1ccccc1SC(C)C)=O 84287,Cc1cc(N2CCCC2)ccc1NC1CCCC(OC(C)C)C1 84288,c1(C(N(CCCNC(c2c(C)cns2)=O)C)=O)cc(CO)oc1C 84289,C12(CNC(C(C=C)(C)C)=O)CCCC1CCN2C(=O)CC1(O)CCC1 84290,c1(C(=O)OCC2C(C)(C)CCCO2)cc(C#N)ccn1 84291,C1(NC(CC=C)=O)CCN(C(c2ccc(-c3cc[nH]n3)cc2)=O)CCC1(F)F 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84380,c1(C(=O)NC2CC3N(C(C4C(=C)CC4)=O)C(CC3)C2)cc(S(N)(=O)=O)ccc1C 84381,C1(NC(c2ccc(C#N)[nH]2)=O)CN(C(=O)CCc2cccc(O)n2)CC1C1CC1 84382,CCC(C)(C#N)C(=O)NCCN(CC(C)O)C(=O)Cn1nc(C)cc1C(F)F 84383,c1(C(=O)NC(C(CO)NC(CCCC(CC)C)=O)C)cc2ccoc2cc1F 84384,N1(C(c2ccc(NC=O)cc2)=O)CCCC(NC(C2CCC2C(F)F)=O)CC1 84385,C1(NC(C2(CNC(C3CCN(C)C3=O)=O)CC(C)(C)C2)=O)CCn2cnnc2C1 84386,C(=O)(N=c1ccn(C(F)F)[nH]1)C1CCCC(NC(C(CC)Cl)=O)CC1 84387,c1(C(=O)NC(C2CCN(C(CCN(CCC)C)=O)C2)C)c(C(C)C)n[nH]c1C 84388,c1(C(=O)NCC(CNC(Cc2c(C)cco2)=O)F)cccn(C)c1=O 84389,c1(C(=O)NCCCC(=O)NCC(C(C)C)C)ccnc(CO)c1 84390,c1(C(N(C(CCCN(CC)CC)C)C)=O)nc2c(s1)CCC2 84391,c1(C(=O)NC(C(=O)NC(CCCC)CC)C)ccn2ccccc12 84392,C(=O)(CC(C)CNC(C1CCC(=O)CC1)=O)NCc1n(CC)ncn1 84393,C1(CC(=O)NC2C(CNC(c3ccc(C(C)(C)C)[nH]3)=O)CC2)CCCOCC1 84394,c1(N(C(C(CCC)N(C)C)=O)C)cccc(Cl)c1C(F)(F)F 84395,CC1CCN(C(C2CC2F)=O)CC1CNC(c1cnn(CC2CC2)c1)=O 84396,C1(C(=O)NCC(C)(O)C2(C)CC2)(CC)CCN(C(=O)CC2COCC(C)O2)CC1 84397,Cn1ncc(C(=O)NC2(CCC(=O)NOCC3CCCOC3)CCC2)cc1=O 84398,N1(Cc2nc(NC(c3c(F)ncc(C)c3)=O)sc2)CCCC2(C1)NC(=O)NC2=O 84399,CC(C)CC(=O)NCC(F)(F)CNC(=O)COCC(=O)OC(C)(C)C 84400,c1(CNC(=O)Nc2ncc(OCC)c(Cl)c2)ccc(S(C)(=O)=O)s1 84401,c1(CC)ccc2oc(C(=O)NCCC(CSC)OC)c(C)c2c1 84402,N1(C(CC2(OC)CC2)=O)CCN(C(c2snc(C)c2Br)=O)C(C)C1 84403,N1(CC(=O)NCC(CC)NC(c2nc(C)sc2C)=O)CCC(C)CC1 84404,c1(CC)c(C(N2CCC(CF)(NC(=O)CCC3(C)CC3)C2)=O)cnc2ncnn12 84405,C(C(CC(F)(F)F)NC(c1nnc(O)cc1O)=O)NC(CC1CCCC(C)O1)=O 84406,S1(=O)(=O)c2csc(n2)N1.c1(OC)ccc(-c2nc(CC3CC3)sc2C(=O)OC)cc1 84407,N1(C(c2cc(CC)on2)=O)CCOCC(C(N2CCC(CC(=O)OC)C2)=O)C1 84408,c1(C(=O)NCC(CNC(COC2(C)CCC2)=O)CO)ccc([N+](=O)[O-])s1 84409,N1(C(CCC#C)=O)CCCC(O)(CNC(C23CC(CN2C2CC2)C3)=O)C1 84410,c1(C(N2CCC(NC(c3ccc(C(C)=O)o3)=O)C2C)=O)ccc2nccnc2c1 84411,C12(C(=O)NCCC)CCCC1CCN2C(=O)Cc1cccnc1 84412,c1(C(N2CCN(C(C3C(CC)C3)=O)C(C)C2C)=O)cc(OC)cc2c1CCCC2 84413,c1(C(=O)NCCCc2nc[nH]n2)ccc(CCNC(=O)C2CC2)cc1 84414,c1(C(=O)NCC(C)(O)C(F)F)[nH]nc2ncccc12 84415,Cc1noc2cc(C(=O)NCC(c3ccc(Cl)cc3)c3ccccc3)nc(C)c12 84416,C(=O)(C1=CNC2=NCCC2=C1)NC1(C)CCN(C(C(COCC)(C)C)=O)C1 84417,S(=O)(=O)(CCCCCl)N1CC(O)(CNC(c2ccc(NC(C)=O)nc2)=O)C1 84418,C1(C(N(CCCNC(C2C(C)C2C)=O)C)=O)CC12CC(F)(F)C2 84419,C(CC(=O)NOCCC(C)O)OC(CNC(C(COCC)C)=O)(C)C 84420,CCC(C)CCCC(=O)NCC(C)(C)CC(=O)NC(C)(CO)C1CCCC1 84421,C1(C(=O)NC23CCCCC(C(=O)OC)(C2)C3)COc2c(OC)cccc2C1 84422,C1(NC(COC2CCN(C(c3ccn(C4CC4)n3)=O)C2)=O)CCC(F)(F)CC1 84423,N1(C(c2ccc(CC)cc2N)=O)CCN(C(c2cc(C(N)=O)on2)=O)CC(C)(F)C1 84424,C1(NC(C2C(NC(C(C)OCOC)=O)C=CCC2)=O)CCCC2(CC1)CC2 84425,c1(C(N2CC(C)CC(NC(COCCC=C)=O)C2)=O)cc(S(C)(=O)=O)cnc1O 84426,CCCC(C)CC(=O)NC(CNC(=O)CCc1ccsc1Cl)(CC)CC 84427,c1(C(C)=O)ccc(S(=O)(=O)OCC(O)COc2cccc(F)c2Br)cc1 84428,C1(NC(C(C)OCCC=C)=O)CCCC1NC(c1cc(CC(C)C)on1)=O 84429,C1(NC(C(C)(C)OC)=O)C(C)OCC12CCN(C(=O)Cn1ccc(C)n1)CC2 84430,C(=O)(C(C(C)CC1CCCC1)N(c1ccc(Cl)c(C(=O)O)c1)C)NCCSC 84431,N1(C(C2C(=C)C2)=O)CC(C(N2CCC(CC(=O)OC)C2)=O)CC(C)(C)C1 84432,N1(C(C(C)OCC)=O)CCN(C(=O)Cc2cccc(OCC(F)(F)F)n2)CC1C 84433,C(=O)(C1SCCc2sccc21)N1CCC(N(C(=O)C(O)CC(F)F)CCC)CC1 84434,C(=O)(CC(CC)C(C)(C)C)NCC(CCCC)NC(=O)C1=CCCC1 84435,CN1CCC(N2CC(NC(=O)OC(C)(C)C)C2)CC1.C12(CC1)CC(=O)NC2 84436,C(=O)(C(C)(C)C(C)C)NCC1CC(NC(c2c(C(=O)OC)c(C)[nH]n2)=O)C1 84437,CC1CCN(C(=O)NCC2(OC(C)(C)C)CC(F)C2)C1.c12cc(cs1)CNC2=O 84438,CCC(CNC(C1CCCN1CC)=O)N=c1[nH]c(Cl)nc2c1S(=O)(=O)CC2 84439,c1(C(=O)NC(CC=C)CNC(=O)CN2CC=CCC2)cnn(C2CC2)c1C 84440,C1(CCCNC(=O)COCC2CCOC2)CN(C(C23CC(F)(C2)C3)=O)CCO1 84441,C(=O)(C1=C(Cl)CCOC1)N1CCC(O)(C(C)NC(CCC=CCC=C)=O)C1 84442,c1(C(=O)OC)ccc(S(=O)(=O)N)c(Br)c1.C(C(O)C(N)=O)CCOC 84443,N1(C(CNC(CCC)=O)=O)CC(N(C(=O)C(C)Cc2ccccn2)C)C2(CC2)C1 84444,C1(NC(c2cc(C)no2)=O)COCCC1NC(=O)CCc1cc(Br)cs1 84445,Cc1onc(C(=O)NCC(C)N(C)C(C2CC(C)(F)C2)=O)c1Br 84446,N1(C(c2ccc([N+](=O)[O-])[nH]2)=O)CC2(CCC(C(N3CCC(CO)C(O)C3)=O)O2)C1 84447,C(c1cccc(O)c1)=CC(=O)NC1CN(C(=O)C(F)(F)CO)CC12CC2 84448,N1(C(CCSCCCC)=O)CCC2CN(C(=O)C(C3CCC3)OC)CC12 84449,N1(C(c2c(CC)ocn2)=O)CCCC2(CCN(C(C3CCC(=O)C3)=O)C2)C1 84450,C1(CNC(=O)C=CCF)CCCN(C(=O)CNS(=O)(=O)C2CC2)CC1 84451,c1(N2CCN(C(C=C(C)C(=O)O)=O)C(C(F)(F)F)C2)ncnc2[nH]c(C)nc12 84452,N1(C(C2(OC)CC2)=O)Cc2ccc(C(N3COC(C)C3)=O)cc2C1 84453,c1(NC(CC2C(NC(C(C=C)O)=O)CCCC2)=O)ccc(C)c(CC)c1 84454,c1(OCCC)ccc(NC(c2cscc2-c2c(SC)cccc2F)=O)cc1OC 84455,c1(NCC(C2CCCC2)NC(c2ccc(OC)nc2)=O)c([N+](=O)[O-])cnn1C 84456,Cc1ccc(C(=O)NCC(O)CNC(c2c(C)noc2N)=O)cc1[N+](=O)[O-] 84457,Cc1cc(Br)cc(S(=O)(=O)N2CC3(CCC(NC(c4nccs4)=O)C3)C2)c1 84458,N1(C(c2c(C)ncnc2C)=O)CCN(C(c2cc3ccccc3s2)=O)CC(O)C1 84459,C1(C)(CNC(CN2CCC(OC)C2)=O)CCCN(C(c2cncc(F)c2)=O)C1 84460,C(=O)(C1=CC2(CN(C(=O)C(C)(C)CC(F)F)C2)OC1)N(C(CC)COC)C 84461,C1(NC(C=C(COC)C)=O)CC12CCN(C(=O)C(C)C(=O)OC(C)(C)C)CC2 84462,Cc1ccc(C23CC2CN(C(=O)NCCc2noc(C)n2)C3)cc1 84463,Cc1cncnc1C(=O)NC1(C(=O)NCCOc2ccccn2)CC(F)(F)C1 84464,C1(NC(N(CC(C(C)C)OC)C)=O)CCC2(CC1)CC2C#N 84465,Cc1c(O)c(=O)ccn1CC(N1CC(N(C)C(C2CC=CCC2)=O)C(C)(C)C1)=O 84466,c1(C(N2CC(N(C(=O)Cc3ccns3)C)C2)=O)cc(Cl)cn1C 84467,N1(CC)CC(NC(=O)C(CN(C)C)NC(c2cccs2)=O)CC1=O 84468,c1(C(N2C(C)CC(NC(C=CCN(C)CC)=O)C2)=O)ncc([N+](=O)[O-])cc1C 84469,CC1(C)CC(NC(C2CC2C2CCC2)=O)CC(N)C1 84470,NS(=O)(=O)c1cccc(C(=O)NCCNC(=O)CCSCc2ccccc2)c1 84471,Cc1cc(F)sc1C(=O)NC1(CNC(c2cc(C(F)(F)F)[nH]c2C)=O)CCCC1 84472,C(=O)(CC1C(=O)Nc2cc(Cl)ccc21)NCC1(OC(C)=O)CCOC1.C1C(=O)N1 84473,C(CC(O)CNC(=O)Cc1csc(-c2cnccn2)n1)NC(CN(C(C)=O)C)=O 84474,CC(C)C1=NOC(C(=O)N(CC(=O)NCC2CCC(=O)O2)C)C1 84475,CN=c1[nH]cc(C(=O)NCC2CCC(C(=O)NC(C(C)C)C3CC3)C2)o1 84476,c1(CN2CC(C(=O)NC(C3C(=O)OCC3)CO)(CC3CC3)C2)ccccc1F 84477,c1(C(C(=O)NCCCCCC)N(C2CCOC(C)C2)C2CC2)ccc(C#N)s1 84478,c1(C(=O)OC)ccc(N2CCCC2CCNC(=O)C(C)N(C)C)nc1 84479,c1(CSCC(=O)NCC2(NC(=O)C(C3CCCCC3)F)CC2)ccncc1 84480,c1(COC)cc(C(=O)NCC2C(C)CCN2C(c2ccc[nH]2)=O)c(C)o1 84481,C1(CC)CCN(C(=O)C(CC)N(C)C)C1CNC(c1ncncc1Cl)=O 84482,C1(NC(C2(C(C)C)CCN(C(c3c(C)cc(C)s3)=O)C2)=O)C=CC(C)(C)CC1 84483,C12(C(=O)NCCCCCNC(C3CC34CCOC4)=O)CCN(CC1)CC2 84484,N1(C(COC(C)C)=O)Cc2nccnc2CC1C(N1CCC(O)C(F)(F)C1)=O 84485,CC1(C(=O)NC2(C(=O)NCCC(=O)NCCO)CCOC2)CCOCC1 84486,C1(C(C)NC(c2c(CC)cns2)=O)CCCN(C(c2n[nH]cc2Cl)=O)C1 84487,Cn1ncc2c1CCN(S(=O)(=O)c1c[nH]c(C(=O)O)c1)C2C(=O)OC(C)(C)C 84488,C=CC(C)CC(=O)NC1COCC1NC(c1cc(C)sn1)=O 84489,N1(C(CSSC)=O)CC2(CCC(CNC(=O)CNC(=O)CCC(C)C)O2)C1 84490,N1(C(C(CO)NC(C(C)C)=O)=O)CC(O)CC1(C)C(=O)N(CCO)CCO 84491,C#CCC(C)(C)C(=O)NCC1CCN(C(=O)CSCc2cscn2)C1 84492,C1(CNC(=O)NC(c2c(OC)cccc2)CO)CCC2C(C1)C2(F)F 84493,CCC(C)CCCCC(=O)N1CC(NC(=O)C=Cc2cn(C)nn2)C2(CCC2)C1 84494,C(=O)(C1c2c[nH]nc2CN1C(c1cnc(C)c(C#N)c1)=O)NC1CCC(CC)C1 84495,c1(C(=O)Nc2cccc(CNC(C=CCN(C)CC)=O)c2)nnc2ccccn12 84496,C(=O)(CCCCC(F)(F)F)N1CCC(CNC(CS(=O)(=O)N(C)C)=O)C1(C)C 84497,C1(C(=O)NCC(O)CNC(c2cccnc2O)=O)(OC)CCCC(C)(C)CC1 84498,C(C1c2ccccc2CN1C(C1C2COCC12)=O)NC(C(NOC)=O)=O 84499,N1(C(Cc2c(C)ccs2)=O)CC2CC(NC(C3CCC(C)(C)O3)=O)CC1C2 84500,N1(C(C(CC=CCC)C)=O)CCC(N=[N+]=[N-])(C(=O)NC2(CCC)CC2)C1 84501,Cc1cc(C(=O)N(C(C)(C)CC(=O)NC2CCCC2(F)F)C)nc(O)c1 84502,C1(C(=O)NCC2(C(C)NC(Cc3c(C)ocn3)=O)CC2)CC2C=CC1CC2 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84662,n1(CC)nc(C)c(C(=O)NC23CCOC(CNC(=O)C(F)C(F)(F)F)(C2)C3)c1Cl 84663,N1(CC2(C)CCN(C(Cn3c(C)cc(C(F)F)n3)=O)C2)CCC(O)C(C)C1 84664,Cc1cc(C(=O)NC2(C)CC(NC(C3CC(=O)NC(C)C3)=O)C2)cc(C)n1 84665,COn1cnc(C)c1C(N1CC(NC(c2c[nH]nc2C(C)(C)C)=O)C(F)C1)=O 84666,N1(C(C2CC(OC)C2)=O)CCC2(CC2)CC1C(=O)NC(CCO)C1CCC1 84667,CC1OCCC1(F)C(=O)NCCC1CCCN(Cc2nccn2C)C1 84668,C1(CNC(c2ccc(C(C)(C)C)[nH]2)=O)CN(C(=O)CSC2CC2)CCC12CCC2 84669,c1(N2CC3C(CNC(c4ccsc4Cl)=O)(C3)C2)ncnc2[nH]c(Br)cc12 84670,N1(C(c2c(CC)occ2)=O)CC(NC(C2CC(C#N)C2)=O)CCC1C 84671,CC1CCOC1CCNC(=O)C(C1(C)CC1)NC(=O)Cc1ccon1 84672,C1(CNC(CCC#C)=O)(OC)CCN(C(c2ccc(-c3ccccc3)nc2)=O)C1 84673,c1(C(N2CC(C)(NC(C)=O)C2)=O)ccc(NCc2ccc(Cl)s2)cc1 84674,C1(C(=O)NCCC2(C)CCCO2)CCN(C(=O)CC2CCCC3CC23)CCO1 84675,C1(C(=O)NCC2N(C(CC(C)C)=O)CCC2)CC2CCCC2C1 84676,S(=O)(=O)(c1cccc(=NCC(C)C(C)C)[nH]1)N1CCC(C(C)C)CC1.C(CCO)N 84677,N1(C(C)(C)C)CCC(NC(c2ccc(C(F)F)o2)=O)C1.C1(=O)CCC2CC(C2)N1 84678,c1(C(=O)NCC(C)(O)CNC(C2(Oc3ccccc3)CC2)=O)cccnc1Cl 84679,C1(CNC(=O)C(N2CCCC2c2ccc(Cl)cc2)=O)CCCS(=O)(=O)C1 84680,C1(=CCNC(C=CCCC(C)C)=O)CCN(C(c2c(C(C)C)cnn2C)=O)CC1 84681,C(=O)(C(F)CC(CC)CC)NC1(CNC(CNC(CC)=O)=O)CCOCC1 84682,CC1(C(N2CCCC(F)CC2)=O)CCCN(C(=O)COc2ccsc2)C1 84683,N1(C(c2cnn(C(C)(C)C)c2)C(=O)NC(C)C)Cc2ccccc2C(C)(C)C1 84684,CC1C(NC(=O)CNC(C2CCCCC2)=O)CC2CCC1N2C(=O)CCC1CC1 84685,c1(C(C(=O)NCC#CCNC(C2OCCN(C)C2)=O)=O)ccc(F)cc1F 84686,C1(C(=O)NCC2(O)CCN(CC3CCCCCCC3)C2)CCOCC12CCC2 84687,Cc1cc(C)c(NC(=O)C(c2cccnn2)N(C)CC2CCCOC2)c(C)c1 84688,C(=O)(NNc1ccc(Br)c(F)c1F)NCCC1(C(=O)OCC)CCOCC1 84689,C1(C(N(CCC(F)(F)F)CC)=O)CCOCC1NC(=O)C(C)OCCSC 84690,CC1CN2CCN1C(C(=O)NC1CC(C)(CNC(c3cn(C)ccc3=O)=O)C1)C2 84691,C1(CNC(c2cc(OC)n(C)n2)=O)CN(C(=O)C(C)n2ccnn2)CC1(C)C 84692,C(C(C)(O)CC(=O)N1CCC1CNC(=O)C(C)(C)Nc1ccc(Cl)cc1)OC 84693,N1(CC(=O)NC(C(CC)C)CO)CC(C(=O)O)C2(CN(C(=O)CC3CCC3)C2)C1 84694,N1(C(C2OCCN(C(CC3CC(CC)C3)=O)CC2)=O)CCC2CN(C)CC2C1 84695,C1(NC(CCC)=O)CC(C)(C(=O)NCC(CO)C2CCC2)C1 84696,c1(N2CC(CN(C(C(COC)(C)O)=O)C)OCC2)cc(=O)n(C)c(O)n1 84697,C1(N(C(C)(C)C)C(N2C(CC)C(C(=O)O)CC2)=O)CC(C)(C)C(C)(C)C1 84698,C1(CCC(=O)O)CCCC1C(=O)NC(c1cccnc1)C1CCCCC1 84699,FC1CC2CC1CC2NC(Cc1ccc(Br)cc1)CCC1CC1 84700,N1(C(=O)CC2CCCC2(F)F)CC2CCCC(C1)N2C(c1cncc(Cl)c1)=O 84701,c1(C(=O)NC(C)CCNC(c2cc(Br)co2)=O)n[nH]cc1[N+](=O)[O-] 84702,c1(C(=O)NCCCNC(C2(COCC)CC2)=O)sc(C#N)cc1Cl 84703,Cn1cc(C(=O)NC2C3CC2N(C(=O)Cc2ccc(C#N)nc2)C3)ccc1=O 84704,C#CCCCCCC(=O)N1CC2CC2(NC(=O)CCCCC2CC2)C1 84705,N1(CC)CC(C(=O)NCCOCCNC(C2CC(=O)N(O)C2)=O)c2ccccc21 84706,c1(C2OCCN(CC(=O)Nc3nnc(NC(=O)C4CC4)s3)C2)ccc(F)c(F)c1 84707,N1(C(c2n(CC)cc(Cl)c2)=O)CCCC(N(C(=O)CCN2CCCC2)C)CC1 84708,c1(C(N2CC(C)N(C(C3(C)CCNC3=O)=O)CC2)=O)cccc2c1NC(=O)CC2 84709,c1(C(=O)NC(C2CCN(C(=O)CCF)CC2)C)ccnc2nccnc12 84710,N1(C(c2c(C)cno2)=O)CCC2(CCCN2C(c2ccc(C(C)C)c(Cl)c2)=O)C1 84711,C1(F)(CNC(c2ccoc2)=O)COCCN(C(=O)Cc2ccc(Br)cn2)C1 84712,C1(SCC)CC(C(=O)NCC(C)(C)CCNC(c2nc(O)c(C)s2)=O)CCO1 84713,c1(C(N2CCN(C(C(C)=C3CC3)=O)CC2C2CC2)=O)cc2cc(Br)ccc2[nH]1 84714,N1(C2CCN(C(CSCC(N)=O)=O)CC2)CCN(C(=O)CO)CC1=O 84715,CC(=O)CCCC(=O)N1CCC(C)C1CNC(=O)C(O)C1CCC1 84716,C1(NC(Cc2cc(OC)no2)=O)CS(=O)(=O)CC1NC(=O)Cc1c(Cl)cnn1C 84717,c1(CN(c2ncc(OC)cn2)CC2(O)CCCNC2)cc(F)ccc1Br 84718,N1(CC(C)(C)O)CCN(C(CC2CCCC2)C(=O)NCCc2ccccn2)CC1 84719,CS(=O)(=O)C1CC(C(=O)NCC2CCN(C(=O)CC3C=CCC3)C2)C1 84720,C1(CNC(c2c(CC)non2)=O)CCN(C(c2cc(OC)cc(C)c2)=O)CC1C 84721,C(=O)(C1CC(=O)c2c(F)cccc21)NCC(CNC(c1c(C)cccc1Cl)=O)C 84722,c1(C(c2n(CCCSCC)nnn2)NCCC(=O)NC)c(N)cccc1Br.C1(SC)CC1 84723,C1(OC(C)(C)C)CC(N=c2ccn3nccc3[nH]2)C1(C)C 84724,N1(C(C2N(C)CCOC2)=O)CC2(C)CN(C(C3CC(F)(CO)C3)=O)CC2(C)C1 84725,N1(Cc2c(OC)cccc2OC)CC2CN(C(c3c(F)ccc(F)c3C)=O)CC2C1 84726,c1(C(N2CC(OC)C(NC(C3(C)CC=CCO3)=O)C2)=O)cc(Cl)cc2c1CCC2 84727,C(=O)(C=CS(C)=O)N1CC(CNC(N(CC(=O)NCCc2ccccc2)C)=O)C1 84728,c1(C(=O)NC2C(C)CN(C(=O)C(Cl)=CCl)C2)ccc(O)c(CO)c1 84729,C1(OC)CC(CCNC(C23CC(c4ccccc4)(C2)C3)=O)N(C(C23CCC2C3)=O)C1 84730,C(=O)(C(CNC(=O)C1=CCCC1C)C(C)C)NC(COC)(C)C(N)=O 84731,CN1CCn2ncc(C(=O)NC3(C)CCCN(C(=O)COCC(C)(C)C)C3)c21 84732,N1(C(c2ccc(N)cc2F)=O)CCC2(NC(=O)C=C3CC3)CCCCCC12 84733,C1(C(N(CCNC(CCC)=O)Cc2ccccc2F)=O)CCc2cnnn2C1 84734,Cc1ccc(C(N2CCC(NC(=O)CC3CCC(C)(C)C3)CC2)=O)c(O)c1 84735,CC1CC=C(C(=O)NC2(CO)CCCN(C(c3ccoc3C3CC3)=O)C2)CC1 84736,c1(C(C2(C(=O)NCCCNC(=O)CC3CSC3)CC2)=O)ccccc1 84737,CN1CCCC(CCC(=O)NCC(C2CC2)NC(=O)COC2CC=CC2)C1 84738,c1(C(=O)NC2CC(NC(c3cc(C)c(Br)s3)=O)C2)cccc(Br)c1O 84739,N1(C(C(Cc2c(C)nc[nH]2)O)=O)CCC(NC(=O)CCCCCN(C)C)C12CC2 84740,O=C(C1=CS(=O)CCC1)NCC1CC(F)(F)CN1C(=O)Cn1cc(Cl)cn1 84741,N1(C(c2c(C(C)C)cco2)=O)CC(NC(c2ccc(Cl)s2)=O)C2(CCOCC2)C1 84742,N1(C(CC=CCCCCC)=O)CCCC(N(C)C(C2CCCNC2=O)=O)C1 84743,c1(CC)ncccc1NC(=O)CC1CCCN1C(c1cncc(Br)c1)=O 84744,c1(C(=O)NC2CCN(C(CC(n3ccc(C)n3)C)=O)C2)cccnc1SC(F)F 84745,CC1=C(C(=O)NCc2ccnc(C(=O)NCC3COCC3(C)C)c2)SCCO1 84746,C1(CNC(C(C(C)C)N2CCCCCC2)=O)CN(C)CCN1C(C1CC(O)C1)=O 84747,c1(C(c2nnnn2C)NCc2c(OCC)cccc2)cc(Cl)ccc1[N+](=O)[O-] 84748,C(CC(=O)N(C1CC2(CC2)C1)C)(C(C)CC)NC(c1cn(CC)nn1)=O 84749,c1(OC)cccc(C2CCN(C(=O)NC3CCN(c4ccccc4)C3)CC2)c1 84750,c1(C(=O)NC2CCN(CCNC(CC(C=C)C)=O)CC2)c(F)ccc2n[nH]cc12 84751,C1(C(C)C)CN(C(C2CC(=O)C2C)=O)CCN1C(C1CS(=O)(=O)C1)=O 84752,C(=O)(C(C)(C)C(=O)N1CCC(C(C)NC(=O)C(C)C2CCCO2)CC1)OCC 84753,c1(C(N(CC=CC(N2C(C(C)O)COCC2)=O)C)=O)coc2ccccc12 84754,c1(C(=O)NCC(CC=C)NC(=O)C(C)(F)CCCC)cnc2c(ccn2C)c1 84755,N1(CC(N2C(C#C)CCC2)=O)Cc2ccccc2C1.C12(CCCCC1)C(=O)N2 84756,c12ccc3c(c1)CC(C3)NC(=O)CCCn1cc(nn1)CNC2.C1(CO)CC1 84757,N1(C(C2CC(=C)C2)=O)CCC2(CCC2NC(c2ccc(F)c(CO)c2)=O)CC1 84758,C=CC1(C(=O)NCCCCCN(C(=O)Cc2csc(Cl)c2)C(C)C)CCC1 84759,C1(NC(Cc2c(C)noc2)=O)CCCC(NC(=O)C(C)C=Cc2ccccc2)C1 84760,C1(C)(C(=O)NC2CCC(C(=O)NC(CCC)c3ccco3)C2)CCC(=O)N1 84761,C1(C(=O)NCC(c2ncc[nH]2)C)CC2CC2N1C(C1(C)CCCCC1)=O 84762,c1(CNC(C(C)N(C(C2C(CC)C2)=O)C)=O)ccnn1C 84763,c1(C(N2CC3C(CNC(c4ncnc5sccc45)=O)(C3)C2)=O)ccc2cc[nH]c2c1 84764,c1(C(N(CCCNC(c2cc(C)nnc2)=O)C)=O)ccc2[nH]c(=O)c(=O)[nH]c2c1 84765,c1(C(=O)NCCC(C)NC(C2CC(CCC)OCC2)=O)nc(O)nc(O)c1OC 84766,C1(C)(NC(C2C(C)OCC2)=O)CCCN(C(c2c[nH]cc2Br)=O)C1 84767,C(N=c1[nH]c2c(c(=NCc3ccc(C)c(F)c3F)[nH]1)CSC2)c1nnc(C)n1C 84768,Cc1ccc(C)c(C(=O)NC(C)CN2CCN(C(=O)CCNC(N)=O)CC2)c1C 84769,N1(C(C2CCC(=O)NC2)=O)CCN(C(=O)Cc2cc(Cl)ccc2Cl)C(CCO)C1 84770,Cc1cc(C(=O)NC2COCC2NC(=O)C#CC(C)C)c(C)c(O)c1 84771,C1(NC(CC=C)=O)CN(C(C2CCN(C(C)C)CC2)=O)CC12CCC2 84772,c1(C(=O)NCC(N(C(c2cc(C)ncn2)=O)C)C2CC2)ccc(Cl)cc1O 84773,c1(C(N2CC(O)(CN(C(CC(C)NC(N)=O)=O)C)C2)=O)cnccc1C(F)(F)F 84774,CC1CC(NC(c2cnc(Cl)n2C)=O)CCN1C(c1cc(F)cc(Cl)c1)=O 84775,C1(CNC(c2ccc(CSC)o2)=O)CCCCC1NC(=O)CCc1n[nH]c(=N)s1 84776,C1(NC(=O)C2=CCOC2)COC2(CCCN(C(=O)CCCC3CCCC3)C2)C1 84777,c1(C(N2C(C(C)NC(C(CCSC)N(C)C)=O)CCC2)=O)cnc2sccc2c1 84778,C1(c2n(CCSCC)nnn2)(NCC(c2nncn2C)(C)C)CCCC1CSC 84779,C1(C(N2CCC(N(C(C3C(=C)C3)=O)CC)C2)=O)CC2(C1)CS(=O)(=O)C2 84780,CCC(C)C(C(=O)NC(=O)C(C)C)NC1CCN(c2ccccc2)C1 84781,C1(NC(CCC=CC)=O)CN(C(C2(F)CCCC2)=O)CCC1CO 84782,N1(C(CCC2N(C(C(C)CN(C)C)=O)CCC2)=O)CC(S(C)(=O)=O)C1 84783,N1(C(C2CC(NC(c3ncc(C)[n+]([O-])c3)=O)C2)=O)CC2CC3CC2C1C3 84784,C1(CNC(CSCC)=O)CN(CC(CC)CC)CCC1(F)F 84785,Cc1cn2c(n1)CC(C(=O)NC1CCC(CNC(=O)Cc3cc[nH]c3)CC1)CC2 84786,c1(OCCOC)cc(NC(=O)C(CCF)NC(C2CCOC2)=O)ccc1CO 84787,C1(CCNC(C2CC(C#N)C2)=O)CCCN(C(=O)Cn2cnc(C(N)=O)n2)C1 84788,N(C1CCCc2ccc(C(C)(C)C)cc21)C(c1n(CC)nc(-c2cccs2)c1)=O 84789,c1(C(C)C)ccc(CNCC(=C2CCCC2)F)c(F)c1 84790,CCCC(C(=O)N(C)CC1CC(O)C1)NC(c1cn(C)cc1C)=O 84791,c1(NC2C(C)(C)C(Oc3nccs3)C2)cc(Cl)cc(Cl)c1 84792,n1(CCC)cccc1C(=O)N(CCO)Cc1ccn(CC)n1 84793,C=CCC(C)(CC)C(=O)N1CCC(N2CCN(C)CC2)C(C)C1 84794,C1(N(C(c2c(OC)cnnc2)=O)CCN2CCN(C)CC2)CC12CCNCC2 84795,C1(S(C)(=O)=O)(C(=O)NC(CNC(C(CC)(C)OC)=O)C)CCOCC1 84796,c1(C(=O)NCC2CCN(c3nc(C(=O)O)cs3)C2)cc(Br)cc2ccccc12 84797,N1(C(c2c(C)cn(C)c2)=O)CCN(C(C2(F)CC3(CCC3)C2)=O)CC1CC(F)F 84798,N1(C(C2CCC(CC)C2)=O)CCCN(C(c2cnn(C(C)C)c2F)=O)CC1 84799,C(=O)(C1=CCCC1C)NC(CSCC)C(=O)Nc1cnc(N(C)C)nc1 84800,C1(N(C(CN(C(C=C(CC)CC)=O)CC2CC2)=O)C)CCOCC1 84801,c1(C(=O)NCC2CCN(C(CSCC=C)=O)C2(C)C)ccc2c(C)noc2c1 84802,N1(OC(c2nc(C3(C(=O)OC)CC3)sc2C2CC2)=O)CC(C)(C)OC(Cl)C1 84803,C=CCCCCC(C(=O)NCCC)N(C1CCN(S(C)(=O)=O)CC1)C 84804,c1(CC(=O)NCC(C2CC2)NC(C(C)(O)C2CC2)=O)ccc2c(c1)OCCCO2 84805,C1(CC)(NC(=O)C(c2nc(C)cs2)C)CCN(C(C2CN(C(=O)N(C)C)C2)=O)C1 84806,C1(C(=O)OC)CCCCCN1C(=O)CN1CCCNS1(=O)=O 84807,NC(=O)C(O)CNC(C1CSCN1C(C1CCC2CC12)=O)=O 84808,C=CC(C)(CC)NC(C1CC(N(C(=O)C(C)N2CC(C)C2)C)C1)=O 84809,c1(N(C(C2CCOC2)C)C)nc(=NCCCCCO)[nH]c2c1SCC2 84810,C(C(CC(F)(F)F)NC(C1(c2cc[nH]n2)CCC1)=O)NC(=O)Cc1cn[nH]c1 84811,C(C)(CC(=O)NOCCCO)N(C(C1C(C(C)=O)C1)=O)C 84812,c1(C(=O)NCC(CNC(c2cc(OC)cc(F)c2)=O)O)cc2n(n1)C(C)CCC2 84813,C(=O)(C#CC1CCOCC1)N1C(C(N2CC(C=C)C2)=O)CN(C)CC1 84814,C1(OC)CN(C(c2ccc(O)nn2)=O)C(C)(CNC(c2ccnc(S)c2)=O)C1 84815,C(=O)(C1=CCN(C(C23CC2CCC3(F)F)=O)CC1)OCC 84816,c1(OC)cnc(F)c(C(=O)NCC2CCN(C(=O)CN3CSCC3=O)C2)c1 84817,N1(C(C(CCC)(C)C)=O)CCOC2(CCN(c3nc(O)c4ccccc4n3)C2)C1 84818,N1(C(C2C(C)=C2)=O)CCC(C2CCN(C(c3cccnc3N)=O)CC2)CC1 84819,c1(C(=O)NCC2N(C(C#CC3(C)CC3)=O)CC(O)C2)cc2c(F)ccc(Cl)c2[nH]1 84820,C1(NC(c2cnc(C)nc2)=O)C(C)(C)C(NC(=O)CC2CC2(Cl)Cl)C1(C)C 84821,c1(C(N(C)CCOCCNC(C2(C(F)F)CCCC2)=O)=O)c(Cl)cccc1[N+](=O)[O-] 84822,c1(NC(c2ccccc2Cl)CSC)ccc(S(=O)(=O)N(C)C)cc1[N+](=O)[O-] 84823,c1(C(=O)NC2CC(CCNC(c3c(Cl)nc(OC)s3)=O)C2)cnc(O)cc1C 84824,N1(C(C=CC(=O)NCC2CC2)=O)CCSC2CCC12.C12(CCCC1)C(=O)N2 84825,CCCCC(C(=O)NCc1cccc(OC)n1)NC(=O)CC(COC)COC 84826,C(CC(C)(C)C(=O)N1CCC(C)(CNC(c2c(OC(F)F)cccc2F)=O)C1)OC 84827,c1(C(C)(C)C)cnc(CNc2nccn2CC(F)(F)F)o1 84828,C1(C(=O)NC2CCC(NC(c3cccc(Cl)c3Cl)=O)C2)CCC2CC1CO2 84829,N1(C(CNC(c2[nH]cc(C(C)=O)c2)=O)C)CCC(C(=O)NC(C)(C)C)CC1 84830,CC1(C)C(C(=O)NCC(C)(C2CC2)NC(c2cc(F)cc(F)c2)=O)CCS1(=O)=O 84831,C1(C(N(CC(C2CC2)OC)C)=O)CNC(=O)CN1C(=O)Cc1cc(C)ccc1C 84832,Cc1cc(CN(C(N2CCCCC2c2ccc(C(F)(F)F)cn2)=O)CCl)cc(C)c1 84833,Cc1c(NC(C2(c3ccc(-c4ccc(I)cc4)c(F)c3)CC2)=O)cccc1Br 84834,C1(NC(Cc2c(C)non2)=O)CCCC2CN(C(c3cn(C)nn3)=O)CC12 84835,C1(C(N(C2CCN(C(=O)CCC(=O)C3CC3)C2)C)=O)CCc2cnn(C)c2C1 84836,Cc1cc([N+](=O)[O-])cc(C(=O)NCC2CCN(C(=O)C#CC3CC3)C2)c1Cl 84837,C#Cc1ccc(F)c(C(N2CC(C)C(NC(=O)CC3CCSC3)C(C)C2)=O)c1 84838,c1(OC)cccc(CN(C2CC(O)C2)C(=O)CC2CCNC2)c1Cl 84839,C1(C(=O)OCC)CCCC(NC(=O)C(C)OC(=O)CCc2scnc2C)C1 84840,n1(CC)cc(C(=O)C(=O)NCC(C)(C)OCCNC(C2(C)CCCS2)=O)cn1 84841,C1(OC(C(c2cn(CC)nc2)C)=O)CCN(c2ccc(Br)cc2)C1=O 84842,C1(C#N)(C(N2CC(C(C)NC(c3c(CC)con3)=O)OCC2)=O)CCCCC1 84843,c1(C(=O)OC)nn(C)nc1C(N1CC(CNC(C2(C)CCOC2C)=O)(OC)C1)=O 84844,CCC(CC(=O)NCC1(C(=O)Nc2cccc(O)c2)CC=CC1)SC 84845,N1(C(C=C(C)Cl)=O)CCOCC(F)(CNC(c2cn(C3CCC3)nn2)=O)C1 84846,C1(C(C)C)CC(N=c2[nH]c(=NC(CF)c3cccc(F)c3)c3sccc3[nH]2)C1 84847,C(CSC)(C(=O)N(C)CC1(O)CN(C(=O)C(C2CC(F)(F)C2)O)C1)OC 84848,N1(C(c2ccn(CCOC)n2)=O)CCSCC1CCNC(=O)C(C)CC1CCC1 84849,C(=O)(CC1=NNC(=O)C1)N1CCC(C(C)NC(c2ccc(OC(C)C)cn2)=O)C1 84850,N1(C(CCNC(C)=O)=O)C(C(=O)NCc2ccco2)C2CC(O)C1C2 84851,C(CCC)(CCCNC(c1nccn1C)=O)NC(C(CC=C)NC(C)=O)=O 84852,c1(C(=O)NC(CC)CN(C(=O)CCC(C)C)C)cccc(F)c1C#N 84853,N1(c2snc(C)c2C#N)CCC2(NC(=O)CCCN3CCCC3)CCCCCC12 84854,c1(-c2cn(C(C(N3C(OCCC)CSC3)=O)C)nn2)c(C)[nH]c2ccccc12 84855,N1(Cc2c(OC)cc(Br)cc2)CC2CCN(C(c3cncc(C)c3)=O)C2C1 84856,CCC(CC(=O)N1CCCC1C(C)(C)NC(C1CCC2CC12)=O)CC(C)C 84857,n1(CC)cnc(C(=O)N(CCCN(C(=O)CN(C)CCOC2CC2)C)C)n1 84858,c1(C(=O)NCCC(=C)CNC(c2oc(Br)nc2C)=O)cn2ccccc2n1 84859,N1(C(C(C)OCCCC)=O)CCC2(C1)CN(C(C1(C)CCN(C)CC1)=O)CCO2 84860,N1(C(C(CC)C#N)=O)CCC(c2cn(-c3cccc(C(F)(F)F)n3)nn2)C12CC2 84861,C1(C(C)C)COCCN(C(C2CCN(C(=O)C(C)(C)C3CC3)CC2O)=O)C1 84862,C1(NC(C(CC)C2CCOC2)=O)CCC(N(C(=O)C(=O)NC2CC2)C)CC1 84863,c1(CC)nc(C(=O)NCC2C(CNC(=O)C(F)C3CCCC3)C2(F)F)cs1 84864,C1(C(=O)NCCC2CCC(C)(C)C2)(CNC(C2CC(C)(CC)C2)=O)CC(C)(C)C1 84865,C1(CC(=O)N(C(C(N2CCC(CSC)C2)=O)C2(C)CC2)C(C)C)CCN(C)CC1 84866,N1(C(=O)CN(C)Cc2c(C)noc2)CCCC1(C)C(F)(F)F.C(C)(=O)O 84867,c1(C(N(CCNC(c2c[nH]nc2Br)=O)CC)=O)nccc(OC)c1N 84868,N1(C(c2ccc(C#C)o2)=O)CCC(C2CCN(C(=O)CCc3ccsc3)C2)C1 84869,c1(CNC(Cn2cc(-c3cnc(OC)c(C)c3)nn2)=O)c(C)nn2c1NCCC2 84870,C(=O)(C(C)C(O)CC(C)C)N(C1CC(C#N)C1)CC(=O)NC(C#C)CC1CC1 84871,C(=O)(CCC(=O)c1cc(Cl)sc1Cl)OCCCO.CC(C)NCCN(C)CCNCF 84872,C1(CNC(C(COCC)NC(=O)CC2CC2(C)C)=O)CCC(=O)NC1C 84873,N1(C(c2c(C)c(O)ccc2)=O)CC(CNC(C2(C)CCN(C)C2)=O)CC(C)(C)C1 84874,c1(-c2nc(CC(C)OCC(C)C)n(CCN(C)C)n2)ccc(Cl)c(Cl)c1 84875,C=CCC(CO)NC(=O)C(C)CN(C(=O)CCC1CC1C)C 84876,N1(C(c2c(CC)scc2)=O)CC(C)(C)OCC1CNC(=O)C(c1ccc(C)o1)C 84877,C=CC(CCC)CC(=O)NCCOC1CN(C(c2cn3ccnc3s2)=O)C1 84878,c1(N2CCC(NC(C)=O)CC2)nc(N2CCCOC(C)C2)c2c(n1)c(C)nn2C 84879,C1(C(=O)NC(CC)CNC(=O)CC2(C)CCCO2)CCC12CCC2 84880,N1(C(C2N(C)CSC2)=O)CC2(CNC(=O)C(C)(C)c3nccs3)CC1CO2 84881,N1(C(c2c(CC(=O)OCC)occ2)=O)CCCC(CNC(c2oncc2C)=O)C1 84882,C1(CC(=O)NCC2CC(O)(CNC(C3CCCN(C)C3)=O)C2)CCCS(=O)(=O)C1 84883,N1(C(c2csc(C)c2N)=O)CCC(NC(C2(C(N)=O)CC2)=O)CC(O)C1 84884,C1(C(=O)NC2CC(NC(c3c[nH]nc3C3CC3)=O)C2)COCCN1CC(F)(F)F 84885,c1(C(=O)NCC(C)CNC(c2cnc(-c3cccs3)o2)=O)csc2nnsc12 84886,CCC(C(=O)NC1(C)CC1)n1ccnc1.C12(CC1)C(=O)NCC(=O)N2 84887,Cc1sc(N)c(C(=O)NCC2CCCC2NC(c2cnn(C)c2C(C)C)=O)c1C 84888,N1(C(c2cccc(CC)c2F)=O)CC2(CCCN(C(c3cccc(C)c3)=O)C2)C1 84889,N1(C(C(C2CCOCC2)OCC)=O)CCN(C(c2ccoc2)=O)C2COCC12 84890,N1(C(CC)=O)CCCC(C2(NC(=O)CCCCCF)CC2)C1 84891,Cc1n[nH]cc1C1CC1C(=O)NCC1(NC(=O)CCc2cncs2)CCC1 84892,C12(CNC(CC=CCC)=O)CC1CN(C(C13CC(c4ccccc4)C1C3)=O)C2 84893,c1(OC)ccccc1C(=O)N(C)CCSC.c12csc(c1)CNC2=O 84894,N1(C(C(=O)NC(C2CCCC2)CN)=O)CCC(n2cccn2)CC1 84895,c1(C(N2C(CNC(c3n(C)ccc3)=O)CC3(CC3)C2)=O)cc2cc(N)ccc2[nH]1 84896,c1(C(N2CC(NC(Cc3c(C)cnn3C)=O)C(F)CC2)=O)ccc2occc2c1 84897,Nc1ccc(Cl)c(C(=O)NCC2CC(NC(=O)C3=CCCOC3)C23CCC3)c1 84898,N1(C(c2n(CCC)ncc2)C(=O)NC2CC2)CCCC(O)C1 84899,CC1(C)NC(=O)N(CCC(=O)NC2CCN(C(=O)C3CC3)C(C3CC3)C2)C1=O 84900,S(=O)(=O)(c1cc(NC(C2CN(C(=O)C(O)CF)CCO2)=O)ccc1OC)NC 84901,c1(CCC)cccc(C(N2CC3(NC(c4cc(C5CC5)ccn4)=O)CC2C3)=O)c1 84902,N1(C(C(c2cnn(C)c2)OC)=O)C2CC=C(C(=O)NC3CCC4CCC34)C1CC2 84903,C1(NC(C(Cn2ccc(C)n2)C)=O)CN(C(c2cc(O)ccc2C)=O)C(C)(C)C1 84904,C(N=c1cc(C)nc(N2CC(CO)C3(CC3)C2)[nH]1)C1CC(OCCOC)C1 84905,c1(CN(C(=O)C(F)(F)c2nccs2)CCNC(COC)=O)ccc(F)cc1F 84906,N1(C(C=CC(=O)NCC23CC4CC2C3C4)=O)CCN(C(c2cscn2)=O)C2CC12 84907,CCN=C(NCC1(CS(C)(=O)=O)CCC1)N(C)CCC(F)(F)CO 84908,C1(NC(CC(C)CF)=O)CCC2(CCN(C(c3cc[nH]c4nccc3-4)=O)CC2)C1 84909,C1(C(N(CC#C)CCF)=O)CN(C(=O)Cc2c[nH]nc2C)CC1F 84910,c1(C(NOCC(CC)O)=O)cc(Br)ccc1OC(F)(F)F 84911,C1(CC)C(=O)NCCN1C(C1CCCN1C(=O)CCCc1cnn[nH]1)=O 84912,CCCC(C)C(=O)NC1CCCC1CNC(c1sc(=N)[nH]c1C1CC1)=O 84913,c1(N2CCC(NC(C(C#N)=CC(C)C)=O)C(C)C2)ncnc2onc(C)c12 84914,C1(NC(c2c(Br)cn(C)n2)=O)CN(C(c2ocnc2C2CC2)=O)CCC1F 84915,C1(CNC(C(C)(C)c2cnsc2)=O)COCCN1C(=O)C=Cc1cccs1 84916,S(=O)(=O)(c1cccc2c1OCCO2)Nc1ccc2c(c1)N(C)CC2 84917,C=CC1OCCCC1C(=O)NCC1CN(C(=O)CSCC(C)C)CCC1(F)F 84918,C(C(C(=O)NCC1(O)CC(N(C)C)C1)NC(=O)C(O)C1CCCC1)OC(C)C 84919,C1C(C)C(=O)N1.C(CN(C)C)(C(=O)NCCCSCCC(C)C)OC 84920,Cn1ncc(C(N2CC=C(CNC(C3CC34CCOCC4)=O)CC2)=O)c1C#N 84921,C1(CCCN(C2CCCN(C(C)(C)C)C2C)CC)CCC(F)(F)CC1 84922,N1(C(C(C)SCC)=O)CC2CCC1(C(=O)OC(C)(C)C)CC2 84923,Cc1c(O)nnc(N2CCN(C)C3CC23)c1C 84924,N1(c2n(-c3oc4cccc(C(=O)O)c4n3)nc(C)c2)CCNCC12CCOCC2 84925,c1(CCC(N2CC=CC(NC(c3cc(C(C)C)sn3)=O)C2)=O)ccc(F)cc1F 84926,C1(C(N(CC#C)CC)=O)CC2CC1CN(C(C1CCC(=O)CC1)=O)C2 84927,c1(CC(N2CCC(CN(C(C(C)(C)OC(C)=O)=O)C)C2)=O)cc2ccccc2o1 84928,N1(C(CC(CC)(C)C)=O)CCCCC12CC(NC(=O)C1=CS(=O)(=O)CCC1)C2 84929,N1(C(COCCCC)=O)CC2CN(C(=O)C(c3ccccc3F)(C)F)CC2(C)C1 84930,c1(N2CCC(COC)(NC(=O)C(CO)N(C)C)CC2)ccc([N+](=O)[O-])cc1C#N 84931,N1(C(CC2(C=C)CCC2)=O)CCC2(NC(c3ccnc(C)c3)=O)CCCC12 84932,C1(NC(C(CSC)OC)=O)CC2(C1)CC2C(=O)NCC1COCCN1C 84933,C(=O)(C#CC1(C)CCCO1)NC1C(NC(Cc2n(C(C)C)cnn2)=O)CCCC1 84934,N1(C(C(CNC(c2c(C)nsc2C)=O)OC)=O)CCCC(C2(C)CC2)C1 84935,c1(OC(C)C)ccc(C(=O)NCCC2(NC(C34COCC3C4)=O)CC2)cc1 84936,c12ncc(Br)c(n1)C(=O)NC1(C)CN2C1.c1(CCNN(C)C)cccs1 84937,Cc1ccnn1CC(=O)NCC(O)C(=O)NC(c1cn[nH]c1)C 84938,N1(C(CC(C(C)C)O)=O)CCN(C(c2ccn(C(C)(C)C)n2)=O)C(C)C1C 84939,CCC(C#N)C(=O)NCC(C1CCNCC1)(C)O 84940,c1(C(N2CC(C(C)NC(c3nsnc3O)=O)C2)=O)ccc(C2CC2)nc1O 84941,C1(CC(N2CCCC(N(C)C(c3n[nH]cc3F)=O)C2)=O)NC(=O)CNC1=O 84942,C1(C(N(C)Cc2ccc(C)cc2)=O)CN(C)CCN1C(=O)C(F)=CC1CC1 84943,C1(CNC(CC=CC=C)=O)CCC2CN(C(c3ncc(C(C)=O)s3)=O)CCC2C1 84944,C1(NC(C2C(CC)CCC2)=O)CCC(NC(c2cc(OC)c(Cl)s2)=O)CC1 84945,S(=O)(=O)(c1cccc(F)c1)NCCNC(c1cn(CCOC)nc1)=O 84946,N1(C(=O)CCCCCn2cc(C3CCCOC3)nn2)CCCC2(CCNC2)C1 84947,N1(C(c2cccc(OC)c2OC)=O)CCCCC12CN(C(c1ccoc1C)=O)C2 84948,C1(C(N(CC(N)=O)C)=O)CN(C(=O)NC(c2ccc(F)c(F)c2)=O)CC(C)(C)C1 84949,Cn1ccc(CNC(=O)C(O)CCCNC(C2(CO)CC3CC3C2)=O)cc1=O 84950,N1(C(C)C(=O)NCC(F)(F)F)CCC2(CN(C(=O)C(C)(C)C3CCCO3)C2)C1 84951,C1(O)(CCNC(C(C)OCC#C)=O)CN(C(=O)Cn2nccn2)C1 84952,CCC(CC(=O)NC1(CC(=O)NCC2CC[Si](C)(C)C2)CC1)C(C)C 84953,Cc1cccc(Br)c1C(C(=O)NC1CC1(C)C)NC(C1CCC2(CC2)C1)=O 84954,Cc1ccc(C)n1CC(=O)NC1C=CC(C(=O)NCCC2CCC(C)C2)C1 84955,c1(OC)cc(O)c(CN2CCCC2CC(=O)NC(C)CCCC(C)C)cc1O 84956,C1(C(N2CC(N(C(C(CC)CC)=O)C)C(C)CC2)=O)CCCC2(CCC2)C1 84957,c1(C(=O)NC2CCC(NC(CC=C=C)=O)C2)csc(C)c1CC 84958,CC(C)(C#N)CCCC(=O)NC1CCCC1NC(C12CCC(CC1)C2)=O 84959,C(=O)(C1COc2ccccc21)NC1CCN(C(C2(C)CC2)=O)CC1CO 84960,C(=O)(CC1OC(=O)c2ccccc21)N(CCCCNC(CC(CCC)(C)C)=O)C 84961,C1(NC(C2(F)CCN(C(CC3N(C)CC=CC3)=O)CC2)=O)CC2CC1CC21CC1 84962,c1(C(=O)NC(CNC(C(CC)=CC)=O)CC)nccc(C)c1N 84963,N1(C(CCCNC(N)=O)=O)CC(NC(=O)C=Cc2ccccn2)CC(O)C1 84964,C(N=c1[nH]c(N2CCC(COC)CC2)nc2c1CCC2)c1nnc(CC)s1 84965,c1(C(N2C(C)CC(NC(=O)CS(N)(=O)=O)CC2)=O)ccc2n[nH]cc2n1 84966,O=C(CC(F)(F)F)N1CCC(N2CCN(C(c3c[nH]c(=O)cn3)=O)CC2)C1 84967,C(=O)(C1=NOC2(CCOC2)C1)NCCC1(OC)CN(C(C2(C#N)CCC2)=O)C1 84968,N1(C(C2C(C(=O)OC)C=C2)=O)CCC(O)C(NC(C2CCCN(C)C2)=O)C1 84969,C1(NC(CCOCCCOC)=O)CN(C(=O)C=CSC)C(C)(COC)C1 84970,N1(C(C2C(C)OCC2)=O)CCC(C(F)F)(CNC(=O)COC(F)(F)F)C1 84971,N1(C(c2ncccc2Cl)=O)CCC2(CCCC2Nc2nccc(CO)n2)CC1 84972,c1(C(N(C(C)CNC(C2(C(=O)OCC)CCCCC2)=O)CC)=O)ccc(N)cc1C 84973,C1(CNC(CCC(=C)Cl)=O)COCC2(CCN(C(=O)CC3=CCCCC3)C2)O1 84974,CC1CN(C(C2CCC(n3cc(-c4ccn(C)n4)nn3)C2)=O)CC1CO 84975,C1(C)(CC)C=C(C(=O)NC2CCCC(NC(c3nnn(C(C)(C)C)n3)=O)C2)C1 84976,N1(C(c2[nH]c(=NC)sc2)=O)CC(C)CN(C(c2coc3c2COC3)=O)CC1C 84977,N1(C(C=Cc2ccc(C)o2)=O)CC2(C1)SCCC2NC(=O)C1=CC2CCCC12 84978,N1(C(c2c(C)ncnc2O)=O)CC(O)(C2(CNC(=O)C3=CCCC3)CC2)C1 84979,C1(NC(CC(=O)OC)=O)CC2CCC(C1)N2Cc1ccnc(Cl)c1F 84980,C12(NC(COCCCCC)=O)CC(C(=O)NCC3(F)CC3)(C1)C2 84981,C1(O)(CN(C(c2ncn(CC)c2)=O)C)CCN(C(c2ccoc2Cl)=O)C1 84982,C=C(C)CC(C(=O)NC1CCN(C(=O)CN(C)C2CC2)C(C)C1)OC 84983,C12(CNC(CNc3[nH]c(=N)sc3)=O)CNCCN1CCOC2 84984,C(=O)(CS(=O)(=O)CCO)NCC(CCNC(c1cc(CC)ncc1)=O)O 84985,N12CCC3CCN(CC13)C2=O.c1(OCCOCC#C)cc(F)c(C)cc1C#N 84986,C1(C(=O)O)(C(=O)NCc2cncnc2)CC2CCC1CC2 84987,N1(C(C(CC=CC)C)=O)CC(C)N(C(=O)CN(C)S(N)(=O)=O)CC1C 84988,Cn1ccn2ncc(C(=O)NC3CCN(C(C4(CO)CCCO4)=O)CC3)c12 84989,N1(C(C2CCC(NC(c3nc(CC)oc3)=O)C2)=O)CCC(CO)C(F)(F)CC1 84990,C=C(C)CCCC(=O)NCC(CC(=O)N1CCCC1(CO)CO)OC 84991,N1(C(c2c(CC)scn2)=O)CCC2(CCCN(C(c3nncs3)=O)C2)C1 84992,c1(NC(=O)CC2(CO)CCN(C(=O)C=CC(F)(F)F)C2)cncc(C2CC2)c1 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85010,C(=O)(C(C)CC(F)(F)F)NC1CCCCN(C(C2CC(OC)C(OC)C2)=O)C1 85011,CCCC(CNCC(C)(CC)C(=O)N1CC2CC1C2C(=O)OC)C(=O)OC 85012,N1(C(C(=C(C)C2CC2)F)=O)CC(CCNC(C2(C)CCN(C)CC2)=O)OC(C)C1 85013,N1(C(CCNC(=O)OC)=O)CCC(C(=O)Nc2cc(Cl)ncn2)C(O)C1 85014,C12CC3CC(C1NC(O)C(=O)C3)CC(CC1(C)CCC1)(CF)CNC(=O)N2 85015,C1(C(=O)NC2C=CC(C(=O)NC)C2)(CNC(CCCSCC)=O)CC2(CC2)C1 85016,C(=O)(C(Cl)=CCl)NCC(C1CCOC1)NC(CC1CN(C)C1)=O 85017,C1(NC(c2nc(CC)oc2)=O)CC(CNC(c2ncc(F)cn2)=O)C1(C)C 85018,c1(N2CCC(C3CC3)(CNC(C=COCC)=O)C2)[nH]c(=O)n(C)c(=O)c1C#N 85019,Cc1ncc(C#N)c(NC2CN(C(c3ccc(O)c(O)c3Cl)=O)CC2C#N)n1 85020,C1(NC(c2nn(CC)c(O)c2)=O)CC(C(=O)NC2CCCC2CF)C12CCC2 85021,C1(NC(Cc2nc(C)sc2Cl)=O)CCN(C(=O)CC(C)(F)F)C(C)C1 85022,C1(CCC=C)(C(=O)NCCc2ncccn2)CN(C(=O)CCC2CC2)C1 85023,c1(NC(C2(F)CCN(C(CCSC)=O)CC2)=O)c(C=O)c(C)nn1C 85024,C(=O)(C1=Cc2ccccc2C1)NC(C(=O)NC(C1CSC1)C)c1ccoc1 85025,C(=O)(C1=CCN(C(C2CC(=O)C23CCC3)=O)CC1)N1CC(CCC)C(CO)C1 85026,CCC(C(=O)NC1(CO)CN(C(=O)CCCNC(=O)CNC(C)=O)C1)OC 85027,Oc1cc(N(C(Cc2ccoc2)C(=O)Nc2ccccc2)C2CC2)cc(F)c1F 85028,N1(C(c2scnc2Cl)=O)CCCN(C(=O)C(O)c2ccco2)CC1 85029,N1(C(C(C2CC2)OC)=O)CC2CCC1C(CNC(=O)CC1CCCC(C)C1)C2 85030,CC(C(=O)N(CCC(=O)NCCC1CC(=O)N(C)C1)CCCO)C(F)F 85031,N1(C(CC(C(C)OC)NC(C23CCC(CC2F)C3)=O)=O)CCC2(CC1)CSC2 85032,CC1CCn2cc(C(=O)N(C3CC4CCC(C3)N4c3nccnc3F)C)nc2C1 85033,CC1CN(C(=O)C(C(C)O)NC(=O)C(=O)NC2CC2)C(C)C1C 85034,C(C1CCN(C(=O)CC23CCCC2C3)CC1)=CC(=O)NC1CCCC(C(C)C)C1 85035,Cc1cc(C(N2CCCC(NC(=O)CCS(C)=O)C2)=O)ncc1Cl 85036,N1(C(C(C)Oc2ccccc2)=O)CCC2(CCC2NC(c2ccc[nH]2)=O)CC1 85037,Cc1cc(-n2cncn2)ccc1CNC1CNC(=O)C1 85038,CCC(F)(F)CC(=O)N1CCC(C)(C)C1CC(=O)NCCN1CCOCC1 85039,C1(NC(C=C(CCC)C)=O)CC2(CCN(C(c3cncc(N(C)C)n3)=O)C2)C1 85040,C#Cc1cccc(C(N2CC(COCC)CC(c3cnn(C)c3)C2)=O)c1 85041,c1(C(=O)OCC)cnc(Cl)cc1NC(=O)CCC1CCCCNC1 85042,c1(CC)noc(C(N2CCOC(CCNC(C3CCCC34CC4)=O)C2)=O)c1C 85043,c1(NC(N(C2CC(OC)C2)C)=O)ccc(Br)c(C(F)(F)F)c1 85044,N1(CCn2cc(COC)nn2)CCN(C(C2CN(C)C2)=O)CC1 85045,c1(C(=O)NCC2CCN(C(C3(CC(F)F)CCCC3)=O)C2)ccc(CO)cc1F 85046,C1(C(N2CC(c3nc(C)on3)C2)=O)CC(C)CN1C(=O)Cc1cnc(C)s1 85047,CC1OCCOC1C(N1CCC(CCNC(=O)CN2CCOCC2=O)CC1)=O 85048,CCCCC(F)C(=O)NCCn1cc(CNC(c2nn(C(C)C)cc2Cl)=O)nn1 85049,C(=O)(C(CO)N(C)C)NC(CC1CN(C(C(C)OC2CCOC2)=O)C1)C 85050,N1(C(C2(CCCC)CC2)=O)CC2C3CCC(C2C1)N(C(C12CC(F)C1C2)=O)C3 85051,C(=O)(C(C)(F)C(=O)NCC1(F)CC(CNC(c2ncc(Cl)cc2Cl)=O)C1)OCC 85052,N1(C(C(C2CCCC2)NC=O)=O)CC2CC(NC(C3(F)CCCCC3)=O)C1C2 85053,N1(C(CCCNC(=O)OC)=O)CC(NC(C2(C(N)=O)CC2)=O)CC12CCC2 85054,c1(NC(C(=O)NC2CC(N(C)C)C2)CC2CC(F)(F)C2)ccc(N(C)C)cc1 85055,C1(C(=O)OCCCc2n(C)ncc2)CCN(C2CC2)C1=O 85056,C1(C)(C(=O)NCC(COC)O)CCN(C(c2cccnc2O)=O)C1 85057,C1(C)(CNC(c2c(OC)c[nH]n2)=O)CN(C(=O)CN2CC(C)(OC)C2)C(C)(C)C1 85058,c1(CC)nccnc1C(=O)NC1(CCNC(=O)C(C)C2CCC2)CCCC1 85059,Cc1cncc(C(=O)NC(C)CNC(c2scc(C)c2Br)=O)c1 85060,CC1CCC(C)(C(=O)NCC2CCC2NC(C2(N(C)C)CCCC2)=O)CC1 85061,Cc1ccc2oc(C(N3CCN(C(C4CC=CCO4)=O)C4CCCC34)=O)cc2c1 85062,CC1CCN(C(=O)C(C)Sc2ccc(Br)cc2)C(CNC(N)=O)C1 85063,S(=O)(=O)(CCC(=O)NCCN(C)C(c1ccc(Cl)s1)=O)NCCNC(C)=O 85064,C(CCC(C)C(=O)N(CC(C)NC(=O)Cn1cnccc1=O)C)OC 85065,CC(CNC(=O)CN(C)C(c1ccoc1)=O)CN(C(=O)CCn1cccc1)C 85066,Nc1cc(F)c(C(=O)NC(CNC(c2cnc(O)o2)=O)C2CCC2)cc1Cl 85067,c1(C(N2CC(CCCCNC(C3C(F)(F)C34CC4)=O)C2)=O)cc2c(cc1O)OCO2 85068,N1(C(CC(c2ccc(F)cc2)C)=O)C2CCC1(CNC(C1CCC(=O)N1)=O)CC2 85069,CC(C(=O)N=c1cc2n([nH]1)CCCC2)C1CCCN(C(=O)C(C)(C)C2CCC2)C1 85070,C12(NC(Cc3nc(CC)sc3)=O)COCCC1CN(C(=O)C=C(C)c1ccsc1)C2 85071,N1(C(CCC=C)=O)CCC(C)N(C(=O)CC2CCOC(C)(C)C2)CC1 85072,C1(NC(C(C)N2CCCC2)=O)CCN(C(=O)CC2CC2)CCC1CO 85073,c1(OC)ncc(C)c(C(=O)NC(C)CNC(c2nc(C3CC3)cs2)=O)c1Cl 85074,c1(NC2CCCN(C(C(C)OCC3CCOC3)=O)C2)cc(Cl)ccc1Cl 85075,C#CCC(C)C(=O)N1CCCC1C(C)NC(c1ccc(C2CC2)nc1)=O 85076,c1(NC(=O)NC(CCCCC)c2ccccc2)cc(F)ccc1NC(C)=O 85077,CCC(C)C(C)C(=O)N(C)Cc1ccccc1CNC(=O)Cn1cnnc1O 85078,N1(C(=O)CC2CSC2)CCN(C(c2cnccn2)=O)C(CC(F)F)C1 85079,c1(C(N2CCCC2C(=O)N(C)C)C(=O)NC(CC)C)nc(C)ns1 85080,C1(NC(c2cncc(C)n2)=O)CN(C(=O)C=CC2CCCN2C)CC(F)(F)C1 85081,c1(NC(C2(OC)CC2)=O)cc(N)cc(F)c1.c1(C2C(=O)N2C)ccc(F)cc1.SC 85082,CC1CC(NC(C23CC(C(F)(F)F)(CO2)C3)=O)CCN1C(c1cncc(Cl)c1)=O 85083,C(=O)(C(C)(F)C(=O)OC)NCC1C(CNC(c2c(CC)ccs2)=O)C1 85084,C(=O)(CC1=NNC(=O)C1)NC1CCN(C(c2c(C)nsc2C)=O)CC1C 85085,c1(C(=O)OC)sc(C(=O)NC2CN(C(C3CCC4CC34)=O)C2)cc1C 85086,C(=O)(C1Cc2ccccc21)N1CC(CCC=C)(C(N2CCC(F)(F)CC2C)=O)C1 85087,c1(CC)c(C(=O)NCC2CCCN2C(C2CC2C2CCC2)=O)cnn1C(C)(C)C 85088,C1(NC(COC(CC)C)=O)COCCN(C(c2ccc(O)nc2C)=O)C1 85089,CC(C#N)CCC(=O)NCC1CCC(NC(=O)Cc2cccc(Cl)c2Cl)CC1 85090,N1(CC)CCOC(C(N2CC(O)CC2C(=O)N(C)CC2(C)CCC2)=O)C1 85091,C1(CNC(CC(C)NC(=O)COc2cccnc2)=O)CCCNC1=O 85092,n1(Cc2cn(CC(c3cnc(C)o3)C(C)C)nn2)cnc2ccc(Br)cc2c1=O 85093,CC1(C)NC(=O)CCC1CNC(=O)CC(F)(F)CC1CCCO1 85094,N1(C(C(C)N2CCCC2)=O)CCC2CCC(C1)N2C(=O)Cc1ncn(C)n1 85095,C1(C)(C(=O)NCC(CCCC)NC(=O)COC)Cc2ccc(C)cc2C(=O)O1 85096,N1(C(CC2C(CC)C2)=O)CC(CO)(NC(=O)CNC(C)=O)C1 85097,C1(C#N)(C(=O)NCCC(C)NC(c2n[nH]cc2C2CC2)=O)CC2(CCC2)C1 85098,c1(C(=O)NCC2CN(C(Cn3c(=O)ccc(C)n3)=O)C2)nc2ccccn2c1F 85099,CC(C)C(C(=O)NC(C)C(=O)NO)C(C)NC(c1c[nH][nH]c1=N)=O 85100,C(C(C(=O)NC1CC1)N1CCC(O)(C(=O)OC)C1)(C1CCCC1)OC 85101,c12cc(n(C)n1)C(=O)NCC1C(C1)C(=O)NC2.C1(COCC)CCCC12CC2 85102,CCCCCC(C)CC(=O)NCC(C(C)(C)C)NC(c1ncc2[nH]ncc2n1)=O 85103,c1(OC)c(Cl)ccc(C(N2CC(C3CC3)(NC(=O)C(F)(F)F)C2)=O)c1N 85104,CC1(C(N2CCC(CCCO)CC2)=O)CCCN1C(c1cc(=O)cco1)=O 85105,C(=O)(C(F)(F)C(O)C(C)C)NC(CC)CNC(c1nc2nc(C)ccn2n1)=O 85106,C1(CNC(C=CC=CC)=O)CC2(CO1)CN(C(c1ccc(OC)c(Cl)n1)=O)C2 85107,c1(C(=O)NCC(CC)NC(C2(N(C)C)CCC2)=O)cc(C)cc(Br)c1 85108,c1(C(=O)NCC(C(C)C)NC(CC(CC)C2CCC2)=O)ccc2ncncc2c1 85109,c1(CC(=O)NC2C(NC(c3c(SC)cnn3C)=O)CCC2)nc2ncccn2n1 85110,C1(C(N2CCC(C)(CNC(c3n(C)ncc3)=O)C2)=O)CCC(S(N)(=O)=O)CC1 85111,CCC(C)(C)C(C)CC(=O)N1CC(C(C)NC(c2c(C)n[nH]c2C)=O)C1 85112,C1(O)(CC)CCC(NC(=O)CC2(N(C(=O)C(C)CC3CCC3)C)CC2)CC1 85113,C1(C(=O)NCc2cnnc(O)c2)CC2CN(C(CCCCCO)=O)CC2C1 85114,C(CC(C)N=c1[nH]c2c(c(=NCC3COC(C)(C)C3)[nH]1)CCC2)SC 85115,N1(C(C(CC)=CCCC)=O)CC2CC(C)N(C(=O)CC=Cc3ccccc3)C2C1 85116,c1(OC)cccc(C(N2CCN(C(=O)C(O)C(C)(C)C)CC2CC(F)F)=O)c1C 85117,C1(C(=O)NC(C2CCCC2)CNC(c2nc(Cl)cs2)=O)CCNC1=O 85118,C1(NC(c2c(C(C)C)n[nH]c2)=O)CC2CC1N(C(=O)CC(C)F)C2 85119,C(C(C)(C)C(=O)NCC(C)CN(C)C(C1CCCC(=O)C1)=O)NC(C)=O 85120,C(C(N=[N+]=[N-])C(=O)NC1C2CC3C(C2)C13C(N1CCC1(C)C(=O)OC)=O)OCC 85121,c1(C(=O)OC)ccc(C(=O)NCC(C)N(C)C(c2nn(C)c(Cl)c2Cl)=O)c(Cl)c1 85122,C1(NC(C(c2c(C)cccc2)C)=O)CC2CC1CN(C(c1ccsc1)=O)C2 85123,c1(C(N2CCC(CCNC(c3cc(CC)sn3)=O)CC2)=O)cn2ccsc2n1 85124,C1(NC(c2ccc(C)n2C)=O)CCCCN(C(=O)Cc2nnn(C(C)(C)C)n2)C1 85125,C(=O)(C1=CC(O)C(NC(=O)CCc2cncnc2)C1)N(C)CCO 85126,C1(NC(=O)OC(C)(C)C)CCCCC1N=c1[nH]nc(CO)n1CCSCCO 85127,c1(C(N(C(C)CNC(C2CC2[N+](=O)[O-])=O)C)=O)ccc(Br)nc1O 85128,C1(C(N2CCC(OC)CC2)=O)CC2CCN(C(c3cc(OC)n(C)n3)=O)CC12 85129,N1(C(C2CC(C)=C(C)CC2)=O)CCC=C(C(=O)N2CCOCC(C)(O)C2)C1 85130,N1(CC(=C)C2CCOCC2)CCC2(CC=CCO2)CC1 85131,CC(C)CC(C(=O)N1CC(S(C)(=O)=O)C1)ONC(C1(C#N)CCCCC1)=O 85132,N1(c2snc(CCSC)n2)CCCCC(CNC(=O)CCN2CCOCC2)C1 85133,N1(C(C2(CC(C)C)CC2)=O)CCC2C(CCCN2C(c2cnn(CCF)c2)=O)C1 85134,C1(CN(CC=CC(N2CCC(C(=O)NC)C2C(C)C)=O)CC)CCCCCCC1 85135,C(c1ccccc1Cl)=CC(=O)N(CCC(C)(C)C#N)c1ccc(C(F)(F)F)cc1 85136,c1(NC(CCCN(C(C(CNC(CC(=O)OC)=O)O)=O)C)=O)ccc(C)c(Cl)c1 85137,N1(C(C2(C)C(C)(C)C2)=O)CCC(C(N2CCC(CO)(CO)C2)=O)C(O)C1 85138,N1(C(CCC(=O)OC)=O)CCN(C(c2cnnc(O)c2)=O)C2CC12 85139,O=C(C1=CCCS1)NCC(C1CCN(C(C2(F)CCOC2)=O)CC1)F 85140,c1(NC(C)CCOC)ccc(S(=O)(=O)NCC(c2ccco2)O)cc1Br 85141,CC(CC(=O)N1CCC(CN(C(=O)C=Cc2ncc[nH]2)C)C1)P(C)(C)=O 85142,c1(OC)c(C(N2CC3CC2CCC3NC(c2ocnc2C)=O)=O)cc(Cl)cc1C 85143,N1(C(C2CC(SC)C2)=O)CCn2c(CNC(=O)C(C)=C3CC3)nnc2C1 85144,c1(NCC(C2CC2)OC)ccc(S(=O)(=O)NCCN(C)C)c(Cl)c1 85145,c1(N2CC=CC(NC(C(C)CC(C)(C)C)=O)C2)ncc([N+](=O)[O-])cc1F 85146,C1(CNC(C(Cn2ccc(C)n2)C)=O)CC2(CCOCC2)CN1C(=O)C=C(Cl)Cl 85147,c1(CNC(=O)OC(C)(C)C)c(C(=O)NC2(C)CCS(=O)(=O)C2)cncc1F 85148,C1(CN(C)C(C2(Cl)CC2(F)F)=O)CCN(C(C2(c3cc[nH]n3)CC2)=O)C1 85149,C(=O)(C1CCCc2nc[nH]c21)N1CC(NC(=O)COCCCN(C)C)CC(C)C1 85150,c1(SCCCC(=O)NCC(C)(CC)NC(C(C=C)O)=O)nc2ccccc2[nH]1 85151,c1(CC(=O)NC(CNC(C(C)C(C)(F)F)=O)C2CC2)noc2ccccc12 85152,C(=O)(C(Cc1cnc[nH]1)NC(=O)C(C1CCCCC1)=O)NCC(C)CC1CC1 85153,C1(C(=O)NC(CN(CC)CC)C)CC12CCN(C(=O)Cc1sc(C)cc1C)C2 85154,c1(C(=O)NC2CCCN(c3nccc(C)n3)C2C)cn2nc(C)cc2[nH]c1=O 85155,CCC(C)C(C(=O)N1CC(C)(C)CC1CC(=O)NC1CC(=O)NC1=O)N(C)C 85156,C1(NC(C(CC)CC(F)F)=O)CN(C(=O)Cn2nccn2)C2CCCCC12 85157,Cc1c(C(N2CCC(NC(=O)C(O)C3CC3)C(C)(C)C2)=O)cc(N)cc1O 85158,C1(CC=C)(NC(=O)CSC(C)(C)C)CCCN(C(c2cc(Br)c[nH]2)=O)C1 85159,c1(-c2ccc(C(N3CCCC(F)C3)=O)cn2)cc(O)cc(Cl)c1 85160,C1(NC(c2cnc[nH]2)=O)CN(C(=O)Cc2cnccc2Cl)CC12CCC2 85161,C1(NC(C(C)(C)C(F)(F)F)=O)CN(C(C2CCC(C)(C)O2)=O)CC12CCOCC2 85162,Cc1cncc(CC(=O)NCCCNC(=O)C=CCn2cncn2)c1 85163,C(=O)(C(F)CC(C)C)NCC(C)(C(C)C)NC(C1CCN(C(C)=O)CC1)=O 85164,N1(C(C2C(C#N)C2)=O)CCCCCC1CO.C1(NC(=O)CO)CCN(C2CC2)CC1 85165,C(C)(C)(CC(=O)N1CCCCC1C(C)NC(=O)C=Cc1scnc1C)OC 85166,C1(C2(O)CN(C(=O)CC3CCCS3(=O)=O)C2)(CNC(C(C)C(C)(F)F)=O)CC1 85167,c1(C(N2CC3CN(C(c4c(C)nsc4)=O)CC32)=O)cc2cc[nH]c2cc1Cl 85168,CC(C)(O)C(C)(C)NC(C1CCC(CNC(c2cnn[nH]2)=O)O1)=O 85169,C(CCC(=O)N(CCCC1CCCN1C(=O)C(CC)OC)CC)N(CCOCC)C 85170,c1(NCC=CCNC(C(c2cccc(Cl)c2)CC)=O)cc(C)ccc1[N+](=O)[O-] 85171,c1(N2CC(C)(C)C(NC(=O)C(F)OC(F)(F)F)C2)ncc([N+](=O)[O-])c(=N)[nH]1 85172,c1(CCC(=O)NCC2C(NC(Cn3c(C)ccn3)=O)CC2)ccc(O)nn1 85173,C1(COC)(NC(=O)Cc2nnc(S)n2C)CCN(C(c2c(O)noc2C)=O)CC1 85174,Cn1nnnc1SCCC(=O)NCC1CC(F)(CNC(=O)Cc2cnoc2)C1 85175,C1(C(N2CCC(CC=C)(NC(c3ccccc3CO)=O)C2)=O)CN2CCC1CC2 85176,c1(N2CCC(CC=C)C2)nc(=NCCC(C)(C)OC)[nH]c2c1SCC2 85177,C1(N(C(=O)CCNC(=O)CO)CC)CCCN(C(=O)CCCC2CCCO2)CC1 85178,C(c1ncc[nH]1)=CC(=O)NCC1(OC)CN(C(=O)CSCCc2ccccc2)C1 85179,Cc1ccc(O)c(CC(N2CCOC(CN(C(=O)CC(C)O)C)C2)=O)c1 85180,N1(C(c2cc(CCC)on2)=O)CCC(NC(=O)CC2CC2(C)C)C(O)C1 85181,Cc1ncc2c(n1)CCN(S(=O)(=O)c1ccc(O)cc1)C2 85182,CN1CC(C(=O)NCC=CCNC(C2(C(F)(F)F)CC2)=O)C1 85183,c1(C(=O)NC23C(CN(C(CC4ON=C(C)C4)=O)C2)CC3)csc2c1CCC(C)C2 85184,N1(C(C(=O)NC2CC(NC(c3cc(C)no3)=O)C2)C)CCCCCC1 85185,C12(C(=O)NCc3c(C)nn(C)c3)CCCC1CN(C(C1CCCCS1)=O)C2 85186,O=Cc1ccnc(NC(=O)NC2CCS(=O)(=O)C2)c1 85187,CCC(C(=O)OC1CCC1)C(C)N=c1[nH]nc(C(F)(F)F)o1 85188,c1(SCC)cncc(C(=O)NC(C)C(C)NC(c2ccnnc2NC2CC2)=O)n1 85189,c1(C(=O)NCC(CC)NC(=O)C=CC2CCC2)cc2cc(C)cc(C)c2[nH]1 85190,CCCCCCC(F)C(=O)N(C1CCN(C(c2cccc(Cl)c2N)=O)C1)C 85191,C1(C(N(C2CCN(C(=O)Cn3cc(Cl)c(C)n3)CC2)CC)=O)CC(C2CC2)C1 85192,O=C(C1=CCCCC1)N1CCC1CC(N1CCC(n2cccn2)C1)=O 85193,CN1CCN(C(c2nccn2C)=O)C(CNC(=O)COC2(C)CCCC2)C1 85194,C=CC(CC)CC(=O)NCC=CCC(=O)NCC(C)N(C)C(C)C 85195,C1(CC)CN(C(c2ccncc2F)=O)CC1NC(=O)C(N1CCCC1)C1CC1 85196,c1(NC(C(CC)NC(=O)C(Cc2ccoc2)SC)=O)cccc(CCO)c1 85197,C1(C(=O)NC2CCCN(C(c3oc(C)c(CO)c3)=O)CC2)CC2CC1CC2(F)F 85198,CCCC(CCCNC(C1(C(=O)N(C)C(C)C)CC1)=O)NC(C1OCCCO1)=O 85199,CC1CN(C(C2(O)CC(F)(F)C2)=O)CC1NC(C1(F)CC1)=O 85200,CCC(O)C(C)(C)C(=O)NCCC1CCCN(C(=O)COCC2CCC2)C1 85201,C12(C(C)=O)CCCC1CCN2C(=O)Cc1c(C)nn(CC(C)C)c1C 85202,CON=C(C(=O)NCC1CC1CNC(c1coc(S(N)(=O)=O)c1)=O)c1ccco1 85203,C1(NC(C2C=C(C)CS2)=O)CC2CCC1C(NC(c1nnccc1C)=O)C2 85204,C1(NC(=O)NC2CCCC(C(C)C)C2)CC2(CCCCCC2)C1 85205,C(=O)(CC(C(F)F)NC(C1C2CCC(C2)C1C)=O)NCCc1ccc(C)s1 85206,c1(C(N(CC(CC)NC(=O)Cn2ncccc2=O)C)=O)cc(C)c(C(N)=O)cn1 85207,c1(CC)nc(CCNC(c2csc(C)c2)=O)no1.c1(CC=O)ccccc1 85208,N1(C(C2N(CC)CC2)=O)CC2CCC1(CNC(=O)CC(CN(C)C)CC)CC2 85209,N1(C(C2N(C(C=C(CCC)CCC)=O)CCC2)=O)CC(O)C(O)C1C(=O)OC 85210,O=C(C1CCCc2scnc21)N1CCCCC2(CCOCC2)C1 85211,c1(C(=O)NC(C(C)C)CCN(C)C(c2cnn[nH]2)=O)ccccc1N=S(C)(C)=O 85212,C1(C(=O)NC(Cc2ccco2)C(=O)N2CCC(CCO)C2)CC2(CCC2)C1 85213,c1(C(N2CC(NC(=O)CCC(=O)N3CCOCC3)C2)=O)ccc2c(c1)CC2 85214,c1(C(N2CCC(NC(CCc3cc(C)[nH]n3)=O)C2C2CC2)=O)c(O)cccc1F 85215,c1(C(=O)OC(C)(C)C)nocc1C(=O)OCCNS(=O)(=O)Cc1ccon1 85216,N1(C(C(=O)N(C(C)COC)CCOC)=O)CCCCCCCCCC1 85217,c1(C2(C(=O)NCCCN(C(=O)CCC3CCCO3)C)CCC2)cc(Cl)cc(Cl)c1 85218,c1(CC)ccccc1C(=O)NC1CC(C)N(C(=O)CC2CN(C)C2)C1 85219,O=C1CCC(CC(=O)N(CCCNC(c2ccc(F)o2)=O)C2CC2)C(=O)N1 85220,c1(CC)ccccc1-n1nnnc1C1(NCc2ccc(COC)o2)COC(C)C1 85221,C(CCC)(C(=O)N1CCC(C(=O)NCCOCCOC)C1)=CC 85222,C12CCCCC1NCCOCCN(C)C2=O.C1(OCC)CC(C(=O)N(C)C)C1 85223,CC(C(=O)N1CCC(NC(c2csc(-c3ncc[nH]3)n2)=O)C1)C(F)(F)F 85224,C(=O)(CCCCC(=O)OC)N1CCC(N(C(CC(CCC)O)=O)CC)CC1 85225,c1(C(=O)NCC2N(C(C3OCC(C)C3)=O)CCN(C)C2)nnc2n1CCCC2 85226,C(=O)(C(C)(C)C(C)(C)C)NC1CC(C)(CNC(C2(SC)CC2)=O)C1 85227,C1(C(N(C(CC)C(C)O)C)=O)CCOC(CNC(C)=O)C1 85228,c1(C(N2CC(CNC(c3cn(C)nc3O)=O)C2)=O)c[nH]c2cccnc12 85229,c1(C(=O)NC2C(NC(CCc3ccc(C)cc3)=O)C2)ccc(S(N)(=O)=O)cc1 85230,c1(CCC(=O)NCCOCCC2=NCCCC2)cnc2cccc(Br)n12 85231,CC(=O)CCN=C(NCc1ccccc1F)NCC1CCC2(CCOC2)O1 85232,c1(N(C2CCN(C(C3(C)C=CCC3)=O)CC2)C)ncc2ncnc-2[nH]1 85233,c1(C(N2CC(C)C(NC(c3cnn(C)n3)=O)C2)=O)nc(O)[nH]c(=O)n1 85234,C(=O)(CCC(=O)NCC1CC(O)CN1C(=O)CCc1cnc(C)s1)NCCC 85235,c1(OCCCC)ccc(C(=O)NCC2CCN(C(C3CCCOC3)=O)C2)c(Cl)c1 85236,CC(CC(C)(F)F)C(=O)NCCC(C)NC(=O)CCC(=O)c1ccccn1 85237,c1(OC)ccc(C(=O)N(C(CNC(=O)C(C)(CO)OC)C2CC2)C)c(OC)c1 85238,CN1CCCC2CN(C(c3ccnc(Cl)c3Cl)C(=O)NC3CC3)CCC12 85239,C1(CNC(C2C(C)(C)C2)=O)CCCCN1C(=O)Cc1cnsc1 85240,N1(C(C(N2C(CC)CCCC2)=O)=O)CC2CCC(C1)N2C(c1cc[nH]c1)=O 85241,CC1=C(C(=O)NC23CCC(C2)N(C(=O)CC2CC4CCC(C2)N4C)C3)SCCO1 85242,C(=O)(C1=CCC2CCC1N2C(C1CC12CCCCC2)=O)Nc1c(C)c(F)ccc1 85243,C1(C(=O)NC2CC(OCC(=O)NCC3=NOCC3)C2)CC2CCC(C1)O2 85244,c1(C(=O)NCC(C(=O)NC(CCCC=C)C2CC2)OC)ccc(F)c(C)c1 85245,Cc1cc([N+](=O)[O-])cnc1C(=O)NCCN(C(c1cc(CO)c(C)o1)=O)C(C)C 85246,N1(Cc2n(C)cnc2)CCC2(CCCOC2)C1.C12CC(C1)C(=O)N2 85247,C1(C2CCN(C(C3CC3C)=O)CC2)(NC(c2cc(C)cc(Br)c2N)=O)CC1 85248,N1(C(CCN(C(c2n(C=C)nnc2)=O)C)=O)CCN(C)C(C)C1C 85249,CC1CC(NC(c2cc(C(N)=O)co2)=O)CN1C(c1snc(O)c1Cl)=O 85250,c1(C(N(CCCNC(=O)Cc2cc(C)on2)CC)=O)ccnc(CO)c1 85251,CCC(CC(F)(F)F)C(=O)NCC(C)(CC)NC(C1CC2C=CC1C2)=O 85252,Cc1ccc2c(c1)CC(C(=O)NC1CC3CN(C(c4ccccc4Cl)=O)CC13)S2 85253,c1(CC(=O)N(C(C)CN(C)C(=O)C2CC2)C)ccc(NC(=O)NC2CC2)cc1 85254,C(=O)(C(Cc1cn(CC(N)=O)nn1)NC(=O)CN(C)C(=O)N(C)C)NCCSC 85255,CCC(F)(F)C(=O)N1CCC(C(C)(C)NC(=O)CN2CC(C)(OC)C2)CC1 85256,c1(C(=O)NC2CC(C)(CNC(CCCOCC)=O)C2)ccc2[nH]cc(C#N)c2c1 85257,CCC(C)C(C)(O)CNC(=O)C(C1(O)CCC1)NC(=O)CCCn1cccc1 85258,c1(NCCCN(C)C)nccc(=NCCc2nncn2C)[nH]1 85259,c1(C(=O)NC(CNC(c2ccc(C)cn2)=O)(C)CO)nn(C)c2c1CCCC2 85260,c1(C(N2C(C(=O)NCCc3ccncc3)CSCC2)=O)ccc(O)cc1O 85261,C1(CC(N2CC(C)(NC(C3C(C)OCCO3)=O)C2)=O)COC2(CCC2)CO1 85262,CC1=C(C(=O)NCc2cc(C(=O)NC(C(O)CO)C3CCC3)on2)CCO1 85263,C1(NC(C=C(CNC(C(CCC)C#N)=O)C)=O)CCc2nnnn2C1 85264,c1(OC)ccnc(F)c1C(=O)NCC1CCN(Cc2csc(Br)n2)C1 85265,C(CC(C)(C)C(=O)N1CCC(C)C(CNC(c2ncccc2F)=O)C1)OC 85266,c1(OC)cccc(C(C)CC(=O)NC(C)CCNC(=O)CCc2ccon2)c1 85267,S(=O)(=O)(c1cccc(=NC2COC3(CCCCC3)C2)[nH]1)NC(c1cc(Br)cs1)C 85268,CC1(C)CC(CC(=O)NN2CCC3CC23)CN1C(=O)C(F)C(F)(F)F 85269,C#CCCC(C(=O)NCCOCCF)NC(=O)C(O)CCC 85270,c1(C(=O)NCC(=O)NC(C)C(=O)NC(C)(C)C)cn(C2CC2)cn1 85271,C1(CC(=O)NC2CCN(C(c3ccc(CCC=C)cc3)=O)C2)CC(F)(F)C1(F)F 85272,C1(CCC)CN(C(C2(Cl)CC2(C)C)=O)CCN1C(=O)C=CBr 85273,N1(C(C(C)Oc2ccccc2)=O)CC2CCC(C(=O)NCC3(C)CSC3)(C2)C1 85274,N1(C(c2c(CNC(C(C)(C)n3cnnn3)=O)cco2)=O)CC2C=CC2C1 85275,C(=O)(C(C)S(=O)(=O)C1CCOCC1)NC1CCC(NC(C(C)NC(C)=O)=O)CC1 85276,c1(C(C2CCC2)NC(=O)NC(C)CC2CCC2)ccc(F)cc1F 85277,N1(C(c2c(C)oc(C3CC3)c2)=O)CCCC(c2ccccc2)CC1 85278,c1(CCC(=O)NC2CCC(N(C(CC=C=C)=O)C)CC2)ccc(C)c(C)c1 85279,C(=O)(C(CCOC)SC)NCCOC(C(=O)N(CCCCC)C)C 85280,N1(CC(=O)NC(CNC(CSC(C)C)=O)(C)C2CCC2)CCC(F)(F)C1 85281,CC1CCCN(C(c2cccnc2)=O)C1CNC(C12CC3CC1C2C3)=O 85282,CC1OCCOC1C(=O)NC(C1CCCN1C(c1cc(C(N)=O)co1)=O)(C)C 85283,CCC(O)CN(C(=O)C(=O)NC(COC)C1(C)CC1)C 85284,c1(CC)[nH]c(=N)sc1C(N1CC(NC(=O)Cc2ccnc(F)c2)C(C)C1)=O 85285,Cc1cc(NC(C2CCCCN2C(=O)OC(C)(C)C)c2nn[nH]n2)ccn1 85286,C(CC(C)C(=O)N1CCCC(NC(C2(CCS(N)(=O)=O)CCC2)=O)C1)=CC 85287,Cc1nc(CN2CC(C(=O)OC)C(O)C2)c(C(C)(C)C)s1 85288,Cc1ccc(C(=O)NC(CNC(=O)C(Cc2ccccc2)C2CC2)CO)c(Cl)c1 85289,c1(NC(C2CC(OC)CN2C(=O)Cc2ccc(O)cn2)=O)ccc(O)cc1Br 85290,N1(C(C(=O)NCC2CCSCC2)=O)CC=C(c2ccc(Br)cc2)CC1 85291,C#CC1(NC(=O)CCC2(NC(=O)Cn3cnnn3)CCCC2)CCCCCC1 85292,c1(C(=O)NC2CCN(C(CCC)=O)CC2C)c(Cl)nc2cc(Cl)ccn12 85293,c1(C(=O)NCCN(CCC)C(C2(C)CCOCC2)=O)ccc(C2(C)CC2)cc1 85294,c1(C(N2CC(CO)OCC2C)C(=O)NC)cc(OC)cc(OC)c1Br 85295,c1(-n2c(CCN3CCCC3)nc(C(CC)C)n2)ccc2nccnc2c1 85296,CC1(C)CC(C(=O)NOCC(=O)NC2CC23CCCCC3)CN1CCC1CC1 85297,Cn1ncnc1CCNC(C1(CCNC(=O)CC2(C)CCOC2)CC1)=O 85298,c1(CNS(CC)(=O)=O)cn(CCCN(C(=O)CC2CNC(=O)O2)C)nn1 85299,C(=O)(CCCCCF)NCC1C(NC(c2c(CC)ncs2)=O)C1 85300,C1(C(=O)NCC=C(C)C2CC2)CC12CCN(C(=O)CCN1CCOCC1)CC2 85301,C(=O)(C1(C)OCCc2ccccc21)N1CC(CC)(NC(=O)C(C(C)(C)C)SC)C1 85302,Cn1nnc2c1CCN(C(=O)C(C1(C)CC1)NC(C1CCCOC1)=O)C2 85303,C1(C)(C(C)C)C(=O)N1.n1(C(CC)C)c2nnc1SC2.c1(CO)ccc(Cl)cc1.CC 85304,C(=O)(CCN(OC)C(=O)C=Cc1cncn1C)NCC1(OC)CCOC1 85305,n1(CC)ccc(CC(=O)NC2CCN(C(=O)C(C)(C)c3cscc3Cl)C2)n1 85306,CC1CC(N(C(=O)C(C2CC2)N(C)C(c2ccoc2Cl)=O)C)CC(C)C1 85307,N1(C(C(C)S(N)(=O)=O)=O)CCN(C(C2Cc3ccccc3C2)=O)C2CCCC12 85308,Cc1c(C(=O)N(CCCN(C(=O)CC2(C)CCCCC2)C)C)cnn1CCO 85309,C1(Nc2nc(C)c(Br)cn2)(CNC(=O)C(C)(C)CN(C)C)CC2CCC1CC2 85310,C(=O)(CCCC(CC)CC)N1CC(CC(=O)NCCC(CCC)C2CC2)C(C)C1 85311,C1(CCNC(CC(C)C2CC2)=O)CSCCN1C(=O)CCCc1cccs1 85312,N1(C(Cc2ncc(CC)[nH]2)=O)CCC(C)C(CNC(c2nc(C)sc2C)=O)C1 85313,c1(C(=O)NCCOCCN(C(C2C(C)CCO2)=O)C)ccc(F)c(F)c1O 85314,N1(C(C2(c3cccc(Br)c3)CCCCC2)=O)CCC(F)CC1 85315,c1(C(=O)NC2C(CC)N(C(=O)CNS(N)(=O)=O)CC2)cn(C)c2ccccc12 85316,C(=O)(CN=S(C)(C)=O)NCC(CNC(C(C(C)O)N(C)C)=O)CO 85317,C(=O)(C(CC(C)C)C(C)C)NC1C(NC(CCCCC=CC)=O)C1 85318,N1(C(C(=O)NCCOC)CCC2CC=CCC2)CC2CC1CN2C1CC1 85319,C12(C(=O)NC3CCN(C(C4CCSCC4)=O)C3)CC(CO)(C1)OC21COC1 85320,N1(C(CCCC#CC)=O)CC2(CNC(C3CCCSC3)=O)CC1CCO2 85321,c1(C(N2CCC(CC(N3CCCC(CCO)C3)=O)C2)=O)ccncc1Cl 85322,Cc1nc(C(=O)NCC(C)(C2CC2)NC(c2ccn(-c3ccncc3)n2)=O)co1 85323,CC1(C)CCCCC1=CC(N1CC2CC1C2CNC(c1ccc(Cl)cc1)=O)=O 85324,CC(CC(=O)NC1CCC(CNC(C2CCOCC2)=O)C1)C(C)(C)C 85325,c1(CC(=O)NC(C2CCN(C(CCCC(C)C)=O)C2)C)ccc2cnccc2c1 85326,c1(CNC(c2nccn2-c2ccccc2)CCC)ccc(C(=O)O)o1 85327,c1(C(=O)NCCCNC(C2CC(CC)C2)=O)cc([N+](=O)[O-])cnc1N 85328,Cn1nc(Cl)c(C(=O)NCC2CCCN2C(c2ccncc2O)=O)c1Cl 85329,CC1CC(NC(C2CCCCC2)=O)CCN1C(C1CC(=C2CCC2)C1)=O 85330,CC1(C)CC(NC(=O)CC2CCCN2C(C2CCCN2C2CCCC2)=O)C1 85331,C(CC(C(=O)NCC1CCCO1)NC(=O)C(c1ccnn1C)C)=CC 85332,C1(CC)C(NC(c2ncnc(C)c2C)=O)CCCN1C(=O)CN(C1CC1)CC 85333,N1(C(C(COC)NC(C)=O)=O)C2CCC1C(NC(=O)Cc1nc(=N)[nH][nH]1)C2 85334,C(C(CC1CC1)C(=O)N(C(C)CNC(C)=O)C)NC(Cc1c(CC)con1)=O 85335,Cc1nc(C(=O)NC2CN(C(c3ccc4snnc4c3)=O)C2)ccc1[N+](=O)[O-] 85336,N1(C(CC#N)=O)CC2(CNC(=O)C(O)Cc3ccncc3Br)CCCC1C2 85337,N1(C(COCCCCC)=O)CC(NC(=O)CN(C)CCC)CC2COCC12 85338,C=CCC(C)C(=O)NCC(C(C)C)NC(c1cc(C(C)=O)c(C)o1)=O 85339,S(=O)(=O)(c1cc(C(N2CC3(C2)CN(C(=O)OC(C)(C)C)CCO3)=O)c(C)o1)NC 85340,Cc1scc(C(=O)OCC(O)CN(c2ccc(OC(F)F)cc2)C=O)c1C 85341,c1(C(N(C2CCN(C(C(CC)F)=O)C2)C)=O)cc(C(F)F)ccn1 85342,C(C(=O)NNc1ncnc2c1ncn2C)NC1C(C)Cc2ccccc21 85343,CC1(CNC(c2ncn(C(C)(C)C)n2)=O)CC(NC(C2(c3cccs3)CC2)=O)C1 85344,c1(CC)c(OC)cc(C(=O)NCC2CCN(C(=O)C=CC(F)(F)F)C2)cc1OC 85345,CC(C)CC(=O)NCCC(C)N(C(=O)C(n1cc(Br)cn1)C)C 85346,c1(CNC(C(C)C)(CCN2CCOCC2)c2nnnn2C)cc(C#N)ccc1[N+](=O)[O-] 85347,c1(C(N(OCC(C)C)Cc2ccccc2)=O)ccc(CC(=O)OC(C)(C)C)cc1 85348,c1(C(=O)NCC(C)N(C)C(c2cn(C3CCCCC3)nn2)=O)cccn(C)c1=O 85349,C1(CNC(CC(CC)OC)=O)CN(C(=O)CN(C)C(C)C)C2COCC2O1 85350,C1(NC(C(c2scc(C)n2)C)=O)CN(C(=O)CC2CC2(Cl)Cl)C2CCCCC12 85351,C1(NC(c2c(C)nco2)=O)COC2(CCN(C(c3ccnc(O)c3)=O)C2)C1 85352,c1(C(N(CCCC(C)C)C)=O)ccc(CN2CC(N)C2)cc1 85353,CC1CC(C(=O)NCC2CCCN2C(=O)CCn2cccn2)CCS1(=O)=O 85354,N(C1CCCc2nc(C)sc21)C(C(=O)OCCC)C(C)C 85355,N1(C(c2c(C)[nH][nH]c2=N)=O)CC2(C1)CN(C(c1ccc(C(C)(F)F)cc1)=O)C2 85356,N1(C(c2cnc(C(C)(C)CF)o2)=O)CCC(NC(C2(C3CCCO3)CC2)=O)CC1 85357,c1(N(C(=O)C(=O)NC(c2c(F)cccc2Cl)C(=O)O)CC)cccc(OC)c1C 85358,c1(CC(=O)N(CC(C)(C)CNC(C2CC3CC3C2)=O)CC)ccccc1Cl 85359,c1(COC)cc(N2CCCC(C(=O)Nc3cccnc3C)C2)ncn1 85360,c1(C(=O)NCC(CO)NC(c2c(C)nc(CC)s2)=O)nc(C)n(C)c1C 85361,N1(C(C(C)C)=O)CCN(C(=O)C(c2ccc(O)cc2)N(C)C(=O)OC(C)(C)C)CC1 85362,C(CCCC(=O)N1CCCC(CCS)C1)N.C(=O)(C(C(C)C)NC=O)CCC=C 85363,c1(NCCNC(=O)NCc2cc(F)cc(F)c2F)ccc2c(c1)OCO2 85364,Cc1cccn2nc(C(=O)NCC(C)N(C(=O)CCC3CC3(Cl)Cl)C)cc12 85365,C(CC(=O)NOCC(=O)NCCCCC(C)C)N(CC)CC 85366,c1(CCC)nc(=NCC2CN(C(=O)CCCc3ccc(C)cc3)C2)s[nH]1 85367,c1(C(N2CCCC(C3(C)N=N3)C2)=O)cc2cc(C#N)ncc2[nH]1 85368,C1(C)(C(N(CC(CN(C)C)(C)C)C)=O)CCN(C(C2CC2C2(C)COC2)=O)CC1 85369,c1(C(=O)NCCCNC(C2CCC(C)(O)CC2)=O)cc2n(n1)CC(F)C2 85370,C(=O)(CS(=O)C(F)(F)F)N(CCNC(c1c(C)ccs1)=O)CCOCCO 85371,c1(-c2c(-c3cn(CC=C)nn3)cccc2)ccc(F)cc1F 85372,N1(C(C2(C)CCN(C)C2)=O)CC(C2CCCN(C(=O)C(C)(C)CS(N)(=O)=O)C2)C1 85373,Cc1cc(CNC(c2ccc(-c3n[nH]c4ccc(C)cc34)cc2)=O)c2n[nH]cc2c1 85374,Cc1n[nH]c(C)c1CC(C)C(=O)NCC(O)CN(C(=O)CSCC(N)=O)C 85375,C1(C(N2CCCC(N3CCC3)C2)=O)C2CCCC2CN1C(c1cccc(F)c1)=O 85376,C(=O)(C(CC(C)(C)C)OC)N(CCOC)CCNC(C1COCOC1)=O 85377,c1(OC)cc(OC)cc(C(N2CC(CN(C)C(C3CCCC3(C)C)=O)C2)=O)c1 85378,N1(C(CC(CC)(C)C)=O)CCCC2(CCN(C(=O)Cn3cc(CO)nn3)CC2)C1 85379,C1(C(N2C(CC=C)CCCC2)=O)C(C2CC2)CCN1C(C1CC(C)C1)=O 85380,Cc1nccnc1C(=O)NC(C1CC1C(=O)NC(CCO)C1CCCC1)C 85381,c1(C(=O)NCC2N(C(=O)CC3CC(=O)C3)CCN(C)C2)cc(O)c2ccoc2c1 85382,C1(CN(CC)CC)CCN(C(C2(NC(c3[nH]ccc3C)=O)CC2)=O)CC1 85383,c1(C(=O)NC23CCCC2CN(C(c2cc(O)cs2)=O)C3)cnc(O)c2ccsc12 85384,CC(C)(C)CCC(F)C(=O)N1CC(CNC(c2cnc(S)[nH]2)=O)C2(CCC2)C1 85385,C(=O)(C(C)(CNC(C)=O)CC(C)C)N(C(c1ccccc1)C(OC)OC)C 85386,C(C(O)C(F)(F)F)NC(CC1N(C(C2C(C)(C)C2)=O)CC1)=O 85387,c1(OCc2cn(C3CN(C(c4scc(C)n4)=O)C3)nn2)ccc(I)cc1Cl 85388,c1(NC(C(OC)OC)=O)nc(C)c(C(=O)N(CC2CCCCC2)OC)o1 85389,c1(SC)ncc(N)c(C(=O)NC2CCN(C(=O)C(C)NS(C)(=O)=O)C(C)C2)n1 85390,c1(N2CCC(CC)(CC)CC2)nc(NCCC2OCCC2(C)C)c2ncsc2n1 85391,C(=O)(C(C(C)(C)C)NC(=O)OC(C)(C)C)Oc1cc(N(S(C)(=O)=O)C)c(N)cc1 85392,CC1(C)CN(C(=O)COC2CCOC2)CC1C(=O)NCCn1cccnc1=O 85393,c1(OC)ccn2[nH]c(=NC(=O)C3CCCN(C(=O)Cc4nc[nH]n4)C3)nc2c1 85394,Cc1c(Br)ccc(NC(C2CC2C(=O)NCc2ccc(Br)cc2Cl)=O)c1F 85395,C=CC(CC(=O)NC12CC(C1)N(C(c1cnccc1OC)=O)C2)c1ccccc1 85396,c1(OC)c(F)cc(C(=O)NCC2CC2NC(=O)C(C2CC2)C2CC2)cc1Br 85397,C1(CNC(C=Cc2ccc(C)nc2)=O)CN(C(c2ns[nH]c2=O)=O)CC(C)(C)C1 85398,c1(C(N(CCN(C(C(CCSC)OC)=O)C)C(C)C)=O)cc2scc(Cl)c2[nH]1 85399,CC(CC(=O)NCC12CCCC(CN1C(C1COCCOC1)=O)C2)CC(F)(F)F 85400,CC(C)C(C(=O)N(C1CN(C(=O)CCF)C1)C)n1cccc1 85401,C(CC(C(=O)NCC1(O)CCSC1)NC(=O)CN(C)C1CC1)N(C)C 85402,C=CCC(CNC(c1c[nH]c(C(N)=O)c1)=O)NC(C1CC(CF)C1)=O 85403,c1(CCNC(C(CCN(C)C)N)=O)nc2ccc(O)cc2o1 85404,CCC(CC(=O)N1CC(C(=O)NCCC(C)C(C)C)C2(CCC2)C1)C(C)(C)C 85405,N1(C(COCC=C)=O)CCC(C)(C)CC1C(=O)N(CC(F)(F)CC)C 85406,Cc1c(S(=O)(=O)N2CCCC(C)CC2)sc2cc(F)ccc12 85407,c1(C(N(C2CN(C(CC(C)C3CC3)=O)CC2O)C)=O)cc2c(cnn2C)nc1O 85408,N1(C(C(=O)N(C)C)=O)CCN(C(C2CCC3CC23)=O)C2(CC2)C1 85409,C1(C(=O)NC2CC(CCNC(C=CC(C)(C)C)=O)C2)CCCCNC1=O 85410,c1(C(N2CCC(NC(c3n(CC)nnc3)=O)(CO)C2)=O)c(OC)ccnc1O 85411,Cc1cn2cc(C(=O)NCC(CC(C)C)NC(=O)C(C)n3cnnn3)sc2n1 85412,Cc1cc(C)c2nc(NC3CCN(C(c4cnc(C(C)O)s4)=O)C(C)C3)sc2c1 85413,c1(C(=O)NC(CNC(C(CCC)OC)=O)CC)c(N)sc(C)c1C 85414,Cc1cc(Cl)nc(N)c1C(N1CCCC(O)(CNC(=O)CC2CCCC2O)C1)=O 85415,c1(CC)ccccc1OCC(=O)N(CC(C)(C)CNC(=O)C=C1CC1)C 85416,c1(C(=O)NCC2CC(NC(CCc3cnc(C)o3)=O)C2)ncn2cc(Cl)ccc12 85417,c1(NCc2cc(C)ncn2)nc(N2CC3CC3C2)nc2sccc12 85418,C1(C)(NC(c2ncn(C)c2)=O)CCN(C(c2nnc(C(C)(C)C)s2)=O)C1 85419,N1(C(C2N(C)CC(O)C2)=O)C2CC=C(C(=O)NCc3n[nH]c4c3CCC4)C1CC2 85420,c1(C(N(C(CN(C(c2nc(C(C)=O)sc2)=O)C)C)C)=O)ccc2sncc2c1 85421,C(C(CC(C)C)C(=O)N1CCSC2CCCC12)NC(CCn1ncc(C)c1)=O 85422,N1(C(CC(C)C)=O)CCCC(N(C(=O)Cn2ccccc2=O)CCO)C1 85423,N1(Cc2c(CC)noc2CC)CCC(NC(=O)CC2CCCC2(F)F)C(C)C1 85424,C#Cc1ccc(C(N2CCCC(CNC(=O)C(C)CS(C)(=O)=O)CC2)=O)cc1Cl 85425,C1(CNC(c2c(C)nc(O)[nH]2)=O)CCC12CCN(C(=O)Cc1csc(Cl)c1)CC2 85426,C1(N(CCCc2nccc(C)c2)CC(=O)OC(C)(C)C)CCC2(CC1)CNC2 85427,Cc1cc(C(=O)NC2CCC(NC(c3ccc(O)nc3C)=O)C2)cnc1C 85428,C=C(C)CN=C(NCC12CC3CC1C2C3)N(C)CCCc1ccccc1 85429,C1(C(=O)NC(CN(C(C=C(C)C2CC2)=O)C)C)CC(c2cc(F)ccc2F)=NO1 85430,C#CC1(O)CCN(C(C2(CF)CCN(C(=O)CCc3cn[nH]c3)C2)=O)C1 85431,Cc1ccc(O)c(NC(C2(CNCC3(Cc4ccccc4)CC3)CC=CC2)=O)c1 85432,Cc1ccc(C(=O)NC23CCC2CN(C(=O)CCN2CCCCC2)C3)nc1C 85433,N1(C(c2cccc(C(C)C)n2)=O)CCCC(C)C1CNC(=O)CC1(C)CC1(Cl)Cl 85434,Cn1ccc2[nH]c(C(=O)OC3CN(C(=O)NC(=O)NC(C)(C)C)C3)cc12 85435,N1(C(c2c(OC)cc(N)cc2)=O)CCC2(CCC2NC(c2cc(F)n[nH]2)=O)CC1 85436,c1(NC(=O)NC(c2n(C)ncc2)C2CC2)cccc2c1CNC2=O 85437,N1(C(c2cnc(SC)s2)=O)CC2CS(=O)(=O)CC2(CNC(=O)C(C)C)C1 85438,S(=O)(=O)(c1c[nH]ccc1=NCCn1cnc(C)c1C)NCC1C(CCC)CCC1 85439,c1(OCCNC(N(CC(C)C)CCC)=O)cc(O)ncc1Br 85440,C1(OCC(=O)NC(CNC(c2cnn(C)c2F)=O)C(C)(C)C)CCC(F)(F)CC1 85441,C(CC(C)(O)c1ccccc1)NC(c1nc(-c2ccncc2)cs1)C 85442,c1(C(=O)NCC2(F)CC(CNC(C3C(C)C3)=O)C2)ccc2nc(=N)[nH]n2c1 85443,C=CCCCC(C)(C)C(=O)NC1CCCC(NC(=O)C(CC2CCCC2)CC)C1 85444,C1(NC(Cc2cnc(C)o2)=O)C(C)CCN(C(=O)CCS(N)(=O)=O)C1C 85445,Cc1cn2cc(C(=O)NCC3CCN(C(c4ccc(N(C)C)nn4)=O)C3)sc2n1 85446,N1(C(C(C2CCOC2)OC)=O)CCN(CCNC(c2cnc(C)s2)=O)CC1 85447,c1(OC)ncc(C(=O)N(C)CC2CCCN(C(C3CC4CCC3O4)=O)C2)cc1Cl 85448,C=CCCCCCCCCC(=O)NCC1CC(NC(=O)CC(C(=O)OCC)SC)C1 85449,c1(C(=O)NC2CC(CCNC(COC)=O)C2)cc(C2CC2)nc2onc(C)c12 85450,CC(O)C(F)(F)C(=O)NC1CCN(C(=O)Cc2ccc(Br)cc2)C1 85451,Cn1nccc1C(F)=CC(=O)NC12CC1CN(C(=O)CSc1nccs1)C2 85452,N1(C(C(CC#C)CC#C)=O)CC2(C1)CN(C(=O)COCC1CC1)CCO2 85453,N1(C(C2(NC(C(CC=C)C)=O)CCSC2)=O)CC2CN(C)CC2C1 85454,N1(CCCCCC)C(=O)CN(CC2CCC(C)(C)O2)C1=O 85455,C1(C(=O)NC2CCCC(NC(=O)CCCC3CC3)CC2)CCn2ncnc2C1 85456,C(=O)(C(C(F)(F)F)C(F)(F)F)N1CCC2(C(CNC(CC(CC)CC)=O)C2)CC1 85457,C1(CCNC(C2(CC=C)CC=CC2)=O)CCCN(C(=O)CC2C(C)C2(F)F)CC1 85458,C12(NC(C(C)CF)=O)CCCC1N(C(c1ccnc(S)c1)=O)CC2 85459,c1(C(=O)NC2CN(C(CCN(CC)CC)=O)C3C2C3)cc([N+](=O)[O-])cnc1O 85460,C(C(COC)CC(=O)NC1CCCN(C(=O)Cn2nc(C)ccc2=O)CC1)OC 85461,N1(C(C2(N(C(c3c(C)con3)=O)CC3CC3)CCC2)=O)CCCC(C(C)(C)O)C1 85462,C(CC(C)C(=O)N(C1CCCN(C(c2cnn(CCSC)c2)=O)C1)CCO)OC 85463,N1(C(CN(OC)CC)=O)CC(C(=O)NCCN2CCCCC2)(COC)C1 85464,C1(OC)CC2CC(NC(=O)CC3CCCN3C(=O)CC(=O)NC3CC3)CC12 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85483,Cc1ccc(=O)n(CC(N2CCC3C(NC(=O)CCc4cn(C)nc4C)C23)=O)n1 85484,c1(C(C(=O)NC2(c3cn(C(C(=O)OCC)C)nn3)CCC2)O)ccccc1Cl 85485,N1(C(c2c(CC)ocn2)=O)CC2CCC(C1)N2C(C1(C)CCCC1C)=O 85486,c1(-n2ccc(CN(C(Cc3c(C)cccc3)C)C)n2)ccc(F)cc1F 85487,c1(CC)cc(C(=O)NC2CN(C(c3coc(C)n3)=O)C2)oc1CC 85488,Cc1cccc(CC(=O)NCC2(C)CCN(C(c3nc(C4CC4)sc3C)=O)C2)c1 85489,c1(OC)ccc(C(=O)NCC2CCN(C(=O)C(C)=C(C)C)CC2C)c(F)c1Cl 85490,C1(C#N)(C(N2CCN(C(c3n(C)nc(C4CCC4)c3)=O)CC2)=O)CC2C=CC1C2 85491,N1(C(C2C(C)OC(=O)N2)=O)CC2CC1CN2C(=O)CC1CC2CC2C1 85492,c1(OC)cc(Cl)c(C)cc1CNC(=O)C(N1CCC1NC(=O)OCC(C)C)=O 85493,N1(C(c2cc(C)ns2)=O)CCC(CCNC(=O)CCC#N)CC1C 85494,c1(C(N2CC3(CN(C(c4c(C)nc(C)o4)=O)C3)C2)=O)cc(C)c(Br)cc1C 85495,N1(C(c2cc(OC)n[nH]2)=O)C2CCC1(CNC(=O)C(C)CC1CCCO1)CC2 85496,c1(C(N(CC(C2CCC2)OC)C)=O)cc(O)nc2c(Br)cccc12 85497,C1(C(F)(F)F)(COC)CN(C(C)C(=O)Nc2cc(Cl)cc(Cl)c2)CCO1 85498,c1(C(=O)NCC(CNC(C2CCC(C)O2)=O)(C)C)ncccc1N 85499,Cc1cc(C)c(C(=O)NC(C2CCN(C(=O)CNC(c3ccsc3)=O)C2)C)[nH]1 85500,c1(C(=O)NCCCN(C(=O)Cc2cnccn2)CC)cc(C2(C)CC2)n[nH]1 85501,Cc1sc(C(=O)NCC2(F)CCN(C(=O)CNC(N)=O)C2)cc1Br 85502,C(CN=C(NCC1CCCCN1S(C)(=O)=O)NC(c1ccc(Cl)nc1)C)SC 85503,CC(CCCCNC(c1cc(C2CC2)[nH]n1)=O)NC(=O)Cc1ccnn1C 85504,N1(C(C2(C#C)CCCC2)=O)CC2CC(O)C1C2NC(=O)Cc1n[nH]c(=N)s1 85505,Cc1ccc(OCC(O)CNCCCC2CC2C)c(C)c1Br 85506,c1(NC(C2CC(=C)CN2C(C2(C)CC2)=O)=O)cccc(Br)c1OC 85507,C1(NC(=O)C(F)CC2CC2)CC2CCC1N(C(c1cc(O)c(O)c(O)c1)=O)C2 85508,c1(C(=O)NCC2CCCN(C(C(CC=C)(C)C)=O)CC2)c(Cl)nc2ccccn12 85509,c1(C(N2CCOC3(CCSC3)C2)=O)cc(F)c(Cl)c([N+](=O)[O-])c1 85510,CC1(C(=O)NCC2(NC(=O)CSCC3CCCCO3)CCOCC2)CC=CCC1 85511,n1(CC)cc(Br)c(C(N2CC3CC2C3NC(C2CCC(=O)N2)=O)=O)n1 85512,N1(C(c2cc(C3CC3)[nH]n2)C(=O)NC2(C)CC2)CC(CCO)C(CO)C1 85513,N1(C(c2c(C)oc(C(C)(C)C)c2)=O)CCC2C(C1)CN2C(=O)C(=O)C(C)(C)C 85514,C1(CS(=O)(=O)NCC2CCC3(COC3)O2)CC2CCCC(C1)C2 85515,n1(CC(=O)NC2CCN(C(C(C)(C)C3CC3)=O)CC2O)cccc([N+](=O)[O-])c1=O 85516,C1(C(=O)NC(C(=O)OCC)C2CC2)CCC(C)(C)N(C(c2cccc(CC)n2)=O)C1 85517,C(=O)(C(C)(CC)CO)NCC1(Cc2cn(CCCC(=O)OCC)nn2)CC1 85518,N1(C(C(=O)NC(C2(CCF)CC2)=O)=O)CCCCC1CCSc1cccc(F)c1 85519,c1(CCC)nccc(N(C(C2CCNCC2)C)Cc2cc(C)n(C)n2)n1 85520,CN1CCCC2C1CC(C(=O)NCc1cnc(C(F)(F)F)nc1)C2 85521,C1(C(=O)OC)CC(NC(=O)NCCOCc2ccccc2)C2CC12 85522,N1(C(CCCOC)=O)CCCN(C(c2cnc(C3CCCC(C)(C)C3)[nH]2)=O)CC1 85523,c1(C(N2CCN(C(C(C=C)(C)O)=O)CC2CC(F)F)=O)n[nH]c2ccc(C)cc12 85524,N1(C(=O)C(F)n2cccn2)CCN(C(c2ccc(F)c(F)c2)=O)C(CF)C1 85525,N1(C(CN(C(C)C)CC)=O)CCC2(CCC2)C1.C1C(C)OCCNC(=O)N1 85526,Cc1cc([N+](=O)[O-])cnc1C(N1CC2CCC(C1)N2C(C1(O)COC1)=O)=O 85527,c1(-c2cc(-c3n(-c4onc(C5CN(C)C5)n4)ccn3)n[nH]2)ccc2ncc(I)n2c1 85528,C1(CCNC(c2cc(COC)sc2)=O)CCCCN1C(C1COC(=O)N1)=O 85529,CCC(C)C(O)C(=O)NCC1(NC(c2cn(C)nc2Br)=O)CCOCC1 85530,c1(-n2cc(SC(C)C)nn2)ccc(C)c(C(=O)NC(Cn2c(C)cc(C)n2)C)c1 85531,C1(C(N2CC(=C)C2)=O)CCN(C(=O)C(CCC)OC)O1 85532,C(c1cnc(C(C)(C)C)s1)=CC(=O)NCC(CC)NC(C1(CC(C)C)CCC1)=O 85533,CCC(Cc1ccc(N)cc1)C(=O)NCCNC(=O)CCc1nnc(C(F)F)o1 85534,c1(-c2cc(C(C)C)no2)nc(C2CCCO2)nn1CC1CCSC1 85535,c1(CC(=O)NCC(C2CCCCC2)NC(CSCCCC)=O)cccc(Cl)c1 85536,C1(OC(C2OCCO2)=O)CC2(CCOC2)C1 85537,c1(OC)ccc2nc(N3CC4CC3C3CC43)[nH]c(=NCCC(O)C3CC3)c2c1 85538,C1(C(=O)NC(c2ccc(F)cc2)CNC(C(CO)N(C)C)=O)CSCC(=O)N1 85539,c1(C(N2CCC(CN(C)C(C3C(C#N)C3(C)C)=O)CC2)=O)cncc2nc[nH]c12 85540,CC1=NOC(C)(c2nc(-c3cc(C)c(-c4cccc(NS(C)(=O)=O)c4)s3)no2)C1 85541,c1(C(=O)NCC(n2cc(C3OCCO3)nn2)C)cnc2ncnn2c1O 85542,C1(C(C)(C)C)CN2CCN1C2=O.c1(OC(=O)NOC(C)(C)C)cc(Br)c[nH]1 85543,C1(C(=O)NC(CN(C)C(C2CC23CC3)=O)(CO)CO)CCCCCCC1 85544,C(CCN(C1(C)CC(C)(C)C1)C(c1ccccc1Cl)=O)(C(C)(C)C)NC(C)=O 85545,C1(NC(c2ccc(OC)cc2F)=O)CCCCN(C(=O)C(=O)NC2CC2)CC1 85546,C1(C(=O)NCCCN(C(=O)CCc2cccn2C)CCC)CCNC1=O 85547,C1(C(N2C(CNC(Cc3cn(CC)nn3)=O)C(C)CC2)=O)CCn2cncc2C1 85548,c1(COC(C2(C3(O)CCC3)CC2)=O)ncc(C(F)(F)F)cc1Cl 85549,N1(C(C(C(C)C)SC)=O)CCC2(CC1)CCN(C(C1CCC3CCCCN13)=O)C2 85550,Cc1nccc(C)c1CCC(=O)NCC1CC(F)(F)CN1c1nnc(C(F)F)s1 85551,C1(NC(C2(CNC(=O)CC34CCCC3C4)CCC2)=O)CC2CC1C(O)C2O 85552,c1(CN2CCCC(C(=O)NC(CCC)=O)C2)nc2ccc(C(F)(F)F)cc2o1 85553,N1(C(C(C)CN(C)C)=O)CCCC(NC(=O)Cn2cccnc2=O)CC1 85554,C(=O)(C(C)(O)C(C)C)N(C)CC1N(C(c2cc(CCOC)on2)=O)CCCC1 85555,C1(=CC(=O)NCC2C(CNC(C(CCSC)O)=O)C2)CCCCC1(C)C 85556,c1(CNC(C2CN(S(CC)(=O)=O)C2)=O)ccc2c(c1)oc(=O)n2C 85557,Cc1cc(CC(N2CCN(C(=O)C3=CCCCC3)C(C)C2)=O)cc(C)c1 85558,c1(CC(=O)NC(C2CC=CCC2)C(=O)NCCOCC(C)C)ccnc(O)c1 85559,c1(C(=O)NC2CCN(C(CN3CC(CC)C3)=O)C2)c(C)noc1Cl 85560,C1(NC(C2N(C(C)C)CCC2)=O)COC2(C1)CN(C(c1cncs1)=O)C2 85561,C(=O)(C1CCOc2ccc(Br)cc21)N1C(c2cn(C)nc2)C(=O)N(C)CC1 85562,C1(C)(CC)CC(NC(c2ccc(C(F)F)cn2)=O)CN1C(=O)C=CC1CCCC1 85563,c1(CNC(C(=O)N(CCc2scc(C)n2)C)=O)csc(C#N)c1 85564,C1(C(N)=O)CN(C(C2CCC(NC(=O)CCSC3CCCC3)C2)=O)CCO1 85565,C1(C(N(CC(NOC)=O)C2CC2)=O)CCC2CCC1N2C(=O)Cn1ncccc1=O 85566,CC(C)C(C)(O)C(=O)N1CCC(C(C)(C)C)(CNC(c2nc(Cl)ccc2N)=O)C1 85567,C1(C(C)C)(C(=O)NCC2CC(C)(C)C2)CCN(C(c2cc(Cl)n(C)n2)=O)C1 85568,C1(N(c2n[nH]c3c2CCC3)C(=O)Cc2cccc(O)c2)CCC2(CCNC2)CC1 85569,C1(NC(=O)OC(C)(C)C)CCC2(CC1)CCN(c1nc(C(C)(C)C)no1)CC2 85570,N(C1CCc2ccc(Cl)cc21)C(c1ccc(C#N)c(C(F)(F)F)c1)=O 85571,C(=O)(C(C)(O)C(F)(F)F)NCCCC(C)(C)NC(C(CCC#C)O)=O 85572,C12(C(N3C(C4(NC(c5n(C)ncc5)=O)CC4)CCC3)=O)CC(C)(C1)OC21COC1 85573,C1(C(N(CCOCCC(=O)N(CC=C)CC)C)=O)COC(C(C)C)C1 85574,c1(C(=O)NCCCCCNC(=O)C=Cc2ccccc2)c[nH]c2c(F)cccc12 85575,C1(C(=O)NC(CC)(CNC(c2cnc(OC)s2)=O)CC)CC2(CCCC2)CO1 85576,c1(C(c2n(CCC)nnn2)NC(C)C)ccc(CNC2CC2)cc1 85577,Cc1cc(NCCC(C)C)n(CC(N2CCC(SC(C)(C)C)CC2)=O)n1 85578,CCC(CCC(=O)NCC1CC(C(N2CCOC(C)C2CO)=O)C1)OC 85579,C1(C(CNC(C2C(OC)CCC2)=O)(C)C)CCN(C(=O)C(C)(C)C)CC1 85580,CC1CC(NC(=NCCN2CCOCC2)NCCOC(C)(C)C)CCN1C.C1CCO1 85581,c1(C(=O)NCCCN(C)C(C2CCCN2C2CCOCC2)=O)ccncc1N 85582,c1(NC(C(C)(C)NC(c2cn(CC)nc2)=O)=O)cn(C)nc1C 85583,Cc1nocc1C(=O)NC1(C(N2CC(c3ccccc3)C2)=O)CC1C 85584,c1(C(=O)NC(CCOC)CNC(C2CC3(CCCO3)C2)=O)[nH]nc2cnccc12 85585,C(C)(CCCC(C)C)N(C(C1(CC#C)CCOC1)=O)CC 85586,CN=c1ccc(C(=O)NC2(C(=O)Nc3cnccc3C)CCCC2C)c[nH]1 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85798,C#CC1(NC(C2COCCN2C(c2c[nH][nH]c2=N)=O)=O)CC2CCCC12 85799,Cn1nnc2c1C(C(=O)N1CC3(CCN(C(C4CCCOCC4)=O)C3)C1)CCC2 85800,c1(C(=O)NC2CN(C(C(C)OCC(C)C)=O)CC2F)cc2c(nc1O)CCOC2 85801,c1(C(N2CCC(N(C(Cn3c(CCC)ncc3)=O)CC)C2)=O)cnn(CC)c1C 85802,C(=O)(C(CC(C)C)ONC(c1cnn(C(C)C)c1)=O)NC(C(=O)OC)(C)CO 85803,CCCCCCn1cc(C2CC2)nn1.C12CC(C1)N(C)C(=O)C1(CC1)C2 85804,C(=O)(CCCCCC(C)O)N1C(CNC(c2c(C)[nH][nH]c2=N)=O)CCC1 85805,C1(O)(C(C)NC(c2nc(CC)oc2)=O)CCN(C(c2ccc([N+](=O)[O-])o2)=O)CC1 85806,C1(O)(C(N2CCCC(CCCCNC(C(C)(C)OC)=O)C2)=O)CN2CCC1CC2 85807,C1(C(=O)NC2C(C)(COC)C2)CN(C(=O)C=Cc2ccoc2)CC12CC2 85808,C1(C(=O)NCC2CC(NC(CCc3c(C)noc3)=O)C2)CCN(C)CC1 85809,c1(C2(C(N(CC(C)NC(c3cc(Cl)n(C)n3)=O)C)=O)CCC2)ccc(F)c(Cl)c1 85810,C(=O)(CCC(=O)N(C1CCCN(C(=O)CSCC(F)(F)F)C1)CCF)NCC 85811,n1(C(C(=O)NCCC)C)cc(CNC(C)(CC)OCCN(CC)CC)nn1.CC 85812,c1(NC(=O)CNC(=O)NC(C2CCCNC2)CC2CCCCC2)ccc(F)cc1 85813,C1(C(N2CCC(NC(=O)C(c3cncn3C)=O)C2)=O)(OC)CCOC1 85814,c1(C(=O)NCC2C(NC(C(CCC)(C)O)=O)C2)ccc(Br)c2ccccc12 85815,C1(CCNC(C(CC)C)=O)CCN(C(C2(F)CC2(Cl)Cl)=O)CC1(F)F 85816,c1(OC)c(C(N2CC(NC(=O)C(C)Cc3ccco3)CC2(C)C)=O)occc1=O 85817,c1(N2CCCC(NC(C3CC(O)C3)=O)C2)ncnc2c(F)cccc12 85818,Cc1ncc(C(=O)NC2CCC2CNC(c2cc(O)cs2)=O)n1C(F)F 85819,N1(C(C(CC)OC)=O)CCN(CCNC(c2ccc(OCC(C)C)nc2)=O)CC1 85820,N1(C(c2c(C)snn2)=O)CCC2(CC1)CC2NC(=O)CC(C)n1cccn1 85821,N1(C(CN(CC(C)(C)C)C)=O)CCC(NC(=O)CC2CCC3CC3C2)C(F)C1 85822,C=CCC(CC)C(=O)NCC(CNC(=O)Cn1nccc1C)C(F)(F)F 85823,O=C(C1CCc2ccccc21)NC1(C2CN(C(C3CC4CC3CO4)=O)C2)CC1 85824,c1(C(=O)NC2CCC(NC(CCCCCSC)=O)C2)onc2c1CCCC2 85825,C1(NC(=O)CCCF)CC2CCC1CN2C(=O)Cn1cnnc1 85826,c1(CC(=O)NC2CCN(C(c3cn(C)nc3)=O)CC2O)c[nH]c2cccc(Cl)c12 85827,C(=O)(C1Cc2ccc(F)cc21)N1C(CNC(c2c(C)cc[nH]2)=O)CCC1 85828,c1(OCC(=O)NCC#CCNC(C2OCC(C)C2)=O)ccccc1C(C)(C)C 85829,C1(C(=O)NCC2CCC(NC(C3(CCCC)CC3)=O)C2)CCS(=O)CC1 85830,C12(CCNC(C=CSC)=O)CCC(C1)N(C(c1ccco1)=O)C2 85831,CC1(C)CCCCCC1NC(C1(F)CCN(C(=O)Cc2cccnc2)C1)=O 85832,Cc1ccc2c(c1)CCN2C(C)Cc1ccnc(N2CC(CO)CCC2C)n1 85833,c1(C(=O)NCCC2CCC(NC(C3CSC3)=O)C2)ccc(F)cc1OC(F)F 85834,C1(CC(=O)NC2C(NC(c3cccc(C)c3)=O)CCOC2)CC2(CCO1)CC2 85835,N1(C(CC(C)C(C)(C)C)=O)CCCC2(CCCN2C(C23CCC(C2)C3(C)C)=O)C1 85836,c1(CN2CCC(O)(C(=O)Nc3ccc(F)cc3Br)C2)c(F)cc(O)cc1F 85837,C1(NC(c2ncn(C3CCN(C)C3)n2)=O)CCCCN(C(=O)CCCCCF)C1 85838,C1(N(C(C(C(C)C)C)=O)C)CC2CCC(C1)N2C(c1cccn2nnnc12)=O 85839,CCCCCCCC(C)NC(=O)C(C)(C)CN(C(=O)C(CSC)OCC)C 85840,C1(NC(=O)CCc2nc(-c3nc[nH]n3)no2)C2CC1CN(C(C1CC1CF)=O)C2 85841,N1(C(CC)C)CCC(C)(CNC(c2ccc(OC)c(-c3ccc(N)nc3)c2)=O)CC1 85842,C1(C(=O)NCCC2N(C(C3(O)CC3)=O)CCC2)CCc2nnc(O)n2C1 85843,c1(C(N2CC3CCN(C(c4cnc(S)nc4)=O)CC32)=O)ccc2oc(S)nc2c1 85844,C1(C(=O)NC2(CC(N3CC4CC3(c3ncc[nH]3)C4)=O)CCC2)C2CC3C(C2)C13 85845,C1(O)(CNC(CCN(C(=O)Cn2ccnn2)CC#C)=O)CCOCC1 85846,c1(C(=O)NC2CC(NC(c3cccc(C)c3)=O)C2)coc2c1N(C)C(=O)CCC2 85847,C(C)(C)(CC(C)NC(=O)CC1CCC(NC(=O)C(F)CC2CCOC2)C1)OC 85848,C1(CC(=O)NC(C#C)C(C)OC)CCC(NC(=O)C=C2CCC2)CC1 85849,CC(CC(C)(C)O)NC(=O)C(Cc1cc[nH]n1)NC(=O)CC1CC=CC1 85850,S(=O)(=O)(c1ccc(C(C)(C)C)cc1)NC1CN(C(CC(C)C)=O)CC1C#N 85851,C1(CC(=O)NCc2cn(CC)nn2)CN(C(=O)C(C)SC(C)C)CC12CC2 85852,C(=O)(C#CC(C)(C)O)NCC1(C)CCC(NC(C(C)NC=O)=O)C1 85853,CC1C(NC(=O)CC(F)(F)Br)CCN1C(c1cnn(C)c1)=O 85854,c1(C(N2CC(CCCCNC(C=C(C)C)=O)C2)=O)coc2c1CS(=O)(=O)C2 85855,C(CCCCNC(C1(CC2CC2)CCCC1)=O)N(C(=O)CCc1nccs1)C 85856,N1(C(=O)NC)CCCC1C(=O)N(CCCN(C(=O)C(C)OCC(F)(F)F)C)C 85857,c1(C(=O)NC2CCCCN(C(c3cncc(OC)c3)=O)C2)onc2c1CCCC2 85858,c1(C(=O)NC(CC=C)CNC(=O)CC2CC2)c[nH]c2ccccc12 85859,N1(C(C(C2CCC2)OC)=O)CCC(NC(c2csc(Cl)n2)=O)CC1 85860,Cc1cccc(C)c1NC(=O)C1=CCN(C(C2COCC2C(N)=O)=O)C1 85861,CC(C)(CC(=O)N1CCCCC1CF)NC(=O)CSc1nc[nH]n1 85862,c1(C(N2CC(CC(C)NC(C3(C)CCOC3)=O)C2)=O)ccc(F)cc1F 85863,CC1(CNC(=O)CC2(C)CC2(F)Cl)CCN(C(c2cnoc2-c2ccco2)=O)C1 85864,C1(C)(CC)CCC(C(N2CC(OCC(=O)NCCc3c(C)n[nH]c3C)C2)=O)O1 85865,C(=O)(C1CCCc2nc(C)[nH]c21)N1CCCC(N2CCN(C(C=C)=O)CC2)C1 85866,c1(NCC2(C(F)(F)F)COCCN2)cc(C2CC2)nc2ccnn12 85867,N1(C(Cc2c(C)cnn2C)=O)CC(O)CCC1C(=O)NCC(F)(F)C(N)=O 85868,c1(C(N2CC3(CCCCN3C(=O)Cc3cnns3)C2)=O)ccc2ncccc2n1 85869,N1(C(c2c(N)nccn2)=O)CCN(C(c2csc(CC(F)(F)F)n2)=O)C2CC12 85870,N1(C(CC(C)OC)=O)CCOCC(C)(CNC(c2c(C)nsc2C)=O)C1 85871,CC1CC(NC(=O)CC(=O)NC2CC2)CN(C(c2cc(CCO)on2)=O)C1 85872,c1(C(=O)NC(C2CN(C(C3(CF)CC3)=O)C2)C)cccc(C2COC2)c1 85873,C1(CNC(N(CCC#CCC)C)=O)CCC(F)CC1 85874,c1(C(=O)NC2(C)CC(NC(=O)C=C3CCSCC3)C2)ccc(-c2cc[nH]n2)cc1 85875,CC1(C)CN(C(=O)Nc2csc(-c3ccc(Cl)cc3)n2)C1C1CCCO1 85876,Cc1cc(C(=O)NC2CC3CC2N(C(=O)C=C2CCC(C)C2)C3)cc(C)c1 85877,c1(C(=O)NCC(C)(C2CCC2)NC(C2CCCC2)=O)ccc2nc(O)[nH]c2n1 85878,C1(CNC(C(n2cc(C)nc2)(C)C)=O)C(C)CCCN1C(=O)CC(=O)N(C)C 85879,C(=O)(C1CCc2c[nH]nc21)OC(N1CCCC(CCCCC)CC1)=O 85880,N1(Cc2nc(C)on2)CCC2(CCCN(C(=O)CCc3ccncc3)C2)C1 85881,CCC(CC(C)C)C(=O)NCc1nocc1C(=O)N1CC(C)(O)CO1 85882,CCCC(CCCNC(=O)Cn1nnc(C)n1)NC(=O)C(C#N)C1CC1 85883,C(=O)(C1=C(F)CN(C(C2CC=C(C)CC2)=O)CC1)NCC(CC)C#N 85884,C1(C(N2CC(CC(C#C)C)C2)=O)CC(C)N1C(=O)C(C1CC1)C1CC1 85885,C(=O)(C(CO)C(C)(C)C)NCC1N(C(c2cc(C)cc(C)c2)=O)CCC1 85886,N1(CCn2cc(NCN3C(C)CCCC3)nn2)CCN(C)CC(C)C1 85887,N1(C(C2CC(C)(NC(c3cc(C(C)=O)[nH]n3)=O)C2)=O)CCC(O)(C(C)C)C1 85888,CC(CN=c1[nH]c2c(c(=NCc3cocn3)[nH]1)CSC2)Oc1ccccn1 85889,c1(C(=O)NCC(C)CN(C)C(c2coc(C(F)F)n2)=O)cnn2c1OCC(O)C2 85890,C12CCN(C(NCCSC)=NCCCO1)C2.C12(CC)COC(C)(C1)C2 85891,c1(C(=O)NCC2CC(COC)CN2C(=O)Cc2nc[nH]n2)cc(C(=O)OC)n(C)c1 85892,C1(C(N2CC(O)(CNC(Cc3cc(COC)on3)=O)C2)=O)CCCC(=O)N1C 85893,C1(CCNC(CNC=O)=O)(NC(C2CCN(CC(C)C)CC2)=O)CCOCC1 85894,C(=O)(C(C)C(C)(F)F)NCC1(F)CC(CNC(C(C)C2CCC2)=O)C1 85895,C1(c2scc(C)n2)CN(C(=O)C(n2cc(C(C)(C)C)nn2)C)CCO1 85896,N1(C(COc2cc(C)on2)=O)C2CCC1CC(F)(CNC(=O)C(O)C(F)(F)F)C2 85897,c1(C(=O)NCC(CO)NC(C(COC)N(C)C)=O)ccc(=N)[nH]c1 85898,c1(OC)nc(C(=O)NCC2CC(C)N(C(c3ccc(Cl)nn3)=O)C2)cc(O)n1 85899,C1(NC(c2n(CCC)ccc2)=O)CC2C1CCN2C(c1cc2cscc2s1)=O 85900,c1(C(=O)NC(CCCC)CNC(=O)C(C2CCC2)OCC)occc1S(C)(=O)=O 85901,C(=O)(CCC(=O)NC1(CNC(C2C(C)C2(F)F)=O)CC1)NCCC 85902,c1(C(N2CCCC(C)(O)C2)=O)cc(OC)nc(-c2cnc(OC)c(C3CC3)c2)c1 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85991,C1(NC(c2cncc(-c3ccccc3F)c2)=O)CCCC(C(F)F)CC1 85992,c1(C(=O)NC(C(C)NC(c2c(C)nn(CCO)c2)=O)C)cnc2ccncc2c1 85993,C1(NC(C2(C(C)NC(c3nn(C)cc3Cl)=O)CC2)=O)CN2CCC1(F)CC2 85994,N1(C(=O)CC2CCC3CC23)CCN(C(C2CC2(Cl)Cl)=O)C2(CC2)C1 85995,C1(CNC(C(C)(C)NC(=O)OC)=O)COCCN1C(c1cnc(OC2CC2)s1)=O 85996,CC1CN(C(C2COCC(=O)N2C)=O)c2ccc(C(F)(F)F)cc2O1 85997,C(=O)(C#CC1CCCCC1)N1CC(CCNC(c2nc(C)sc2)=O)OC(C)C1 85998,CC1CC(CNC(C2(C)C=CCCC2)=O)CCN1C(c1cc2scnc2[nH]1)=O 85999,C(=O)(CCC(C)C)NC1CC1.C12CCN(C1)CC(=O)N2C(C=C)C1CC1 86000,C(=O)(CC(O)CC(C)(C)C)N1CCCC(C(=O)NC2CC3(CCC3)C2)(CC)C1 86001,c1(CC(C(=O)N(CC(CNC(COC(C)=O)=O)O)C)C)c(C)noc1C 86002,CCN=c1[nH]c(C(=O)NCC2CCC(C)CN2C(c2nccc(Cl)c2F)=O)cs1 86003,Cc1cc2ccc(C(N3CCCC3CNC(C3CC34CCOCC4)=O)=O)cn2c1 86004,CC(C)(C)CCCCCC(=O)N1CCN(C(=O)C#CC2CCC2)CC1C(F)F 86005,O=C(C(O)C(F)(F)c1ccccc1)N1CCN(C(=O)C(Cl)=CCl)C(CC(F)F)C1 86006,C(c1cncnc1O)=CC(=O)N(CCCCNC(CC1C(C)OCC1)=O)C 86007,O=C(C(CO)C(F)(F)F)NCCC1(NC(=O)CC2(O)CCOC2)CCC1 86008,Cc1cc(Cl)cc2cc(C(N3CCC(C)C3CNC(C3(CO)CC3)=O)=O)[nH]c12 86009,C1(C(=O)NCCCCOCC)(CO)CCN(C(C2CCC(O)CC2)=O)C1 86010,c1(OCC=C)cccnc1C(=O)NCCC1CCC(NC(c2cc(C)c[nH]2)=O)C1 86011,C(CN=c1[nH]nc(O)s1)C1CCC(NC(Cc2c(CC)noc2CC)=O)C1 86012,c1(C(=O)NCc2cccc(NC(C3(CC=C)CCOC3)=O)c2)cc2sccc2[nH]1 86013,Cc1nc(-c2ncc[nH]2)sc1NCCOC1CNC(=O)C1 86014,C=C(C)CC1C(=O)N1.C1(C(C)(C)OC)CC=CC(n2cc(C(CC)OC)nn2)C1 86015,C1(CC)CN(C(=O)C=C(C)Cl)CCC1NC(C1CCS(=O)(=O)C1)=O 86016,CC1CC(C(N2CC(F)(CNC(=O)CNS(=O)(=O)C3CC3)C2)=O)Cc2nn[nH]c21 86017,N1(C(C(=O)Nc2cccc(F)c2)C2C(C)C2)CCC(N(C)C)CC1 86018,C1(NC(=O)Cc2ccc(Cl)nc2)CN(C(C2(F)CCC2)=O)CC2(CC2)C1 86019,CC1CN(C(=O)C2=CC3C=CC2C3)CC(C)N(C(=O)CC2CC(C)C2)C1 86020,C1(NC(CC(C)OC)=O)C2CC1N(C(=O)CCc1cncn1C)C2C 86021,C1(OC)CC(CNC(=O)CCCc2ccc(Cl)cc2)N(C(C2CCCC2C)=O)C1 86022,C1(NC(CC(CC=C)NC(c2cncc(C)c2)=O)=O)COC2(CCCC2)C1 86023,N1(c2ccc(S(=O)(=O)NCC3(COC)CCC3)cn2)CCCC2(CCN(C)C2)C1 86024,C1(N(C)C(c2n[nH]cc2Cl)=O)CCCN(C(C2CC23CC3)=O)CC1 86025,C1(CNC(COCC=C)=O)CN(C(C2(NC(C)=O)CCC2)=O)C(C(F)(F)F)CO1 86026,C1(NC(c2ccc(COC)[nH]2)=O)CC2CC(C1)N(C(=O)CC1NC(=O)NC1=O)C2 86027,c1(OC)ccccc1OCC(C1CC1)C1CC1.N12CCCCC1NC(=O)C2=O 86028,c1(N(C(CNC(CCOCCCOCC)=O)C)C)ccccc1 86029,N1(C(Cc2cc(C)nn2C)=O)CCCN(C(c2c(Cl)n[nH]c2C)=O)CC1 86030,N1(C(CC2CC(NC(=O)C=C(C3CC3)C3CC3)C2)=O)CCOCC(C2CC2)C1 86031,c1(C(C)(C)C)noc(CCC(=O)NCC2(NC(c3cc(C(F)F)no3)=O)CC2)n1 86032,C12(C(N(CCOCC)CC)=O)CC(CN(C(C3CCSC(C)C3)=O)C1)C2 86033,N1(C(CCCCSC)=O)CCC2CN(C(c3cnc(C)cn3)=O)CCC2C1 86034,C(=O)(CCCNC(=O)CSC1CC1)NC(C1CCC1)C 86035,c1(C(=O)NCC(C)NC(c2c(C)nccc2)=O)ccc([N+](=O)[O-])c(S(N)(=O)=O)c1 86036,N(C1CCOc2ccc(Br)cc21)C(c1c(N)cccc1)=O 86037,Cc1ccc(Cl)c(C(=O)NC(CNC(C2(C(F)F)CC2)=O)CC(C)C)c1N 86038,c1(N(C(CC2(C=C)CCOCC2)=O)CC)ccc2c(c1)ncn2C 86039,C(C)(N=c1[nH]c2c(c(=NCCNC(=O)NC3CC3)[nH]1)COC2)c1cc(C)c(F)cc1 86040,C1(NC(C2(C(=O)OCC)CCO2)=O)CC2CCC(C1)N2C(=O)C(C)CC(F)(F)F 86041,N1(C(c2c(C)cc[nH]2)=O)CCCC(C(=O)Nc2cnn(CCO)c2C(C)C)CC1 86042,C1(C2CCC2)(C(N(CC)CC2CCN(C(=O)OC(C)(C)C)C2)=O)OCCO1 86043,CC1CN(C(=O)COc2ccccc2)CCC1CN(c1nnc(C(=O)N(C)C)o1)C 86044,C1(C2CCN(C(c3[nH]cc(C)c3)=O)C2)CCCCN1C(=O)CCn1cncn1 86045,c1(C(=O)NC(CC#CC)C(=O)NCCP(C)(C)=O)cc2cc[nH]c2cn1 86046,C1(NC(C(CC)(C)F)=O)COC2(C1)CN(C(=O)C(C)(C)C(=O)OC(C)(C)C)C2 86047,C1(C(=O)NCc2ncc(C(N3CC(OC)(CO)C3)=O)cn2)CCOCC1(C)C 86048,N1(C(CCC2(C)CC2)=O)CCC2(C1)CN(C(=O)CC13COCC(C1)C3)CCO2 86049,c1(OC)ccc(F)c(C(C(=O)NC(CCO)C(F)F)N(CCC#N)C)n1 86050,C1(CC(=O)NC2CC(CNC(C3C(C)C3)=O)C2)CC2(CCC2)CCO1 86051,Cc1cc(C(N2CC(O)(CNC(=O)CC(c3ccccc3)N(C)C)C2)=O)n[nH]1 86052,N1(C(C2(C)CC2)=O)CC2(CCN(C(C3(c4ccncc4)CCCCC3)=O)CC2)C1 86053,c1(OC)ccc(C(N2CCCC2CC(N2CCc3sccc3C2)=O)SC)c(F)c1F 86054,C1(CCNC(c2n(C=C)nnc2)=O)CCCN(C(=O)C(F)CC2CCOC2)CC1 86055,C1(NC(c2cc(OC)ncc2)=O)(CNC(c2ccc(Cl)cc2)=O)CCCCC1C 86056,CC1(C)C(CC(=O)NC2(C)CCN(C(c3ccccn3)=O)C2)C1(C)C 86057,N1(C(CC(CC)C2CCC2)=O)C2CC=C(C(=O)NCC3C(C)C3(F)F)C1CC2 86058,N1(C(C(C(C)C)CO)=O)CC2(CCC2)CC1CNC(=O)COC1(C)CCCC1 86059,c1(C(N2C(CN(C(=O)CCn3ccccc3=O)C)CCC2)=O)cncc(O)c1Cl 86060,C12(CNC(C3(CC=C)CC3)=O)CCC1CN(C(=O)C=Cc1c(Cl)cccc1Cl)C2 86061,N(C(=NCC1CCC1)N1CCC(C)(C(=O)NC)C1)CC1OCCN(CC)C1 86062,C1(F)(C(=O)NCc2occ(C(=O)NC(CCC=C)C)n2)CCCCC1 86063,c1(CNC(C2C(NC(C=C(COC)C)=O)CCO2)=O)cccc(C#N)n1 86064,CC(CC(=O)NC1CN(C(=O)NC2CCC2c2nc(S)n[nH]2)C1)c1ccncc1 86065,CCCCCCCCCC(=O)N1CC(C)(NC(=O)C(c2ccccn2)O)C1 86066,C1(CN2CC(C(OC)OC)C2)CCCCC1SCCCN=[N+]=[N-] 86067,C1(CNC(c2ccccn2)=O)CCN(C(c2cnnc(O)c2)=O)CC1O 86068,Cc1cc(C)c2cc(C(N3CC(NC(c4c(C)[nH][nH]c4=N)=O)C3)=O)sc2n1 86069,C(=O)(C(C)(CC)C(N)=O)N1CCC(N(C(C(C)OCC#C)=O)CC(C)C)CC1 86070,N1(C(c2c(C)nc(C)s2)=O)CC(NC(=O)COCC(F)F)C(C2CC2)C1 86071,c1(N(C(=O)C(C)=CC2CC2)CCOC(CC)C)ccc(F)cc1C#N 86072,C1(NC(c2nc(C(C)C)sc2)=O)CCCC1(C)NC(=O)C(C)C1CC1 86073,c1(C(=O)NCC2CC(O)(CNC(C3(COC)C=CCC3)=O)C2)ccc(C)nc1C 86074,c1(CNC(=O)NCC2(c3ccc(OC)cc3)CC2)c(Cl)nc(C)nc1Cl 86075,C1(N(C(C2C(c3ccn(C)n3)C2)=O)CCO)CCN(C(c2cccs2)=O)CC1 86076,n1(CC(N2C(CCNC(C(C)(C)F)=O)CCC2)=O)cnc(C#N)n1 86077,N1(C(c2n(C(CC)C)ncc2)=O)CCCC(N(C(C2CCC(=O)O2)=O)CC)C1 86078,N1(C(C2C(C)C2C)=O)CCN(C(=O)C(Cl)=CCl)CCC1C 86079,C1(NC(c2cc(C)n(C)n2)=O)CN(C(=O)C(Cl)=CCl)C2(CCC2)C1 86080,N1(C(C(C)SC)=O)CCN(C2CCCN(C(c3ccc(CO)o3)=O)C2)C(=O)C1 86081,CC1(CNC(c2cnoc2C2CC2)=O)CCN(C(c2ccccc2Br)=O)C1 86082,C(CCCC#N)(c1nnnn1C1CC1)NC(c1ccc(N2CCCCC2)cc1)C 86083,c1(C(N(CCn2cc(CCC(CC)O)nn2)CC)=O)ccccc1C(C)(C)C 86084,N1(C(Cc2c(COC)cccc2)=O)CCN(C(=O)C2=NOCC2)C2CC12 86085,C12(CC(=O)NCCCC(C)O)CCC1CN(C(=O)COc1ccn(C)n1)C2 86086,CCCC(CNC(C1CSCCN1C(c1ccccc1C)=O)=O)CCO 86087,c1(C(=O)NC(CC)CNC(=O)CC(F)(F)F)sc2ccccc2c1COC 86088,C=CCC(CNC(=O)COC1CC1(F)F)C(=O)N(C)Cc1nc[nH]n1 86089,N1(C(C(CC)N(C)C)=O)CC(NC(c2ccnc(OC)n2)=O)C2CCCCC12 86090,N1(C(c2c(C)cco2)=O)CCC(N=[N+]=[N-])(C(=O)N(C)CC2CC2(C)C)C1 86091,c1(C(N2CCC(N(C(=O)C(C)CC)CC)C2)=O)cc(=O)n(C)cc1Br 86092,C12(CNC(C3(CC=C)CCC3)=O)CCCC1N(c1ncncc1C#N)CCC2 86093,CCN=C(NCCCC(C)(F)F)NCC(C1CCCC1(C)C)(C)O 86094,Cc1ccc(C(=O)NC(CC(=O)NCc2c(F)cncc2F)C(C)C)c(C)n1 86095,C1(CNC(C=CCC)=O)CCC2(CO1)CC(NC(c1cc(O)ccc1C)=O)C2 86096,N1(c2c(C)c(NC3CCC4(CC4)C3)ncn2)CC2CC3CC2C1C3 86097,c1(C(=O)NCC2(OC)CN(C(=O)Cc3c(C)noc3C)C2)cc[nH]c(=N)n1 86098,c1(OC)ccc(C(N)=O)cc1C(=O)NCC(C)(C)NC(=O)C=CCO 86099,Cc1cc(C(=O)NCC(C2CCCCC2)NC(=O)CC23CC(C2)C3)ccc1[N+](=O)[O-] 86100,c1(OC)ccc(C=CC(=O)NC(C)CC2CN(C(=O)C(C)C(C)(C)C)C2)cc1F 86101,c1(C(N2CCCCC(NC(C3C(C)C3)=O)C2)=O)cccnc1S(=O)(=O)C(F)(F)F 86102,c1(CC)ncccc1C(=O)N(C1CCC(NC(c2cccnc2)=O)C1)C 86103,c1(SC)ncc(C(=O)NC2CC(NC(C3(n4ccnn4)CC3)=O)C2)c(O)n1 86104,c1(C(=O)NC(C(=O)NC2CC(C(C)C)OC2)CC2CC2)ccn2ccccc12 86105,c1(C(=O)NCCNC(c2c(C)ccc(Br)c2F)=O)coc2c(C)cccc12 86106,C=C(C)CC(C(=O)NCC(C)(O)CC)NC(c1cc(OC)sn1)=O 86107,CC1CC(NC(c2cccc(=O)o2)=O)CN1C(=O)Cc1ccccc1Br 86108,N1(C(CCCOCCOCC)=O)CC(NC(c2c(N)cccc2Cl)=O)CC(O)C1 86109,Cc1ccc2sc(N(C)CC3CN(C(=O)C(C)(O)C4CC4)C3)nc2c1 86110,c1(C(N2CC3C(CNC(CC(C)(C)C4CC4)=O)(C3)C2)=O)cc(O)ccc1Cl 86111,S(=O)(=O)(c1cnc(NCC23CCCC2OCC3)c(Cl)c1)N(C)CC1(CSC)CC1 86112,c1(C(=O)NC2CCN(C(CCC(=O)NCC)=O)CC2F)cccn2c(C)nnc12 86113,c1(C(N2CC3(C2)CN(C(C2CCNC2=O)=O)C3)=O)c[nH]c(=O)c2ccncc12 86114,CC(F)(F)CCNC(=O)CNCC1CCN(C(N2CCCC2)=O)C1 86115,CC1(NC(c2coc(Br)n2)=O)CCN(C(=O)CCCn2ccccc2=O)C1 86116,N1(C(CCC(=O)OCC)=O)CCC(CO)C(NC(=O)CCCn2ccnn2)C1 86117,N1CC2CC3CC2C1C3NC(=O)C(F)C1CCC1.O=CCCCc1ccncc1 86118,N1(C(c2c(C(C)C)cccc2)=O)CC(NC(c2cc(F)ccc2I)=O)C(C#N)C1 86119,N(C(=NCCC1CS(=O)(=O)C1)NCc1noc(C2CC2)n1)CC1(C)CCC1 86120,c1(C(=O)NC(CNC(c2c(OCC)oc(C)n2)=O)C2CCC2)cc(C)cc(C)c1 86121,N1(C(C(C=C)(C)O)=O)CC2CC(NC(c3ccc(CC)c(Br)c3)=O)C1C2 86122,C1(C(=O)O)CCCC(CNC(c2occc2-c2ccccc2)=O)C1 86123,c1(N2CCN(C(C)C)C(=O)C2)nc(N2CC=CC(C)C2)c2ccsc2n1 86124,N(C(=NCCF)NCc1cc(Cl)ccc1Br)CCC1CCN(C)CC1 86125,c1(C(C)(C)C)ncncc1C(=O)NCCC1(O)CN(C(=O)C(F)(F)CC2CC2)C1 86126,CC(C)(CCCNC(=O)CC(F)(F)F)C(=O)NCC1CCC(F)C1 86127,c1(OC)cc(C(=O)NC2CC3CC(NC(=O)C(C)SC)C2C3)cc(Br)c1 86128,c1(CNc2cccc(CN3CC4C(C(C)=O)C4C3)c2)nccc(C#N)n1 86129,N1(C(=O)NCC2(C)COC2)CCC(O)(C(F)(F)C(N)=O)C1 86130,CN(Cc1c[nH]c2nccc(Cl)c12)N1CC=C(C(C)(C)C(=O)N2CCCC2)CC1 86131,N1(C(C2C(C(C)(C)C)CC2)=O)CC2CC2(NC(C2CC(OC(F)F)C2)=O)C1 86132,c1(C(N2C(C)C(=O)NCC2)C(=O)NCc2ccco2)cc2ccccn2n1 86133,N(C(=NCCCC(C)(F)F)NC(C)C1CC1)C(c1cccnc1)C 86134,C1(CC(N2CCCC(CCC#C)C2)=O)CN(C(c2c(C)csc2C)=O)CCC1C 86135,c1(OCCc2nc(CC(CC)C)nn2-c2c(F)cccc2Cl)cc(CO)ccc1C 86136,C(CCCCOc1cccc(C)c1)(c1n(C(CC)(C)C)nnn1)COC 86137,FC1(F)CCC2C(CCCN2c2nc(-c3ccncc3)nc3ccccc23)C1 86138,c1(C(C(=O)OC)N(C(=O)CC(N)CC2CCCC2)C)cccc2ccsc12 86139,C(=O)(C1=COc2ccccc2O1)N(C)CC1C2CN(C(=O)C3=CCCC3)CC12 86140,N1(C(CCC2C(C)(C)C2)=O)CCC(CN(C(c2ccc(F)cc2)=O)C2CC2)CC1 86141,c1(C(N2CC(CCNC(C3C(C)C3C)=O)C(C)C2)=O)cc2c(cn1)OCCO2 86142,C=C(Br)CCC(=O)NC1CCC(CNC(c2ccc(C(F)F)nc2)=O)C1 86143,Cc1c(O)c(=O)ccn1CC(N1CC2CC(NC(=O)C(F)C3CC3)C1C2)=O 86144,c1(C(=O)NC2(C)CC(NC(C3(Cl)C(C(C)=O)C3)=O)C2)c(C(F)F)cnn1C 86145,Cn1c(O)ncc(C(=O)NCC2CC3(CO2)CN(C(C2CC(C)(C)C2)=O)C3)c1=O 86146,C(CC(C(C)(C)C)NC(=O)C(C)OC1CCOC1)N(C(c1c(C)noc1N)=O)C 86147,CC(C)(CC(=O)N1CC(NC(C2CCCCN2N=O)=O)CC(F)C1)CC(F)F 86148,C1(NC(C(C)O)=O)CC2(C1)CC(NC(c1c[nH]cc(F)c1=O)=O)C2 86149,c1(C(N(C(C)CNC(C2CCCN2c2ncccn2)=O)C)=O)ccnnc1S 86150,C1(NC(C(CCC)F)=O)Cc2ccccc2C1NC(=O)CC1C=CCC1 86151,CC(Cc1ccccn1)N=c1[nH]c(=NCCN2CCC(O)C2)[nH]c2cccnc12 86152,N1(Cc2cnc(OC)nc2)CCN(C)C(C(N2CC(O)CC2C(=O)O)=O)C1 86153,c1(C(N2CC(NC(CCC(C)O)=O)C(C)CC2)=O)ncnc2sccc12 86154,c1(C(=O)NC2C(NC(Cn3ncn(C)c3=O)=O)CCC2)c(N)cccc1[N+](=O)[O-] 86155,C(C1C(=O)N(C)CC(=O)NCc2cn1nn2)OC.N1(CC(F)F)CCCC1 86156,c12ccc3nc(O)n(c3c1)C(C)C(C)C(=O)N2.C1(CC)CN(C(C)=O)CC(CC)O1 86157,C1(OC(CCC(C)(C)OC)=O)CCC2CN(C(c3c(OC)noc3CO)=O)CC2C1 86158,c1(C(N2CCC(N(C(=O)C(C)(C)C#N)C)C2)=O)ccc(Cl)cc1Cl 86159,N1(C(c2occ(CC)n2)=O)CC(c2nc(COC3CCCC(C)C3)no2)C(C)(C)C1 86160,C1(C(N2CC(COCC)(NC(=O)Cc3ccccc3)C2)=O)CC2CCC(C1)C2 86161,N1(C(c2cnc(C)o2)=O)CC=CCC1C(=O)NC(C)C1CC1 86162,c1(CC(=O)N(C)CC2CCCN2C(=O)CN2CCOC2=O)c(F)cccc1Cl 86163,c1(OC)ccc(C(N2CCC(O)(CNC(=O)CCC3CC(F)(F)C3)C2)=O)nc1 86164,C(=O)(C1=CCCOCC1)N1CCC(COC)(NC(c2cnc(C(C)(C)C)o2)=O)C1 86165,C1(CC(=O)NCC2N(CC)CCC2)N(C(c2cccnn2)=O)CCC1(C)C 86166,C(=O)(C1=NNC(=O)CC1)NC(CC)(CNC(=O)Cc1ccccc1CC#N)CC 86167,N1(C(c2cc(CN(C)C)on2)=O)CCC2CN(C(=O)Cn3ccnn3)CCC2C1 86168,N1(C(c2c(CC)n(CC)nn2)=O)CC(O)(C2(CNC(C3CC(C)CO3)=O)CC2)C1 86169,c1(CC(N2C(CN(C(CN(CC)CC)=O)CC)COCC2)=O)cc(C)ccc1O 86170,CC(C)C(C(=O)NCCC(C(C)C)NC(=O)C(C)N(C)C)NC(=O)OC(C)(C)C 86171,C1(C(=O)NC(CN(C(c2cc(C)nc(N(C)C)n2)=O)C)C)CCc2nnnn2C1 86172,c1(C(N(C2CCN(C(=O)C(C#N)CC)C2)CC#C)=O)cn(C)nc1CC 86173,C1(C)(CN2CCC(C)(CC)C2)CCCN(CC2CCCCCC2)C1 86174,C1(NC(C(C)CN2CCOCC2)=O)CCC2CN(C(=O)CC3CSC3)CC2C1 86175,Cc1cccc(C)c1C(C(=O)O)NCc1cc(Br)sn1 86176,N1(C(CN(C)CC)=O)CCC2CCCC(C1)N2C(c1cc2c(nn1)CCCO2)=O 86177,c1(C(=O)NCC(C)CN(C)C(c2cc3sccc3n2C)=O)cc(F)c(F)cc1F 86178,N1(C(C(COC)OC)=O)CC(C(=O)N(CCCO)C(C)C)C(C)C1 86179,C1(C(=O)NCC2C(NC(Cc3ccn(CC)n3)=O)C2)C(C)(C)C1(C)C 86180,N1(C(CCCCC(C)C)=O)CC=C(C(C)(C)C(=O)NCC2CCC(F)C2)C1 86181,c1(C(=O)OC)cc2n(n1)CCCC2NC(c1nc(-c2ccccc2)sc1N)=O 86182,c1(CC(N2C(CNC(C=C(CC)C)=O)CC(OC)C2)=O)ccc(F)cc1[N+](=O)[O-] 86183,C12(CNC(C(CCC)C#N)=O)CN(C(c3c[nH]nc3C3CC3)=O)CC1CCO2 86184,Cc1nc2cncc(C(N3CC4(CCN(C(c5c[nH]cc5Br)=O)C4)C3)=O)c2[nH]1 86185,CC(C)CCCCCC(=O)NCC(C)(C)C#CC(=O)NC(C)C(O)C(F)F 86186,C1(NC(CC2(OC)CCC2)=O)COCCC1NC(C1CCC(C(C)C)CC1)=O 86187,c1(C(=O)NC(CC(C)NC(C2C(C)C2)=O)C)n[nH]c2c1CC(C)CC2 86188,C(CNC(=O)CCC1CCC1)(C(C)(C)C)NC(c1cc(CCCCC)[nH]n1)=O 86189,c1(-c2n(C)nc(CO)n2)cc2c(s1)C(C)(C)CCC2 86190,C=CC(C)CC(=O)NCCC1CC(NC(=O)CCc2ccccc2O)C1 86191,c1(OC)cc(C(=O)OCCCCCNC(=N)N)ccc1F 86192,Cc1cc(C(=O)NCC2(NC(C3CCN(C)S3(=O)=O)=O)CCCCC2)ncc1N 86193,N1(C(C)C)CC(NC(C2CC(CCNC(=O)C(C)SCC3CC3)C2)=O)CC1=O 86194,N1(C(c2c(C)n[nH]c2C)=O)CCC2(CCNC2)C1 86195,c1(CCCC)cc2c(C)cc(=O)oc2cc1N(C(c1ccc(N)cc1)=O)CC 86196,c1(C(=O)NC(CC)(C)CNC(=O)C#CC(=O)N(C)C)n[nH]c2ccc(O)cc12 86197,N1(C(C(COC)OC)=O)CCOCC(NC(=O)CCCCCO)C1 86198,C1(O)(CC(=O)NCCCCNC(CSc2nc(C)[nH]n2)=O)CCCOC1 86199,Cc1ccc2cc(C(=O)N(C)CCN(C(=O)C=CC(F)F)C)nn2c1 86200,CC1CC(C(N2CCOC(CCF)C2)=O)N(C(=O)CCC2(C#N)CCC2)C1 86201,C=CC1(CC(=O)NCC(C)OC(F)F)CN(C(c2c[nH]ccc2=O)=O)C1 86202,c1(N2CCCCC(NC(CC(=C)C)=O)C2)nccc(S(C)(=O)=O)n1 86203,c1(C(N2CCCC(CCNC(C=C(C)C)=O)C2)=O)cccc2[nH]c(=N)oc12 86204,N12CCCC(C1)N(C)C(CC1C=CCC1)C2=O.c1(C2(NCCO)CC2)ccccc1 86205,C1(CNC(CCC=C)=O)CCN(C(=O)CCc2nc3ccccc3o2)C12CCC2 86206,C(=O)(CC(C)(C)C=C)NCC(=C)CCNC(=O)CC(CC)c1ccccc1 86207,N1(C(C(C(=O)NC)(C)C)=O)CCc2sc(CNC(=O)CSS(C)(=O)=O)nc2C1 86208,C1(CCC(=O)N(CC)Cc2cnn(C)c2)CCCCN1C(C1C=CCCC1)=O 86209,c1(C(=O)OCC)nn(C)[nH]c1=NC(=O)c1noc(C)n1 86210,N1(CC)C(=O)CCC1CC(=O)NC(C)(CNC(c1c(C)ncn1O)=O)C1CC1 86211,CC1(C)NC(=O)CCC1C(=O)N(C(=O)CNc1ncccn1)CC1CC(F)(F)CS1 86212,C1(NC(c2c(C)snc2)=O)CCC12CN(C(C1CCN(C3CC3)C1=O)=O)C2 86213,C=CC(O)C(=O)NC(C)(CNC(c1cc(OC)ns1)=O)CO 86214,O=C(CCCCCCc1ccccc1)NCC(C1CC1)NC(=O)C#CC1CCOC1 86215,N1(C(CCCC#CC)=O)C(C(=O)N(CC(C)C#N)C2CC2)C2CC(O)C1C2 86216,c1(C(N2C(C)C(NC(=O)Cn3cccnc3=O)CC2)=O)cccc(S(N)(=O)=O)c1 86217,C1(C(N(CCN(C(c2cc(C(C)(C)C)on2)=O)CC)CC)=O)CCc2nnnn2C1 86218,CC1CN(C(=O)CCn2ccnc2)CC1CNC(=O)CN1CC(=O)NC1=O 86219,c1(C(N2C(C)C(C)N(C(C3CC(=O)CCO3)=O)CC2)=O)cn2cc(Cl)cnc2n1 86220,c1(C(=O)NCC2CC(OC)CN2C(=O)CSCCN(C)C)cc(C)n(C)c1C 86221,c1(-n2cc(C3(OC)CCOC3)nn2)nc2c(C(N)=O)cccn2n1 86222,C(=O)(CCCC(=O)OC(C)(C)C)NC(CNC(C1CN(C(C)C)C1)=O)(C)CO 86223,C1(CNC(CC(C)=C(C)C)=O)CC(F)(F)CN1C(=O)C=Cc1cncn1C 86224,CCC(F)(F)CC(=O)N(C)CC1CCCC(NC(=O)CCc2ccoc2)C1 86225,c1(C(N2C3CCC(NC(C=CC=CCC)=O)C(C3)C2)=O)cnn2ccc(O)nc12 86226,c1(NC(C2CC3CC3N2C(=O)CC2CCCCO2)=O)ncc(Br)nc1Br 86227,Cc1cc(=NCCOc2ncccn2)[nH]c(NC2CCC3(C(C)C)CC23)n1 86228,c1(C(=O)OC)cc(NC(c2nc(C(c3ccccc3F)C)no2)C)ncc1OC 86229,c1(N2CCC(N(C(=O)Cc3cncn3C)CCC)CC2)ccc(C#N)nc1 86230,C1(CC(=O)NC(C2CCCN2C(c2c[nH]nc2C(F)F)=O)(C)C)CCC2CC2C1 86231,C1(NC(c2cc[nH]n2)=O)CCCC(NC(C23CSC(C2)C3)=O)C1 86232,N1(C(CC)C(=O)Sc2nc(CN)ncc2C(F)(F)F)CCc2ccccc21 86233,c1(NC(=O)NC2CC(c3ccc(Cl)cc3)C2)ccc2nc(O)sc2c1 86234,CC1NC(=O)C(C)N(CC(c2nccn2-c2ccccc2)=O)C1C 86235,c1(NC(C)CCCCN(C(=O)OC(C)(C)C)C2CC2)snc(C(F)(F)F)c1C#N 86236,N1(C(C(C)Cn2ccnc2)=O)CCCCC(C(=O)NCC(C)(C)C2CCCO2)C1 86237,C#CC1CN(C(C2COC(=O)N2)=O)CCN1C(=O)CCCCC(=O)OCC 86238,N1(C(c2c(C(=O)OC)nccn2)=O)CCCC(CNC(=O)CN2CC=CC2)CC1 86239,Cn1cc2ccc(C(=O)NC3CC3C(=O)Nc3nccc(I)n3)cc2n1 86240,C1(c2n(C)cnc2)CN(C(=O)C=CC(F)(F)F)CC1NC(C1(C)CNC(=O)C1)=O 86241,c1(C(N2CCC(OC)C2)C(=O)NCCSC2CCOCC2)ncc(C)cc1C 86242,Cc1noc(CCC(=O)NC(Cc2nnc(C)o2)C(=O)O)n1 86243,CC(F)(F)C(C)(C)CNC(=O)NCc1c(C2CC2)cccc1F 86244,C(C(C(=O)N(CC(C)(C)CNC(=O)C(C)OC)C)c1ccccc1)OCC=C 86245,C12(NC(CCCSC)=O)CCCC1N(C(c1ccnc(F)c1N)=O)CC2 86246,C(CCCCC(=O)NC1(CNC(=O)Cc2cncnc2O)CC1)SC 86247,C(=O)(C1CCCc2scnc21)NCC(CC)(CC)Nc1nc(Cl)nc2c1CCC2 86248,N1(C(CC2C(C(=O)OC)CC2)=O)CCC(c2n[nH]cc2COC=O)C1.C(C)(C)(C)O 86249,CCCC(C(O)C(=O)N1C2COCC1C2)NC(C12CCCC1CCC2)=O 86250,N1(C(CC2(N(C)C)CCC2)=O)CCOC(CC(=O)NCC2CCCC2(C)C)C1 86251,C1(C(C)NC(=O)Cn2ccc(C)c2)CN(C(=O)CC2CCC2)CCO1 86252,Cc1cc(CNC(C2CC(C)CN(C(c3c[nH][nH]c3=N)=O)C2)=O)cc(F)c1 86253,N1(CC)C(C)CN(Cc2c(OC)nsc2OC(C)C)CC1(C)C 86254,CCCC(C)(CC)C(=O)N1CC(C(=O)NC(CCO)CC(C)C)C(C2CC2)C1 86255,N1(C(c2cc(Br)ncc2Cl)=O)CCn2c(cc3cc(Cl)ccc23)C1 86256,c1(C(N2C(CNC(=O)CCC(C)C)CC(OC)C2)=O)nccc2c(F)cccc12 86257,C1(C2CCCCC2)(NCCOc2c(C(N(C3CCNCC3)C)=O)nccc2)CCCCC1 86258,c1(CN2CCC(C)C(C)(C)C2)ccc2cc(F)cc(Br)c2n1 86259,C1(NC(C2CCN(C(CC3CCCN(C)C3)=O)CC2)=O)CC2CCCC2C1 86260,N1(C(C(CCCCC)F)=O)CCOC2CCN(C)CC12 86261,Cc1nn(C)c2sc(C(=O)NC3CC(C)N(C(=O)CC(C)(C)F)C3)cc12 86262,Cc1c(C(=O)NC(CNC(c2ccsn2)=O)CO)cnc2ncnn12 86263,C1(NC(C=CC(=O)N(C)C)=O)C=CC(C(=O)NCC(F)Br)C1 86264,c1(C(N2CC(NC(C(C(C)C)n3ccc(C)c3)=O)C2)=O)cnn2c1OCCC2 86265,c1(C(N2CC3CN(C(c4cscc4Br)=O)C3C2)=O)cc2n(n1)CCC2 86266,C12(CNC(C3(SCC)CC3)=O)CCC1CN(C(=O)Cc1ncsc1Cl)C2 86267,CC(C)(CO)C(=O)NC1CC1NC(c1ncoc1C(C)(C)C)=O 86268,C=C(Cl)CC(C(=O)NC1CCC(=O)NC1)NC(=O)C(F)CCC 86269,Cc1c(C(=O)NC(C)C(CO)NC(C2(C)CC(C)C2)=O)cnn1C(C)C 86270,C1(NC(c2c(C)n(CCO)nc2)=O)CC2(CCN(c3ccnc(C#N)n3)C2)C1 86271,Cc1nc(NCCc2nnc3n2CCS3)cc(=NC(C)c2cc[nH]n2)[nH]1 86272,Cc1cccc(C(O)C(N2CC(C)(NC(c3cncc(N(C)C)c3)=O)C2)=O)c1 86273,N1(C(C(C(C)(C)C)O)=O)CCN(C(=O)CC2=NNC(=O)C2)C2COCC12 86274,N1(C(C2N(CC)CCC2)=O)C2CCC1CC(C(=O)NCC(F)C1CCC1)C2 86275,c1(C(N(CCCCCNC(=O)COC2(C)CCC2)C)=O)c[nH]nc1[N+](=O)[O-] 86276,C12(C(N(C(C)C)C)=O)CC1CN(C(=O)CN1CCN(S(C)(=O)=O)CC1)C2 86277,Cc1nncn1NC(=O)CCC1CCCN(C(=O)CC2(C)OCCO2)C1 86278,CC1CCN(C(c2c(F)cccc2Cl)=O)CCC1N1CCN(C2CC2)CC1 86279,c1(C(=O)OC)cc(SC)c(C)cc1NC(=O)COc1cc(C)c(C)cc1 86280,C1(C(=O)NCC(C)CNC(c2ccncn2)=O)C(C)CCN1C(=O)OC(C)(C)C 86281,C(=O)(CC1=CCN(C(=O)CC2CCOC2(C)C)CC1)NCC 86282,N1(C(c2cc(CC)c(Cl)cc2)C(=O)NC(C)C)C2C=CCC1CCC2 86283,c1(C(=O)NCc2cn(CC(=O)NC(C3CC34CC(O)C4)=O)nn2)ccnc(F)c1 86284,c1(C(N2CCC(CCC(=O)N(C(C#C)C)CCCC)C2)=O)cc(C#C)ccn1 86285,c1(NCC2C(C)CCC2)[nH]c(=NCc2ccc(=N)[nH]c2)nc2scnc12 86286,CCCC(C(O)C(=O)NC1CCN(C(C)(C)C)C1)NC(=O)CC(C)(C)COCC 86287,CN1CCC(CC(=O)Nc2cccc(CNC3CCN(S(C)(=O)=O)CC3)c2)C1=O 86288,c1(C(=O)NC(CNC(c2cnn(C(CC)C)c2C)=O)C)cncc2ccsc12 86289,O=C1CS(=O)(=O)CC(C(=O)NC2CC2NC(=O)C(C2CC(F)(F)C2)O)N1 86290,c1(C(C)NC(C2(CNC(=O)C(c3cnn(C)c3)=O)CCCC2)=O)ccc(Cl)nc1 86291,N1(C(C(CCC)OCC)=O)CC2(C(=O)NCC(CO)C3CCC3)CC1CO2 86292,Cc1cnc(C)c(NC(C2C=CCN2C(=O)Cc2ccccc2Cl)=O)n1 86293,c1(C(=O)NCCOCCCC#C)ccnc(CNC(C2(C)CC3CC3C2)=O)c1 86294,N1(C(C(C)C)=O)CC(CNC(C2NC(=O)CC2C(F)(F)F)=O)C(C)C1 86295,C(=O)(C1=CCCN(Cc2cccc(F)c2Br)C1)Nc1ccc(OC)nc1OC 86296,C1(C)(C(=O)NCCN(C(=O)CCC2CC2(Cl)Cl)CC(C)O)CCCCC1 86297,C1(NC(c2cn(CCC)nc2)=O)C(C)CCN(C(c2cnnc(C)c2)=O)C1C 86298,c1(C(N2C(CNC(c3nc(C4CC4)cs3)=O)CC(O)C2)=O)cc(F)ccc1Cl 86299,C(C(C(=O)NCC(C)(C1CC1)NC(c1cncnc1O)=O)C(C)(C)C)OCC=C 86300,C(=O)(C1=CCCCC1)N(C)CC1COCCN1C(c1nccnc1O)=O 86301,N1(C(C)C)CCCCC1C(=O)NC1(C)CN(C(C2(S(C)(=O)=O)CC2)=O)C1 86302,CC(CN(C)C)CCC(=O)NCc1ccc(C(=O)NCC2C3CCCC23)o1 86303,N1(C(C2(C)CN(C(=O)CCC(N)=O)C2)=O)CCCC(C(=O)NC)C1 86304,C(=O)(C1CCCc2scnc21)NCC(CC)NC(C1CCc2nncn2C1)=O 86305,c1(C(=O)N(C(C2CCNC2)(C)C)Cc2ncccn2)ccc(C#N)c(F)c1 86306,C1(C(N(CC#C)CC=C)=O)CCCN(C(=O)CCc2ccoc2)C1C 86307,N1(C(CCC)=O)CCN(C(c2cc(Cl)cn2CCOC)=O)CC(C)(C)C1 86308,Cc1noc(C)c1-c1cn(C2CCC(C(=O)N(C(C)C)C(C)C)C2)nn1 86309,N1(CC(=O)NCC2(C(=O)NCC3(SC)CCC3)CC2)CCNC(=O)C1 86310,c1(NC(COCC(=O)OC)=O)cccc(NC(=O)C(O)Cc2cnc[nH]2)c1 86311,CC1(CCCCNC(c2ccccc2Sc2ccc(Cl)c(Br)c2)=O)NC(=O)NC1=O 86312,Cc1c(C(=O)NCCCCN(C)C(c2cncc(C(C)C)c2)=O)ncn1C 86313,c1(C(=O)NCCNC(C2CCCOC2)=O)ccc2c(Br)cccc2c1 86314,C1(C(=O)NC2CN(C3CN(C(CC4CC(=C)C4)=O)C3)C(=O)C2)CCCC1C1CC1 86315,c1(C(=O)NCC(C)NC(=O)CC23COC(CF)(C2)C3)nc(C2CC2)sc1Br 86316,CCC(CNC(C1CN(C(N)=O)C1)=O)(CC)NC(C1CCNC1=O)=O 86317,C1(CNC(C2(COCC)CC2)=O)CC(C)(C)CN1C(c1ccc(CO)cc1)=O 86318,c1(NC(N2CC(C)OC(C3CC3)C2)=O)cc2ncccc2[nH]1 86319,c1(-c2ccn(CCC(F)(F)F)n2)nc(-c2ccccn2)nn1C1CC2CCC1C2 86320,c1(C(N2CCOC(CC)C2)C(=O)NCCC)cnc2cnccn12 86321,c1(C(=O)NC(C)CNC(c2ccncc2O)=O)cc2nccc(C(F)(F)F)n2n1 86322,C1(NC(C(C)OCC=C)=O)CCS(=O)(=O)C12CN(C(=O)CSCC)C2 86323,N1(C(c2cnc(COC)o2)C(=O)NC(C)C)CCc2c3cc-3cc21.C1(OC)CC1 86324,C(=O)(CCS(=O)(=O)CC(C)C)N(CCCNC(C1ON=C(C)C1)=O)C1CC1 86325,Cc1cc(C(N2CCOCC(NC(c3ncc(Cl)s3)=O)C2)=O)c(N)c(Cl)c1 86326,N1(C(C2(C=C)CCC2)=O)CCCC(N2CCN(C(=O)C(F)C3CCOC3)CC2)C1 86327,C1(CCCNC(C(CO)OC)=O)CCN(C(C2(C)CC3CC3C2)=O)CC1 86328,C(=O)(C1=CC(O)CCC1)NCC1CC(OC)CN1C(c1ccsc1Cl)=O 86329,CC(C)CCCCCC(=O)NC(C(N1CCC1(CO)CO)=O)C1CC1 86330,c1(C(N(C(c2ccc(Br)cn2)C)C)=O)cc2c(C(F)(F)F)cc(N)cc2s1 86331,c1(CC)sc(C(=O)NCC(C)(C2CC2)NC(=O)C(C2CCC(=O)N2)C)cc1C 86332,N1(OC)CCC(C23CC(C2)C3)C1.c1(-n2c3nc(n2)OC3C)ccc(C)c(F)c1 86333,CC1Cc2sc(C(=O)NCC3(F)CN(C(c4ccncc4O)=O)C3)cc2C(C)C1 86334,C1(C(C(=O)NCCCOC)N(CC(CC)(C)OC)C)CCC(C)(C)C1 86335,c1(C(N2CCC2CNC(CN(C(=O)CC2CCCN2C)C)=O)=O)ccncc1 86336,N1(C(C2(C(=O)OCC)CC2)=O)CCN(C(C2CC3CC(OCC)CC23)=O)CC1C 86337,c1(CC(=O)NC2CC(CCNC(C3(C)CCCS3)=O)C2)ccc(C#N)c(F)c1 86338,C1(OCC#C)CCN(C(=O)CC2CN(C(c3cnc(Cl)[nH]3)=O)CCO2)CC1 86339,C1(c2cn(C3CN(C(c4c(OC)c[nH]n4)=O)C3)nn2)C2CCCCC12 86340,c1(C(=O)NCCC2CCN(C(C(C)=CC3CC3)=O)CC2)c(F)ccnc1Cl 86341,CC1(C)CC(CNC(=O)COC2CCCCC2)CN1C(c1cccc(F)c1N)=O 86342,C(=O)(C(O)CC(C)(C)C)N1CC2C(CNC(C(C)N=[N+]=[N-])=O)(CC2)C1 86343,c1(C(=O)NCC(C)NC(=O)CCCCNC(N)=O)ccc2cccc(F)c2n1 86344,c1(CC)ccc(C(=O)NCC2(NC(=O)Cc3c(C)nn(C)c3C)CCC2)cc1N 86345,N1(C(CSCCC(C)C)=O)CCC2CC1CN2C(=O)C(c1cncc(F)c1)C 86346,N1(C(c2cc(C)cs2)C(=O)Nc2c(CC)cccc2C)CC2(C)COCC2(C)C1 86347,C1(OC)CC(NC(c2cnn(-c3nccs3)c2)=O)CN(C(C2CCCSC2)=O)C1 86348,c1(C(C)C)[nH]ccc1C(=O)NC1CCN(C(c2cc(C(F)(F)F)n[nH]2)=O)C1 86349,C1(CC(N)=O)(NC(C(C)SCC)=O)CCN(C(=O)C(O)CC(C)C)CC1 86350,C(=O)(C(C)(O)C(C)(C)C)N(CC(CN(C(C1CC2(CC(=C)C2)C1)=O)C)O)C 86351,Cc1ncc(C(N2CCC(OCC(N3CC(=O)NCC3C(N)=O)=O)C2)=O)c(C)n1 86352,CC1(C)CCN(C(C2C3CCCOC23)=O)CC1NC(c1cccc(Cl)c1)=O 86353,c1(C(N2CCC(C(CNC(CC(C)OC)=O)F)CC2)=O)cc(N)c(F)cn1 86354,Cc1cc(C(N2CCOC3(C2)CN(C(=O)C2=CCC2)C3)=O)c2cc(F)ccc2n1 86355,N1(C(CCCCCC#C)=O)CCc2[nH]nc(CNC(=O)C(C(C)C)N(C)C)c2C1 86356,N1(C(C(C)NC(c2c(C)occ2)=O)=O)CC2CC1C2NC(C1CC1C)=O 86357,c1(Nc2ccc(CNC(c3cnc(C)s3)=O)s2)ccc(C(N)=O)cc1 86358,N1(C(CCCNC(CC2(NC(C)=O)CC2)=O)=O)CC(C)C(C)C1C 86359,N1(CC(=O)N(CCC=C)C)CCC2(CCCC(CO)O2)CC1 86360,C1(NC(C(C(C)C)O)=O)CC2CCC(C1C)N2C(=O)Cc1c[nH]c2cccnc12 86361,C1(NC(C(N)=O)=O)CCCC2CN(C(=O)CC3CCCCCC3(F)F)CC12 86362,c1(C(C)C(=O)NCCN(C(C2CC(C)(C)O2)=O)C2CC2)ccc(F)cc1F 86363,C1(C(=O)NCC2CC(C(=O)NC3CCS(=O)(=O)C3)C2)(CC)CNC(=O)C1 86364,C(CC(C)(C)CBr)(c1n(CCOC)nnn1)Nc1cc(CN(C)C)ccc1OC 86365,C1(CC=C)(NC(=O)C(O)C=CC)CCN(C(c2cccc(=O)o2)=O)C1 86366,Cc1cc(C)n(C(C)C(=O)NCC2CN(C(C3OCCOC3C(F)(F)F)=O)C2)n1 86367,C1(CC2CN(C(CNC(C3C(C)C3)=O)=O)C2)CCOC1C.N1CCC1C 86368,Cn1cnc2cc(C(N3CCC(c4ncc(Br)cn4)CC3)=O)cnc12 86369,N1(C(CC(CC)OC)=O)CCC(CNC(c2ccc(Cl)c(Cl)c2)=O)C(C)C1 86370,N1(C(Cc2c(C)nc(S)s2)=O)CCCN(C(C2(C(F)F)CCCO2)=O)CC1 86371,c1(C(=O)NCC2CCC(CNC(C(C)C(C)(F)F)=O)CC2)cccc2occc12 86372,C1(CC(C)C)CCN(C(C2(CNC(=O)CCn3cnnn3)CCCC2)=O)C1 86373,CN1CCC(NC(=O)CCN(C(=O)Cn2c(O)nnc2O)CCO)C(C)(C)C1 86374,c1(C(CC(=O)NCCC(=C)CNC(=O)C(O)CC)O)ccc(Cl)cc1 86375,c1(C(=O)OCCCC#C)nn(CC)c2c1COCC2 86376,N1(C(c2c(CCC)nco2)=O)CC2CCC(C1)C2NC(=O)COC(C)C 86377,C1(NC(C2CC(=C)C2)=O)CCCC12CCN(C(c1cnc(N(C)C)cc1F)=O)C2 86378,N#Cc1ccc(C(=O)NCC2CC(NC(c3c[nH]c(Br)n3)=O)C23CCC3)c(O)c1 86379,C1(CC(N2CCC(CN(C(=O)CSCc3ccccc3)C)C2)=O)NC(=O)NC1=O 86380,C(=O)(C(C(=O)N1CCC(CCCCCNC(=O)C(C)CF)CC1)OC)OC 86381,CCC1=NOC(C(=O)N(CC(C)NC(c2ccccc2CC(F)(F)F)=O)CC)C1 86382,CC(C)(C(=O)N1CCC(NC(C2CCOC2C(F)(F)F)=O)C1)c1cccs1 86383,Cc1cc(=NCCc2nc(-c3cnn(CC4CC4)c3)nn2CC(F)(F)F)[nH]cn1 86384,C1(C(=O)NCc2cc(C)n(C)n2)CCCCCCN1C(c1ccn(CCF)n1)=O 86385,N(C(=NCc1cc(C2CC2)on1)NC1CC(=O)N(c2ccccc2)C1)C(C=C)C 86386,C(C(=O)N(C)OCC(=O)OC)C1N(C(C2C(=C)C2C(=O)OC)=O)CCC1 86387,c1(CC)cccc(C(=O)NCCCCCCN(C)C(C23CCCC2C3)=O)c1 86388,c1(C(=O)NC2CCN(C(c3cc(CC)no3)=O)C23CC3)cc2cccc(C)n2n1 86389,c1(C(N2CC(C(=O)OC)OCC23CC3)=O)[nH]nc2c1COC2(C)C 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86529,CCC(CCC(=O)N1CC(F)(CC)C1)OC.c12ccccc1NC2=O 86530,N(C1COc2ccc(Cl)cc21)C(=O)CC1CCN(c2ncc3cn[nH]c3n2)C1.CN 86531,c1(CC)cnc(NC(=O)Cn2cncn2)c(C)c1 86532,c1(C(=O)NCCN(C)C(c2ccc(F)nc2)=O)cnc(O)c(Br)c1 86533,S(=O)(=O)(c1ccc(N2CCOC3CC23)c(C#N)c1)NC1C(OC)CN(C)C1 86534,c1(OC)ccc(C)cc1C(=O)N(C1(CC(=O)N(CC(O)C2CC2)C)CC1)C 86535,c1(NC(COC)(C)C)nccc(=NCC2CCc3cccc(OC)c32)[nH]1 86536,c1(NC(=O)NCCC#CBr)ccc2cccc(Br)c2c1 86537,N1(C(CC(C)C)=O)CCC(CNC(c2cncc(N)n2)=O)C12CC2 86538,C1(=CCNC(=O)CC(F)F)CCN(C(C2(F)CCOC2)=O)CC1 86539,C(CCC(=O)N(C1CCCC1)CCNC(=O)C=CC1CCC1)N(C(C)=O)C 86540,N1(n2cc(C=O)scncc2)CC(F)(F)CC1CCNC(C1(C(N)=O)CCC1)=O 86541,C(=O)(CCC(=O)NC1(C(N2CCC(OCCNC(=O)NC)C2)=O)CCC1)NC 86542,c1(C(N2CCN(C(COC(CC)C)=O)CC2C)=O)nc(C)c(C)nc1C 86543,C=C(Cl)CCC(=O)N(CC(C)NC(=O)C(c1ccc(O)cc1)OCC)CC 86544,c1(C(=O)NCC(CC)NC(=O)C(C)SC(F)(F)F)ccc(OC)c(OC)n1 86545,c1(C(=O)NC(C)CCN(C(=O)C(C)CC(F)(F)F)C)ccc2nnc(S)n2c1 86546,c1(C(=O)NC(CNC(c2cocn2)=O)C2CCC2)cc(Cl)nnc1O 86547,c1(C(C)NC(=O)N(C2CC2c2cn[nH]c2)C(C)C)cccc(O)n1 86548,c1(NC(C(C(CC)C)O)=O)nc(C2=CCC(N3CCOCC3)CC2)cs1 86549,c1(NC(C2(CC)CC2)=O)cn(C)c(C(=O)NCc2cocn2)n1 86550,CC1=C(C(=O)NCCOC2CCN(C(c3oc(C)nc3C)=O)C2)CC1 86551,N1(C(c2ccc(CC)s2)=O)CC(C(=O)NC2CCOC(C)C2)CC1(C)C 86552,c1(N2CCCC(C(N)=O)C2)nc2ccc(Cl)cc2c(=NCCSC2CCCC2)[nH]1 86553,C1(NC(C(CSC)(C)C)=O)CN(C(=O)CN(C(=O)COC)C)CC1O 86554,c1(OC(C)=O)cc(NC(C2CCCN2Cc2cc(C)on2)=O)ccc1N 86555,c1(C(N(C)CC2CN(C(C3CCOC3)=O)C2)=O)csnc1Cl 86556,n1(CC)nnc2cc(C(N3CCCCCC(NC(C4CC(F)C4)=O)C3)=O)ccc12 86557,CCCCC(O)CC(=O)NC1(CC(N2CCCN(CCC)CC2)=O)CC1 86558,CC(CCCc1cn(CCN(C)C)nn1)C(=O)NC1(c2ccn(C)n2)CC1 86559,C(=O)(C1=C(C)Oc2ccccc2C1)N1CCC(C(C)NC(CC(=O)OCC)=O)C1 86560,N1(C(C(CC(C)C)ONC(c2cc(C)no2)=O)=O)CC2(CCNC(=O)O2)C1 86561,N1(C(CCCC#C)=O)CCCC(C2CCN(C(c3cscc3Cl)=O)C2)C1 86562,C1(C)(CC(=O)N(CCC(=O)NC(c2ccn(C)n2)C)C)OCCO1 86563,N1(C(C(C2CCC2)OC)=O)CCC(C(=O)NC(c2ccccc2F)C)C12CCC2 86564,N1(C(C23CC(C2)C3)=O)CCC12CCN(Cc1cccc(F)c1O)CC2 86565,N1(C(c2c(CCC)n(C)nc2)=O)CCCN(C(=O)CC=C(Cl)Cl)CC1C(C)C 86566,c1(NC(C(n2nc(C3CC3)nc2-c2cnc(Cl)s2)C)=O)ccc(C(F)(F)F)cc1 86567,C1(C(N(C)CC2N(C(C3CC(=C)C3)=O)CCC2)=O)C(C=C(C)C)C1(C)C 86568,S(=O)(=O)(c1cc(Cl)c(Br)cc1F)N1CC(C(=O)Nc2cncnc2O)SCC1 86569,c1(CN(CC(=O)N(C)Cc2ccccc2)C(C)(C)C)ncccc1Br 86570,c1(C(=O)NCCCNC(C(c2c(C)ccc(F)c2)O)=O)ccnc2c1ccn2C 86571,C(=O)(C(CC1CC1)NC(C1CCNC1=O)=O)N(CCCc1ccco1)C 86572,c1(N2CCN(C(=O)CCc3cnc4ccccn34)CC2)cccc2ccccc12 86573,N1(C(=O)NC(C2CCC3CCC23)C)CCC(C(C)(C)C)(NC(=O)OC(C)(C)C)C1 86574,c1(NC(=O)OCC)cccc(NC(=O)CN(C)CCO)c1.N12CC3CC3(C1)C2=O 86575,c1(CNC2C(C)CN(C(=O)CCc3ccc(OC#N)cc3)C2)cc(Cl)cc(Cl)c1 86576,c1(-c2cn(CCN3C(N4C(=O)OCC4)COCC3)nn2)ccc(F)c(Br)c1 86577,N1(C(Cc2c(C)cco2)=O)CC2CC(C1)C2NC(=O)CNS(=O)(=O)N(C)C 86578,c1(C(N2CCC(NC(C(CCC)OC)=O)C2)=O)cc2c(nc1O)CCSC2 86579,C1(NC(=O)CCF)COCC1NC(c1cn(-c2ccccc2)nn1)=O 86580,Cc1c(C(N2CC(C)N(C)C(C)C2)C(=O)NCCC2CC2)cc(F)cc1[N+](=O)[O-] 86581,CCCCCCC[SH](=O)(CCCC)CC(=O)N1CCC1Cc1ccccc1 86582,N1(C)CCN(C(=O)C(C)N2CCCC2)CC1.c1(C(C)=O)ccc(C(F)(F)C(=O)OC)cc1 86583,n1(CC)ccc(=NC(=O)C2CCC(C(C)C)N2C(C2CC2Cl)=O)[nH]1 86584,C1(c2c(C(N3CC(CCS(N)(=O)=O)C3)=O)c[nH]n2)COCCN1C(=O)CC1CC1 86585,c1(OC)cc(O)ncc1C(=O)NC(CNC(C1(C#N)CCC1)=O)CC(C)C 86586,C(=O)(CC(O)C(C)CC)NCC(CC(=O)N(CC(C(=O)NC)C)C)O 86587,C(C(CNC(=O)C=NOC)S(C)(=O)=O)NC(C1N(C(C(CC)C)=O)CSC1)=O 86588,CCCCC(O)CC(=O)NC(CNC(=O)C(C)(C)c1ncco1)CO 86589,C1(OCc2c(C)csc2Cl)CCN(C(=O)OCc2ccccc2)CCC1CO 86590,N1(C(C2CCC(F)(F)CO2)=O)CCC2(CC1)CCN(C(C1C=CCCC1)=O)C2 86591,c1(C(=O)NCC(C)NC(c2cc(=NC)[nH]cc2)=O)csc(=NC2CC2)[nH]1 86592,CS(=O)(=O)c1ccc(F)c(C(=O)NCC2CN(C(=O)NS(C)(=O)=O)C2)c1F 86593,C1(CN(C)C(c2cnn(C3CCC3)c2)=O)CN(C(C2CC(F)C(=O)N2)=O)CCO1 86594,c1(N(C)C)ccc(C(=O)NCCCCCCNC(=O)Cc2cnn(C)c2)nc1 86595,CC1OC2(CNC(=O)C(C)NC(C)(C)C)CC1(NC(C1CCN(C)C1)=O)C2 86596,C1(NC(C(CCSC)O)=O)CCN(C(=O)Cc2ccc(Cl)s2)C12CC2 86597,C=CCC(C)(C(=O)NC1(CNC(=O)C(C)CC)CCC1)N(C)C 86598,C(=O)(C1Cc2ccccc21)NC1CN(C(C=C(C)C)=O)CC12CCC2 86599,c1(C(=O)NC2C(NC(c3c(C)noc3C3CC3)=O)CC2)onc2ccccc12 86600,C1(C(=O)NC(c2ncccn2)CC)CN(C(C2(C)CNC(=O)N2)=O)CCO1 86601,c1(C(N2CCC(NC(CC(=O)N(C)C)=O)CC2)=O)noc2c1CCCC2 86602,CC1(C)CCC(CNC(C2CCC(=O)N2)=O)N(CC2CCCOCC2)C1 86603,S(=O)(=O)(C(Cl)(Cl)Cl)NCC(N1C(C(=O)Nc2scc(C)n2)CCC1)=O 86604,N1(C(C2(NC(CC(C)OC)=O)CC(F)C2)=O)CCC(C)(F)C1 86605,N1(C(C2N(C(C3(CCCC)CC3)=O)CC(O)C2)=O)CCN2CCCCC1C2 86606,C1(CNC(C(CSC)(C)C)=O)CC(C)CN(C(=O)CC2CC(F)C2)C1 86607,C(CC(=O)NOC1CCOC1)(C(F)(F)F)NC(C(C)NCC)=O.C(C)(=O)OC 86608,C(=O)(C1=CCCC1(C)C)NC(C)CCNC(c1cc(OCC(F)F)ccn1)=O 86609,C1(CCC(=O)NCC(=O)NC(C(=O)OCC)OC)(COC2CC2)CCCO1 86610,C1(O)(CC(=O)NCC(CCOC)NC(C2(CC=C)CCC2)=O)CCCCC1 86611,Cc1nnc(NCC2CCC(NC(=O)Cc3nc(C)c(C)s3)C2)c(C#N)c1C 86612,O(NC(=O)C(C)(C)CCCNC(=O)CCC(C)CC)C(C=C)C 86613,c1(NC(=O)NCc2nccc(OC)c2)ccc(I)cc1Br 86614,C1(C)(NC(=O)COC(C)(C)C)CN(OC(C)=O)C1.C12(CC1)C(=O)N2 86615,C1(F)(C(=O)NC2CC(NC(c3cc(C(=O)OC)[nH]c3)=O)C2)CCS(=O)(=O)C1 86616,c1(OC)ccnc(C(=O)NCC(C)N(C(=O)CC(C)n2ccnc2C)C)c1F 86617,C1(C(N2CC(NC(c3ccccc3)=O)C2)C)CCC(C)(C)CO1 86618,Cc1ccc(CN2CCOCC(C(=O)NCC3=CCCCC3)C2)c(C)c1 86619,N1(C(C=CC)=O)CCOC(CN(C)NC(C2CC2C(N)=O)=O)C1 86620,C1(NC(c2ccc(C)s2)=O)CC12CCN(c1cc(=O)n(C(C)C)c(O)n1)CC2 86621,C1(NC(C2(CC=C)CCCC2)=O)CN(C(C2CC2(C)C(F)(F)F)=O)CC(C)(C)C1 86622,N1(C(c2ccnn2C)C2CC(=C)C2)CCCCC1C1CCCN1c1ncns1 86623,c1(OC)ccc2ncccc2c1C(=O)N(C(C)CCNC(C1(O)CCOC1)=O)C 86624,c1(C(C(=O)NC2C(NC(CC(C)SC)=O)C2)NC(C)=O)c(F)cccc1F 86625,C1(NC(C=CCC)=O)CN(C(c2ccc(-n3ccnc3)cc2)=O)CCC1C 86626,C1(C(N2CC=CC(NC(c3cc(Cl)c(Cl)s3)=O)C2)=O)(OC)CCCCC1 86627,c1(CCc2n(CCCC)nc(CC3CCC3)n2)c(Cl)ccc(Br)c1F 86628,c1(C(N(CC(C)NC(=O)Cn2cc(C#N)cn2)C)=O)ncccc1OC(F)F 86629,c1(SC)ccc(C)c(C(N2CCCC3(NC(c4ccn(C)n4)=O)CC23)=O)c1 86630,CS(=O)(=O)c1ccc(CN2CCC(O)(C(=O)Nc3ncc(I)nc3Cl)C2)cc1 86631,c1(CNc2c(C#N)ncc(C(=O)OC)n2)ccc2ncn(C)c2n1 86632,C(C)(CCC(=O)NOCCCC(=O)OC)NC(c1c(CC)cco1)=O 86633,C1(NC(C2(CC=C)CC2)=O)CC2CC1CC2C(=O)NC(CO)C1CC1 86634,C1(NC(C2CCN(C(=O)CNc3cccnc3)C2)=O)CCS(=O)(=O)N1 86635,C1(NC(C2CCO2)=O)CCC2(CC1)CN(C(c1ccc(C3CC3)cn1)=O)C2 86636,C1(NC(CC(C=C)CC)=O)CC(C2CCN(C(C3(C)CC4C=CC3C4)=O)CC2)C1 86637,C=CCC(CNC(C1CCCCS1)=O)C(=O)Nc1ccc[n+]([O-])c1 86638,C(=O)(C#CC1CCCOC1)N1CCN(C(c2c(COC)scc2)=O)C(COC)C1 86639,N1(C(CC2C(=C)CC2)=O)CCC2(CC(NC(c3cc(C)c(Cl)cc3C)=O)C2)C1 86640,c1(C(=O)NC(c2nc[nH]n2)C)c(CNC(=O)CC(C)(C)N(C)C)cnn1C 86641,CS(=O)c1ccc(C(=O)NCC2(NC(=O)CC(F)F)CCCC2)cc1 86642,N1(C(c2ccc(C)cc2O)=O)CC2CCC(C1CO)N2C(=O)Cc1ccco1 86643,C12(C(=O)NC(C)CNC(=O)Cc3cc(F)ccc3F)CC=CCN1CCC2 86644,Cc1cc(F)c(Br)cc1NC(C1CC(C)CN1C(c1cccnc1F)=O)=O 86645,C1(C(=O)NC(C)C(N)=O)CC(F)(F)CN1Cc1cccc(-n2ccnc2)c1 86646,c1(OC(C)C(=O)NCCC2CN(C(c3ccnn3CCF)=O)C2)cccc(Cl)c1 86647,N1(C(C2C(C)C2C)=O)CCC(CCCNC(C2(C)CCCOC2)=O)CC1 86648,c1(NC(CC(C)(C)n2cc(CNC(C(C)O)=O)nn2)=O)ccc2ncsc2c1 86649,C1(CNC(c2c(C)csc2C)=O)COCCN(C(=O)Cc2cnn(C(C)C)c2)C1 86650,c1(NC(C(=O)NNC(=O)C2CC3CCC2O3)=O)cc(-c2ccccc2)ccc1Cl 86651,c1(C(=O)NC(c2cn(C(C)C)nc2)C)cccc2c1CCO2 86652,C1(C(=O)NCCCOCCNC(C2C=CC=CC=C2)=O)CCC2(CCOC2)O1 86653,C(=O)(C(CCC(C)C)NC(C1CCC(=O)C1)=O)NC1(CCOC)CC1 86654,N1(C(C2C(C(N)=O)COC2)=O)CCC(C2CN(C(C3CCO3)=O)C2)CC1 86655,C1(C(=O)NC2C(C=O)C2)CCN(C(c2ccc(CC)[nH]2)=O)CC1.CCOC 86656,C1(NC(C2(CC=C)CCCC2)=O)CCN(C(c2cc(C(F)F)[nH]n2)=O)CC1CO 86657,Cc1cnccc1C(=O)NCC12CC1CN(C(c1ccc(C(F)(F)F)o1)=O)C2 86658,C1(C(=O)NC(CCC)CC)CCCCCCN1C(C1CC2C=CC1O2)=O 86659,C(CCC(O)CO)N(C(CC1(C)N(C(C=CC=CCC)=O)CC1)=O)C1CC1 86660,N#Cc1cccc(F)c1NC(C1CC(F)CN1C(c1ncccc1Cl)=O)=O 86661,C1(NC(=O)OC(C)(C)C)CCCC1C1CC1NC(c1cc(C(F)(F)F)cnc1Cl)=O 86662,N1(C(=O)OC(C)(C)C)CC(C(N2CCC3(CCC3)C2)=O)C(C2CCCC2)C1 86663,C(=O)(C(CC(C)(C)C)OC)NC(C(=O)NCCOC)(C)CO 86664,C1(C(=O)NCCCN(C(=O)CC2CCCC(=O)N2)C)Cc2c[nH]cc2S1(=O)=O 86665,N1(CC)CCC(CN(C)CC)C1.n1(CCOCC(CCOC)O)nnnc1C.C1CC1 86666,C1(C(=O)NC2(CCNC(C(C)OCC(F)(F)F)=O)CCCC2)CCCC1(C)C 86667,C1(C(=O)NC(CCCC=C)C)CC(C)(C)CN1C(c1cnc(O)c(C)c1)=O 86668,C1(C(N(CC(N2CCCC2)C)C)=O)CCN(C(=O)CCN=[N+]=[N-])C(C)C1 86669,CCS(=O)CC(=O)N1CCC(C(=O)N(C(C)C(N)=O)C)(CF)C1 86670,N1(C(c2cnn(C)c2C#N)=O)CCCC2(CCCN2C(C2CCC2(C)C)=O)C1 86671,Cc1ccc(NC(=O)C(C2CC2)N(C(=O)C(O)C(F)(F)F)C)cc1Cl 86672,c1(C(=O)NCC(CN(C)C(C2CC2(C)Br)=O)O)ccc(N)cn1 86673,C1(C(=O)NCC2(C#C)CC2)CC(C)(NC(C2CC(O)(C(F)(F)F)C2)=O)C1 86674,c1(CNC2C(C(=O)NC(C=C)CO)C2)csc(Br)n1 86675,CN1N=C(CC(=O)N2CC(=O)NCC2C(N2CC3C(C(N)=O)C3C2)=O)CC1=O 86676,Cc1cc(C)c(NC(=O)NC2CC3CC2CN3C(c2cc(C)[nH]n2)=O)c(C)c1 86677,C#CC1(c2ccccc2)COCCN1C(=O)NC.C12CCCN(C1=O)C(C1CC1)CC2 86678,c1(OC)nc(Cl)ccc1C(=O)NC1CC(C)(CNC(=O)CN2CCSCC2)C1 86679,C1(NC(C2CC(C#N)C2)=O)CCC(NC(=O)CN2CCS(=O)CC2)CC1 86680,C(=O)(C(F)C(C)(F)F)N1CCC(CC(=O)N(C2CCS(=O)(=O)C2)C)CC1 86681,N1(C(CC2(OC)CN(C(=O)CC3CCCSC3)C2)=O)CCC12CN(C)C2 86682,N1(C(C(C=C)OC)=O)CCC(C(=O)NC2CC3(CC3)C2)C12CCC2 86683,Cc1cc(C(=O)NCC(C)(O)CNC(=O)CCSCC(C)C)nn1C(C)C 86684,C(=O)(CCC(C)(C)C)NCCCCN(C(=O)CC(O)c1cnc(Cl)s1)C 86685,C1(C(NOCCCN(C)C)=O)CCOCCN1C(C1CC(=O)NC1(C)C)=O 86686,N1(C(C=CCN(C)C(c2ncccc2F)=O)=O)CCC2CC2CC1 86687,c12cc(nc(Cl)n1)N2CCNC(CC(C=C)c1ccccc1)=O.C(C)(=O)NC 86688,c1(CC(N2CC(N(C(C(CCC)C)=O)C)C(O)C2)=O)c[nH]c2ccc(OC)cc12 86689,c1(N(C)C)cnccc1C(N1CC(NC(C2CCC23CCC3)=O)C1)=O 86690,C(CC(C(=O)NC(CC1CCCC1)CO)NC(C12CC(F)(C1)C2)=O)=CC 86691,CC(C(=O)NCC1CCN1C(c1csc(C(N)=O)n1)=O)P(C)(C)=O 86692,C(C(C)(C)C(=O)NCC(C(=O)NCCC1CCCCO1)N(C)C)OCC 86693,C(C(C)CC(=O)NC1CCN(C(C2CCSCC2)=O)C1C1CC1)OC 86694,c1(C(=O)NC2C(CNC(C(C)OCCCCCC)=O)CC2)ccn2cccc2c1 86695,C1(CNC(c2cnn(C)c2Cl)=O)CCC2(CN(C(c3coc(C(N)=O)c3)=O)C2)O1 86696,N1(C(C(C=CC)O)=O)CC2CCN(C(c3nn(C)c(Cl)c3Cl)=O)C2C1 86697,c1(C(N(C2CCC(NC(C3CC4(C3)CC4F)=O)CC2)C)=O)cc(N)c(Cl)c(O)c1 86698,c1(C(N2C(CN(C(c3cccc(C#C)c3)=O)C)CCC2)=O)ccc2c(c1)OCC2 86699,Cc1nc(C(=O)NCC(CC(C)C)NC(=O)CC2(C)CC2)c(C)s1 86700,N1(C(C=C(CC)C)=O)CCCC(O)(CNC(=O)CC2CCCN(C)C2)CC1 86701,N1(C(C2(C)CCN(c3nc(SC)c(F)cn3)C2)=O)CCC2(CCCO2)C1 86702,c1(CCC(=O)Nc2cc(OC)c(F)cc2)ccc2[nH]ccc2c1 86703,c1(C(=O)NC2CN(C(C(C=C)(F)F)=O)CC2C(F)F)ccc(Cl)c(C)c1N 86704,N1(C(C)=O)CCc2c(NC(C3(C)CCCOC3)=O)cccc21 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86776,CCCC(C(=O)NCC1(COC)CN(C(=O)C#CC2CCCO2)C1)C(C)C 86777,C(CC1CCC1)(C(=O)NCC1CC(O)C1)NC(C(C)OCCCC)=O 86778,c1(C(=O)NCC2CC(NC(C3CCC(C)NC3=O)=O)C2)ccc2n[nH]cc2c1 86779,N1(C(CC=CC=C)=O)CC=C(C(=O)N(CCCN(C)C)CC)CC1 86780,CC#CC1CCN(C(=O)C(F)CC2CN(C(c3cnn(CC)c3)=O)C2)CC1 86781,C1(C(N2C3(CN(C(c4cn(C5CCC5)nn4)=O)C3)CC2)=O)CC2CCCCN2C1 86782,N1(C(C(C2CCCCC2)OC)=O)CC2C(CNC(C3CCC(C)(C)C3)=O)C2C1 86783,C1(NC(C2CC(Cl)(Cl)C2)=O)CCC2(CCCN(C(c3ccncc3)=O)C2)C1 86784,c1(NC(C(CCSC)NC(c2sccc2C#N)=O)=O)cc(C)cnc1C 86785,N(C1c2ccccc2CC1NC(=O)C(C)C(O)CC)C(c1cn(CCC)nc1)=O 86786,C1(C(=O)OCCCOC)CCC=CC1NCc1ccc(C)cc1 86787,c1(C(N2CCCC(N(C)C(C3C4CCC34)=O)C2)=O)ccc(C(F)(F)F)cc1Br 86788,N1(C(CC(C)C)C(=O)Nc2ccccc2)CCS(=O)(=O)CC(C)C1 86789,N1(C(CN2CCN(Cc3ccnc(C)n3)CC2)=O)CCN(CC(C)(C)O)C(C)C1 86790,CC(O)CCCC(=O)N(C(C)CCNC(C1(S(C)(=O)=O)CCC1)=O)C 86791,C1(C(=O)NCC(C(=O)Nc2c(CCC)cccc2)C)CC(=O)OC1(C)C 86792,c1(C(=O)NCC(CNC(COCCOCC)=O)(C)F)ncncc1C 86793,C(=O)(C(CO)C(C)(C)C)N1CCCC(F)(C(=O)NCC(N2CCCCC2)CC)C1 86794,C(=O)(C1=NOC(C)(C)C1)NC1CN(Cc2nc(C)sc2C)C(C)CC1 86795,CC(CC(F)F)C(=O)N1CCCCC(NC(=O)COCC2CCC2)C1 86796,CC(C)S(=O)(=O)CC(=O)NC(C)C(CO)NC(c1ccccc1Br)=O 86797,c1(NC(=O)CC(F)(F)Cc2cccc(Br)c2)[nH]nc([N+](=O)[O-])c1Br 86798,c1(C(C(=O)NCCN(C(COC(C)C)=O)CC(C)O)C)ccccc1C(F)(F)F 86799,C1(OCC#C)CCN(C(C2CCOCC2NC(C2CCN(C)C2C)=O)=O)CC1 86800,Cc1ccncc1C=CC(N1CC2CC(NC(=O)CC3CCC4CC34)C2C1)=O 86801,CS(=O)(=O)C1CCCC1C(=O)NCC1(NCC(F)(F)F)CCC1.C1(=O)C=CCN1 86802,C1(CC(=O)NCCC2(O)CN(C(CC#N)=O)C2)CC2(CCC2)CCO1 86803,c1(C(=O)NCCCC(c2ccccc2)NC(CN(CC)CC)=O)sc(C)cc1Cl 86804,C1(NC(C(CCSC)N(C)C)=O)CC12CCN(C(C1(C#N)CC1)=O)CC2 86805,C1(C(=O)NCCCOCCN(C(CC=C=C)=O)C)Cc2ccccc2O1 86806,CC(C)C(C(=O)N1CCC(c2cccc(F)c2)(NC(c2cocn2)=O)C1)NC=O 86807,C(=O)(N=c1cc(C2CCC2)[nH][nH]1)C1(C)CCN(C(=O)Cn2ccnn2)C1 86808,C12(CC)CN(C(=O)CCCSC)C(CNC(c3sc(C)c(C)c3C)=O)(C1)C2 86809,C1(C)(CC)CC(C(=O)NC2CC(CCNC(c3csc(S)n3)=O)C2)C1 86810,c1(Nc2cccc(CC(N)=O)c2)ccc([N+](=O)[O-])c(OC2COC2)c1 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86828,c1(C(=O)NC2CCCC2CSc2ccc(CO)o2)ccc2c(c1)CCC2 86829,c1(C(=O)NCC(C)(C)OCCNC(C2CCN(C)C2)=O)cccc(C#N)c1 86830,N1(C(C#C)=O)CC2CCN(Cc3ccc(O)c(O)c3)CC2C1 86831,CC1=NNC(=O)C1CCC(=O)NCC(C1CCC1)NC(C1(n2cccn2)CC1)=O 86832,N1(C(C(C)N(C(CC2ON=C(C)C2)=O)CCO)=O)CC(S(C)=O)C1 86833,C1(C(N(C2CCN(CC)C2)C)=O)CCN(C(c2cc(F)cc(F)c2)=O)CC1O 86834,N1(C(C2(N(C)C)CC2)=O)CCC(F)(CNC(=O)CC2COC(C)(C)C2)CC1 86835,N1(C(=O)C=Cc2cncnc2O)CCN(C(c2cc(F)ccc2F)=O)CC(O)C1 86836,C1(CC(=O)N(C2CC(NC(CN(c3ccccc3)CC)=O)C2)C2CC2)OCCCO1 86837,C(=O)(CCCCOC(C)C)N1C(Cc2cn(CC(=O)OC)nn2)CCC1 86838,C1(NC(=O)C=Cc2ccncc2)CN(C(=O)Cc2csc(S)n2)C2(CCOC2)C1 86839,C(=O)(C1=COCCO1)N(CCN(C(=O)C(N1C(C)CCC1C)C)C(C)C)C 86840,c1(C(c2n(C(CC)(C)C)nnn2)NCc2sccc2Br)ccc2nc(O)[nH]c2c1 86841,C1(CC#C)(C(=O)N(C2CCN(C(=O)CCC=C(C)C)C2)CC)CCCCC1 86842,N1(C(C(CCC)OC)=O)CC(CNC(=O)CCn2cncn2)C2(CCOCC2)C1 86843,N1(C(CCN(C)CC)=O)CC2(CC(NC(=O)C(C)C3CC3)c3nccn32)C1 86844,C(=O)(CC(OC(C)C)OC)NC(CN(CC)CCC(N1CCCCC1)=O)C 86845,CON(C)C(=O)C1(C(=O)NC(=O)C(C)=CC(C)(C)C)CCC1 86846,c1(OC)cncc(C(=O)NCC(C)NC(=O)CC2CC2c2ccc(F)cc2)n1 86847,C(=O)(C1Cc2ccc(Cl)cc21)N1C(C)(CNC(=O)CC2CC3(CC3)CO2)CCC1 86848,C1(CCNC(c2cn(CCC)nn2)=O)COCCN1C(=O)C(C)n1ccnn1 86849,c1(C(N(C(c2cn(-c3cccnc3Cl)nn2)C)C)=O)cccc(Br)c1 86850,N1(C(CCCc2cn(C(c3ccc(F)cc3)C)nn2)=O)CCCC(O)(C(=O)NC)C1 86851,Cc1cc(=NCc2ccc(CCCc3ccco3)o2)[nH]cc1S(=O)(=O)N(C)C 86852,c1(CC(N)C(N2CCNC(=O)C2c2ccccc2Br)=O)cn2c(n1)CCCC2 86853,c1(C(c2nnnn2C2CC2)NC(CC=C)C2CC2)ncc(Br)cc1OC 86854,c1(CC)sc(C(N2CCC2CNC(=O)CCF)=O)cc1Br 86855,c1(N(C)Cc2c(OC)nsc2OC)nc(=NC2CCC(CO)C2)[nH]c2c1CCC2 86856,Cc1nc(C(N2CCC(F)(CNC(=O)CC3NC(=O)NC3=O)C2)=O)sc1C 86857,c1(C(=O)NCC(C2CCCC2)NC(C(C)c2ccon2)=O)c(F)cccc1F 86858,C1(C)(C(=O)Nc2cccc(CC)c2F)COC(C)(C)OC1 86859,c1(SCC(=O)NC2CCCC2CNC(=O)C(O)c2cnc[nH]2)nnc(S)s1 86860,C#CC1(C(=O)NOCC2CCCO2)CN(C(=O)C=CC(C)C)C1 86861,Cc1cc(CC(N2CC(C(C)(C)O)(CNC(C3(C)CC3(F)Cl)=O)C2)=O)c(C)s1 86862,CC1CC(C(N2CCC(CCNC(=O)CC3CCCCO3)CC2)=O)CCO1 86863,Cn1nccc1C1CC1C(=O)NC(C)(CNC(=O)COc1cccnc1)CO 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86899,C(=O)(C(Cn1cccn1)NC(=O)C(c1ccccc1)=O)N(C)C 86900,N1(C(CC(C)OCC)=O)CCN(C(c2ccc(OC(C)C)nc2)=O)CC12CC2 86901,C1(C(N2CC(O)(C(C(=O)N(C(C)C(=O)NC)CC)F)C2)=O)CC12CCOCC2 86902,C1(NC(Cc2cccc(CC)c2)=O)CCN(C(=O)C(=O)NC2CC2)CC1C 86903,CC(CCC(C)(C)C)C(=O)NCC1CC(C(N2CC3(CC(F)C3)C2)=O)C1 86904,C1(NC(c2c(C)n(C3CC3)nc2)=O)CCCC2CN(C(=O)CC3(C#N)CC3)CC12 86905,c1(C(=O)NC2CCCC2NC(C2SCCCS2)=O)cccc(CCO)c1 86906,Cc1sc(C(=O)NC(C)CCCNC(=O)C(C(C)O)N(C)C)nc1O 86907,C1(COC)(NC(c2cc(C)nn2C)=O)CCN(C(C2CC23CCC3)=O)CC1 86908,c1(NC(CSCCNC(C(=O)NCCC2CCCC2)=O)=O)cc([N+](=O)[O-])n[nH]1 86909,C=CCC(C(=O)NC1CC1NC(=O)Cc1sccc1C)NC(=O)OC(C)(C)C 86910,C1(NC(C2CC(CNC(C(n3ccc(C)n3)C)=O)OC2)=O)CCC=CCCC1 86911,CC(CC(F)F)C(=O)N1CC(NC(c2cnc(Cl)s2)=O)C(C(F)F)C1 86912,C1(C(=O)NC2CCN(C(C(CCC)NC(N)=O)=O)C2)CCC2(CCCCC2)CC1 86913,c1(C(N2CCC(COC)(NC(=O)CC34CC(C3)C4)CC2)=O)cc2c([nH]1)CCCC2 86914,c1(-c2nnn(C34CCC(CC3C)C3CC(CCCSC3)N4)n2)ccc2c(c1)OCO2 86915,CC1CN(C(C2(CNC(=O)C(C3(O)CCCC3)F)CCCCC2)=O)CC1O 86916,Cc1cc(C)c(C=CC(=O)NC2CCC2CNC(c2cc(C)[nH]c2C)=O)c(C)c1 86917,O=C(CC1=CCN(C(c2coc(CO)c2)=O)CC1)N1CCC(c2nc[nH]n2)C1 86918,C1(NC(c2nnc(C)s2)=O)CN(C(c2ccc(N(C)C)cc2F)=O)CC1C1CC1 86919,C12(C(=O)NCC34C(CN(C(c5cc(CCC)ncc5)=O)C3)C4)CCC(CC1)OC2 86920,C1(CCN(C)C(C2(C)SCCCS2)=O)CCN(C(=O)CC2CCCCO2)CC1 86921,C1(OC)CC(C(=O)NCc2cc(CC(C)C)on2)N(C(=O)CCOC(C)C)C1 86922,CON(CCC(=O)N1CCC(N(C)C)C1)C(=O)CC1CC2CCC2C1 86923,c1(CC(=O)N(C(CNC(c2cn(C)nn2)=O)C2CC2)C)noc2ccccc12 86924,N1(C(C(C=C=C)C)=O)CC(C2CCN(C(=O)Cn3ccc(=O)n(C)c3=O)CC2)C1 86925,C#Cc1ccc(NC(C2COCCC2NC(=O)CNC(C)=O)=O)c(C)c1 86926,C1(C2CN(C(C3CCC(C)C3)=O)C2)CN(C(c2ccco2)=O)CCO1 86927,C12(NC(CC(C(=O)OC)C)=O)CCC(CN(C(C3(CCF)CCC3)=O)C1)C2 86928,C(=O)(CCCC(=O)NC(C(C)NC(=O)CSCc1ncc[nH]1)C(C)C)OCC 86929,CS(=O)(=O)c1ccccc1NCC1C2CC(O)C1NC2 86930,N1(CC(=O)NCc2nocc2C(=O)N(C2CC2)Cc2ncon2)C(=O)CCC1=O 86931,Cc1nnc2n1CC(C(N1CC3(C1)CN(C(=O)CC(C)C)CC3CO)=O)N(C)C2 86932,c1(CC(N)C(F)F)ccc(C2CCC23CCC3)cc1 86933,C1(CNCc2cc(F)c(Cl)cc2Cl)CCC2COCCC2C1 86934,C(=O)(CCC(C)N=C(NC1CC1)NC1CC1c1cc(Cl)cc(Cl)c1OC)NC 86935,c1(C(N(C)CC2OCCN(C(C(CC)(C)F)=O)C2)=O)ccc(S(N)(=O)=O)s1 86936,c1(C(=O)NCC2N(C(C(C)=C3CCC3)=O)CC(C)CC2)ccc2sccc2c1 86937,c1(C(=O)NC(C2CCCN2C(=O)Cc2cncs2)C)nc[nH]c2ncnc1-2 86938,C(=O)(C1CCc2nccn21)NC1(C)CCCN(C(c2cccc3ncsc23)=O)C1 86939,CON(C(=O)C1=CCC(NC(C23CCC(C2)C3)=O)C1)C1CCC1 86940,c1(CN2CC(NC(C(CCC)C)=O)C(F)C2)cc(Br)cc(Cl)c1O 86941,c1(CNC2(c3n(CCCSC)nnn3)CCCC2CC(C)C)nc(F)ccc1Br 86942,c1(C(=O)NC(C2(CNC(C3(CF)CCC3)=O)CC2)C)ccc2n[nH]cc2c1 86943,N1(CC)CCC(N=c2[nH]c(C(F)(F)F)nc3cc[nH]c23)C(C)C1 86944,N1(C(Cc2cc(C)on2)=O)CC(NC(C2(C)CC2(C)C)=O)C(C)C1 86945,n1(CC)ccc(C(=O)NCC(C)CNC(c2scc(C)c2Cl)=O)cc1=O 86946,CN1CCOCC1CC(N1CCC(O)(C(=O)NC2(c3cccnc3Cl)CC2)C1)=O 86947,Cc1nsc(NCC2(C(=O)NCc3nn(C)c(C)c3Br)CC2)c1C#N 86948,N1(C(C=C(C)Cl)=O)CCCC2(C1)CN(C(c1cnc3c(Cl)cccn13)=O)CCO2 86949,C=CC1(C(=O)NCC2C3CCCCCC23)CCN(C(C2CCC(C)(O)CC2)=O)C1 86950,c1(C(=O)NCC(=C)CCNC(c2cc(-c3cccnc3)on2)=O)oc(C)cc1C 86951,C1(C(=O)OC)CCC2(CC2)N(C(CCc2ccccc2F)C(=O)NCCCF)C1 86952,C1(CN(C(=O)CC2CCCCC2O)C)COCCN1C(=O)CC1CC=CC1 86953,Cc1nn(C)c(C)c1CC(=O)NC(CNC(C1CC1c1ccsc1)=O)C1CC1 86954,c1(C(N2CCC(CC#C)(C(=O)N(CCF)CCOC)C2)=O)cc(F)ccc1F 86955,N1(C(C)(C)C)CCOC(C(=O)NCCNC(=O)C(c2ccc(F)cc2)C2CC2)C1 86956,C=C1COc2c(-c3nc(CCCN)no3)cnn2C1 86957,C1(NC(CCC#CC)=O)C2CCN(C(=O)Cn3cccn3)CCC12 86958,n1(C23OC(C)C(C2)C3)c(-c2ccoc2)csc1=Nc1ccc(Cl)c(F)c1 86959,C1(C2CCN(C(C(CC)C)=O)C2)CCCCN1CCOCCOCCOCC(C)(C)F 86960,c1(C(=O)NCC2CN(C(CCN(S(C)(=O)=O)C)=O)C2)ccc(C#N)cc1Cl 86961,C1(F)(CNC(C2CC=CCC2)=O)CN(C(=O)C(F)(F)c2csc(Cl)c2)C1 86962,c1(NC(C2CCN(C(=O)CCF)C2)(C)C)cnc(C(=O)OCC)s1 86963,N1(C(C(CNC(C2CCCC(F)C2)=O)N(C)C)=O)CCn2cncc2C1 86964,c1(CC)ccc(OCC)c(C(=O)OCC2COC(C)(C)CO2)c1 86965,c1(CC(=O)NC)ccc(C(=O)NC(C)(C)CCCNC(=O)C(O)C(C)SC)cc1 86966,c1(C(C(N2CCC(CNC(C(CC)(C)C)=O)C2)=O)(C)C)ccc2ccccc2c1 86967,C1(C(N2CC(CC)N(C(=O)COCCOCCO)CC2)=O)CCC12CCOCC2 86968,C=CC1CN(C(=O)C(C(C)C)NS(C)(=O)=O)CC1NC(C1CC(=C(F)F)C1)=O 86969,n1(CCCSCC)nnnc1C(c1cnccn1)NCC(C)C(C)C 86970,C(=O)(C#CC1CCCOC1)N1CCC(C)C(NC(C2CC(C)OC2C)=O)C1 86971,C1(C(N(CC(C)O)C(C)C)=O)CCC(C)(C)N(C(=O)CC2CCCO2)C1 86972,c1(SCCc2c(C)cc(C(=O)NC(=O)CCc3cscn3)o2)nn(C)c(=O)n1C 86973,N1(C(CCc2ccc(C)o2)=O)CC(O)CC1(C)C(=O)N(CCC(C)C)C 86974,c1(CC(N2CC(n3cc(CC(=O)OC)nn3)C2)=O)ccc(C#N)cc1 86975,O=C(C1c2ccccc2CN1c1ncnc2c1CCC2)N1CCC2(CCC2)C1 86976,N1(C(c2ccc(CNC(Cc3cc(C)sc3)=O)cc2)=O)CC(O)CC12CCC2 86977,c1(CC)cc(C(=O)NC2COCCN(C(C3CCCC(C)(C)C3)=O)C2)c(C)nn1 86978,C1(C(N2CC(S(C)=O)C2)=O)CC2C=CC1N(C(c1csc(C#N)c1)=O)C2 86979,O=C(CCS(=O)(=O)c1cccc2scnc12)NCC1COC2CC1C2 86980,c1(CNC(c2cnn(C)c2)CC)cccc(CC(F)(F)F)c1 86981,C(=O)(C(CCCCCCO)N(CCc1ccccc1)C(C)C)NC(C)C 86982,c1(C(N(CC)CC2CCCO2)=O)oc(CNC(=O)CC(C)C2CC2)nc1C 86983,C1(NC(COCCC(C)C)=O)CCCC(C(N2CCC(C)(C)C2C)=O)CC1 86984,N1(C(c2cnc(CC)nc2)=O)CCCC(C)(C)C1C(=O)NCC(F)C(C)(C)O 86985,c1(N2C(C(N3CCC(Cl)C3)=O)CC(O)C2)ncnc2c1ccn2-c1ccccc1 86986,c1(N(CC(=O)N(C2CCN(C(C)=O)CC2)CC)[NH+](C(C)(C)C)[O-])cc(C)c(Cl)c(C)c1 86987,C1(CNC(C(CC)NC(c2n[nH]cc2Cl)=O)=O)C2CCCCCC12 86988,N1(C(C2C(C=C)C2)=O)CCC2(C1)CN(C(=O)Cc1ccc3nn[nH]c3c1)CCO2 86989,N1(C(CN(C)C2CC2)=O)CCC(CCNC(C2CC=CC2)=O)C(F)(F)CC1 86990,c1(C(=O)NC2CCCC3CCC2N3C(C2CCO2)=O)[nH]c2ccc(Cl)cc2c1Cl 86991,C1(F)(C(N(CCN(C(C)C)C(C23CC(CO)(C2)C3)=O)C)=O)CC1(Cl)Cl 86992,CC1(C)c2ccccc2CC1C(N1CC2CCC(C1)N2C(=O)CCC(F)(F)F)=O 86993,c1(C(=O)NCC(CCOC)NC(C2(C#N)CCC2)=O)cncc2nc(C)[nH]c12 86994,C(C)(C)(C(=O)NNC(=O)CN1CCC(OCC(F)F)CC1)OC 86995,C(C(=O)OC)(C(=O)OC(C)(C)C)OC.c1(C23CN(C2)C(=O)O3)cccc(C)c1 86996,c1(C(=O)NC2C(OC)CN(C(c3sccc3SC(F)F)=O)C2)cnc(C)c(C)c1 86997,CP(C)(=O)c1cncc(C(N2CCCC(NC(=O)COC3CCOC3)C2)=O)c1 86998,N1(C(C2CNC(=O)N2)=O)CC(CNC(c2cnccc2Cl)=O)C2(CCC2)C1 86999,C1(C(=O)OCC)CCCC(NCc2cc(CCC(=O)OC(C)(C)C)cs2)C1 87000,c1(NC(C2(C)CCN(Cc3cnc(OC)c(Br)c3)C2)=O)ccc(F)cc1[N+](=O)[O-] 87001,N1(C(Cc2c(C)nccc2)=O)CCC2C1CCN2C(c1cc2cccnn2n1)=O 87002,c1(OC)cc(F)c(C)cc1NCc1ccnc(Br)c1Br 87003,C(CCCC(=O)N1CCC(F)(CNC(c2cc(C(C)(C)C)no2)=O)C1)OCC 87004,N1(C(COC(CC)C)=O)CC2(C1)OC1(C)CC2(NC(=O)C(c2ccccc2)F)C1 87005,O=C1CCC(O)CN1CCC(=O)N(C1CC1)Cc1cn(CC2COCCO2)nn1 87006,C(C(CC(=O)N1CCC(N2CCC2)C1)NC(C1CCC(C)(C)C1)=O)OC 87007,C1(O)(C(C)NC(CCN(CCC)C)=O)CCN(C(=O)CNC(=O)C(F)(F)F)C1 87008,Cn1cnc2c1CCNC2C(=O)NC12CCC(CN=[N+]=[N-])(CC1)CO2 87009,C1(NC(CC2(C#N)CC2)=O)CC(O)CN(C(=O)Cc2csc(C3CC3)n2)C1 87010,N1(C(CCCCOCCC=C)=O)CCC2CN(C(=O)CC(COC)C(F)F)C2C1 87011,C(=O)(C(CCS(C)(=O)=O)c1ccccc1)N(C(C(C)O)(C)C)CC(F)F 87012,C1(NC(C2(C)C=CCN2C(C2CN(C3COC3)C2)=O)=O)(CO)CC2CCCC12 87013,C1(CNC(c2c(CC)oc(C)c2)=O)CCCC2CN(C(c3sccc3Cl)=O)CC12 87014,CC(C)CC(O)C(=O)NCC1(F)CCCN(C(=O)C(N2CCCCCC2=O)C)C1 87015,Cc1ccc(O)cc1C(=O)NC1CCC(CCC(=O)NC2CCCCC2(C)O)C1 87016,C#CCCCC(C)C(=O)N1CC2CCC(CNC(c3cc(C)n(CC)n3)=O)(C2)C1 87017,N1(C(CNc2cncc(C(N)=O)c2)=O)CCC(NC(c2ccoc2Cl)=O)C12CC2 87018,N1(C(c2cc(C)no2)=O)CCC(C)(CC(=O)NC2CC(N3CCC3)C2)C1 87019,N1(C(C(Br)=C(C)C)=O)CC2CCC(NC(=O)Cc3cccc(F)c3F)CC2C1 87020,c1(C(=O)NC(C2CCCCN2C(=O)Cc2ccccc2)C)cc2c[nH]cnc-2n1 87021,c1(C(CNC(c2cn(C3C(OC)COC3)nn2)=O)F)cc(F)cc(Br)c1 87022,C(=O)(C1CCCc2nccn21)N1CCC(CNC(c2ccc(CC)cc2)=O)CC1 87023,N1(C(CC=CC)=O)CCC2CCC12CNC(c1c(O)cccc1Cl)=O 87024,C(CCCC(=O)NCC(C)(Cn1cccn1)NC(=O)CCF)SC 87025,C(=O)(CCCCCCC)NCc1cc(C(N2C(C=C)CCC2)=O)sc1 87026,c1(SC)cn(C)nc1C(N1CC(F)CC1CN(C)C(C1CCOC1)=O)=O 87027,C=CC(C)(CC)C(=O)NCc1csc(CNC(c2[nH]c(C3CC3)nc2C)=O)n1 87028,N1(CCOC)CC(C(=O)NC2CCCC2NC(C23CC(CCO2)C3)=O)CCC1=O 87029,C1(NC(CC2N(C)CCC2)=O)CCC2(CC1)CN(C(=O)CC1CC3(CC3)CO1)C2 87030,C1(C(N(C2CCCN(C(CCn3ccc(C)n3)=O)C2)C)=O)CN2CCC1(C)CC2 87031,Cc1oc(C#N)cc1C(=O)NCC1(C)CCN(C(C2CCCCC2(C)C)=O)CC1 87032,C(=O)(C(C(C)C)NC(N)=O)N(CCCN(C(C(C)=CC)=O)C)C 87033,c1(C(N2C(COC)(CNC(C3CC4(CSC4)C3)=O)CCC2)=O)cc(C)ncc1Cl 87034,N1(C(c2n(CC)ccc2)=O)CCC2CC1CN2C(=O)CC(C)SC 87035,C(CCC(=O)NC(c1cn(C)nn1)C(=O)NCc1ccn(CC)n1)=CC 87036,N1(C(CCCOCC)=O)CCN(C(c2ccc(C)cn2)=O)C2CC12 87037,N1(C(=O)NC(c2[nH]nnc2C)CC)CCSCC1c1ccccc1 87038,C1(C(N(C)CC2CN(C(=O)C(O)c3ccsc3)C2)=O)CCCN1C1CCCCC1 87039,[N-]=[N+]=NC1CCC2(C(=O)NCc3cnc4ncccn34)CC12 87040,c1(C(=O)OC2C=CS(=O)(=O)C2)cc2cc(Cl)ccc2[nH]1 87041,N1(C(c2c(C)[nH]nc2C(F)(F)F)=O)CCN(C(=O)Cc2cc[nH]n2)C(C(F)F)C1 87042,C1(NC(c2cccc(-c3nnc(C)o3)c2)=O)CCCCCN(C(=O)C2CC2)C1 87043,c1(OC)ccc(C2(C(N3CCC(Oc4ccnc(C)n4)CC3)=O)CC2)nc1 87044,CC(C(=O)NCC1CC(NC(=O)Cc2cccs2)CCO1)C(F)(F)F 87045,C(=O)(C(C)S(C)(=O)=O)NCCC1CCCN(C(CC(C)c2ccccc2)=O)C1 87046,C#CCC(CC(=O)OC)NC(=O)CC(CCC)NC(=O)C1=C(Cl)CC1 87047,C1(CC(N2CCC(NC(C3(F)CCOC3)=O)C(CO)C2)=O)CN2CCN1CC2 87048,c1(C(N2CCN(C(C3CC(C#C)(O)C3)=O)CC2)=O)cc(Cl)c(Cl)n1C 87049,c1(OC)c(C(N2CC3CCN(c4ncncc4Br)C3C2)=O)cccc1[N+](=O)[O-] 87050,c1(C(=O)NCC(CN(C(=O)CC23COC(C)(C2)C3)C)O)c(N)cccc1Cl 87051,S(=O)(=O)(c1ccc(CNC(=O)C(=O)Nn2c(O)nc3ccccc23)cn1)N(C)C 87052,CC1=NNC(=O)C1CCC(=O)N1CCC1CC(=O)NOCC(C)(C)C 87053,N1(C(C2=NNC(=O)C2)=O)CC2(CCC2)CC1CNC(C1CC1C(F)F)=O 87054,C(C(=O)NNC(=O)C#CCN)C1Oc2c(OC)cccc2S1(=O)=O 87055,C1(CNC(c2cn(C)nc2)=O)CC2CCCCC2N1C(=O)Cc1nnc(O)s1 87056,C1(C(N2CC(O)(CCNC(C3(OC)CCSCC3)=O)C2)=O)CCN(C)S1(=O)=O 87057,c1(C(=O)NC2CC(C(=O)C)C2)cnc(NC2CC2C(=O)N)cn1.C(C(F)F)OC1CC1 87058,C#CCCN=C(NCC(C(C)(C)C)OCCO)N1CCC(N2CCCC2)C1 87059,Cc1n[nH]c2cc(C(=O)NC(CNC(=O)CCC3CCCO3)C(C)C)ncc12 87060,C(=O)(C(=O)N(C)C)N(C(CNC(C1(CC(C)C)CC1)=O)C)C 87061,c12ccc(cc1)s2.c1(CCN(CC=C)C)ccon1.C1CC(=O)N1C 87062,N1(C(c2ncoc2C(F)(F)F)=O)C2CCCC1CC(NC(C1(O)CCCC1)=O)C2 87063,C(C)(C)(CCC(=O)NC1CC(C)CCC1O)NC(c1ncn(CC)c1)=O 87064,C1(C(C)C)CN(C(=O)C2=NNC(=O)C2)CCCN1C(c1coc(C(C)(C)C)n1)=O 87065,Cc1ccc2c(C(=O)NC(C)CCCNC(C3CC(F)C(=O)N3)=O)c[nH]c2c1 87066,c1(C(=O)NC2C(NC(C(CC)OCC)=O)C2)ccc(-n2cccc2)nc1 87067,C#CC(CNC(=O)C(C(C)(C)C)n1cc(C2(O)CCCC2)nn1)CC(C)(C)C 87068,C(=O)(C(C)S(N)(=O)=O)NCC1(O)CC(NC(c2c(C)ccn2C)=O)C1 87069,n1(CC(=O)N(CCCCN(C(c2cnc(C)s2)=O)C)C)ncc2ncccc12 87070,N1(C(C2C(C)C2C)=O)CCN(CC2CCCN(C(C3CC(F)(F)C3)=O)C2)CC1 87071,CC(C(=O)N1CCCCO1)C1CCCN1C(c1cccn1C)=O 87072,c1(C(N(C2CC(NC(C3CCCCS3)=O)C2)CCC)=O)cccn2cc(C)nc12 87073,c1(C(=O)NC2CCCCN(C(CC(CC)SC)=O)C2)ccnc2c(F)cccc12 87074,N1(C(C(C)(C)CCl)=O)CCC2(CCC(N3CC(F)C(F)C3)O2)CC1 87075,N1(C(c2cc(Cl)on2)=O)CCCC2(CCN(S(=O)(=O)c3cnc(Cl)c(Cl)c3)C2)C1 87076,CCC(COC)C(=O)NCCC(C)N(C(=O)CC1CC=CCC1)C 87077,C1(O)(C(C)NC(=O)C=CC(=O)N(C)C)CCN(C(C2CC(=O)CO2)=O)CC1 87078,O(C1CCc2c(Br)cccc21)C(c1ccc(C2CCC2)cc1)=O 87079,C1(C(=O)NC2CCN(C(N)=O)C2)CC2(CCN1C(=O)COC1CCCOC1)CC2 87080,C(c1c(F)ccc(Cl)c1F)=CC(N1CCC(NC(C(C)=C(C)C)=O)C1C1CC1)=O 87081,c1(C(N2C(C(=O)Nc3ncccn3)CC3CC32)=O)ccc2nccc(Cl)c2c1 87082,N12CCOC(C)C1NC2=O.C(CCF)OCC 87083,CCC(CCC(=O)N1CCC(C)(N(C)C)C1)NC(=O)C(c1ccnn1C)C 87084,C(=O)(C#CC1CCCCO1)NC1(C)CN(C(c2c(C)c(N)cc(O)c2)=O)C1 87085,Cc1nccc(CN(C)CC2CCCCN2C(c2nc(Cl)oc2C)=O)n1 87086,C1(NC(C(C=CC)O)=O)CC12CCN(C(c1ccc(Cl)c(C)c1)=O)CC2 87087,c1(C(=O)NCCN(C(=O)CCc2cnoc2)CC(C)O)cccc2ccccc12 87088,C=CCCC(C(=O)NCCCS(C)=O)NC(=O)Cc1cccs1 87089,Cc1cncc([N+](=O)[O-])c1N1CCC(NC(=O)CCc2cccnc2C)C(O)C1 87090,C12(C(=O)NC(C3CCCO3)CC)CCC(NC(=O)CCc3cn(C)cn3)(CC1)C2 87091,N1(CC=O)CCCC2(CCc3ccccc3O2)C1.CC1C(C(F)(F)F)CCCN1 87092,C(=O)(CC(C(F)(F)F)S(=O)(=O)NC(c1cccc(Cl)c1F)CO)OCC 87093,CC(CC(C)(F)F)C(=O)OCC1OCCCO1 87094,N1(C(CCc2cc(C)no2)=O)CC2CCC(C1)N2C(c1cc(C)c(Cl)cc1C)=O 87095,N1(C(CC(C)=C(C)C)=O)CCC2(CC2C(=O)Nc2ccc(O)c(Cl)c2)C1 87096,C12(C(=O)NCCn3c(C)nnc3)CCC(CC1NC(C1CC3(C1)CC(O)C3)=O)C2 87097,c1(C(N2C(CNC(=O)C3=COCCC3)CC(C)(C)C2)=O)ccc2c(c1F)CCC2 87098,C(=O)(CCCCN(C)C(c1ncccc1Cl)=O)NCC(CC1CC1)OC 87099,C(C(=O)N(CCC(=O)N(C)CCn1ccnc1)CCCO)(C(C)C)NC(C)=O 87100,c1(C(=O)NC(CN(C(C2CC(=C)C2)=O)C)(C)C)cc(CC)nnc1C 87101,c1(N)c[nH]nc1C(=O)NC1C(NC(C2(C(N)=O)CC2)=O)CC1.C(N)=O 87102,C#Cc1ccc(CC(=O)NC2CC3C2CCN3C(=O)C(=O)CC(C)C)cc1 87103,CS(C)(=O)=Nc1ccc(C(N2CCN(C(=O)CC3CC3(Cl)Cl)C(CF)C2)=O)cc1 87104,Cc1nc(C(=O)NC2(CCC(=O)N(CCCC(C)O)C)CCC2)c(C)o1 87105,c1(NC(C2CN(Cc3ncc(Br)cc3Br)C2)=O)ncnc2occc12 87106,c1(CC)ncncc1C(=O)NC(C1CCN(C(=O)CCc2cccnc2)C1)C 87107,C(C(C)C(F)C(=O)Nc1cn(C)nc1C#N)NC(c1ccnc(OC)n1)=O 87108,c1(C(=O)OC)ccnc(NC(C2CCCC(NC(c3cscc3C)=O)C2)=O)c1 87109,C12(C(N3C(C)(C(=O)NC)CC3)=O)C(NC(=O)C(C)C#N)C3CC1C2C3 87110,C1(NC(C2(C)CC=CCC2)=O)CN(C(c2cc(Cl)cnn2)=O)CCC1F 87111,C1(NC(c2c(C)scc2)=O)CCN(C(C2CCOC3(CCC3)C2)=O)CC1(C)C 87112,c1(C(OCC)OCC)ccccc1C(=O)NC(c1cn(C(C)C(=O)O)nn1)C 87113,Cn1nccc(C(=O)NC2CN(C(=O)Cn3nccn3)CC2O)c1=O 87114,N1(C(=O)C=Cc2ccccc2)CC(Nc2ncc(Br)cn2)CC(F)C1 87115,N1(C(c2nc(C)n(C)c2)=O)C2CCCC1CN(C(=O)CC1CCCC(C)C1)C2 87116,c1(NC(c2ccc(SC(F)F)cc2)c2n(CC)nnn2)c(CO)cccc1Cl 87117,C1(C)(C(=O)NCC(=C)CCNC(c2cc[nH]c2C(=O)OC)=O)CC(O)CN1C 87118,C1(c2n(CCSC)nnn2)(NCc2c(C)ncn2C)CCC(c2nc(C)no2)C1 87119,C12(C(N3CCCCC(NC(CC4N(C)CCC4)=O)C3)=O)CCC(CO)(CC1)CC2 87120,N1(C(C2N(CCCC)CCCC2)=O)CCC(C)(C)C(C(=O)N(C)C)C1 87121,C(C(C(=O)NC(c1nn(C)cc1O)C)C(C)(C)C)NC(C(C(=O)OCC)(C)C)=O 87122,c1(CNc2cc(C(N3C(C(=O)OCC)CC(O)C3)=O)no2)ccc(O)cc1O 87123,c1(CC)cccc(NC(=O)COC2CCN(C(c3c(Cl)cnn3C)=O)C2)c1F 87124,[N-]=[N+]=NC1CN(C(=O)CC2CC(=O)NC2=O)CC1NC(=O)Cc1cncnc1O 87125,N1(C(CCOCC)=O)CCN(C(c2cccc(C(F)(F)F)n2)=O)C(C)C1 87126,CC1(C)CCCC(CC(N2CCN(C(c3ccnc(S)c3)=O)CC2C2CCC2)=O)O1 87127,c1(C(=O)NC(C2N(C(CC(C)C(F)(F)F)=O)CCC2)C)c2c(nn1C)CCCC2 87128,C1(F)(C(=O)NC(c2cn(C)nc2)CO)CCN(C(c2cnn(C(F)F)c2)=O)C1 87129,c1(CC)nc(O)c(C(N2CCC3(NC(=O)CC4CCSCC4)CC3C2)=O)cc1C 87130,N1(C(CCC(CC)CC)=O)CCCCC2(C1)CN(C(c1cnnn1C)=O)C2 87131,C1(NC(C(CN(C)C)(C)C)=O)CC2(CCCN(C(=O)C=Cc3cccnc3)C2)C1 87132,Cc1scc(C(=O)NCC2CN(C(C3(Cl)CC3(F)F)=O)CC2O)c1N 87133,C(=O)(C(CNC(=O)CN1CCCCC1=O)(CC)CC)NC(C#C)C(C)(C)C 87134,C1(N(C(=O)CCOCC(F)F)C)CCCCN(C(=O)Cc2cnc[nH]2)C1 87135,Cc1nc(N)cnc1C(=O)NCCNC(=O)CC(C)NC(c1ccccc1)=O 87136,C1(NC(c2cnn(C)c2F)=O)CN(C(C2C3COCC23)=O)CC2(CCC2)C1 87137,c1(C(C)C)cc(N2CCC(NC(=O)C3=CCCCC3)C(C)C2)n2ncnc2n1 87138,CC(C)CCCC(C)C(=O)N1CC(CCNC(c2scnc2Cl)=O)C(C)C1 87139,C(CCCCC(=O)NCCCNC(=O)CCC(=O)Nc1cc(CO)n(C)n1)SC 87140,C1(CN(C(C(C)OCCC(C)C)=O)C)CN(C(=O)CC=CC(C)(C)C)CCO1 87141,CC1CCN(C(=O)CC(C2CC2)NC(=O)CS(C)(=O)=O)CCS1 87142,C1(NC(=O)Cc2ccc(O)cn2)CC2CN(C(C3C(F)(F)C34CCC4)=O)CC12 87143,c1(C(N2CCC(C(=O)Nc3c(C)cc(O)cc3)C2)=O)c(F)c(F)c(O)c(F)c1F 87144,C1(NC(CN2C(C)CCC2)=O)CCC2(CC1)CC2NC(C1C2CC3C(C2=O)C13)=O 87145,c1(C(=O)NCCCC(C)(C)NC(CCC#CC)=O)ccc(N)c(Br)n1 87146,N1(C(C(C#C)(C)C)=O)CCOCC(C)(CNC(C2CCC3CCC2O3)=O)C1 87147,c1(C(=O)NC2CCC(F)(CNC(CC3ON=C(C)C3)=O)C2)ccc(F)cc1Cl 87148,c1(NC2CC(NC(=O)OC(C)(C)C)C2(C)C)c(C(=O)O)cc(Br)cc1C#N 87149,N1(C(C)C)CC(C(=O)N(CCCN(C)C)CCNC(C2(C)CCOC2)=O)CC1=O 87150,N1(CC(COCC)O)CCCCC1CC.N12CCCCC1C1CCC(CC1)C2=O 87151,C(CN=c1[nH]c(=NCCC2CCCCO2)[nH]c2cc[nH]c12)c1ccc(SC)cc1 87152,c1(C(N2CC(CNC(=O)Cc3cccc(Br)c3)C2)=O)cc(F)c(Cl)c(Cl)c1 87153,N1(C(CC(c2nc(C(=O)Nn3ccnn3)co2)C)=O)CCCC[Si](C)(C)C1 87154,CCCCN=C(NCc1c(C)cccc1F)NCC1(CO)COC1 87155,c1(C(=O)NCC2CCCCN2C(c2n[nH]cc2F)=O)c[nH]cc(Br)c1=O 87156,N1(C(CC(C(F)F)NC(c2cc(C)c(F)cc2)=O)=O)CCC2CCCC2CC1 87157,Nc1sc2c(c1C(N1CCC3(NC(=O)CCCC4CC4)CCCC13)=O)CCC2 87158,[N-]=[N+]=NCCCCCC(=O)N1CCOC(C2CN(C(=O)C3=NOCC3)C2)C1 87159,c1(C(=O)NCC2C3N(C(C4C(CCC)C4)=O)C(CC3)C2)ccc2oc(O)nc2c1 87160,c1(CC=C)ccccc1C(N1CCC(CNC(=O)C(C)n2cncn2)(OC)C1)=O 87161,C1(NC(=O)C=CC(F)(F)F)CCCCC12CCN(C(=O)C=Cc1cccs1)C2 87162,c1(OCCC)ccc(C(N2CCCC2C(C)NC(=O)CC2CN(C)C2)=O)cc1 87163,C(=O)(CCC=CBr)NCC1N(C(CCc2ccc(C3C(C)C3)s2)=O)CC1 87164,Cc1nc(C(=O)NCCCN2CCN(C(=O)COC3CCCC3)CC2)c(C)s1 87165,N1(C(c2cc(C)c(Cl)s2)=O)CC2CC1CN2C(C1CC(C2CC2)=NO1)=O 87166,N1(C(C2CC(=O)C2)=O)CC(C2CC2)(C(=O)NC2C3C=CC(C3)C2CO)C1 87167,c1(CNC(CN2C(C)(C(=O)OC)COCC2)=O)c(F)ccc(Br)c1F 87168,c1(C(N(CCCCNC(C2CCC2)=O)C)=O)csc(C2CC2)c1 87169,N1(C(CCn2ccc(C)n2)=O)CCCC(NC(c2nnc(O)cc2C)=O)CC1 87170,C(C1=CCN(C(c2cc[nH]c2C2CCC2)=O)CC1)NC(C(F)OC)=O 87171,c1(COC(CC2(NC(c3nnnn3CCOC)CCC)CC=CC2)=O)ccccc1 87172,C1(F)(CNC(C(C)OCC=C)=O)CCN(C(c2cccs2)=O)CC1 87173,N1(C(C2N(C(CCC)=O)CCCC2)=O)CC2(CCCCN(C(=O)C(C)CO)C2)C1 87174,C1(NCC(c2ccc(F)c(F)c2)C(C)C)CC2CCC1C(N)C2 87175,C(=O)(CC(O)CC(C)(C)C)NCC(=O)NCC(=O)NCCCOCC=C 87176,C1(CNC(C(C)c2cn[nH]c2)=O)CC(O)CN1C(=O)CCc1cc(Cl)no1 87177,N1(C(C2N(C(CC(C(CC)C)O)=O)CCN(C)C2)=O)CCC2CN(C)CC2C1 87178,C(=O)(CCCCCOC)N1CC(CCC)C(C(N2CCCCC2C2CCC2)=O)C1 87179,c1(NC(CCC)CCCNC(=O)Cn2cnnn2)c([N+](=O)[O-])c(CC)nn1C 87180,CC1(CC(N2CC(O)(CCNC(=O)C(N)=O)C2)=O)CC1(F)F 87181,N1(C(CN(C)S(N)(=O)=O)=O)CCC2(CC1)CC2NC(=O)CCSc1nccn1C 87182,N1(CC(CC(=O)OC)Sc2noc(C3CC3)n2)CCCN(C(=O)OC)CC1 87183,C1(CNC(CN(C)C(c2ccccc2)=O)=O)CCCCC1NC(=O)CC(F)F 87184,c1(OCCN(C)C)ccc(CC(N2CCC(CN(C3CC=CC3)C)CC2)=O)cc1 87185,CC(C)(CCC(=O)NC1(CNC(=O)C(O)(C2CC2)C2CC2)CC1)[N+](=O)[O-] 87186,CC(CC(=O)NC1CCN(C(C2CC(F)(CO)C2)=O)C1(C)C)C(F)F 87187,c1(C(C(=O)N2CC(CC(C)(C)C)C2)NC(CCOCC)=O)cnn(C)c1 87188,C12(NC(c3c[nH]c(=O)cn3)=O)CCC1CN(C(=O)COC1CCCCCC1)C2 87189,c1(C(=O)NC2(C)CCCN(C(c3c(OC)c(C)sc3)=O)C2)cc2ccncn2c1 87190,N1(c2cn(C)nc2)CCCC(N2CC(CC3CCCCC3)C2(C)C)C1=O 87191,C(CN=c1cc(C)nc(C)[nH]1)C1(O)CCN(C(C=CC=CC=CC)=O)CC1 87192,c1(-n2ncc(CNCC(C=C)O)c2)ccc(C)cc1 87193,CC1c2ccc(F)cc2CCN1CC(=O)N(c1cccc([N+](=O)[O-])c1)c1cncs1 87194,c1(C(c2n(CCCSC)nnn2)NCC2(OC(C)C)CCSC2)c(OC)ncnc1Cl 87195,CC(CC(C)NC(C1CCCN1c1cnccn1)=O)NC(=O)C(C)(C)C 87196,c1(C(N2C(C(CNC(CC3CC(=C)C3)=O)(C)C)CCC2)=O)nn(C)cc1NC 87197,c1(C(=O)NCCC(=O)NC(CC)C)c[nH]nc1CCNC(=O)CC1CC1 87198,C1(C(=O)NC(c2ccccc2)CC)CC2(CCC2)CN1C(=O)C(CO)C(F)(F)F 87199,C1(C(=O)NCC2(F)CN(C(C(N3CCCCC3)C)=O)C2)CCC(=O)NC1 87200,C1(C2CCCN(C(=O)C(C)(C)CC#N)C2)(NC(C(c2ccccc2)C)=O)CC1 87201,CC1CN(C(=O)CCC2CC(NC(C3C4CCC(=O)C34)=O)C2)c2cccnc21 87202,C(=O)(C(CNC(C1CNC(=O)C1)=O)CC1CC1)N(CC(C1CCC1)OC)C 87203,c1(C(=O)NC(CC)CN(C)C(C2(CCF)CC2)=O)cc(C)c(Cl)c(C)c1 87204,CC(CNC(c1ccc(O)cn1)=O)C(F)C(=O)NCCc1cccnc1F 87205,N1(Cc2c(OC)nccc2)CC2CC1CN2C(c1ccc(O)c(F)c1)=O 87206,c1(COC)nc(N2CCCC(NC(=O)Cn3cc(C(C)O)nn3)CC2)cc(O)n1 87207,c1(C(C)NC(C(CC)NC(c2ccccc2)=O)=O)cc2ccccc2s1 87208,C1(C(N2CCN(C(c3c(C)ccs3)=O)CC2C)=O)CC2CC1C1C2C1(F)F 87209,C1(CC(=O)NCCC2(O)CN(C(COCC=C)=O)C2)CCOC(C)(C)C1 87210,C1(C(=O)NC(C=C)C2CC2)CN(C(=O)C(CC)=CCOC)CCC1(C)C 87211,c1(C(N(C2CN(C(c3cc(Cl)cnn3)=O)C2)C)=O)cncc2nc[nH]c12 87212,CN1CC2(CN(C(=O)NC3CC3c3cccc(OC(F)(F)F)c3)C2)OC1=O 87213,C1(NC(NC(C=C)C)=NCC2CC(=O)N(c3ccccc3)C2)CCOC(C)(C)C1 87214,CON(CCCO)C(=O)C1(CO)CCCN(C(c2cnnc(C)c2)=O)C1 87215,C1(CCCNC(C2(CSC)CC2)=O)CCCN1C(=O)C=CC1CC1 87216,CC1CN(C(C2CCC(C)(C)CC2)=O)CC1(C)C(N1CC(C)(F)C1)=O 87217,c1(NC(C(CC)NC(=O)CC(F)(F)F)=O)ccc(OC)cc1Br 87218,C=C(C)C1CCC(C)(O)C(NC(=O)NCc2cccc(Br)c2Cl)C1 87219,c1(CC)oc(C(=O)NC2(C(=O)NCCCN3CCC(O)C3)CCN(C)C2)cc1C 87220,C1(CC)CCN(C(=O)CCC2(C)CC2)C1C(=O)N(CC(C)(C)COC)C 87221,c1(NC(C(C)Cc2ccnn2C)=O)ncccc1OCC(F)F 87222,c1(C(=O)NC23CN(C(CC=C)=O)C(C2)C3)cc(C#N)c(O)nc1N 87223,C1(N(CC#C)C(=O)OCC)CCN(C(=O)C(C)Cc2ccccc2)CC1 87224,N1(C(CC=CC=C)=O)CC2CC1CC2NC(C1(Cn2cccn2)CCCC1)=O 87225,C1(CN(C)C(c2sc(F)cc2Cl)=O)CN(C(=O)Cc2cncs2)CCO1 87226,N1(C(C2CC(CC)(CC)C2)=O)CC(C(=O)NC2CCCC2O)CCC1C 87227,C1(C)(OC)CCCN(C(=O)CC=CCNC(=O)C2=C(C)OCC2)CC1 87228,Cc1c(C(=O)NCC2COCCN2C(=O)Cn2cc(Br)cn2)cncc1Br 87229,C1(CC)CN(C(c2cocc2C)=O)CCC1NC(C1(C)CC=CC1)=O 87230,c1(C(N2CCC(F)(CNC(C(CC)OCC)=O)C2)=O)cccc(S(N)(=O)=O)c1 87231,C(=O)(CCCCN(C(=O)C(C)(F)c1ccon1)C)NC(c1cc[nH]n1)C 87232,c1(OC)ccc(CCC(=O)N(C2CN(C(=O)CC3CC(C)C3)C2)C)cn1 87233,CC(CC(=O)N(C)CC1(O)CCN(C(=O)C(F)(F)CO)C1)C(F)(F)C(F)(F)F 87234,c1(C(=O)OC)ccc(C=CC(=O)NC2CCCN(C(c3ncncc3Cl)=O)C2)o1 87235,N1(CC2(NC(C=COCC)=O)CC2)CCN(C(=O)C(F)(F)c2ccccn2)CC1 87236,Cc1cc(C(=O)NCC(=C2CN(C(=O)Cc3ccn(C(F)F)n3)C2)F)n(C)n1 87237,C(CO)(CCCCNC(C1(C)COC(=O)OC1)=O)NC(C=COCC)=O 87238,C1(CNC(CC=CC=C)=O)(CNC(=O)CCNC(=O)CC(C)C)CC12CCC2 87239,CC(C)CCCCC(=O)NC1CC1CNC(c1ccnc(OC(C)C)c1)=O 87240,CC1(C)CC(C(=O)NCC(O)CC(F)(F)F)CCN1C(C1CC(=O)CC(=O)N1)=O 87241,Cc1cc(NC(=O)C(=O)NCc2ccc(=N)[nH]c2)ccc1Br 87242,c1(C(=O)NCCOC2CN(C(=O)CCOC3CCC3)C2)nnc2ccccc2n1 87243,C12(C(=O)NCC#CCNC(Cc3cc(C(C)C)no3)=O)CCCC1CC2 87244,c1(C(N2CCC(OC)(CN)C2)=O)c2c(nn1C)CCS(=O)(=O)C2 87245,CCCC(C)C(CC)(c1nnnn1CC)NCC1(c2ccc(OC)cc2)CC1 87246,N1(C(C=C(CC)CC)=O)CCC2CN(C(c3cn4cccnc4n3)=O)CC12 87247,c1(C(N2CCC(N(C(c3cncc(SCC)n3)=O)CC)C2)=O)ccc(C)nc1O 87248,c1(CC(=O)NC(c2cccc(OC)n2)C(C)C)ccc(S(C)(=O)=O)c(C(=O)O)c1 87249,CS(=O)(=O)CC(=O)NC1CCCCC1NC(=O)CNC(=O)C(F)(F)F 87250,C12(CNC(c3n(C)cnc3)=O)COCCN1CCN(C(c1cnsc1)=O)C2 87251,CCC(C)CCCCC(=O)N1CC2(C1)CN(C(=O)CN1CCCS1(=O)=O)C2 87252,c1(C(=O)NC(c2nnc(Cc3ccccc3)o2)C)ccoc1C1CC1 87253,N1(C(c2cc(C3(C)CC3)on2)=O)CCCC(C2CC2NC(=O)CCP(C)(C)=O)C1 87254,C1(NC(C2CCC(=O)S2)=O)CCc2nncn2C1 87255,C(=O)(C(C)(F)C(=O)NC(CO)C(C)NC(c1ccnc(C(C)(C)C)c1)=O)OC 87256,N1(C(C2C(C(C)C)CCC2)=O)CCCC(C)(C)C1C(=O)NC1CCC2(CCC2)C1 87257,c1(C(=O)NC(C2CCN(Cc3cccnc3Br)CC2)C)cc(Cl)cnc1Br 87258,C1(C(=O)NC(C(C)(C2CC2)OC)C)C=CCCN1C(=O)CCCNC(=O)OC 87259,N1(C(CC=CC=C)=O)CC(C2CC2)(C(=O)NCC2CC(C)C2)C1 87260,Cc1ccc2c(c1)C(C(=O)NC(CNC(=O)Cn1cc(C(N)=O)nn1)C(C)C)C2 87261,c1(OC)ncccc1CC(N1CCCC1C(C)NC(C1CCN(C)CC1)=O)=O 87262,C(=O)(NNc1ncc(Br)cn1)C(C)(C)C.C12CC3(CCC(O3)CNC(=O)N1)C2 87263,C1(C(N(CC(=O)NCCCC2CCCO2)CCOC)=O)CCCN1C 87264,C12(NC(c3nc(CNC(C45COCC4C5(F)F)=O)cs3)=O)CCC(CC1O)C2 87265,N#CCCCC(=O)NC1CCN(C(=O)COc2ccc(Cl)cc2)C1 87266,c1(CC(N2CC(CNC(C3(C)CC(C#N)C3)=O)C2)=O)ncn2c1CCCC2 87267,c1(CNC(c2cc(CC)[nH]n2)=O)nnn(C)c1C(=O)NC1(C(=O)OC)CC1C 87268,C=CC1(C(N2C3C=CCC2CC3)=O)CCN(C(=O)CC(C)COC(C)=O)C1 87269,c1(CC(=O)NCCCCCNC(c2sccc2F)=O)ccc2n[nH]cc2c1 87270,C1(NC(c2cc(Cl)c[nH]2)=O)CC2CCC1N(C(c1ccc(C3CC3)cc1)=O)C2 87271,C(CCCCCO)NC(CC(C)N(C(CN1CCC(C)C1)=O)C)=O 87272,C(=O)(C(C)C(C)c1ccc(F)cc1)NC(C1(O)CN(C(c2cccs2)=O)C1)C 87273,CN1CCOC(CC(=O)NC(CCN(C)C(c2ccco2)=O)c2cccs2)C1 87274,Cc1cc(S(=O)(=O)NC(C2COC3CNCC23)=O)c(Cl)cc1F 87275,N1(C(C#CC2(CC)CC2)=O)CCCN(C(c2cccc(C3(C)CC3)c2)=O)C(C)C1 87276,C12(C(=O)NC(C#C)CC)CCC(NC(C3CC34CCOCC4)=O)(CC1)C2 87277,Cc1cc(Cl)cc(C(=O)NC2CC2CNC(c2cncc(O)c2Cl)=O)c1C 87278,CN1CCOC(C(=O)NCC(O)CCNC(c2cnccn2)=O)C1=O 87279,c1(CC)ccsc1C(=O)NCC1CCC1NC(c1cncn1-c1ccccc1)=O 87280,Cc1ncc(N)cc1C(N1CC(C(C)NC(c2nc(Cl)c(Cl)s2)=O)C1)=O 87281,c1(C(N(CCCCNC(C(CC)C(C)(F)F)=O)C)=O)noc2c1CC(C)CC2 87282,c1(C(N2C(CC)CN(C(=O)CC(C)F)CC2)=O)cnc2scc(C)n2c1=O 87283,c1(C(C(=O)NCC(C(C)C)NC(=O)C(=O)NCC(F)(F)F)C)cncc(F)c1 87284,c1(CC(N2CCC(C(C)NC(c3nc(C)sc3)=O)C2)=O)ccc2c(c1)ncn2C 87285,c1(OC)cc(SC(c2nc[nH]n2)=O)cc(OCC(N2CC(CN)C2)=O)c1OC 87286,C(=O)(C(C)(C)C(N)=O)NCC(N1C(C)C(=O)N(CCN)C1)=O 87287,CN1CCN(C(=O)C(O)CCC2CC2)CC1CNC(C1(N2CCCC2)CC1)=O 87288,c1(SCC(=O)NC2CCN(C(CC(CCC)C)=O)C23CC3)nnc2ccccn12 87289,c1(C(=O)NCCN(C(=O)C(C2CCC(=O)N2)C)C(C)C)ncc(F)cn1 87290,Cc1cc(=O)n(CC(=O)NC(C2CCC(C)(C)CC2)C(N)=O)cn1 87291,C1(NC(C=CCC)=O)CCC12CN(C(=O)C(CC)NC(=O)OC(C)(C)C)C2 87292,N1(C(c2c(COC)n(C)nc2)=O)CCCN(C)C(=O)C1 87293,Cc1ccc(C(C)C(=O)N(C2CCN(C(=O)CC(O)C3CCCC3)C2)C)s1 87294,N1(C(C(F)=CCC)=O)Cc2occ(C(=O)NC3CN(C)CC3OC)c2C1 87295,C#CCCCC(C)C(=O)N(CCN(C)C(C1(C)COC(C)(C)CO1)=O)C(C)C 87296,C(CCCCCNC(C1CCC(C#N)C1)=O)NC(c1cc(C)sn1)=O 87297,n1(C(C)(C)C)ncnc1CNC(=O)NCC1CCCCS1 87298,CC1CN(C(=O)C=Cc2ccncc2)CC(C(=O)NCc2ccon2)O1 87299,c1(C(c2n(CC(=C)C)nnn2)NCC2(OCC)CC=CC2)ccnn1C=C 87300,Cn1nc(CNC(=NCc2ccccc2-n2ccnc2)NC2CC2)cc1Cl 87301,CN1CCCCC(C(=O)N(C)CCN(C)C(c2cn(CC(F)(F)F)cn2)=O)C1=O 87302,C(=O)(CCCCN1CCCC1)N1CC(OCCNC(C(C)CC2CCCO2)=O)C1 87303,c1(C(N2CCC(O)(CN(C(C3C(CC)N(C)CC3)=O)C)C2)=O)cc(O)ccc1C 87304,N1(C(c2c(Cl)ccc(C#C)c2)=O)CCCC2(NC(=O)Cn3ccc(C)n3)CC2C1 87305,Cc1cc(C)n(C(C)CC(=O)N(C)CC2CCN(C(c3ccc(F)o3)=O)C2)n1 87306,C1(NC(C(C)C(F)F)=O)C2CC3C1C3C2C(=O)Nc1cc(O)cc(F)c1 87307,Nc1c(C(N2CC(NC(=O)C#CC3CCOC3)CC(F)(F)C2)=O)ccc(Cl)c1Cl 87308,S(=O)(=O)(c1c[nH]ccc1=NC1COCc2cccnc21)NCC(CC)OC 87309,C1(C(N(CCCCCC)CC(N)=O)=O)CCC(CC2CCCN2C(C)=O)CC1 87310,C(=O)(C(C)(C)C(C)(F)F)N1CC2C(C(N(C3CCC3(C)C)C)=O)C2C1 87311,N1(C(CNC(=O)NC)=O)CCC(C)C(N(C(=O)C(C)(C(C)C)OC)C)C1 87312,C(=O)(C(CC)C(C)(C)CC)N1CCCC(N(C(CCCC(=C)C)=O)CC)C1 87313,C(CC(C)C)(C(C(=O)Nc1ccc2c(c1)OCO2)N1CCC(C(N)=O)C1)OC 87314,c1(OC)cc(C)c(C(CNCc2cc(N(C)C)nc(C)n2)(O)c2ccco2)cc1C 87315,S(=O)(=O)(c1ccc(Br)s1)N1C(CNC(=O)C=CCBr)CCCC1 87316,C(=O)(C(CC(C)C)NC(N)=O)NCC(=O)NCC1(CC)CC1 87317,CCCCCC(O)C(C)C(=O)NC1CCCC1NC(c1nncn1C1CC1)=O 87318,CN1CC2C(CCCN2c2nnc(-c3ccc(S(N)(=O)=O)cc3)n2C)C1=O 87319,CC1(C)CCC(C(=O)NC(CCO)C2CC2)CN1C(C1(O)CCCC1)=O 87320,CCC(C)(COC)C(=O)NC1CC1CNC(=O)Cc1nn(C(C)C)cc1Br 87321,C(=O)(C=C1SCC(=O)N1C)NCCC(C)NC(C1CCCCC(=O)N1)=O 87322,C1(CNC(c2c(CC)nccn2)=O)CN(C(C2CCOC(=O)CC2)=O)CCCO1 87323,N1(C(C=C)=O)CCCCC1C(C)(C)CNC(c1ccc(N(C)C)cn1)=O 87324,C1(F)(CNC(C(C)OC)=O)CN(C(=O)CCNC(c2ccsc2)=O)C1 87325,N1(C(=O)Nc2cc(C)on2)CCN(C(=O)C(C)N(C)Cc2ccccc2)CC1 87326,c1(OC)cc(N(C)C)ccc1C(=O)NC(C)CCNC(=O)Cc1cnns1 87327,C1(CNC(C(CCC)OC)=O)COC(C)(C)CN1C(=O)CCc1ccn(C)n1 87328,c1(C(CC)=O)ccc(C(=O)N(CC(C)NC(C23CC2C3)=O)C)cc1 87329,C12CN(CC1(C)C)C2=O.C(c1ccccc1)=C.c1(NC(C)C(=O)N)ccc(Cl)cn1 87330,c1(C(N2CCC(N(C(C3C(C=C)C3)=O)CC)C2)=O)cc(Cl)ncc1N 87331,C=C=CC(C)C(=O)NCc1ccc(CC(C)NC(=O)Cc2csnc2C)cc1 87332,c1(C(=O)NCC)noc2c1CN(C(=O)OC(CC(=O)OC(C)(C)C)C(F)F)CC2 87333,O=C(C1=CCCCCC1)NCc1cc[nH]c1C(=O)NCC1OC(=O)CC1O 87334,CC(C)S(=O)(=O)CC(=O)NC1CCN(C(C2CCCCCS2(=O)=O)=O)CC1O 87335,c1(-c2ccc(CNC(N3CCC(c4nn[nH]n4)(CF)C3)=O)o2)cccc(Cl)c1 87336,Cc1cc(C(=O)N(C2CCCCC2)CCNC(=O)CCCF)cc2c[nH]nc12 87337,c1(C(C2CC2)N(C(c2cccc(C)n2)C)C2CC2)c(F)cccc1F 87338,CC(C)CCCC(=O)N1CCC(NC(=O)C=CC2CCCCC2)C(O)C1 87339,CC(C)C(CCC(=O)N1CCC(C(C)CO)CC1)NC(C1CC2(CSC2)C1)=O 87340,C1(C)(C(N(CC(C)NC(C2(CC#C)CCC2)=O)CC)=O)CCCOC1 87341,N1(C(C)=O)CCCC(CC(=O)NCC(CNC(=O)C(C)(C)C2CC2)CO)CC1 87342,c1(OC)nccc2c(NC(c3c(O)ccc4c3OCC4)=O)cccc12 87343,O=C(CC1NC(=O)c2ccccc21)NCCC1CCN(C(C2SCCS2)=O)C1 87344,C(CCC(C)CC(=O)NCC1(NC(=O)COC(C)(C)C)CC1)=C(C)C 87345,c1(CC)cc(Br)ccc1C(=O)OC(C)C(=O)NC1CC1 87346,N1(C(CNC(CC(c2c(C)n[nH]c2C)C)=O)=O)CCOC(C)(C(F)F)C1 87347,N1(C(C=CSC)=O)CC(NC(=O)Cc2cccc(C#N)c2)CCC1C 87348,CC(CN=c1[nH]cnc2c(Br)c[nH]c12)c1cccc(OC(F)F)n1 87349,N1(C(C(C2CCOC2)NC(Cn2ncc(C)c2)=O)=O)CCCC2(CC1)CC2 87350,C(=O)C1=CC2C=CC(C1)C2.N1(N2CCC(CC)C2COC)CCCC(C)(C=O)C1 87351,C(C)(CCS(C)(=O)=O)NC(=O)Nc1ccc(N(CC)C)nc1 87352,c1(C(=O)NC(CNC(C2CCCSC2)=O)C2CCC2)cccc(OCC(F)F)n1 87353,C(=O)(C1Cc2ccc(F)cc21)NC1(CO)CN(C(CC(C)C2CCCCC2)=O)C1 87354,Cc1cccc2nc(NC(=O)CCC3CCCN3C)[nH]c12 87355,N1(C(c2ccc(F)c(F)c2)=O)C2CCC1CN(C(c1ncsc1Br)=O)C2 87356,N1(C(C)=O)CCC(CC(=O)NCCCN(C(c2cncn2C)=O)C(C)C)C1 87357,C=CCCC(=O)N(CC(C)NC(c1cscc1Cl)=O)CC 87358,C1(C(=O)O)COC2CN(C(c3ccccc3-n3cc(C4CCCC4)nn3)=O)CC12 87359,N1(C(C=C(CCC)CCC)=O)CCCCC(N(C)C(C2C=CCC2)=O)C1 87360,C1(C(=O)NCCC(=O)NC)CCOCC1NC(c1ccc(O)cn1)=O 87361,C#CC1(C(=O)N(CCNC(=O)CC(=O)NCC)CC)CCCC1 87362,c1(OCC(=O)NCCN(C(C2(CC(C)C)CCCC2)=O)C(C)C)cccc(O)c1 87363,Cc1nc2ncnn2c(NC2CC3CC(C2)N(C(=O)CC2CSCCS2)C3)c1C 87364,c1(C(=O)NC2CN(C(C(CCC)N(C)C)=O)CC2O)ncnc2cc[nH]c12 87365,C12(C(=O)NCC3CCN(C(C4CC5(CCOC5)C4)=O)C3)CC3CC1(CO)CC3C2 87366,c1(CC)nc(C(N2CCCC2CNC(=O)C=CCOC)=O)c2ccccn12 87367,CCC(C)C1C(=O)N1.C1(CNC(=O)C(C)OCCOC)CCOC(C)(C)C1 87368,C(CN=C(NC(C)CN(C)C(C)C)N1CCC(c2nncs2)C1)OC.CSC 87369,C1(COC)CC(CNC(=O)C=C2CCSCC2)N(C(C2CSCN2C(C)=O)=O)C1 87370,c1(SC)ccccc1CC(N1CC=CC(NC(=O)C=C(C)C(F)F)C1)=O 87371,C12(CC(F)(F)C1)C(=O)NC2.C1(C(=O)OCC)OCCC1C(F)(F)F 87372,c1(SC)nc(C(F)(F)F)cc(=NCC2CCCCN2Cc2cnco2)[nH]1 87373,C(=O)(C1=C(SC)CCCC1)NCC1CCN(C(c2c(CC)csc2)=O)CC1C 87374,C1(OC)(OC)CCN(C(C)C(N2CCCCCC2)=O)CC1O.c12ccc(Cl)cc1N2 87375,c1(C(N(C2CCCN(C(c3cc(F)n(C)n3)=O)C2)CC)=O)cccc(C#N)c1C 87376,c1(CC)ncc(C(=O)NC2CN(C(C3CCC(C)(C)CO3)=O)CCC2C)c(O)n1 87377,C1(CN(C(C(c2cnccn2)C)=O)C)CCCN(C(c2ccc(=O)oc2)=O)C1 87378,N1(C(C(C)C#N)=O)CCC2(CCC2)C(CNC(c2cc(C(F)(F)F)n(C)n2)=O)C1 87379,Cc1cc(=NC(=O)C2CC(F)CN2S(=O)(=O)Cc2cccc([N+](=O)[O-])c2)cc[nH]1 87380,C1(CNC(C2(C)CCC2)=O)C2CN(C(=O)CCc3cccs3)CC12 87381,C1(C)(NC(CC2CCC(N(C)C(C3CC4CC4C3)=O)CC2)=O)CCC2(CC1)CC2 87382,N1(CC)CCC(NC2CCC(CC(F)(F)F)CC2)CC1 87383,CC1=C(C(=O)N2CC(NC(c3ccc(C(N)=O)c(Cl)c3)=O)C(F)C2)CCO1 87384,C(c1cc(Cl)c2c(c1)OCO2)=CC(N1CCC(C)C(NC(=O)C(C)N(C)C)C1)=O 87385,C(c1ccc(C#N)cc1)=CC(=O)NC1(CNC(C2CC(C)OCC2)=O)CC1 87386,Cc1cc(O)cc(C)c1C(N1CC(F)(CNC(C2(C)CC3CC3C2)=O)C1)=O 87387,C(=O)(C(C)(C)CC(C)C)N1CC(C(N2CCC(C=C)(O)C2)=O)OC(C)C1 87388,C1(OC)CC(NC(C2CCCC(CF)C2)=O)CN(C(=O)COC(F)F)C1 87389,C(N=c1cccc(S(=O)(=O)NCC2(SC)CCC2)[nH]1)c1n(CC)ncc1 87390,N1(C(=O)NC(C2CCOCC2)F)CCC2(CC1)CC2(C)Cn1c(C)ncc1 87391,Cc1cc(Cl)c(C(N2CC(F)(CNC(C3CNC(=O)N3)=O)C2)=O)cc1C 87392,c1(OC)cc(COC(c2cc(C)ccc2N2CCCC2=O)=O)ccc1O 87393,c1(CCCN(CCC)C(N2CCC(c3noc(C)n3)(NC)C2)=O)ccc(Br)cc1 87394,C1(NC(C(CN=[N+]=[N-])NC(=O)C(=O)NC2CC2)=O)CC2(C1)CC21CCC1 87395,CC1(C)CC(c2ccccc2)CN(C(CCc2ccccn2)C(=O)NC2CC2)C1 87396,N1(CC#C)CCN(C(C2CSCN2C(=O)CCc2cnoc2)=O)CC1=O 87397,c1(C2(CNCCC(=O)OC(C3CC(N(C)C)C3)=O)CCC2)cc(Cl)ccc1F 87398,C(=O)(C#CC(C)(C)CNC(=O)C(O)c1ccsc1)NC(c1ccc(C)cc1)C 87399,N1(C(C(C)OCC#C)=O)CCN(C(c2cnn(CC)c2C)=O)C2CS(=O)(=O)CC12 87400,C1(NC(c2cc(OC)cc(Cl)c2)=O)CN(C(c2nncs2)=O)C2(CCCOC2)C1 87401,C(=O)(CCCCC(N)=O)NC1(C)CCN(CCC(=O)Nc2ccccc2F)C1 87402,C1(NC(C(CSC)OC)=O)CCC2(CC1)CN(C(=O)C1=COCC1)C2 87403,N(C)(C1CCc2cc(F)ccc21)CC(=O)N(c1ccccc1)CCOCCOC 87404,C(COC)(CC(C)(C)C(=O)OC)NC(C1CCC(CCCC)C1)=O 87405,c1(C(N2CCCC(C)(NC(C(C)=C3CCCC3)=O)C2)=O)ccn2cc(C)nc2c1 87406,C1(F)(C(=O)NC(CNC(C(CC)CC2CCCCC2)=O)CO)CCC(F)(F)CC1 87407,c1(N2CCCN(C(C)=O)CC2)nc(=NCC2CNC(=O)C2)[nH]c2cc(C)ccc12 87408,CCCCC(O)CC(=O)NCC(C1CCCC1)NC(c1ncccc1Cl)=O 87409,C1(n2cc(CN(CC(C)(C)OC)C)nn2)CCCCCC1O 87410,N1(C(CC(c2cccs2)N(C)C)=O)CC2CC1CCC2NC(C1CCCCC1)=O 87411,C(=O)(C1=CCC2(COC2)OC1)N(C(C)C)CCNC(C1CC(n2ccnc2)C1)=O 87412,C(c1cn(C)cn1)=C(C(=O)NC1(CC)CN(C(C2C(OCC)CCC2)=O)C1)F 87413,Cc1nc[nH]c1C(=O)NC(CNC(=O)CCN(c1ccncc1)C)CO 87414,c1(C(N2CC3C(C2)N3c2ncncc2I)=O)cccc2ncsc12 87415,Cn1c(O)ncc(C(=O)NC(c2ccccc2)c2ncon2)c1=O 87416,c1(C(N2CCC(C3N(C(CC(CC)C)=O)CCC3)C2)=O)ncc(F)c(OC)n1 87417,C#Cc1ccc(CC(N2CCC(NC(c3c(C)csc3Cl)=O)C(CC)C2)=O)cc1 87418,c1(OC)ccnc(C(N2CC(O)(CCNC(=O)C(C3CCOCC3)C)C2)=O)c1F 87419,C1(CNC(=O)NC2CN(C3COC3)C2)CCCC(F)C1 87420,N1(C(c2cc(C)ncn2)=O)CCN(C)CC1CNC(c1ccoc1CC(N)=O)=O 87421,c1(CCC(=O)NCCCCNC(CC2C(CC)C2)=O)cccc(O)n1 87422,Cc1cnc(F)cc1C(N1CCCC(CNC(=O)C(C)(C)n2cnnn2)C1)=O 87423,N1(C(C(C(C)C)CCc2ccccc2)=O)CCC2(CCOCC2)C1 87424,C1(C(N(CCCN(C)C)CCOCCOC)=O)CCN(C(=O)C(C)(C)C)CC1 87425,c1(CCC)cc(=NC(CNC(c2coc(COCC)n2)=O)C2CC2)[nH]c(Cl)n1 87426,c1(C(N2C3CCN(C(C4(OC)CC4)=O)C3CCC2)=O)ccc2c(c1)OCC(=O)N2 87427,C=Cc1cncc(C(N2CC(O)(C(F)C(=O)NCC(c3ccncc3)O)C2)=O)c1 87428,N1(C(CC(CC)SC)=O)CCC(O)C(NC(=O)CCC(C)C)C1 87429,C(=O)(CC(C)(C)NC(c1sccc1CC)=O)NC(C1CCOC1)C#C 87430,CC(C(=O)NC1(CN2CCN(C(=O)C=Cc3ncc[nH]3)CC2)CC1)C(F)F 87431,C1(=O)CC2=CCN(CC2)N1.C1(C)(C(NOCCCC(C)C)=O)CCC(C)C1 87432,c1(NC(CC2C(NC(C=CCOC)=O)CCCC2)=O)cc(C2CC2)ccc1C 87433,Cc1sc(C(N2CCCC2C(C)NC(=O)C2=NOCC2)=O)cc1Br 87434,N1(C(C(C(=O)OC)(C)F)=O)CCC(C)N(C(c2cnn3c2CCC3)=O)CC1 87435,c1(OC)ccc2nc(S(C)=O)[nH]c(=NCc3cnn[nH]3)c2c1 87436,c1(CN2CCN(CCN(CC)CC)CC2)ccc(Cl)cc1Cl 87437,C(=O)(C(C)(C)CS(N)(=O)=O)N1CC(NC(C(C2CCOC2)OC)=O)C(C(F)F)C1 87438,Cn1cncc1C=CC(=O)NCC(C1(O)CN(C(C2C3CNC(=O)C23)=O)C1)(C)C 87439,Cc1ccc(N(C(=O)CC2CC(C)N(C(c3cnn4c3CCC4)=O)C2)C)cc1C 87440,C#Cc1cnn(C)c1C(=O)NCC1CN(C)CCN1C(C1C2COCC12)=O 87441,C1(CC(=O)OCC)CC(NCCC2N(C(=O)CN3CC4CC4C3)CCC2)C1(C)C 87442,c1(C(N(C2CC(NC(C(C(CC)CC)C)=O)C2)C)=O)cnn2cccc(OC)c12 87443,CN1CCc2ccc(C(=O)NC3CC3CNC(=O)C3=NNC(=O)CC3)cc21 87444,CCC(C)C(C(=O)NCC1CN(C(c2cn3ccnc3s2)=O)CC1(C)C)N(C)C 87445,C(=O)(C(C)CC(F)(F)F)NCC1CN(c2cc(C)nc(C(C)(C)C)n2)CC1(C)C 87446,C(=O)(CCS(C)(=O)=O)NC1(C(=O)NC(CC)CN2CCCC2)CCSC1 87447,c1(C(=O)NC2CC(NC(=O)C=Cc3cc[nH]n3)C2)ccc(C2CC2)nc1 87448,N1(C(c2c(C)n(C)cc2)=O)CCC(NC(=O)C(O)C(F)F)C2(CCC2)C1 87449,c1(OC)ccc2nc(N3CCCC3)[nH]c(=NCC3CCCc4ccccc43)c2c1 87450,N1(C(c2c(C)n(-c3ccn(C)n3)nn2)=O)CCC(CNC(C2CCC2)=O)C12CC2 87451,c1(CC(=O)NC2CC2NC(c2csc(-c3ccccn3)n2)=O)ccc(O)cn1 87452,c1(C(N(C2CCN(C(C3CC(OC)C(OC)C3)=O)C2)CC)=O)ccn2ncccc12 87453,O=C(C1=CS(=O)CCC1)NCC1CCN1C(=O)CC1CCC(F)(F)CC1 87454,O=[N+]([O-])c1ccc(Br)c(Cl)c1N(C)CCc1nccs1 87455,c1(CC=C(C)C)ccccc1C(=O)NCC(C)CNC(c1snnc1C1CC1)=O 87456,Cc1cc(N(C)CC2CC(Cl)(Cl)C2)nc(N2CC=CCC2)n1 87457,N1(CC(=O)NC2C(CC(=O)NCCN3CC=CC3)CCC2)CCOCC1=O 87458,C(N=c1ccnc(C)[nH]1)C1CCCC(NC(C(c2cc(C)c(F)cc2)(C)C)=O)C1 87459,c1(C(=O)NC2C3(CN(C(c4cnc(C)o4)=O)C3)CC2)coc(S(=O)(=O)N(C)C)c1 87460,N1(C(C(c2ccc(OC)nc2)(F)F)=O)CCC2(NC(=O)CC(C)(C)O)CCCC12 87461,N1(C(c2cc(C)c(C)s2)=O)CC2(CC(NC(=O)CS(=O)(=O)N(C)C)C2)C1 87462,N1(C(Cc2ccc(C)cc2)=O)CC(NC(=O)C(C)CC(C)(C)C)CCC(O)C1 87463,C1(CC(=O)NCC2CCC(C(N)=O)O2)CN(C(=O)COc2cccnc2)CCO1 87464,c1(OC(CCSC)=O)ccc(OCC(N)=O)cc1.c1(O)ccc(F)cc1 87465,O([Si](C)(C)C(C)(C)C)CC.C1(CC(C)C)(C(=O)NCCCOC)CC(=O)C1 87466,CCC(CNC(=O)C(C(=O)OC)OC)(CC)C(=O)Nc1ccc(O)cc1Cl 87467,C(=O)(C#CC1(CC)CC1)NC(CNC(C(C)SCCCC)=O)C(C)C 87468,N1(C(c2c(CC)ncs2)=O)CCCC2(C1)CN(C(c1cccc(C)c1Cl)=O)C2 87469,CC1CN(C(=O)CS(=O)(=O)NC(C)(C)C)C(C)CN1C(=O)Cc1cnnn1C 87470,CN1CCN(C(C2CC(C3CC3)=NO2)=O)C(C(=O)N(C2CCN(C)C2)C)C1 87471,CCCCN=C(NCCc1ccc(Cl)c(Br)c1)NCCc1nccs1 87472,C1(C)(C(=O)NC2C=CC(CC(N3C(C)(C(=O)OC)CC3)=O)C2)CCCCC1 87473,c1(C(N(C2CCCCN(C(C3(C)CC=CC3)=O)C2)C)=O)cc(Br)cnc1O 87474,N1(C(c2c(COC)cco2)=O)CCCCC1CCN(C(=O)C(C)NS(C)(=O)=O)C 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87545,C1(CNC(C)=O)CCC(F)(CNC(=O)C(C)CCN(C)C)CC1 87546,c1(CNC(C(CO)O)C2CC(F)(F)C2)ccc2ccccc2c1 87547,C(=O)(CCCN(C)C)N(C1CCC(NC(C2(F)CCC2)=O)C1)C 87548,C1(F)(CNC(C(COC)OC)=O)CCC(CNC(=O)C(c2cnccn2)C)CC1 87549,C1(NC(c2ccc(OC)s2)=O)C(C)CN(C(c2cn(CCO)nn2)=O)CC1C 87550,C1(NC(c2ccnc(F)c2Cl)=O)CCN(c2ncncc2I)CC1F 87551,N1(C(C)=O)CCCC(CCNC(c2sc(F)cc2C)=O)CC1 87552,C(C(=O)N1OC2CCC1C2)C1(C)N(OC(CCCCN(C)C)=O)CCC1 87553,CC1=NOC(CCNC(=O)CCN(CCO)C(C23COCC2C3)=O)C1 87554,N1(C(C=C2CCC(C)C2)=O)CCCN(C(=O)COc2cncc(Br)c2)CCC1 87555,N1(C(c2ncn(C(C)C)n2)=O)CCC2(CCC2NC(c2cnncc2O)=O)CC1 87556,c1(C(=O)NC(c2cnc[nH]2)C)coc(CNC(c2ccsc2Cl)=O)n1 87557,Cc1cc(C(=O)NCCN(C(=O)Cc2cncc(C#N)c2)C2CC2)ccc1Cl 87558,O=C1CC(C(=O)NC23CCN(C(c4cccc(Cl)c4F)=O)CC2C3)CC(=O)N1 87559,c1(C(=O)NCC(C)CNC(=O)C(c2ccccc2)O)cc(Cl)c(Cl)cc1N 87560,C1(C(N2CC(Cn3cc(C(C(=O)OC)(C)C)nn3)C2)=O)(NC(C)=O)CCNCC1 87561,Cc1cn2cc(C(=O)NC3CCC3CNC(c3cnc(C(C)(C)C)s3)=O)nc2s1 87562,N1(C(C(CCC)O)=O)C2CCCC1CN(C(=O)C(O)C1CCC1)C2 87563,c1(C(=O)NCCOC2CCN(C(C(C=C=C)C)=O)CC2)ccc(C#N)c(C)c1 87564,N1(C(N(c2sc(C)cc2Cl)C(C(=O)OC)Cc2ccccc2)=O)CCCC(C#N)C1 87565,C=CCC(C(=O)N1CC(N(C)C(c2ccn(CCC)n2)=O)C1)c1ccccc1 87566,C=CCCCCCCCC(=O)NC1CCCC(CNC(=O)CCSCCOC)C1 87567,c1(OCC)cccnc1C(=O)NCCCCNC(C1(C)CCC(=O)N1)=O 87568,CC(C)CCC(O)C(=O)NCCCCC1CCN(C)CC1.C1CO1.C(CO)O 87569,c1(N(C)C)n[nH]c(=NC(=O)N2CC(C(N)=O)C(c3ccccc3)C2)s1 87570,N1(C(C(CC)COC)=O)CCCC(C)(C(=O)NCc2nocc2C(C)C)C1 87571,c1(CC(=O)NC(C)CNC(c2cncc(N(C)C)c2)=O)ccccc1S(C)=O 87572,C1(C(N2CC(CCNC(C3C4(CC(C)(C)C4)C3)=O)C2)=O)CCc2ncncc2C1 87573,C1(NC(c2occ(C)c2)=O)COC2C(NC(=O)C(F)F)COC12 87574,C1(C(=O)NC)COCCN1C(C1CCCCN1C(C12CSCC1C2)=O)=O 87575,c1(CC)nc(C(=O)NCC2CCCCC2NC(=O)Cc2ccccc2F)c(C)o1 87576,c1(C(=O)NC2(CNC(c3n[nH]cc3F)=O)CCOC2)cnn2c1OCCC2 87577,c1(SCC)cc(C(=O)NCCC2(NC(=O)CC(CC)SC)CCC2)ccc1F 87578,N1(C(c2n(C)ncc2)=O)CC2CC1(C(N1CCC(C(F)F)CC1)=O)C2 87579,C1(CNC(c2ccc(C#C)cc2)=O)COC(C)(C)CN1C(=O)C(C(C)C)N(C)C 87580,C1(CNC(C(C)(C)Br)=O)CCN(S(=O)(=O)Cc2cccc(Br)c2)CC1 87581,c1(C(C)C)ccc(C(N2CC(O)(CCNC(=O)CCC3CC3(F)F)C2)=O)c(F)c1 87582,C1(C(N(CCO)CC)=O)CC2CN(C(C3CCCCC3)=O)CC2C1 87583,CC1CN(C(c2ccc(C3CC3)nn2)=O)CCN(C(c2cnnn2C)=O)C1 87584,n1(CCC(=O)N(CCCN(C)C(C23CCC2C3)=O)C)ccc(O)nc1=O 87585,N1(C(c2c(OCCC)cccc2)=O)CC(NC(=O)C(C)c2ccco2)CC(C)C1 87586,C=CCC(CC(C)C)C(=O)N1CCOC(CN(C(=O)CCc2cnn[nH]2)C)C1 87587,C1(CC)CN(Cc2c(C)coc2CBr)CCN1Cc1ccccc1 87588,c1(CC(=O)NCC(C)N(C(Cc2ccc(C)cc2)=O)C)nn(C)cc1[N+](=O)[O-] 87589,C1(CNC(CCCCSC)=O)CCN(C(=O)C(C)(C)C2(C)CC2(F)F)CC1C 87590,N1(C(C2(OC)CCC(C)C2)=O)CCC(C=CC(=O)Nc2cc(C)ccc2F)CC1 87591,C1(C)(C(N(C)CC2CCCN(C(CC(=O)OC)=O)C2)=O)CCS(=O)(=O)CC1 87592,C1(C(=O)NCCc2ccc(C)s2)(NC(COCCOCC)=O)CCN(C)C1 87593,C(CN=c1[nH]c2c(c(=NCc3nn(C)cc3C)[nH]1)CSC2)c1nnc(COC)s1 87594,C1(CNC(c2c(C(=O)OC)scc2)=O)CN(C(=O)C(C)CCOC)CCCO1 87595,N1(C(C(C(C)C)C)=O)CC(CC(=O)NCC2(CCO)CC2)CC1(C)C 87596,c1(OC)ccccc1C=CC(=O)NCC(C)(CO)NC(c1cc(F)ccc1C)=O 87597,C1(C(=O)NCC(C(C)C)NC(c2cc(CCO)on2)=O)CCC(C)CC1 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87616,c1(C(=O)NCC(C(=O)N(C)CC2CCCC3CC23)N(C)C)c(F)cccc1F 87617,c1(OC)cc(C(=O)NC2CCC2CNC(C2CCCOCC2)=O)cc([N+](=O)[O-])c1 87618,C12(C(C)NC(=O)C(c3ccco3)NC(c3coc(C(F)F)c3)=O)CCC(CC1)C2 87619,Cc1cccc(C(C(C)C)NC(c2ccnn2CC(F)F)=O)c1 87620,CCC(CC(=O)N1CCN(C(=O)CCc2ccc(C)s2)CC1COC)C(F)F 87621,c1(OC)cccc2c(CC(=O)NCCCN3CC(C)CC(C)C3)c[nH]c12 87622,Cc1cccc(N)c1C(=O)NCC1C(C)CCCN1C(=O)Cc1cccc(F)c1 87623,c1(CC)onc(C)c1C(N1CC2CC2(C(=O)NCc2cccc(Br)n2)C1)=O 87624,c1(C(N2CCCC(OC(C)(C)C)C2)C(=O)NC(CC)(C)C)ccc2c[nH]nc2c1 87625,c1(C(=O)NCC(C)CNC(c2cnc(C(C)O)s2)=O)cnn(C)c1-n1cccc1 87626,C1(C(N(C2CCC2O)C)=O)CC(O)C(O)CC1CNC(C1(N(C)C)CC1)=O 87627,C1(NC(C2CCn3ccnc3C2)=O)CCCC12CCN(c1nncs1)CC2 87628,Cc1cc(N)c(C(=O)NC(C2CN(C(c3cccc(F)n3)=O)CCO2)C)cc1F 87629,c1(C(N2CCC(NC(CC(=C)C)=O)(CF)C2)=O)ccc2c(c1O)CCCC2 87630,C1(NC(C(CC#C)C)=O)CC2(C1)CN(C(c1ccnc(OCC)c1)=O)C2 87631,c1(C(=O)NCC(C(C)C(C)C)NC(Cc2cnc(C)[nH]2)=O)cc2ccccc2o1 87632,c1(C(C(N2C(CN(C(C(CC)N(CC)CC)=O)C)CCC2)=O)=O)ccc(O)cc1 87633,c1(OC)cc(OC)cc(C(=O)NCC(C)(C(C)C)NC(c2ccc(Cl)cc2)=O)c1 87634,C1(NC(C(=O)Nc2ccc(C3CCCNC3)cc2)=O)CCNCC12CC2 87635,CC(CCC(=O)NC(C)(CNC(=O)C(N)=O)C1CC1)NC(=O)OC(C)(C)C 87636,C(C1c2ccccc2CN1C(=O)CSc1nncs1)NC(C1C2CCCOC12)=O 87637,c1(C(N2C(C)CN(C(C3CCC(=O)N3)=O)CC2)=O)ccnc(P(C)(C)=O)c1 87638,C1(CN(C)C(c2cccc(O)n2)=O)CCCCN1C(C1(C)CCC(=O)C1)=O 87639,c1(C(=O)NCC2C(C(=O)NCC(=O)N(C)CC)CCC2)ccccc1CC#N 87640,C1(C(N2CCCC(N(C(c3cc(Br)c[nH]3)=O)CC)C2)=O)CC2CCCCCCC12 87641,c1(CSC)ccc(C(C)(C)C)cc1.C12(CCOC1)CN2 87642,c1(CCC(=O)NCCOc2ccc3cccnc3c2)cccc2c1OCCO2 87643,C1(CNC(=O)CNC(=O)CNC(C)=O)C=CCOC1.C(=O)(C(=O)N)NCCNC(C)=O 87644,N1(C(C2CCC(=O)N2)=O)CC2(CCCC2NC(c2ccc3ncsc3c2)=O)C1 87645,c1(OC)cccc(C(F)F)c1C(=O)N(C)CCN(C)C(C12CC1COC2(C)C)=O 87646,C1(C(=O)NC2CCN(C(CC3C(C)C3)=O)CC2F)CC2C=CCC(C1)C2 87647,N1(C(CNC(CC)=O)=O)CCC(C(C)NC(c2sc(C)nc2CC(C)C)=O)CC1 87648,C(=O)(C1=NOC2COCC12)N(CCNC(C(C)SC)=O)CC1CC1 87649,C=CCCCCC(=O)NC1COCC1CNC(c1c[nH]c(Br)c1)=O 87650,N1(C(c2occ(C)c2)=O)CC2OCCN(C(c3cnn(CCF)c3)=O)C2C1 87651,C(C1=CCCOC1)NC(C(CNC(c1cnccn1)=O)O)=O 87652,Cc1cc(C(=O)NCc2cc[nH]c2C(=O)NCC(c2cnc[nH]2)C)[nH]c1C 87653,c1(NC(C(=O)N(C2CC3CCC2C3)C)=O)cncc(SC(C)(C)C)c1 87654,N1(C(C(C(C)C)O)=O)CC2CN(C(=O)COCC3CCCCC3)CC2C1 87655,c1(CN(C(c2c(COC(C)=O)ocn2)=O)C)cccc(C)c1C.C12(CC1)C(=O)N2 87656,C1(NC(CC(C)(C)C)=O)CC2(C1)CN(C(c1nc(Br)cnc1N)=O)C2 87657,Nc1cccnc1C(=O)NCC1COCCN1C(=O)CN1CCOC1=O 87658,C1(C(=O)NC2CCCC(CNC(CNC(=O)OCC=C)=O)C2)CN(C)CC(C)O1 87659,N1(C(c2c(C(C)C)occ2)=O)CC(CNC(C2CCCCN2C)=O)C(O)C1 87660,c1(CCC(=O)NC2CCN(C(CCC(=C)C)=O)C2)cn2ccccc2n1 87661,c1(OC)cc(OC)[nH]c(=NC2CCC(C)N(C(c3coc(C4CC4)n3)=O)C2)n1 87662,c1(CN(C(NC(CC)C)=NCc2cc(C3CC3)no2)C)ccc2c(c1)CCCC2 87663,c1(C(N2C(CCNC(C(N3CCNC3=O)C)=O)CCC2)=O)cccc(O)c1F 87664,C=Cn1nccc1C(N1CC(CC(C)NC(C2CCN(C(C)=O)C2)=O)C1)=O 87665,CCCCCCCCC(=O)NC1(C(N2CCOC(CF)C2)=O)CC1 87666,c1(OC)ncc(S(=O)(=O)NCC(c2ccccc2Cl)O)cc1C 87667,c1(C(N2CCN(C(=O)C3=CCCSC3)C(CCO)C2)=O)cccc2c1NCC2 87668,C1(CC)CN(C(=O)CCOC(C)C)CCN1C(c1ccnc(C)c1N)=O 87669,N1(C(C=CCOC)=O)CCC(CNC(c2ccc(Cl)c(C(F)(F)F)c2)=O)C12CC2 87670,Cc1csc2ncnc(N3CCCC(C(=O)NCC(C)O)C3)c12 87671,c1(CC(=O)NC(C)CCNC(c2csc(-c3cnc[nH]3)n2)=O)c[nH]c(=N)nc1O 87672,C12(CNC(C=Cc3ccc(C)o3)=O)CCCC1N(C(=O)Cc1nc[nH]n1)CC2 87673,C(CC(F)F)(C(=O)NC(C)C(=O)N(C)C)NC(CCOCC)=O 87674,C=CCC(C(=O)NCC(F)C1CCC1)NC(=O)CCCN(C)C 87675,Cc1nc(NCCc2nc(-c3cccs3)n[nH]2)cc(=NCc2ccc(F)cc2)[nH]1 87676,C1(C(=O)NC(CC(C)NC(c2cnn(C(C)C)n2)=O)C)CCCCC1C 87677,c1(CC)nc(N2CC(CNC(C3CN4CCN3CC4)=O)(OC)C2)cc(C)n1 87678,c1(NC(C)=O)ccc(C(N2CCCC(N(C)C(C3CCCSC3)=O)C2)=O)c(Cl)c1 87679,c1(C(=O)NC(CNC(CC2(CC=C)CCCC2)=O)C(C)C)coc2c1COC2 87680,N1(C(C2CC(C)C2)=O)CC2CC1(C(=O)NCCC1CC3C=CC1C3)C2 87681,c1(C(CO)NC(c2cnn(C(CC)C)c2C)=O)cc(F)cc(Cl)c1 87682,c1(OCC(N2C(C3(NC(c4c(CC)non4)=O)CC3)CCC2)=O)ccc(C#N)cc1 87683,c1(CC)nn(C)c(CC)c1CC(=O)NCC(C)(C)NC(c1cc(N)cnc1C)=O 87684,N1(C(C2CC=C(C)CC2)=O)CCC2C(C1)CN2C(c1cc(C)cnc1C)=O 87685,C(c1c(C)nn(C)c1Cl)=CC(=O)NCC(CC)NC(C1CN2CCCN1CC2)=O 87686,C1(CN(C(COC(CC)C)=O)CC)CCN(C(C2CCCC3CC23)=O)CC1 87687,N1(Cc2onc(CCOC)n2)CCC2(CC1)CN(C)C2(CC)C(=O)O 87688,c1(C(=O)NC(C(C)C)C(C)NC(=O)Cc2cncs2)cccc2c1OCC2(C)C 87689,CC1CCN(C(C2CCC=CO2)C(=O)Nc2ccc(Cl)cc2F)CCS1 87690,FC1(F)CCCC(c2nc(-c3ncccc3Br)no2)CC1 87691,C(=O)(C1CCCc2ccccc21)NC(CN=c1[nH]nc(C(=O)OC)s1)C 87692,CCC(C)C(O)CC(=O)N1CCC(CC(=O)NCC=C(Cl)Cl)CC1 87693,C(CO)(CCCNC(c1ccc(=N)[nH]c1)=O)NC(c1c(CC)cco1)=O 87694,c1(NCC(=O)N(C2CCN(C(C3(CC)CC3)=O)C2)CCO)ccccc1[N+](=O)[O-] 87695,C1(NC(CCc2cnc(C)o2)=O)CCCC(C(=O)N(CC(C)O)CC(C)O)CC1 87696,Cc1cnn(C)c1CC(=O)NCCOCCN(C)C(C1(CC(C)C)CCCC1)=O 87697,CCCCC(C(=O)N1CCCc2nccn21)NC(C1CC(=O)CS1)=O 87698,c1(OC)ccc(CSC2CCCN2c2cc(C(F)(F)F)ncn2)c(Cl)c1OC 87699,C(CNC(=O)COCC1CCOC1)(CC(C)C)NC(c1c(C)ccnc1)=O 87700,c1(NC(C2(CC)CN(C(=O)Cc3ccoc3C)C2)=O)cnccc1CO 87701,C(C)(CCCC(C)C)NC(CC(C)(C)NC(Cc1c(C)noc1C)=O)=O 87702,C1(C(N2C(C(N(CCO)CC)=O)CC2)=O)CCCSC1 87703,Cc1cc(C)c(C(=O)NCC(F)CNC(=O)C=C(C2CC2)C2CC2)o1 87704,c1(N(CCOCC=C)C)nc(=NC2C(OCC)CCC2C)[nH]c2c1CCC2 87705,c1(OC(C)C(=O)OCC23COC(c4ccccc4)(C2)C3)cccc(Cl)c1 87706,CC1(C(=O)NCC2(c3nn[nH]n3)CC3CCC(C2)S3)CCn2ccnc21 87707,N1(C(COC(C)=O)=O)CC2C3CCC(C2C1)N(C(=O)CC1CCC2CC12)C3 87708,N1(C(c2c(CC)nccc2)=O)CCC2(CCCN2C(C23CCC2CC3)=O)C1 87709,N1(C(C(C)OC2CCCCC2)=O)CCC(N(CCO)CC(c2ccoc2)=O)CC1 87710,CC1(C)CC(NC(c2coc(C3CC3)n2)=O)CN(C(=O)Cc2n[nH]c(=N)s2)C1 87711,C1(C(=O)NCCCSCC)CN(C(=O)CC2CCCSC2)CC12CCC2 87712,c1(OC)ccc2c(c1)OCC(C(N1CC3CC1CCC3NC(C1(C)CC1)=O)=O)C2 87713,C1(CC(=O)N(CCNC(=O)CCn2cncn2)CC)CC(C2CC2)C1 87714,Cc1ccc(C#N)cc1S(=O)(=O)N1CCC(C)(C(N2CCCCC(C)(F)C2)=O)C1 87715,CC#CCC(C(=O)NCC1CC(C(=O)OC)C1)NC(=O)CCSCC 87716,c1(OC)ccc2c(c1)c(CCNCCC1(O)CCOC1)cn2C 87717,C(=O)(CS(=O)(=O)CCOC)NCC(CCOC)NC(=O)CC1CC2CCC1CC2 87718,c1(C(=O)NC2C(CNC(C(C)NC=O)=O)COC2)cc(F)cc(F)c1 87719,C1(C(=O)NCC(O)CO)(OC)CCN(Cc2ccc(F)cc2)CC1 87720,C1(CCC)CN(C(C2CCCSC2)=O)CCN1C(=O)CC1CCC1 87721,c1(C(N2C(CCNC(c3c(CC)nn(C)c3)=O)COCC2)=O)ccc(F)cc1Cl 87722,C1(NC(C(CC#C)C2CC2)=O)CC2CC1N(C(c1ccoc1Br)=O)C2 87723,C(=O)(C(CCC1CCC1)NC(=O)CC1CCC(=O)NC1)NCc1ccn(C)n1 87724,c1(NC(C23C(CN(Cc4ccc(OC)nc4)C2)C3)=O)cccc2c1OCC(=O)N2 87725,C1(C(N2CC(NC(=O)OC)C2)=O)CCC(O)CN1C(=O)CC1CCN(C)CC1 87726,N1(C(CS(CC)(=O)=O)=O)CCCN(C(C2CC(F)C2)=O)C(CO)C1 87727,C(=O)(C1OCCn2ccnc21)NCC1C(NC(COc2c(C)cccc2Cl)=O)CC1 87728,c1(C(CC(=O)NC2(C)CN(C(C(CCC#C)O)=O)C2)C)ccc2c(c1)OCO2 87729,N1(C(=O)NC(=O)NCC=C(CCC)C)CCC(C)(NC)CC1 87730,N1(C(CC(C(=O)OC)C)=O)CCC(C)(C)CC1C(=O)NCC(CO)OC 87731,c1(OCCCNC(CNC)=O)ccc(Br)nc1 87732,C1(CNC(COCCOC)=O)COCCN(C(=O)C=CC(C)(C)C)C1 87733,c1(SC)cccc(C(N2CCC(C)C2CNC(=O)C2=CCSC2)=O)n1 87734,c1(-c2nc(CCNC(=O)NCC3(CO)CCOCC3)sc2)cccc(F)c1 87735,Cn1c(NC(=O)C(O)Cc2ccccc2Cl)nnc1C1CCCCC1 87736,C(C)(C)(CC(F)C(=O)N(C1CCC2(CC1)CC2)C)NC(C(CCCC)O)=O 87737,CC1(C)CCCCN(C(C2N(C(=O)CC3OCCCO3)CC23CCCC3)=O)C1 87738,C1(C(=O)NC2(C)CN(C(=O)CC3(O)CCOC3)C2)Cc2c(F)cccc2O1 87739,N1(C(c2c(C)c[nH]c2)=O)CCN(C(=O)CCc2cncnc2)CC(C)C1 87740,C1(C(N2C(CNC(C3(N(C)C)CCC3)=O)CC2)=O)CCCOC1c1cn(C)nn1 87741,C=CC1(O)CCN(C(=O)CC(C(C)OC)NC(c2cncc(CC)c2)=O)C1 87742,C(=O)(C(C1=CCSC1)N(CCS(=O)(=O)C(C)C)C)NCCC 87743,c1(OCC)ncc(Cl)cc1CNC(=O)Nc1oc(C2CCC2)nc1C 87744,C(C(C)(C)CC1COC1)N(C(=O)C(C)(C)C)C(=O)NC1C(C(C)N)C1 87745,c1(OCC(C)C)cccc(C(N2CC(NC3(C)CC3(C)C)C(C(F)F)C2)=O)c1 87746,C(C(CC(=O)N(CC(=O)N(C)C)C)NC(C1C=CCS1)=O)OC 87747,c1(NC(CCC)=O)cncc(C(N2CCN(CC(F)(F)F)CC2)=O)n1 87748,c1(C(F)(F)F)ccc(CNC2CCC(Sc3ccccc3)C2)cc1 87749,C1(C(=O)NC(c2ccc(OC)cc2)C)CC12CCN(c1nc(Cl)ncc1F)CC2 87750,CC(C(=O)Nc1cnc(F)nc1)C(C)NC(c1ncc(F)cn1)=O 87751,CCCC(C)(C)C(=O)NCC(CNC(c1cnn(C)c(=O)c1)=O)OC 87752,CC1C(C(=O)N(C2CC(OC(C)(C)C)C2)C)SC(C(F)(F)F)C1 87753,N1(C(C(c2ccc(C)cc2)=O)=O)CCC2C(CCCN2C(C2CCS2(=O)=O)=O)C1 87754,N1(C(CCSCCC)=O)CCC2CCN(C(c3nc(C)c(N)cc3C)=O)C2C1 87755,N1(C(C(C(CC)C)O)=O)CCN(C(c2cnn(CC(F)F)c2C)=O)CC(C)(C)C1 87756,CC(C)C(CNC(C1CCOC1(C)C)=O)C(=O)NCc1c(F)cccc1F 87757,c1(C(C)=O)ccc(CC(N2CC=CC(NC(=O)CCN3CCC(F)C3)C2)=O)cc1 87758,c1(CCC(=O)NC2C(CNC(CC)=O)C2)cccc(CC(C)C)c1 87759,C1(CNC(CCC#CC)=O)CC(C)CN(C(=O)C=Cc2ccc(OC)cc2)C1 87760,C1(N(C(=O)CCN2CCCC2)C)CN(C(=O)CC2CCC(F)(F)CO2)CC1(C)C 87761,C(N=c1[nH]c(=NCC(C(C)C)NC)[nH]c2c1CCCCC2)C1N(CCC)CCC1 87762,CC1(CN(C2CCCO2)CC(=O)NC(=O)CCN)CC1(F)Cl 87763,c1(C(=O)NC2CCN(C(C3CC4C(C3)C4(F)F)=O)CC2F)occ2c1CCOC2 87764,C(c1cccc(C#N)c1)=CC(=O)NC1C(OC)CN(C(C2CCCO2)=O)C1 87765,N1(C(C2(C)C(C)(C)C2)=O)CC2COCC(C1)C2NC(=O)C1=C(Cl)CC1 87766,N1(C(C(C)N=[N+]=[N-])=O)CCCC2CN(C(=O)CN3CCCCC3=O)CCC12 87767,c1(C(N2CC(COC)(CNC(=O)C(C#N)C(C)C)C2)=O)nc2ncccn2n1 87768,c1(C(=O)NC(C(=O)NCCN(C(=O)CC(C)(C)SC)CC)C)cccc(F)c1F 87769,C1(OCC)CCCC1(c1nnnn1CCCF)NCC(C)(CC)CC 87770,c1(C(C(=O)NCCC(C)F)NC(C2CC(=C3CC3)C2)=O)cccnc1 87771,N1(C(C(C)(C)CO)=O)CCC2(CCOCC2)C(CNC(=O)CCc2cnc[nH]2)C1 87772,C1(CC)CCN(C(=O)C=Cc2ccnn2CC)C1C(=O)NCc1cc(C)sc1C 87773,N1(C(COCC(N2CCOCC2)C)=O)CCC(NC(=O)C(C)(C)NC(N)=O)C(C)C1 87774,C(CCCCCC(=O)NCC1CCN(C(c2ccc(C(=O)CF)cc2)=O)C1)SC 87775,N1(C(C(NOC)=O)=O)CC(C(=O)NC2(c3nc(C)no3)CC2)C(C)(C)C1 87776,Cc1ccc(C=CC(=O)NCC(C)CN(C(=O)CCSCC(C)C)C)cc1 87777,CCS(=O)(=O)CC(=O)NCC1(C(=O)Nc2cc(OC)cc(C(F)(F)F)c2)CC1 87778,C(CC(C)(C)C)(C(=O)N1CCC(C)(C(N2CCCCC2)=O)C1)OC 87779,C12(C(N(C)Cc3ccoc3)=O)CCC(CC1NC(=O)CSC(F)F)C2 87780,c1(C(N2CC(CN(C)Cc3ccc(Br)c(F)c3F)C2)=O)cc2cccnn2n1 87781,C(CCCCC(=O)NCC1CCC(C#N)C1)n1cc(C2(CC)CCC2)nn1 87782,N1(C(CN2CCC(C)(C)C2)=O)CCC2(CC1)CN(C(=O)CC1CCOC1(C)C)C2 87783,N1(C(=O)N(CCS(C)(=O)=O)CCO)C2CCC1C(NC(c1ccccc1)C)C2 87784,C1(n2cc(Cc3c(C)nn(C)c3)nn2)CC(N=c2ccnc(S(C)(=O)=O)[nH]2)C1 87785,c1(C(=O)NC2CCC(C)N(C(=O)Cn3ncnn3)C2)ccn2c1CSCC2 87786,C1(NC(C(=Cc2cccnc2)C)=O)CCN(C(=O)CC2(C)CCC2)CCC1CO 87787,CC1CN(Cc2cc(-c3cc[nH]c(=N)c3)ccc2F)C(C)(C)C1 87788,C(=O)(N=c1ccn(C2CCS(=O)(=O)C2)[nH]1)C1(CC#C)CCCCO1 87789,c1(C(CNC(C(n2cc(C(C)O)nn2)C)=O)=O)ccccc1[N+](=O)[O-] 87790,C(c1ccccc1)=CCN(CC(=O)N(C1CN(C(=O)CC2(C)CC2)C1)C)C1CC1 87791,c1(C(=O)NCC(CN(C(C(=O)NCC)=O)C)C)n[nH]c(C(C)C)c1[N+](=O)[O-] 87792,C(=O)(C1=C(C#N)CCC1)N1CC(NC(c2c(CCC)n(C)nn2)=O)C(SC)C1 87793,N1(C(C2CC(NC(c3c(OC)cc(F)cc3)=O)C2)=O)Cc2cc(Br)cnc2C1 87794,C=CCC(C)(CC)C(=O)NC1CCCC1CNC(c1cnnn1C1CC1)=O 87795,c1(OCC)nc(C)ccc1C(=O)NC1CCC(F)(CNC(=O)CCC(C)C#N)C1 87796,c1(C(N2CCC(N(C(c3cc(C)on3)=O)C)C2)=O)c(-n2nccn2)cccc1F 87797,C1(CC=C)(NC(=O)CCC2(C)CC2)CN(C(=O)COC(F)(F)F)C1 87798,Cc1nc(C(C)C)ccc1C(=O)NC1CCCC(NC(c2cc(F)n(C)n2)=O)C1 87799,C(=O)(C(C)(C)C(=O)NC1CC(C)(NC(C2CCCC(C(N)=O)CC2)=O)C1)OC 87800,c1(C(C(=O)OC)N(C(=O)COC2CCCOC2)C)ccccc1F 87801,C1(CCC)CN(C(=O)CCNC(=O)COC)CCN1C(C1CCCOCC1)=O 87802,C(=O)(CS(=O)(=O)C1CCCC1)NCCC(C)N(C)C(C1CC2(C1)CC2(F)F)=O 87803,Cc1ccc2snc(C(=O)N(CC(C)NC(C3CC4CCCCN4C3)=O)C)c2c1 87804,C1(C(N2CC(C)(C)C2)=O)COC2(C1)CN(C(=O)CC1CCCOCC1)C2 87805,CC1OCCCC1C(=O)NC1(CC(=O)NCC(C)(O)C2CC2)CCCCC1 87806,Cc1ncnc(C)c1CC(=O)Nc1ccc(N2CCN(C)CC2)nc1 87807,CCC(COC)C(=O)N(C(C)(C(=O)NC(C)C(C)(C)CN(C)C)C1CC1)C 87808,C(CN=C(NC(C1CC=CCC1)C1CCCC1)NC1CCCCC1)N(CC(C)C)C 87809,Cc1cccc([N+](=O)[O-])c1N1CC2CC1CN(C(=O)Cn1cc(S(N)(=O)=O)cn1)C2 87810,N1(CCC(C)NC)CCCC(NC(N2CCC(C(=O)OC)CC2)=O)C1 87811,c1(C(C)(C)C)cc(Br)ccc1NC(c1ccnc(C2CC2)n1)=O 87812,CC1(C(=O)NCc2ccccc2)CCCN1Cc1cccc(F)c1 87813,C1(O)(CNC(c2cc(OC)no2)=O)CCN(C(=O)C(C)(C)Sc2ccccc2)C1 87814,C1(C(=O)NCCC2(NC(=O)C(C)OCC3CCCO3)CCC2)(SC)CCC1 87815,N1(C(c2ncn3c2CCC3)=O)CCC2(CCSCC2)C1 87816,CC1CN(C(c2occ3c2CCC3)=O)CCCN1C(C12CC1COC2(C)C)=O 87817,C1(C(=O)NCCOCCO)(NC(C(COCC)C)=O)CCCCC1 87818,c12cc(C)c(c(C)c1)-c1nc(C3CSC3)nn1C2.c1(CC)onc(CSC)c1C 87819,C1(C(N(CCNC(=O)Cc2csc(S)n2)Cc2ccccc2)=O)CCCC1(F)F 87820,N1(C(C(CCSC)OC)=O)CC2CC1CN2C(c1ncn(C(C)(C)C)n1)=O 87821,C1(CC)CCC(O)(C(=O)NCCC2(CNC(=O)C=Cc3ccc[nH]3)CC2)C1 87822,C#CCCC(O)C(=O)N1CCC(C(C)(C)NC(=O)C(C)CC=CCC)CC1 87823,C12(c3cn(C)nc3)CCC(C1)C2C(N1CCC1CNC(C1(CF)CC1)=O)=O 87824,C(CCC(=O)N1CCCC1C(=O)N(C1CCC1)C)OC(C)C 87825,CP(C)(=O)C(O)C(=O)N1CCC(NC(=O)Cc2cccc(Br)c2)C(O)C1 87826,c1(C(N2C(C)(C(=O)NC3(COC)CC3)C=CC2)=O)cc([N+](=O)[O-])c[nH]1 87827,c1(C(=O)NC(C(=O)NC2C(CC=C)COC2)CO)cc2cc[nH]c2cn1 87828,c1(OC)ccc(Cl)c(C)c1C(N1CCC2CN(C(=O)C3=COCC3)CC12)=O 87829,Cc1cc(C(=O)NCC2CCN(C(=O)C=Cc3cncs3)C2)no1 87830,CC(C(F)F)N(C)N1CCC(CN2CCOC(C)C2)CC1 87831,c1(C(=O)NCC(CC)NC(CSCC#C)=O)cn(C)nc1OC 87832,Cc1cncc(C)c1C(=O)NCC(O)CNC(C1CCC(C(C)(C)O)CC1)=O 87833,N1(C(c2c(CN=[N+]=[N-])ccs2)=O)CCN(C2CCN(C(C3(CO)CC3)=O)C2)CC1 87834,c1(CC(=O)N(C2CCCC2)CCNC(C2C(C)CCCO2)=O)ncc(F)cc1F 87835,Cc1nc(C(N2CC(O)C(O)C2CNC(=O)CCCc2ncco2)=O)cc(O)n1 87836,CC1=C(C(=O)N2CC=CC(NC(C3CCCSC3)=O)C2)CCCO1 87837,c1(N(CCCS(C)(=O)=O)C)nc(-c2ccccc2)nc(=NC2CCOC2C)[nH]1 87838,C1(C(N(CCOC)CCO)=O)CCC2(CC2)N1C(C1Cc2nccn2C1)=O 87839,N1(C(Cc2cccc(C#C)c2)=O)CCC2(CCCN(C(=O)CCCOC)C2)C1 87840,N1(C(c2ccc(C)cn2)=O)CC2(CCOCC2)CC1CNC(=O)C(C)C1CC1 87841,C1(CNC(C=C(C)C(C)C)=O)CN(C(C2CC=CC(O)C2)=O)CCO1 87842,C1(NC(C(C=CCCC)O)=O)CCCC(NC(C2CC(=O)N(C(C)(C)C)C2)=O)C1 87843,c1(C(=O)NC(C)CCN(C(=O)CN2CCOCC2)C)cc2c(F)c(F)ccc2s1 87844,c1(C(=O)NCC2C=CC(NC(CCCN(C)C)=O)C2)ccc(F)c(F)c1 87845,C1(CNC(CNC(CNC(CC=CC)=O)=O)=O)CCCC(C#C)C1 87846,c1(OCC(=O)NC(C2CC2CNC(=O)CC2CCC2(C)C)C)ccc(C#N)cc1 87847,C1(CNC(c2cc(C)n(C)n2)c2n(C(C(=O)OC)C)nnn2)CCN(C)CC1 87848,c1(Nc2c(C(=O)NCC(C)(C)C)cc(OC)nc2)ncc2[nH]ncc2n1 87849,c1(C(N2CCC(C)(NC(C3CCC4CC4C3)=O)C2)=O)cc2n(n1)CCNC2=O 87850,C(=O)(C(F)CCC(C)C)NCC(CC(F)(F)F)NC(CCCC=C)=O 87851,C1(c2nn[nH]n2)(C(=O)NC(C(C)C)Cc2cccnc2)CC12CCCC2 87852,c1(C(=O)NCCOCCNC(c2c(C)nncc2)=O)cccc(CO)c1C 87853,c1(OC)cc(S(=O)(=O)N2CC(CNC(c3cc4cccnc4[nH]3)=O)C2)ccc1Br 87854,n1(CC(=O)NCC(=C2CN(C(C3CCC(=O)O3)=O)C2)F)c(=O)oc2ccccc12 87855,c1(C(=O)NC(C2CCCC2)CNC(c2n(CCC)ccc2)=O)ncccc1CC 87856,C=CC1(C(=O)NCC(c2ccc(F)cc2)NC(C2CC2C)=O)CCOCC1 87857,C1(C)(CN(C)C)CCN(CC(=O)NC2(C(C)(F)F)CC2)CC1 87858,CC1CCCC(C(N2CCOCC2CN(C)C(c2cn(C)nc2C(F)F)=O)=O)C1 87859,c1(C(C(=O)NC(C(=O)NCC(=C)Br)C2CC2)C)cncnc1 87860,N1(C(C(CCC)N(C)C)=O)CCC2(CC1)CN(C(=O)Cc1ccc(CC)cc1)C2 87861,N1(C(c2c(OCC)nccc2)=O)CCCCC12CC(NC(=O)CCC(C)(C)C)C2 87862,C1(CCNC(c2c(C)cc[nH]2)=O)CC2CCC(C1)N2C(=O)CCCc1cncs1 87863,CCC(CC)C(C)C(=O)NC1(C)CN(C(=O)CSC(F)F)C1 87864,Cn1cnc2nc(N3CCN(S(C)(=O)=O)CC3)nc(NCc3cc(Cl)ccn3)c12 87865,CN1CCC(CNC(C2C=CCC2)=O)C1c1cccs1 87866,N1(C(c2nccc(OC)c2)=O)CCCC(O)(CNC(C2CC3(CCC3)CO2)=O)C1 87867,C12(C(=O)NC3CC(CNC(COCC(C)C)=O)C3(C)C)CCC(CC1)CC2 87868,n1(CCC(N2CCC(CCNC(C(C(C)OC)O)=O)CC2)=O)cnc([N+](=O)[O-])c1 87869,CC1CC(NCCC(=O)NCC(c2ncccn2)=O)c2nccn21 87870,c1(C(=O)NC(C)CCNC(c2nnn(C(C)(C)C)n2)=O)cc(Cl)ccc1[N+](=O)[O-] 87871,C(=O)(C(CO)C(F)(F)F)NC1C2C(C(=O)NC(C(=O)NC)CC3CC3)C3C(C2)C13 87872,C1(c2ccc(CC)o2)NC(=O)N(C2CC2C(F)(F)F)C2=C1C(=O)OC2 87873,c1(C(N(CCN(C(C(=O)OC)C)C2CC2)C)=O)cc(Cl)ccc1OC(C)C 87874,c1(C(N2C3CCC2CC(CC(F)(F)F)C3)=O)ccc(OC(F)(F)F)cc1[N+](=O)[O-] 87875,c1(C(=O)NCC(O)CNC(C2CC2c2cccs2)=O)ncoc1C1CC1 87876,c1(COCC)cn(CCNC(=O)N(CCC(C)(C)O)C)nn1 87877,Cc1c(N(C)CC2CCCC(C)C2)ncnc1N1CCC(C(C)C)CC1 87878,C1(C(=O)OC)CCOC1C(=O)N(C)CC1(O)CN(C(=O)C(C)CN(C)C)C1 87879,c1(C(=O)NCC2(COC)CN(C(=O)CC(C)(C)C)C2)cc(F)ncc1OC 87880,C1(C)(CNC(C(C(C)C)OCC)=O)CCN(C(=O)CCc2ccoc2)CC1 87881,Cc1nc(CCC(=O)NCC2C(C)CCN2c2nnc(C3CC3)o2)[nH]c1C 87882,CCCCC(C)CCC(=O)N1CC2C(NC(=O)C(C)CC(N)=O)C2C1 87883,C1(C(N(C)CCNC(=O)Cc2cncnc2)=O)CCNC(=O)C1 87884,N1(C(C(=O)NCC=C)C)CCC(O)(C(=O)NCC(C2CCCCC2)C)CC1 87885,c1(CC(=O)NCC(CNC(=O)Cc2cn(C)nc2C)OC)ccnc(F)c1F 87886,Cc1ccc(Br)c(NC(C2CC(NC(=O)Cn3cc(Cl)cn3)C2)=O)c1 87887,C1(C#N)(C(=O)NCC(Cc2ccccc2)N(C)C(c2ccsc2)=O)CCOCC1 87888,CON=CC(=O)N1CC(CNC(c2csc(C(F)F)n2)=O)C1 87889,C1(C(=O)NCc2ccc(C)o2)CSCCN1C(c1cccc(O)n1)=O 87890,n1(CCC)ncc(-c2nc(C3CCCCCC3)nn2C(C)C(C)C)c1C 87891,Cc1[nH]c(C)c(C(=O)N(C)CCOCCN(C)C(C2(C)CCN(C)C2)=O)c1C 87892,C1(CNC(Cc2cc(C)ns2)=O)CCCCN(C(=O)C(N2CCSCC2)C)C1 87893,CC#CCCC(=O)N1CCC(C(COC)NC(=O)C(C)C(C)O)CC1 87894,CC(C)(C)CCCC(C(=O)NCCCF)N1CCCCC1Cc1ccccc1Cl 87895,N1(C(c2c(O)cc(C)nn2)=O)CC(C)CN(C(C2(C#N)CC23CCC3)=O)CC1C 87896,C(CCC(C)C(=O)NC1CCN(C(=O)CCCC2CCCC2)C1C)OC 87897,C1(F)(C(=O)NC(C2CCOC2)CC)CCN(C(c2ccn(COC)n2)=O)CC1 87898,N1(C(c2c(CNC(CNC(CC)=O)=O)ccs2)=O)CCC(O)CC(C)(C)C1 87899,N1(C(CCSCCC)=O)CC2(CCCN(C(=O)C(C)(O)Cc3ccccc3)C2)C1 87900,C(=O)(C1=C2CCCN=C2NN1)NC(C1CCCN(C(CCC=C(C)C)=O)C1)C 87901,C1(CC(=O)N(C2CCN(C(C3CCC(OC)C3)=O)CC2)C)SC2=NCCN2C1=O 87902,C(=O)(CCCC(F)(F)F)NC(CSCC)C(=O)NCCC1CCN(C)C1 87903,C1(NC(c2ccc(CNC(c3ccc(C#C)o3)=O)s2)=O)CCC(C)(C)CC1 87904,c1(CNC(=O)NCc2c(OC)n(C)nc2)cc(F)ccc1C 87905,N1(C(=O)Cc2cc[nH]c2)CCC2CC12C(=O)NC1CCCC1CN=[N+]=[N-] 87906,CN1CC(CC(=O)N(C)CCc2cn(-c3ccc(I)cc3)nn2)C(O)C1 87907,N1(C(c2nnn(CC)c2C)=O)CC(C)N(C(c2cccc(COC)c2)=O)CC1C 87908,C(=O)(C(C)(C)C(F)F)N1CC2C(Cc3ccccc3)(C2)C1.n12nc(cc1O)C(=O)NC2C 87909,O=C(C1=CCCC1)NCC1(O)CC(C(=O)NC2(c3ncccn3)CC2)C1 87910,C1(CC(=O)N(C2CCN(C(C3(Br)CC3)=O)C2)CC)CCC(=O)N1C1CC1 87911,N1(C(c2n(CC(C)C)ncc2)=O)CC2CN(C(=O)Cc3cnc[nH]3)CCC12 87912,c1(OC)c(C(N2C3CCC2CC(NC(c2cc[nH]n2)=O)C3)=O)ccc(Cl)c1C 87913,C1(C(=O)NC2C(CC(=O)NC(C#C)CCC)C(O)C2)NC(=O)OC1C 87914,C1(N(C(CCC2(C#N)CCC2)C(=O)NC(C)(C)C)CC=C)CCN(C(C)=O)CC1 87915,C#CC1(C(=O)NCc2nnc(O)n2C)CCN(C(C2C(C)(C)C2(C)C)=O)C1 87916,Cc1nc2ccc(C(N3CC(NC(C4(C)COC(=O)C4)=O)C3)=O)cc2o1 87917,C12(C(=O)NC3C(CN(C)C(c4ccc(C(N)=O)nc4)=O)CCC3)CCC(CC1)C2 87918,C(=O)(C(C)(C)CCS(C)(=O)=O)NC(Cc1ccc(OC)cc1)(C)CO 87919,N1(C(c2c(N=[N+]=[N-])cccc2)=O)CC2CC(C1)CN(C(=O)C=CS(F)(F)(F)(F)F)C2 87920,CC1(C)CCCCC(NC(=O)C(O)C2CN(C(=O)CNc3ncccn3)C2)C1 87921,CC1CN(C(=O)C(F)C2CCCC2)CC1CC(=O)NC1(C(F)F)CCC1 87922,C1(C(=O)NCC#CC(=O)NCc2cc(OC)no2)CCC(C2CC2)C1 87923,C12(C(N(C(C=C)C)C)=O)CC1CN(C(=O)C=Cc1ccoc1)C2 87924,N1(C(C2C(C)(C)C2)=O)CC2CCCC(NC(c3csc4cc(Cl)cnc34)=O)C2C1 87925,C1(CC)CCCC1(C)C(=O)NCCCN(CCCCNC(C1CCCCC1)=O)C 87926,C12CCCN(C1)C2=O.c1(SC2C(OCP(C)(C)=O)CCC2)ccccc1 87927,c1(CN(C2CCN(C)C2)CC(OC)OC)ccc(F)nc1 87928,Cc1ncc(C(N2CCC(C)C(CNC(c3ccc(O)cc3O)=O)C2)=O)c(C)n1 87929,c1(C(N(CCNC(c2cc(S(=O)(=O)NC)oc2)=O)C)=O)ccc2sc(C)nc2c1 87930,n1(CC(N2C(CNC(C3CC(CC)C3)=O)CC2)=O)ncc(=O)c2ccccc12 87931,Cc1ncnc(C)c1OCC(N1CCN(C(C2CC2F)=O)C(CO)C1)=O 87932,c1(CC)cnc(C(N2CCC(NC(=O)C(C)(C)n3cnnn3)C2C)=O)cn1 87933,C=CCC(C(=O)NCc1nccn1C)NC(C1CCCC1CCC)=O 87934,c1(CC(=O)OC)cccc(C(=O)NCC2C3CN(C(C)C=C(C)C)CC23)c1 87935,c1(C(=O)NCC(CNC(c2c(C)onc2)=O)(C)C)nn2c(c1Br)CCC2 87936,CCCC(CC(=O)Nc1cscc1C)NC(C1CCCN(C)C1)=O 87937,c1(C(C(=O)NCCOCC)N(CCCCCCCO)C)cc(NCC)nc(Cl)c1 87938,C1(NC(CSCC)=O)CCCC(N(C(=O)CC2CN(C)C2)C)C1 87939,C=C1CC(C(=O)NCc2ncco2)(CNC(=O)C(N2CCOC2=O)C)C1 87940,c1(C(N2CCCC(C)(NC(C3ON=C(C)C3)=O)C2)=O)cccc2c1OCCN2C 87941,Cc1ncnc(C(N2CCSCC2C(N)=O)=O)c1C.C1(CCF)C(=O)N1 87942,Cc1cc(-c2ccsc2)ncc1C(=O)NC1CCC(NC(c2cocn2)=O)CC1 87943,N1(C(CN2CCN(C(CC3N(C)CC=CC3)=O)CC2)=O)CC(=O)NCC12CC2 87944,N1(C(CCOC(C)C)=O)CC2C(C(N3CCOCC3CC3CC3)=O)C2C1 87945,c1(OC)ccc2c(c1)CCC2C(=O)NCC(CNC(C12CC(F)(C1)C2)=O)C(F)(F)F 87946,C1(NC(C2CCN(C(C(C3CCOCC3)C)=O)CC2)=O)CC2(C1)CN(C)C2 87947,Cc1cc(NC(=O)CS(=O)(=O)C2CC2)ccc1S(C)(=O)=O.C1CO1 87948,c1(C(CNC(c2cccc(P(C)(C)=O)n2)C)=O)ccc2c(c1)CC(C)O2 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88002,C1(CC(N)=O)(NC(=O)C2=COCC2)CCN(C(c2n[nH]c3c2CCC3)=O)CC1 88003,c1(C(=O)NCCC(C)NC(C=Cc2c(C)cncc2)=O)ccc(P(C)(C)=O)cc1 88004,CCCCN=C(NCCc1ccc(F)cc1F)NCC1CCCN1CCC 88005,CCCCC(C(=O)NCC1CCN1C(C1CCC1(F)F)=O)C(C)C 88006,Cc1csn1CC(=O)NCCN(C(=O)CC1CCCC1)C1CC1 88007,N1(C(CC(C)F)=O)CC2(CCN(C(=O)CNN)C2)C1.c1(C(CNC=O)=O)ccccc1 88008,C(CC(=O)NCC1CN(C(=O)C=C2CCCCC2)CC1O)(C(C)C)OCC 88009,S(=O)(=O)(c1cnn2ccc(=NC(C)CCOC)[nH]c12)NC(C(CC)CC)C 88010,C1(C(=O)NC2CC(C)(NC(c3cn(C)nn3)=O)C2)C2CCN(CC2)S1(=O)=O 88011,c1(C(N(CCCn2cc(-c3nc(C)c(C)s3)nn2)C)=O)ccc2ncsc2c1 88012,N1(C(=O)Nc2ccnn2C2CNC2)CCC2(CCCCO2)C1 88013,C(c1ccc(F)cc1Cl)=CC(N1CC2CN(C(CCCC#C)=O)CC21)=O 88014,Cc1c(NC(=O)CC2CN(C(C3CCCO3)=O)CCO2)ccc(Br)c1Cl 88015,n1(CC)nc(C)cc1C(N1CC(C)(NC(c2cccc(C(C)=O)c2)=O)C1)=O 88016,c1(C(=O)NCC2CCCN(C(C3(C)N(C)CCC3)=O)C2)ccc2nc(O)[nH]c2c1 88017,N1(C(c2cncc(OC)c2)=O)CCC(C)C(NC(C2CCCN2C2CC2)=O)C1C 88018,C1(CNC(CC2(C)CCC2)=O)CC(F)CN1C(=O)CNC1CCCC1 88019,c1(CCCNC(N2CCC(c3cnccn3)C2)=O)cnccn1 88020,Cc1ccc(F)c(O)c1CNCCC(C)(C)NC(=O)Cn1cc(C2CC2)cn1 88021,CCC1=NOC(C(N2CC=CC2CNC(c2cnoc2COC)=O)=O)C1 88022,CCCCC(C(=O)NC1CCN(c2cc(F)ncn2)C1C)NC(N)=O 88023,N1(C(CC)=O)CC2CCOC2(CNC(c2cc(C)ccc2NS(C)(=O)=O)=O)C1 88024,c1(OC(Cn2cc(C(=O)OC)nn2)=O)ccc(C)c(N(C)C)c1 88025,c1(C(=O)NCC2N(C(c3ccccc3N3CCCCC3)=O)CC2)cc(I)ccc1O 88026,c1(OCCCC)ccc(C(=O)NCC2(C)CC2(Cl)Cl)cc1OCCC 88027,c1(CC(=O)N(C(C)C)CCN(C)C(c2ccoc2Cl)=O)cn(C)nn1 88028,C1(NC(C=C(C)C(C)C)=O)CC2(CCCN(C(C3(C#N)CC(C)C3)=O)C2)C1 88029,N1(C(CC)=O)CCS(=O)(=O)C(CNC(=O)Cc2csc(-c3ccc(F)cc3)n2)C1 88030,N1(C(CNN2C(C)CCCC2)=O)CC2(C1)CC(C)(O)C2 88031,C1(C(=O)NCc2ncc(C3CC3)s2)CC(N=[N+]=[N-])CN1C(C1CCC(O)CC1)=O 88032,CC(C)CCC(O)C(=O)N(C(C)C(N1CC(O)CC(O)C1)=O)C 88033,c1(OCCNC(=NC)NCC(c2cnccn2)(C)C)ccccc1C#N 88034,N1(C(COCCC)=O)CCC(C)(C(=O)NCC2CN(C(C)C)CCO2)CC1 88035,C1(C)(CNC(C(C(C)C)NC(C)=O)=O)CN(C(=O)C(C2CCCCC2)C)CC1C 88036,Cc1ccc(N)c(C(=O)NC2CN(C(=O)C(n3nc(C)cc3C)C)CC2(C)C)c1 88037,C1(N(C(=O)CCc2csc(C)n2)CC#C)CCN(C(C2CCC(C)S2)=O)CC1 88038,c1(CC(N2CC3CC(NC(CN(C)CC)=O)C3C2)=O)ccc2n[nH]cc2c1 88039,N1(C(CC(C)(C)C)=O)CC2CCCC(NC(c3coc4c(F)cccc34)=O)C2C1 88040,N1(C(CCN(C)CC)=O)CC(NC(c2cc(C(C)C)no2)=O)CC(O)C1 88041,c1(C(=O)NCC2C(NC(CCC=C)=O)CC2)c(C)ccc(F)c1O 88042,c1(C(c2nnnn2C2CCCCCC2)NCC(COCC)C)oc(CC)nc1C 88043,c1(NCc2cc(C)oc2)nc(=NCc2cc(C)n(C)c2C)[nH]c2c(C)nn(C)c12 88044,C(=O)(C1CNC(=O)c2ccnn21)N(CCCCCCNC(C(CC)(C)CO)=O)C 88045,CC(C(=O)NC1CCCOC1C1CCN(C(C2CCCC2)=O)CC1)C(C)(F)F 88046,C(C)(C)(CCCC(=O)N1CCC2C(C(N)=O)C2C1)NC(CCc1n(C)cnn1)=O 88047,C(=O)(C(F)CC(C)(C)NC(c1cc2ccccn2n1)=O)N(C)CCc1cccs1 88048,C1(OC)CCCC2(COC3CC3)CC12.c12ccc(cc1)Cc1nc-2no1 88049,C(C(COC)C(=O)N1CCCC(CCCO)C1)OC 88050,CCC(C)C(O)C(=O)NC(C)Cn1cc(C)cn1 88051,c1(CCC)nc(C(=O)NCC(C2CCCN2C(C2CC2CN(C)C)=O)(C)C)cs1 88052,C(=O)(C(CCF)NC(C1(C)CCC(=O)N1)=O)N1C(C)(CCC)CC1 88053,N1(C(CN(C2CC2)CC)=O)CCC2CC1CN2C(C1CCCCC12CCC2)=O 88054,C(=O)(CC1OCCc2ccccc21)NC(CN(C(c1[nH]cc(CC)c1)=O)C)C 88055,C1(C(=O)NC2CCCC(CNC(Cc3c(C)non3)=O)C2)C(C)(C)OC1(C)C 88056,Cc1cc(C(N2CCC(NC(=O)CC(C)O)C2C2CC2)=O)c(N)s1 88057,C(C(=O)OCC(c1nn[nH]n1)=O)(C(C)C)NC(C(n1cc(C)nc1)(C)C)=O 88058,C#CCC(CC(=O)NCCN(C(C)C)C1CC1)NC(C1C2CCCC12)=O 88059,C(=O)(CCCCCC#N)NC1CC2(CN(C(Cc3c(Cl)cn(C)n3)=O)C2)C1 88060,CC(c1cccnc1)=CC(=O)NC1CCN(C(c2conc2C)=O)CC1F 88061,Cc1cc(C(N2CCC(NC(c3cncc(N4CCCC4)n3)=O)C2C)=O)c(C)nn1 88062,N1(Cc2c(OCC(=C)C)cccc2)CCC(O)C(C(N2CCOC(O)C2)=O)C1 88063,C(CCN=C(NC1CC1C(F)F)N1CCN(c2ccc(F)c(F)c2)CC1)OC(F)F 88064,CC1CC(CNC(C2(N3CCCCC3)CCCC2)=O)CN1C(=O)Cn1cnnn1 88065,C(=O)C(C)P(C)(C)=O.C(C(CO)N)N(C(=O)CSC(C)(C)C)C 88066,N1(C(C(CC)O)=O)C(C(=O)NCCc2ccc(C)s2)CC2CCCCC12 88067,C(CO)(C(=O)N1CC(NS(N)(=O)=O)C1)NC(CCC(=O)N(C)C)=O 88068,CN(C)NC(=O)CCC(=O)NC1(C)CCN(C(c2ccc(C#N)o2)=O)CC1 88069,c1(C(=O)NC2CCN(C(C3COC3)=O)CC2O)ncn2ccccc12 88070,C1(C(N(C2CCN(C(=O)C(=O)N3CCCC3)C2)C)=O)CCc2cncn2C1 88071,C1(N(c2ccc(-c3ccccc3)cc2)C)CCCN(C(=O)C(=O)NC2CCCC2)C1 88072,C(=O)(CC(C)(F)F)NC(C=CC(=O)N(CCCC#C)CC)(C)C 88073,c1(CC(N2CC3CN(C(c4c(C)coc4)=O)CC3C2)=O)coc2cc(O)ccc12 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88160,c1(CC)[nH]c(=N)sc1C(=O)N(CC(C)N(C)C(c1cncnc1C)=O)C 88161,N1(Cc2c(C)nc[nH]2)CCc2nc(C(=O)NC3CCC(N(C)C)CC3)cn2CC1 88162,N1(C(c2n(CC=C)ccn2)=O)CCCC2(NC(c3ccc(COC)s3)=O)CC2C1 88163,c1(C)cccc(OC(F)(F)C(F)(F)F)c1.C1(C(C)N)CCCN(c2nccs2)C1 88164,c1(C(N(CC(O)CNC(=O)C#CC2CC2)C)=O)cnc2c(F)c(F)ccc2c1 88165,c1(C(=O)NCCC(C(C)C)NC(C(COC)C)=O)cccc2ncc(Br)n12 88166,C1(C(=O)NC(C(=O)OC)CC2CC2)CCCN(C(c2cc(OC)n(C)n2)=O)C1 88167,CCC(C)(C)CCCC(=O)NCC1CCCC(NC(=O)C(C#N)C(C)(C)C)C1 88168,c1(NC(C(C)C)=O)cccc(C(=O)NC2CCCC(CNC(C3(O)CC3)=O)C2)c1 88169,c1(C(N(C)CC2(O)CCN(C(=O)Cn3cnnn3)C2)=O)cc2c(ccn2C)[nH]1 88170,N1(C(=O)NCc2cn(C(CC)C)nc2)CCc2cc(C)ccc2C1C 88171,N1(C(C(CN(C(CN(CCC#C)C)=O)C)(C)C)=O)CC2OCCN(C)C2C1 88172,N1(c2c(C)cccc2)CCC2(CCN(c3nccc(N4CC=CCC4)n3)C2)C1 88173,c1(C(=O)NC2CCC(NC(c3c(OC)cc(Cl)nc3)=O)C2)cc(C)c(F)cc1Br 88174,c1(C(=O)NC2(C3N(C(CN(CCOC)C)=O)CCC3)CC2)cc(C)cc(F)c1 88175,C1(C(=O)NC(C)(C)CNC(C2CC(C)(F)C2)=O)CCCC1(F)F 88176,c1(C(N2C(CCNC(=O)C3=CCCCC3)CCC2)=O)cc2cccn2cn1 88177,C#CC1(C(=O)NCC(C)N(C)C2CC2)CCN(C(=O)CC(C)C2CCCC2)C1 88178,CCC(CC(=O)NCC(CC(C)C)NC(C12CC(OC(C)=O)(C1)C2)=O)C(C)(C)C 88179,c1(C(=O)NC(CCNC(C2(CC)CCCC2)=O)C)nn(C)c2c1CC(C)(C)CC2 88180,C1(C(=O)NCC(CCNC(=O)CCc2cnco2)O)CCc2ccccc2C1 88181,C1(C(=O)NCC2(NC(Cn3nc(C)n(C)c3=O)=O)CC2)CCCCN1S(N)(=O)=O 88182,C1(C(=O)NC2(CC=C)CCOC2)CCCC(NC(=O)CNC(=O)CN(C)C)C1 88183,c1(C(=O)OC)cnc(NC2CC3(C2)CC3NC(c2[nH]nc(OC)c2Cl)=O)cn1 88184,C1(C(F)(F)F)(C(=O)NC(CC)CNC(c2ccnnc2)=O)CC=CCO1 88185,N1(C(C)COc2ccccc2)CCC(O)(C(=O)NC2CSC2)CC1 88186,N1(C(c2c(C(=O)OCC)n[nH]c2)C(=O)NCC)CCOC2(CCN(C(C)=O)C2)C1 88187,N1(C(COCC(=O)OC)=O)CCCCC1CNC(=O)C(C)(O)C1CC1 88188,c1(OC)nn(C)cc1N(C)C(C1CC(CNC(=O)CCCC2CC2)C1)=O 88189,N1(C(CCCOCC)=O)CCC(NC(c2ccc(SCC)cc2)=O)C12CCCC2 88190,N1(C(C=CCC)=O)CCCCC1CN(C(C1(C)COC1)=O)CC 88191,N1(C(c2cc(CCNC(c3cnc(C)o3)=O)on2)=O)CCOC2CC12 88192,c12ccccc1N(C)C(COC(=O)NC)C(=O)NCC(OC)CCNC2=O 88193,C1(CC)CC(C(=O)NCC(C)CC(=O)OC)CCN1C(c1c[nH]c(=N)c(C)c1)=O 88194,N1(C(CSCC#C)=O)CCC(O)(CCNC(=O)C(c2nc(C)cs2)C)C1 88195,C1(CC#C)(C(=O)NCC(CCOC)NC(=O)C=Cc2nccs2)CCCCO1 88196,C1(CNC(C(CO)OC)=O)C2CN(C(=O)C(F)(F)c3ccccc3)CC12 88197,N1(C(C(C(CCN2C(CC(=O)N)CC2=O)C)F)=O)CC(C(N)=O)C2(CC2)C1 88198,n1(CC)nc(C(=O)NC2COCC2CNC(=O)COCC(C)(C)C)c2c1CCOC2 88199,n1(CC)cnc(C(=O)NCC2(NC(c3ccn(CC(C)C)n3)=O)CCCC2)n1 88200,c1(OCC)cc2ccc(-c3ccc4c(c3)CC(=O)N4)cc2s1.n12nccc1c1cccn21 88201,N1(C(c2c(C)noc2N)=O)CCC2(CCC(NC(=O)Cc3cocn3)C2)CC1 88202,C1(C2CN(C(=O)CN=S(C)(C)=O)C2)(NC(C(=C(C)C2CC2)F)=O)CC1 88203,c1(C(N2CC(C)C(O)C2)C(CCCCCC)=O)cccc2c1CCO2.N 88204,N1(CC(N2C(CC(=O)NC(COCC)CO)CC2)=O)CC(=O)NC1=O 88205,c1(CC(N2CC(N(C(C3N(CC)CC3)=O)C)C(O)C2)=O)cc(C)ccc1OC 88206,C1(C(N2C(CC)CN(C(=O)CCCF)CC2)=O)CCC(C2CC2)CC1 88207,C1(CCNC(c2csc(C3CC3)n2)=O)CCCCN1C(c1cc[nH]n1)=O 88208,C#CC1(O)CC(C(=O)NC2(C(=O)NCCNS(=O)(=O)CC)CCSC2)C1 88209,CCC(C(=O)NCC1(OC)CC1)N(C(=O)C(C)(F)c1ccon1)C 88210,c1(OC)ncc(C(N2CCC(C)(C(=O)OC(C)(C)C)C2)=O)cc1[N+](=O)[O-] 88211,C1(OC)CCCC1C(=O)NC(C)C(=O)NCCc1cccnc1 88212,CC(CNC(C1CN(C)CCN1C)=O)C(F)C(=O)NC1CCNC(=O)C1 88213,c1(NCC(CC)CCO)ccc(S(=O)(=O)NCC(C2CCOCC2)OC)c(Cl)c1 88214,c1(C(=O)NC2CCC(CNC(CS(N)(=O)=O)=O)C2)cnc2nccn2c1 88215,C1(CNC(CSCC#C)=O)COC(CNC(=O)COCCC(C)C)C1 88216,C1(C(=O)NC(C2(CNC(c3cc(C)n(C)c3)=O)CC2)C)CCC(C)(C)OC1 88217,N1(C(CN(C2CC2)CC)=O)CC2CC2(C(=O)NC(CO)C(=O)O)C1 88218,N1(N2CC(C(N(C)C)=O)C2)CC2CC1CN2C(=O)CC1(C)CC1 88219,N1(C(C2(C#C)CCCC2)=O)CCC2(CCCC2CNC(C2CCNC2=O)=O)CC1 88220,N1(C(=O)OC)CSCC1C(=O)NCC1(NC(=O)CCCc2ccccn2)CCC1 88221,C1(NC(C(CNC(C2C(Cl)(C(=O)OC)C2)=O)OC)=O)CC(C)(C)C12CCC2 88222,N1(C(C(C=C)c2ccccc2)=O)CC2(CCC(NC(c3cnncc3O)=O)CC2)C1 88223,CC1OC2(C(=O)NC3CCN(C(c4cc(C(N)=O)co4)=O)C3)CC1C2 88224,C#CCCCCC(=O)NC1CCC(NC(C2(CCOC)CC2)=O)C1 88225,CCC(CC)CCC(=O)NCCCN(C(c1cc(OC)ccc1CC)=O)C1CC1 88226,Cc1cc(C(N2CC3CC3(CNC(=O)CC3CCCC3O)C2)=O)n(C2CCC2)n1 88227,N1(C(COCCC)=O)CCC(C)CC1CNC(=O)CCc1cccnc1 88228,N1(C(C=C(COC)C)=O)C2CCCC1CC(NC(C1CC(n3cnnc3)C1)=O)C2 88229,c1(-c2nnc(N3C(CCC)CCC3)n2CCC#N)cc2ccccc2o1 88230,C1(F)(C(N2CC=CC(NC(c3c(CCCC)ocn3)=O)C2)=O)CCS(=O)(=O)C1 88231,CC1(C)CCC(NC(c2cncnc2)=O)C(CNC(=O)C2=CCCOC2)C1 88232,c1(C(N2CCC(NC(C3C4(CC4)C34CC4)=O)C(F)C2)=O)cccc2c1COCC2 88233,C1(CC(=O)NCC2(O)CN(C(c3c[nH]nc3C(F)(F)F)=O)C2)CC2CCC(C1)C2 88234,N1(CC(=O)NCC2C(C)CN(C(=O)C=CC3CCOC3)C2)CCCCCCC1=O 88235,Cc1cc(F)ccc1C(F)(F)C(=O)NC1C2CN(C(C3CCCOCC3)=O)CC12 88236,CCC(C)(CO)C(=O)NCc1cncc(C(=O)NCCCCCC2CC2)c1 88237,CN1CCC2CCC(C1)N2C(=O)CC1CCCCC1NC(=O)C1=COCCC1 88238,C1(CNC(C2(C)ON=C(C)C2)=O)CN(C(=O)CC2(C)CCCCC2)CC12CCC2 88239,N1(C(C(=O)NC(CC)C)CCC2CC2C)CC(C(=O)OC)C(C2CCCCC2)C1 88240,c1(NC(C(F)=CC)=O)ccc(NC(c2cc(CC(C)C)c[nH]2)=O)cc1C 88241,N1(C(CCN(CCC)C)=O)CCC(C2(O)CN(C(=O)C=CI)C2)CC1 88242,N1(C(c2cnc(C(C)=O)s2)=O)CC2CC1CCC2NC(=O)C(C)SC(F)(F)F 88243,c1(OCC(N2CCC(NC(C3C(COC)C3)=O)C2)=O)ccc(C)cc1Cl 88244,c1(OC)ccc(F)cc1C(=O)C(=O)N(C1CCCN(C(c2cc(F)n(C)n2)=O)C1)C 88245,N1(C(CCc2n(C)ncc2)=O)CCOCC1CNC(c1cnc(Cl)s1)=O 88246,CC(F)(F)C(C)(C)C(=O)NCCC1CC(F)(F)CN1C(C1COCCN1C)=O 88247,c1(C(N2CCC(N3CCOC3=O)C2)C(=O)NCCOC)cnc(OC)c(Cl)c1 88248,C(=O)(C(O)C(F)(F)F)N(CC(CC)NC(=O)C(O)Cc1ccccn1)CC 88249,c1(C(=O)NC2CCC(NC(C3N(C)CCCCC3)=O)CC2)cnc2c(c1)COC2 88250,N1(C(C(CCC)F)=O)CC(CNC(c2c(C)noc2C2CC2)=O)CC(C)C1 88251,C(CO)(C(N)=O)NC(CC)Cc1nnnn1C 88252,c1(NC(CN2C(CO)CC(NC(C3N(C)C(=O)OC3)=O)C2)=O)ccc(Cl)cc1F 88253,C(C(C(C)(C)C)NC(=O)C=CCOC1CCOCC1)NC(COCCC#C)=O 88254,CCC(C)C(=O)NCC(=O)NCC(c1ccccc1)CNC(=O)CCCC1CC1 88255,CCCCCC(C)C(=O)N1CCN(CSc2nn(C)c3ccccc23)CC1C#N 88256,C(=O)(C(F)C(F)(F)C(F)(F)F)NCC1C(NC(C(=O)NCC)=O)CC1 88257,N1(C2CN(C(COC)=O)C2)CC(NC(=O)CC2(C)CC2)CC1=O 88258,C1(NC(=O)CCc2cc(C3CCC3)on2)(CO)CCN(C(=O)CC(F)F)C1 88259,c1(C(=O)NCC2OCC(CNC(=O)C(C)(C3CC3)OC)C2)n[nH]c2c1CCCCC2 88260,C1(CC(=O)NCC2N(C(C3(O)CC(C)(C)C3)=O)CC2)Cc2ccc(Br)cc2C1 88261,C1(C(=O)NCCN(C(C2CCCN2C(=O)NC)=O)CC)(C)CC(F)(F)C1.CC 88262,c1(NC)cnncc1C(=O)NC1CCC(CNC(c2cc(O)ncn2)=O)C1 88263,CC(CC(=O)N(C)CCNC(=O)C1=NNC(C(F)F)C1)C(C)(C)C 88264,CCC(CC(=O)N1CC2(C)CC1(C(=O)NCc1ncnn1C(C)C)C2)CC(C)C 88265,C1(NC(c2cc(C(N)=O)[nH]c2)=O)CC2CCC1(NC(C1CC=CC(O)C1)=O)C2 88266,C(=O)(C1c2c[nH]nc2CN1C(=O)C#CC1(C)COC1)N1C(C)C(N(C)C)CC1 88267,c1(CC(=O)NC2CN(C(C3CC(CC)C3)=O)CC2F)c[nH]c2ccc(Cl)cc12 88268,O=C1CCCC(C(N2CCC(O)CC2C(=O)NC2CCN(CCF)C2)=O)CC1 88269,CON(C)C(=O)C(C)N1CCC(F)(CN)C1 88270,N1(C(C(C)C2CC2)=O)CC2(CCC(CNC(=O)Cc3ccc(Cl)c(F)c3)O2)C1 88271,c1(C(N2CC(SC)C(NC(C3(C)CCCO3)=O)C2)=O)ccc2n[nH]c(C)c2c1Cl 88272,N1(C(CCNC(C)=O)=O)CCOC2(C1)CN(C(c1cc(C)cc(Cl)c1)=O)C2 88273,CC1=NOC(CC(=O)NC(C)(C)CN(C(=O)C=Cc2cncs2)C)C1 88274,N1(C(CCOCC)=O)CCOCC2(COCCN2C(=O)C(O)Cn2cncn2)C1 88275,CC(C)C(C)CC(=O)NC(CC1CC1)C(=O)N(C1(c2cc[nH]n2)CC1)C 88276,c1(CC(=O)N(CCC(=O)NC2CCSC2)CC=C)ccnn1C 88277,c1(NC(CC2CC(OC)C2)=O)ccc(C2CCCN(S(=O)(=O)CCCl)C2)cc1 88278,N1(C(CC(=O)OCC)=O)CC(NC(=O)Cc2ncc(C)s2)CC1(C)COC 88279,CN1CCC(NC(c2ccc(N3CCCC(C)(N(C)C)C3)cc2)=O)C(C#N)C1 88280,c1(N(C2CCN(C(=O)C(c3ccccc3Cl)O)C2)C)cnc(C#N)cn1 88281,C12(CNC(C(CCO)N(C)C)=O)CCC1CN(C(=O)Cc1cc[nH]c1)C2 88282,N1(C(c2cc(C)c(Cl)cc2F)=O)CCC(NC(C2CC(C)C2)=O)CC(C)(C)C1 88283,CC(C(C)(C)C)=CC(N1CCC(NC(=O)CCc2cc[nH]n2)C1)=O 88284,CCC(CO)C(=O)NCCC1(O)CN(C(=O)C(F)(F)C2CCOCC2)C1 88285,N1(C(=O)NC(C(=O)OC)C)CCC(F)(F)C(NC(c2cc(Br)ncc2F)=O)C1 88286,C(CCC(=O)NC1CCOC2(CCC2)C1)(C(C)C)NC(C(c1ccn(C)n1)C)=O 88287,c1(CC(=O)NCC2CCCC(NC(c3csnn3)=O)C2)nc([N+](=O)[O-])n[nH]1 88288,N1(C(C2(C)CC3CC3C2)=O)CCN(C(=O)CCCN=[N+]=[N-])C(CCO)C1 88289,c1(NCCCC)ccc(C(N2CC(F)(CNC(C3CC3C#N)=O)C2)=O)cc1 88290,C1(N(C(=O)CCN2CCOCC2)C)CCC2CN(C(c3ccoc3Cl)=O)CC12 88291,n1(CCCN(C(=O)CSC2CCCCO2)C)cc(C2CCCO2)nn1 88292,O=C(CC1=CCCCC1)N1CCC(F)(CNC(=O)C(F)(F)C(O)C2CC2)CC1 88293,C1(C(=O)NC(CC=C)C(=O)N(C(C)CCO)C)CCCC12CCC2 88294,C1(C(F)(F)F)(NC2CCCO2)CCN(C(C2CCC(F)(F)C2O)=O)CC1 88295,CC(O)(CNC(c1conc1CNC(C1(CO)CCOC1)=O)=O)C(F)(F)F 88296,c1(C(N2CCC(N(CCC)C(c3ccc(C)cc3)=O)C2)=O)cc(F)c(N)cc1F 88297,c1(C(=O)NCCCCC(C)NC(=O)C(F)(F)C2CC2)cccc2c1CCC2=O 88298,C1(NC(=O)CCc2ncc[nH]2)CCC(c2cn(CCC(F)(F)CO)nn2)CC1 88299,C1(NC(c2scc(C)c2)=O)C2CC1N(C(=O)CSc1nnnn1C1CCCC1)C2 88300,c1(C(=O)NCC2(CCCNC(COCC=C)=O)CCCC2)cc2sccc2cn1 88301,CN1CCN(C2CCCC2c2ccc(NC(=O)COC3CCCCC3)cc2)CC1 88302,c1(CC)ccc2c(c1)C(CC(=O)N1CCCC1CCNC(=O)C(C)(C)O)C(=O)N2 88303,N1(C(CCOCC#C)=O)CCC2CN(C(C3OCCN(C)C3=O)=O)CC12 88304,C1(CC)CCCN(C(C2CC(SC)C2)=O)C1C(=O)NC1CCN(OCC)CC1 88305,c1(CNC(=O)CC2CCCN2C(=O)CC2CCCC3CC23)ccc(F)c(F)c1 88306,C1(C(=O)NC2C(CNC(CSCCCC)=O)CCC2)COCCN1C(CC)CC 88307,C1(C(=O)OCC)(C(C(c2cc(OCC)cs2)=O)=O)CCCO1.C(C(C1CC1)NC)N 88308,C(=O)(CS(=O)(=O)C1CC1)NCC1CCN(C(C(N2CCCOCC2)C)=O)CC1 88309,CN1C2CCCC1CN(C(=O)C(c1ccccc1)NC(=O)CC1=NNC(=O)C1)C2 88310,c1(N(C(c2cnc(C)[nH]2)=O)CC2CC2)ccc(Cl)cc1 88311,C(=O)(C1CCCn2cnnc21)N1CCC(C2N(C(C(C)CO)=O)CCC2)CC1 88312,CC1(C(=O)Nc2cnccc2Cl)CCCN(C(=O)CCc2cnccn2)C1 88313,c1(C(=O)NC2CCN(C(CSCCCC)=O)CC2)ccnc2c1ccn2C 88314,N1(C(Cc2c(C)cccc2)=O)CCC2CCC12CNC(c1c(C)nc(C)n1O)=O 88315,C(=O)(CS(=O)(=O)CCO)NCC1(C(C)(C)C)CCN(C(C(F)OC)=O)C1 88316,C(CCCC(C)NC(c1cnn(CC)n1)=O)NC(C(C)(C)OCC)=O 88317,c1(NC(C)CCc2ccccc2F)nccc(=NCC2(CCO)CC2)[nH]1 88318,c1(C(COC)C)nc(-c2ccc(C3CC3)cc2)nn1CC1CCCCC1 88319,N1(CC(=O)NCC(N(C(CCCCC#C)=O)C)C2CC2)CCc2ccccc21 88320,C1(C(=O)NCCc2ccc(F)cc2)CCN(Cc2ccc(F)cc2O)CC1O 88321,N(C(=NC1CCS(=O)(=O)C1)NCC1CC(C)(C)C1)C1CC(OC)C1 88322,C#CCCCCCC(=O)NCC1C2CN(C(=O)CC(C)N(C)C)CC12 88323,S(=O)(=O)(CC(=O)NC1CCCC1NC(c1nccn1C(C)C)=O)NC 88324,C1(CC(=O)N(CCCC=C)C)CCCN(C(C2CCCN2CC)=O)CC1 88325,C(=O)(C1CCCc2ncnn21)N1CC(O)CC(NC(CC2(C)CCC2)=O)C1 88326,Cc1nn(CC(=O)NC2C3CN(C(=O)C(C)CC4CC4)CC23)c(C)c1Cl 88327,Cc1cc(C(=O)NCc2cn(C(C)C(C)O)nn2)n2nccc2n1 88328,c1(-c2cn(CCCNC(CC3CCC(=O)N3)=O)nn2)cccnc1Cl 88329,N1(CCC(=O)NC)CCCC(NC(=O)C(Cc2ccccc2)NC)C1 88330,Cc1n[nH]c2cnc(C(=O)NCC(C(C)C(C)C)NC(c3nocc3Cl)=O)cc12 88331,N1(C(C(CSC)OC)=O)CC(NC(=O)CCc2cncc(O)c2)C(C2CC2)C1 88332,C1(C(=O)OC)CC(NC(=O)NC(c2ncc(Br)cc2C)C)CC(C)(C)O1 88333,N(C1CCCc2cc(CNC(=O)C=Cc3ncco3)ccc21)C(C(C)=C(C)C)=O 88334,C1(OC)(OC)CCC1C(=O)NC(C)C=CC(=O)NC(C)CC1CC1 88335,C(=O)(C(=O)CCC(C)(C)C)N1C(C)CN(C(c2cc([N+](=O)[O-])nn2C)=O)CCC1 88336,N1(C(CC2C(OC)CC2)=O)CCN(C(C2CS(=O)(=O)CN2C(C)=O)=O)CC1CO 88337,N1(C(C(C)(C)C)=O)CCC2(CC1)CN(C(C1Cc3cccc(F)c3O1)=O)C2 88338,c1(C(N2C(C(N(CCCO)CC#C)=O)CC2C)=O)ccc(CC)cn1 88339,C1(C(=O)NC2(C(=O)NC)CCCC2)COCCC1NC(c1cnsc1)=O 88340,Nc1ccc(C(N2CC3CC(NC(=O)Cc4ccoc4)C3C2)=O)c2c1CCCC2 88341,C1(NC(CN2CCC(C)CC2)=O)CC(F)CN(C(c2cc(C(N)=O)no2)=O)C1 88342,CC(CC(F)(F)F)C(=O)Nc1ncc(C(C)(C)O)s1 88343,c1(OC)ccccc1C(C)(C)NC(=O)NCc1ncccc1C(F)F 88344,c1(C(=O)NCC(C2C(C)C2(F)F)=O)cc(-n2ccnc2)ncn1 88345,C1(OCC(=O)NCCC(C)NC(C2(CCF)CCOCC2)=O)CCC(F)(F)CC1 88346,c1(-c2nc(C(C3CCCCC3)C)n(CCF)n2)ccc2ccccc2n1 88347,N1(C(=O)Cn2ccc(C3CC3)n2)CCCN(C(c2n[nH]cc2[N+](=O)[O-])=O)CC1 88348,CC1=C(C(=O)N2CCC(NC(C34CCCC3C4)=O)CC2C)C(=O)OC1(C)C 88349,c1(CC(=O)NCCN(CCC)C(c2csc(Br)c2)=O)cc(OC)no1 88350,C1(CC(C)(C)C)CN(C(=O)Cc2cn[nH]c2)CC1NC(C1(C)CCCCO1)=O 88351,CCC(CC(F)F)C(=O)N1CCN(C(c2cscc2C(N)=O)=O)CC1 88352,N1(C(CCC#C)=O)CCC(N(C(=O)CCC=C(C)C)CC#C)CC1 88353,CC(CN(C)C)N=c1[nH]c2c(c(=NC(C)c3ncc(C(F)(F)F)[nH]3)[nH]1)CCC2 88354,n1(CCCNC(C(=O)NCCNC(CCNC(N)=O)=O)=O)cc(Br)cn1 88355,c1(CC(=O)NCC2(OC)CN(C(C3OCCCC3(C)C)=O)C2)ccnc(F)c1F 88356,c1(CC)[nH]nc(C(=O)NCCC(C)NC(=O)C(c2ccnn2C)C)c1[N+](=O)[O-] 88357,N#CC1(C(=O)NCC2(NC(=O)Cc3ccccc3)CCC2)CCOCC1 88358,Cc1cc(CNC(c2conc2C(C)NC(=O)C2CC2)=O)n(C)n1 88359,Cc1nc(F)ccc1NC(N1CC(SCC(C)C)C1)=O 88360,Cc1c(F)cc(C(N2CCC(NC(C3CCc4n[nH]cc4C3)=O)C2)=O)c(F)c1N 88361,Cc1nc(C(N2CCCC(n3cc(CNC(=O)C(F)C4CC4)nn3)C2)=O)c(C)o1 88362,c1(CNC(c2cc(CCNC(COCC(=C)C)=O)on2)=O)ccc(O)c(F)c1 88363,c1(C(=O)NC2C(CNC(C3C(C(C)(F)F)C3)=O)C2)ccc(CC2SCCS2)cc1 88364,C(C(=O)NCCc1cn(Cc2cc(C)no2)nn1)(C(C(C)C)OC)OC 88365,Cc1nc(CO)sc1C(=O)NCC(C)NC(c1nc(=N)cc[nH]1)=O 88366,c1(C(N(CCOCCNC(C(C(C)O)C)=O)C)=O)ccc(F)c2ccoc12 88367,Cc1nc[nH]c1CNC(=O)CCNC(c1cccnn1)=O 88368,C1(NC(C(C)=C(CC)C)=O)C=CCN(C(=O)C(C)NC(c2cccs2)=O)C1 88369,Cc1[nH][nH]c1C(=O)NCCCc1cn(C2CC(O)C2)nn1 88370,C1(O)(CNC(C2(F)CN(C(c3c(C)nc(CC)o3)=O)C2)=O)CCC(C)(C)C1 88371,C=CCC(C)(C)CC(=O)NCCCCNC(c1c(C)ncnc1O)=O 88372,C1(NC(=O)CC2CNC(=O)O2)CN(C(c2ccnc3[nH]cnc23)=O)C2(CCC2)C1 88373,Cc1cnc(Cl)c(S(=O)(=O)N2CCSCC2C(=O)Nc2ccnc(Cl)c2I)c1 88374,C=CCC(C)(C)CC(=O)N1CCN(C(c2coc(COC)c2)=O)CC1CC 88375,c1(NC(C2CCN(C(c3n(CC)nc(C)c3)=O)C2)=O)cc(Br)c(O)cc1F 88376,Cn1cnc2cc(C(N3CCCC(NC(=O)C4=CCCOC4)C3)=O)ccc12 88377,c1(C(C)NC(=O)C(c2ccccc2)Oc2cnn(C)c2)ccnc(F)c1 88378,C1(COC)(NC(c2cc(C(N)=O)co2)=O)CCN(C(c2cc(=O)cc[nH]2)=O)CC1 88379,c1(NC(C(C2CC(F)(F)C2)OC)=O)cccc(-c2nc(O)n[nH]2)c1 88380,N1(C(c2cnc(SC)s2)=O)CCN(C(C23CCCC2C3)=O)CC(C)(C)C1 88381,c1(OC)cc(C(=O)NCC2CCN2C(c2cccc3occc23)=O)cc(N)c1N 88382,C12(C(=O)NC3CCC(NC(C4C=CCC4)=O)CC3)C3CC(CC13)C2(F)F 88383,CC1CN(C(=O)CNC(c2ccccc2)=O)CC1NC(C1(F)CC=CCC1)=O 88384,N1(C(C(c2ncc(Br)cn2)N(C)C)=O)CC(S(C)(=O)=O)CC1(C)C 88385,N1(C(=O)Cn2ccnc2)CC2CN(Cc3ccc(C4(C)CC4)cc3)C2C1 88386,Cc1cc(F)ccc1C(=O)NCCC1CCCN1Cc1ccncc1 88387,C(CC(F)F)(C(=O)N(C1CCCC1C#N)CC)N(C(CCCOCCC)=O)C 88388,c1(C(N2CCOC(CNC(C34CCCN3CCC4)=O)C2)=O)ccc2nccn2n1 88389,CC1COCCN(C(=O)CCN(C(=O)COC2(C)CCC2)C2CC2)C1 88390,N1(C(CCC(=C)C)=O)CCC2(CCOC2)C(CNC(c2csc(COC)c2)=O)C1 88391,N1(C(C(CCOC)NC(=O)CCCCNC(C)=O)=O)CCNC(=O)C1C 88392,c1(C(=O)NC2CC(CNC(C(C)C3CCC3)=O)C2)n[nH]c2ccc(Cl)cc12 88393,c1(C(=O)NCCCC(C)NC(=O)CC2CC23CC3)nn(C)nc1Br 88394,C(C(=O)NCc1cccs1)(C(C)CC(C)C)N1CCC(C(=O)NC)C1 88395,CC1(C)CCOC1CS(=O)(=O)NC(c1cnc(CN2CC(N)C2)o1)=O 88396,Cc1cccc2c1CCOC2C(=O)NC1COC2CN(C(=O)C3=CCOC3)CC12 88397,C(=O)(CC(C)(C)C(=O)OC)NCC1C(NC(CCC=C)=O)CC1 88398,C=Cn1ncc(C(N2CCC(C=CC(=O)NCCC(C)C(C)C)CC2)=O)c1N 88399,C1(CNC(CCCC(C)=O)=O)CN(C(=O)C(C)(C)C2CCCCO2)CCC1(F)F 88400,c1(OC)coc(C(=O)NC2CC(CNC(=O)Cn3cc(C#N)cn3)C2)cc1=O 88401,C(CC(C)(C)C)(C(=O)N1CCC(C)(C(=O)N(C)CC2(C)CCC2)C1)OC 88402,C#Cc1cccc(C(N2CC(CN(C)C(c3cnn4ccn(C)c34)=O)C2)=O)c1F 88403,c1(C(N(CC(CN(C(=O)CCC2CCCO2)C)O)C)=O)nccc2cccnc12 88404,CCCCCC(F)C(=O)N1CC(NC(=O)CCCCCn2cnnn2)C(C)(C)C1 88405,C1(N(C(c2cn(CC)nn2)=O)C)CCCN(C(c2cc(C)c(CC)o2)=O)C1 88406,N1(C(CC)CC)CC(C(=O)N(C2CCC(CNC(=O)C(F)CC)CC2)C)CC1=O 88407,c1(OC(C)C)cc(C(=O)NC2CN(C(C3(c4ccccc4)COC3)=O)C2)ccn1 88408,C(=O)(CC(C)(F)F)N1C(C2(NC(COC3(C)CCC3)=O)CC2)CCC1 88409,C1(NC(C(CC)NC(C)=O)=O)CCC2CC1CN2C(=O)C(C)OCCC(C)C 88410,N1(C(C(CC)(F)F)=O)CCc2ccccc2C(NC(=O)CC(O)C2CCCC2)C1 88411,C1(C)(C(N(CC(C)NC(Cc2c(C)non2)=O)C)=O)CC(F)(F)C1 88412,c1(C(C)=O)[nH]c2ccccc2c1C(=O)NCC1CC1(Cl)Cl.C12CCCC1NC2=O 88413,Cc1ncnc(C(=O)NCC(CC2CC2)C(=O)NC2(c3nn[nH]n3)CC2)c1C 88414,C12(NC(C(C)C3CCCC3)=O)CCC(CNC(=O)CN3C(=O)CCC3=O)(C1)OC2 88415,C(=O)(C(O)CC(C)(C)C)NC1C(CC)CN(C(=O)C2=CCCO2)CC1 88416,C1(NC(c2coc3c(-c4cn[nH]c4)cccc23)=O)CCc2ccc(O)cc2C1 88417,N1(C(C)=O)CCCc2cc(NC3(c4nnnn4C)CC(C(C)C)C3)ccc21 88418,CC(C(=O)NCC1C2CN(C(=O)CCN3CCCCCC3)CC12)S(C)(=O)=O 88419,C1(C)(c2cn(CCc3ncn(C)n3)nn2)COCCN1C(=O)Cc1nc(=N)[nH][nH]1 88420,C(=O)(C1CCCc2ncnn21)N1CC(N(C)C(c2csc(S)n2)=O)C1 88421,C(CC(C(C)(C)C)C1CC1)N(CC(C)(C)NC(=O)C1CC1)C.C1(=O)C=CC(=O)N1 88422,N1(C(C(C)(C)C2CC2)=O)CC(CO)C2(CCN(C(C3C4CCCC34)=O)CC2)C1 88423,c1(C(=O)NCCCN(C(=O)CCc2ccnc(Cl)c2)C)cnn2ccn(C)c12 88424,C(=O)(C(C)(C)C(C)C)OCCCC(=O)NC1CCC1CNCC=C 88425,c1(Cc2nc(C3ON=C(CC)C3)on2)ccc2c(c1)CCCO2 88426,c1(OC)ccc2c(c1)CC(C(=O)NCC(C)(C)NC(=O)C1=CCOC1)O2 88427,c1(C(N2CC(C)(NC(C3(CC(C)C)CC3)=O)C2)=O)ccc(-c2cn[nH]c2)cn1 88428,C(=O)(CCC(=O)NC1CC(C)(NC(=O)CCC(=O)Nc2nnc(C)s2)C1)OC 88429,Cc1cc(C(N2CCCC2(C(=O)N(C(CO)C2CC2)C)C(C)C)=O)nc(O)c1 88430,c1(CNCC(=O)N(CC(=O)N(C)CC2(CO)COC2)C)ccccc1 88431,N1(C(C(C)n2ccnc2)=O)CCC(O)C(NC(c2cc(=O)cc(Cl)[nH]2)=O)C1 88432,CCCCC(CC(=O)N1CCC(C)CC1C)NC(C1CC2CC(=O)C1C2)=O 88433,S(=O)(=O)(c1ccc(NC2CCC(CO)C2)cc1Cl)NCCc1nc(C)sc1 88434,N1(C(C(CC)OC)=O)CCCC(CNC(=O)CCn2ccnc2C)C1 88435,N1(C(CCCOCCC)=O)CC(C(=O)NC(CF)C(F)(F)F)C(C)C1 88436,C1(NC(=O)CCCc2cccs2)CCN(C(=O)Nc2ccc(O)c(O)c2)CC1O 88437,CC1=C(C(=O)NCC2CN(C(C3CC(NS(C)(=O)=O)C3)=O)CCC2C)SCCO1 88438,C1(C(N(C)Cc2ccc(Cl)s2)=O)C=CCN(C(C2CCCCO2)=O)C1 88439,C1(NC(COCCOC)=O)CC12CCN(C(=O)Cc1cnc(C)s1)C2 88440,C1(NC(C2N(C)CCC2)=O)CCC2(CC1)CCN(Cc1c(F)cc(F)cc1F)C2 88441,C1(NC(CC(C)(C)C2CC2)=O)CCCN(C(c2ccc(Br)c(O)n2)=O)CC1 88442,Cc1cnccc1C(N1CCC(N(C(=O)CCSc2nccn2C)CCO)C1)=O 88443,c1(C(c2n(CC)nnn2)NCCN2CCOC2=O)cc2nccc(Cl)c2s1 88444,C1(NC(c2cncnc2)=O)C(CC2CC2)CCN1C(=O)CCC1CC1 88445,C(=O)(CCC(F)(F)C(=O)N1CCN(C(C2C=C2C)=O)CC1COC)OCC 88446,Cc1cccc2c1CCN2C(C1(F)CCN(C(C2COC(=O)N2)=O)CC1)=O 88447,c1(CC)cccc(C(N2CCCC(CNC(=O)CSC3CCOC3=O)C2)=O)c1F 88448,C1(NC(CCCCCNC(C2(SC)CCOCC2)=O)=O)Cc2ccncc2N1 88449,C(C(CC(C)C)NC(c1cc(-c2ccc(C)cc2)no1)=O)NC(C(COC)OC)=O 88450,C1(CC)CCCC1(C)C(N1CCC(CC(=O)NC(c2n[nH]c(C)n2)(C)C)C1)=O 88451,N1(Cc2cnc(CCC)s2)C(C(N2CCOC3(CC3)C2)=O)CC2CCCCC12 88452,c1(-c2cn(C(C(=O)NC(C(CCCOC)C)=O)(C)C)nn2)cccc(C#N)c1C 88453,C(C)(C(=O)NC1CC(CNC(C2CCC2c2nc[nH]n2)=O)C1)OCCCC 88454,C(CC1CCCCC1)(C(=O)NCCCCCN(C(=O)C=Cc1cscn1)C)OC 88455,N1(C(C(CCOC)(C)C)=O)CCC2CC(NC(C3(O)CCSC3)=O)CCC2C1 88456,Cc1cn2c(n1)CC(C(=O)NCC13CC1CN(C(c1cnn(CCF)c1)=O)C3)C2 88457,C1(N(C(=O)CC2(C(=O)NC)CC2)CC)CCN(C(C2(C)CCOC2)=O)C1 88458,N1(C(C(P(C)(C)=O)O)=O)CC(NC(=O)C(F)(F)C(F)F)CC12CCCC2 88459,CCC(C(=O)Nc1cn(C)nn1)NC(=O)CC1CCN1C(=O)C1CC1 88460,c1(C(N(CCOCCN(C(c2cn(CC=C)nn2)=O)C)C)=O)cc[n+]([O-])cc1 88461,c1(OC)ccc(Br)c(F)c1S(=O)(=O)N1CCC(c2ccc(Br)s2)C1 88462,C(CC(CC1CC1)N=c1ncc2ccccc2[nH]1)NC(Cc1n(C)ncc1Cl)=O 88463,C(CC(=O)N1CCCC1C(C)(C)C#N)(C(N)=O)C(=O)OC(C1CCOCC1)C 88464,C1(CNC(COC)=O)CN(C(=O)COc2cccc(C#N)c2)C2(CCC2)C1 88465,C1(CC)(NC(c2cc(CNC(C3CC(C)(C)C3)=O)on2)=O)CCCC1 88466,c1(C(=O)NC(CNC(CC(C)OC)=O)(C)Cn2cccn2)cccc(N)n1 88467,c1(SC)c(C(=O)NC(C(=O)NOCC(C)(C)O)C2CC=CCC2)cnn1C 88468,C(=O)(C(CC=C)CC(C)C)NC1(CC=C)CCN(C(c2cccnn2)=O)CC1 88469,NS(=O)(=O)c1ccc(C(=O)NC2CN(C(=O)C(O)C(F)F)C2)cc1F 88470,CCC(C)(CNC(C1COCCO1)=O)C(=O)NC(C)Cc1cccnc1 88471,c1(OC)ccc(NC(=O)CCC2CCN(C(C3CC3F)=O)CC2)cc1C 88472,N1(C(C(COC)C)=O)CCN(C(c2nc(Cl)c(Cl)s2)=O)CC(C)(F)C1 88473,Cc1cc(C(N2CC(CCNC(C3CC(O)C3)=O)OC(C)C2)=O)nc(O)c1 88474,C(CCCCCN(C)C(=O)OC(C)(C)C)NC(C(=O)NC(CC)C)=O 88475,Cc1cc(C(=O)NCCC2(O)CCCN(C(C3CSCC(=O)N3)=O)C2)ncc1N 88476,C1(CNC(c2c(Cl)cn(CCC)n2)=O)CN(C(C2C(C#N)C2(C)C)=O)CC12CC2 88477,c1(C(N(CC)CC2CCCN2C(C2CC(SC)C2)=O)=O)ccc(N(C)C)cn1 88478,C(=O)(CCCC(C)(C)NC(C1CCN1C(C)(C)C)=O)N1CC(OCC#C)C1 88479,N1(CCN(C(c2cc(CC)no2)=O)C)CCN(C(c2cn(CC)nn2)=O)CC1 88480,N1(C(CNC2CC(C(C)C)C2)=O)CC2(CC2)C1 88481,C1(C(c2n(CCCC)nnn2)NCC2CCN2CC)CC12CCOCC2 88482,c1(OC)cc(F)c(CC(=O)N(CC(C)NC(c2csc3nccn23)=O)C)c(Cl)c1 88483,c1(C(N2CC3CCC(C2)N3C(=O)CC2CC3CC3C2)=O)ccn2cccc2c1 88484,N1(C(CN2CCC(O)(C(C)CNC(C(C)CO)=O)C2)=O)C(C)CCCC1C 88485,C1(C(=O)NCc2cncc(CC)c2)CC12CCN(C(=O)CC1(O)CCC1)C2 88486,C1(CNC(CN(C)C(N)=O)=O)CN(C(=O)CC2C=CCCC2)CCC1(F)F 88487,Cc1cc(NC(C2C3CN(C(=O)CC4CSCCO4)CC23)=O)cc(C)c1 88488,N1(C(CC2C(=C)C2)=O)CCC2(CC1)CN(C(=O)CCOCC)C2C(C)C 88489,C1(CNC(c2ncccc2F)=O)CCN(C(C2C3CCC(=O)C23)=O)CC1 88490,c1(N(C(C)C)C)cc(N(C)C)nc2c1CCCC2.C1(=O)CO1 88491,C1(COC)(NC(C2CCC(=C3CCC3)CC2)=O)CCN(C(C2CNC(=O)N2)=O)C1 88492,C(=O)(CCC(F)(F)CN=[N+]=[N-])N(CCC)CCNC(C1CCc2nnnn2C1)=O 88493,n1(CCCSCC)nnnc1C(C(C)(C)C)NCC(C)C1CCC1 88494,c1(C(=O)NC2CCN(C(C34CC(CCO3)C4)=O)CC2F)cc2cc(F)ccc2o1 88495,C1(C)(OCC(=O)OC)CN(C(=O)CCCF)C1.C1=CC(=O)NC1(C)C 88496,C(=O)(CC(C)CC(=O)NC(C)C(C)C(=O)N(C)Cc1cnco1)OC 88497,c1(C(N(C(C)CCNC(=O)CCc2cncc(O)c2)C)=O)cccn2nncc12 88498,C1(OCC)CCCC1N=c1[nH]c(=NC2CCC(C)(C)CC2)[nH]c2c1COCC2 88499,n1(CCNC(=O)NCC(C)CN(C)C(=O)OC(C)(C)C)cccc1C=O 88500,c1(C(N2CCC(N(C(C3(C4CC4)CC3)=O)CC)C2)=O)cccn2c(C)cnc12 88501,N1(C(CC(C(CC)C)O)=O)CC2(CCN(C(=O)CC3CC(F)C3)CC2)C1 88502,Cc1cc(CNC(=O)NC2CCC(C(=O)O)CC2)c(F)cc1Br 88503,c1(C(C(=O)NCC2CCOC2)N(CCSC)CC)ccc(OC)c(C)n1 88504,CN1CC2(CC2)CC1C(=O)NOCC(N1CCC1C1CCC1)=O 88505,S(=O)(=O)(C1CCS(=O)(=O)C1)NCC1(N(C)C(=O)OC(C)(C)C)CC1 88506,C(CCC(=O)N(CC(O)CN(C(=O)C(C)n1ccnn1)C)C)N(C(C)C)C 88507,N1(C(C=Cc2nc(C)sc2)=O)CCN(C(=O)Cc2csc3nccn23)CC(C)(F)C1 88508,C1(C(=O)NC(c2nc(C)[nH]n2)C)CC(O)CCN1C(c1ccncc1Cl)=O 88509,N1(C(c2[nH]cc(C)n2)=O)CCCC(CCn2cc(CCCC(C)O)nn2)CC1 88510,c1(C(C)C)ccc(CCC(=O)OCc2nc(C(C)(C)C)n[nH]2)cc1 88511,N12CC(CC1(C)C)CC2=O.C(=O)(C(F)C(C)(F)F)NC1CC(OCC)C1 88512,Cc1[nH]nc(C(=O)N(C(C)C(=O)N2CCC2CC2CC2)C)c1O 88513,C1(NC(C(C(C)C)c2cnn(C)c2)=O)CN(C(c2ns[nH]c2=O)=O)CC12CC2 88514,C(=O)(CCCC(C)(C)C)NC1CN(C(Cc2ccc(C(=O)NC)cc2)=O)CC1C 88515,C(=O)(C1=CCCCC1)NC1(CNC(=O)C(c2ccc(C)s2)C)CC(OC)C1 88516,C(CC(C(=O)N1OC2CCC1C2)OC)NC(c1c(CC)cno1)=O 88517,C1(CNC(c2cccc(CC)c2)=O)CC2(CO1)CN(C(=O)C(C1CCC1)OC)C2 88518,c1(N(C)CC2COC(=O)O2)nc(N2CC3CC2C3)c2cnn(C)c2n1 88519,C1(NC(c2c(C)nn[nH]2)=O)CN(C(c2ccc(-c3ccc(Cl)cc3)[nH]2)=O)CC1C 88520,CC(C)C(C)(CNC(C1CC1C(C)(C)C)=O)NC(=O)C(O)CC1CCC1 88521,Cc1[nH]c(=N)ccc1C=CC(=O)NCCC(C)NC(C1CCCC12CC2)=O 88522,C1(CNC(C2CCC2(F)F)=O)CC2(CCN(C(c3cccc[n+]3[O-])=O)CC2)CO1 88523,C(=O)(C1=CCOC1)NC(C)CCCNC(c1cn(C2COC2)nn1)=O 88524,C12(NC(c3cnc(C(C)=O)s3)=O)CCN(C(=O)CCn3cnccc3=O)CC1C2 88525,C#CCCCC(C)C(=O)N1CCC(C(C)(C)NC(c2ccc(O)nc2)=O)C1 88526,Cn1nc(Cn2cc(CN3CCCC(F)CC3)nn2)c2c1CCC2 88527,c1(OC)ccccc1OCCC(=O)NCC1CC(NC(C2COCC(C)O2)=O)C1 88528,c1(NC(C2(F)CN(c3nc(C)cc(OCCOC)n3)C2)=O)nc(C)c(Br)c(Cl)n1 88529,N1(C(C2C(C)C2)=O)CCCC(N(C(=O)CCC2CCCOC2)CCF)C1 88530,c1(C(C)CN2CCNC(=O)CC23CC3)ccc([N+](=O)[O-])cc1-c1nn[nH]n1 88531,C1(C(N(C)CCC2CCCCN2C(c2cncc(Cl)c2)=O)=O)CCC(C)(C)CC1 88532,n1(CC(=O)NC)cccc(NC(C2CCC(O)(CC(C)C)CC2)=O)c1=O 88533,c1(CC(=O)NCC2N(C(C(N3CCC(O)CC3)C)=O)CC2)cccc(F)c1F 88534,CCCC(C)(CCC)C(=O)NCC12CCC1CCN2C(c1cc(C2CC2)on1)=O 88535,C(c1ccsc1Br)=CC(=O)NC1CCC(CNC(c2ccon2)=O)C1 88536,N1(C(Cc2c(C(C)C)con2)=O)CCN(C(C)CNC(C2(C)CC(C)C2)=O)CC1 88537,N1(C(C(C(C)C)n2ccc(C3CC3)n2)=O)CCN(C(=O)C(N)=O)C2(CCC2)C1 88538,C(C(C)(O)CC(=O)NC1CCCN(C(c2cc(C#N)cs2)=O)C1)OC 88539,c1(NC(Cn2c(C)cc(C)n2)=O)ccc(NC(c2cnc(C(N)=O)cn2)=O)c(F)c1 88540,C=C(C)CN=C1NCC(C)(C)N2CCN(CC2)CCC2(CC)C(C(CO)CN1)C2.OC 88541,N1(C(C2CC(C)(C(=O)OC)C2)=O)CCN(C(=O)CC=C(Cl)Cl)C(C)C1C 88542,C(=O)(CC(CC)CC(F)(F)F)N1C(CN(C(CC(=O)NCC)=O)C)COCC1 88543,N1(C(CNC(c2n(C(C)C)ccc2)=O)=O)CCN(C(=O)CN(C)C(N)=O)CC1 88544,C12(C(N(C)CC3CCCN(C(=O)C=CC4CCC4)C3)=O)CCCN1S(=O)(=O)CC2 88545,C12(C(N3CC(NC(CSC(C)C)=O)C(CC4CC4)C3)=O)CCCCCC1OCC2 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88616,N1(C(=O)CCOC2CCC2)CC2CC1CN2C(C12CCC1CC2)=O 88617,c1(CN(C(N(CCC(=O)NCCCOC)C)=O)C)cncn1C 88618,c1(C(C)C)ccc(C(=O)NC2CCN(C(=O)CN(C(=O)OC(C)(C)C)C(C)C)C2)o1 88619,C1(CC=C)(C(=O)N(C)C(C2CCCO2)C)CN(C(=O)CCOC2COC2)C1 88620,N1(C(c2cccc(N(C)C)c2)C(=O)NCCC)CCC2(CC1)OCC(C)(C)CO2 88621,c1(C(N2CCN(c3c(C)cc(Br)cc3)CCC2=O)=O)cc(=O)c2ccccc2o1 88622,CCCC(C)C(=O)NC(C)CCCNC(c1cnn(CCN(C)C)c1C)=O 88623,CC(C(C)C(=O)NCCc1cnco1)NC(=O)C=Cc1cnccn1 88624,c1(C(C2CC2)NC(CONC(CC2ON=C(C)C2)=O)=O)ccc(F)cc1 88625,c1(C(=O)NCC(CNC(CCNC(C(C)(C)C)=O)=O)CO)ccnc(O)c1F 88626,CC(CF)CC(=O)NCC1CCN(C(c2cn(-c3cccc(Cl)c3)nn2)=O)C1 88627,C(C#Cc1cnn(C)c1)NC(C1CC(NC(C(c2ccnn2C)C)=O)C(O)C1)=O 88628,Cc1cc(C#N)cnc1C(N1CCOCC(NC(=O)C2=COCCO2)C1)=O 88629,C1(F)(C(N(C2CC(C)OCC2)C)=O)CCCN(C(C2COC(=O)NC2)=O)C1 88630,c1(C(=O)NCC(C)NC(C(C)SCCCC)=O)ccc([N+](=O)[O-])cc1 88631,Cc1cn(C)cc1C(N1CCCC(CC(=O)N(C)Cc2cccnc2)C1)=O 88632,C1(NC(CC(C=C)c2ccccc2)=O)(CO)CCCN(C(=O)C(C)C(O)CC)C1 88633,Cc1nn(CCc2ccccc2)c(C)c1CNC1CN(C(=O)C(C)O)CC1C 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88652,C(=O)(C1=NOC2(CCC2)C1)NC(C)CC(O)c1ccco1 88653,C1(C(=O)NCC2(C)CCN(C(CCc3cncc(C)c3)=O)C2)CN2CCC1CC2 88654,c1(C(N2CCC(OCCNC(c3cnc(CC)[nH]3)=O)C2)=O)nnccc1C 88655,C1(C(=O)NC2CN(C(C=C(C)C)=O)C(C)(C)C2)CN2CCN1CC2C 88656,C1(N(C(=O)CCC2CCC(=O)NC2)C)CN(C(C2CC(=O)C2)=O)CC12CC2 88657,C1(S(=O)(=O)N2CCCC2COC)(CC=C)CC1.N1(C=O)CC=CC1(C(=O)OCC)CO 88658,N1(C(C2(C)CNC(=O)C2)=O)CCOCC(NC(c2cc3sccc3s2)=O)C1 88659,CC(C)CC(O)C(C)C(=O)N1CCC(F)(C(=O)NCC(C)(C)C#N)CC1 88660,C1(NC(c2n(CC)ncc2Br)=O)CCN(C(=O)Cn2ncnn2)C(C)C1 88661,CC(C)CCC(O)C(=O)NCC1(C)CCCN1C(c1ccn(CC(C)C)n1)=O 88662,c1(CC)nc(C)c(C(=O)NCc2cccc(CN(C)C(C3(O)CCOC3)=O)c2)o1 88663,c1(C(N2CC(CNC(C(CCC)C)=O)C(C)C2)=O)cc(C)cc(Br)c1 88664,C12(C(=O)NCC3(CCNC(C(N4CCCC(O)C4)C)=O)CC3)CCOC(C)(C1)C2 88665,C(=O)(C(CC1CCCCC1)N1CCC1c1ccccc1)NCCC(=O)OCC 88666,c1(OC)ccc(OCCC(=O)NCC(CO)NC(=O)C(C#N)C2CC2)cc1 88667,C1(CNC(c2c(CCC)occ2)=O)CCC(C)(CNC(c2c(C)n[nH]c2C)=O)C1 88668,c1(C(N2C3CN(C(CSc4ccc(C)cc4)=O)C(C3)C2)=O)cnc2occc2c1 88669,CCC(O)C(C)C(=O)NC(C)CCN(C(=O)CNC(c1ccccn1)=O)C 88670,CC(C(=O)N1NC2CCC1C2)C(F)(F)c1ccccc1 88671,N1(C(C(C(CC)CC)C)=O)CCN(C(c2ccc(CO)o2)=O)CC2(CC2)C1 88672,C(=O)(C1(C)CCc2ccccc21)NCC1(F)CCN(C(CCC=C)=O)CC1 88673,c1(OC)ccc(F)c(C(=O)NC(C)CNC(=O)C=CC2CCOC2)c1 88674,N1(C(C2CCCC(C)C2)C(=O)Nc2c(C)cccc2C)CCS(=O)CCC1C 88675,CC(C)(C(=O)NCC1CCC1NC(C1(CC2CCC2)CCCO1)=O)c1cc[nH]n1 88676,CC1CC(CO)(NC(C2(F)CN(C(C3CCSC3C)=O)C2)=O)C1 88677,Cc1cnn(C)c1N(C(=O)CNC(=O)C(CN(C)C)N(C)C)Cc1ccco1 88678,C1(C(N2CCC(N(C(=O)CC3CC(C)(C)C3)CCC)C2)=O)CC2CCC1CC2 88679,C1(CC(=O)NCc2occ(C(N(C3CSC3)CC#C)=O)n2)CC(O)C1(C)C 88680,C=CC1CN(C(c2ccccc2CC(C)(C)C)=O)CC1NC(=O)C(O)C(F)F 88681,C#Cc1cnc(C(=O)NC2CC(CCNC(=O)C=C(C3CC3)C3CC3)C2)c(C)c1 88682,Cc1c(C(=O)NC2(c3ccccc3Br)CC2(F)F)cc(Br)cc1I 88683,c1(C(=O)NC2CCN(C(CCCCOC)=O)C2C)n[nH]c2ccc(OC)nc12 88684,Cc1ccc(C)c(C(=O)NC2(C)CCN(Cc3ccc(C#N)cc3)C2)c1 88685,CC1CC(C)(C(N2CC(N(C(=O)CC3CCCC3(F)F)C)C2)=O)CC(C)O1 88686,c1(C(=O)NC(CC(C)C)CNC(C2CNC(=O)N2)=O)cc(O)ncc1Br 88687,CC(C)C(O)C(C)C(=O)N1CC2C(C(N3CCN(CC(C)O)CC3)=O)C2C1 88688,C1(C(=O)NCCOCCNC(CN2CCC(C)(C)C2)=O)CC12CCCOC2 88689,C1(NC(=O)CCOC2CCC2)CCC2(CC1)CC2NC(c1cc(CCO)on1)=O 88690,NC(=O)CC(C(=O)NCC1C=CCCC1)NC(C1CC(C2CC2)C1)=O 88691,CC1=C(C(=O)NCCC(C)NC(=O)CCC2=CCCCC2)S(=O)(=O)CCO1 88692,C1(CNC(COCCC)=O)CC2CCC1N(C(=O)C(F)CC1CCCC1)C2 88693,CCC(C)C(O)CC(=O)NC(C1CC1C(=O)NCC12CCC(CC1)OC2)C 88694,c1(C(N(CCCN(C(C2C(CC)CCCC2)=O)C)C)=O)cc(C)cc(C#N)c1 88695,CCCCCCCCC(C)CC(=O)NC1C2CCN(C(=O)CS(=O)(=O)CC)C12 88696,C1(C(N2CC(NC(C(F)OC)=O)C(C(F)(F)F)CC2)=O)C(C)(C)CCCC1(C)C 88697,C1(CNC(CC(CC)(C)C)=O)CCCC2CN(C(=O)CC3CC4CCC3C4)CC12 88698,n1(CC(=O)NC(CCC)CNC(c2ccnc(CC)c2)=O)cc([N+](=O)[O-])cn1 88699,N1(C(Cc2nc(C)[nH]n2)=O)CCC(NC(c2nc(C)nn2C)=O)C12CCC2 88700,C1(C(N2C(CNC(C3CC(C)(F)C3)=O)CC2)=O)CCN(c2ccncn2)CC1 88701,c1(C(N2CCC(N(C(=O)CCc3ccnc(Cl)c3)CC)C2)=O)cc(C)cnc1N 88702,C(=O)(C1CCCc2nnn(C)c21)NCCCOC.N12CCN(CC1)c1cccc(c1)C2=O 88703,c1(CC(=O)NC2C(NC(CC(C=C)C)=O)COC2)ccc(Cl)c(Cl)c1 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88846,c1(C(=O)NCCCOCC(C)(C)NC(C2C=CCCC2)=O)cnn2c1CCC2 88847,O=C(CC1=CCCC1)NCC1(O)CC(NC(c2cn(-c3ccccc3)cn2)=O)C1 88848,C12(NC(CSC)=O)CCCC1N(C(=O)COc1ccc([N+](=O)[O-])cc1)CCC2 88849,Cc1ncccc1CCC(N1CCCC(NC(c2ccncc2Cl)=O)C1)=O 88850,C(=O)(NNc1ccc(Br)c(F)c1F)c1c(OC)nc(F)c(Br)c1 88851,c1(OC)cnncc1C(=O)NCC(O)C(=O)NCc1cccc(OC)n1 88852,c1(CNC(c2n(C(C(=O)OC)C)nnn2)CC(C)C)cc(F)ccc1Cl 88853,C1(OC(C(C)OCc2ccc(C)o2)=O)CCOC2(CCOCC2)C1 88854,C(=O)(N1CCC(C(=O)NCCCn2cnnn2)O1)c1cc(OCC)no1 88855,C1(C2CCN(C(=O)Cc3ccco3)C2)(CCC(C)C(=O)NS(C)(=O)=O)CC1.CC.CN 88856,c1(C(=O)NC2CC(C)(CNC(C(CC)(C)CO)=O)C2)cc(F)cc2nn[nH]c12 88857,C1(C(N2CCC(CCCC)C2)=O)CCN(C(=O)CCCCC(C)=O)CC1(C)C 88858,Cc1cc(O)c(C(N2CCC(NC(c3ccc(CF)cc3)=O)C(O)C2)=O)nn1 88859,N(C1CCOc2ncccc21)CC(O)CC1(O)CCCC1 88860,C1(CC)(NC(=O)CC(C)C(C)C)CCCN(C(c2csc(Br)c2C)=O)C1 88861,Cc1cc(C(=O)NCC(C)NC(=O)CC(C)(C)CN(C)C)cc(O)n1 88862,c1(NC(C2C(NC(C(CC)OCC)=O)CCC2)=O)ccc(-c2cscn2)cc1 88863,CC1CC(c2ccsc2)CN1Cc1sc(Cl)cc1Br 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89020,CC(C)(CCF)C(=O)NC1CC(O)(CNC(C2CC(CC3CC3)C2)=O)C1 89021,c1(C(N2C(CCNC(=O)Cc3cccnc3)COCC2)=O)ccn2ccnc2n1 89022,N1(C(C(c2ccc(C)o2)C)=O)CC(N(C)C(c2nc(C3CC3)oc2C)=O)C(O)C1 89023,O=C1OC2CC1N(C(=O)CCC1CCCCO1)C2 89024,c1(C2C(C)C2)nc(SCCOCC(C)(C)NC(=O)OC(C)(C)C)n[nH]1 89025,C1(N(C)C(c2cnn(Cn3cc(CC4CCCCN4C)nn3)c2)=O)CCC2CCCC12 89026,C(CC1=CCN(C(C2CCc3ccnn3C2)=O)CC1)NC(C(C)(O)C1CC1)=O 89027,C(=O)(CCC(=O)NN(C)C)NCC(CC(=O)NC(COCC)(C)C)C 89028,c1(C(N2CCCC(CF)C2)C(=O)NCCSC)ccc(F)c(C2CC2)c1 89029,c1(C(=O)NC2CC(NC(C3C4CC5C(C4=O)C35)=O)C2)ccc2c(n1)CCO2 89030,Cc1c(C(=O)NC(CN(CCO)C2CC2)C2CCC2)cccc1Cl 89031,c1(C(N(CC(CC)NC(c2cccnc2S(C)=O)=O)C)=O)cc(C)n(C)c(=O)c1 89032,N1(C(CC=C(C)C)=O)CCOC(CNC(=O)CC23COCC(C2)C3)C1 89033,Cc1cc(C)c(C(N2CC(N3CCN(C(C4CC(F)C4)=O)CC3)C2)=O)[nH]1 89034,N1(C(CSc2nc(C)[nH]n2)=O)C(CNC(c2coc(C3CC3)n2)=O)CC2COCC12 89035,C(=O)(CC(C)C(F)(F)F)N(CC(CNC(C(F)=C(C)C)=O)(C)C)C 89036,C1(O)(C(=O)NC2CC(C(N3C(C)(C(=O)OCC)CCC3)=O)C2)CCOC1(C)C 89037,Cn1c(C(N2CC(CNC(C3CC(C)(C)CO3)=O)C2)=O)cc2sccc12 89038,C(=O)(C(CCNC(C1C2CCCOC12)=O)OC)NCCC1(COC)CCC1 89039,c1(OC)nc(C)ccc1C(N1CC(NC(=O)CC2CC(SC)C2)C(F)C1)=O 89040,N1(C(c2c(C)nn(C(C)C)c2)=O)CC(NC(=O)CC=C(Cl)Cl)CCC1C 89041,C(c1c[nH]c2ccccc12)=CC(N1C(C(N2C(C)C(O)CCC2)=O)CC(O)C1)=O 89042,C1(CC(=O)N(CC#C)CCF)CCN(C(=O)C(C)C2CCC2)C1(C)C 89043,c1(C(C)C(=O)NC2(CC(=O)NCC(=O)OCCO)CC2)cnn(C)c1 89044,C(=O)(C(C)(CCF)NC1(c2ccn(-c3c(F)cccc3F)n2)CCC1)OC 89045,C1(NC(Cc2c(C(C)C)cccc2)=O)CC2(C1)CN(C(=O)Cn1cnnc1O)C2 89046,N1(C(c2c(C)ncn2C)=O)CCC2(CCCN2C(c2cncc(Cl)n2)=O)C1 89047,CC1CN(C(=O)COCC2CC2)CC(C)C1NC(=O)CCCN(C)N=O 89048,C1(NC(=O)C=CCF)CC2CCCC(C1)C2.C12(CCCCC1)C(=O)NC2 89049,c1(C(=O)NC(CC)CN(C(c2sccc2C)=O)CC)ccc(F)c(C)c1C#N 89050,c1(NC(CCC)C)ncnc(NCCc2ncccc2C)c1C 89051,Cc1ncc(C(=O)NCC2CCCCN(C(c3cncs3)=O)C2)cc1N 89052,c1(C(=O)NC(CC)CN(C)C(C2CCCO2)=O)c[nH]c2c(Cl)cccc12 89053,N1(C(C2ON=C(C(=O)OC)C2)=O)CCOCC(C)(CNC(=O)Cc2cnc[nH]2)C1 89054,S(=O)(=O)(c1cccc(C)c1)N1CCCC(C(N2CC(OCC)C(O)C2)=O)CC1 89055,C1(C(=O)NCC(CO)NC(C2(C=C)CCCCC2)=O)CNC(=O)CC12CCC2 89056,C1(NC(c2cnc(COC)s2)=O)CC2CC1CN2C(c1cn(C)c(C)n1)=O 89057,Cc1csc2ncc(C(=O)N(C)CC3CC(F)CN3C(=O)CC3(C)CC3)n12 89058,C=Cc1cnn(C)c1C(=O)NCC1CN(C(=O)C(F)(F)CC)CC1C(F)(F)F 89059,Cc1cc2c(C(N3CCSCC3CCNC(C34CC(C)C3C4)=O)=O)cccc2o1 89060,c1(C(=O)NCC(C)(O)C2CCC2)[nH]ccc1CNC(C1CC=CCC1)=O 89061,Cc1nc(C)n(CCC(=O)NCC2(C(C)(C)O)CN(C(=O)CC(F)(F)F)C2)n1 89062,N1(C(C)=O)CC2CC1CN2C(C1C=CCN(C(=O)C(C)(C)CCF)C1)=O 89063,n1(CC)nnc2c(N3CCC(CN(C(=O)C(C)CC(N)=O)CC)CC3)ncnc12 89064,N1(C(C(COCC)(C)C)=O)CC2(CNC(=O)CC(C)(O)C3CC3)CC1(COC)C2 89065,C1(C(=O)NCC2(F)CC(NC(C3(CF)COC3)=O)C2)CCCCCC1 89066,c1(NC(C2(OC)CCN(C(C(CCCOC)C)=O)C2)=O)cn(C)c(=O)nc1O 89067,C1(C2N(C(=O)CCCOC(C)C)CCC2)CCN(C(c2c[nH]c(=S)cn2)=O)CC1 89068,N1(C(c2ccncc2O)=O)CCCC2C1CCN2Cc1ccc(F)c(F)c1Cl 89069,C(CCCC(=O)NC1(CN(C)C(C2(OC)CC2)=O)CC1)OCC 89070,C1(Nc2cccc(-c3c(C)ncn3C)c2)CCC2COCCC2(C#N)C1 89071,CC1(C)CC(C(=O)NCCNC(=O)CCc2ccc(Cl)cc2)C(C)(C)O1 89072,CC(C)C(CNC(=O)CP(C)(C)=O)C(=O)NC(C)(CO)C(C)(C)O 89073,c1(CC)nn(C)c(Cl)c1C(N1CCC(O)(C(C)NC(=O)C(F)(F)CN(C)C)C1)=O 89074,CC12CC(C(=O)NCC(CNC(c3cn(CCCF)nn3)=O)CO)(CCO1)C2 89075,c1(CNC(CCc2cn(C(CN3CCC(C)CC3)C)nn2)=O)ccc(Cl)cc1F 89076,C(C)(C)(CCC(=O)N(C)CC1CN(C(=O)C(c2ccc(Cl)s2)C)CCO1)OC 89077,c1(OC)cc(CNC(=O)CC2(C)CN(Cc3cc(CO)ccc3O)C2)ccc1F 89078,c1(C(N2CC=CC(C(=O)NCCC34CCC(C3)C4)C2)=O)cc(O)ncn1 89079,Nc1cc(Cl)cc(Cl)c1C(=O)NCCC(O)CNC(c1cnc(C2CC2)[nH]1)=O 89080,c1(C(N2CCN(C(=O)Nc3cccc(C)c3)CC2)=O)cc(Br)cc2ncoc12 89081,c1(OC)ccc(C(C2CCCO2)NCc2oc(C)nc2C)c(C(F)(F)F)c1 89082,c1(C(=O)NCCN(C(COCCC#C)=O)CCCN(C)C)cnnc(O)c1 89083,C(=O)(CCCCN1CCCC1)NC(CC(C)NC(c1[nH]cc(CC(C)C)c1)=O)C 89084,C1(C(=O)NC2CN(C(C3CCN(C)CC3)=O)CC(O)C2)CCc2ccccc2C1 89085,CCC(C)N(OC)C(=O)COC(=O)C1=NOC(C)C1C.C1CO1 89086,c1(NC(N(CC(F)(F)F)CCCOC)=O)ncc2cnccn12 89087,CC(C)C(C)C(CNC(=O)COC1CC1)NC(c1c(Cl)n[nH]c1C1CC1)=O 89088,C(C(=O)Nn1nnc(C)c1C)(C1CCCC1)N(C(C(NOC)=O)=O)C1CC1 89089,CC(C)C(C)(CNC(=O)C(C)Oc1ccc(F)cc1)NC(=O)C=Cc1cocn1 89090,N1(C(CCCOCC)=O)CC(NC(c2nc(C)n(C)n2)=O)CCC1C 89091,Cc1cccc(CCCNC(c2nc[nH]n2)C)c1 89092,c1(-c2nc(C(CC)O)nn2-c2ccc(F)nc2)ccc2ocnc2c1 89093,C(=O)(C1=CCc2ccccc21)NC1C(NC(C(c2ccc(Cl)cc2)C)=O)C1 89094,c1(C(=O)NCC(C)(C)CS(C)(=O)=O)ccc(C#CCN)cc1 89095,C1(S(N)(=O)=O)(C(=O)NC(C(C)NC(C2CCCC(=O)N2)=O)CO)CCCC1 89096,C(=O)(CCC(CC)CC)N(CCNC(CCn1ncc(C(=O)OC)c1)=O)C(C)C 89097,c1(OC)ccc(O)c(CN2CC(NC(=O)CCCCCBr)C2)c1 89098,C1(CC)CN(C(c2occc2CNC(=O)C(n2cc(C)cn2)C)=O)CC(=O)N1 89099,c1(C(=O)NC(C2CCCN(C(=O)C=CS(C)=O)C2)C)cc(C(C)(F)F)ccc1Cl 89100,C1(NC(C(CC)C(C)C)=O)CCC2CCN(C(=O)C(O)C(C)C)C1C2 89101,c1(C(=O)NC2(CC=C)CN(C(C3(OC)CCOCC3)=O)C2)cnc(S(C)(=O)=O)s1 89102,c1(OC)n[nH]c(NC(C2CN(C(C3CCCC3C)=O)CCS2)=O)c1C#N 89103,N1(C(CSC(C)C)=O)CC2(C(N3CCOC(C(C)(C)C)C3)=O)CCC1CC2 89104,N1(C(c2cncc(C#C)c2)=O)CCC2CN(C(c3ncc(OC)cn3)=O)CC12 89105,C1(C(=O)NC23C(CN(C)C2)C3)CC1C1CN(C(c2c[nH]nc2C2CC2)=O)C1 89106,N1(C(=O)OC)CC(NC(C2(n3cc(CSC)nn3)CCC2)=O)CC(O)C1 89107,CC1C(NC(C2CC(O)C2)=O)CC2CCC1N2C(C1(CF)CCC1)=O 89108,Cc1c(NC(=O)Cn2cc(C(=O)O)nn2)cccc1N=[N+]=[N-] 89109,N1(C(c2nccc(N(C)C)c2)=O)CC=C(CNC(=O)C(O)C2CCC2)CC1 89110,C1(N(C(c2ccc(CC)o2)=O)C)CCCCC1NC(C1CCCC1C(=O)OC)=O 89111,C(CC(C(C)(C)C)NC(c1cc(F)cs1)=O)N(C(c1c(CC)n(C)nc1)=O)C 89112,C1(CNC(c2cccc(NC)c2)=O)CCC2(CCC2)C1NC(C1CS(=O)(=O)C1)=O 89113,N1(C(CC(C)SC)=O)CC2CC(C1)CN(C(=O)CC1CCN(C)C1=O)C2 89114,C1(C(=O)NCC(=O)OCc2ccc(F)cc2)CCC(F)(C(=O)OC)CC1 89115,c1(CC)cc(C(=O)NCCCOCCNC(C2COC(=O)N2C)=O)ccc1F 89116,C1(NC(C(CC)O)=O)C=CCCC1C(=O)NCC1CCCC12CC2 89117,c1(C(=O)NC23CCN(C(c4c(N)non4)=O)CC2C3)cc(O)nc2c1CCCC2 89118,CC(O)CC(=O)NCC1(C(=O)NCCCC2CCCC2O)CC1 89119,C1(N(C(C(C)C2CCC2)=O)C)C2CN(C(=O)CCc3ccc(N)cn3)CC12 89120,Cc1cc(F)c(C(=O)NCCN(C(c2ccnc3c2CCC3)=O)C2CC2)cc1F 89121,C1(C(=O)NCC(=O)NC(C)C)CCN(C(=O)C(N2CCOC2=O)C)C1 89122,c1(SC)cncc(C(N2CCCCC2Cc2[nH]c(-c3cnccn3)nc2C)=O)n1 89123,N1(C(C2C(CC)CCC2)=O)CCC(C2(O)CN(C(c3coc(CO)c3)=O)C2)CC1 89124,c1(C(=O)NCCC(=C)CNC(c2cc(COC)[nH]n2)=O)ccc(C2CC2)c(F)c1 89125,c1(C(=O)NC2CCC(NC(C(C)OCCC#C)=O)C2)ccnc2c1ncn2C 89126,Cc1c(C(C)C(=O)NC2(C)CN(C(C3CCCN3C=O)=O)C2)cccc1Br 89127,c1(C(=O)NCCNC(Cc2c(C)ccc(F)c2)=O)cccc2c(C)ccnc12 89128,Cc1c[nH]cc(C(=O)NC(C(C)NC(c2cn(C)nc2C(C)C)=O)C(C)C)c1=O 89129,c1(C(N2C3CC(N(C)C(c4nncs4)=O)CC2CC3)=O)cccc2c1ncn2C 89130,N1(C(CC(=O)OC)=O)CCC(CC(N)=O)(NC(c2ccsn2)=O)CC1 89131,C(=O)(C1CCc2cccc(F)c21)NCC(=O)Nc1c(C)noc1C 89132,CCC(CCCC(=O)N(CC(O)(CC)CC)C)NC(=O)CC1CCCC(=O)C1 89133,N1(C(C(=O)NC(C)(C)C)C2C(C)C2)CCC(C(=O)OC)C(C(N)=O)C1 89134,N1(C(c2n(CC)nc(C)c2)=O)CCC2CCC(NC(=O)C=CC3CCC3)C12 89135,N1(C(CCOCCC)=O)CCCC(C2CCN(C(=O)CC(F)F)CC2)C1 89136,N1(C(=O)OC(C)(C)C)CCC(C)(CC(O)C(=O)N2CCC2C(F)F)C1 89137,N(C1CCCc2ccoc21)C(C1(NC(C(C)C2CCCO2)=O)CCC1)=O 89138,Cc1cc(=NC(=O)N2CC(C)CCC2CO)[nH]nc1-c1ccccc1 89139,c1(C(N2CCC(NC(C=CCC)=O)(CO)C2)=O)nc2ncccn2n1 89140,C1(C)(CNC(C(c2cn(CC)nc2)=O)=O)CCCN1C(=O)CCOCC(F)(F)F 89141,C1(C(N)=O)C=CC(NC(c2coc(CNC(c3csc(O)n3)=O)c2)=O)C1 89142,N1(C(C2CCC(C)N2C(=O)CN2CCOCC2=O)=O)CCc2cnccc2C1 89143,C1(C(=O)NC(C(C)NC(C=Cc2ccc(CC)o2)=O)CO)CCn2nnnc2C1 89144,N1(C(C(CC=C)N(C)C)=O)CCCCC2C1CCCN2C(=O)COC1CCC1 89145,N1(C(=O)CCc2cnn[nH]2)CCC(NC(=O)COC2(F)CC2)CC1 89146,c1(CN2C3CCN2C3)ccc(OC(F)F)cc1F.CC(CCO)c1cnn[nH]1 89147,N1(C(CCC(CC)OC)=O)CC2CCCC2(NC(c2c[nH]nc2Cl)=O)C1 89148,c1(SC)cc(CN(C(=O)CC(N2CCCCCC2)C)CCO)ccn1 89149,c1(C(=O)NCC(=O)NCc2cccc(OCF)c2)c[nH]c2ncccc12 89150,C(=O)(CCC(C(C)C)NC(C1(C)CC(=O)C1)=O)Nc1ccc(C#C)nc1 89151,C1(C(C)C)CN(C(=O)CCC(=O)NCC(N2CCCC2)=O)CCC1NC(=O)CO 89152,C1(CNC(C2N(C(CCCNC(=O)OCC)=O)CC2)=O)CCCC1(F)F 89153,N1(C(Cc2cn(C)nn2)=O)CCC(F)C(NC(=O)CN2CCOCC2)C1 89154,c1(C(C)NC(=O)C(=O)N(C)CC2CCOC2C)cccc(Cl)n1 89155,N1(C(c2c(C(=O)OC)cccc2)=O)CCN(C(=O)CC2CC2C)CC(O)C1 89156,c1(C(N(C2CCCC(NC(C3CC(=C)C3)=O)C2)C)=O)cnn2cc(C)cnc12 89157,O=CN1CCCC1C(N1CCOCC1C(=O)NCCC1(O)CCC1)=O 89158,Cc1c(Cl)sc(Cl)c1C(N1CC(O)(CNC(=O)Cn2ccnn2)C1)=O 89159,C1(NC(C(C)CC2CC2)=O)CC2CCC1CN(C(c1ccc(=O)n(C)c1)=O)C2 89160,CCCCCCC(C)C(=O)NCC(C(=O)N(C(C)CO)CC)OC 89161,N1(CC(=O)NCCCN(C(C(C)N2CCCC2)=O)C2CC2)CCC(C)(C)C1 89162,CC1CCCn2c(C(N3CCCC(N4CC(O)C4)C3)=O)cnc21 89163,C1(NC(c2n(C)ncc2)=O)CCCCC1NC(c1ccncc1F)=O 89164,N1(C(C2C(CC)CCC2)=O)CC2CCCC(C1)N2C(c1ccc2cnsc2c1)=O 89165,C12(C(=O)NC3CCCN(C(c4ccc(NC)c(F)c4)=O)C3)CCCCN1CCC2 89166,N1(C(C(Cc2ccoc2)NC(c2c(OC)cnnc2)=O)=O)CC(O)CC(O)C1 89167,C1(NC(=O)NC2(CC)C(c3ccccc3)CC2)C2CCC3C(C2)C13C(=O)OCC 89168,c1(C(C)OC)nc(NC2(CO)CCCN(C(=O)C(C)C(C)COC)C2)cc(Cl)n1 89169,N1(C(C=CC(CC)C)=O)CC2CCC(C1CO)N2C(=O)CCC1CCCCCC1 89170,CC1CCN(C(c2c[nH]nc2C(C)(C)C)=O)CCN1C(C1CN(C)CC(C)O1)=O 89171,c1(C(N(C2CCCCN(C(CC3(CSC)CC3)=O)C2)C)=O)cc2ccccc2o1 89172,CC1CN(C(=O)NCCCCc2ccc(F)cc2F)CC(C)S1(=O)=O 89173,C1(NC(c2ncn(C)c2)=O)CN(C(C2CC(=C(F)F)C2)=O)CC2(CCC2)C1 89174,c1(CC(=O)NCC2C3CN(C(C(C=C)(F)F)=O)CC32)noc2ccc(F)cc12 89175,N1(C(c2cc(C)sc2)=O)CCCC1C1CCCN1C(C1CCc2nc[nH]c2C1)=O 89176,C1(C(C)NC(c2c[nH][nH]c2=N)=O)CCCN(C(c2cc(N)cnc2)=O)C1 89177,Cn1cnc2cc(C(=O)NC3CC4(NC(=O)CC5(CO)CC5)COC3C4)ccc12 89178,C1(NC(c2ccc3cnnn3c2)=O)COC2(C1)CN(C(c1cc(Cl)ncc1O)=O)C2 89179,C(C#Cc1ccccc1)O.C(=O)(NNC(=O)C1(C2CC2)CCOC1)N(C)CC1CC1 89180,C(=O)(C1=NNC(=O)CC1)N1CCN(C(C=Cc2cc(OC)ns2)=O)C2C1C2 89181,C1(C(=O)NC(CCCNC(c2onc(COC)n2)=O)C)CCCCNC1=O 89182,O=C(CC(C(F)F)NC(=O)CN1CCCC1)NC1CC2OC1C1CC21 89183,c1(C(N(C(CCNC(c2c(SCC)cccn2)=O)C)C)=O)cnc(O)n(C)c1=O 89184,C1(NC(CCCN(C)C)=O)CN(C(c2ccc(O)cn2)=O)CC1N=[N+]=[N-] 89185,C1(C(=O)NC2CC(C)(NC(C(C(C)C)C)=O)C2)CC(F)(F)C1(C)C 89186,c1(C(N(CCCN(C(c2nccc(C)c2O)=O)C)C)=O)cc2cccc(F)c2o1 89187,C#CCC(O)C(=O)NC(C)(C)CNC(=O)C(=Cc1ccccc1)NC(C)=O 89188,C12(C(N3CC(F)(CC)C3)=O)CCC(CC1)N(C(C1CC1(C)C(F)F)=O)C2 89189,c1(C(N(C)CC2COCCN2C(C2SCCCS2)=O)=O)cccc2nc[nH]c12 89190,CC(C(=O)NCCCN(C(=O)Cc1ccc(Br)s1)C)C(F)(F)F 89191,c1(CNC(c2[n+]([O-])ccc(OC)c2)=O)ccc2c(c1)CN(C(=O)C(C)C(C)O)C2 89192,C1(CC(=O)NC2C(C)N(C(=O)Cc3csc(=N)[nH]3)CCC2)SC2=NCCN2C1=O 89193,Cc1c(CN2CCC(N3CCCC3=O)CC2)cc([N+](=O)[O-])cc1[N+](=O)[O-] 89194,C1(NC(CC(C)OC)=O)CC2CCC(C1C)N2C(c1ccc(C(=O)CF)cc1)=O 89195,c1(C(=O)NC(C(N2CCC(N(C)C)C2)=O)C2(O)CCC2)ccc2c(c1)CC2 89196,c1(OCC(=O)NC2CC2CNC(c2ccnn2C2CCC2)=O)cccnc1 89197,N1(C(CCN(CCC)C(C)=O)=O)CCC(O)(CC)C1 89198,N1(CCOC)CCC(NC(=O)Nc2cc(-n3ccnc3C)ccn2)CC1 89199,C1(CNC(C(c2n(C)ncc2)(C)C)=O)CN(C(C2CCC(C)CC2)=O)CCO1 89200,n1(CC)cc(C(=O)N(CCCCCCNC(=O)OC(C)(C)C)C)c(OC)n1 89201,n1(C(CC)(C)C)nnnc1C(c1c[nH]nc1C(C)(F)F)NCCc1cnn(C)c1 89202,C1(NC(C(C)(C)OC)=O)(COC)CCN(C(=O)C(O)Cc2cccc(Cl)c2)C1 89203,C1(C(=O)NC(C2CC(NC(C=C(C)C)=O)C2)C)C2CCCC12 89204,c1(C(=O)NC2(CCNC(C3CCOC3)=O)CCCC2)cnc(-n2cccn2)cn1 89205,C1(CC(N2CCOC(CNC(=O)C(n3ccc(C)n3)C)C2)=O)(OC)CCCCC1 89206,c1(SC(C(=O)NC2CCC(NC(C)=O)C2)C)ccc(Cl)cc1 89207,C(CCC(C)NC(c1ccnn1C)=O)NC(CC1C(CC)C1)=O 89208,C1(C(N2CCN(C3CCOCC3)CC2)=O)(CN)CC2(CC(F)C2)C1 89209,c1(C(=O)NC(CC(C)NC(c2nnn(C)c2C(F)(F)F)=O)C)cc2n(c1)CCC2 89210,C1(CC(C)NC(C2CSCCS2)=O)CCN(C(=O)C(C)(C)N2CCCCC2)CC1 89211,C1(C2CC2)(C(N(CCCOC)C)=O)CN(C(=O)CC2CCCSC2)C1 89212,C#Cc1cnn(C)c1C(N1CCOC(C(=O)NC(c2cn(C)nc2C)C)C1)=O 89213,C1(NC(c2cc(CNC(C34CCN(CC3)CC4)=O)[nH]n2)=O)COCC1C1CC1 89214,c1(NC(C2CCCN2C)COC)nc(NCc2nnc(O)n2C)c2ncsc2n1 89215,c1(C(=O)NCCC(CNC(c2ccc(C)cc2Cl)=O)(C)C)ccn2nncc2c1 89216,c1(C(=O)NCC(CC=C)NC(=O)C(C)(CC)CO)ccc(CC)c([N+](=O)[O-])c1 89217,c1(CNC(C(CC)NC(N)=O)=O)cnn2c1CN(C(C1CC1CN(C)C)=O)CC2 89218,c1(C(C(=O)NC(CN(C(C(n2ccc(C)n2)C)=O)C)(C)C)F)ccc(F)cc1 89219,C12(COC)COC(C(N3CC(CNC(=O)C(C(C)C)ONC(=O)OC)C3)=O)(C1)C2 89220,c1(-c2c(C)ccs2)csc(=Nc2cccc(OC)c2)n1CC1CCC(C(F)(F)F)C1 89221,C(=O)(C(C(C)O)N(C)C)NCCC(=C)CNC(=O)CCCCN(C)C(C)=O 89222,c1(C(C)=O)cc(C(=O)N(CC(C)CNC(=O)Cc2cnc(C)o2)C)co1 89223,CC1CCC(C)(C(N2CCC(=CCNC(=O)CC3(C)OCCO3)CC2)=O)C1 89224,C1(NC(CN(CCOC)C)=O)CN(C(=O)CCc2scnc2C)C(C)(C)C1 89225,Cc1cc([N+](=O)[O-])ccc1C(=O)Nc1nnn(C(F)(F)F)c1C(N)=O 89226,C1(OC)CC(N=c2[nH]c(=NC(C)c3ccncc3F)c3ncccc3[nH]2)C1 89227,N1(C(c2sc(C)c(O)n2)=O)CCN(C(c2cc(O)c(F)cc2N)=O)C2COCC12 89228,n1(CC)cc(Br)c(C(=O)N(CC(C)NC(=O)CCc2ccncc2)CC)n1 89229,c1(C(N2C(CC(=O)NCCNC(C)=O)CC3(CC3)C2)=O)ccc2c(c1)OCCCO2 89230,Cc1cc(C(=O)NC2CCC2NC(=O)C=Cc2nnn(C)n2)n(C2CCC2)n1 89231,CC(C(=O)NC1CCN(C(c2ccc(Cn3ccnn3)cc2)=O)CC1)C(C)(F)F 89232,C1(CNC(CNC(=O)OCC)=O)CN(C(C2COCCO2)=O)CC1(C)C 89233,C1(C)(C(N2CC(C(C)OC)C2)=O)CCN(C(=O)C=C(C)C(C)C)C1 89234,c1(C(N(CC(CC)NC(c2c[nH]c3ccncc23)=O)C)=O)onc2ccccc12 89235,N1(C2CN(C(c3ccc(SC)cc3)=O)C2)CC(NC(=O)COC(F)(F)F)CC1=O 89236,c1(C(=O)NCc2cn(C)nc2C(F)F)c(F)ccc(O)c1F 89237,c1(C(=O)NC2CN(C(=O)OCCN(C)C)C(=O)C2)ccc2occc2c1 89238,CC1(C)CCCC(C)(C)C1C(N1CCCC1CNC(C1CCN1S(C)(=O)=O)=O)=O 89239,C12(CNC(=O)CC3CCC(O)C3)CN(C(c3cc(C4CC4)on3)=O)CC(F)(C1)C2 89240,c1(C(N(C2CCN(c3nnc(CO)s3)C2C)CCC)=O)ccc(C)cc1Cl 89241,C1(NC(C2C(CC(C)C)C2)=O)CCC(CNC(=O)C(C)Cc2cccnc2)CC1 89242,C(=O)(C(CCOC)OC)NC.c1(C(=O)NC(CC)COC)nc(C(=O)NCC)oc1C 89243,CC(C)C1CCC(=O)N(C)CCO1.c1(SCC(=O)NCC2CC2)nc[nH]n1 89244,N1(C(C(C)OCC#C)=O)CCOC(CC(=O)NCCc2ocnc2CO)C1 89245,c1(OC)c(C)ccc(C(N2CC3(C2)CN(C(C2CC(C)OC2=O)=O)C3)=O)c1F 89246,c1(C(=O)NCC2C(C)CCN(C(CC(CC)(C)C)=O)C2)c(N)cc(Cl)cc1F 89247,c1(C(=O)NCC2CN(C(CC(C=C)(C)C)=O)C(C)C2)cc(C)c(C)cc1N 89248,C1(NC(C23CCC(NC(C(COC)N(C)C)=O)(CC2)C3)=O)CC2(C1)CC(C#N)C2 89249,C1(CNC(=O)CC2CCNC2=O)CN(C(C2(O)CCCCC2)=O)CCO1 89250,N1(Cc2c(C)n[nH]c2)CCCC2(CCCN(C(c3ncsc3C)=O)C2)C1 89251,Cc1cccc(Br)c1C(=O)N(CCCNC(=O)C(F)C(C)C)C 89252,N1(C(C2CCC(=C)CC2)=O)CCCC1C1CCCCN1C(C1CSC1)=O 89253,CC1CC(C(N2CC(NC(c3nc[nH]c3C(C)(C)C)=O)C2)=O)C1(C)C 89254,N1(C(CN2C(C)CCC2)=O)CC(N(C(=O)Cn2ccc(O)nc2=O)C)C(C)(C)C1 89255,c1(C(N2C(CCC)CN(C(=O)CS(=O)CC)CC2)=O)c(Cl)ccc2cccnc12 89256,N1(C(C=C2CCN(C(c3c(OC)ccs3)=O)CC2)=O)CCNC(=O)CC1 89257,Cc1c[nH]nc1CNC(=O)CC1CCC(NC(=O)C(C2CCOCC2)O)C1 89258,C(=O)(C(C)C(O)C(C)C)NCC1CC(Cn2cc(Cc3c(C)nc(CC)o3)nn2)C1 89259,CC(CO)C(=O)NCC1(C(=O)NC(CN2CCCC2)CO)CCC1 89260,N1(C(C2N(CC)CCC2)=O)CCCC(O)(CNC(=O)CCc2ccncc2)CC1 89261,N1(C(C2=NOC(C)C2)=O)CCCN(C(=O)COC2(C)CCCC2)C(C)C1 89262,CC(C)(O)C(CCO)NC(C1CC2(CC2)CN1C(=O)CCc1cncs1)=O 89263,N1(C(C2(CC)CCCN2C(c2ccc(CC#N)cc2)=O)=O)CCCC2(CCO2)C1 89264,[N-]=[N+]=NC1CN(C(C2CC2CF)=O)CC1NC(=O)COCc1ccccc1 89265,N(C(=NCC1CCC(=O)NC1)N1CCC(CCC#N)CC1)CC(=O)NC 89266,C1(NC(Cc2nc(C)oc2)=O)CC=CCC1C(=O)NCC(N1CCCC1)C 89267,c1(CC(C(=O)NCCC(C)NC(c2cn(CC)nc2)=O)O)cc(Cl)cc(Cl)c1 89268,C1(CNC(C2N(C=O)CC2)=O)CC2COCC2N1C(c1ccc(Cl)cn1)=O 89269,N1(C(c2c(CC)ocn2)=O)CCC2CN(C(c3ccc(N)cc3O)=O)CCC2C1 89270,C(=O)(C1=CCCOCC1)NCC1(F)CCN(C(c2cc(N)cc(F)c2)=O)C1 89271,N1(C(c2nc(C(C)=O)sc2)=O)CC(NC(C2CCC(C)(C)O2)=O)C2(CC2)C1 89272,N1(C(c2c(N)ccc(C)c2)=O)CC(NC(c2cc(F)cs2)=O)C(S(C)(=O)=O)C1 89273,c1(CC)ncc(C(=O)NC23CC(NC(=O)CC4CC4(C)C)(C2)C3)c(C)n1 89274,Cc1nc(C(=O)N(C)CC2CCCN2C(=O)C(C2CCCO2)C2CC2)c(C)o1 89275,c1(Nc2ccc(C(CCC(=O)OC)(C)C)cc2)cc(O)nc(SCC(F)(F)F)n1 89276,C=CC1(CNC(=O)NC2CC2C#N)CCCCC1 89277,S(=O)(=O)(c1cccc2c1OCCC2)N1CC(O)CC(OCC)C1 89278,N1(C(C(C)(CO)OC)=O)CCC2OCCN(C(=O)C=C(C)C(F)F)C2C1 89279,c1(CC)cc2c(NCCCCCCNC(c3ccc(C)cn3)=O)nc(C)nc2s1 89280,c1(C(=O)NCC2CN(C(CC(C)(C)OC)=O)CC2O)cc(=O)c2ccccc2o1 89281,c1(C(=O)NC2(CF)CCN(C(C3CCC(CC)O3)=O)C2)ccc(=O)n(CCO)c1 89282,N1(C(Cc2ccc(SC)cc2)=O)CCC2(C)CN(C(=O)CCc3cnc[nH]3)CC12 89283,Cc1ccc(N(C(C)C(C)C)C(=O)NC2CCN(C(C)C3CC3)C2)cc1N=[N+]=[N-] 89284,N1(C(c2c(CN(C)C)cccc2)=O)CC2(C1)CN(C(C1CCC3CC3C1)=O)C2 89285,N1(C(CCC=C)=O)CCN(C(=O)Cn2cc(Br)ccc2=O)CC1CC1CC1 89286,C1(C(N2CCC(CC#C)C2)=O)CN(C(=O)C(C)CSC)C(C)(C)C1 89287,CCC(CNC(=O)C(c1cccs1)NC(=O)C#CC1CC1)C(C)C 89288,C(c1cnc(O)nc1O)=CC(N1CC(C)C(NC(=O)C(C)C(C)(C)C)CC1)=O 89289,c1(C(N2CC(CC)C(C(=O)NCC(O)CO)C2)=O)cc([N+](=O)[O-])c[nH]1 89290,N1(C(CSCCOC)=O)CC2(C1)CN(C(c1nscc1C)=O)C2 89291,C1(OC)CN(C)C(C)(C(N2CCC(CN(C)CCOC)CC2)=O)C1.c1ccccc1 89292,C=C(CNC(C12CC(CO1)C2)=O)CCNC(=O)C(C1CCCO1)OCC 89293,CCC1=C(C(=O)NCC2CN(C(C3CCCN3C(C)=O)=O)CCN2C)CCCO1 89294,N1(C(C)=O)CCC2(CC1)CCN(c1ncnc(=N)[nH]1)CC2.c1cc(F)ccc1F 89295,c1(CCC(=O)NCC(c2ccccc2)NC(C2CN(C3COC3)C2)=O)nc(O)n[nH]1 89296,c1(C(=O)NC(C2CCN(C(C3(C)CC(=C)C3)=O)CC2)C)ccc(C)c(C)c1Cl 89297,Cc1cc(C(=O)NCCCCN(C(=O)Cc2ccnn2C)C)c2cnn(C)c2n1 89298,N1(C(C(CC)(F)F)=O)C2CCC(C2)C1CNC(c1nc(Br)cnc1N)=O 89299,n1(CC(N2C(CNC(COCCOCC#C)=O)CC2)=O)cc([N+](=O)[O-])cn1 89300,N1(C(C(=O)NCC)=O)CCC2OCCN(C(=O)CCSCc3ccccc3)C2C1 89301,N1(C(C(CO)NC(N)=O)=O)CC2CC1CN2C(=O)Cc1cc(Cl)ccc1Cl 89302,CCC(C)CC(=O)C(=O)NC(CO)C(=O)NCC1CCc2nccn21 89303,C(=O)(CCCCC(=O)OC)N1CC(O)(C(C(=O)NCc2c(C)nc(CC)o2)F)C1 89304,c1(N2CCC(NC(c3c(C)ccc(C)n3)=O)C(C)C2)ccc([N+](=O)[O-])c(C#N)c1 89305,C#Cc1ccc(C(=O)NCCC2(O)CCN(C(C3(CC)CC3(F)F)=O)CC2)cc1 89306,C(CCCCC(=O)N1CC(NC(=O)CC2CC2(Cl)Cl)CC1(C)C)OCC 89307,C#CCCC(C(=O)N1CCC(=C)CC1)NC(=O)CC1CCOC1=O 89308,Cc1nc(Nc2cc(Cl)n3nccc3n2)c2c(n1)CNCC2 89309,C(C(C)(C)C(=O)N1CC(F)CC1CNC(=O)C(C)Oc1ccc(Cl)cc1)OC 89310,C1(NC(CC=C)=O)CN(C(c2ccc(C(N)=O)o2)=O)CC1C(F)F 89311,C1(CCCC)(NC(c2cn(CCC)nc2)=O)CCN(C(=O)C(O)COC)C1 89312,N1(C(Cn2cc[n+](C)c2)=O)CC2CC1(CO)C2.C1(C(=O)N)CC12CCOC2 89313,c1(C(N(CC(C)NC(C(C=C)CC)=O)C)=O)ccn(C)c(=O)c1 89314,C1(O)(COC)CCN(C(=O)C(=O)Nc2cccc(-c3ccccc3)c2)CC1 89315,N1(C(C(c2ccoc2)OCC(=O)NCC2CCCC2)=O)CCCC(O)CC1 89316,CC1(C)C(CNC(c2cc(C3CCC3)no2)=O)CCN1C(C1CC1C(F)(F)F)=O 89317,c1(CNC(=O)NCCSCC(F)F)ccc2c(c1)CCO2 89318,N1(C(=O)OC(C)(C)C)CCC2CC(NCC3CCOC(C(F)F)C3)CCC12 89319,c1(NC(C(C)NC(c2cccc(CC)n2)=O)=O)cnc(CO)nc1C 89320,C1(NC(C2N(C(C)C)CCC2)=O)CCC2CN(C(c3cnnc(O)c3)=O)CC2C1 89321,C(C1c2ccsc2CCN1C(C1CCCOC1)=O)NC(Cc1nc(CC)sc1)=O 89322,Cc1cn(CC(=O)NC2CC23CCC(NC(=O)C(C)O)CC3)c2ccccc12 89323,C(C)(CO)(C(F)(F)F)NC(c1cn(CCNC(c2cc(OC)n(C)n2)=O)nc1)=O 89324,C1(CN(C(=O)CC23CC(C2)C3)C)CCN(C(=O)CCc2ccncc2)C1 89325,C1(CC(N2CC(CNC(CN(C)C3CC3)=O)C2)=O)CC2(CCCC2)CO1 89326,c1(C(CC)C)nccc(=NCC23CC(NC(c4[nH]ccc4COC)=O)(CO2)C3)[nH]1 89327,C1(C(N(c2ccc(C(=O)OC)cc2)C)=O)CC(=O)N(C)C1c1cnn(C)c1 89328,C(=O)(C1=CC2(CCN(C(c3ccsc3Cl)=O)C2)C1)N(C1C(C)CCCC1)C 89329,N1(C(C(F)=C(C)C)=O)CCOC(CCNC(=O)CCc2nccn2C)C1 89330,C12(C(=O)NCCC(C(=O)OC)C)COC(C1)C(NC(c1scnc1C)=O)C2 89331,N1(C(CCC(CC)C)=O)CC2CCOC2(CNC(c2cc(C)ccc2Cl)=O)C1 89332,Cc1c(C(N2CC(CO)OC(CO)C2)=O)[nH]c2cc(Cl)ccc12 89333,CCS(=O)(=O)c1ccccc1C(=O)NCc1ncoc1CCNC(=O)C(C)(C)O 89334,C1(CNC(C(Cc2ncn(C)c2)O)=O)CCC(NC(c2cnc(O)n2C)=O)CC1 89335,N1(C(COCP(C)(C)=O)=O)CCC2CCN(C(C3CSC3)=O)C2C1 89336,c1(C(=O)NC2CCC(C(N(C)CC#N)=O)CC2)c(Cl)cc(F)cc1Cl 89337,Cc1cc(C(=O)NCC(C)N(C)C(C2CCOC(=O)N2)=O)c2c(n1)CCCC2=O 89338,N1(C(C(C)NC(C)=O)=O)CCN(C(=O)CCCc2nccs2)C(c2cn[nH]c2)C1 89339,N1(C(c2cccc(NC)n2)=O)CCC2(CCCCC2NC(=O)CC(C)C2CC2)C1 89340,S(=O)(=O)(c1ccc(Br)cc1F)NCCC(=O)NCCCc1cnon1 89341,C12(C(=O)NC(C3CCN(C(Cc4cc(C)no4)=O)C3)C)CC3CC1C2C3 89342,c1(C(c2n(CC)nnn2)NCCOC(C2CC3CC3C2)=O)ccc(F)cc1 89343,C1(CNC(C(C)=C2CCC2)=O)CN(C(c2cccc(Br)c2)=O)CCC1(C)C 89344,Cc1c(C(N2CC(NC(c3cnc(C(C)(C)CF)o3)=O)C2)=O)nn(C)c1C1CC1 89345,c1(C(N2CCN(C(C3CC4CCCCCC34)=O)CC2)=O)cc(O)ccc1Cl 89346,C(C(C)(C)C(=O)NCCF)N(C(=O)C(C1CCOCC1)=O)C 89347,c1(C(=O)NCC2CC2NC(C2(Cl)CCC2)=O)ccc2c(n1)CCC2 89348,c1(C(N(CC(CC)NC(=O)C(CC)SC)C)=O)cc(C)c2c(O)n[nH]c2n1 89349,C(CC1=CCCCCC1)NCC1(CO)CCN(Cc2ccc(F)cc2)C1 89350,c1(C(C)C)cc(=NC2CC(NC(=O)CCOCC(F)F)C2)[nH]c(C(C)(C)C)n1 89351,N1(C(C(CC=C)(C)O)=O)CC(NC(c2c[nH]c(C(N)=O)c2)=O)C2(CCC2)C1 89352,C(=O)(CC1=CCCC1)NC(C1CCN(C(c2conc2C(F)(F)F)=O)CC1)C 89353,CC1(C)CCC=C1C(=O)N1CCCN(C(c2ccc(F)c(Cl)c2)=O)CC1 89354,c1(NCN(C(C(=O)N(C(CC)C)CC)C)CC)ccc2cccc(F)c2n1 89355,N1(C(C(C)(C)N2CCC2)=O)CCOCC(C(N2CC(SC(F)F)C2)=O)C1 89356,c1(C(=O)NCCC(CNC(=O)Cc2c(F)cccc2Cl)O)ccn2nncc2c1 89357,c1(C(=O)NCc2cccc(C(N(CCC(=O)OC)C)=O)n2)c(O)cccc1F 89358,N1(C(C(C=C)O)=O)CC2(C(=O)NCC(O)C(=O)OC)CC1CO2.C 89359,c1(C(=O)NC(CCNC(c2ccc(CC)[nH]2)=O)C)ccc2c(=O)n(C)cnc2c1 89360,Cn1ncc(C(N2CC(CNC(=O)CCOCC(F)(F)F)C(O)C2)=O)c1Cl 89361,c1(C(N2CC(CCCNC(C(C)SCC)=O)OCC2)=O)cc(=O)c(O)c[nH]1 89362,C(CCNC(C1(NC(C2C(C)(C)C2(C)C)=O)CC(O)C1)=O)(C(C)C)OC 89363,C(CC(=O)NC(c1cscn1)CO)(C(F)(F)F)NC(=O)CC1COCCOC1 89364,C1(CC(C)NC(c2cnc(CC)s2)=O)CCN(C(=O)C(C)(C)c2ccns2)CC1 89365,Cc1ccnc(CN2CCCC2CCNC(c2cccc(-c3nn[nH]n3)c2)=O)c1 89366,c1(NC2(C3CN(C(C4C5CCCC45)=O)C3)CC2)ccc2cnccc2c1[N+](=O)[O-] 89367,Cc1nnc2cc(N3CC(NC(C4CSC4)=O)CC3C)ncn12 89368,N1(C(C(CCCC)C)=O)CC2(CCCCN2C(=O)CCOCC(F)F)C1 89369,CC(C)C(CNC(C1CCCCO1)=O)C(=O)Nc1cccc(OC(F)F)c1 89370,N1(C(c2c(Cl)cnc(-c3cccc(C)c3)n2)=O)CCCC2NC(=O)CCCC12 89371,C1(C)(CNC(C=CCCC)=O)CCCN(C(=O)C=Cc2nc(C)cs2)C1 89372,C(=O)(C(CC)C(C)(C)CC)NC(CCC)CNC(=O)C(CC)N(CC)CC 89373,c1(CC)c(C(=O)NC(C)CN(C(=O)C(C)(C)C2CCOC2)C)nnn1C 89374,c1(C(CNC(=O)CCC2CCCO2)=O)csc(Sc2ccco2)n1 89375,Cc1ccccc1NC(=O)C(N1CCOC(Cc2cccs2)C1)c1ccc(Cl)s1 89376,c1(-n2cc(CCC#N)nn2)ccccc1CC(N1CC(C(=O)O)C2CC12)=O 89377,c1(N(C(N(C)C)=O)C)ccc(NC(=O)NCc2cn(CCCCO)nn2)cc1 89378,Cc1cc(C=CC(=O)NC(C)C(C)NC(=O)C(C)(Cl)Cl)ccc1C(F)(F)F 89379,C1(CC=C)(NC(c2occc2CC)=O)CCCN(C(c2cncc(N)c2)=O)C1 89380,c1(C(=O)OCc2cc(OC)nn2C)cccc(S(=O)(=O)N(C)C)c1 89381,N1(C(c2n(C)cnc2)=O)CCC(CNC(c2ccn3ncnc3c2)=O)C(F)(F)C1 89382,CC(C)CC(CC(=O)NCC1CC(C)(C)CN1C(c1cnc(O)o1)=O)CC(N)=O 89383,c1(OC)ccc(C(=O)NCC(O)CN(C(=O)C2=CCCSC2)C)cc1OC 89384,C=CCC(C(=O)N1CC(O)CC1C(=O)NC1(C2CCCO2)CC1)OC 89385,CC1C(C=CC(=O)NCCOCCNC(C2(C(=O)N(C)C)CC2)=O)C1(Cl)Cl 89386,C1CCO1.C1(C(=O)OCC)(NCCOC)CC1 89387,CCC(CC)C(F)C(=O)NC(CCCC)CC(=O)NCC#Cc1cnn(C)c1 89388,C1(CN(C(=O)Cc2cn(C)nc2C(F)(F)F)C)CCN(C(=O)CCS(C)=O)CC1 89389,CCC(C)(CNC(=O)Cc1csc(Br)c1)NC(=O)C(C)CO 89390,c1(OC)ccc(CC(=O)NC2CCCC(CNC(=O)Cc3ccsn3)C2)c(F)c1 89391,c1(C(=O)NCC2CCCC(NC(c3cc(Cl)no3)=O)C2)cccc2c1CCCN2 89392,c1(OC)cc(F)c(-c2ncccc2C(=O)N(C)Cc2cccc(SC)c2)c(F)c1 89393,C1(CNC(CC(C)(C)O)=O)C2CCCCCC12.C12CCCCC1NC2=O 89394,C1(C)(Nc2ccc(CNC(CCC(=O)OC)=O)cc2)CCCS1(=O)=O 89395,C1(C(=O)Nc2cccc(NC(=O)C(F)Cc3ccccc3)c2)CCCCCCC1 89396,N1(C(C(COC)C)=O)CCC(C(=O)NCC2CC23CCOC3)CC1C 89397,N1(C(C2(CC)CC2)=O)CC(CNC(C2CC(=O)N2)=O)(OC)C1 89398,C=C1Cn2c(C(=O)N(CC(C)CNC(=O)CC3CCN(C)C3=O)C)nnc2S1 89399,c1(NC(c2csc(NS(=O)(=O)C(F)(F)F)n2)=O)ccc(Br)c2c1CNCC2 89400,c1(CCC)occc1C(=O)NC1CN(C(C2CC2n2cnc(C(=O)OC)n2)=O)C1 89401,c1(CC(=O)N(C2CCN(C(=O)C(O)CSC)CC2)CC)cn2ccsc2n1 89402,CN1CCOCC1C(N1CC(NC(c2ccnn2C)=O)C(C(F)(F)F)C1)=O 89403,C1(C(N2CC(NC(CCSCCC)=O)C(CC)C2)=O)COC2(CCC2)C1 89404,C1(NC(C(C)=C(CC)C)=O)CC(N=c2[nH]cnc3c(C(=O)OC)nsc23)C1 89405,c1(CC)c(N2CCN(C(C3CC3C(C)O)=O)CC2)nc(C)nc1Cl 89406,C1(C)(CNC(C(c2cccnc2)N(C2CC(NC(N)=O)C2)C)=O)C(C)(C)C1(C)C 89407,c1(C(=O)NCC2CC(c3ccccc3)CO2)ccc(Br)cc1 89408,N1(CCC(=O)NCCCN(C(c2cnc(C)o2)=O)C(C)C)CCCCC1=O 89409,C1(C(=O)NCC2(CNC(=O)C(F)OC(F)(F)F)CC2)CCC2(CC1)CC2(F)F 89410,C1(C(=O)NC2C(F)CCN(C(CC(C=C)(C)O)=O)C2)CN(CP(C)(C)=O)C1 89411,C(CC(C)CCNC(C1CCN(C(N)=O)CC1)=O)NC(C(N1CCOCC1)C)=O 89412,c1(OC)c(C(=O)NCCC(C)(C)NC(=O)Cn2cnnc2O)cc(Br)cc1F 89413,C1(C(=O)NC(CC=C)CO)CC(N=[N+]=[N-])CN1C(=O)C(O)CN(C)C 89414,C(=O)(C(CCSC)NC=O)NCCCCCN(C(CC)=O)C 89415,CCC(CC)CC(F)C(=O)NC(CNC(C1(C)CCOC1)=O)CCOC 89416,CN1CCCC1C=CC(N1CCOC(CCNC(=O)CSc2n[nH]c(=N)s2)C1)=O 89417,C1(C(=O)NCC2(NC(CCSC)=O)CCCCC2)CN2CCN1CC2C 89418,c1(Cn2c(C(CC(=O)OC)NCCNC(=O)OCC)nnn2)ccc(Br)cc1 89419,N1(C(c2c(OC)scc2)=O)CC2CN(C(C3CCN3C(C)C)=O)CC2(C)C1 89420,c1(C(=O)NC2CC(NC(c3nccc(Br)n3)=O)C2)cccc2c1OC(F)(F)O2 89421,N1(CC=C)CCN(C(=O)CC(CC2CC2)NC(=O)CC2C=NN(C)C2=O)CC1 89422,C1(NC(C(=O)Nc2cccc(C)c2)=O)COCCN(C(C2(C)CC2)=O)C1 89423,C1(N(C)C)CC2CCC(C1)N2C(c1ccncc1-c1ccc(F)cc1F)=O 89424,c1(C(C(=O)NCCCCCC)N(C)CC2(C#N)CC2)cc(C)nc(C)n1 89425,C(CS(=O)(=O)C(C)C)NC(N1C(c2onc(C)n2)CCCC1)=O 89426,Cc1c(CNC(=NCCC2COC3(O)CCOC23)NC2CCC2)c(Cl)nn1C 89427,c1(N2C(C)C(NC(c3ccc(CO)cn3)=O)CCC2)ncc(C#N)cc1Cl 89428,C(C)(CC(=O)NC1C2CC1N(C(c1ccc(CO)s1)=O)C2)(C(F)F)N(C)C 89429,c1(CC)ccc2cc(C(=O)NCC(C)CNC(C3(c4cc[nH]n4)CC3)=O)[nH]c2c1 89430,CC1(C)CN(C(=O)CSS(C)(=O)=O)C1C1CCN(C(C2CCCSC2)=O)CC1 89431,C1(C(=O)NCC(n2cc(C3CCOCC3)nn2)C)CC12CCC(C)(C)CC2 89432,c1(CC(=O)NC2CCCC2CNC(C2CCC3CC23)=O)ccccc1CC1CC1 89433,C#Cc1ccc(CCC(=O)NC2CC(NC(=O)C=Cc3ccc(C)cn3)C2)cc1 89434,C1(C(=O)NCC(C(C)C)NC(C2CCCCC2)=O)CCCCN1C 89435,CCCC(C)CCCC(=O)N(C1(C(=O)NC2(c3cc[nH]n3)CC2)CC1)C 89436,C1(CNC(CSCC#C)=O)Cc2ccccc2CN1C(c1cc(F)n(C)n1)=O 89437,c1(C(N2CC(CC=C)(NC(=O)Cc3ccsn3)C2)=O)c(C)cccc1[N+](=O)[O-] 89438,N1(C(C(C)SCC)=O)CC(NC(=O)CCCn2nc(C)cc2C)CC2(CC2)C1 89439,N1(C(C(C2CC2)OCC)=O)CCc2ccc(C(=O)N(C(CC)CO)C)nc2C1 89440,c1(NC(C(CC)(C)C#N)=O)ccc2c(c1)CN(C(=O)C(=O)Nc1ccccc1)C2 89441,N1(C(C(C(CC)C)NC(=O)C2=CCN(C)C2)=O)CC(F)(F)C(F)(F)C1 89442,Nc1cc(Cl)ccc1C(N1CC2CC(NC(c3ccc(F)s3)=O)C2C1)=O 89443,C1(NC(=O)C2=CCCCC2)CCCC12CN(C(c1ccn(CC(F)(F)F)n1)=O)C2 89444,C(=O)(C#CC(C)(C)CNC(=O)Cc1ccoc1)N1CCOCC(C(C)C)C1 89445,c1(C(=O)NCC2N(C(Cn3ncc(C)c3)=O)CCN(C)C2)cccc2c1CCC2 89446,c1(C(=O)NC2CC(NC(c3c(C)c(F)ccc3)=O)C2)cnc2[nH]c(=N)sc2c1 89447,C1(C)(C(=O)OCC)CCN(C(C(=O)NC2CC2)C(C)C2CCCOC2)C1 89448,CC1(CNC(c2ncoc2Br)=O)CCCN1C(C1CC(F)C(=O)N1)=O 89449,C1(C(=O)N(C(C)C(=O)NC(C)CN(C)C)C)(CC)CCNC1=O 89450,c1(CC)cccc(C(=O)NC2CCCC(CNC(C3CNC(=O)N3C)=O)C2)c1O 89451,c1cc(=NCCCSCCOCC2CCCO2)[nH]c(NC2CCCCCC2)n1 89452,c1(C(=O)O)cccc(CN2CCC(F)(C(N3CCS(=O)CC3)=O)CC2)c1F 89453,CN1CC(O)(CNC(C2CCC(CNC(c3cc(C(N)=O)[nH]n3)=O)O2)=O)C1 89454,CC1CCN(C(C2CCC(=O)N(C)C2)=O)CCN1C(c1csc(Cl)n1)=O 89455,N1(C(C(CC)N(C)C(c2cc(COC)[nH]n2)=O)=O)CCCC(COC)C1 89456,c1(C(N(CCCNC(C(CCOC)C)=O)C)=O)cnc2nc(O)nc(O)c2c1 89457,c1(C(=O)NC2C(OC)CN(C(c3occc3CN(C)C)=O)C2)cc(F)ccc1O 89458,C1(CNC(C2CCC(C)(C)C2)=O)CN(c2ncnc(O)c2Br)CCC12CCOC2 89459,N1(C(C2CC(SC)C2)=O)CCC(CC(=O)NC2CC(C#N)C2)CC1 89460,c1(C(N(CC(CNC(C2(CC)CC2(F)F)=O)O)C)=O)nn(C)c2c(=O)[nH]cnc12 89461,c1(C(N2CCC(NC(C3(O)CCC(CC)C3)=O)CC2)=O)cn2ccsc2n1 89462,c1(N2CCC(N(C(=O)CNC(=O)NC)CC)C2)nc(C#N)ncc1C 89463,C1(CNC(Cn2c(C)csc2=O)=O)CN(C)CCN1C(c1cccc(O)n1)=O 89464,c1(CC)ccc(N)c(C(N2C3CCC2C(NC(C2(C)CCCC2(F)F)=O)C3)=O)c1 89465,c1(C(C(=O)N(C(CNC(=O)C(=O)NCCNC(C)=O)C)C)C)cccnc1 89466,Cc1nn(C)c(N2CCNCC2)c1CN1CCCN(c2ccc(C(N)=O)s2)CC1 89467,N1(C(CN2CCCC(CC)C2)=O)CC2(CCCC2NC(C2C=C2C)=O)C1 89468,N1(C(C2C(C)C2)=O)CCC(OCCCNC(C2CC2c2ccoc2)=O)CC1 89469,C(CC(C(C)(C)C)NC1(c2n(CCCC)nnn2)CCC2(CC2)C1)SCC 89470,C1(C(=O)NC(c2ccnn2C)C(N2CC(OC(C)C)C2)=O)C=CC=CC=C1 89471,CCC(C)(C)OCC(=O)NCC1CC1NC(=O)C=C(C)C(F)F 89472,Cn1cc(-c2cccc(CC3CCN(n4cccn4)CC3)n2)c(C(F)(F)F)n1 89473,C1(C(=O)NCC2(C)CCC(NC(C3CN(C(N)=O)C3)=O)CC2)OCC2COCCC12 89474,N1(C(c2ccnc(C)c2N)=O)CC2CC(NC(=O)CCN3CCCCC3)C(C2)C1 89475,Cc1ccc(CNC(C)CCc2ccc(Br)cc2)c(Br)c1 89476,C12(C(=O)OCC(c3ccc([N+](=O)[O-])cc3)=O)CC=CCN1CCC2 89477,N1(C(CC)=O)CCCC(C(=O)NC2CCCC2NC(c2cc(C(N)=O)no2)=O)C1 89478,N1(C(c2c(C(C)CCO)noc2)=O)CC2CCC2(NC(=O)CC=CC(C)(C)C)C1 89479,C1(C(N(CC(CNC(COc2cccc(CC)c2)=O)C)C)=O)C(F)(F)C12CCC2 89480,C1(CNC(c2n(C)ncc2)=O)CC(F)CN1C(c1ccnnc1)=O 89481,c1(C(N2CCC(N(C)C(c3cc(-c4ccco4)[nH]n3)=O)C2)=O)cc(F)cc(F)c1 89482,C1(CNC(CCC=C)=O)CN(C(=O)C(C)CCO)CCC12CCOC2 89483,c1(OCCCCC2(n3cc(C(C(C)C)O)nn3)CCC2)cccc(C#N)c1 89484,O=C(CCCn1cncn1)NC1C=CCCC1.n12cc(nn1)C(=O)N1CC2C1 89485,N1(C(c2ccc(CCCC)cc2)=O)CCC(NC(C2COCC2(C)C)=O)C(O)C1 89486,C1(C(N(C2CCN(C(c3csc(O)n3)=O)C2)C)=O)CCS1(=O)=O 89487,C1(C(=O)NCCCN(C(CCC(CC)OC)=O)CCO)CCCC(C)(C)CC1 89488,N1(C(CC)CO)CC(=O)N(CC(N)CF)C1 89489,c1(C(=O)NCC(CC)N(C(=O)Cn2cnnc2O)C)cccc(C(C)(C)C)n1 89490,N1(C(C(F)OC)=O)CCOCC(CNC(c2cnoc2)=O)C1 89491,N1(C(C(=O)NCCC2CC(NC(C=C(CCC)C)=O)C2)=O)C(C)CCCC1C 89492,C(=O)(C(O)CC(C)C)NCC1(CNC(COC(CC)(C)C)=O)CC1 89493,Cc1cc(C(=O)NCC2CC(F)(CNC(=O)CC(C)F)C2)ns1 89494,C1(C)(C(=O)NCCCOC)CCCN(C(=O)Cn2nc(C)cc2C)C1 89495,C1(NC(CSCCC)=O)CC(N=c2[nH]cnc3cnccc23)C1 89496,c1(OC)ccc(F)cc1C(=O)NC1(CNC(C2CC23CCC3)=O)CCCC1 89497,C12(CN3CCC(c4cccc(Br)n4)C3)CCCCCC1NCC2 89498,Cc1cncc(C(=O)NC2CN(C(=O)CCC3CC3(C)C)CC23CC3)c1C 89499,C12(C(=O)NC(c3cc4ccccc4cn3)C)CCC(O1)c1ccccc12 89500,CCCC(O)CCN=c1nc(N2CCC(C(C)(C)C)C2)c2sccc2[nH]1 89501,Cc1cc(CC(=O)NC23CC(C2)N(C(=O)CC(C)n2cccn2)C3)cc(C)c1 89502,c1(OC)ncc(S(=O)(=O)NC(=O)COc2ccc(Oc3ccccc3F)cc2)s1 89503,c1(C(C(N2CC(N(C(CCS(C)=O)=O)C3CC3)C2)=O)O)cc(F)cc(F)c1 89504,C1(C(=O)O)CC(C(=O)NCc2ccccc2OC2CC2)C12CCCC2 89505,C(=O)(C1=CCSC1)NCc1c(C(=O)NCCC(CC)C)cco1 89506,C=CC(CC)CC(=O)NCC1CCN(C(=O)C(COC(C)(C)C)N(C)C)C1 89507,C(C)(C(O)C(F)F)NC(C(C)(C1CCC1)NC(C(CC)O)=O)=O 89508,C1(n2cc(C3CCOCC3)nn2)(C(N(CCC2CC2)CC)=O)CCOCC1 89509,C1(CNC(C2C(CC)C2)=O)CC(C)N(C(=O)C=Cc2cncs2)C1 89510,C(=O)(C(C)C(C)(C)O)NC1C(NC(c2c(C)[nH]c(C(C)(C)C)c2)=O)COC1 89511,N1(C(CCCCN(C)C)=O)CCC(NC(c2ccn(CC(F)(F)F)n2)=O)C(O)C1 89512,C(=O)(CCC(=O)N1CCCC1C1CCC1)Nc1nnc(CC(=O)OC)s1 89513,C#CC1(C(N2CCOC(COC)C2)=O)CN(C(=O)CC(F)(F)F)C1 89514,CC1(C(N2CCC(N3CCN(C(=O)Cc4ccsc4)CC3)C2)=O)CC2CCC1O2 89515,c1(C(C(=O)NCCSCC(=O)OC)NC(=O)CCOC2CC2)cnn(C)c1 89516,c1(-c2ccn(CC)n2)nnc(CN(C)C)n1-c1ccccc1C 89517,N1(C(c2c(C)cc(C)[nH]2)=O)CCC(NC(c2cnc(C(F)(F)F)nc2)=O)C12CC2 89518,N1(C(C2CC(C#N)C2)=O)CC(O)C(O)C1CNC(=O)CCc1cccc(Cl)c1Cl 89519,N1(C(C(CC2CCC2)NC(c2c(C)non2)=O)=O)CCC(O)C(C)(C)C1 89520,c1(C(=O)NCCC(C)NC(C=C(C)c2cccs2)=O)cnc(O)cc1C 89521,c1(C(=O)Nc2cc(OC)c(C)cc2C)c(Cl)nc2cc(Cl)ccn12 89522,O=NN1CCCCC1C(=O)NC(CO)C(C)NC(C1(c2ccccc2Cl)CC1)=O 89523,C1(CC(=O)NC2(C)CC(NC(C(C)Cn3ccnc3)=O)C2)CCC(C)(C)C1 89524,N1(C(c2c(CC)n(C)nn2)=O)CCC(C2CCCN(C(c3cc(Cl)ns3)=O)C2)C1 89525,O=[N+]([O-])c1ccc(CNc2ccccc2-c2ccccc2)cc1-c1nn[nH]n1 89526,N1(C(C(C)NC(CC)(C)C)=O)CCC(C(=O)NC(C)C2CC2)CC1 89527,C1(NC(=O)COC2COC2)CCC2CC1CN2C(C1CC1C(F)(F)F)=O 89528,c1(CN(C(=O)C(c2cccnc2)O)CCC)cc(Br)ccc1OC 89529,c1(C(=O)NCC(CO)NC(c2coc(C3CCC3)n2)=O)ccnc(C(F)(F)F)n1 89530,CCC(C)(C(=O)NCCC(N1CCCCC1)=O)C(F)F.C(CCNC(=O)CNC(N)=O)O 89531,C(=O)(CC(F)F)N(CC(C)N(C(=O)CNC(c1ccoc1)=O)C)C 89532,c1(CC)nc(C)cc(=NCCC2CCN(C(C3CCCCN3C(C)=O)=O)C2)[nH]1 89533,C(=O)(C1=CCN(C)C1)N1CCC(n2cc(C3(F)CC(SC)C3)nn2)C1 89534,Cc1cccn2cc(C(=O)NC3CCN(C(c4cncc(Br)c4)=O)CC3C)nc12 89535,Cc1ccc(C(F)(F)F)cc1C(N1CCC(C)(NC(c2ccccc2)=O)C1)=O 89536,c1(C(N2CCCCC(CNC(c3ccc[nH]3)=O)C2)=O)ccc2c(=O)ccoc2c1 89537,[N-]=[N+]=NCCCCC(=O)NC1(C(=O)NCC2CCCC2O)CCC1 89538,C#CC1(C(=O)NCC2CCCCCC2)CCN(C(=O)C(F)C(C)(F)F)C1 89539,C#CC1CN(C(C2(NC(C3CCC(C)O3)=O)CCCCC2)=O)CCN1C 89540,c1(OC)ccc(CC(C)C(=O)NC(C)CNC(c2cnc3n2CCC3)=O)cc1F 89541,c1(N2CCCC(C)(OC)C2)nc(=NC(Cc2cncs2)CCO)[nH]c2c1ncn2C 89542,N1(C(C23CC(C2)C3)=O)CCC12CN(Cc1cccc(C(F)(F)F)c1O)C2 89543,Cc1noc(C)c1C(C)(C)C(=O)N(CCCNC(=O)C(C)NC(C)(C)C)C 89544,C(C(=O)NN1CCCC1C(=O)N(C)Cc1cnnn1C)OCC=C 89545,C1(NC(=O)Nc2c(OCC)cc(F)cc2)CCCC2OCCC12 89546,C1(NC(C(C)(C)C2CC2)=O)C=CCN(C(C2CCN(C3CCCCC3=O)C2)=O)C1 89547,C#Cc1ccc(C(=O)NC(Cc2cn[nH]c2)C(=O)NCCCN2CCOC2=O)o1 89548,CN1CCOC(N(C(C(=O)NCCCF)C(C2CC2)C2CC2)C)C1 89549,CC#CCC(C)N=c1[nH]c(=N)[nH]c(=NCC(c2cccs2)N(C)C)[nH]1 89550,c1(C(N2CC(CCNC(C3CCC3CF)=O)(OC)C2)=O)ccc(Cl)c(O)c1 89551,c1(CN=C(NCCOC)NCC2SCCc3ccccc32)ccc(S(N)(=O)=O)c(Cl)c1 89552,C1(CCC(=O)NCC(C)(C)F)CCN(C(c2cc(Cl)ncn2)=O)CC1 89553,CC1Cc2ncccc2CN1S(=O)(=O)c1cc(C(=O)N(C)C)co1 89554,c1(OCCC)ccc(OCC(N2CC(N(C(=O)C(C)(CO)OC)C)C2)=O)cc1 89555,Cc1ccc(SCC(=O)NCC2CCCN2C(c2nccnc2Cl)=O)cc1 89556,C(=O)(C(C)(C)CCCN=[N+]=[N-])N1CC2(CN(C(C3(F)C(C)(C)C3(C)C)=O)C2)C1 89557,CC1(C)COCCC1C(N1CCOCC1)=O.N12CCCC(C1)C2=O 89558,c1(C(=O)NC2C(CNC(Cc3cc(C)sc3C)=O)C2)c[nH]c2ccccc2c1=N 89559,c1(C(C(C)C)NC(CCn2cc(CCCOCC)nn2)=O)c(F)cccc1F 89560,C1(C(N2CCCC(F)(CNC(C3(O)CC3)=O)C2)=O)Cc2cncn2C(=O)N1 89561,c1(OC)cc(C(=O)NCC(Cc2ccc(F)cc2F)C(N)=O)ccc1Br 89562,CCCCC(C)CCC(=O)N(CCCN(C(=O)CCc1c(F)cccc1F)C)C 89563,c1(C(N2CC(SC)C(NC(c3csc(Cl)c3)=O)C2)=O)ccc2cc[nH]c2c1 89564,Cc1coc(OCCOCCNC=O)c1-c1ccccc1.C(=O)(CN(C)C1CC1)N 89565,Cn1c(CNC(C2CCC(CNC(c3ncccn3)=O)C2)=O)nnc1O 89566,Cc1c(C(C(=O)NC2CCCC2)N(c2nc[nH]n2)CCC#N)cnn1CC(F)F 89567,C1(C2CCCN(C(=O)CCN(c3ccccc3)C)C2)(NC(C(COC)C)=O)CC1 89568,n1(C(C)C)cnnc1CC(=O)NC1(C(=O)O)CC1 89569,N1(c2nnc(CC)s2)CCC(NC(=O)C(C)OCC(C)C)CC(C)(C)C1 89570,N1(C(C(C)=C(C)C)=O)CCN(C(=O)C=CC2CCCN2C)C2CCCC12 89571,N1(C(c2nncc(OC)c2)=O)C2CCC(C(=O)NOCC(N)=O)C1CC2 89572,c1(OC)noc(C)c1C(=O)NC(CNC(=O)C(C)(C)COCC(F)F)C1CCC1 89573,c1(CC)cc(C(N2CCC(C(C)C(=O)NC(CCOC)C(C)C)C2)=O)ncn1 89574,N1(CC)CCOCC1C(=O)NCc1cccc(CN2CCOCC2)c1 89575,N1(CC(=O)NCCN(C(c2snc(O)c2Cl)=O)CC)CCC(CO)CC1 89576,N1(Cc2cccc(C)n2)CCCC2CN(Cc3cccnc3)CCC12 89577,C1(C(CNC(c2cnc(O)o2)=O)F)CCN(C(=O)C(c2cccnc2)O)CC1 89578,Cc1ccc2[nH]nc(C(=O)NC(CNC(C3CCC4CC3CO4)=O)C3CC3)c2c1 89579,CC1=C(c2ccccc2)CN(C(c2cccc(F)c2)C(=O)NCC2CC2)CC1 89580,N1(C(C2(CC)CCCCO2)=O)CC(NC(=O)CCC2(C)COC2)C2(CC2)C1 89581,N1(C(C(CC)COC)=O)CCC2(CC1)CCN(C(C1(C)COC(=O)C1)=O)C2 89582,c1(CNC(=O)NCC(C2CCCN(CC)C2)(C)C)ccc(F)c(C)c1F 89583,C12(C(N3CC(C=C)OCC3)=O)CCCC1CCN2C(c1cn(C2CC2)cn1)=O 89584,Cc1nc(O)nc(O)c1CCC(N1CCC2(C1)CN(C(=O)CCCCO)C2)=O 89585,C1(NC(C2(C=C)CCC2)=O)CC2CC(NC(C3(C(C)(F)F)CC3)=O)CC12 89586,c1(NC(c2ccnc(C)n2)C)ncc(Cl)cc1C(N)=O 89587,Cc1ccc(CC(C)C(=O)NC(C)CCCCNC(c2cncn2C)=O)cc1 89588,N1(C(c2cc(Br)ccn2)=O)CCC2(CC2C(N2CCOCC23CC3)=O)C1 89589,C(=O)(CC(O)C(C)C)NC(COCC)C(=O)NCCc1[nH]cnc1C 89590,C(=O)(C(F)(F)CF)NCCOC1CN(C(C(C)N(CC)CC)=O)C1 89591,c1(C(=O)NC2CCC(NC(c3cn(CC)nc3C)=O)CC2)ccnc(C)c1Cl 89592,C(=O)(C1=C(C)OCCC1)NC(C(=O)NCc1cccc(OC)n1)(C)C1CCC1 89593,Cc1ccc(Br)cc1C(N1CCCC(C)(C)C1)=O.C12CCCN1C(=O)C21CC1 89594,C(=O)(CCC(F)(F)C(F)F)N(C)CC1CCN(C(=O)CC2CCC2C2CC2)CC1 89595,CCCCC(CCCC)C(=O)N(C(C)CN(C(=O)CN1CC(C)C1)C)C 89596,CN1CCN(C(C2CC3(CCO2)CC3)=O)C(C(N2CCCC(C#N)C2)=O)C1 89597,C(=O)(C(C)(C)C(O)CC)NCC(CNC(c1cc(C(=O)OC)on1)=O)OC 89598,CCCC(C(=O)NCCN(C1CCCC1)C(c1ccsc1)=O)OC 89599,Cc1cnc2cc(C(N3CCN(C(C4CC=CC4)=O)C(CO)C3)=O)ccn12 89600,C#Cc1ccc(Br)c(C(=O)NC(C)CN(C)C(C2(C)C=CCCC2)=O)c1 89601,C1(CC)CN(C(=O)CCc2cnoc2)CCN1C(=O)C=CC1CCCO1 89602,c1(C(N2CCC(NC(C(C)C)=O)CC2)=O)c(F)c(F)c(F)c(F)c1F 89603,N1(C(C(C)CN(C)C)=O)CCN(C(C2(CC3CC3)CC2)=O)CCC1C 89604,c1(C(N2CC(CCO)(NC(Cn3cnc(=N)[nH]3)=O)C2)=O)ccc(N(C)C)c(F)c1 89605,N1(C(C=O)NCCN(OC)CC)CCC(NC(=O)OC)C1.CC(C)C 89606,c1(C(N2CCN(C(CC=C)=O)CC2CC2CC2)=O)cc2ccc(F)cc2cn1 89607,CCC(CC)(CCNC(c1ccon1)=O)NC(=O)C(Cc1ccccc1)N(C)C 89608,C1(NC(CC(C)c2ccccc2)=O)CN(C(c2ccc(O)nc2Cl)=O)CC12CC2 89609,c1(OC)ccc(Cc2ccc(CC(N3CC4(CC4C(N)=O)C3)=O)s2)cc1OC 89610,C12(CC(F)(F)C1)NC(=O)C1C(=C)C1C(=O)NC2.c1(CN(C)C)c(C)cnn1C 89611,CC(C(=O)N1CC(C(=O)NCC2C(C)C2C)C(F)(F)C1)C(C)(C)C 89612,N1(C(C(C)ONC(=O)OC(C)(C)C)=O)CCC2CC12CNC(c1cn[nH]c1)=O 89613,c1(OC)cccc(CCCCCNC(C2(c3ccc(Br)cc3)CCCC2)=O)c1 89614,C1(c2cccc(C)c2)CCCN1NC(=O)c1cnn(C2CCC2)c1C 89615,C(=O)(C(C)(C)c1cccs1)N(CCOCCNC(CSCC)=O)C 89616,C1(C(=O)NCC(CCNC(=O)Cc2cn[nH]c2)O)CC12C1CC3CC(C1)CC2C3 89617,C1(COC)CN(C(c2cc(O)ncn2)=O)CCN1C(=O)C(C)n1cccn1 89618,CCC(COC)C(=O)N1CCCC(NC(=O)C(=Cc2cn[nH]c2)C)C1 89619,C1(NC(c2cncc(COC)c2)=O)CN(C(=O)CN2CCCC2=O)CCC1(C)C 89620,C(=O)(C(O)CCC(C)C)N1CCN(CC(C)NC(C2(C#C)CC(=O)C2)=O)CC1 89621,c1(CC(=O)NCC(C)CCc2nn[nH]n2)cccc(-c2nnco2)c1 89622,c1(C(=O)NC(CC(=O)NCC2CC2(F)F)C2CC2)ccccc1O 89623,c1(N2CC(CNC(C3(C)CCNC3=O)=O)OCC2)cncc(C#N)n1 89624,c1(C(N(C)CCOCCCN(C)C(C2CCCC2O)=O)=O)cc2ccccn2c1 89625,C1(CCC(N)=O)CCCCN1C(C1CCN(C(=O)C=C(C2CC2)C2CC2)CC1)=O 89626,N1(C(c2ccn(C(F)F)n2)=O)CCOC(C2CC2)C1 89627,c1(C(=O)NC2C(NC(c3ccc(CCC)s3)=O)CC2)cccc(C)c1F 89628,N1(C(c2cnn(CC)c2C)=O)CCCC(NC(=O)C(C)(C)n2cccn2)C(F)C1 89629,c1(C(N2CCC(NC(c3c(C)ncnc3)=O)C2)=O)ccc(N)cc1C(C)(C)C 89630,N1(C(C(CNC(c2cc(OC)n[nH]2)=O)N(C)C)=O)CCCC12CCNC2=O 89631,N1(C(C2CSCCN2C(c2cccs2)=O)=O)CCc2ncncc2C1 89632,C(CN=c1cccc(S(=O)(=O)NCC2CCC3(CCC3)C2O)[nH]1)c1n(CC)cnn1 89633,Cc1c(C(=O)NCC(C)CN(C(=O)CC2CCC2)C)c(-c2ccccc2)cn1C 89634,c1(C(=O)NC2COCC2CNC(=O)C(O)C(F)(F)F)cc(O)cc(Br)c1 89635,N1(CC=C)C(=O)NC(CSc2ccccc2)C(C(=O)OCC2CC2)=C1C1CC1C 89636,C1(CN(C)C(C2CC(C(F)(F)F)C2)=O)CCCN(C(C2C3CC(=O)CC23)=O)C1 89637,C(=O)(C1CCCn2cncc21)NC(CC=C)CNC(c1c(Cl)ccc(C)c1N)=O 89638,C#CCC(C)(CC)C(=O)N1CC(CNC(=O)CCc2ccc(F)cc2)C(C)(C)C1 89639,C1(CC(=O)NCC2CN(C(C(N(C)C)C3CC3)=O)C2)Cc2ccc(Br)cc2C1 89640,N1(C(C2OCCN(C(CCCOC)=O)C2)=O)CCC(C2CCC2)C1 89641,Cc1c(CNC(N2CC(N3CCOCC3)CC2C)=O)cnn1CC(F)(F)F.C=O 89642,C(C(C)N=c1ccc(C(F)(F)F)n[nH]1)NC(c1c(C)nc(CO)nc1)=O 89643,N1(C(c2n(C)ncc2C#N)=O)CCC2(CCCN2C(=O)CCS(N)(=O)=O)C1 89644,C(CN=c1[nH]c(C(F)(F)F)cs1)(c1ccccc1OC(C)C)OC 89645,O=C1CC(CC(=O)NCC2CC(O)(CNC(c3cccc(Cl)c3)=O)C2)C(=O)N1 89646,C1(CNC(c2c(C)cc(C)o2)=O)CN(C(=O)CNC(=O)CC(C)C)CCC1(F)F 89647,N1(C(C2CC23CC(O)C3)C(=O)NCCC)CCCC2(CCCNC2=O)C1 89648,c1(CNCC(C)CF)ccc2nonc2c1 89649,c1(C(N(C2CCN(C(C3CC(O)C3)=O)C2)CC)=O)cnn(CC2CCCCC2)c1 89650,c1(C(=O)NC2C=CC(CNC(C=CCCC)=O)C2)c(C)cc(O)nc1C 89651,CC(O)(C(=O)NCC1CC2CN(C(=O)CCCc3ncco3)CC12)C(F)(F)F 89652,C1(C#N)(C(=O)NC2C(C)N(C(c3cccnc3OC(F)F)=O)CC2)CC12CCC2 89653,Cc1nnn(CC(=O)NCCCN(C(=O)C(C2CCOCC2)O)C2CC2)n1 89654,c1(C(N(C)CC2CN(C(C3COC(=O)N3)=O)CCO2)=O)ccc2[nH]ccc2n1 89655,c1(NC(N2CCC(=CC(=O)NC3CN(C)C3)CC2)=O)cccc(Cl)c1F 89656,C#Cc1ccccc1CC(=O)NCC1CC(CNC(C2C=CC=CC=C2)=O)CO1 89657,C(=O)(C1CCCc2sccc21)NC1CCC(CNC(c2ccc(N)c(F)n2)=O)C1 89658,n1(C(C(=O)NC2CCCN(C(C)=O)C2)C)cc2ccccc2n1 89659,N1(C(=O)OC(C)(C)C)CCCCC(NC(=O)NC(CO)C2CC2)C1 89660,C1(C(C)NC(C(F)=CC)=O)CCCN(C(C2CN(CC(F)(F)F)C2)=O)C1 89661,C(=O)(C1=CCC(F)(F)CC1)NC1CC(CCNC(=O)OC(C)(C)C)C1.C(CO)O 89662,c1(C(N2CCCC2CN(C(C23C=CC(CC2)C3)=O)C2CC2)=O)cccc(O)c1F 89663,c1(C(N(CCNC(C2(CCOC)CCCC2)=O)C)=O)ccc(-n2ccnc2)cn1 89664,C1(C)(C(=O)NCCN(C(C(C)Cc2cccnc2)=O)CC(C)O)CCCN(C)C1 89665,N1(Cc2cccc(OC(C)=O)c2)CCC2CN(S(=O)(=O)C(Cl)(Cl)Cl)CC2C1 89666,c1(NC(C2C=CCN(C(CCC3CC(C)C3)=O)C2)=O)cn(C)nc1C#N 89667,C(C)(CNC(=O)CC1CCSCC1)(CO)NC(C(C)=CC)=O 89668,C#Cc1cccc(C(N2CCC(O)(C(C)NC(=O)CCC3CCCOC3)C2)=O)c1 89669,Cn1cnnc1CC(N1CC(CO)(NC(c2ccc(C3CCOC3)s2)=O)C1)=O 89670,c1(C(N2CC3(C2)CN(C(=O)C(F)CC2CC2)C3)=O)cccc2nc(O)oc12 89671,C(=O)(C1CCCc2nccn21)NC1CC(OC)CN(C(=O)C(C)NS(C)(=O)=O)C1 89672,N1(C(=O)CN2C(=O)CCC2=O)CC(C2CN(C(C3CCc4n[nH]cc4C3)=O)C2)C1 89673,N1(C(CS(=O)(=O)NCC)=O)CCCC2(CNC(=O)CN3CC(C)C3)CCCC12 89674,C1(CC2NC(=O)N(Cc3c(C)ncs3)C2=O)CC2(CCCC2)CO1 89675,c1(CC)cnccc1C(=O)NCC(N1CCCCC1CSC)=O.N12CC(C1)C2=O 89676,C(=O)(N=c1ccnc(N(C)C)[nH]1)C1CCN(Cc2n(C)cnc2)C1 89677,C1(C(N2C(C(=O)NCC3(O)CC3)(CC)CCC2)=O)C2CCC(C2)C1C 89678,CC(Cn1ccnc1)C(=O)N(CCC(N1CC(C#N)(N(C)C)C1)=O)CCCO 89679,C=CC1(C(=O)NCC2CCOCC2)CCN(C(c2cc(C)c[nH]2)=O)C1 89680,Nc1cc(C(N2CCCC2CNC(C2CCCC23CC3)=O)=O)cnc1Cl 89681,Cc1cnn(C)c1CC(=O)NC(CC(F)(F)F)c1ccccc1 89682,c1(C(c2nnnn2Cc2cccs2)NCCC=C=C)ccnc(OC)c1 89683,CCCC(C(=O)NC12CC(NC(c3cnn(CC(C)C)c3)=O)(C1)C2)N(C)C 89684,N1(C(CC2C(C)OCC2)=O)CCC(NC(=O)Cn2cncn2)C(C)(C)C1 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89720,C1(CC=C)(NC(c2sccc2OC)=O)CCCN(C(=O)C(C#N)CCC)C1 89721,Cc1cc(Br)ccc1CCC(N1CCOC(CNC(=O)C2=C(Cl)CC2)C1)=O 89722,C(=O)(CCCC(=O)N(CC(C)NC(c1ccc(OC)c(Br)n1)=O)C)OC 89723,C1(CCNC(C(CC)n2cncn2)=O)CCCN(C(c2oncc2C)=O)C1 89724,c1(OC)ccc2[nH]nc(C(N3CCC34CCC4)C(=O)NC3(C)CC3)c2c1 89725,C(=O)(C1=C(Cl)CCOC1)N1CCC(N(C(=O)Cn2nc(O)ccc2=O)CCO)C1 89726,c1(CC(=O)NC(CN2CCC(CC)CC2)(C)C)c(OC)ccc(Br)c1F 89727,C1(C(N(C)CCNC(=O)C2=CCC2)=O)CC(C)(C)CCO1 89728,C12(CNC(c3cncc(C)n3)=O)CCC1CN(C(=O)CC1CNC(=O)C1)C2 89729,c1(C(N(C2CCC2)CC#C)=O)ccoc1CNC(=O)C(CC1CCC1)OC 89730,CCC(C(=O)NC1CN(C(c2nccn2C)=O)CCC1C)C(C)C 89731,C(C(N=[N+]=[N-])C(=O)NC1CC(C)N(C(=O)C(C)C2CCCO2)C1)OCC 89732,O(NC(=O)C(C)NC(=O)CCSc1ccccn1)CC(C)O 89733,c1(OC)cccc(O)c1C(=O)NC(C)CNC(=O)COCCSc1ccccc1 89734,N1(C(c2c(Br)ccc(N)c2)=O)CCC(NC(C2CCC2)=O)C2(CCC2)C1 89735,N1(C(c2c(CC)scc2)=O)CCC(CNC(=O)C=Cc2cccc(O)c2)C(C)C1 89736,CC1(CCNC(=O)Nc2cccc(I)c2)CC(F)(F)C1 89737,CS(=O)(=O)c1cc([N+](=O)[O-])ccc1NCC(c1ccc(F)c(F)c1)O 89738,N1(C(CC2CCCC(=O)N2)=O)CC2CCC(C1)N2C(C1C(Cl)(Cl)C12CC2)=O 89739,CC1=C(C(=O)NCC2COCC2NC(=O)CCCNC(N)=O)CCO1 89740,CC(C)(C)CCC(=O)N1CC(C)(C)CC1CNC(=O)Cn1ccc(C2CC2)n1 89741,N1(C(Cc2cccc(C(N)=O)c2)=O)CC2CC1CN2C(=O)CC1CCCO1 89742,N1(C(c2ccc(OC)s2)=O)Cc2ccccc2C(NC(c2ccc(Cl)cc2)=O)C1 89743,N1(C(C2CC3(C2)OCCO3)C(=O)NC(COC)C2CC2)CCc2c(C)cccc21 89744,N1(C(CC2CCCN(C(C(C(=O)OC)(C)F)=O)CC2)=O)CCC(C)C(C)(C)C1 89745,c1(OC)ncc(S(=O)(=O)N2CCCC(C(=O)N(CCC#N)C(C)C)C2)cn1 89746,CN1CCC(NC(=O)COC2CN(C(c3ccc(O)cn3)=O)C2)C1(C)C 89747,c1(C(=O)NC2CC(F)(CNC(CC3(C)CC3F)=O)C2)ncn2ccccc12 89748,N1(C(c2cn(C)c(O)n2)=O)CC2(CCC(NC(=O)CN3C(=O)CCC3=O)CC2)C1 89749,N1(C(CN(CCOC)C)=O)CC(C)(C(N2CC(F)(F)CCC2C)=O)CC1(C)C 89750,Cc1cncc(C(N2CC(C(C)NC(=O)C(C3CC3)C3CC3)C2)=O)n1 89751,CC1CC2(CO1)CN(C(c1cncc(CNC(=O)Cc3cnsc3)c1)=O)C2 89752,CCC(CC)=CC(=O)NC1(CNC(C)=O)COC1 89753,C#CC1CCCC(NC(C2CC2C(C)NC(c2cnn(C3CC3)c2)=O)=O)C1 89754,C(=O)(C(C)S(N)(=O)=O)NC1(CNC(c2cnc(OC)s2)=O)CCOC1 89755,C(CCC(C)(C)C(=O)NNc1c(C)cccc1[N+](=O)[O-])OC(CC)C 89756,C1(C(=O)NC2CCC(CCNC(c3cc(Cl)cs3)=O)C2)C2CCC3C(C2)CC13 89757,Cc1nc(Cl)ncc1CN(CCC(N1CCCCCC1)=O)C 89758,C1(COC)CC2(CCN2C(C2CSCCN2C(c2cn(C)nn2)=O)=O)C1 89759,c1(C(=O)NC2CCN(C(C3CCC(=C)CC3)=O)C(C)C2)cnc2ccccc2c1 89760,c1(CNC(C(C2(C)CC2)NC(CCn2ncc(C)c2)=O)=O)cc(C)ccc1O 89761,C1(NC(c2cc(C(=O)OC)sc2)=O)CCCCC1NC(c1n[nH]cc1F)=O 89762,c1(C(=O)NCCCCNC(C2(C3CC3)CCC2)=O)cnc2cc[nH]c2c1 89763,c1(C(CC)C)nc(N2CCC(NC(=O)COC(C)CC)C(C)C2)cc(C)n1 89764,Cc1nscc1CC(N1CC(NC(c2cn(C3CCOCC3)cn2)=O)C1)=O 89765,C=CC(C)(C)CC(=O)N1CCOCC1CCNC(C1CCCCN1CC(F)F)=O 89766,c1(CC)nc(=N)[nH]cc1C(=O)NC1CC(CCNC(C2CC(C)(O)C2)=O)C1 89767,c1(C(=O)NC2CN(C(Cc3c(C)ncs3)=O)C(C)C2)cc(N)ccc1C(F)(F)F 89768,C1(CC)C(C(=O)NCc2ccsc2C)CCN1C(=O)Cc1cc[nH]c1 89769,c1(OCCC(=O)NC2CC(C)N(C(=O)CC3CC3)C2)ccc(Cl)cc1Br 89770,c1(C(C)(C)C)ccc(C(N2CCCC2CNC(C2C3(CC3)C23CC3)=O)=O)cn1 89771,c1(CN2C3C(C(=O)Nc4ccc(F)nc4)C(C3)C2)cccc2nc[nH]c12 89772,CC1(CO)CCN(C(=O)CCC2CC(NC(=O)Cc3ccon3)C2)CC1O 89773,C(=O)(CCCC(C)C)N1C(CCC2C(SC)CCN2C(=O)C#CC(C)C)CCC1 89774,c1(C(N(CCC(C)NC(=O)CCS(C)(=O)=O)C)=O)cc2ncccc2cc1Cl 89775,CC1CN(C(=O)Cc2cnns2)CC(C)C1NC(=O)CCc1ccncc1 89776,c1(C(=O)NCC(C)N(C(C(C(C)C)NC(=O)OC)=O)C)cc(Cl)cc(Cl)c1 89777,c1(CNC(CNC(C2C(C)C2)=O)=O)cnn(C)c1C(=O)NCCc1cscn1 89778,C#CCC(O)C(=O)NC1CCC1NC(c1cnn(C)c1-n1cccc1)=O 89779,C1(CNC(C(C)OCC)=O)CN(C)CCN1C(=O)Cn1cnc(=O)cc1C 89780,Cc1ncc2n1CCC(C(=O)NCC1CCCN(S(C)(=O)=O)C1)C2 89781,Cn1ncc(C(N2CCC(C(F)C(N)=O)CC2)C(=O)NCCCC2CC2)c1Br 89782,C1(C(N(CC(F)F)CCC)=O)CCCC2(CCC2)O1 89783,N12CCC3CC(C3C1)C2=O.N1(C(=O)CSC2CC2)C2CCC1CC2 89784,C1(C(=O)NCC2CCC(NC(c3c(C)nns3)=O)C2)CC(c2ccncc2)=NO1 89785,c1(C(=O)NC2C3CN(C(C(CCCC)C)=O)C2CC3)cc(Cl)c2c(c1)OCCO2 89786,c1(OC)ncc(CNC2(c3nnnn3CCSC)CCOCC2)cc1Br 89787,C1(C(CN(CCCCNC(=O)C(=O)Nc2ccccc2)C)=O)CC1C1CCCC1 89788,Cc1cc(C(=O)NCc2c[nH]nc2C(=O)NCC(N2CCCCC2)C)nc(C)c1 89789,C(=O)(CC(C)CC(C)C)NC(CCC)CC(=O)NCC1(OC)CCCC1 89790,c1(CCC(=O)NCC(CC)NC(C2CC(OC(C)(C)C)C2)=O)cccnc1 89791,CC1CC(NC(=O)CC2CSCCS2)CN(C(=O)CCN(C2CCCCC2)C)C1 89792,c1(OC)ccc(F)c(C(N2CC(c3cn(CC(=O)NCCC#N)nn3)C2)=O)c1F 89793,C#CC1(C(=O)NCCCn2nccn2)CN(C(c2coc(SC)c2)=O)C1 89794,c1(C(N(CCNC(CCC2C(C)C2)=O)C)=O)ccc(N2CCCC2)cc1 89795,C1(N(C(=O)Cn2ccnn2)CCOC)CCN(C(=O)C(F)C2CCCC2)CC1 89796,C1(C)(C(=O)NC(CC(C)NC(C(c2ccc(C)cc2)=O)=O)C)CCCS1(=O)=O 89797,C(=O)(CC(C)(C)CNC(=O)CCc1ccco1)NCC(CC(C)C)O 89798,c1(-c2onc(C3(Cc4cccc(Br)c4)CCCC3)n2)c(Cl)ccc2c[nH]nc12 89799,c1(C(N(C2CCN(C(=O)C3=CCN(C(C)=O)C3)C2)CC=C)=O)cc2n(n1)CCO2 89800,C1(C(=O)NCCN(C(CC(C)C2CCCO2)=O)C)(CF)CCC(F)(F)CC1 89801,c1(CC)nc(C)c(C(=O)NC(CCN(C)C)C(=O)NC(C)CCF)o1 89802,c1(C(=O)NC2CCN(C(CCc3ncc(C)[nH]3)=O)C2)cn2ccn(C)c(=O)c2n1 89803,N1(C(CNC(N)=O)=O)CCCC2CCN(C(c3cn4c(n3)CCC4)=O)CC12 89804,C1(CC(=O)OC)CCCC2(CN(C(c3c[nH]c(-c4ccc(Cl)cc4)c3)=O)C2)O1 89805,Cc1cc(F)c2cc(C(=O)NCCN(C(=O)CC3CC=CC3)C)[nH]c2c1 89806,C(CN=c1cc[nH]c(C(N)=O)n1)(c1ccc(F)cc1)NC(C)=O 89807,c1(N2CC(CC)OCCC2)ccc(Br)c(S(=O)(=O)NCC(C)(C)C2CCCO2)n1 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89825,C1(O)(CC#C)CC(C(=O)NC(C2CCN(C(c3occc3C(F)(F)F)=O)C2)C)C1 89826,C1(CC)CC(C)CN(C(C23CC(CN2C(=O)C2=CCSC2)C3)=O)C1 89827,c1(C(N2CCC(NC(C(C(=O)OCC)(C)F)=O)CC2)=O)c(C)cc(Br)cc1F 89828,N1(C(C(C)OCCN(C)C)=O)CCC(CN(C(=O)Cn2cc(C3CC3)cn2)C)C1 89829,Cc1nc(C(=O)NC2CN(C(=O)CCc3ccoc3)CCC2C)c2ccccn12 89830,CCCCCCC(C)CC(=O)NCCN(C(C1CCC2CC2CC1)=O)CC1CC1 89831,C(C(F)(F)C(F)(F)F)NC(=O)CCNC(=O)C(O)c1ccco1 89832,C=CCC(CC)C(=O)NC1(C)CCN(C(c2c(C)cccc2O)=O)C1 89833,c1(C(=O)NCCC2OCCN(C(C=Cc3occ(C)n3)=O)C2)cccc(C)c1N 89834,C1(C(=O)NC(CNC(c2nc(O)c(C)s2)=O)CO)(COC)CCCCO1 89835,C1(C(=O)NC2C(NC(C(C)(C)OC)=O)CCCC2)CC2C=CC1CCC2 89836,Cc1cccn2cc(CC(=O)NCC3CCCCN3Cc3ccccc3F)nc12 89837,c1(C(=O)NC(C(C)NC(c2c(C)nccn2)=O)C)ncc([N+](=O)[O-])cc1Br 89838,C(=O)(CC(CC)C(=O)OC)NC(CNC(CCCC#CC)=O)C(C)C(C)C 89839,N1(C(C(C)(Cl)Cl)=O)CC2(C)CN(C(=O)C(O)C3CCCC3)CC2(C)C1 89840,O=C(CN1CC(O)CO1)NCCN(C1CC1)Cc1ccccc1Cl 89841,n1(CC)cc(CN(C(=O)C(CC2CCC2)NC(C2CCO2)=O)C)cn1 89842,c1(NC(=O)NC(c2ccccn2)C2CCCC2)ccc(Br)c(F)n1 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89860,Cn1ccc2sc(C(=O)NC3CC(NC(=O)OC(C)(C)C)C3(C)C)cc12 89861,N1(C(c2ncccc2C(F)(F)F)C)CC2(CCN2CC2(C)CCCC2)C1 89862,CCCCCCC(C)(CC)C(=O)NCC1CN(C(c2sccc2Cl)=O)CC1(C)C 89863,Cc1nc(CO)sc1C(=O)NC1COCC1CNC(C1CC(=O)N(C)C1)=O 89864,C1(NC(CC2(C=C)CCCCC2)=O)COC2(C1)CN(C(C1CCCC1(F)F)=O)C2 89865,N1(C(C2CCC(C)O2)=O)CCCC2CN(C(=O)CCc3ccn(C)c3)CCC12 89866,c1(N2CC(C(C)C)NC(=O)C2)nc2c(c(=NCc3ncc(Br)cn3)[nH]1)CCC2 89867,C(=O)(C1=CCCN(C(c2cncc(Br)c2)=O)C1)Nc1nc(OC)c(Br)cc1 89868,C1(CC(=O)NC2(C(=O)OCC)CCC2)CCN(C(c2ccsc2)=O)C1 89869,N1(C(C2(CC(=O)OC)CC2)=O)CCC(O)(C(C)NC(=O)C(C2CCCCC2)F)C1 89870,c1(CC)nc(C#N)cc(=NCC2C(C)CCCN2C(c2cnnc(O)c2)=O)[nH]1 89871,C1(C(=O)NC(C2(N(C)C)COC2)C)CCCC(F)(F)C1.C12CCC(CC1)C(=O)N2 89872,N1(C(C2(SC)CC2)=O)CC(NC(=O)C(CC)c2ccccc2)CC2(CC2)C1 89873,N1(C(C(=O)NC)C)CC(O)(C(C)NC(c2cn(CCC(C)C)nn2)=O)C1 89874,n1(CC)ccc(C(N2CCC(NC(=O)C(CC3CCCC3)OC)C2C)=O)c1C 89875,Cc1cc(C(C)C(N2CCC(Cn3cc(CCCC(C)O)nn3)C2)=O)c(C)o1 89876,CCCCC(CCCC)C(=O)NC1(C)CC(NC(=O)CSc2cccc[n+]2[O-])C1 89877,c1(OC)c(F)ccc(C)c1CNC(=O)NCc1ccc(Br)cc1OCCN(C)C 89878,C12(CCNC(CCC=C)=O)CCC1CN(C(c1csc(O)n1)=O)C2 89879,CCCCCCCC(=O)NC1CC(NC(=O)C(C)(C)C2CCCO2)CC1O 89880,CC1CC(=O)NC1C(=O)NCCCNC(C1CCC(C)CC1)=O 89881,CC(C)C(O)C(C)C(=O)N1CCC(NC(=O)CCC2CCC2)CC1 89882,N1(C(c2c[nH]nc2C(F)F)=O)CCC2(CCCN(C(=O)C3=CSCS3)C2)CC1 89883,C1(C)(CNC(C2(CCN(C)C)CC2)=O)CN(C(=O)CC2CCCO2)CCO1 89884,c1(CC(N2C(CNC(Cc3c(C)n[nH]c3C)=O)COCC2)=O)ccc(C#N)cc1 89885,CN1CC=C(CC(=O)N2CC3(CCC3NC(c3csc(Cl)c3)=O)C2)CC1 89886,N1(S(CC(C)C)(=O)=O)CC2CCC1C1CN(C(c3cncs3)=O)CC21 89887,N1(C(CCC#C)=O)CCC2(CCCCC2NC(=O)C2=C(Cl)CCC2)C1 89888,n1(CC)cc(C(=O)NCC2CC(COC)CN2C(=O)Cc2cnc(C)o2)c(C)n1 89889,C1(NC(c2c(OC)n[nH]c2)=O)CC2CN(C(=O)CC34CC(C3)C4)CCN2C1=O 89890,C(C(=O)N(C)CC1CCCN(C(c2csc(COC)n2)=O)C1)(C(C)C)SCC 89891,N1(C(CCC2CCN(C)CC2)=O)CCC(NC(C2CC3CC3C2)=O)C(C(N)=O)C1 89892,C1(CC)(CC)CC(NC(=O)C(C)C(C)C)CN1C(c1cnc(OC(C)C)nc1)=O 89893,C=CC1(CC(=O)NC(C)(CNC(=O)Cc2cncs2)C2CC2)CC1 89894,N#CC1(C(N2CCN(C(c3ccc(F)s3)=O)C(CC(F)(F)F)C2)=O)CCOCC1 89895,c1(C(=O)NC(CNC(C(CC)(C)CO)=O)CO)ccc2c(c1)OCO2 89896,N1(C(C(C)NC(CC)=O)=O)CC(CNC(=O)CC(O)C(C)C)OC(C)(C)C1 89897,c1(SCC(=O)NC(CNC(C2CC3C=CC2O3)=O)CO)ccc2ccccc2c1 89898,Cc1cccc(Cl)c1C(N1CCC(C(=O)O)C(C(=O)C(C)C)C1)=O 89899,C1(CNC(C(=O)NCC=C(C)C)=O)CC(CNC)CO1 89900,c1(CC)ccc(C(=O)NC(CNC(=O)CCc2cnn(C)c2)CC)cc1Cl 89901,c1(C(=O)NCC(C)C2CCC2)cnccc1-n1cccn1 89902,c1(C(=O)NCC2OCCN(C(C(C)C(F)(F)F)=O)C2)noc2ccccc12 89903,N1(C(c2c(CC)c[nH]c2)=O)CC2CCCCC2(CNC(=O)CSCC(F)(F)F)C1 89904,C1(NC(c2csc(-c3cn[nH]c3)n2)=O)CN(C(c2cc(Cl)no2)=O)C2(CCC2)C1 89905,CC1CCc2onc(C(N3CC(O)C(O)C3CNC(=O)CSC(F)(F)F)=O)c2C1 89906,N1(C(C2C(OC)(OC)CC2)=O)CC(NC(=O)Cn2nnc(C3CC3)n2)C2(CC2)C1 89907,C1(NC(Cn2cc(COCCC(N)=O)nn2)=O)CCn2c(O)nnc2C1 89908,C1(NC(Cc2n(C)ccn2)=O)CCN(C(C2OCC2(C)C)=O)C12CCC2 89909,CC(F)(F)CC(=O)NCc1ccoc1C(=O)NCc1nc(C(N)=O)no1 89910,C1(NC(C(C2CN(C(=O)C(C)Cc3ccoc3)C2)OC)=O)CCC(CO)C1 89911,c1(NC(C2CCN(C(C(C)(CO)CO)=O)C2)=O)c(Br)cc(OCF)cc1[N+](=O)[O-] 89912,C1(CC(=O)NC2CCOCC2NC(C2(c3cc[nH]n3)CCC2)=O)CCC(=O)NC1 89913,C#CCC(C)(CC)C(=O)NC1CCN(C(c2ccc(O)c(C)c2C)=O)CC(O)C1 89914,N1(C(CCOCC(C)C)=O)CCCC(C2(NC(C3CCNC3=O)=O)CC2)C1 89915,S(=O)(=O)(c1ccc(=NCC2COCCCO2)[nH]c1)N1CC(N(C)C)C(O)C1 89916,c1(C(N2CCC(N(C(CC=C=C)=O)CC3CC3)CC2)=O)cc(C)ncc1C 89917,c1(C(=O)NCC2N(C(CSCCC)=O)CC(F)C2)c(C)cc(OC)cc1F 89918,N1(C(C(c2ccccc2)OC)=O)CC(NC(c2cc(C)cc(C)c2)=O)CC(F)C1 89919,CCC(C(=O)N1CCOCC(C(=O)NCC2CCOC2(C)C)C1)C(F)(F)F 89920,c1(OCCC(=O)NCCCC2CCCN2CC2CCCC2)ccccc1Cl 89921,N1(C(c2c(C)nc(CO)s2)=O)CCC2CN(C(=O)Cn3cc(CO)nn3)CCC12 89922,CC1Cn2nc(C(=O)N(CCCNC(C3CCCC(=O)O3)=O)C)cc2C(=O)N1 89923,c1(C(=O)NCC(C)NC(=O)CNC(=O)C2CC2)cccc(-c2ccccc2)c1O 89924,N1(C(C(C)CC#N)=O)C2CCC1CC(n1ccnn1)C2.N12CCCC(C)(C1)C2=O 89925,N1(C(C(C)n2ccnn2)=O)C2CCC(C2)C1C(=O)NCC1(F)CCOCC1 89926,C(C(C(=O)NCCC#N)N1CCCC(c2ncc(C)s2)C1)(C1CC1)OC 89927,N1(C(CCCC)=O)CCN(C(=O)C(C)N(C(C2(c3ccccc3)CC2)=O)CC)CC1 89928,N1(C(c2cccc(-n3cncn3)c2)=O)CCC(F)C(NCC2CCOC2)C1 89929,C1(N(C(C=CC(CC)C)=O)C)CCCN(C(c2cc(C(N)=O)no2)=O)CC1 89930,N1(C(Cc2nc(C)[nH]n2)=O)CCC(C)(NC(=O)Cc2nc(C3CC3)no2)C1 89931,C1(NC(c2c(C)nsc2N)=O)CC2(C1)CN(C(=O)COc1cccc(Cl)c1)C2 89932,c1(C(N2CCC(C)(NC(C3CCC(CC)C3)=O)CC2)=O)[nH]nc2c1CCC2(C)C 89933,C1(C(=O)NC2(c3cnc(CCC(=O)OCC)o3)CC2)Cc2ccccc2N1 89934,c1(CN2CC(C#N)N(C(c3ccccc3S)=O)CC2)ccc(F)c2ccoc12 89935,C(=O)(C(O)CCCNC(=O)CC1C(=O)NN=C1C)N1CCN(CC#CC)CC1 89936,Cc1cscc1C(=O)NCCC1CCCN1C(c1sccc1F)=O 89937,C1(NC(CC(C)c2ccccc2)=O)CN(C(=O)CSc2nncs2)CC1C 89938,N1(C(CSCCC)=O)CCN(C(=O)C(O)CC(N)=O)C(C(C)(C)C)C1 89939,c1(C(N2C(C(N(C3CCC3)C)=O)CSC2)=O)cc(C#N)cs1 89940,c1(CCC(n2c(C)cc(C)n2)C)ccc(=NCCCN(C)C)[nH]c1 89941,c1(CNC(C(N2CCC(OCCC)CC2)=O)=O)cc(C)c2ncn(C)c2n1 89942,CN1CCN(C(=O)Cc2cncnc2)C(CNC(=O)CC2CCC3CC3C2)C1 89943,Cc1cn2cc(C(=O)NCCOCCNC(c3ccn4ccnc4c3)=O)nc2s1 89944,N1(C(C(c2cccc(OC)c2)(C)C)=O)CC2(CC(NC(=O)CCC(C)OC)C2)C1 89945,c1(C(=O)OC)nc(OC)cnc1C.C12C3CC1CN(C3)C2=O 89946,N1(C(c2c(C)noc2)=O)CCCC(CCC(N2CC=CC2C(N)=O)=O)C1 89947,c1(OC)nn(C)cc1C(=O)NCC1(NC(=O)C=CS(C)=O)CCOC1 89948,Cc1c(CC(N2CCOCC(C)C2)=O)sc2ccccc12 89949,C1(C)(CNC(C2CC(NC(C(C3CCOCC3)OCC)=O)C2)=O)CCCCCC1 89950,C(=O)(CC(C)CNC(C1CCS(=O)CC1)=O)N(C(C#C)C1CCC1)C 89951,c1(C(=O)NCC2CCCN2C(c2cccc(Cl)c2O)=O)c(F)cccc1[N+](=O)[O-] 89952,Cc1ccc(C(=O)NCC(C)(C)C(=O)NCc2nn(C)cc2CO)n1C 89953,N1(S(CC)(=O)=O)CCCC(C(N2CC3CC3(NC(=O)CCCCC3CC3)C2)=O)C1 89954,c1(C(N2CC3C(NC(C4OCC(C)C4)=O)C(CC3)C2)=O)csc2c(Cl)cccc12 89955,c1(NC(=O)Cc2cccc(F)c2O)ccc(-c2ccc(Cl)cc2C(=O)O)cc1F 89956,C(=O)(C1=NOC(C)(C)C1)N1C(C(N(C)C)=O)CC(O)C1 89957,C1(C(=O)NCC2C3CCC(C3)N2C(=O)CCC=CBr)CCc2n[nH]cc2C1 89958,N1(C(CC2C3CN(C(c4c(COC)cc[nH]4)=O)CC32)=O)CC=CC12CCOCC2 89959,C#CC1CCCCN1C(C1(C(C)NC(=O)C(=O)CC(C)C)CC1)=O 89960,c1(C(=O)NCCC2(C)CCN(C(COCCC=C)=O)C2)cccc2c1OC(C)C2 89961,C(=O)(C#CC(C)(C)O)N1C(C(=O)NCc2ccncc2F)CC(OC)C1 89962,N1(C2C(C(=O)OCC)C2)C(C(=O)NCc2cc(COCC)no2)CC2CC12 89963,c1(C(=O)NC(C2CC=CCC2)C(N2CCC(=C)C2)=O)cnc(O)cc1C 89964,c1(CC)nc(C)c(CC(=O)NC(C)(C)CCNC(=O)Cc2csc(C)c2)c(C)n1 89965,C1(NC(CCS(C)=O)=O)CCSC12CN(C(=O)CNC(c1cccnc1)=O)C2 89966,N1(C(CCc2cccc(C)c2)=O)CCCC(C(=O)NCC2CSCCO2)CC1 89967,C=CCCC(C(=O)NCC1(C2CC2)CCC1)NC(=O)CC1COC(=O)C1 89968,c1(C(=O)NCC23CC(NC(C(COC)C)=O)(C2)C3)cccc(Cl)c1 89969,C1(CNC(N(c2c(C)ccc(F)c2)C)=O)CCC2(CCCOC2)O1 89970,c1(C(=O)NCCC(C)(C)NC(C2CC2(Cl)Cl)=O)cnc2occc2c1 89971,N1(C(C(C(C)(C)C)OC)=O)CCC(C(=O)NCC(CC(C)C)N(C)C)C12CCC2 89972,C(C)(C(C)(C)C(=O)N(C)Cc1cnn(C)c1C)NC(C1N(CC)CC1)=O 89973,Cc1cc(NC(=O)NC2CCCC2c2cnn(C)c2)ccc1NC(=O)CCF 89974,N1(C(C2=C(C)CCC2)=O)CCC2CCC(NC(C3CC4(C3)CS(=O)(=O)C4)=O)C1C2 89975,CC(CCN=c1cc[nH]cc1S(=O)(=O)NCc1cc(Cl)ccc1OC)P(C)(C)=O 89976,C1(CNC(C#CC(C)C)=O)CCCC12CCN(C(=O)CC1OCCC1C)CC2 89977,C1(NC(C2(SC)CC(O)C2)=O)CN(C(c2ccc(F)cc2)=O)C2(CCC2)C1 89978,N1(C(C(CC)C)=O)CC(CO)C2(C1)CN(C(=O)C(c1cccc(Cl)c1F)(C)C)C2 89979,c1(C(N2C3CN(c4c(Br)ccc(C#N)c4)CC23)=O)cc2ccccc2cc1O 89980,CC(C)C(C(C)NC(=O)CCc1cc[nH]n1)NC(=O)Cc1ccc(O)cc1 89981,C1(C(N(CCC)C(C)C)=O)CN(C(=O)C(C)NC(C)(C)CC)CCO1 89982,CCC(C(=O)N(C(C)CCNC(c1ccc(S(N)(=O)=O)o1)=O)C)C(F)(F)F 89983,CN1CCC(O)C(NC(C2CC(NC(c3cnn4c3CCC4)=O)C2)=O)C1 89984,c1(C(N(CCCNC(C(C)c2cncs2)=O)CCO)=O)cc([N+](=O)[O-])ccn1 89985,C1(NC(=O)OC(C)(C)C)CC2(C1)CC(N=c1ccc([N+](=O)[O-])c(O)[nH]1)C2 89986,CN1CC(C(=O)NC(C)(C)COCCCNC(=O)Cc2cscn2)CCC1=O 89987,C1(C)(C(N2CCC(n3cc(CCC(=O)OC)nn3)C2)=O)CC2CCC1C2 89988,c1(-c2scc(Nc3nc(C)cc(OC)n3)n2)cc(F)c(Cl)cc1Cl 89989,N1(C(Cc2ccnc(OC)n2)=O)CCN(Cc2ccccc2)C(CCO)C1 89990,C1(NC(C(C=C)(F)F)=O)CN(C(c2cc3c(s2)CCC3)=O)CCC1C 89991,C1(NC(=O)COCC2CCOC2)COCCN(C(=O)CCOC2COC2)C1 89992,C1(CC(C)(C)C)CCCCN1S(=O)(=O)CCCO 89993,c1(C(=O)NC2COCC2NC(C2CC3CCC2C3)=O)cc2c(F)ccc(F)c2[nH]1 89994,CC1(C)CN(C(C2(Cl)CC2)=O)C1C1CCN(C(C2CCS(=O)(=O)N2)=O)CC1 89995,c1(C(N2CC(F)(CNC(C(Br)=C(C)C)=O)C2)=O)ccnnc1O 89996,S(=O)(=O)(c1cc2c(Br)cncc2s1)NC(C1(C)CCN1)C 89997,CC(C)(CS(C)(=O)=O)C(=O)NCC(C)(C)CNC(c1cnc(N)c([N+](=O)[O-])c1)=O 89998,Cc1nc(C(=O)NCC(=O)Nc2ccccc2Cl)c(C)n1C 89999,Cc1cccc(C(O)C(c2ccccc2)NCc2cc(C#N)no2)c1 90000,Cc1cc(=NCCC(C)(O)C2CCC2)[nH]c(=NCc2c[nH]nc2C)[nH]1 90001,c1(N(CC(=O)NOC2CCOC2)C(C2CCC2)=O)cccc(S)c1.C(CCO)N 90002,c1(OC)ccc(-c2ccccc2)cc1CN(CC(O)C1CCC1)C 90003,C=CCC(CC(F)F)NC(=O)COC1CCN(C(=O)C(C2(O)CCCC2)F)C1 90004,Cc1ccn2ncc(C(=O)NC(C)CNC(=O)C(O)CC(N)=O)c2c1 90005,C(=O)(CCC(CF)CF)N1C(C(=O)NC2C(C)C2(C)C)CC1 90006,c1(CC)nc(Cl)[nH]c(=NC2CC(NC(=O)C(c3ccc(C)s3)C)C2)c1Cl 90007,C(C(CC(=O)NCCNC(N)=O)C1CCC1)NC(C(CC)N(C)C)=O 90008,C12(n3cc(C4(C)COC4)nn3)CCC(C(=O)NC3(c4ccc(F)cc4)CC3)(CC1)C2 90009,C1(N(C(=O)Cc2ccn(C)n2)C)CN2CCC1CC2 90010,Cc1cc(C(=O)N(C2CCN(C(c3ccc(C#N)cc3)=O)C2)CCO)ccc1Br 90011,C1(NC(C2(CNC(c3cc(CCC)on3)=O)CCC2)=O)CCCCC1C(N)=O 90012,N1(C(C2N(C(COc3ccn(C)n3)=O)CC=C2)=O)CCn2nncc2C1 90013,N1(C(CCCCNC(C)=O)=O)CCCCC(C(N2CCCC(O)C2C)=O)C1 90014,c1(C(=O)Nc2c(C)cc(C)c(O)c2)cc2n(n1)CCCN(C(=O)C(C)O)C2 90015,CCC(C)C(C)C(=O)NCC1(F)CC(CNC(=O)CCc2ncc(F)cn2)C1 90016,CC(C)CC(O)C(=O)NCCC1CN(C(=O)CCCn2ccccc2=O)C1 90017,C(=O)(CC(C(F)(F)F)NC(c1ccccc1F)=O)NC(C)Cn1cncn1 90018,N1(C(c2c(CC)ocn2)=O)CCC(F)(F)C(CNC(c2ccc(Cl)s2)=O)C1 90019,N1(C(CCOCCOC(C)(C)C)=O)CC=CC(NC(C2CCCN2C=O)=O)C1 90020,C1(C(N2CC(CNC(CC3(OCC)CCCC3)=O)C2)=O)CCCS(=O)(=O)C1 90021,c1(C(N2C(CNC(C3C4CC5C(C4=O)C35)=O)CC2)=O)ccc2c(c1)CCOC2 90022,C(=O)(C(C)(C)CCCN(C)C)NCC(C)(C)OCC(NOCCCOC)=O 90023,c1(C(=O)NCC(C(C)(C)C)CO)cnc2cnc(Cl)cc2c1 90024,CC1(C)CN(C(=O)Cn2cccnc2=O)CC1NC(c1c[nH]cc(F)c1=O)=O 90025,c1(C(N(C(C)CN(C)C)CC)=O)cccc(-c2n[nH]c(C)n2)c1 90026,c1(N2C(CNC(CS(CCOC)(=O)=O)=O)CCC2)cc2c(cn1)C(=O)CCC2 90027,N1(C(CNC(C)=O)=O)CC(c2ccccc2)(N)C1.C1(C=O)CC1Br 90028,c1(C(=O)NCC(C)N(C(=O)CCn2cnnn2)CC)ccc(Br)cn1 90029,N1(C(c2[nH]nc(OC)c2Cl)=O)CCCN(C(=O)C(c2ccc(C)cc2)C)C(C)C1 90030,CCC(C)(CCNC(=O)Cc1ccccc1F)NC(=O)CC1CCCCO1 90031,Cc1ncc(CC(=O)N(C2CC(NC(C3CNC(=O)C3)=O)C2)C)c(O)n1 90032,C(=O)(C1=CCCC(C)(C)C1)NC(C1CCCN(C(c2ccc(SC)cc2)=O)C1)C 90033,N1(C(CCCC(=O)OC)=O)CC2CN(C(C3CCC(C)CC3)=O)CC2(C)C1 90034,c1(C(N)=O)cccc(N(C(C2CN3CCC23)=O)Cc2ccccc2)n1 90035,c1(C(N(CC(C)O)CCNC(c2ccc(C3CC3)nn2)=O)=O)cc(Cl)nnc1O 90036,C1(NC(CCNC(C)=O)=O)CCN(C(=O)CCS(C)=O)C1C 90037,c1(OCCC)cccc(-c2cccc(NC(C3(C)CC3)=O)c2)c1 90038,CC(C)(C(=O)NC1CCC(CNC(C2(CO)CCCO2)=O)C1)S(C)(=O)=O 90039,c1(C(C(=O)N(CCC)CCNC(=O)Cc2ccno2)N(C)C)ccccc1 90040,CC1(C(=O)NC2CC(CNC(=O)Cn3nnc(-c4ccccc4)n3)C2)CC(F)C1 90041,C1(N(C(CCC=C(C)C)=O)C)CN(C(=O)C=CC(=O)NC2CC2)CCC1O 90042,N1(C(CCCOCC)=O)CC2CC(NC(c3cc(C(F)F)ncn3)=O)CC2C1 90043,N=c1nc(C(N2CCCC(CC(=O)NCc3nc(=O)o[nH]3)C2)=O)cc[nH]1 90044,C1(C2CCCN(C(=O)C3=CCC(C)CC3)C2)(NC(c2c(CC)cccc2)=O)CC1 90045,c1(C(=O)NCC2OCCN(C(CC3(C=C)CCC3)=O)C2)cc(C#N)c(O)nc1N 90046,Cc1cccc(NC(C2CCC(NC(c3cc(Cl)c(Br)s3)=O)CC2)=O)n1 90047,N1(C(C2(CC)CC(C)(C)C2)=O)CC(C)OC2(CCN(C(=O)CSC(C)C)CC2)C1 90048,C(=O)(C1=NOC(C)C1C)NCC1(CN(C(c2c(C)ccnn2)=O)C)CC1 90049,N1(C(=O)Cc2nc(Cl)cs2)CCN(C(c2ncncc2Cl)=O)CC(O)C1 90050,N1(c2n(CCC#C)c(N3CC4CC3CC4O)nn2)CCc2ccccc2CC1 90051,C(=O)(C(CC(C)C)NC(c1ncn(C(C)C)n1)=O)Nc1c(C)nsc1 90052,C(C(C(=O)NCCC(C)CO)C(C)(C)C)NC(C(CC)(C)CC)=O 90053,C1(NC(C(C=C)CC)=O)CC2CCC(C1F)N2C(c1ccccc1F)=O 90054,c1(C(N(CC(C)NC(=O)C=Cc2ccoc2)CC)=O)cnc2[nH]ncc2c1 90055,C1(NC(C=CC(C)NC(C2CC(F)(CCCO)C2)=O)=O)COCC1F 90056,N1(C(C2C(CC)OCC2)=O)CC2CCC(C1)N2C(C1CCC(C)(C)O1)=O 90057,C1(CNc2c(OC(CC)C)cccn2)CCCC2(CC(C(=O)O)C2)O1 90058,C1(C(=O)OC(C(N2CC(NC(=O)OC(C)(C)C)C2)=O)=O)CCCCC1 90059,C(=O)(C1Cc2ccccc21)NC(CNC(c1c(NC)cccc1C)=O)(C)CO 90060,CCC(C)CCC(=O)N1CCOC(CNC(c2ncoc2C(F)(F)F)=O)C1 90061,Cc1nn(C(C)C)c(C)c1C(C)NCCC(C)(O)c1ccccc1 90062,C(CC1CCCC1)(C(=O)NCC(CO)NC(C1CCCSC1)=O)OC 90063,c1(C(=O)NCCCC(C)NC(CCC=C=C)=O)cc2c(nc1O)CCCC2 90064,C1(CC(=O)NC2(C)CN(C(C(C)Cn3ccnc3)=O)C2)CCCC1(F)F 90065,Cc1cncc(C=CC(=O)NCC(C2CC2)NC(=O)CC2CCCC(C)O2)c1 90066,c1(C(=O)NC(C2CCC(NCC3CCCCO3)CC2)=O)cccc(F)c1I 90067,Cc1cc(C(=O)NCC(C)(C2CC2)NC(=O)CNC=O)cc(C)c1N 90068,N1(C(c2c(OC)c[nH]n2)=O)CC2CC(O)C1C2NC(c1ccc2nnnn2c1)=O 90069,c1(N2CCC=C(C)C2)[nH]c(=NCCc2cccs2)nc2c1ncn2C(C)C 90070,C1(CNC(c2n(C(CC)C)ncc2)=O)CN(C(c2snnc2C)=O)CCCO1 90071,N1(C(C(C)NS(CCC)(=O)=O)=O)CCN(C(=O)CCCCC2CC2)C(CCO)C1 90072,N1(C(CCC2(C)CCCN2C(C2CCOC(=O)CC2)=O)=O)CCC2(CCC(O)C2)C1 90073,N1(C(CC=CC=C)=O)CCC(C)(C)C(CNC(C2CCOC(CC)C2)=O)C1 90074,N1(C(C(COC)O)=O)CCC(C2CCN(C(=O)C(C)(C)C(C)(F)F)C2)CC1 90075,CCCC(C)(C)CC(=O)N1CCC1CNC(=O)CCc1cn(C)nc1C 90076,c1(C(N2CC(C)CC(NC(CCCC=C)=O)C2)=O)c(C)[nH]c2ccc(Cl)cc12 90077,C1(C(=O)NC2(C3N(C(C(C(CC)C)C)=O)CCC3)CC2)CN2CCN1CC2C 90078,c1(C(=O)NCC(CCOC)NC(C2(C#N)CC2)=O)ccc(C(F)F)c(OC)c1 90079,c1(C(N(C)CCNC(=O)CCC2CCCOC2)=O)cccc(S(N)(=O)=O)c1 90080,C(c1cccnc1)=CC(=O)N(C1CCN(C(=O)CCC(F)F)CC1)CC#C 90081,c1(NCC(C(C)C)(C)NC(=O)Cn2cc(CO)nn2)ncc2c(n1)COC2 90082,C1(C(=O)NCC(CNC(=O)C(C)CN(C)C)OC)CC2CC1CC2(F)F 90083,c1(C(=O)NCCC(CCNC(C(C)N(C)C)=O)C)cnn2c1S(=O)(=O)NCC2 90084,c1(C(=O)NC2(CCNC(C(C)(C(C)C)OC)=O)CCC2)cc(F)cc(N)c1F 90085,C1(C(=O)NC(CC#C)(C)C)CCC2(CC2)N1C(C1CC(=O)CS1)=O 90086,c1(OCC)ccc([N+](=O)[O-])nc1N1CCC(O)C12CCCC2 90087,C1(N(CCC(=O)N(C)C)C(CN(CCC#C)C)=O)CC2CC2C1 90088,c1(OCC#C)ncccc1C(=O)N(CCNC(C1CC1Cl)=O)Cc1ccccc1 90089,CCC(C#N)(CC)C(=O)NC(C)CCNC(C1CC2(C1)CC1(CC1)C2)=O 90090,C1(F)(C(=O)OC)CCC(Nc2cc(-c3ccc(Cl)cc3)no2)C1 90091,C=CCC(CC(C)C)C(=O)NCC1CCCC1NC(C1(C(=O)NC)CCCC1)=O 90092,C=CC(C)(C)CCCNC(=O)C(CC1CCOCC1)NC(=O)C(F)CC 90093,C12(C(N3CC(NC(C4CC5(CCC5)C4)=O)C3)=O)CC3CC(CC1C3)C2 90094,c1(C(N2C(CNC(CN=S(C)(C)=O)=O)CC2)=O)cc(Cl)ccc1[N+](=O)[O-] 90095,C#CC1CC2(CC2)CN1C(c1cc(CCN(C(=O)C(Cl)Cl)CC)on1)=O 90096,C1(NC(CCCCC(CO)NC(=O)OC(C)(C)C)=O)CS(=O)(=O)CC12CC2 90097,c1(SC)cc(Cl)nnc1Cl.C12(CC1)C(=O)N(C)CC(C)NC2=O 90098,c1(CC=C(C)C)ccccc1C(N1CC=CC(NC(=O)CC2CCCCC2)C1)=O 90099,N1(C(C2CCC(=C)CC2)=O)CC2CCOCC2(NC(=O)CCC(C)C)C1 90100,C1(N(C(C2CN(C(C)C)C2)=O)C)CN(C(=O)CC=CC(C)(C)C)CC12CC2 90101,C=CC(CCC)CC(=O)NCC=CCC(=O)N(CC(C)C#N)C1CC1 90102,c1(C(N2CC(C=C)(CC(=O)N(C3COC(C)(C)C3)C)C2)=O)nccc(C)c1N 90103,c1(CN(C(c2ccc(-c3cccnc3)cc2)C(=O)NCC)C)ccc(Br)cc1F 90104,N1(C(c2n(CCC)ccc2)=O)CC(NC(c2cc(OC)ccc2F)=O)C(C)(C)C1 90105,c1(NC(=O)NC2CC(OC)C23CCC3)ccc(C)c(NCCSC)c1 90106,C=C(C)CCC(=O)N1CC(=C(F)CNC(=O)CCn2cc(C)cn2)C1 90107,c1(OCC)cc(NC2CCN(C(=O)CC3CC(C)(C)CO3)CC2)ncn1 90108,CC(C(=O)N1CCC(C(C)(O)CNC(=O)C#CC2CCC2)CC1)C(C)(F)F 90109,c1(OCC(N2CCC(Oc3ccc(C)cc3)C2)=O)c(F)cc(I)cc1F 90110,c1(NC(C2N(Cc3ccc(C)[nH]3)CCCC2)=O)nc(Cl)c(C)cc1[N+](=O)[O-] 90111,C1(NC(C2(N(C)C)CC2)=O)CCC2(CC1)CN(C(c1cc(=O)cc(Cl)[nH]1)=O)C2 90112,CCCCC(C)C(=O)NC1CCCCCC1C(N1CC[Si](C)(C)CC1)=O 90113,N1(C(CCC#C)=O)CCCCC(C(=O)NC2CC23CCCCC3)C1 90114,S(=O)(=O)(c1cccc2ccccc12)N1CCOCC(NC(C(C=C)O)=O)C1 90115,C(CCC(CCC)NC(c1oc(C(F)F)cc1C)=O)NC(CC(=C)C)=O 90116,N1(C(C(C)SC)=O)CC2(CCCCN2C(c2cnc3c(c2)CCCC3)=O)C1 90117,N1(C(C2(CC#C)CCN(C(=O)C(=O)NC)C2)=O)CCCC(CC)(CC)CC1 90118,N1(C(c2ncc(Cl)cc2F)C(=O)NC(C)(C)C)CCC12CCOCC2 90119,c1(C(=O)NCCC(C)OC)ccc(CNC(C2CCCCC2O)=O)cn1 90120,c1(C(=O)NC2C(CNC(c3ccc(C#N)s3)=O)C2)cnc2ccc(F)cn12 90121,C1(N(C)C(C2CC(F)(CF)C2)=O)CCCN(C(=O)COCCCF)C1 90122,c1(C(C(=O)NC(c2cnn(C)c2)C)O)ccc([N+](=O)[O-])cc1 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90266,N1(C(C2(C#N)CCCC2)=O)CC(C2CN(C(C34CC(CO3)C4)=O)C2)C1 90267,c1(C(=O)NCC2(NC(C(CCSC)O)=O)CC2)c(C)ncnc1C 90268,N1(C(C(C)OCC)=O)CCOCC1CC(=O)NCc1conc1C 90269,c1(-c2nc(C(CC)C)nn2C2CC(OC(C)(C)C)C2)ccn2c1CSCC2 90270,C1(C(=O)NCC(c2cn(C)cn2)O)(NC(C(C)c2cc[nH]n2)=O)CC1(C)C 90271,C1(C)(COC)CC(NC(c2c(Cl)cccc2Cl)=O)CN1C(=O)CCC(C)C 90272,C1(OC)CC(CNC(=O)Cc2cncs2)(NC(=O)CC23CC(C2)C3)C1 90273,n1(CC(N2CC(CCNC(C3CC3C3CCCO3)=O)(OC)C2)=O)nc(C)oc1=O 90274,C1(C(=O)NC2(C)CCN(C(=O)C=CBr)C2)CC2CC(O)CC(C1)C2 90275,CON(CCC(=O)N1CCN2C(=O)OCC2C1)C(=O)c1ccc(C)c(C)c1 90276,N1(C(C)=O)CCN(C(=O)CC2CCCN2Cc2nccc(C)n2)CC1 90277,N1(C(CC=C)=O)CCC(CNC(=O)CCc2cnn(C)c2)CC1C 90278,C1(C(N2CCCC(F)C2)=O)CCC2(CN(Cc3ccc(F)c(F)c3Cl)C2)O1 90279,c1(C(N(C(C)(C)CCC(=O)N2CC3CCC3(C)C2)C)=O)ccc(C#N)cn1 90280,C=C1CCN(C(c2cc3n(n2)CCO3)=O)C(C(=O)NC2CN3CCC2CC3)C1 90281,c1(SC)cc(C(N2CC(NC(=O)Cc3cc[nH]c3)C(C)C2)=O)ccc1[N+](=O)[O-] 90282,c1(CCOCCO)ccc(SC2CCN(CCCF)C2)cc1 90283,CC1OC(=O)NC1C(=O)NC(C)(C)C=CC(=O)N(CCC(C)(C)C)C 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90422,c1(C(=O)NCC2C(C)CN(C(=O)CCCSC(C)(C)C)C2)cccc2c1CCC2 90423,c1(C(N2CC(N3CCN(C(C(CSC)(C)C)=O)CC3)C2)=O)cc(N)cc(N)c1 90424,N1(C(CC=CCC)=O)CCCCC1CN(C)C(c1cc(C(=O)OC)nn1C)=O 90425,c1(C(=O)NCCc2ccc(COC)cc2)cnc(C)c(C#N)c1 90426,Cc1cc(CC(N2CC(C)(NC(=O)C(C)Nc3ccccn3)C2)=O)ccc1O 90427,C1(C(N2CC(CCC)C(NC(=O)C(c3ccccc3)C)C2)=O)CC(C(C)C)=NO1 90428,C#CCCCC(C)C(=O)NCCn1ccc(C(=O)N(C2CCN(CC)CC2)C)c1 90429,CC1CN(C(c2cnc3[nH]nnc3c2)=O)CC(C)CN1C(=O)C1=CSCCO1 90430,N1(C(c2c(C)c[nH]n2)=O)CCOCC1CNC(c1csc(C(F)F)c1)=O 90431,c1(CNC(C(Cn2cncn2)NC(C(C)N2CCCC2)=O)=O)nccc(O)n1 90432,c1(CC)nc(C)oc1C(=O)NCCC(C)N(C(=O)CSc1ccccc1F)C 90433,c1(CCC(=O)NC(CNC(C(CCC)C#N)=O)C)ccc2c(c1)OC(F)(F)O2 90434,c1(C(=O)NC2CCC(NC(CC=CCC)=O)CC2)cnc2c(c1)CCOC2 90435,CC(CCNC(C1(C)CCN(C(c2c[nH]c3nccc-3c2)=O)C1)=O)CC(C)(C)C 90436,N1(C(C2(C(C)(F)F)CC2)=O)CCCC1CNC(=O)CCC1CCOC1 90437,c1(C(=O)OCCc2cc(OC)ncc2)ccc(C2CC2)c(Cl)c1 90438,C(C(CC(=O)NCC(C)(C)NC(=O)Cc1cc(F)ccc1Cl)C(F)(F)F)N(C)C 90439,C(=O)(C(F)(F)CCn1cc(C(CC)OCC)nn1)NCc1nnc(CC)s1 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90510,c1(C(N2CCCC(N(C(=O)CS(C)(=O)=O)CC)C2)=O)cc(CC(C)C)nc(O)c1 90511,c1(C(N(CC(N2CC(=C)C2)=O)CC#C)=O)cc(F)ccc1C 90512,N1(C(C(C(COC)C)C)=O)CC(CO)C2(C1)CN(C(c1cccc(C)n1)=O)C2 90513,C(=O)(CCCN=[N+]=[N-])NC1(CNC(C2C(C)C2C)=O)CCCC1 90514,c1(CC)[nH]nc(Cl)c1C(=O)NCC(C)(C)NC(C1CN(C)CCO1)=O 90515,c1(CC)cc(C(N2CC=CC(C(=O)NC3(C)CC(F)(F)C3)C2)=O)nn1C 90516,CC#CCCCC(=O)N1CCC(C)(NC(c2cnc(C3CCC3)cc2C)=O)C1 90517,CC(C)CCC(=O)NC1CCCC1(C)CNC(=O)CC1CC2CC2C1 90518,C1(N(C(C2(CC=C)CC=CC2)=O)C)CC2CCC(C1)N2C(=O)CS(=O)(=O)CC 90519,N#Cc1[nH]c(=NCC2(O)CCCN(C(C3CCCSS3)=O)C2)sc1Cl 90520,C1(C(=O)NCCCN(C(c2c(CC)c[nH]n2)=O)C(C)C)COCCN1C 90521,CCC1=NOC(C(=O)NCc2nc(CNC(=O)CC(O)c3ccccc3)cs2)C1 90522,c1(C(=O)NC(CC=C)CNC(=O)C(CC)OCC)sc2nccn2c1C 90523,C1(OCC)(OC)CC2(CC(CNC(C)CCc3ccsc3)C2)C1 90524,C(=O)(CCS(=O)(=O)C1CCCC1)NCCC(C)NC(C1SCCS1)=O 90525,C12(NCC3CCN(C(CNC(N)=O)=O)C3)COC(CC(C3CCCCC3)=O)(C1)C2 90526,C1(C(=O)NCCC#C)OCCC1NC(=O)CSCC 90527,C1(NC(c2ncccc2F)=O)CN(C(c2cccnc2)=O)CC2(CC2)C1 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90580,c1(C(=O)OCC2CN(S(=O)(=O)CC)C2)c(C(=O)NCC)nn2ccccc12 90581,N1(C(c2c(Cl)cn(CCC)n2)=O)CCCC(NC(C2CCOC2CC)=O)C1C 90582,C1(C(N2C3CC(NC(c4c(C)cc(C)o4)=O)C(C3)C2)=O)CCC(C2CCC2)CC1 90583,c1(OC)ccc(Br)cc1CC(=O)NC1CC1CNC(c1coc(C)n1)=O 90584,c1(C(N(CCCN(C)C(C2CC(F)C(=O)N2)=O)C)=O)cnc2c(c1)NC(=O)CO2 90585,C1(C(N2C(CN(C(C3(C(C)C)CCC3)=O)C)CCC2)=O)C(C#N)C1(C)C 90586,N1(CC(C)NC(C2CCC2C(N)=O)=O)CCN(C(C2CCCCC2)=O)CC1 90587,C1(CNC(c2ccc(C(F)(F)F)cc2Br)C)COC2(CCNCC2)C1 90588,N1(C(C=CC(=O)N(C)C)=O)CC(C2CN(C(=O)CCCOC3CCOCC3)C2)C1 90589,Cc1cnc(C(=O)NC2CC3CC(NC(=O)C4=CCSC4)C3C2)cc1C 90590,N1(C(Cc2cc(C(=O)OC)sc2)=O)CCC2C(C1)CN2C(=O)C1=C(C)OCC1 90591,C(C(C(C)C)C(C)C)NC(C(C)(CO)NC(CS(CC)=O)=O)=O 90592,C(=O)(C(CC)C(F)(F)F)N(CCC)CCNC(C1C2C(C2CC)C1(F)F)=O 90593,C(CC(=O)NCCN(C(=O)C(C1CCOC1)OCC1CC1)CCOC)SCC 90594,C(=O)(C1=CCCC1(C)C)NC1CC(NC(c2cn(CCCC)nn2)=O)C12CCC2 90595,Cc1nc(C(=O)NCC2CCCN2C(=O)C(F)(F)c2cscn2)c(C)n1C1CC1 90596,C(C)(c1cccs1)=CC(=O)NCC1C(NC(C2(CSC)CC2)=O)CCC1 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90863,C=CCC(F)(F)C(=O)NCC1CC1NC(C1CCCN(C(=O)OCC)C1)=O 90864,C1(C)(CNC(CCC=C(C)C)=O)CN(C(C2C3CCCCC23)=O)C(C)(C)C1 90865,C(=O)(CC(C(C)C)OCC)NCc1c(CNC(C(CC#C)C2CC2)=O)cccc1 90866,n1(CC(N2CC(NC(CC(C)c3cnn(C)c3)=O)C(F)C2)=O)cccc(O)c1=O 90867,c1(NC(C(C)OC)Cc2ccccc2)ccc(C2CCOCC2)cc1 90868,CCCC(C)(O)CC(=O)NC1CCC(F)(CNC(c2nc(C)ccc2F)=O)C1 90869,Cc1ccc(OC(C)(C)C(=O)NC2CN(C(C3CC(O)C3)=O)C3CC23)cc1 90870,Cc1ccc(C(=O)N(C)CCNC(c2ncccc2N)=O)c(F)c1F 90871,C(=O)(C(C)(C)C(=O)N(C)C)NC(C1CCCN(CCCc2c(C)con2)C1)=O 90872,N1(C(CC(C)O)=O)CCCCC1CCN(C)C(c1ccc(OCC2CC2)cc1)=O 90873,c1(C(=O)NC2CN(C(c3c(C)ncc(C)c3)=O)CC(O)C2)cnc2[nH]cncc1-2 90874,CC(C)C(F)C(=O)NCC1CCC(C(=O)NCC2COCC(C)O2)CC1 90875,c1(CC)c(C(=O)N(CCCN(C(=O)C=Cc2ccsc2)C)C)oc2ccccc12 90876,CC1CC(C(=O)N(CCCNC(C23CC(CC(F)F)(C2)C3)=O)C2CC2)CCS1 90877,c1(C(N(CC(=O)NC2CC(C)OC2=O)CC2CC2)=O)cccc2c1CCC2 90878,c1(N(CC(C)C)C(=O)OC2COC2)ccc(OC(F)(F)F)cc1 90879,c1(C(N2C3CCN(C(CSC)=O)CC3CC2)=O)c[nH]c2c(F)c(F)ccc2c1=O 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91056,N1(C(c2cncc(Cl)c2Cl)=O)CCC2(CC(NC(C3(O)CC3)=O)CO2)C1 91057,C1(NC(C2OCC(C)C2)=O)CCN(C(c2cn(C)[nH]c2=N)=O)CC12CCC2 91058,N1(C(C2C(COC)CC2)=O)CCCCC(C2CN(C(C3(F)CC3)=O)C2)C1 91059,N1(C(C=CCOC)=O)CCC2(C1)CN(C(=O)CC(C)CN(C)C)C2 91060,CC1(C)CN2C(NC3CC3)=NCC1CC2.C1(CO)CC2CC1C2.c1ccccc1 91061,Cc1cc(C(N2CCCC2C(=O)NC2(C)NC(=O)NC2=O)=O)cc2ccoc12 91062,N1(C(c2[nH]n(C)c(=O)n2)=O)CC(F)(F)CC1CNC(=O)C1CC1 91063,c1(CC)nc(C(=O)NCC2CC(F)CN2C(=O)CC2CC2CC)c(N)s1 91064,CC(C)CC(CNC(c1ccn(CCN(C)C)n1)=O)NC(C1(CO)CC1(F)F)=O 91065,N1(C(Cn2c(C)ccn2)=O)CCCC12CCC(NC(=O)C=Cc1cnc[nH]1)CC2 91066,CC1CCC(C(N2C3CCC2C(CNC(=O)CC2COC(C)(C)C2)C3)=O)CC1C 91067,C1(NC(=O)Cc2cnoc2)CCCN(C(=O)C(O)Cc2cnc[nH]2)C1 91068,C(=O)(C(C)(C)C(F)F)N.N1(S(C(C)CO)(=O)=O)CCCCCC1 91069,c1(CC)occ(C)c1C(=O)NCC1CC1NC(C1CC1c1ccsc1)=O 91070,c1(OC)cc(C(N2C3CCC2(CNC(=O)C(F)OC)CC3)=O)ccc1[N+](=O)[O-] 91071,N1(C(CCN(C(C)=O)C)=O)CCc2cc(CNC(C3(C)CC(C)=NO3)=O)ccc21 91072,c1(C(=O)NC(C(=O)N(CC(C2CCC2)OC)C)C)cncc(O)c1 91073,C1(NC(=O)CN2CCCC2)CN(C(=O)Cn2ncccc2=O)C2(CCCOC2)C1 91074,c1(CNC(C(n2cc(C3CC=CCC3)nn2)C)=O)cncc(C(C)(C)C)c1 91075,c1(C(=O)NCCCN(C(C2COCC(C)O2)=O)CCO)cc2cccn2c(O)n1 91076,c1(CNC(N2CCC(NS(=O)(=O)C3CC3)CC2)=O)ccc2nonc2c1 91077,c1(C(N2CC(C)C(NC(=O)C(CO)NC(N)=O)C2)=O)c[nH]c2c(F)cccc12 91078,C1(NC(c2c(C)sc(Cl)n2)=O)CCN(C(=O)COC2(C)CCOCC2)CC1F 91079,c1(OC)cc(C)cc(C(=O)N(C2CC(NC(=O)CN(C)C3CC3)C2)C)c1N 91080,CCCCCCC(C)CC(=O)NC1CCN(CCOc2cccc(F)c2)CC1 91081,C1(CNCc2cc(OC)c(OCC)cc2)(CNC(=O)C(N)=O)CCCNS1(=O)=O 91082,C(=O)(CS(=O)(=O)CCO)NC(C)CNC(C1(N(S(C)(=O)=O)C)CCCCC1)=O 91083,CN1C(=O)CN(CC(=O)NC2CCCC(NC(C3CCOCC3(C)C)=O)C2)C1=O 91084,N1(C(Cc2cc(C)no2)=O)C2CCC(C2)C1CC(=O)NC(C)(C)CC(C)C 91085,CCCCC(C(=O)NC1CCCC1NC(c1cccn1C1CC1)=O)C(C)C 91086,c1(OC)ccc(C(=O)NC(CCNC(c2cnc(C(C)(C)C)o2)=O)C(C)C)cc1 91087,C1(NC(N2C(CC(=O)OC)CN(C(=O)C(F)(F)F)CC2)=O)CC(=O)CC12CCC2 91088,c1(CCNC(C2C(CC)CCC2)=O)ccc(S(=O)(=O)N2CCCN(CC)CC2)s1 91089,C1(CC)CN(C(=O)C(N2CCOC(CC(=O)OC(C)(C)C)C2)=O)CCN1C 91090,c1(C(=O)NC(C2CCCN(C(C3CC4(CC(=O)C4)C3)=O)C2)C)ccc(Cl)c(Cl)c1 91091,C1(NC(C=C(CC)C)=O)CCCC(NC(c2ccc(OCCF)cc2F)=O)CC1 91092,CC(=Cn1ccnn1)C(=O)N1CCCCCC1CCNC(=O)C(C)C1=CCCC1 91093,N1(C(CC2CC=C(C)CC2)=O)CCC(C(=O)N(c2cc(F)ccc2C)C)C(O)C1 91094,CC(C(=O)N1CCC(CN(C)C(c2cc(C(C)(C)C)nn2C)=O)C1)C(F)(F)F 91095,C#Cc1cncc(NC(C2(CNC(c3cc(C4CC4)no3)=O)CC=CC2)=O)c1 91096,N1(C(C(CC)NC(N)=O)=O)CC2CCC1C(CNC(=O)CCc1cccs1)C2 91097,O(C1CCc2ccc(Br)nc21)Cc1cc(C)c(C(=O)OCc2cccnc2)cc1 91098,c1(C(C(=O)NC2CCN(CCSC(C)C)CC2)OCC)ccc(F)cc1C 91099,Cc1cc(C)n(CC(=O)NCCN(CCCNC(=O)CC2CCCCC2)C)c(=O)n1 91100,c1(OC)cccn2ncc(C(N3CC4C(NC(=O)C(F)CC5CC5)C4C3)=O)c12 91101,N1(C(CC)=O)CCCC(CC)C1C(=O)NCC=CC(C)(C)C 91102,C1(C(=O)NCc2nc(C)ns2)(CC)CCCN1C(c1nccn1C)=O 91103,Cc1ccc(C#N)cc1C(=O)NC1CC(NC(=O)C(c2ccccc2)F)C1 91104,C1(CNC(CCC(C)OC)=O)CC2(CC2)CN1C(c1cncc2c1CCC2)=O 91105,c1(CC(C(=O)NCC(c2c(F)cccc2Cl)N(C)C)O)cc(Cl)ccc1Cl 91106,Cc1cccc(C)c1C(=O)NCCC(O)CNC(C1CC(CN(C)C)C1)=O 91107,C1(NC(c2c(SC)scc2)=O)CCN(C(c2[nH]nnc2C)=O)C(C)C1 91108,C1(N(C)C(c2ccccc2N2CCOCC2)=O)CN(C(C2COC2)=O)CC1(C)C 91109,c1(C(=O)NCCN(C(c2n(CC)cnn2)=O)C2CC2)ccc(S(=O)C(C)C)cc1 91110,Cc1ccncc1CC(=O)NCCC1CC(NC(=O)CCc2cc[nH]n2)C1 91111,O=C(C1=C(c2ccccc2)CCC1)NC1(C2CN(C(=O)C(F)C3CC3)C2)CC1 91112,N1(C(c2cc(Br)cs2)C(=O)NC(CC)C)CC2CCC(C)(C1)C2(C)C 91113,Cc1cccc(C(=O)N(CCCNC(c2cnn(CC(F)F)c2)=O)C2CC2)n1 91114,C1(NC(=O)Cc2cc[nH]n2)CCCC(NC(=O)Cc2nc(C3CC3)cs2)C1 91115,C1(OC)CN(C(=O)C(C(C)C)NC(c2ccco2)=O)CC1NC(c1ccon1)=O 91116,c1(C(=O)NC2CCC2NC(c2nsnc2O)=O)cc2nccn2c(O)n1 91117,C(=O)(C(O)CC1CCCCC1)N(CCC(C)NC(c1coc(C2CC2)n1)=O)C 91118,C1(NC(=O)C=Cc2cocn2)CC12CCN(C(c1cnn3c1CCCC3)=O)CC2 91119,O=C(CC1CC2(C1)CN(C(=O)CC1CCOC1=O)C2)Nn1cnnc1 91120,C1(NC(=O)Cc2ncc(Cl)cc2Cl)CCN(C(C2COCCOC2)=O)CC1F 91121,C1(CC)CCC(O)(C(=O)N(CCCNC(c2cc(C(=O)OC)cn2C)=O)C2CC2)C1 91122,c1(C(C)(C)C)ccc(NNC(=O)NCc2ccc(NC3CCOCC3)cc2)cc1 91123,C(CC1CC1)(C(=O)NC(C)C(=O)NCC(C)F)OC 91124,c1(C(=O)OC)ccc(S(=O)(=O)NC2C3CCC(O3)C2N=[N+]=[N-])cc1 91125,N1(C(C2N(NC(=O)C3(SC)CCC3)CCC2)=O)CCC(C2(C)CC2)C1 91126,N1(C(c2ccnc(C3CCCC3)c2)=O)CCC(NC(C2(F)CCOC2)=O)C(F)C1 91127,C1(C(C)CNC(c2cccnc2)=O)CCN(C(=O)CCCN2CCOC2=O)CC1 91128,Cc1c(C(=O)NC(C)CC2CN(C(C3CCCO3)=O)C2)cccc1N 91129,Cc1[nH]c(C(C)(C)C)cc1C(N1CC(C)(NC(C2CCCSC2C)=O)C1)=O 91130,c1(C(=O)Nc2cnc(Br)c(F)c2)cnc2c(C3=CCCCO3)cccc2c1 91131,C(=O)(CCC(=O)OC1CC(C)OC1=O)c1ccc(C)s1.C123CC(C1)(C2)CNC3=O 91132,Cc1cc(C(N2CCC(C(=O)NC3CN(c4ncco4)C3)C2(C)C)=O)nc(O)c1 91133,C(c1cc(C(N2CC3(CNC(=O)CC)CC2CO3)=O)cc(OC)c1OC)=CC 91134,N1(C(CNC(CCCN(C(C)C)C)=O)=O)CCCCC1C(C)O 91135,Cn1cccc1C(=O)NCC1(C(=O)NOCCOCCF)CCC1 91136,Cc1ccc(C(N2CC(C(C)NC(C3CCC(C(F)(F)F)CC3)=O)C2)=O)n1C 91137,c1(CNC(C2C(CCC)C2)=O)ccc(NC(=O)C(c2ccn(C)c2)C)nc1 91138,C12(C(=O)NC3C(OC)CCC3)CC(CN(C(c3ccc(C4CC4)o3)=O)C1)C2 91139,c1(C(=O)NC2CC(C)N(C(=O)CC(C)(C)O)CC2)cccc2ccncc12 91140,C1(C2CCCN(c3nc(C)ncc3C)C2)(NC(C2CC(C#C)(O)C2)=O)CC1 91141,N1(CCCn2ncc(NC(C(=O)NCC(COC)C)=O)c2)C(=O)CNC1=O 91142,N1(C(C(C)OC)=O)CCC(CNC(c2cnn(C)c2)=O)(OC)C1 91143,N1(CC)CC(NC(=O)C=CC2CCCN2C(C23CC(C#N)(C2)C3)=O)C(C)C1 91144,C#Cc1ccc(C(=O)NC(C(=O)N(C(C)C(=O)OC)C)C(C)(C)C)cc1 91145,C1(NC(C=CC(C)C)=O)CC2CC(C1)N(C(=O)Cc1cc(F)ccc1Cl)C2 91146,Cc1sc(=O)n(CC(=O)NCC(C2CC2)NC(=O)CC2CCCS(=O)(=O)C2)c1C 91147,Cn1c(COCC(=O)NCC2CCC(NC(c3ccco3)=O)C2)nnc1S 91148,c1(CC(=O)N(CCCCNC(C2CCCC2O)=O)C)c(F)c(F)cc(F)c1F 91149,C1(NC(c2nn(CC)c(O)c2)=O)CC(NC(=O)C(C)(C)C2CCCC2)C12CCC2 91150,C(=O)(CCC(=O)c1ccncc1)N1CCC(CNC(c2ccc(Cl)nc2)=O)C1 91151,N1(C(C(Cn2cccn2)NC(c2ccccc2F)=O)=O)CCCC2(CCCC2)C1 91152,c1(OCOC)cc(-c2nc(C(=O)Nc3nnccc3C#N)ccc2F)ccc1C 91153,Cc1cc(Nc2ccsc2C(=O)NC(c2ccccc2)CO)nc(Br)c1 91154,C1(NC(c2ccc(OC)s2)=O)CCC(O)CN(C(C2CC(=O)NC(C)C2)=O)C1 91155,N1(C(c2ccnc(C)c2C)=O)CCC(C(=O)NCc2nnnn2C)=C(F)C1 91156,Cc1cn2c(C(N3CCC(CNC(c4sc(F)cc4C)=O)C(C)C3)=O)cnc2s1 91157,CC1CN(C(c2cnncc2C(F)(F)F)=O)CC1NC(c1ncc[nH]c1=O)=O 91158,c1(C(=O)NC2CCCCN(C(CCSC)=O)C2)cc2n(c(=O)c1)CCS2 91159,C(N=c1cc(Cl)nc(C)[nH]1)C1N(C(C=CCOC)=O)CCCC1C 91160,N1(C(=O)C2=CCCCC2)CC2CC(C1)CN(C(c1ccsc1Br)=O)C2 91161,C1(C(=O)Nc2ccc(OCCOC)c(OC)c2)CCn2c(cnc2Br)C1 91162,C1(C(N(CC(C)NC(c2cc(-c3ccccc3)cs2)=O)CC)=O)CC2(CCC2)C1 91163,C(=O)(CC(C)(C)C(=O)N1CC(OC)C(NC(=O)C(COC)CC)C1)OC 91164,Cc1nc(N(C)C)sc1C(=O)NCCC1CN(C(C2CC(C)(C)O2)=O)CCO1 91165,C1(=CC(=O)NCC2N(C(C(C)C3CCC3)=O)CCC2)CCC(C)(C)CC1 91166,C1(NC(=O)NCc2c(C)nc[nH]2)CN(C(=O)OC(C)(C)C)CC1O 91167,CCC(C#N)(CC)C(=O)NCC1CN(C(=O)C(C2CCOCC2)O)C(C)(C)C1 91168,C1(C(=O)N(C2CC2C)C)(NC(CN(CC)CC)=O)CC(O)C1 91169,CP(C)(=O)C(CC(=O)NC1CCOCC1NC(=O)Cc1cncnc1)P(C)(C)=O 91170,C1(NC(Cc2n(C)ccc2)=O)CCC(C)(CNC(=O)CC2CC(=O)NC2=O)CC1 91171,N1(C(C2CC(NC(C3CC(CCC)C3)=O)C(O)C2)=O)CC2CC2C2CC12 91172,N1(C(c2c(C(C)C)noc2)=O)CC(C(=O)NCC2(C)CCCC2O)C(F)(F)C1 91173,c1(C(=O)NC(C2CCN(C(=O)CCn3ccnc3)C2)C)ccc(Br)cn1 91174,N1(C(C(CC)N(C(=O)C=C(C)C(C)(C)C)C)=O)CCCCC(COC)C1 91175,c1(N2CC3C(CC)(C3)C2)ncccc1S(=O)(=O)NCC(c1ccc(F)cc1)O 91176,C(=O)(C(F)CC(C)(C)NC(=O)CCC1CCOC1)NCC=CCSC 91177,N1(C(C(CC)N(C)C)=O)CCC(O)(CCNC(c2[nH]c(C)nc2C)=O)C1 91178,C(CC(=O)N(C)CC1CN(C(=O)CCc2nnc(C)n2C)C1)(C(F)(F)F)OC 91179,c1(OC)ccc2c(C(=O)NC3CC4CC3N(C(=O)Cn3cnnc3)C4)csc2c1 91180,CCC(C)C(C(=O)N(O)Cc1cn(-c2ccccn2)nn1)Oc1ccc(F)nc1 91181,C(=O)(CC(O)C(Cl)(Cl)Cl)N(C(c1ccc(OC)nc1)CCC)C 91182,c1(NC(C2(C)CCN2C(c2ccc(F)nc2F)=O)=O)c[nH]c2ccc(Cl)cc12 91183,S(=O)(=O)(CC(=O)NCCCNC(=O)CC1OCCCO1)N(CC)CC 91184,CC1CC(NC(C2CCC(NC)C2)=O)CN1C(c1ccc(OCC2CC2)cc1)=O 91185,C1(C(N2CC(=C)C2)=O)CC(C)N1C(=O)CC1(COC)CC1 91186,CCC(O)(CC(=O)NCCN(c1cncc(Cl)n1)CC1CC1)c1ccccc1 91187,C#CC1(C(=O)NC2CCC(CO)C2)CCN(C(C2CC3(CCC3O)C2)=O)C1 91188,c1(OCC)ccc(C(=O)N(CC(CC)NC(c2nc(Cl)c(Cl)s2)=O)C)cc1 91189,C1(C(=O)NC(C)CCCNC(C2CCS2(=O)=O)=O)CCCC(C#N)C1 91190,Cc1sc(N)c(C(N2CCCC(CO)(CNC(=O)C(O)CN(C)C)C2)=O)c1C 91191,C1(C)(CCOC)CCN(C(=O)NCC(C)(O)CCO)CC1 91192,N1(C(C23CC(OC)C2C3)=O)CCC2(CC1)CN(C(=O)C=C(C)C)C2 91193,c1(OC)ccc2c(c1)CC(OC(C)C)CN2C(c1c(F)c(C)cc(F)c1F)=O 91194,N1(C(CCN(C(C)=O)C)=O)CC(NC(c2nnc(S)n2C)=O)CC2(CC2)C1 91195,C#CCCCCCCC(=O)NC(C)CN(C)C(C1CCCN(C(C)C)C1)=O 91196,Cn1cnc(C=CC(=O)NC2CC(F)(CNC(C3CCCC(F)C3)=O)C2)c1 91197,C(=O)(C1Cc2c(Cl)cccc21)N(C(C)CNC(=O)CNC(=O)OC(C)(C)C)C 91198,CCCCCC(C)(C)C(=O)N(CC(C)CNC(=O)CC1CC(O)C1(C)C)C 91199,N1(C(CCCNC(C)=O)=O)CC(F)(F)CC1(C)CNC(=O)C(F)OC(F)(F)F 91200,N1(C(CSC)=O)CCC(C)(CCNC(=O)CN(C(c2ccccc2)=O)C(C)C)C1 91201,c1(C(=O)NCCN(C(=O)CC2CCCCN2C)C)cn(C)c(O)n1 91202,C#Cc1ccc(C(=O)NC(CNC(c2cn(C(C)C)nn2)=O)CCCC)cc1 91203,N1(C(c2cc(CC)no2)=O)CCC(NC(=O)CC(F)F)C(CC)C1 91204,C(=O)(C(CCO)N(C)C)NC1(C2N(C(CC(=O)OC)=O)CCC2)CC1 91205,C1(CC)CN(C(=O)C(CC(F)F)N(C(=O)C=C(C)C(C)C)C)C(C)CO1 91206,c1(C(=O)NC2CCN(C(CC(CC)C)=O)CC2O)nc2ccccc2cc1Br 91207,C(=O)(CS(=O)(=O)C1CCCC1)N1CC(NC(C(C(CC)C)O)=O)C(OC)C1 91208,N1(C(C(CCC)OCC)=O)CCN(C(c2n[nH]cc2OC)=O)C2(CCC2)C1 91209,C(=O)(CCCCCF)NCCNC(C1(SC)CCC1)=O 91210,c1(C(N(C)CC2C=CC(NC(=O)Cn3cccn3)C2)=O)cnc(C(C)(C)C)[nH]1 91211,N1(C(Cc2nnc(C)o2)=O)CCN(C(=O)C=CCn2cncn2)C2CC12 91212,C1(NC(c2ccncc2O)=O)COC2(CCN(C(c3cc[nH]c3)=O)C2)C1 91213,C1(CCC(=O)N(CC(=O)OC)C)CCCCN(C(c2ccncc2)=O)C1 91214,c1(SC)cc(C(=O)NC(CCNC(C2(C(F)F)CC(O)C2)=O)C(C)C)ccc1N 91215,N1(C(CNC(=O)OCC)=O)CCN(C(c2cccc(Cl)c2OC)=O)C(C2CC2)C1 91216,c1(CC(=O)NC2CC3(C(NC(COC)=O)C3)C2)c(C)nc(Br)nc1O 91217,c12cnc(nc1)C(=O)N1CCCC(C1)Cc1cn(nn1)C2C.n1(CO)cccc1 91218,N1(C(C2CC(=C)C2)=O)CC=CC1C(N1CCC(N2CCC2)C1)=O 91219,C1(NC(C(COC)C)=O)CCN(C(=O)C(c2ccc(OC)c(OC)c2)C)CC1O 91220,N1(C(C)C)CCCC(C)(C(N2CCCC2CC(=O)N(C)Cc2cn[nH]c2)=O)C1 91221,CC(C)C1=CCC(C(N2C3CCC2CC(CCNC(=O)CSC2CC2)C3)=O)CC1 91222,N1(C(CC=C)=O)CCC2(CCC2NC(=O)C=C2CCSCC2)CC1 91223,Cc1nccn1C(C)C(=O)NC1CCCC1NC(=O)CCOC1CCCCC1 91224,CN1CCn2ncc(C(=O)NCC3CN(C(=O)CC(C)(C)C)CC(C)(C)O3)c21 91225,c1(C(N2C(C(C)NC(CC3(C#C)CCC3)=O)CCC2)=O)ccc(OC)cc1Cl 91226,c1(CC(N2CCC(C)(CCNC(CCC#C)=O)C2)=O)c(C)[nH]c2ccc(F)cc12 91227,S(=O)(=O)(CC(=O)NC1(C2CCCCN2C(C2(C)CCN(C)C2)=O)CC1)NCC 91228,C1(NC(c2ccc(C(C)=O)cc2)=O)(CO)CCCN(C(C2CC(O)C2)=O)C1 91229,Cn1nc(C(=O)NC2CCCN(C(C3(N4CCOCC4)CC3)=O)C2)cc1Cl 91230,c1(C(N2CC(OCCNC(C3C(OCC)C3C)=O)C2)=O)cnnc(C)c1 91231,C12CC(F)CCN1C2=O.c1(C(=O)NCc2ncccn2)cncc(Cl)c1 91232,n1(CC)cnc(NC(=O)CC2CC=CCC2)cc1=O 91233,c1(CSCC)cc(C(=O)N(CCC(=O)NCCC(=O)OCC)C)no1 91234,c1(C(=O)NC(C(=O)NCCC(CC)O)C2CCOC2)c[nH]c2ccccc12 91235,c1(CNC(CN2CCN(C(C(CCC)NC(C)=O)=O)CC2)=O)ccc(Cl)c(Cl)c1 91236,C(=O)(C(C)C(C)N)NC(=O)C=CCOCCOC.C(CC(=O)N)SCC 91237,CC(C)C(CC(=O)NC1(CCO)CCCCC1)NC(C1CCC2(CCC2)C1)=O 91238,N1(C(c2c(CC)cno2)=O)CCC(C)(C(=O)N(CC(C)C(F)(F)F)C)C1 91239,c1(CC(=O)NC2CN(C(=O)C3=CCCCC3)CC3CC23)ccc(F)cc1[N+](=O)[O-] 91240,N1(C(c2ccc(CC)s2)=O)CCC(CO)(NC(=O)C(C)(C)c2ccccn2)C1 91241,CC1CN(C(=O)CCC(N)=O)CCC1NC(C12CC(c3ccccc3)(C1)C2)=O 91242,C1(C(=O)Nc2ccnc(F)c2Br)Cc2cc(O)ccc2CN1Cc1cn[nH]c1 91243,C(=O)(C#CC1CCCCC1)NCC(C)(CO)NC(C(CCCC)CC)=O 91244,C1(C(N(CC(COCC)O)C)=O)C2CN(C(C3(F)CC=CCC3)=O)CC12 91245,N1(C(C2(N(C)C)CCC2)=O)CCCC(C)(C(=O)NCCc2ccccn2)C1 91246,N1(C(c2cc(C)c(C)s2)=O)C(C(=O)N(C2CCCC2)CCO)CC2CCCCC12 91247,N1(C(C2C(C)C2C)=O)CCC(CC(=O)NCCF)C1 91248,c1(C(N2C(CN(c3nnc(C)o3)C)CCCC2)=O)c(O)nnc2c1CCCC2 91249,Cc1ccc(CCC(=O)NC2CC2NC(c2c(C)noc2N)=O)cc1C 91250,C1(CNC(C2(C)C=CCCC2)=O)CN(C(c2cc(O)ncn2)=O)C2CCCCC12 91251,N1(C(COCCCCC)=O)CC2CCN(C(c3ccc(F)c(F)c3N)=O)C(C2)C1 91252,Cc1cc(=O)n(C)cc1C(=O)NCC1C(CNC(=O)C=CC2CCCN2C)C1(F)F 91253,c1(NC(C(C2CCN(C(C3C(C)(C)C3(C)C)=O)C2)F)=O)ccc(O)cc1F 91254,c1(NCC(N2CCN(CC)CC2)(C)C)ccc(S(=O)(=O)NC2CC2)cc1C#N 91255,c1(C(=O)NC2C(CNC(c3c(C)nc[nH]3)=O)C2)cn2c(n1)CCC2 91256,c1(C2(C(=O)NC3CC(C)(c4ccccc4)OCC3)CC2)nnc2n1CCCCC2 91257,Cn1ncc(C(=O)NCc2occc2C(=O)NCC2CCCSC2)c1N 91258,c1(C(N2CC(NC(C(CC=C)OC)=O)C(O)C2)=O)cccc(OC)c1F 91259,C(=O)(C(C)CCCC(C)=O)N(C1CCN(C(=O)Cn2nc(C)oc2=O)C1)CC#C 91260,c1(C(=O)NC23C(CN(C(Cn4c(C)cnc4)=O)C2)CC3)nc2nccc(C)n2n1 91261,C(=O)(C1=CCCCC1C)NCc1ccc(C(N2CC=C(C)C2)=O)cn1 91262,C1(NC(C(c2n(C)ccc2)=O)=O)CCCC(NC(c2cnsn2)=O)C1 91263,C12(CCC(C)(C)C1)C(=O)N2CC.C(=O)(C=CSC)NC1CC(C(=O)OCC)C1 91264,Cc1cc(Br)c(CN2CCN(c3ccc(CN)cc3)CC2)cc1O 91265,C(=O)(NN1CCC(F)(F)CC1)N(C(c1cn(C(C)C)nn1)C)C 91266,N1(C(C2C(CC)C2)=O)CCCC(C2CN(C(C34CC(C)(C3)OC43COC3)=O)C2)C1 91267,CC1CCC(CO)(NC(c2cncc(CNC(=O)C(C)OC(C)(C)C)c2)=O)C1 91268,C(=O)(C1Cc2ccccc21)N1CC(N(C)C(c2ccc[nH]2)=O)C1 91269,C1(CCC)(NC(C2CC3(CCC3)C2)=O)CCCN(C(C2CS(=O)C2)=O)C1 91270,N1(C(C2CC3CC(OC)C3C2)=O)CC23CCCC2(C1)CN(C(=O)C1=COCC1)C3 91271,c1(C(C)(C)CNc2ccnc(N3CCCCC3)c2)cc2cccc(F)c2[nH]1 91272,CC(C)C(C(=O)N1CCC(CCNC(=O)C(C)NS(C)(=O)=O)C1)C(C)C 91273,c1(C(=O)NC2CCN(C(C3C(C=C)CC3)=O)CC2CO)cccc2c1CCC2 91274,C(=O)(C1=CC2(CCOC2)C1)N1CCC(N(C23CC(C2)C(C)O3)C(C)=O)C1 91275,c1(C(=O)OCc2c(C)cccc2F)cc2ccc(Cl)cc2c(=O)o1 91276,C1(NC(Cc2scc(C)c2)=O)CC2CCC(C1C)N2C(c1ccc(C2CC2)o1)=O 91277,C1(C(=O)NC(C)CNC(=O)Cc2cn(C)nc2Cl)CCc2nnc(O)cc2C1 91278,C1(CNC(c2ccc(CC(C)(C)O)s2)=O)CCCCN(C(C2CC=CCC2)=O)C1 91279,c1(NC(C(C)(O)C2CCCCC2)=O)cc[n+]([O-])cc1 91280,O=C1CCc2cc(C(N3CC(=O)NC(CO)C3)=O)sc21 91281,C1(NC(=O)CSCc2ccccc2)CCN(C(C23CC(F)(C2)C3)=O)C12CCC2 91282,N1(C(CCS(CC)=O)=O)CC2(CCC(NC(C3CCCN(CC)C3)=O)CC2)C1 91283,C1(NC(c2c(C)onc2)=O)CCC2(CCCN2C(c2cccc(Cl)c2F)=O)CC1 91284,N1(CC)CCCC1C(=O)NCCCSc1cc(C)no1 91285,c1(C(N2CC(NC(c3cc(Br)ncc3Cl)=O)C(O)C2)=O)ccc2ccncc2c1 91286,Cc1cc(NC(C2CCN(C(c3cnn4cc[nH]c34)=O)C2)C)ncc1[N+](=O)[O-] 91287,C#CC1(C(=O)NCCC2CCCC2(F)F)CCN(C(=O)C(O)CC(C)(C)C)CC1 91288,c1(C(=O)NCC(n2cc(C3(C)CCOC3)nn2)C)cccc(F)n1 91289,c1(CNCC2CN(c3nc(C)[nH]n3)CCO2)cnc(N(C)C)cc1Cl 91290,N1(C(C2CCCCO2)=O)CCNC(C(N2CCCC(F)C2)=O)C1 91291,N1(C(=O)OC(C)(C)C)CCc2ncc(NS(c3c(C)nn(C)c3C)(=O)=O)cc2C1 91292,C1(NC(c2on(C)c(=O)c2)=O)CCCCC12CCN(C(c1cccs1)=O)C2 91293,c1(C(=O)NC2CN(C(c3cnc(Cl)[nH]3)=O)CC2F)cc2cc(F)cc(F)c2[nH]1 91294,C1(CC(=O)N(C(C)CC2CNC2)Cc2ccccc2)CCCCC(=O)N1 91295,c1(N(CCN(C(C2C(=C)C2)=O)C)C)nc2c(C(=O)OCC)cccc2o1 91296,CN(C)NC(=O)CCC(=O)NCCOCCCNC(C1(C#N)CC2CC2C1)=O 91297,c1(C(=O)NCC(CO)NC(c2c(CC)scc2)=O)cc(F)cc2cc[nH]c12 91298,C(=O)(C(CC(C)C)C(C)C)NCCC(C(=O)NC1C(CCC)C1)OC 91299,c1(C(=O)NCC2OCCN(C(CNC(C)=O)=O)C2)cnn2cccc(Cl)c12 91300,C(=O)(CCCCCF)NCCC1CCC(NC(CN2CCC(OC)C2)=O)C1 91301,N1(C(c2c(CC)nc3n2CCCC3)C(=O)NCCC)CCC(C2CCOC2)CC1 91302,c1(C(=O)NC(CC=C)CNC(=O)C(C)CC2CC2)cnn2ccnc(C)c12 91303,C12(C(=O)N(CC(C)(C)C)C(C#C)C3CCC3)CCCC1N(C(=O)CN)CC2 91304,C12(NC(Cc3ccc(C)o3)=O)CCCC1CN(C(=O)Cc1ccno1)C2 91305,c1(OC)cccc(C)c1C(=O)NC(C)C(c1ccccc1)NC(C12CCC1C2)=O 91306,CCN=C(NCCNc1cc(OC)cc(OC)c1)N1CCC(CN2CCCC2)C1 91307,C1(CNC(CCC=CC)=O)CCN(C(c2cnc(C(F)(F)F)s2)=O)CC1C 91308,N1(C(c2cc(C(=O)OC)sc2C)=O)CCC2C(C1)CN2C(=O)CSc1cn[nH]c1 91309,Cc1ccc(Cl)cc1C(=O)NC12COC(CNC(c3cnn(C(F)F)c3)=O)(C1)C2 91310,c1(C(N2CCC(NC(C(CC)O)=O)CC2)=O)c(Br)sc(C)c1C 91311,c1(-c2n(C(C)C(F)(F)F)nc(C3CCC3)n2)cc(Cl)cc(C#N)c1 91312,N1(C(COCCCC)=O)CCCC(NC(=O)C(C)N2CCC2)C1 91313,C1(N(C(c2n(CCOC)ncc2)=O)CC)CCCN(C(C2CC=CCO2)=O)CC1 91314,C(CCC(C)C)(C(=O)N(C1CCCN(C(=O)CC2OCCO2)C1)C)NC(C)=O 91315,c1(C(=O)NC2CN(C(Cn3nc(C)oc3=O)=O)CC2(C)C)ccc2c(c1)CCC2 91316,C(=O)(C(CC(C)C)ONC(=O)CC1CC(F)C1)N(CC)CC1(O)CCC1 91317,C12(NC(COCC(=C)C)=O)CCCC1N(C(=O)Cc1ccc(O)cn1)CC2 91318,CCC(C)(CC)C(=O)NC1CN(C(=O)C(C)Cc2ccnn2C)CC1OC 91319,c1(OC)ccc2c(c1)OC(C(=O)OCC(C1CC(F)(F)C1)OC)C2 91320,C(c1ccc(C(F)(F)F)c(O)c1)=CC(N(CC)OCCOc1ccccc1)=O 91321,N1(C(c2c(SC)cccn2)=O)CC(NC(c2csc(C)c2)=O)CCC1C 91322,c1(SC)cc(C)c(C(=O)NC2CCCC2CNC(C2CCCO2)=O)o1 91323,c1(C(=O)NC2C(NC(c3cscc3F)=O)CCCCC2)cnc2[nH]nnc2c1 91324,CCCCCCC(CC)C(=O)NC(C)CCCNC(=O)C(C)C(C)S(C)(=O)=O 91325,c1(C(=O)NCCN(C(c2c(OCC)nc(C)cc2)=O)CC)c([N+](=O)[O-])cnn1C 91326,CCCC(C#N)C(=O)NCC1(NC(=O)C=Cc2ccc(C(=O)N(C)C)cc2)CC1 91327,C1(C2CC2)(C(=O)NCC(c2ncn(C)c2)O)CN(C(=O)Cn2ncnn2)C1 91328,Cc1ccc(Br)cc1CC(N1CCC(F)(C(N2CCOCC2C)=O)C1)=O 91329,c1(C(N2C(C(N(CC#C)CCF)=O)CC2C)=O)coc2c1COC2 91330,C1(NC(=O)C(F)=C2CCC2)CC2CC1CN(C(c1coc(C3CC3)n1)=O)C2 91331,c1(C(=O)NC2C3CN(C(c4c(C)cc(C)[nH]4)=O)CC32)cc2c(ccn2C)s1 91332,N1(C(CCC(=C)Cl)=O)C(C(=O)NCc2cc(C)c(C)o2)C2CC(O)C1C2 91333,CCC(CC1CCCC1)C(=O)N(C)CC1CN(C(c2c(C)[nH][nH]c2=N)=O)C1 91334,c1(C(C)Nc2nc(C)[nH]c(=NCc3n[nH]cc3C)c2)ccc2c(c1)NC(=O)CO2 91335,N1(c2c(C)cccc2)CC(C(N2CC(NC(=O)COC(C)C)C(C)C2)=O)CC1=O 91336,N1(C(C(C)(C)C)=O)CCC2C1CCCN2C(c1cc(O)c(O)c(Cl)c1)=O 91337,c1(CN2CCC(O)(C(=O)Nc3n(CC)ncc3Br)C2)ccc(Br)c(OC)c1 91338,CC(C)CCC(=O)N1CC(CNC(=O)C(C)CC2CCCCC2)C2CC12 91339,N1(C(c2ccc(CCC)cc2)=O)CCN(C(=O)C(C2CC2)OCC)CC(C)(F)C1 91340,Cc1csc2ccc(C(=O)NCCC(C)(C)NC(C3CCC4CC34)=O)cc12 91341,C1(NC(c2c(C)cno2)=O)CCC2(C1)CN(C(C1(C)CC1)=O)C2 91342,C1(C(=O)NCc2ccsc2)CC12CCN(CCC1(F)CCC1)CC2 91343,N1(C(CC2C(C)CC2)=O)CC(NC(C2CC3(CCC3O)C2)=O)CC12CCCCC2 91344,C1(NC(c2ccnc(OC)n2)=O)CN(C(=O)C(C2CCC2)OC)CCC1F 91345,C(CC(=O)NOCC1CCOC1)N(C1CC2(OC)CC1C2)C(C)=O.OCC 91346,CC(C)CC(CNC(=O)C(F)=CCCF)C(=O)NCC(C)(C)CO 91347,c1(C(N(C(C)C)C)=O)n[nH]c2ccc(-c3ccc(-n4ccnn4)cc3)cc12 91348,C1(C(N2CCN(C)CC2CO)=O)CC2(CCC2)CN1C(c1coc(N(C)C)n1)=O 91349,c1(CC(C(=O)N2CCC(C(C)NC(=O)CC3CC3)C2)(C)C)ccc(C#N)cc1 91350,CCCCCC(O)C(=O)NC(C)(CNC(c1cc(C)ccc1C(C)C)=O)C1CC1 91351,N1(C(C#C)C)CCN(C(C2(NC(c3cn(C)cn3)=O)CCOCC2)=O)CC1 91352,Cc1nc(C)c(C(N2CCC(C)(CNC(C3(CC#N)COC3)=O)C2)=O)nc1C 91353,C1(C(N2CC3C(NC(c4cc(C)cc(O)c4)=O)C3C2)=O)(OC)CCC(C)(C)C1 91354,Cc1nn(C)cc1C(O)C(=O)NC1CCN(C(=O)C(=Cc2cccnc2)F)C1C 91355,c1(CCSC)cc(CNC(=O)NC(c2ccc(OC)nc2)C(F)F)cc(F)c1 91356,c1(CCC(=O)NCCN(C(C)C)C(C23CCCCC2C3)=O)ccc(F)cc1Cl 91357,c1(C(N(CCCNC(CSCCCC)=O)CCO)=O)cccc([N+](=O)[O-])c1OC 91358,C1(F)(Cc2ccc(CNC(C3(OCC)CCCCC3)=O)o2)CCN(C(C)=O)CC1 91359,C(=O)(C(F)C(F)(F)C(F)(F)F)N(c1c(OC)c(Cl)ccc1)C 91360,c1(C(=O)NCCSCC(=O)NCC(C(C)C)(C)F)cc(O)cc(F)c1 91361,Cc1cc(C)n(CC(=O)N(CC(CO)(CO)NC(c2cn[nH]c2)=O)C)n1 91362,Cc1cc(NC(=O)CCc2cscc2Br)ncc1Br 91363,CN1CCN(CC(=O)OC(C)(C)C)CC1.C12C=CCN(C1)C(=O)CONC(=O)C2 91364,C1(OC)CC(NC(N2CCN(c3cccc(C(F)(F)F)c3)C(=O)C2)=O)C12CCC2 91365,C1(NC(=O)COc2ccc(Cl)cc2)CCN(C(C2CC2(F)F)=O)CCC1CO 91366,C1(C(=O)NC(CN(C(=O)CCOCC2CCCC2)CC)C)CCCCS1 91367,C(=O)(C1=CCCSC1)N(CC(C(=O)NCCN1CC=C(C)CC1)C)C 91368,C1(C)(NC(C(n2cc(-c3cccnc3F)nn2)C)=O)CC=CCC1 91369,C1(NC(c2ccns2)C)CC2CCC(C1)N2CC1C2CCC(C2)C1(C)C 91370,c1(CC)c(C(=O)NC2CC2CNC(=O)Cn2nnnc2C2CC2)ccn1C 91371,c1(CC(C#C)NC(=O)N(c2cnn(C)c2)C2CC2)cccc(Br)c1 91372,CCC(CCC(=O)NC(CO)CCCO)NC(=O)CCC(C)N(C)C 91373,c1(CCCCC)nc(C(N2CCC2CNC(C2CCC2C(F)F)=O)=O)cs1 91374,c1(C(=O)NCC(N(C(CCOC)=O)C)C2CC2)ccc(S(C)=O)cc1 91375,CCCCC(C)C(=O)NC1CN(c2ncccc2Br)C1 91376,c1(OC)cc(N2CC(CO)(NC(=O)Cc3cnccc3C)C2)nc(C(F)(F)F)n1 91377,C(CNC(c1cnn(CC2CC2)c1)=O)(CC(F)(F)F)NC(C1(C#C)CC1)=O 91378,N1(C(CCN(C)CC)=O)CCC2(CCC(NC(=O)CC(C)CC(C)(C)C)C2)C1 91379,C12=NC=C(C(C)=N1)C2C(=O)NC.C1(NC)CC(C)(C(=O)OC(C)(C)C)C1 91380,Cc1cn2c(C(=O)NC(C)C(CO)NC(C3(F)CCOCC3)=O)c(Cl)nc2s1 91381,C(=O)(C1=CC2C=CC(C1)C2)N1CCC(C(C(NOC2CCN(C)CC2)=O)F)C1 91382,c1(CC)ccnc(C(=O)NC2CC(C(=O)NC3CCC(=O)NC3)C2)c1 91383,c1(SC)ncc(C)c(N2CCCC(C(C)NC(c3cc(Br)ccc3Cl)=O)C2)n1 91384,C(=O)(CCC(C)(C)C#N)NC(CCCNC(CCc1ccc(OC)c(C)c1)=O)C 91385,C(=O)(CCCCCN=[N+]=[N-])N(CCC(=O)N(C)CCOC(F)F)C1CC1 91386,c1(C(=O)NC2C(C)(C)CCN(C(c3cnc(O)o3)=O)C2)cnc2ccc(F)cn12 91387,N1(C(C2ON=C(C)C2)=O)CCN(C(=O)CC(F)F)CC1C(C)C 91388,C=CCCCC(=O)N1CC(CNC(c2cncn2C(F)(F)F)=O)CC1C 91389,N1(C(c2cc(CC)n(C)n2)=O)CCC(CNC(c2csnc2C)=O)C(F)(F)CC1 91390,C=CCCCC(C1CC1)NC(=O)Cc1cccc(-c2nn[nH]n2)c1 91391,c1cnc2ccc(C3CCCN3C3CN(c4nncs4)C3)cc2c1 91392,N1(C(c2cnc(CC(C)C)s2)=O)CC(CNC(C2(CC(F)F)CCC2)=O)C2CC12 91393,N1(C(C)=O)CC2CCC1CN2NCC(C)CS(N)(=O)=O 91394,c1(C(=O)NCC(C)CN(C)C(c2cccc(F)c2)=O)cc2cnccc2[nH]1 91395,c1(C(C(=O)NC(CC)(C)C)N(C)Cc2cncnc2)ccc(C)c(C)c1F 91396,C(CC(C(=O)NCCCC(=O)NCCOC1(C)CCOCC1)NC(N)=O)SC 91397,C12(NC(=O)CCc3cc(Cl)no3)CC1CN(C(=O)C(C1CCC1)C1CCC1)C2 91398,N1(C(CSCC=C)=O)CC2(C1)OC1(C)CC2(NC(c2cc(Cl)c(C)cn2)=O)C1 91399,c1(C(N(CC(C)NC(c2cc(C#N)on2)=O)CC)=O)nn2c(c1C)OCCC2 91400,C(=O)(C(C)(C)CN(C)C)NCc1nc(OCC)oc1 91401,CC1(C)CN(C(=O)CSC(F)F)CC1NC(C1(F)CCCC1)=O 91402,N1(C(C2OCCC(C)C2)=O)CC(NC(c2cnccc2Cl)=O)CC12CCOCC2 91403,N1(NCC2N(C(C(=O)NCC(C(C)C)N3CCCCC3)=O)CC2)C(C)CCC1C 91404,c1(CCC(=O)NCCN(C)C(C2CC2(C)C)=O)ccccc1[N+](=O)[O-] 91405,C1(CNC(C(CN(C)C)NC(C2CC2C(C)(C)C)=O)=O)CCCC12CC2 91406,Cc1c(NCC2(CO)CC2c2cccs2)ncnc1N(C)CC=CCO 91407,C1(NC(c2c(CC)csc2)=O)CC2CC(NC(c3cnccc3N(C)C)=O)C2C1 91408,N1(C(C(C)NC(C)=O)=O)CC(C2(NC(C3CN(S(C)(=O)=O)C3)=O)CC2)C1 91409,c1(CCNC(C(C)N(CCCC)C(c2ncc(C(F)F)s2)=O)=O)ocnc1CC 91410,Cc1nc(C)c(C(N2CCC(CCNC(=O)CC3CC3)C2)=O)nc1C 91411,c1(C(=O)NCC(CO)NC(c2n(CC)ccn2)=O)cccc(-c2ncon2)c1 91412,CN1CCN(C)CC(C(N2CC(n3cc(CNC(C4SCCCS4)=O)nn3)C2)=O)C1 91413,CC(=O)CCN=C(NCCNC(=O)N(C)C)NC1CSCC1C 91414,N1(C(C(CSC)O)=O)CCC(C(=O)NCC(c2nccs2)C)=C(F)C1 91415,C(c1cncc(O)c1)=CC(=O)NCC1CC(CNC(c2c(C)ocn2)=O)C1 91416,C1(CNC(C(C)(C)CO)=O)CCN(C(C2CCN(c3ncccn3)C2)=O)C12CC2 91417,c1(C(=O)NCC2CN(C(COC)=O)C(C)C2)cc2c(Br)cccc2s1 91418,C(=O)(CCS(=O)(=O)c1ccc(C)cc1)N1CC2C(N(C(C(CC)C)=O)C)C2C1 91419,N1(C(C(CC)(F)F)=O)CCCOC(CNC(c2c(OC)ccnc2F)=O)C1 91420,C1(C)(CC)CC(NC(=O)C(=O)N(C)C)CN1C(=O)Cc1ccsc1Br 91421,N1(C(C(C)(C)NC(=O)NCC)=O)CCCC2(CCC(NC(=O)CCCOC)C2)C1 91422,c1(C(=O)NC2(CNC(C3N(C)CCC3)=O)CCOCC2)ccc(N)c(N)c1 91423,CCCCS(=O)(=O)CC(=O)N1CCCC2(CNC(C3(C(C)C)CC3)=O)CCCC12 91424,CCS(=O)(=O)c1cccnc1C(=O)NCCCN(C)C(C12COCC(C1)OC2)=O 91425,c1(CN(c2nnsc2C)CC(=O)NCC(C)(CO)NC(C)=O)ccccc1Cl 91426,C1(CC(=O)NCC(C)(C)C)C2CCCC2N1C(c1ccc(C(N)=O)o1)=O 91427,N1(C(CNC(C)=O)=O)CCCC2(NC(=O)COc3ccc(C#N)cc3)CCCC12 91428,C1(CNC(CN2CC(CC)C2)=O)CC(C)(C)CN1C(C1CCCOC1)=O 91429,c1(NC(=O)NCC2COC3CCCC3O2)c(C(F)(F)F)nc2n1CCCC2 91430,c1(C(=O)NC(C(=O)N2CC(C(C)OC)C2)Cc2cn[nH]c2)ccc(O)nc1 91431,C#CC1(CO)CN(N2CCCC(CC(N)=O)C2)C1 91432,Cc1cc(C)c(C(=O)NS(=O)(=O)CC2CCCC(C3CC3)O2)o1 91433,C(=O)(C(CC(C)(C)C#N)N1CCN(C)CC(O)C1)NCCCCCC 91434,CC(C)(C)CCC(F)C(=O)NCCNC(c1ccc([N+](=O)[O-])cc1Cl)=O 91435,C1(NC(=O)CCc2cnc(O)[nH]2)CN(C(=O)C=CC=C(Cl)Cl)C2CC12 91436,c1(CCC)cc(C(=O)NC2C(CNC(C3(C(=O)NC(C)C)CCC3)=O)C2)no1 91437,C1(CCNC(C=CC=CCC)=O)CCCCN1C(=O)CN1CCCC1C 91438,CC1CCN(C(c2cc3[nH]ccc3s2)=O)CCN1C(=O)C=C1CCCCC1 91439,c1(C(=O)NCCC2C(C)CCCN2C(=O)CC23CC(C2)C3)cc(F)cc(N)c1F 91440,c1(C(N(C2CCN(C(=O)COCC3CCOC3)CC2)C)=O)cccc2sccc12 91441,c1(OC)c(C(=O)NC2CC(NC(C3CCCC3O)=O)C2)cc([N+](=O)[O-])cc1Cl 91442,c1(OC)ccccc1C=CC(=O)NC1CCCCC1N(C(=O)CSC(F)F)C 91443,CCC(CC)C(C)C(=O)NC12CCOC(CNC(c3cc(Cl)cnc3O)=O)(C1)C2 91444,Cc1ccc2c(C(=O)N(C(C)CCNC(=O)C(CN(C)C)C(C)C)C)csc2c1 91445,C1(NC(C=C(C)c2cccs2)=O)CC2(CCCN(C(=O)C(F)(F)C(C)O)C2)C1 91446,CCCC(CCCNC(=O)CC1CCN(C)CC1)NC(=O)CN(C1CCC1)C 91447,Cc1ccc2[nH]c(C)c(CC(=O)NCC3OCc4ccccc43)c2c1 91448,C#CC1CN(C(=O)COCCC)CCN1C(c1n[nH]c(=N)s1)=O 91449,N1(c2cc(C)nc(CO)n2)C2CCC1CC(CNC(C1(n3cnnn3)CC1)=O)C2 91450,CCCC(C(=O)NC1CCCC(NC(c2ccc(N)c(SC)c2)=O)C1)S(N)(=O)=O 91451,C=C=CC(C)C(=O)NC(c1ccc(F)cc1)CNC(c1ccn(C2CCC2)n1)=O 91452,C1(NC(C(C2CCCCCC2)C)=O)C2CC1N(C(=O)COC1(C)CCC1)C2 91453,CCCCCCC(F)C(=O)N1CCC(CN(C(=O)CC2(O)CCOC2)C)CC1 91454,N1(C(C(=O)OC)CCSc2cn(-c3cnn(C)c3)nn2)CCCCCC1 91455,c1(ONC(=O)NC2C(C)C(O)C2)ccc(C#N)cc1 91456,c1(CC(=O)NCC(CNC(CCC(C)N(C)C)=O)O)cc(Cl)cc(Br)c1 91457,c1(NC(C2CC(=C)CN2Cc2cc(C)[nH]c2C)=O)ccc(Br)cc1OC 91458,CCC(C)CCC(O)CC(=O)N1CCC(C)(C)C(CNC(C2(F)CCCC2)=O)C1 91459,C12(CNC(Cc3cncc(C)c3)=O)CCC(C1)N(C(C1CCCCCCC1)=O)C2 91460,Cc1nnc2ccc(C(=O)NC3CCCC(NC(C4CC(F)C4)=O)C3)cn12 91461,C(=O)(CC1C(=O)Nc2ccccc21)NC1CCN(C(c2cnn(C)n2)=O)C1(C)C 91462,c1(OC)ccc(C(=O)NC2CCC(NC(=O)C=Cc3ccco3)C2)nc1Br 91463,c1(NCC=C)[nH]c(=NCC2C(F)(F)C23CCC3)nc2c1ncn2C 91464,CS(=O)(=O)CCC(=O)NCC1CC(CNC(c2cn3ccnc3s2)=O)CO1 91465,N1(C(CC2CC(C)C2)=O)CCc2nc(CNC(=O)C(C)(C)C(C)(C)C)sc2C1 91466,N(C(=NCCN1CCOCC1)NC1CC2(CCC2)C1)CC1(C#N)CCCO1 91467,C12(C(N3CCC(CNC(=O)C=Cc4cccc(O)c4)C3)=O)CCCN(CCC1)C2 91468,C(=O)(CCC(C)(C)C#N)NCC1CC(NC(c2c(CC)con2)=O)C1(C)C 91469,N1(C(c2c(CN(C)C)cco2)=O)CCCC2(CCCN2C(=O)Cc2ccon2)C1 91470,C(=O)(CCCCC(C)(C)C)N1CC(C(=O)NC2(CC)CCOC2)C(F)(F)CC1 91471,N1(C(CCc2nc(C)sc2)=O)CCCC12CCN(C(C1CCC1(F)F)=O)C2 91472,N1(C(=O)NCC2CCN(c3cccc(F)c3)C2)CCCCC(C2CCOC2)C1 91473,C(=O)(C1=CC2CCCCCCC12)NC1C(C)(C)CN(C(=O)C=CC2CCCO2)C1 91474,N1(C(COC2(C#C)COC2)=O)CCN(C(=O)C(C)CC=C)C2COCC12 91475,c1(C(=O)NCCN(c2ncnc3scc(Br)c23)CCC)cnc2ncnn2c1C 91476,c1(C2N(C(=O)N(C3CC4(C3)CC4F)CC3(F)CCOCC3)CC2)ccccc1F 91477,C1(C(N2C3CN(C(C4CSCC(=O)N4)=O)CC2C3)=O)CCCC2(CCC2)O1 91478,c1(CC)c(C(=O)NCCN(C)C(C2CCCN2C2CC2)=O)cnc2ncnn12 91479,C(CC(C)C(=O)NC(CN(C)C(c1cc(CC)c(CC)o1)=O)CC)=CCC 91480,c1(C(N(CCCNC(=O)C(C(C)O)N(C)C)CC)=O)ccc(S(=O)(=O)CF)nc1 91481,Cc1nc(C=CC(=O)NCC(C)CNC(=O)C=Cc2nnn(C)n2)cs1 91482,Cc1cnn(CC(=O)NCC2CC(F)(CNC(c3ccc(C(C)(C)C)[nH]3)=O)C2)c1 91483,N1(CC(C)C)CCC(NC(NC(Cc2ccccc2)C2CC2C(=O)O)=N)CC1 91484,C1(NC(N2C(Cn3cc(C4CCN(C)C4=O)nn3)CCC2)=O)CCc2nccn2C1 91485,c1(OC)c(O)cc(C(=O)NCC2CC(F)CN2C(=O)C(C)OC)cc1C#N 91486,c1(N2CC(C(=O)Nc3nc(C(F)(F)F)cs3)SCC2)ccn2ncc(I)c2n1 91487,C(C(CCO)NC(c1cc(CNC(=O)CCCC2CC2C)ccn1)=O)OC 91488,C(=O)(C(C)(C(C)C)NCC1CC1)OCC(C)SC 91489,C(=O)(C(F)C(C)(C)O)NCCOC1CCN(C(CC2(C(=C)F)CCC2)=O)CC1 91490,C1(C)(NC(C(CC)n2cccn2)=O)CCCN(C(c2ccc(C)n2C)=O)C1 91491,N1(C(C(C)(C)CS(C)(=O)=O)=O)CCC2CCCN(C(=O)CSc3cccs3)C2C1 91492,CC1CN(C(C2(C)CCCN2C(=O)Cc2cncnc2)=O)CC1N=[N+]=[N-] 91493,C12CCN(C(Cc3ccccc3OC(=O)NCC3CC3)C1)C2=O.C(C)(C)(C)OC 91494,Cc1nn(CC(=O)NCC2(O)CN(C(=O)CSCc3ncc[nH]3)C2)c(=O)n1C 91495,C1(C(=O)OC)(NC(=O)Cc2c(I)ccnc2F)CC(C)(C)OC(C)(C)C1 91496,C1(C(=O)NC(C)(CO)c2nn[nH]n2)CCC(C(N)=O)CC1 91497,N1(C(c2cccc(S(C)(=O)=O)c2)C(=O)NC)CCCC2(CC1)CNC(=O)C2 91498,N1(C(c2c(C)cccc2Cl)=O)CC2(C1)OC1(C)CC2(NC(=O)CCF)C1 91499,Cn1nc(C(F)F)cc1C(=O)NC(c1ccccc1)CNC(C1CC2CC1CO2)=O 91500,C(=O)(CCC[N+](=O)[O-])N1CCC(C)C1CNC(=O)C(c1ccccc1)C1CC1 91501,c1(C(N2CCCC(CCCCNC(=O)C3CC3)C2)=O)cnn2c1OCCC2 91502,c1(N2C(C(=O)NCc3nccn3C)CC(C)C2)ncc2ccc(Br)cc2n1 91503,c1(N2C(CNC(C(C)C3CC3)=O)CCCC2)ncnc2sccc12 91504,N1(C(C(C(CC)CC)F)=O)CCC2(CCN(C(c3cccc(F)c3)=O)C2)C1 91505,c1(NC(c2ncn(C)n2)C)ccc(S(=O)(=O)NCC2CSCCO2)cc1Cl 91506,C(=O)(C1=CCCSC1)NC(C(=O)NCc1c(CC)cccc1)C1CCCC1 91507,c1(C(N2CCN(c3nc(C)c(F)cn3)C(CC#N)C2)=O)cc(F)c(C)c(Br)c1 91508,c1(C(=O)NC2C3(CN(C(CCNC(C)=O)=O)C3)CC2)cccc2c1OC(F)(F)O2 91509,CC1CCN(C(=O)CCC2(C)CC2(F)F)CC1NC(C1CC=CCC1)=O 91510,N1(C(CN(CCC)C)=O)CCC(NC(c2cc(C(C)(C)C)on2)=O)CC1C1CC1 91511,C(=O)(C(C)(C)C(C)NC(=O)Cn1ccc(C)c1)NCCCCCOC 91512,c1(C(N2CC(N(C(C3(C)N(C(C)=O)CCC3)=O)C)C2)=O)ccc(P(C)(C)=O)cc1 91513,C1(C(N(CCNC(C2CCCN(C(C)=O)C2)=O)C(C)C)=O)CCCCS1(=O)=O 91514,C=CC(C)(O)CC(=O)NC1CCN(C(c2occc2Cl)=O)CC1CO 91515,c1(-n2cc(NS(CC)(=O)=O)nn2)ccc(OCCN(C)C)cc1 91516,c1(NCc2cc(C(=O)NCCCN(C)C3CC3)no2)nccnc1N 91517,c1(-c2n(CCOC)c(N3CC4CCC3C4)nn2)ccc2cn(C3CC3)nc2c1 91518,CC(C)(C)C1=NOC(C(N2CCOC(CNC(c3nocc3Cl)=O)C2)=O)C1 91519,CCCCC(C(=O)NC)NC(C1CC2CCC1O2)=O.C1(=O)CCCCCN1 91520,N1(C(CCCCOC)=O)CC(F)(F)CC1C(N1CCC1COC)=O 91521,C(CC(O)CC(=O)N1CCCC(NC(C2(C)CCOCC2)=O)C1)SC 91522,C1(C)(C(N2CC(C(=O)NCCNC(CC)=O)C2)=O)CCOC(C)C1 91523,C1(CNC(c2c(SCC)cccc2)=O)CCCCN(C(C2CC2(C)C)=O)C1 91524,C1(O)(COC)CCCN(C(C2CCCN(C(=O)C#CC(C)(C)O)C2)=O)CC1 91525,c1(C(N2CC=CC(NC(C(C)(CO)OC)=O)C2)=O)cccc(C)c1C#N 91526,C1(CCC(=O)N(C2CC(CNC(=O)CCCC3CC3)C2)C)CCC(=O)C1 91527,C1(C(C(CCCCC)=O)=O)CC(C(=O)NC(C)CC(=O)NC)=NO1.NCO 91528,C1(NC(C(CC)(F)F)=O)CN(C(=O)CCN2CCC2)CCC1O 91529,C(=O)(C1=NOC(CNC(c2coc3c2COC3)=O)C1)N(C(CO)CO)C 91530,c1(C(=O)NC(C(C)NC(CCOC)=O)CO)cc(C)c(OC)c(Cl)c1 91531,N1(C(c2c(C(C)C)con2)=O)CC(CNC(=O)C=CCO)CC(C)(C)C1 91532,c1(N(CCC)C(C2(C)CCCN2C(C)C)=O)nc(SC)nc(C)c1Br 91533,C1(NC(CC2C(C)(C)C2)=O)CC1C1CCCN(C(c2ncn3cccnc23)=O)C1 91534,c1(N2C(CN3CCN(C)CC3)CCC2)nc(=NC2CC2F)[nH]c2cccc(F)c12 91535,C1(NC(C(N2C(=O)CCC2=O)C)=O)C2CC1N(C)C2.C1(N(CC=O)C)CCCC1 91536,C1(C(=O)NC(CN(C(=O)Cc2cc(Cl)ccc2O)C)(C)C)CC(C2CC2)=NO1 91537,N1(C(C)C)CCN(C(=NCC2CCCCC2C)NCc2ccc(F)cc2)CC1=O 91538,N1(C(C(CC)SC)=O)Cc2n[nH]cc2C1C(=O)N1CC(C)(C)C1 91539,N1(C(C=CCCC)=O)CC(CNC(=O)C(C)CC(F)F)C(C)(C)C1 91540,N1(C(C2C(C)OC(=O)N2)=O)CC(NC(=O)CCc2ccccc2Cl)CC(C)C1 91541,CCC(O)CC(=O)NCC(C)C(=O)NCCc1ncccc1C 91542,c1(C(=O)NC2C(NC(C(CC)(C)OC)=O)CCCC2)cnc2[nH]cncc1-2 91543,C(C(CNC(C1CCC12CCC2)=O)C(F)(F)F)NC(Cc1[nH]c(=N)sc1)=O 91544,C(C(=O)N(C)CC1COCCN1C(C1(N2CCCC2)CC1)=O)(C(C)C)OCC 91545,c1(C(N)=O)ccc(C(=O)NCCC2CCN(C(C3CC=CCC3)=O)C2)cn1 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91564,C(=O)(C(F)C(C)(F)F)NC(C(C)C)CCNC(c1ocnc1C1CC1)=O 91565,C(=O)(C1=CC2CCCCCC12)NCCCC(C)NC(c1cc(C(C)C)on1)=O 91566,N1(CC)CCCC(C(N2CC=CC2CNC(=O)C=Cc2ccc(Br)s2)=O)C1 91567,c1(C(N2CCC(N(C(=O)CC3CC4CCC3O4)C)CC2)=O)cc2n(n1)CCOC2 91568,C1(CNC(NC(CC(F)F)C)=NCCc2cnsc2)Cc2ccccc2O1 91569,c1(C(N2CC(N(C(=O)C(F)CC3CCC3)C)C(O)CC2)=O)nccn2ccnc12 91570,N1(C(Cc2ccn(CC)n2)=O)CC2CN(C(=O)C=Cc3cccnc3C)CCC12 91571,C(C)(C(C)(C)C(=O)NCCC(O)C(F)(F)F)NC(CC1(CC)CCC1)=O 91572,N1(C(C2=NNC(=O)C2)=O)CC2CCCC(NC(c3noc4c3CCCC4)=O)C2C1 91573,Cc1ncnc(C)c1C(=O)NCC=CCNC(C1CC(c2ccccc2)CO1)=O 91574,c1(OCCCC)ccc(CN(C=O)CC(N2CCC(COC)C2)=O)c(F)c1F 91575,C1(COC)CC(CNC(=O)CC2CC(=O)NC2=O)N(C(c2cc(Cl)c[nH]2)=O)C1 91576,N1(C(CC(C)OC)=O)CCN(C(=O)Cn2nccc2C)CCC1C 91577,C1(C#N)(OC)CC(C(=O)NCC#CC(=O)NCC2CC=CCC2)C1 91578,C(=O)(C(F)CCC(C)(C)C)NCC#CC(N1CCCC(C)C1CO)=O 91579,N1(C(C(COC)N(C)C)=O)CCN(C(c2cn(C)c(=O)n2C)=O)C2COCC12 91580,N1(C(CN)=O)CCC2(CC1)CC2NC(c1cc2ncccc2[nH]1)=O 91581,CC1(C)CC(CO)CN1C(=O)C1=NOC(CNC(=O)C=CC2CCCCC2)C1 91582,N1(C(COCC(=C)C)=O)CC2CCN(C=O)C(C2)C1.c12ccccc1O2 91583,CC(C)(C)C(=O)N1CCCC1CC(=O)NC1CCN(C(c2cscc2C(F)F)=O)C1 91584,C(C(=O)N1CC(CNC(c2ccc(-c3cc[nH]n3)s2)=O)C1)(C(C)C)OCC 91585,c1(CNC(=O)C(c2cccnc2)NC2CCCC2)ccc2nonc2c1 91586,c1(C(=O)NCCC2(O)CCCN(C(c3c(=N)[nH][nH]c3)=O)C2)nc2c(s1)CCCC2 91587,CC1(CNC(=O)C(=O)NC(CCC#N)c2ccccc2)COc2ccccc2O1 91588,O(NC(=O)C1(N(C(=O)C=CC(C)(C)C)C2CC2)CCC1)CCC=C 91589,O=[N+]([O-])c1cccc2c(N3CCN(CCCO)CC3)nc(Cl)cc12 91590,C1(O)(CNC(C2(c3cccc(C)c3)CCC2)=O)CCCN(C(C2CC2(C)C)=O)C1 91591,c1(OC)ccc(S(N)(=O)=O)cc1NC(C1CSCCN1C(c1csc(Br)c1)=O)=O 91592,C=CC(C)(CCOC)C(=O)N1CCCN(C(c2cc(COC)on2)=O)C(CO)C1 91593,N1(C(c2c(C)coc2)=O)CCC(CC(C)NC(=O)CC2CC23CC3)CC1 91594,c1(C(=O)NCC(C23CCC(CC2)C3)O)ccccc1Br 91595,N1(C(C(C)SCCCC)=O)CC(C2CN(C(c3cnc(=N)[nH]c3)=O)C2)C1 91596,N1(C(C2C(C(C)C)C2)=O)CCCN(C(c2ccc(CCF)cc2)=O)CC1 91597,c1(C(=O)NC2CCC(N(CC=C)C(C3CCCO3)=O)C2)ccc(C=CCO)cc1 91598,C12CCC1CN(OC)C2.c1(CN(C=O)Cc2c(C)cccc2)cnc2n1CCC2 91599,c1(OC)cc(OC)c(CNC(=O)CS(=O)(=O)CC2CC3CC3C2)cc1F 91600,CC1(C)C(NC(C2CC(F)(F)C2)=O)C(C)(C)C1NC(c1cncnc1C1CC1)=O 91601,c1(COC(=O)Cc2nnsc2Cl)nccn1-c1ccccc1 91602,c1(CC)cc(N)ccc1C(=O)NC1CCCCC1NC(=O)C(N)=O 91603,N1(C(C(C)C)=O)CCC(CC(C)NC(C2CCCN2C)=O)CC1 91604,N1(C(C=CC(=O)N(C)C)=O)CCCC1C(=O)NCCc1ccncn1 91605,C1(NC(CC2C(C)(C)N(C(=O)Cn3[nH]cnc3=N)CC2)=O)CCC(C2CC2)CC1 91606,C1(C(=O)Nc2ccc(COC)cc2)CC1C1CN(C(c2cn(C(C)C)cn2)=O)C1 91607,c1(CN(CCCC)C(=O)Nc2ncc(F)nn2)ccc(F)c(F)c1 91608,c1(C(CO)NC(C(c2ccccc2Cl)(C)O)=O)cc(Cl)cc(Cl)c1 91609,c1(C(=O)NCC2OCC(CNC(=O)C=Cc3ccccn3)C2)cc(=O)c(O)c[nH]1 91610,C(C)(CNC(=O)Cn1cc(C(F)F)nn1)(CC(C)C)NC(C(CCOC)OC)=O 91611,Cc1coc(C)c1C(=O)NCC(c1ccccc1)NC(=O)CCC1CCCN1C 91612,C1(C)(C(N2CC(CC(=O)NC3CC3(C)C)(OC)C2)=O)CCN(C)CC1 91613,Cc1cc(O)nc(C)c1C(N1CCC2(C1)CN(C(C1(C)CCCOC1)=O)C2)=O 91614,C=C(CC)CN=c1nc(N2CCCN(C(=O)C3CC3)CC2)c2c([nH]1)CCC2 91615,CC1CCc2[nH]nc(C(N3CCC(NC(=O)C4=CCSC4)C3C3CC3)=O)c2C1 91616,C1(NC(c2cccc(OC(F)F)n2)=O)CCOC(CNC(C2CC=CC2)=O)C1 91617,c1(C(C)CNC(=O)N(C2CCOC2)CCON)ccccc1Cl 91618,C1(C(=O)NC(CC(CC)C)C)CN(C(=O)C(=O)NCC2CC2)CCC1O 91619,CCS(=O)CC(=O)NCCCCCNC(C1(F)CCCOC1)=O 91620,c1(OCC(=O)NCC2C(NC(COCC)=O)C2)cccc(C(N)=O)c1 91621,c1(C(n2nnnc2C2(NC3CS(=O)(=O)C3)CCC2)C)ccc(F)c(Cl)c1Cl 91622,C1(NC(c2c(C#N)scc2)=O)CCCC(NC(C2CC2c2ccccc2)=O)CC1 91623,C(c1ccccn1)=C(C(N1CCC(N(C(C2CC(C)(O)C2)=O)CC)C1)=O)C 91624,Cc1cnc(C=CC(=O)N(C)CC2CCN(C(C3CCN3C3CCCC3)=O)C2)[nH]1 91625,C12(C(N(C)CC3CCN(C(C4CC=C(C)C4)=O)CC3)=O)CCCCN1CCC2 91626,C(CC(C)(C)C(=O)NCC(CC)NC(c1ccccc1NC(=O)CC#N)=O)OC 91627,N1(C(CN(C(C#CC2(CC)COC2)=O)C2CC2)=O)CCCC2CN(C)CC12 91628,C1(N(C(=O)CCC2CC(F)(F)C2)CC)CCCN(C(=O)C(C)CNC(N)=O)C1 91629,N1(OC)CCCC(Cc2cn(CC(C)NC(C3CN(c4nncs4)C3)=O)nn2)C1 91630,C1(C(N2CCCC(CNC(Cc3c(C)noc3Cl)=O)C2)=O)COC2(CCC2)CO1 91631,N1(C(C2(CC)CCC2)=O)CCC2(CCCC2NC(c2c[nH]c(=NC)s2)=O)C1 91632,N(C(=NCCCn1cccn1)NC(c1ccc(F)c(F)c1)C)C(C#C)CC 91633,N1(CCNC(c2n(CCC)ncc2)=O)CCN(C(c2cc(CC)ccn2)=O)CC1 91634,C1(NC(C2CC(C(F)F)C2)=O)CCCCN(C(=O)C(O)C(F)(F)F)C1 91635,c1(C(N(CC(C)O)CCNC(C2CC(N(C)C)C2)=O)=O)nnn2c1CCCCC2 91636,c1(OC)ccc(Br)c(F)c1CN1CCOC(C)CC1 91637,c1(CC(=O)NC2CC(NC(C3CCCCS3(=O)=O)=O)C2)ccc2ncccc2c1 91638,C1(C(C)C(=O)NC(C)CCO)CCN(C(=O)C(C)(C)N2CCCC2)C1 91639,C(C)(CO)(C(=O)N(C1CN(C(c2cncc(Cl)c2)=O)C1)C)NC(C)=O 91640,CC1CN(C(=O)Nc2ccncc2Cl)CCN1CCN1CCOCC1 91641,Cc1cc(Cl)cc2cc(C(=O)N(CC(O)CNC(C3CS(=O)(=O)C3)=O)C)[nH]c12 91642,C(=O)(C1=CCCOCC1)NCC1C(Nc2ncc(C(=O)OC)c(C)c2)CCCC1 91643,N1(C(C(C2CC2)OC)=O)CC(C)(OC)C1.C(CCF)N(C(=O)NC)C 91644,CC(C)C(C)CC(=O)N1CC(C(=O)NCCCCn2ccnc2)CC(C)C1 91645,N1(C(CCC(=O)NC)=O)CC(NC(c2c[nH]c(C)c(Cl)c2=O)=O)C2(CCC2)C1 91646,N1(C(c2cn(CCOC)nc2)=O)CCC2(CC(NC(=O)C3=NNC(=O)C3)C2)C1 91647,C=CC(C)(O)CC(=O)N1CCC(c2cn(CCN(C)C(C)C)nn2)CC1 91648,C1(C(=O)Nc2nnc(CCC)s2)CCN(C(c2ccc(SCC)cc2)=O)C1(C)C 91649,c1(SC)ccc(CCCC(N2CC(N(C(=O)C=CCN(C)C)C)C(F)C2)=O)cc1 91650,N1(CC(CC)CC)CCC(C2CCN(C(c3ccc(C)o3)=O)CC2)C1 91651,C=CCCCCCCC(=O)NCC(=C)CCNC(C1CCCCC12CCC2)=O 91652,c1(CC(=O)N(C(C)CNC(c2ccc(C(=O)C3CC3)s2)=O)C)ccc(Cl)nc1 91653,c1(NC(C(C(C)NC(=O)C(C)(Cl)Cl)C)=O)cc(O)cc(F)c1 91654,N1(C(C(C)OC)=O)CCCC2(CCCN2C(c2ccnc3c2nnn3C)=O)C1 91655,c1(C(N2C(C(=O)O)C=CC2)=O)ccc(S(=O)(=O)N2CC3CCC(C2)NC3)cc1 91656,c1(C(N2CC3C(CNC(CCn4c(C)cc(C)n4)=O)C3C2)=O)ccc(Cl)cc1O 91657,c1(C(=O)NC2CCC(N(C(c3nccc(OC)c3)=O)C)C2)ccc(C)c(C)c1O 91658,C(=O)(C1CCCc2scnc21)N1CCC(N(C(=O)CC2C=CCCC2)CC)CC1 91659,c1(CCCNCCNC(=O)NCC(c2ccccc2)CO)ccc(Cl)s1 91660,C1(C(=O)NCCCCNC(C(CC)n2cncn2)=O)CCC2(CCOCC2)CO1 91661,C1(COC)CN(C(c2ccc(Br)nc2F)=O)CCN1Cc1scnc1Cl 91662,c1(CNC(c2cc(C)on2)=O)ccnc(C(N2CCC(C(C)O)C2)=O)c1 91663,C#CCCCC(=O)N1CC(NC(C2(c3cncc(Br)c3)CC2)=O)C(F)C1 91664,Cn1nc2c(c1C(=O)NCCC1CC1)CN(Cc1c(F)ccc(O)c1F)CC2 91665,S(=O)(=O)(c1cccc([N+](=O)[O-])c1C#N)NC(COCC)CC 91666,N1(CC(=O)Nc2snc(SC)n2)CC2CCC2(CC(=O)O)C1 91667,Nc1cc(C(=O)NCc2cc(O)nc(CNC(=O)C=CCO)n2)cc(O)c1Cl 91668,C1(C(=O)NCC(C)(CO)NC(c2cc(F)n[nH]2)=O)CC2CCCC(C1)C2 91669,C(=O)(C1=CC2(CCOC2)C1)N(CCNC(C1(C)CC2(CC(=O)C2)C1)=O)CC 91670,CC1(C)CCCC(CC(=O)NCC2CCCC(NC(c3sccc3CO)=O)C2)O1 91671,C1(OC)CCCC(CC(=O)Nc2cccc(C(=O)C(F)(F)F)c2)C1 91672,c1(OC)cccc(C=CC(=O)NCCCNC(C2(F)C3CCCC23)=O)c1 91673,C=C(Br)CC(C)(C)CNCc1csc(Cl)c1Cl 91674,CC(C)(O)C(C)(C)CNC(C1C=CC(NC(C2(C)CCCO2)=O)C1)=O 91675,N1(C(CC(C)=C(C)C)=O)CCC2(CC1)CC(CNC(c1ncn(C)n1)=O)C2 91676,C1(OC)(CNC(=NCc2ccnn2C)NCC2CC(O)CCO2)CCSCC1 91677,C(=O)(CCCCC(=O)N1CCCC(CCCCNC(=O)C(C)CC#N)C1)NC 91678,c1(C(=O)NCCOC)ccc(NC(=O)C(=O)NC2CCCCC2CCO)cc1 91679,CCCCC(O)C(C)C(=O)N1CCCCC1CC(=O)NC1CC(OC(C)C)C1 91680,c1(C(N2CCC(NC(CNC(C)=O)=O)C(CO)C2)=O)cc2nc(Cl)ccc2o1 91681,C1(CNC(=O)Cc2csc(S)n2)C2CN(C(=O)Cc3nncs3)CC12 91682,C(C)(C)(CC(F)C(=O)N1CC(C)(N(C)C)C1)NC(C(CCC)F)=O 91683,c1(NCC(CC(=O)OC)(C)O)cnc2ncnn2c1.C1(C2(OC)CC2)C(=O)N1 91684,N1(C(CCc2n(C)ncc2)=O)CC2CC2C1C(=O)NCc1nc(N(C)C)n[nH]1 91685,Cc1nc2ncc(C(=O)NC3CC(NC(C4(C)CSC4)=O)C3)c(=O)n2[nH]1 91686,N1(C(=O)NCCc2cccc3[nH]ccc23)CCc2nc(O)cc(Br)c2C1 91687,C1(CNC(C2(C(N)=O)CCCC2)=O)CCCC2(CCC2)O1 91688,c1(CCC(=O)NCCC2CN(C(C3CC4CCC4C3)=O)CCO2)cccc(O)c1 91689,C(CC(C(=O)N1CC(O)C1)NC(C1C(C)C1C)=O)=CC 91690,c1(C(N2CC(C)(NC(c3cn(CC(CC)O)nn3)=O)C2)=O)ccc([N+](=O)[O-])[nH]1 91691,C=CCC(C)C(=O)N=S(C)(=O)c1cnn2c1CN(C(=O)CCCCO)CC2 91692,CC1(NC(=O)CC2CC23CC3)CCCN(C(c2cscc2Cl)=O)C1 91693,C12(SCC(=O)NC3C(NC(C(c4ccccc4O)OC)=O)C3)CCN(CC1)C2 91694,C=CCCC(C)(C)NC(=O)CC1(NC(=O)CC2CCCOCC2)CCC1 91695,CC1(C)C(C(=O)NC(C2CCCCC2)C(N2CCC(F)(F)C2)=O)C1(F)F 91696,S(=O)(=O)(c1ccc(Br)cc1NCc1ccc(-c2nc[nH]n2)cn1)N(CC(=C)C)C 91697,N1(C(C(=CC2CCCC2)C)=O)CC2CCOC2(CNC(c2cncc(C)n2)=O)C1 91698,N1(C(CCN(C)Cc2ccccc2)=O)CCOCC(NC(=O)C(O)P(C)(C)=O)C1 91699,c1(CN(C)C)ccc(C(=O)NCC2CN(C(=O)CC3CCCCO3)CC2C)nc1 91700,CCCC(CCC)C(=O)NC1CC(O)CN(C(=O)C(C2CCOCC2)F)C1 91701,N1(C(c2n(C)nnc2)=O)CCC2(NC(c3ccncc3Br)=O)CCCC12 91702,C(=O)(C(CC(F)F)C1CCC1)NCCN(C(C(C=C)(C)O)=O)CC 91703,N1(C(C(C)=CC(C)(C)C)=O)CCC(C)(C)C1C(=O)NCc1nc(C(N)=O)no1 91704,CC(C)C(F)C(=O)NC1CCCC(C(=O)NCc2cn(C3CCC3)nn2)C1 91705,C1(C(=O)NCc2c(C(=O)NCC(C)O)scc2)CC(=O)CCO1 91706,C1(N(C(=O)CC2CSCCS2)CC)CC2CCC(C1)N2C(=O)Cc1ccsc1 91707,N1(C(C2CC(CCNC(=O)COCC3CCC3)C2)=O)CCOCC2(CC2)C1 91708,c1(C(N2CCC(O)(C(=O)OC)CC2)C(=O)NCCOCC)nc(Br)c(C)cc1Cl 91709,C#CCCN=C(NCC(C)Cc1cccs1)NC1CC(CNC(=O)OC(C)(C)C)C1 91710,C1(CC(=O)N(CCNC(C2CCN(CC(F)(F)F)C2)=O)CC)CCCOCC1 91711,Cc1cc(C(F)(F)F)cc(C)c1C(CC(N1CC(C)(C)C(C(=O)O)C(C)(C)C1)=O)=O 91712,c1(C(=O)OC)ccc(C#N)c(NC(c2cc3ccccc3o2)OC)c1 91713,CCN=c1[nH]c(C)c(C(N2CCCCC2CNC(C2CCNC2=O)=O)=O)s1 91714,c1(C(N2CC(C)N(C(c3cnn4ccsc34)=O)CC2)=O)cccc2ccsc12 91715,CC1CC(CNC(C2(C(F)F)CCC2)=O)CN1C(=O)COc1ccccc1Cl 91716,Cc1cc(=NC(=O)CSCC(N2CCN3C(=O)OCC3C2)=O)[nH]o1 91717,Cc1ccc(C)c(SCC(=O)NCCCC(C)NC(=O)Cc2nccs2)c1 91718,C1(C(N2CCC(N(C(CN(C(C)=O)C)=O)C)C2)=O)COCCN1C 91719,N1(C(C)=O)CCC(NC(c2cc(C(C)C)nnc2O)=O)CC1C 91720,C=CC(CCC)CC(=O)N1CCOC(CNC(=O)CCOCC(F)F)C1 91721,n1(CC)cc(Br)c(C(N2CC(NC(=O)C=Cc3cncn3C)C3CC23)=O)n1 91722,c1(CC)nc(C)c(C(=O)NCCC2CCC(NC(=O)Cc3cccn3C)C2)s1 91723,N1(c2c(C(=O)OC)c(OC)ncn2)CC2CN(c3ccccc3)CC2C1 91724,c1(C(=O)NCCCNC(C2CC(O)C(F)C2)=O)cncc2c1CCCC2 91725,c1(C(=O)NCCC(CCNC(C)=O)C)c[nH]cc(Br)c1=N 91726,N1(C(C2(C)CC2(F)F)=O)CC(OC)C(NC(c2nc(C(=O)OCC)sc2)=O)C1 91727,C(CCC(C)(C)NC(=O)C(C(C)OC(C)(C)C)N(CCCSCC)C)OC.C(C)(C)C 91728,Cc1cccc(S(=O)(=O)CCCN2CCn3c(C(F)F)nnc3C2)c1 91729,C(=O)(C1CC=Cc2ccccc21)NC(C1CCCN1C(=O)CSCC(N)=O)C 91730,N1(C(C(C=CC)O)=O)CCCCC(NC(=O)CN(c2ccc(Cl)cc2)C)C1 91731,C(=O)(C1=CCCCC1C)N1CC(O)(CN(C(CCCOC)=O)C)C1 91732,C1(CNC(c2c(COC)cco2)=O)CCCN(C(=O)C(F)(F)c2csc(Cl)c2)C1 91733,C1(CNC(C(CC)SC)=O)CCCN(C(=O)CSc2ncccn2)CC1 91734,N1(C(=O)Nc2c(C(=O)NC)n(C)nc2)CCC2NC(=O)NCC2C1 91735,N1(C(C(CC)C(C)(F)F)=O)C2CCCC1CN(C(=O)C(C)(C)S(C)(=O)=O)CC2 91736,C1(CNC(COCCC)=O)CC2COCC2N1C(c1c(F)ccnc1F)=O 91737,c1(C(N2CC3CC2CC3O)C(=O)NCCCC)ccc(C)c(Cl)c1 91738,C(=O)(C(O)C1=CCCCC1)NC1(C)CN(C(CC2CC(CC)OCC2)=O)C1 91739,C1(NC(C2(CC)CCCCC2)=O)CN(C(=O)CC2CCN(C)C2)CC1N=[N+]=[N-] 91740,N1(C(C(C(CC)O)C)=O)CC=C(CCNC(c2ccnn2CC2CC2)=O)CC1 91741,CC1(C)CCN(C(=O)CC2CCC(=O)NC2)C1C(=O)NC1(CF)CCC1 91742,CC(O)(CC(=O)NC1CC1C(=O)NCc1cc(F)c(Cl)cc1Cl)CC(=O)O 91743,C(=O)(CC(C(C)CC)NC1(CC)CCOC1)N(CCCCO)CC#C 91744,C1(C(=O)NC(=O)Cc2cccs2)(CO)CCN(C(=O)CSc2ccncc2)CC1 91745,Cn1ncc2ncnc(NCCNS(C)(=O)=O)c12.C12CC(CO1)C(=O)NC2 91746,c1(C2(NC(=O)C(c3cccc(C(F)(F)F)c3)O)CC2)cc(F)c(F)c(F)c1 91747,C1(NC(C2CCCC2CNC(=O)C(c2ccccc2)O)=O)(OC)CCC1COC 91748,c1cc2[nH]c(=NCC3CCCOC3)nc(N3CCOC(CC4CC4)C3)c2[nH]1 91749,CN(CC(=O)NC1CCCCC1)N1CCC(OCCO)CC1 91750,C1(NC(CC2CC(C)C2)=O)COCCN(C(C2(OC3CCOCC3)CC2)=O)C1 91751,CC(C)(C)CC(O)CC(=O)N1CC=CC(C(=O)NCc2ccncc2)C1 91752,C1(O)(C(=O)NC2C(C(c3ccccc3)NC(CCC)=O)COC2)CC(C)(C)C1 91753,CCC(C)(CC)C(=O)NCCC(CNC(c1[nH]ccc1C)=O)OC 91754,CCCC(O)C(=O)N(CCCNC(C1CC1c1cnn(CC(C)C)c1)=O)CCO 91755,c1(CC(=O)NCCC2CCN(C(C(CSC)OC)=O)C2)ccc(C(C)(C)C)cc1 91756,N1(CC(N2C(CNC(Cc3cc(C)ns3)=O)C=CC2)=O)CCNC(=O)C1 91757,Cc1ccc(C#N)c(NC(C2C3CC2N(S(=O)(=O)c2ccncc2)C3)=O)c1 91758,c1(C(=O)NCc2cc(F)ccc2-c2ccc(Cl)c(Cl)c2)n[nH]c2c1COCC2 91759,Cc1c(F)cccc1S(=O)(=O)N1CC(O)CC1C(=O)NC(C)(CO)CO 91760,N1(C(COC2CCCC(C)C2)=O)CCN(C(=O)Cc2ccc(F)nc2)CCC1C 91761,n1(CCC)c(CN(CCCNC(=O)CC2CCCOC2)C)nnc1C 91762,c1(NC(c2ccc(C(c3ccc(C)n(C)c3=O)=O)cc2)=O)sc2ccccc2c1C#N 91763,C1(NC(c2cnc(SC)s2)=O)CN(C(c2cc(C)nc(Cl)n2)=O)CCC1C 91764,c1(C2OCCN(C(=O)NCC3(n4ccnn4)CCOCC3)C2)c(Cl)cccc1Cl 91765,C=CC(C)(CC)C(=O)NC(C1CC1C(N1CCC2(CC1)N=N2)=O)C 91766,c1(C(=O)NCCOC2CCN(C(C(C(CC)O)C)=O)C2)nn(C)c2c1CCC2 91767,C(=O)(C(O)CC(C)(C)C)N1C2CC(C(N(C3CCCC(C#N)C3)C)=O)C1CC2 91768,N1(C(c2c(C)nc(Br)o2)=O)CCCN(C(C2CC23CCCCC3)=O)CC1 91769,c1(C(=O)NCCNCc2cc3c(cc2Cl)OCCO3)ccc(C2=CCCC2)cc1 91770,N1(C(CC=C)=O)CC(NC(=O)CN(C)C(=O)C2CC2)CCC1C 91771,c1(NCCOC)cc(C(=O)NC2CCCC2NC(c2nc(C)cs2)=O)ccn1 91772,C1(C(N(C2(C(N(CC(CC)C)C)=O)CCC2)C2CC2)=O)C2CCC(F)C12 91773,C#CC1CN(C(c2cccc3ccoc23)=O)CCN1C(C1CCSC(C)C1)=O 91774,C1(OCC)CC2(C1)CC2C(N1CCC(C(C)NC(c2nocc2C2CC2)=O)C1)=O 91775,C(=O)(C(CC)CCCC)NCCC=CCN(C)C(c1cccc(SCCCC)c1)=O 91776,C12(CNC(c3c(C)coc3)=O)CCC(CC1)N2C(c1cc2scnc2[nH]1)=O 91777,Cn1[nH]c(=NC(=O)NCC2CCC3(CCC3)CC2)cc1C1CC1 91778,C1(OC)CC2CC1CN(C(=O)CC1(NC(c3cnncc3C)=O)CC1)C2 91779,c1(C(N2CC(OCCNC(CCC3CCC(C)O3)=O)C2)=O)cccc(Cl)c1 91780,C(C(=O)N=c1c(Cl)c[nH]cc1I)c1nn2c3cc(cc(F)c3)c2n1.CC 91781,c1(NCC(CC(=O)NC)C)[nH]c(=NC(C)c2nccc(C)n2)nc2ncn(C)c12 91782,c1(CC(=O)NCC(C)N(C)C(C2CN3CCC2CC3)=O)ccc(Br)cc1F 91783,c1(-n2c(C(=O)NC(C)(C)CNC(=O)CC3CCCCC3)cnn2)ccccc1F 91784,C1(NC(C2C(C)C2)=O)CN(C(c2cc(Cl)cc(Cl)n2)=O)CC1C#N 91785,C(C(C)(C)CNC(=O)N(C)C)(c1n(C(CC)(C)C)nnn1)NC1(C)CCOC1 91786,c1(C(=O)NCC(CC=C)NC(=O)C(C)(C2CC2)OC)n[nH]c(C)c1[N+](=O)[O-] 91787,Cc1cc(O)ncc1C(=O)NC1CC1CNC(c1ccc(O)c(Cl)n1)=O 91788,C1(C(=O)NCCCC(C)NC(c2nn(C)cc2Cl)=O)CC12CC(C)(C)C2 91789,N1(C(c2cc(C)sc2)=O)C2CCC1CN(C(=O)CN1CCC(C(F)(F)F)CC1)C2 91790,N1(C(CC(=C)C)=O)CCC2(C1)CN(C(c1ccnn1C(F)F)=O)C2 91791,Cc1nsc2ncc(C(N3CCCC4(C3)CN(C(C3CCCOC3)=O)C4)=O)cc12 91792,c1(C(=O)OC)cc(Cl)c(N2CCCC(N(C)C(C3CC=CCC3)=O)CC2)nc1C 91793,CC1CCC(C)(C(=O)NC2CC(NC(c3cncc(N)n3)=O)C2)C1 91794,c1(NC(C2CC(O)CN2Cc2ccc(Br)nc2)=O)c(F)cc(F)cc1[N+](=O)[O-] 91795,c1(CC2(CN(C(=O)CSF)CCNC(C3CC(C)(O)C3)=O)CC2)ccc(N)cc1 91796,c1(C(=O)NCC(C(C)C)NC(c2cc(OC)ncn2)=O)sc2cccnc2c1Cl 91797,C(CC(=O)NC12CC1CN(C(c1ncoc1C1CCC1)=O)C2)(C(C)C)OCC 91798,C(CCCCCNC(C1CC(CN(C)C)C1)=O)NC(C)=O 91799,c1(C(N2C(C)CN(C(=O)CC3=CCCC3)CC2)=O)cc2cc(Cl)cnc2[nH]1 91800,c1(CC)ncncc1C(N1CCC(CNC(C23COC(CO)(C2)C3)=O)C1)=O 91801,c1(C(c2nnnn2C(C)CCC)NCC(CC=C)(C)C)c(F)cnc(Cl)c1C 91802,N1(C(c2cc(C)[nH]c2)=O)CC23CCCC2(C1)CN(C(=O)CCc1ncccn1)C3 91803,CN1CCc2cc(CC(=O)NC3(CCNC(=O)CCOCC4CC4)CC3)ccc21 91804,c1(C(N2CC(F)(C(=O)NCC(C)CCl)C2)=O)csc2ccccc12 91805,C(N=c1[nH]c2cc(Br)ccc2o1)C1C(C)CN(C(C2CCOC2)=O)C1 91806,c1(OC)ncnc(N2CCC(N(C(=O)Cn3ccnc3C(C)C)C)C2)c1C 91807,N1(C(c2c(C)cc(Cl)cc2)=O)CCCC(C2CCN(C(=O)C(O)C(C)C)CC2)C1 91808,N1(C(c2ccc(C3CC3)s2)=O)CC2CCC(C1)N(Cc1scnc1C(F)(F)F)C2 91809,c1(C(N(CC(c2ccccc2)CC)CC)=O)ccc(C(F)(F)F)s1 91810,N1(C(CC(C)SC)=O)CCOCC1CC(=O)NOC1CCC(O)C1 91811,CCC(C(=O)N1CC(C)C(C)(CNC(C2CC(O)C2)=O)C1)C(F)(F)F 91812,CCC(C)C(CN(C)C)NC(=O)C(F)CC1CN(C(c2cnn(C(C)C)n2)=O)C1 91813,C1(NC(c2cc(C)[nH]n2)=O)CC(O)CN(C(c2ccc(-c3cnn(C)c3)o2)=O)C1 91814,c1(NCCN2CC(OC)C2)cc(=NC2CCOc3ccccc3C2)[nH]c(C(C)C)n1 91815,C1(CCNC(C(C)C2CC2)=O)CCC(NC(=O)CN2CCOC2=O)C1 91816,c1(C(=O)NCC2CC(NC(C=Cc3n(CC)ccn3)=O)C2)c(Cl)ccc(F)c1F 91817,c1(OC)c(C(=O)NCC(C)N(C(=O)COC2CCOC2)C)cc(Br)cc1F 91818,CN1CCOCC1CC(=O)NC12CC1CN(C(c1cn(-c3ccccc3)cn1)=O)C2 91819,C1(NC2CN(C(COCC=C)=O)C2)CC(F)(CNC(=O)COCC(C)C)C1 91820,c1(C(=O)NC(CCNC(c2cc(C(C)C)no2)=O)(C)C)cc2c(ccn2C)[nH]1 91821,C1(C(N2CCCC(C3N(C(c4c(C)cco4)=O)CCC3)C2)=O)CCCCC1(F)F 91822,C1(C(=O)NCC(CC)(C)O)COCCN1C(c1cc(=O)cc[nH]1)=O 91823,C=CCC(C)(C)CC(=O)NCC1CCCN1C(c1cc(C)c(C)nc1O)=O 91824,C1(CNC(C=C(CCN(C)C)Cl)=O)CN(C(=O)CC(C)(C)C)CC2(CCC2)O1 91825,N1(CC)CCN(CC(=O)NCCN(C(=O)C(N2CCN(C)CC2)C)C)CC1 91826,CC1=NOC2(C1)CC(C(N1CC(NC(C3CCS(=O)CC3)=O)C(C(F)F)C1)=O)C2 91827,C1(C(=O)NC(C(C)C)C2CCC2)(CC)CCN(C(c2c[nH]nc2C)=O)CC1 91828,N1(C(C(CCC)OC)=O)CC2(C1)SCCC2NC(=O)Cc1cnoc1 91829,c1(CNC(C2C(CNc3cc(OCC)ncn3)CCC2)=O)ccc(C)c(Cl)c1F 91830,C1(NC(c2oc(CC)c(C)c2)=O)CCC(C)(NC(c2cc(Cl)ccc2O)=O)CC1 91831,Cc1noc(C)c1CCC(=O)NC1(C)CC(NC(C2CC23CC3(F)F)=O)C1 91832,N1(CC(C)NC(=O)OC(C)(C)C)CCC2(CC1)OCCc1ccccc12 91833,c1(NC(CCC)CCCNC(=O)CCC(N)=O)ccc(S(C)(=O)=O)cc1[N+](=O)[O-] 91834,C1(C(=O)NC2C(C(C)NC(c3sccc3C(C)(C)C)=O)C2)CCc2ccnn2C1 91835,Cc1ccc2[nH]c(C(N3CCC(N(C(=O)C#CC4CC4)C)C3)=O)cc2c1 91836,n1(CC)cc(Br)cc1C(=O)NC(C1(O)CN(C(C2CC23CCC3)=O)C1)C 91837,C1(CC(=O)NCCCN(C(=O)CC2COCCN2C)CC)(OCCO)CCCCC1 91838,CC(CN(C)C(c1c[nH]c2nccc-2c1)=O)N=c1[nH]c2ccc(O)cc2s1 91839,C1(F)(C(=O)OC)CN(C(C(=O)NCCSC)c2nccs2)CC12CCOCC2 91840,O=C1NCC2(CO1)CN(C(=O)Nc1ccc(Oc3ncccn3)cc1)C2 91841,C1(NC(C2CCCNS2(=O)=O)=O)CCN(C(C2CCCSC2)=O)CC12CCC2 91842,CC(C(F)C(=O)N1CCC(NC(=O)CC2CC3CC3C2)C(O)C1)C(F)(F)F 91843,C=CCC(C(=O)N1CCC(C(C)NC(C2(C(C)(C)OC)CC2)=O)CC1)NC(C)=O 91844,C1(C(=O)NC(CCC)CCO)CN(C(C2(SC)CC2)=O)CCC1(C)C 91845,c1(C(=O)NC2(C)CCCN(C(C3C(=C)C3)=O)C2)c[nH]c2ccccc12 91846,c1(NC(N2CCC(n3cc(CO)nn3)C2)=O)cc(Cl)cc2nccnc12 91847,N1(c2nc(NC3COc4cccc(F)c43)cc(C)n2)CCc2nc(C)c(O)cc2C1 91848,N1(C(C2(CCC)CCC2)=O)CCC2C(C(=O)NCC(F)(CC)CC)C2C1 91849,CCCCCCCC(O)C(F)(F)C(=O)NC1CN(C(C)=O)CC(C(F)(F)F)O1 91850,c12ccc(cc1Br)S(=O)(=O)NC1(C)CN2CCO1.C(CCCCC1CC1)OC 91851,c1(OC)c(Cl)nc[nH]c1=NCCN(C1CCC1)C(C)=O.c12cncc(n1)NC2=O 91852,c1(C2(F)CC(C(=O)NC(C)CCN(C)C(C3CC3C)=O)C2)cccc(F)c1 91853,Cc1cccc(C(N2CCC(C(N3CCCCC(C)C3)=O)C2)=O)c1I 91854,N1(C(CNC(N)=O)=O)CCC2(C1)CN(C(c1n[nH]c3c1CSCC3)=O)CCO2 91855,C(=O)(C(C)(C)CCC(C)=O)NCc1c(OC)ccc(F)c1 91856,c1(CNCC2C3CC=CCC32)cccc2c1CCC2 91857,C1(NC(CNC(CNC(C)=O)=O)=O)CCN(C(=O)CC2CC2(Cl)Cl)CC1 91858,N1(C(C(CC=C)OC)=O)CC(C)(C)OCC1CNC(c1c[nH]c(C(N)=O)c1)=O 91859,c1(C(=O)NCC(C(C)C)NC(c2ccsc2Br)=O)ccnc(C2CC2)n1 91860,c1(OC)cccc(C)c1NC(C1(CNC(c2cccn2C)=O)CCCO1)=O 91861,C1(CC=C)(C(=O)Nc2coc(COC)n2)CCN(C(=O)C=CC(C)(C)SC)C1 91862,CC1CN(C(c2csc(Cl)c2Cl)=O)CC1NC(C1CC1F)=O 91863,c1(C(=O)NC(C(=O)NC2(C)CC(O)(CO)C2)CCF)cccc2occc12 91864,C(=O)(C(=O)CC(C)C)NC(C(=O)NCC(CC)C#N)CCF 91865,C12(NC(=O)C(Cl)=CCl)COC(C1)C(NC(=O)C(O)Cc1cnc[nH]1)C2 91866,N1(C(CN(CCCCCC)C)=O)CCCC(Cc2cc(C)sc2C)C1 91867,C1(C(C(=O)N(CCN(C(C)=O)C)C)C)CCCN(C(c2cn(C)nc2C)=O)C1 91868,c1(NC(=O)N(C)C)coc2ccc(Br)cc12.n12cc(nn1)C(C1CC1)C(C)C2 91869,Cc1cc(NC(C2CC(C)(C)CN2C(c2cccc(C)c2N)=O)=O)cnc1Cl 91870,c1(C(=O)NCC2N(C(C3CCC(C(=O)OC)C3)=O)CC=C2)ccc(C)c2c1CCC2 91871,c1(CC)c(C)nc(=N)[nH]c1C.C12CC(C1(C)C)CNC(=O)C1(CC1)CC(=O)N2.CSC 91872,C1(C(=O)NCCC(CNC(=O)C(C)(C)n2cncn2)OC)CCc2c[nH]nc2C1 91873,C1(CC(=O)NCC(C(=O)OC)OC)CCCN(C(=O)C(OC)OC)CC1 91874,N1(C(C(C2CC2)SC)=O)CCCC(O)(CCNC(=O)CCC2CC2(F)F)C1 91875,N1(C(C2N(CCCC)CCCC2)=O)CCCCC(NC(C2(CC(C)C)CC2)=O)C1 91876,C(=O)(C(C(C)(F)F)OC(=O)CCc1ccc(F)c(OC)c1)OC 91877,c1(C(=O)NCC(c2cnn(C)c2)NC(C(C)C)=O)ccc(C(=O)N(C)C)cc1 91878,C1(C(N2C(C)CC(NC(=O)Cc3cnnn3C)C2)=O)CN(C)CCN(C)C1 91879,c1(C(=O)NCC(C)CO)c(Cl)nn(C)c1Cl 91880,c1(CC)cc(C(=O)N(C)CCN2CCN(C(=O)C(O)C(C)OC)CC2)ccc1F 91881,C(=O)(C(C)NC(C)=O)N(C1CCCC1)CCNC(CSCC#C)=O 91882,CCC1=NOC(CC(=O)NCCC2CCN(C(C3C(Cl)(Cl)C34CC4)=O)C2)C1 91883,c1(CC)ccc(N2CC(C(N3CCCC(CNC(=O)CO)C3)=O)CC2=O)cc1 91884,c1(C(=O)NC2CN(C(CSCC=C)=O)CC2N=[N+]=[N-])cnc2c(c1)ncn2C 91885,Nc1cccc(C(=O)NCC2CCC2NC(c2ccnnc2O)=O)n1 91886,c1(C(N2CC(C)C(C)C2)C(=O)NC(CC)C)c(Cl)nc(Cl)n1C 91887,Cc1ccc(C(CNC(=O)CC(C)(F)F)NC(c2ccn(C3CC3)n2)=O)cc1 91888,C1(CN(CCCNC(c2c(C)onc2)=O)C2CC2)CCC(C)(C)CC1 91889,N1(C(CCSC)=O)CCN(C(=O)C(c2ccc(Br)s2)C)CCC1C 91890,C1(C(=O)NC(C2CCN(C(c3cc(Cl)no3)=O)CC2)C(C)C)CN(C)CCN1C 91891,C(CCCCC(=O)NCC(O)CF)NC(C1(C(C)=O)CC1)=O 91892,C1(C(N2CCC(NC(C=CSC)=O)C23CCC3)=O)Cc2nn(C)cc2C(=O)N1 91893,CC(C)C(C(=O)N(C1C(c2ccc(F)cc2O)C1)C(C)(C)C)C(C)C 91894,c1(OCCCC(N2CC(C)C(NC(=O)C(C)C(C)(C)O)C2)=O)ccc(F)c(F)c1 91895,N1(C(C2CCCN(c3ccccc3)C2)C(=O)NC)CCOC2(CCCC2)C1 91896,N1(C(C(C)N(C(CN(CCC#C)C)=O)C)=O)CC2(C1)CC(C)(O)C2 91897,n1(CCCF)nc(-c2ccncc2)nc1-c1ccc(OCC(F)(F)F)cc1 91898,Cc1ccc2cc(C(=O)NCCCNC(=O)C(F)C3CC3)c(C)nc2c1 91899,N1(C(=O)CSC(F)(F)F)CCN(C(=O)CCC(F)(F)F)C2CCCCC2C1 91900,C#Cc1cccc(C(=O)NCc2cccc(CNC(C3CC=CC3)=O)c2)c1F 91901,C(=O)(CC(C)(C)C)NCC(=O)N(C1CCCCC1)CCCNC(C(CC)F)=O 91902,Cn1cc(C#N)cc1C(=O)NC(Cc1ccoc1)C(=O)NCCc1nccn1C 91903,C1(CNC(CCN(C(C)C)C(C2CC3CC(=O)C2O3)=O)=O)CCCC2(CC2)C1 91904,CC(C(=O)NCC(O)CNC(c1cncc(F)c1)=O)C(=O)N1CCOCC1 91905,N1(C(CCOC(CC(C)C)C)=O)CCCC1(C)CNC(C1CN(C)C(=O)N1)=O 91906,c1(CCCC)ccc(CCC(N2CC(c3ccccc3)CC2C(=O)OC)=O)cc1 91907,c1(C(=O)NC2CCC(NC(C(C(C)O)NC(C)=O)=O)C2)c(C)nc(C)n1O 91908,c1(C(N2CC3CCCCC3C2)=O)ccc2c(-c3ccc(CO)o3)cccc2n1 91909,C1(C(=O)NCCN(C(=O)C(C)SC(F)(F)F)C(C)C)CC2CCC(C1)S2(=O)=O 91910,N1(C(Cc2cn(C)nc2)=O)CCOCC(NCc2cccc(O)c2Cl)C1 91911,C12(NC(C3CCN(C)CC3)=O)CCCN(C(=O)Cc3cc(F)cc(Cl)c3)CC1C2 91912,n1(CC(=O)NC2C(NC(CC(=O)N(C)C)=O)CC2)ncn(C)c1=O 91913,c1(-c2nc(C)c(C(=O)NCC3(C)CCOCC3)s2)ccc2ccccc2n1 91914,c1(C(N2CCC(CNC(C3(C=C)CCCCC3)=O)C2)=O)nnn2ccccc12 91915,C(CC(C(=O)O)NC(=O)CCSc1ccccc1)NC(N)=O 91916,N1(Cc2c(C)onc2)CCC2(CC1)CC2C(N1CCC(CO)C(O)C1)=O 91917,Cc1c(NC2CC2c2ccccc2)ncnc1N1CCC(C)CC1 91918,CC1C(C)N(C(c2cnc(F)c(F)c2)=O)CCN1C(=O)CCc1cnccn1 91919,N1(C(c2cncc(-c3ccc(OCCC(C)C)cc3)n2)=O)CCOC(C#N)C1 91920,C=C(C)C1OCCC1C(=O)NCC12CCC(CC1)N2C(c1cnn(C(F)F)c1)=O 91921,N1(C(C(C2CC2)OC)=O)CCC(C2(NC(c3ccccc3C#N)=O)CCC2)CC1 91922,C(CNC(=O)CC(=O)NC1CC1)(CC(=O)NCC(C)CC)OC 91923,c1(C(=O)NCC2CCCN(C(CC(CC)C)=O)CC2)cc(S(=O)(=O)NC)cs1 91924,N1(C(C=C(C)c2cnn(C)c2)=O)CCC(NC(=O)CCC2CC2)C12CCC2 91925,C1(C)(CC)CC(C(=O)NCC2CC3(C2)CN(C(=O)CN=S(C)(C)=O)C3)CCO1 91926,C1(CNC(CN(CC(=O)NC(C)C)C)=O)CCCN(C(C2CC(N(C)C)C2)=O)C1 91927,C1(NC(=O)C(F)C2CCOC2)(CNC(C23CCC(C2)C3)=O)CCCC1 91928,C1(CNC(C2CC3(CCOC3)C2)=O)CCC2CN(C(c3cc[nH]n3)=O)CC12 91929,S(=O)(=O)(CCCN=c1nc2scnc2c(NCCNC(=O)NC2CC2)[nH]1)NC 91930,C1(C(N2CC(NC(=O)CC3CCCS3(=O)=O)(CF)C2)=O)CCCCC1(F)F 91931,c1(C(=O)NCC2(CNC(Cc3ccc(C)s3)=O)CCC2)cc2cn[nH]c2cn1 91932,c1(C(N(C2C(C)CN(C(=O)C(=O)C(C)(C)C)CC2)C)=O)cc2ccc(F)cc2[nH]1 91933,c1(CN2CCC(C(=O)Nc3n(C)cc(Br)n3)CC2)ccn2ccnc2c1 91934,N1(C(c2c(CC)n(CC)nn2)=O)CCN(C(C2CSC2)=O)C(CC(C)(C)C)C1 91935,Cc1cnc(N(C2CCNCC2F)C(c2ncccc2C)=O)nc1 91936,C1(COC)(CNC(=O)COc2cnn(C)c2)CCCN1C(C1CC(C)=NO1)=O 91937,N1(C(CC(COC)(C)O)=O)CCN(C(=O)CCOCC2CCCO2)C2CCCC12 91938,c1(CCCC(=O)NCC2(F)CCC(NC(C3CCC3)=O)C2)cc(Cl)ccc1Cl 91939,N1(C(C2(COCC)CC2)=O)CCC2(CC2C(N2CC(C#N)(CC)C2)=O)C1 91940,c1(C(=O)NCCCNC(C2(S(N)(=O)=O)CC2)=O)ccc(=O)n(CC2CCCO2)n1 91941,C1(NC(C2N(C(=O)NC)CCC2)=O)CCCN(C(=O)Cn2nc(C)nc2C)C1C 91942,Nc1nn2ccccc2c1C(=O)NC1CCC(O)(C(F)(F)F)C1 91943,C1(C)(CC)CC(C(=O)NCc2cc(C(=O)NC(C)Cc3cnccn3)no2)C1 91944,C(=O)(CC(C)CC(C)(C)C)N(C1CC2N(C(CC=CC)=O)C(CC2)C1)C 91945,c1(CC(=O)NCC2=CCN(C(COC(C)=O)=O)CC2)c(C)[nH]c2ccnn2c1=O 91946,CN1CCC(CCNC(C2CC(C)(NC(C3CCCCC3)=O)C2)=O)C1 91947,Cc1cc(N)c(F)c(C(N2CCCC(O)(CNC(C3(O)CC3)=O)CC2)=O)c1F 91948,C1(C#N)(C(=O)NCC(CNC(C(C)=C(CC)C)=O)OC)CCCC(=O)C1 91949,C1(NC(C(C)OCCC(C)C)=O)COC2CN(C(=O)C3=CCCCCC3)CC12 91950,c1(C(=O)NCCN(C(=O)C(C)n2cccn2)CCC)ccc2sccc2c1 91951,C(c1ccc(F)c(F)c1)=C(C)C(N1CCC(NC(=O)CCN2CCC2)C(C)C1)=O 91952,C1(N(C(C=Cc2c(C)cccn2)=O)C(C)(C)C)CCN(C(C)(C)C)CCC1C(=O)O 91953,C12(NC(c3c(OC)cc(F)cc3)=O)CCN(C(=O)CS(N)(=O)=O)CCC1C2 91954,Cc1cc(=O)n(CCC(N2CC(N(C)C(C3C4COCC34)=O)C(O)C2)=O)cn1 91955,Cc1ccc(C(N2CCN(C(=O)C(C)n3cncn3)CC2C2CCC2)=O)c(N)n1 91956,c1(COC)c(C(=O)N(CCCCNC(=O)C(CC)OC)C)sc2ccccc12 91957,C(c1csc(Br)c1)=CC(=O)NC1(CF)CCN(C(C2OCCO2)=O)C1 91958,N1(C(C2(C)CCCCC2)=O)CC(CO)C2(C1)CN(C(c1ccc(C#N)o1)=O)C2 91959,c1(C(=O)NCC(CC)NC(C(C=C)(C)O)=O)cc(OC)cc2c1OCC2 91960,c1(C(=O)NCCN(C(=O)C(C2CCCCCC2)C)CC)cncc(C2CC2)c1 91961,c1(-c2c(C)n(C)nc2)ncn2c1CN(C(c1cccc(Cl)n1)=O)CC2 91962,c1(C(N)=O)ccc(CC(=O)OCc2nccn2CCc2ccccc2)cc1Cl 91963,CC1CC(NC(C2(C(F)(F)F)CC(F)(F)C2)=O)CN1C(c1cncc(O)c1)=O 91964,C(=O)(C1=CCC(C)(C)CC1)N(CCN(C(c1ccc(OC)cc1Cl)=O)C)C 91965,CC1C2C(CCN2C(c2cn3c(n2)CCC3)=O)CN1C(=O)C1=CCSC1 91966,C1(C(=O)NC2(CNC(CCc3onc(C(C)OC)n3)=O)CCC2)OC2CCC1C2 91967,N1(C(c2c(C)n(C(C)C)nc2)=O)CCN(c2cc(OCC3CC3)ncn2)C(C)C1 91968,Cc1nc(Nc2cccc(OCC(C)C)c2)cc2nncn12 91969,N1(C(c2nc(-c3ccc(C)o3)sc2)=O)CCCC1(C)CNC(=O)C=C1CCC1 91970,Cc1cc(C(N2CCOC(C3CCOC3)C2)C(=O)NC2CCCC2)n(C)n1 91971,c1(C(N2CC(Cc3cn(CCC(C)=O)nn3)OCC2)=O)cc2sccc2cn1 91972,CC1COCC(CN(C(=O)CC2CCC(C(F)(F)F)O2)C2CC2)O1 91973,c1(C(=O)NCC(CO)NC(c2cnc(OCC)s2)=O)noc(C)c1[N+](=O)[O-] 91974,N1(C(CCC(C)OCC)=O)CCN(C(c2ccc(C)cn2)=O)CC(CO)C1 91975,N1(C(CC2(OC)CN(C(=O)CC3CCC(C)O3)C2)=O)CC2(CCOC(=O)N2)C1 91976,N#CC1CN(C(=O)CN2CCCCC2)CCN1C(=O)CCc1ccsc1 91977,C1(C2CN(C(=O)CC(C)(C3CCC3)N(C)C)C2)(NC(C(C)CF)=O)CC1 91978,N1(C(c2c(C)nc(C)[nH]2)=O)CC2CCN(C(=O)CC(O)c3ccccc3)CC2C1 91979,c1(SC)cncc(C(=O)N(C(C)CNC(=O)CCc2ccc(C(C)C)cc2)C)c1 91980,CC(C(=O)NCCC1(O)CN(C(=O)CN2CCCCC2)C1)C(C)n1cccn1 91981,CC1(C)CC(NC(C2(CO)CCCCC2)=O)CN(C(c2ncc(F)cc2N)=O)C1 91982,N1(C(c2n(C)nc(Cl)c2)=O)CCC=C(C(=O)N2CC(O)C(F)C2)C1 91983,c1(C(=O)NCC=CCNC(c2cc3n(n2)CCCC3)=O)cc2nc(Cl)ccc2s1 91984,C12(C(N3CC(=O)OCC3)=O)CCC(C(=O)Nc3cc4ccoc4s3)(CC1)C2 91985,c1(CNC(C2(C3CCCN3C(C3CCCS3)=O)CC2)=O)ccc(O)nn1 91986,C1(N(S(=O)(=O)C(C)C#N)C)CN(N2CC(O)(CC#N)C2)CC1c1ccccc1 91987,C1(NC(Cc2cc(C)no2)=O)CC2(CCN(c3ccc(C#N)cn3)CC2)C1 91988,N1(CC)CC(C(=O)NC2CN(C(c3ccccc3C(F)(F)F)=O)CC2C)CC1=O 91989,c1(C(=O)OC)ccc2c(c1)CCC2NC(=O)C(=O)NC1CCC1c1ccccc1 91990,N1(C(C(=O)NCCC#N)C2C(C)C2)CCc2ccccc21 91991,c1(C(=O)NC(COC)C)cnn2cccc(-c3c[nH]c4ncccc34)c12 91992,C=CCC(CC=C)NC(C1CCCC1NC(=O)CN(C)CCC)=O 91993,Cc1nc(C(N2C(C(=O)NCC(O)CF)CC3CC23)=O)cc(O)n1 91994,C1(C)(CCNC(C(C)C)=O)CCN(C(=O)COC2CCN(C)CC2)C1 91995,C(=O)(CCc1nccs1)NCCN(C(CNC(C)=O)=O)C 91996,C1(C(=O)Nc2cn(CC=C)nc2)CN(C(c2cn(CCO)nn2)=O)CCN1C 91997,C(=O)(C(O)(C(F)(F)F)C1CC1)N1CCC(CNC(=O)Cc2ccc(CCF)cc2)C1 91998,Cn1cc2ccc(NC(C3CC34CCN(C(=O)CCCCCBr)CC4)=O)cc2n1 91999,c1(NC(C(C)OC(c2cncc(C(F)(F)F)c2)=O)=O)c[nH]c2ccc(F)cc12 92000,c1(N2CCC(c3ncc(C)[nH]3)CC2)ccc2ncccc2c1[N+](=O)[O-] 92001,CC1CCC(CNS(=O)(=O)c2ccccc2OC(F)(F)F)Cc2ccccc21 92002,c1(C2(C(=O)NCC3(F)CC(NC(c4c[nH]cc4Br)=O)C3)CC2)ccc(Cl)nc1 92003,N1(C(CCc2ccc(C)cc2)=O)CC(N(C)C(c2ccnnc2O)=O)C2(CC2)C1 92004,C(CC(C(C)C)(c1nnnn1CC1CCCO1)NCCNC(C)=O)OC 92005,C(N=c1ccc(C#N)n[nH]1)C1CCCN(C(c2c(C)ccc(C(F)(F)F)c2)=O)C1 92006,C1(CCCNC(C2(C(C)C)CC2)=O)CCCCN1C(c1cncc(N)c1)=O 92007,C1(NC(C(c2cccs2)OCC)=O)CC(NC(c2cc(OC)ncn2)=O)CC1O 92008,N1(C(C(C)SCCCC)=O)CCC(C(C)C(=O)N(CCC2CC2)CC2CC2)CC1 92009,Cc1nc(O)nc(C)c1C(=O)NC1CC(NC(=O)COc2cccc(F)c2F)C1 92010,CCC(CCOC)C(=O)N1CCCC(C)(C(=O)NCCCO)C1 92011,N1(C(C2(C)C(C)CCO2)=O)CCC(NC(C2CCCN2c2cnccn2)=O)CC1 92012,C1(NC(CC2CCN(C)CC2)=O)C2CC3CN(C(=O)CC4CS(=O)(=O)C4)C1C3C2 92013,C1(N(C(C2CC2C(F)F)=O)Cc2ccccc2Cl)CCCN(CC)C1 92014,Cc1cccc(C2(C(N3CCC(CC(=O)N(C)C)C3)=O)CC2)c1 92015,c1(C(C)=O)ccc(Br)cc1NC(C1CCN(C(c2cc(C)n(C)n2)=O)CC1O)=O 92016,c1(C(=O)NCCCCCNC(c2c(C)c(O)ccc2)=O)cn2c(n1)COCC2 92017,CC1(C)C2CCC1(C)C2CNC(c1ccn(-c2cccc(C(F)(F)F)c2)n1)=O 92018,CCC(F)(F)C(=O)NC1CCC(NC(=O)Cn2cc(-c3ccccc3)nn2)C1 92019,c1(C(=O)NCC2(CNC(C(C(=C)Cl)(C)C)=O)CC23CCC3)nnn2c1CCCC2 92020,c1(C(N2CCC(N(C(CN(c3ccccc3)C)=O)C)C2)=O)cc(O)c(F)cc1N 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92075,N1(C(C(C)NC(=O)C(C)(C)C)=O)CC2CC(C1)CN(C(C1CC1(C)C)=O)C2 92076,c1(CC)ncncc1C(N1CCCC1CCNC(=O)C(C)Cn1ccnc1)=O 92077,c1(C(=O)NCCN(C(=O)CCCCC(N)=O)C(C)C)ccc2[nH]cc(C#N)c2c1 92078,c1(CC(=O)OCC)cnc(OC)c(C(=O)N(C2CC(OC)C2(C)C)C)c1 92079,CC1(CNC(c2c[nH]c(=N)o2)=O)CCCN(C(=O)Cc2ccsc2Br)C1 92080,N1(C(C(N2CC(C)C2)C)=O)CCN(C(c2ccncn2)=O)CC1c1nccn1C 92081,Cc1cc(CNC(c2ccc(-c3c(C)noc3C)c(C)n2)=O)ccc1F 92082,C1(C(N2CC(C)(C(NOCCC(=C)C)=O)C2)=O)CCOC1C(=C)C 92083,N1(C(C(CO)N(C)C)=O)CC2(C(=O)NCC(F)Cl)CC1CO2 92084,C(C)(C)(CC(C)(C)O)N(C)C(C1C=CCN(C(C2CC(OC3CC3)C2)=O)C1)=O 92085,C(=O)(C(O)CCCn1cc(-c2ccc(N)cn2)nn1)N1CC(C)C(NS(C)(=O)=O)C1 92086,C(=O)(CCCS(C)(=O)=O)NCC1(CNC(C(C)Cc2cnco2)=O)CC12CCC2 92087,C=CC(C)(C)CC(=O)N1CC(C(=O)NCCNC(C2CCC(C)S2)=O)C1 92088,C(C)(C)(CC(F)C(=O)NC1CCSC1C)NC(c1c(CC)c[nH]n1)=O 92089,C(=O)(C(C)(C)C(C)O)NCCSCC(N1CCC(C)(OC(C)=O)C1)=O 92090,C(N=c1nnc(C)c(C)[nH]1)C1(C)CCN(C(c2nc(C(=O)OCC)sc2)=O)C1 92091,c1(NC(CC)CN2CCCCC2)[nH]c(=NCc2c(Br)cnn2C)nc2scnc12 92092,c1(C(=O)NC(CC=CC)C(=O)Nc2cnccc2OC)c[nH]c(=N)c(C)c1 92093,N1(c2cc(N3CCC(C(=O)O)C3)ncn2)CCCOC(Cn2ccnc2)C1 92094,CC(C)C(C(=O)NC1CCCCC12CCC2)C(C)NC(=O)C#CC1CC1 92095,C1(C(=O)Nc2cn(CC=C)nc2)CC(C)CN(C(=O)CCn2cnnc2)C1 92096,N(C(=NCc1nc(C2CC2)n[nH]1)NC1CCCC(CF)C1)Cc1sccc1 92097,c1(-c2c(C(=O)NCC3C(NC(c4cc(C)no4)=O)CC3)c[nH]c2)ccccc1Cl 92098,c1(CN(C(CSCc2ccccc2)C(C)(C)C)C(CC(C)C)=O)cc(C#N)ccc1N 92099,C1(NC(C2C(OC)CN(C(CCC#CC)=O)C2)=O)CC2(CCCC2)C1 92100,c1(OCC(=O)N(C(CNC(c2c(CC)nco2)=O)C)C)ccccc1C#N 92101,Cc1cccc(CCNC(N2CCC(c3csc(C)c3)C2)=O)c1 92102,C1(C(N(CCNC(c2nc(C)c(C)s2)=O)C2CC2)=O)CC2(CCC2)CO1 92103,C1(CNC(c2scc(C(N)=O)c2)=O)C(O)C(O)CN1C(C1CCCCC(=O)N1)=O 92104,C(C(O)C(=O)NC(Cc1cn[nH]c1)C(=O)N1CCC(CC(N)=O)C1)SC 92105,N1(C(CCNS(CC)(=O)=O)C)CCOCC1.C1CCN1C(=O)OC 92106,C=C(C)CCN(CC(C)NC(=O)NCC)C 92107,CC1CCn2ncc(C(=O)NC(CNC(c3ccncc3O)=O)C(C)(C)C)c2C1 92108,Fc1cc(Cl)cc(Br)c1C(N1CC1)C1CN(c2ncc3cn[nH]c3n2)C1 92109,C1(CC(N2CC(NC(c3coc(C4CCC4)n3)=O)C(O)C2)=O)CC2(CCC2)CO1 92110,c1(CC)cc(C(=O)NCC(O)CCNC(C2CCSC2)=O)cc(C)c1 92111,C(=O)(CC1=CCCCC1)NC1C(C)(CNC(CC2(OCC)CCC2)=O)CCC1 92112,C1(OCC)CC2(CCCN(CC(=O)Nc3ccc4c(c3)OCCO4)C2)C1 92113,C#Cc1cc(C(=O)NCC2(C)CCCN2C(=O)CCC2CC2(C)C)ccc1Cl 92114,C1(CCCNC(C(C2CC(C)(C)C2)OC)=O)CCCCN1C(=O)C=CCO 92115,c1(-n2cc(-c3c(C)cno3)nn2)ccc([N+](=O)[O-])cc1F.N12CC3CC1(C3)CC2 92116,c1(C(=O)NCCCCN(C(=O)C(O)c2ccco2)C)c[nH]c(C#N)c1 92117,N1(Cc2cc(C(=O)OC)c(C)n2C)CCc2ccc(C#N)cc2C1 92118,C(=O)(C(CN(C)C)CC)NCc1c(C(=O)NC(C(=O)OCC)C)[nH]cc1 92119,C(=O)(C(C)S(C)(=O)=O)NCCn1ncc(C(N(CC(CC)C)C)=O)c1 92120,N1(C(=O)CN)CCCC1C1CCCOC1.CC1CC1 92121,C1(C2CC2)(CNC(C2(OC)CCC2)=O)CCN(C(c2c(Br)nnn2C)=O)C1 92122,Cc1nc(C(N2CC(F)CC2CC(=O)NC2CC(CCO)C2)=O)cn1C 92123,CC(C)CC(F)C(=O)N(C)CC1CCCCN1C(c1cc(C(C)C)on1)=O 92124,c1(CNC(=O)CNC(=O)CNC(C2CCCS2)=O)ccncn1 92125,N1(C(CC(C)c2ccccc2)=O)CC(O)CC1C(=O)Nc1ncccn1 92126,C#CC1(O)CN(C(=O)CSCCNC(C2(CF)CC2)=O)C1 92127,CC#CCCC(=O)N1CC(OCC)C(NC(=O)CCCSCCCC)C1 92128,C1(O)(CN(C(=O)CCC2CCC(=O)N2)C)CN(C(=O)CCc2cnoc2)C1 92129,c1(CC)ccc(C(=O)NC2CC(N(C(=O)C=CC3CCOCC3)C)C2)cn1 92130,C1(CC(=O)NCC(C)(CO)NC(C(C)=C2CCC2)=O)COC(C)(C)C1 92131,N1(C(C(C(C)O)NC(=O)OC(C)(C)C)=O)CCOC(C)(CNC(=O)CC(C)(C)O)C1 92132,C1(C(=O)NC(CNC(c2cc(C)[nH]n2)=O)C(C)(C)C)COC2(CO)CC1C2 92133,C#CCC(CC(F)F)C(=O)N1CCCC1CCC(=O)Nc1ccc(C)cc1CO 92134,CCC(CC)CC(F)C(=O)NC(CCCOC)C(=O)N1CCC1CC1CCCC1 92135,N1(C(C2(CC)CCCC2O)=O)CC2(C)CC1(C(N1CC3(CCC3O)C1)=O)C2 92136,c1(C(=O)NC2CC(CCNC(CSC)=O)C2)ccc(N2CCCC(O)C2)cc1 92137,C(CCNC(C1CCCC1)=O)(C(=O)NCCOC1CC1)OC 92138,C1(CC(=O)NCCN(C(CCSCCCC)=O)CC2CC2)CC(OCC)C1(C)C 92139,N1(C(C(C)OCC=C)=O)CC(C(N2CCCC(C(C)(C)O)C2)=O)C(C)(C)C1 92140,N1(C(C2(N(C(c3n(CC)ccn3)=O)C3CC3)CCC2)=O)CC2(CC(CO)CO2)C1 92141,C=CCCCCCCC(=O)N1CCN(C)C(CNC(C2CCCC2CC)=O)C1 92142,C1(S(C)(=O)=O)(C(=O)NC(C)CC(C)NC(c2ccncc2F)=O)CCC1 92143,c1(CC(=O)N(CCC(=O)OCC)CCO)cc(F)c(F)cc1F.C1C(C)N1 92144,C(=O)(CC(C)C(=O)NC1(C)CN(C(=O)CCSc2ccccc2)C1)OC 92145,Cc1nc(CO)ncc1C(=O)NCC1(C)CC(NC(C2(n3ccnn3)CC2)=O)C1 92146,N1(C(C2CC=C(C)CC2)=O)CCCC2CN(C(=O)CC3CC=CCC3)CC12 92147,C1(CCCNC(CC2(OC)CCCC2)=O)CCCCN1C(C1CC(C)(C)C1)=O 92148,N1(C(CCC2(C)CC2)=O)CCN(C(c2cccc3c2CCC3)=O)C2CCCCC12 92149,Cc1ccc(CC(N2CC(CNC(=O)CNS(N)(=O)=O)C(O)C2)=O)c(F)c1 92150,CCC(CCC(=O)NC12CC(C)(C1)C2)NC(=O)CC(C(F)F)SC 92151,CC1CCN(C(=O)C(=O)NCC(F)F)C1CNC(c1c(Br)ncn1C)=O 92152,C(=O)(C(C)S(=O)(=O)C(C)C)NCC(C1CCN(C(CCCC(C)C)=O)CC1)(C)C 92153,N1(C(C(C)=CC)=O)CC(CNC(=O)CC(CC)CCC)OC2(CCC2)C1 92154,c1(N(C)Cc2ccccc2[N+](=O)[O-])ccc(S(=O)(=O)NCC2CCCCS2)cn1 92155,C(CCCC(=O)NCCCCCF)N(C(C1C(C(C)C)OCC1)=O)C 92156,C1(CC(=O)N(C2CCN(C(=O)COCCF)CC2)C)COC(C)(C)CO1 92157,N1(C(C(=O)NCCSC(C)(C)C)=O)CCOC2c3ccccc3OCC12 92158,C1(N(C(CCc2c(C)ncs2)=O)C)CCCN(C(=O)CC2CCSC2)CC1 92159,O(NC(=O)C(F)C1(O)CN(C(c2ccc[n+]([O-])c2)=O)C1)C(C)(C)C 92160,CC1CN(C(C2CCCN2c2cnccn2)=O)CCN1C(=O)C=CBr 92161,N1(CC2CCCC(C(=O)OC)C2)C(=O)NC(Cc2cc(C)cc(C)c2)C1=O 92162,C1(CNC(C2N(C(=O)OCC)CCOC2)=O)COCC(C)(C)O1.C12CCN1C2=O 92163,N12CCN(CC13CCC3)C(=O)CC2=O.C1(C)(SCCCC)CCC(C(F)(F)F)C1 92164,C1(C(C)NC)(CNC(c2ccc(CC(=O)OC)o2)=O)CCN(C(=O)COCC)C1 92165,C1(CCC(N2C(COC)CCC2)=O)CCCN(C(c2c(SC)cnn2C)=O)C1 92166,C1(CNC(C2C(C=C)C2)=O)COCCN1C(=O)CC1CCSCC1 92167,c1(C(N2CC(C)N(C(=O)Cc3c(Cl)cnn3C)CC2)=O)cnn2c1N(C)CC2 92168,O=C(C=CCCc1ccccc1)NNc1ccc(Cl)cn1 92169,C1(NC(C2C(C(N)=O)C2)=O)CC2COCC(C1)C2NC(C1CCCCNC1=O)=O 92170,C1(C(=O)NCCCN(C(C)C)C(C23CSCC2C3)=O)CC2CC(=O)C1C2 92171,c1(C(N(C2CC(C(=O)NC3CCCCC3)C2)C)=O)c[nH]c2cccnc12 92172,Cc1nc(CC2CC2)ncc1NC(=O)C=Cc1ccsc1 92173,C1(SCC)CCN(C(c2cnn(COC)c2)=O)C1CNC(=O)CCN1CCCCC1 92174,C1(CNC(C(c2cccc(O)c2)C)=O)CCN(C(=O)C=CC2CCCC2)CC1 92175,CCC(C)(CC)CN=c1[nH]c2c(c(=NCC(=O)NC3CC3)[nH]1)CCCCC2 92176,c1(C(=O)NCC(COC)NC(c2cc(C(=O)OC)c[nH]2)=O)c(Cl)cnn1C 92177,c1(C(=O)NC(CNC(c2cc(C)ncn2)=O)C2CC2)ccc(F)cc1F 92178,c1(C(C)C(=O)NC(C2(O)CN(C(c3ncccc3Cl)=O)C2)C)c(F)cccc1F 92179,C(=O)(C#CC1CC1)NCC1CC(C(=O)NCC#CCOC)C1 92180,c1(C(=O)OC)coc(C=CC(=O)NCC(C)N(C(=O)Cc2ccon2)C)c1 92181,N1(C(Cc2cc(CC)nn2C)=O)CCN(C(c2cc(OC)n[nH]2)=O)CC(C)(C)C1 92182,c1(C(N(CCN(C(COCC)=O)C)C(C)C)=O)ccc2nc(C3CC3)cn2c1 92183,C1(C(=O)NCC(=O)N(C(c2ccncc2)C)CC)CCC(OC)CC1 92184,C1(CNC(C2CCCC3CC23)=O)CCCC12CCN(C(C1CCCC1O)=O)CC2 92185,c1(OC)n[nH]c(C(=O)NCC2CCC(NC(=O)Cc3cccs3)C2)c1Cl 92186,N1(CCN=C(NCC(CC)CO)NC2CCC2)CCc2ccccc21 92187,C1(CNC(C(C=C)O)=O)CC(F)CN1C(C1CCC(C)O1)=O 92188,C(=O)(CC1=CCN(C(c2c(F)cccc2F)=O)CC1)Nc1ccc(C)nc1C 92189,c1(C(N2CCC(CN(C(=O)C(O)C3CCC3)CC)CC2)=O)onc2ccccc12 92190,c1(CC(C)NC(=O)C(C)(C2CC2)N(C(=O)C(F)OC(F)(F)F)C)ccccn1 92191,N1(C(C(n2cnc(C#N)n2)CC)=O)CC(CNC(=O)CCCF)C(C(F)(F)F)C1 92192,C(=O)(CCCCC(C)CC)NC(CCCC)CNC(c1ncoc1C(F)(F)F)=O 92193,C1(NC(C(CCCOC)(C)C)=O)CCC2CN(C(C3CCCO3)=O)CC2C1 92194,C(CC(F)CN=[N+]=[N-])NC(c1cc(CNC(C(C)NC(CC)=O)=O)ncc1)=O 92195,Cc1nn(CC(N2CCC3CCC23CNC(=O)C=CC(F)(F)F)=O)c(C)c1C 92196,C1(C(N(C(CC)C2CC2)C)=O)COCCC1NC(c1cc(C)sn1)=O 92197,c1(NCc2cnn(CC)c2C)ncnc(NC2CC3CC(O)C2C3)c1C 92198,c1(C(=O)NC2CCC(NC(=O)CC3CCCS3(=O)=O)C2)nc2cnccc2s1 92199,Cc1ccc(Cl)c(N)c1C(=O)NCCC(O)CNC(C12CCN(CC1)C2)=O 92200,CCCC(CCCNC(c1coc(CC)n1)=O)NC(=O)CN(C1CCC1)C 92201,c1(NC(C2(CO)CN(CC3CC3(F)F)C2)=O)ccc(-c2nc(C(F)(F)F)cs2)cc1 92202,CCC(O)CC(=O)NCCC1(CNC(=O)CCc2nc(-c3ccco3)no2)CC1 92203,CC1(C)CC(NC(=O)C=CCO)CCN(C(=O)CC2CCNC(=O)C2)C1 92204,C1(C(C)(C)NC(=O)CC2CNC(=O)C2)CCN(C(C2CC2[N+](=O)[O-])=O)CC1 92205,c1(NC(CC)CNC(C23CC4CC(C(=O)N2)C3C4)=O)ncnc2c1nnn2C 92206,Cc1c[nH]c(C(=O)NCCN(C(=O)Cc2ccoc2)C2CC2)cc1=O 92207,C(CCC(C)C)(C(=O)N(CCCOC(C)C)C)NC(CC(CC)C1CC1)=O 92208,c1(CC)cccc(NC(=O)CC(C2CC2)NC(c2sc(O)nc2C)=O)c1C 92209,C1(C(N(CC(=O)N(C)C)CCC)=O)CCCN(C(=O)C2=C(Cl)CC2)C1 92210,c1(C(N(CCNC(C(c2n(C)ncc2)O)=O)CC2CC2)=O)ccc2c(c1)COC2 92211,c1(C(=O)NC(C2(C(=O)NC3CCCC3(F)F)CC2)C)ccc([N+](=O)[O-])o1 92212,C=CC1CN(C(c2cccc(=O)o2)=O)CC1NC(c1ccc(CO)c(F)c1)=O 92213,c1(C(=O)NC(C(C)NC(Cc2ccc(OC)cc2)=O)C(C)C)c(F)cccc1F 92214,C1(CCC(=O)NCCCSC)CCCN1C(=O)CCn1cccn1 92215,c1(C(=O)C(N2CCN(C3CC(F)(F)C3)CC2)=O)ccc(Cl)cc1 92216,CCC(C)(CNC(c1coc(-c2ccccn2)n1)=O)NC(C1(OCC)CC1)=O 92217,C1(O)(CC2CC=CCC2)CCN(C(=O)NC(c2cc[nH]c2)C)C1 92218,c1(OCC(CN(C)Cc2cnn(C3CCCCO3)n2)O)cccc(Br)c1I 92219,c1(C(N(CCC(C)(C)NC(CC(CC)C)=O)C)=O)cn2ccc(C)cc2n1 92220,c1(NC(C2(NC(C)=O)CC2)=O)c(F)c(F)c(F)c(F)c1F 92221,c1(C(=O)NCC(C2CCCCC2)NC(C(C)OCCOC)=O)ncc(Cl)cc1Cl 92222,c1(OC)ccc(Cl)c(F)c1C(=O)NCCCCNC(C1CC1c1ccoc1)=O 92223,c1(OC)ccnc(NCC(=O)NCC(C)CNC(C2(C)CCCC2C)=O)n1 92224,C1(C(F)F)(OC)CCCN(C(c2nc(Br)nn2C)C(=O)NC(C)(C)C)C1 92225,N1(C(C(C(C(C)C)C)NC(N)=O)=O)CCCC2(C1)CN(C(=O)C1=NOCC1)C2 92226,Cc1c(C(N2CCCC2C(=O)NCCC(CO)C(C)C)=O)cccc1C#N 92227,CC12CC(CCO1)N(C(=O)C(C1CCOC1)NC(=O)CC(O)C1CCCC1)C2 92228,c1(-c2ccc(-n3c(C)cc(C)n3)cc2)cc(F)c2nc(C)cn2c1 92229,CCCCC(O)C(=O)NCC1(C)CCN(C(c2cccnc2OC)=O)C1 92230,c1(N2CC2CC(C)C)ccc(F)cc1C.CCCCC 92231,C(CO)(CC(C)(C)C)NC(C1C(CNC(Cc2nc(C)[nH]n2)=O)C1(C)C)=O 92232,C1(C(=O)NCC2(C=C)CCC2)C2CCCC2CN1C(C1CCC2(CCC2)C1)=O 92233,C(C(CNC(C1CCS(=O)(=O)C1)=O)S(C)(=O)=O)NC(C1(CC#C)CC1)=O 92234,c1(C(=O)NC2CCN(C(C(C)NS(C)(=O)=O)=O)C2)cc(Cl)c(Cl)[nH]c1=N 92235,C=C=CCC(=O)N1CCC(C(C)(C)NC(c2cc(C(C)CC)no2)=O)C1 92236,C(C(CC1CCCC1)C(=O)NCC1CCN(C2CC2)C1)NC(C=CCC)=O 92237,N1(C(c2coc3c2COC3)=O)CCN(C(=O)C(F)(F)C(F)(F)F)CC2(CC2)C1 92238,CC(C)CCC(=O)C(=O)N1CC(CC(=O)NC2CC(F)C2)C(C)C1 92239,C1(O)(CNC(c2cn(CCNC(CCC=C(C)C)=O)nn2)=O)CCC(C)C1 92240,C#CCC(C)C(=O)N(CC(C)NC(c1ccc(-c2cn[nH]c2)cc1)=O)CC 92241,c1(NCC(=O)NC(CNC(COCCCCC)=O)(C)CO)ccccc1Cl 92242,CC(CC(=O)N1CCC(O)(CNC(=O)CC2CN(C)C2)C1)C(F)(F)F 92243,c1(C(C)C)cc(C(N2CC(CO)(NC(c3cccc(F)c3F)=O)C2)=O)ccc1F 92244,C(C1CCCO1)=CC(=O)NCC1CCCC1NC(=O)CC(O)c1ccccc1 92245,C(=O)(CCCN=[N+]=[N-])NCCCCC(C)NC(C1(CCOC)CC1)=O 92246,CCC(C(=O)NCCCCC1(NC(=O)Cc2csc(Cl)n2)CC1)C(F)(F)F 92247,CC(C)(C#N)CCCC(=O)NCC1C(CNC(c2c(F)cccc2F)=O)C1(F)F 92248,C1(NC(CCC)=O)(CNC(c2cscc2OC)=O)CC2CCC1CC2 92249,C12(CNC(COCCOCC)=O)CC1CCN2C(=O)CN1CSCC1=O 92250,N12CCCC(O)(C1)C2=O.C#CC1(NC(=O)CCNCS(=O)(=O)C(F)(F)F)CCCC1 92251,C1(CNC(c2n(CC=C)ccc2)=O)C(C)CCCN1C(c1cc([N+](=O)[O-])n[nH]1)=O 92252,Cc1cc(C(N2CCOCC2C(=O)NCC2CCOC2)=O)oc1C 92253,N1(C(C2CC(C)N2C(C2CC3CCC(C2)O3)=O)=O)CCc2ccccc21 92254,N1(C(c2cc(OCC)n[nH]2)=O)CCC2(CCCN2C(C2CCCCC2(C)C)=O)C1 92255,c1(C(N2CCC(F)(CNC(c3sccc3F)=O)C2)=O)ccc2nonc2c1 92256,C1(NC(C2(COC)CCC2)=O)CN(C(=O)COc2cccc(F)c2)CC2(CC2)C1 92257,C1(C(=O)NCC2C(NC(CC3(C)CC(F)(F)C3)=O)CCC2)CCS(=O)(=O)CC1 92258,c1(C(N2CCCC(N3CCCC3=O)C2)C(=O)NCC(C)C)cnn(C(C)C)c1I 92259,C1(C(=O)NC(c2ccc(C)nc2)C)CCN(C(c2ccccc2F)=O)C(C)(C)C1 92260,C(=O)(C1=CCc2ccccc21)NC(C)CC(C)NC(c1cnc(Cl)n1C)=O 92261,c1(C(C(=O)NC2C(CNC(=O)Cc3cccs3)C2)O)cccnc1 92262,C1(NC(CCC(N)=O)=O)CCC2CCN(C(=O)C(C3CC(F)(F)C3)O)C1C2 92263,N1(C(C(CC(C)C)=O)=O)CCC2CN(C(C3(C4CC4)CC3)=O)CC2CC1 92264,n1(CC)cc(C)c(=NC(=O)c2cn(CCCC(=O)OC(C)(C)C)nn2)[nH]1 92265,N1(C(C(c2ccccc2)OC)=O)CCCOC(CNC(C2(C(N)=O)CC2)=O)C1 92266,c1(C(N2C(C)CC(CNC(CCSC)=O)C2)=O)cc2n(n1)CCCNC2=O 92267,n1(CCCC=C)cc(C(=O)NCC(C)CNC(=O)COCc2nc[nH]n2)nn1 92268,N1(C(C2C(C)(C)CO2)=O)C2CCC1CN(C(C1CC3C=CC1C3)=O)C2 92269,C1(N(C(C(CCC)CC)=O)C)CC2CCC(C1)N2C(=O)C(F)(F)C(O)CC 92270,c1(C(=O)NC(C)CNC(=O)CC2(C#N)CCC2)cc(N2CCNC2=O)c(F)cc1F 92271,c1(SC(C(N2CC(OC)C(C(=O)OC)C2)=O)C)ccc(F)c(C2CC2)c1 92272,C1(O)(C(N(CCNC(=O)Cn2ccc(C3CC3)n2)CC)=O)CCC(C)(C)CC1 92273,Cc1ncc(CCNC(=O)CCN(C(=O)C=CC2CCOC2)C(C)C)[nH]1 92274,N1(C(CC(CC)C(C)C)=O)CC2CCN(C(=O)C(C)OCC3CCCC3)C2C1C 92275,c1(C(C(N2C(C)(CNC(C(C3CC3)OCC)=O)CCC2)=O)=O)ccc(Cl)cc1O 92276,c1(C(=O)NC(C)CN(C(=O)CC(C)(C)C(F)F)C)coc2c1C(O)CCC2 92277,c1(OC)cc(F)ccc1C(=O)NC1CCN(C(=O)Cc2cc(C)nn2C)C12CC2 92278,CC1CN(C(=O)Cc2cc(O)nc(O)n2)CCN1C(c1coc(Cl)c1)=O 92279,c1(C(=O)NC2CC(NC(C3N(C(C)=O)CCCCC3)=O)C2)cnc2n1CCCC2 92280,c1(C(=O)NCC2CN(C(C3(C=C)CC3)=O)CC2O)nc2n(c1Cl)CCCC2 92281,c1(C(=O)NCC2(NC(c3ccsc3)=O)CC2)cccnc1-n1ccnc1 92282,N1(C(C(C)=CC)=O)CCCC2(C1)C(NC(c1cc(F)n[nH]1)=O)CCN2C 92283,c1(C(=O)NCC(CC)(C)NC(c2cc(-c3cnn(C)c3)on2)=O)nc(O)sc1C 92284,N1(C(COCCC#C)=O)CCCC(CNC(C2(CC(=O)NC)CC2)=O)C1 92285,c1(C(N2CC3(C(CNC(=O)Cc4nc[nH]n4)CC3)C2)=O)ccc([N+](=O)[O-])c(Cl)c1 92286,C1(C(=O)NC(CC)(C)C(F)(F)F)CCN(C(=O)CN(C)C2CC2)C12CCC2 92287,C1(C(=O)NC2C(CNC(CNS(NC)(=O)=O)=O)CCC2)COC(C)(C)CO1 92288,Cc1cccn2cc(C(=O)N(CC(C)NC(C3(C(C)C)CCCO3)=O)C)nc12 92289,c1(OC)cc(Cl)ccc1C(N1CCC(CO)C(NC(=O)C2CC2)C1)=O 92290,CCCCCC(C)NC(=O)C(c1cn(C)nn1)NC(c1ccc(F)s1)=O 92291,C1(C(=O)NCC(=C)CCNC(=O)CCCOC)CSC(CC)C(=O)N1 92292,CCC(=O)CCC(=O)N1CCCN(CCNC(=O)C(F)C2CCOC2)CC1 92293,N1(C2CCCN(C(c3c(CC)scc3)=O)C2)CCN(C(=O)C#CC2CC2)CC1=O 92294,c1(C(N2CCN(CCCNC(C3(C)COCCO3)=O)CC2)=O)cnn2c1OCC2 92295,C1(CN2C(CNC(Cc3nc(NC=O)sc3)=O)CC2)CCCCC1(F)F 92296,Cc1cc(C(=O)NCC2(CNC(=O)Cn3ccc(C(F)(F)F)n3)CC2)ccn1 92297,c1(C(N(C)CC2N(C(c3c(C)nns3)=O)CCC2)=O)cnc2nc(O)ccc2c1 92298,N1(C(CC2CCC(C)C2)=O)CC23CCCC2(C1)CN(C(c1cc(CO)[nH]n1)=O)C3 92299,c1(C(C(N2C(C(=O)OCc3ccccc3)CSC2)=O)O)cc(F)c(F)cc1F 92300,C1(NC(c2n(CC)nnc2)=O)CCCC(NC(=O)CC2(N(C)C)CC2)C1 92301,c1(C(C(=O)NC(C)CNC(=O)C=CC(F)(F)F)C)ccn(C)n1 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92319,C1(NC(C=Cc2ncc(C)[nH]2)=O)CN(C(=O)C(C2CC2)C2CC2)CC1C1CC1 92320,N1(C(C23N(C(Cc4nn(C)c(Cl)c4)=O)CC(C)(C2)C3)=O)C2CCC1CC(CO)C2 92321,c1(N(C(CCNC(C2(OC)CCS(=O)(=O)C2)=O)C)C)ccc([N+](=O)[O-])cc1Cl 92322,N=c1nc2c(c[nH]1)CC(C(=O)NCCCCNC(=O)CC13CCCC1C3)CC2 92323,C1(C(=O)NCC2C(OCC)CN(C(CCC=C=C)=O)C2)CCC2(CCC2)CO1 92324,C1(C(=O)NC(CC)CNC(=O)CCC#N)CC(c2ccc(C)cc2)=NO1 92325,C1(NC(C(N2C(COC)CCC2)=O)=O)CCCCN(C(=O)CC(F)F)C1 92326,CC1(C)NC(=O)N(CC(=O)NC2CC(NC(=O)C(CO)NC(N)=O)C2)C1=O 92327,C1(C(=O)NCC(=O)Nc2nncs2)CCCN2CCCC12 92328,c1(NC(c2scc(-c3ccc(C(=O)NC)cc3)n2)=O)cc2n[nH]cc2cc1C 92329,c1(C(N(CC(CNC(CSCCC(C)C)=O)C)C)=O)cnn2c1NCCC2 92330,C1(N(C(c2c(C)coc2)=O)C)CCCCN(C(=O)C(F)C(C)(F)F)C1 92331,c1(C(=O)OC)cnn(C)c1S(=O)(=O)NCC1C2OC(=O)OC12 92332,Cn1ncc([N+](=O)[O-])c1C(N1CC2CC(C1)C(CO)O2)=O 92333,N#Cc1c(NCc2ccc(Br)o2)cccc1F.C1(CN2CC2)CCCO1 92334,C1(NC(c2c(C)onc2CO)=O)CCC2CN(C(=O)CCCN(C)C)CC2C1 92335,C#CC1(C(=O)NC(c2ccc(O)nc2)C)CCN(C(C2CN(C)CCO2)=O)C1 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92354,c1(SCC2CC(NC(c3c(C(=O)OCC)cccn3)=O)C2)nccn2nccc12 92355,C(=O)(CC1OCCc2ccccc21)N1CCC(C)(NC(=O)CC2(O)CCC2)CC1 92356,C(=O)(C(COC(C)=O)C(F)(F)F)NC12CC(NC(C(CCCC)C)=O)(C1)C2 92357,Cn1ncc(C(=O)NC2CCN(C(=O)CC3CC(C)(C)C3)C2)c1-c1ccccc1 92358,N1(C(C2CCC(NC(C3C4C=CC(C4)C3CO)=O)CC2)=O)CCC2(CCOC2)C1 92359,c1(C(N(C(C(C)OC2CCN(CC3CC3)C2)=O)C)C)ccc(S(C)(=O)=O)cc1 92360,CC(CC(=O)NC1(C)CCN(C(c2ncccc2O)=O)C1)C(F)(F)C(F)(F)F 92361,N1(C(C2CN(CC)C(=O)C2)=O)CC2(CCN(C(c3ccc(Cl)o3)=O)CC2)C1 92362,N1(c2ncc(C#C)cn2)CC2(CN(C(=O)CNC(=O)C(C)(C)C)CCO2)C1 92363,c1(C(C)(C)NCc2c(Br)ccc(C)n2)ccc([N+](=O)[O-])cc1 92364,c1(OC(C)C)ccc(S(=O)(=O)N2CCNC3(CCC3)C2)cn1 92365,CC1C2CCC(C2)C1C(N1CCC(C(N2CCC2C(N)=O)=O)C(C)C1)=O 92366,C1(C(C)NC(c2c(C)cns2)=O)CN(C(=O)CCc2cccc(O)n2)CCO1 92367,c1(N(C)C)cc(F)c(C(=O)NCC2CC(NC(=O)C=CC3CCOC3)C2)c(F)c1 92368,c1(C(N2C(CNC(C(c3cncc(F)c3)C)=O)C=CC2)=O)ccc(F)c(F)c1F 92369,N1(C(c2cncnc2)=O)CCOC2(C1)CN(C(c1cc3c(s1)COCC3)=O)C2 92370,C(=O)(C1CNCc2ccc(Cl)cc21)N1CCC2(CC(OCC)C2)C1 92371,C(=O)(CC(C)P(C)(C)=O)N(CCNC(C=CC(C)C)=O)C1CC1 92372,N1(CC)CC(C)N(C(c2cnc(CC)[nH]2)C(=O)NCCCOCC2CC2)C(C)C1 92373,C1(CNC(C(CC)C#N)=O)(NC(c2cc(C(F)F)ccn2)=O)CCCCC1C 92374,C1(NC(COCC=C)=O)(CO)CCN(C(c2cc(-c3cccnc3)on2)=O)CC1 92375,c1(CC)cc(C(N2CC(C(C(=O)NCCc3nccn3C)OC)C2)=O)n(C)n1 92376,c1(CC(=O)N(C2CC(C#N)C2)CC(=O)NC(c2ncco2)CC)csnc1C 92377,c1(OC)cc(Cl)ncc1NC(C1CCC(NCc2cc(Br)cnc2F)CC1)=O 92378,N1(C(C=Cc2c(C)ccs2)=O)CCC2CN(C(C3CC34CCSCC4)=O)CCC12 92379,C#CCCC(O)C(=O)NCC1C2CC1N(C(c1cccc(C)n1)=O)C2 92380,c1(CNC(C2N(C(C3CC(OCC)C3)=O)CCC2)=O)ccc(O)c(C)c1 92381,c1(C(C)NC(=O)NC2CC(C)(COC)C2)cccc(SC)c1 92382,C1(C(=O)NC2C(C)(C)CN(C(=O)Cc3ccsc3)C2)CCc2nccn2CC1 92383,C#Cc1ccc(C(=O)NCCC(C)NC(C2CC(C#N)C2)=O)c(F)c1 92384,C(c1ccccc1[N+](=O)[O-])=CC(=O)NC1CCN(C(C2CCCCC2)=O)CC1F 92385,N1(C(c2c(C)n[nH]c2C)=O)CCCC(C2(NC(=O)C3=CCCCCC3)CC2)C1 92386,CCC(C)C(O)C(=O)Nc1cccc(NC(=O)CC23CCCC2C3)c1 92387,CC1(CCN(C(CCC2OCCO2)C(=O)Nc2ccccc2)C)CCOCC1 92388,c1(C(=O)OC)cccc(CC2CN(C(C3(F)CC(C(=O)OCC)C3)=O)C2)c1OC 92389,c1(OC)cc(C)ccc1OCCc1nc(CCC(F)(F)F)nn1CCCO 92390,NC1CCN(CC(=O)NC2CC2c2cncs2)C(C(F)(F)F)C1 92391,N1(C(C2CCN(CC)CC2)=O)CCN(C(C2CCSCC2)=O)C(CC#N)C1 92392,N1(C(CCC(C)OCC)=O)CCOC2(CCN(C(=O)CC3CCOC3=O)C2)C1 92393,C(C(C)(C)CC(=O)N1CCC(N(CCO)C(c2cnnc(C)c2)=O)C1)OC 92394,C1(NC(c2nc(C)n(C)n2)=O)CC2CC(NC(=O)C3=CCOCC3)CC2C1 92395,Cc1cn(C(C)C(=O)OC(C)C)[nH]c1=NC(=O)c1c[nH]c(-c2ccccc2)n1 92396,C1(CNC(CN(C2(C)CCC2)C)=O)CCN(C(c2csc(CC3CC3)n2)=O)C1 92397,C1(C(N2CC(C(C)NC(=O)Cc3cccc(Cl)c3)C2)=O)CC2CC1C1CC21 92398,O=CN1CCOCC1C(N1CC2CC2(CNC(C2CC(C3CC3)=NO2)=O)C1)=O 92399,N1(C(=O)CC2CCS(=O)(=O)CC2)CCN(C(=O)C2=CCCOC2)CC(O)C1 92400,C1(C(N2CCC(N(C(=O)C=CSC)CCC)C2)=O)CCc2nc(C)cn2C1 92401,c1(OC)ccc(N(C(=O)C(C)N(C)Cc2ccc(Br)s2)Cc2ccco2)cc1 92402,CN1CC2C(C(=O)NCCn3cc(CCCC(C)(C)C)nn3)C2C1 92403,Cc1cc(CNC(=O)NC(Cc2cccc(Br)c2)CO)ncn1 92404,C(C(C)(C)CN=c1[nH]c(=N)[nH]c(=NC(C)Cn2cc(C)cn2)[nH]1)OC 92405,c1(C(=O)NCCC(C(C)C)NC(c2ccc(OC)cc2)=O)cnc(Cl)cc1N 92406,c1(C(=O)OC)cc(S(=O)(=O)NC(c2ccccc2)CF)ccc1F 92407,C1(N(C)C)CCC(C(N2CCCC(C(O)C(F)(F)F)C2)=O)CC1 92408,C=C(C)C(C)(O)C(=O)NNC(=S)NC1CCC12CCC2 92409,Cc1ncnc(C(=O)NC(C)CC(C)NC(=O)CCC(=O)c2cccs2)c1C 92410,c1(C(C(N2CC(C)OC(C)C2)=O)(C)C)ccc(Cl)cc1[N+](=O)[O-] 92411,C(=O)(C(CC(C)C)N(C1CC1)CC1CC1)OC.c1(C2C(=O)N2)ccccc1Br 92412,CC1CN(C(=O)C(C)(CO)NC(c2ccc(C(N)=O)o2)=O)Cc2nncn21 92413,N1(C(C(C(C)C)N2CCCC2=O)=O)CC2CCCN(C(c3cc(O)no3)=O)C2C1 92414,N1(C(CCn2cc(SCC)nn2)=O)CCC(O)(CNC(C(F)F)C(C)(C)C)CC1 92415,c1(C(=O)NCC(=CC(=O)NC(C(CCC)C)CO)C)ccc2cc[nH]c2n1 92416,c1(NC(CC2(C)CN(Cc3c(OC)c(F)ccc3)C2)=O)nccc2[nH]ccc12 92417,c1(CC(N2C(CNC(C=C(C)Cl)=O)CN(C)CC2)=O)ccc2c(c1)COC2 92418,Cc1ccccc1.c1(OCCC(=O)N)cccc(N2CCC2)c1 92419,c1(CCNCCOCCOC(COC)NCC)cn(C(C)(C)C(C)C)nn1 92420,CP(C)(=O)c1ccc(C(=O)NCC23CCCC(CN2C(=O)COC2CC2)C3)nc1 92421,N1(C(=O)CCCC(F)F)CCC2(CCN(C(=O)C3=CCCC3)C2)C1 92422,N1(C(c2ncnc(C)c2C)=O)CCCC2(CCN(C(=O)COCC(F)(F)F)C2)C1 92423,c1(C(N2CCC(C(C)(C)NC(C(F)OC)=O)C2)=O)cccc2ccc(O)nc12 92424,C1(C(=O)Oc2ccccc2)CCCN1Cc1conc1-c1ccccc1 92425,C1(C(N2CC(COC)(NC(=O)C(CCOC)OC)C2)=O)CC(=O)C12CCC2 92426,c1(CC(N2CC(CCO)(NC(c3cc(C)no3)=O)C2)=O)c(C)noc1Cl 92427,Nc1ncnc2c1ncn2CCCCC(=O)Nc1cccc2c1ncn2C 92428,c1(CC(C)=O)nc(C)c(C(=O)NCC2CC(NC(=O)C=CC3CCCC3)C2)o1 92429,c1(CCC(=O)NCCCC(C)NC(C2(C)CCCO2)=O)ccccc1Br 92430,c1(C(N2CCN(CCCNCC3CC=CCC3)CC2)=O)cn2c(Br)cccc2n1 92431,C(=O)(C(C)C(F)F)NC(C(=O)NCCN(C(CC)C)C)CC 92432,CC(C(=O)N(C(C)CCNC(c1ccc(C2CCOC2)cc1)=O)C)C(C)(F)F 92433,C1(C(=O)NCC)CCCN1C(c1ccc(CNC(=O)CCCNC(N)=O)s1)=O 92434,C1(C)(CNC(C2(NC)CCCC2)=O)CCCN1C(=O)COC1CCCCC1C 92435,n1(CC)ccc(C(=O)NCC2CCN(C(=O)C(C)COC)C2)c1C 92436,C1(C(=O)NCC2C(NC(CSCCC#N)=O)CCCC2)CCC2CCCCN12 92437,C#CCCCCC(=O)N1CCN(C(=O)CC(C)c2ccccc2)CC1CCO 92438,C(CC(CC)C(=O)NC(C1CC=CCC1)C(=O)NC1CCCC(CO)C1)=CC 92439,S(=O)(=O)(c1c[nH]c(C(N2CC(CCNC(=O)C(O)C(C)(C)C)(OC)C2)=O)c1)NC 92440,N1(C(C(CC)(C)F)=O)CC(NC(c2ccc(C(C)C)nc2)=O)C(N=[N+]=[N-])C1 92441,C1(C(=O)NC2CC(NC(c3ccccc3CO)=O)CC2O)(OC)CCC(C)(C)C1 92442,Cc1cc(C(=O)NCc2nc(C(=O)NCC3CCCCC3(C)C)co2)nc(C)c1 92443,N1(C(C(CC)=CC)=O)CCCC(C(C)(C)NC(C2CCCCC2C)=O)C1 92444,C(=O)(C1=CC2(CCN(C(C3(CO)CCCC3)=O)C2)C1)NCc1ccc(CC)cc1 92445,c1(NC)cncc(C(N2CCCC(CCNC(=O)Cc3cc[nH]c(=N)c3)C2)=O)c1 92446,c1(NC(C2N(Cc3cccc(C#N)c3)CCSC2)=O)ccc(Br)cc1[N+](=O)[O-] 92447,c1(C(=O)NCCN(C(C(C)OCC=C)=O)C)cc(OCC)cc[n+]1[O-] 92448,C1(NC(CN(C(C)=O)C)=O)COCC1NC(=O)CNc1ccccc1 92449,C1(NC(c2c(C)snc2)=O)CCCC(C(=O)NCC(O)CNC(N)=O)CC1 92450,c1(CC)nn(C)c(OC)c1CNC(=NCc1n[nH]cc1Br)NC1CC1C 92451,N1(C(C2(CNC(=O)CC3C=CCC3)CCCCC2)=O)CC(C2CCCCC2)C1 92452,c1(C(N2CCC(N(C(c3cnc(O)n3C)=O)CC)C2)=O)cccc2nccnc12 92453,c1(NC(CC)CO)ncccc1S(=O)(=O)NCCC(F)(F)CC 92454,N1(C(C(CC)=CCCC)=O)CC(NC(C2(COC)CCCC2)=O)C(COC)C1 92455,N1(C(CS(CC)=O)=O)C2CCC1C(CNC(c1c[nH]cc(Cl)c1=O)=O)C2 92456,N1(C(CC2(CC)CCC2)=O)CCC(C(C)(C)C(=O)NC(CN(C)C)CC(C)C)C1 92457,N1(C(CCCCCC)=O)CC2CCCC2(NC(c2nn(C)c(C)c2Br)=O)C1 92458,CCC(C)C(C(=O)NC1(C)CC1)NC(=O)NCCSC 92459,c1(-c2c(N3CCN(C(CC)=O)CC3)nccc2)ccc2[nH]c(C(=O)OC)c(C)c2c1 92460,C=CCCN=C(NCC(C)C(F)(F)F)NCc1ccc(C2CCCCC2)cc1 92461,C1(C(=O)NCC2CCCN(C(=O)C3=CCCCO3)C2)CC2CC1CC2(F)F 92462,CCC(CCC(=O)NC1CCC(C)CC1)NC(c1cc(C)c(CC)o1)=O 92463,c1(CN2CCN(C(CC(CC)C)=O)C3C2C3)cc(C#N)ccc1Cl 92464,C1(C(=O)NC(C)C(C)(C)NC(c2cncc(Cl)c2)=O)OCCOC12CCC2 92465,Cc1ncc(C(F)(F)F)cc1C(=O)NCC1CCC1NC(C1CC1(F)F)=O 92466,CCC(CC(=O)NC1CCC(NC(c2conc2C2CCC2)=O)CC1)SC 92467,c1(NC(N2Cc3c(cc(C(=O)OC)s3)CC2)=O)cnc2c(Br)cc(Br)cc2c1 92468,N1(C(c2cn(CCCC)nc2C)=O)CCOCC(NC(C2(F)C3CCCC23)=O)C1 92469,C(=O)(CCCC(=O)NCC(CO)NC(=O)C(O)CC1CCOCC1)N(CC)CC 92470,c1(C(c2nnnn2CC2CC2)NC(c2cc(Br)cs2)C)cc(F)cc2c1OCC2 92471,N1(CC(=O)NC(CNC(C(CC=C)NC(C)=O)=O)C)CCCCC(O)C1=O 92472,N1(C(C=NOC)=O)CC(NC(c2cnc(C)c(CC(C)C)c2)=O)CC(O)C1 92473,C1(CC(=O)NCCN(C(C)C)C(C23CC4CC2C3C4)=O)CCCN(C)C1 92474,CCC(C)CCC(=O)N1CCC(C(C)C(=O)N(C)CCC2CCCC2)CC1 92475,C1(CC)C(C(=O)NCc2[nH]cnc2C)CCCN1C(C1CC2(CC2)CO1)=O 92476,n1(CC(=O)N(C)CC2N(C(C(C)N(C)C)=O)CCC2)ccc2ccccc12 92477,Cn1cnc2c1CCC(C(=O)NCC1(CNC(c3ccc(CF)cc3)=O)CC1)C2 92478,N1(C(C(C)CCc2ccc(F)cc2)=O)CC2OCCN(C(C3CC(O)C3)=O)C2C1 92479,C1(CNC(CSCCC(C)C)=O)C2CCC(C2)N1C(C1CC(=O)N(C2CC2)C1)=O 92480,C1(C(N2CC(O)(CN(C(C3C(C(=O)OC)C3)=O)C)C2)=O)C(C)(C)C1(C)C 92481,N1(C(C(=O)NC(C)CN2CCOCC2)=O)CC2CCC1C1CNCC21 92482,C1(C)(CCC)CCN(C(=O)C(C)Cn2cccn2)C1.C1(=O)CC2(CC2)N1C 92483,Cc1ccccc1C(C)CC(=O)N1CC(NC(=O)OC(C)(C)C)C1 92484,Cc1cccc2c1CCOC2C(=O)Nc1ccc(F)c(C#N)c1Cl 92485,CC1CC(CNC(=O)CCC2CC2C)CN(C(=O)C=Cc2ncc[nH]2)C1 92486,CC(CF)CC(=O)N1CCC(C(C)CNC(c2ccn(C3CC3)n2)=O)CC1 92487,c1(N(C)C)nccc(C#N)n1.C1CCCNC1=O 92488,c1(OC)cc(NC(C2CC2NC(c2cccc(O)c2O)=O)=O)ccc1C 92489,CC(CCCCN=c1c(C#N)c[nH]c2cc(F)cc(F)c12)NC(=O)C1=CCCO1 92490,Cc1cc(F)ccc1C(N1CCOC(CNC(=O)C=CCOCC(F)(F)F)C1)=O 92491,C1(C(=O)NCc2c(C(N(C)CC3CCN(C)C3)=O)scc2)CCC(=O)NC1 92492,Cc1c(C=CC(=O)NCCCCC(C)NC(C23CCC(CC2)CO3)=O)cnn1C 92493,C(C(C)(CC(C)C)NC(C1CCOCC1(C)C)=O)NC(c1cccc(C)n1)=O 92494,N1(C(CCSC)=O)CC2CCCC(CNC(=O)CN3CCn4nccc43)C2C1 92495,C(=O)(C1=CC2(CN(C(C3CC=CC3)=O)C2)OC1)NC(CC=C)C(=O)OC 92496,S(=O)(=O)(c1c[nH]ccc1=NCc1ccc(C(N)=O)o1)NCC(COC)C 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92549,CC1(C(N2CCN(CCNC(=O)CC3CCSCC3)CC2)=O)COC(=O)N1 92550,C(c1ccc(C)cc1C)=CC(=O)NC1C(CNC(C2=CC(C)(CC)C2)=O)C1 92551,C1(C(=O)NC)(CC2(C(=O)NC(CC)CN3CCCC3)CC2)CC1(F)F 92552,CCCCCS(=O)(=O)NC(c1cncc(-c2ccncc2)c1)=O 92553,Cc1cc(N)c(F)c(C(=O)NC(CNC(=O)Cc2ccc(Cl)cc2F)CO)c1F 92554,Cc1cc(C(=O)N(CCC(C)NC(C2COCCN2CC(F)F)=O)C)ncc1F 92555,C1(C(=O)NCCN(C(=O)CC2CCCN2C(C)C)CCC)CCC(=O)N(CC)C1 92556,c1(C(N2CCC(O)(CC(=O)NCC3(O)CC(C)(C)C3)C2)=O)ccc(F)c(F)c1 92557,C(=O)(C#CC1CCCCC1)NC1CC2N(C(C(CNC(C)=O)(C)C)=O)C(COC2)C1 92558,C1(NC(CC2(CC)CCC2)=O)CCC(C(=O)N(C)CC2CC(F)C2)C1 92559,N1(C(C(C2CC2)OCC)=O)CCC(O)(C(C)NC(c2ccc(Cl)nc2C)=O)CC1 92560,c1(CC(=O)N(C2CCOCC2)CCOC)ccc(C(C)=O)nc1C 92561,c1(C(N2C(C)C(NC(=O)C=Cc3ncco3)CCC2)=O)ccc2ncccc2n1 92562,Nc1ccc2ccccc2c1-c1cccc(-c2ccccc2F)c1 92563,c1(OC)cc(C)cc(-c2nc(C)c(NCc3cc(F)cc(C#N)c3)s2)c1O 92564,c1(C(N2CCC(F)(CNC(C3(O)CCOC3)=O)CC2)=O)n[nH]c2c1CCCCC2 92565,N1(C(=O)NCCN(C)C)CCN(CCN2CCC(OC)CC2)C(=O)C1 92566,CC1CN(C(=O)CSc2nnc(S)s2)CC(C)C1NC(c1cccc(=O)o1)=O 92567,c1(OC)cc(CC(N2CC3(CCN3C(c3csc(C#N)c3)=O)C2)=O)ccc1C 92568,C(=O)(CC(F)(F)C(F)(F)Br)NCC(C)NC(c1ncc[nH]1)=O 92569,C1(C(=O)NCC(C)CNC(c2ccc(C(F)F)cc2)=O)C(C2CC2)C1(F)F 92570,N1(C(C(C)C)=O)CCOC(CNC(C2CCOC(=O)N2)=O)C1 92571,CCCC(O)C(=O)N1CC(O)CC1CNC(=O)CCC1OCCO1 92572,c1(OC(C)C)cc(=NC(=O)c2ccn(-c3ccccc3)n2)[nH]o1 92573,Cc1cc(CC(=O)NC2COCC2CNC(=O)CN2CCCCC2)cs1 92574,C12(C(=O)NC3(C#C)CCCC3)CCC(CN(C(=O)C(C)CCOC)C1)C2 92575,N1(C(C=NOC)=O)CC2(NC(C3CC3OC(C)(C)C)=O)CCCC2(F)C1 92576,N1(C(C2C(C=C)C2)=O)CC(CNC(c2cc(C(C)(C)C)n[nH]2)=O)C2(CC2)C1 92577,C(C(CC(C)(C)C)C(=O)N(C)C)N(C(=O)C(N)Cc1ccc(F)nc1)C 92578,c1(OCC)ccc(C(N2CC(c3cc(OC)ccc3O)C2)=O)cc1Cl 92579,C1(OC)CC(NC(c2ccccc2C2CCOC2)=O)CN(C(C2(C#N)CC2)=O)C1 92580,CCCC(CCCNC(=O)CC1CCSC1)NC(=O)CSc1cccc(Cl)c1 92581,CCCC(C(O)C(=O)N(CC(C)C#N)CC)NC(c1csnn1)=O 92582,O(NC(=O)CCOC)C(C(=O)N(CCOCC=C)C)C 92583,C(N=c1cc(NCCc2ccnnc2)nc[nH]1)C1(N(C)C)CCSC1 92584,c1(C(N2CC(CNC(C(C)CC#N)=O)C(F)(F)C2)=O)cc2cccnn2c1 92585,C=Cn1nncc1C(N1CCCC1(C)CNC(c1cccc(=O)o1)=O)=O 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92622,N1(C(c2c(C)c(C3CC3)[nH]n2)=O)CC2CCC(NC(=O)CN(C)C)CC2C1 92623,C1(NC(C2C(C)C2C)=O)CCS(=O)(=O)C12CN(C(=O)CCNC(c1ccoc1)=O)C2 92624,C1(CNC(C2(CC(C)C)CCNC2=O)=O)COCCN(C(C2(F)CC2)=O)C1 92625,C1(NC(c2[nH]cc(CC)c2)=O)C(C)CCN(C(=O)CC2CCCC(C)C2)C1C 92626,c1(C(=O)NC2(CCCNC(Cc3ccc(OC)cn3)=O)CC2)ccc(F)cc1F 92627,N1(C(C2CC3OC(C)(C)OC3C2)=O)CC2(CCC(NC(=O)CCCCO)CC2)C1 92628,c1(-n2c(C(C3CC4CCC3O4)NCCCCC)nnn2)ccc(OC(F)(F)F)cc1 92629,Cc1ncncc1C(N1CC(O)(C(C)(C)CNC(C2(C)CCN(C)C2)=O)C1)=O 92630,c1(OC)cccc(S(=O)(=O)N2CCC(C)(C(=O)NCc3c(F)cccc3Cl)C2)c1 92631,Cc1cc(NC(=O)Cc2ccc(C(N)=O)nc2)cc(C)c1 92632,Cc1nccc(C(=O)NC2CCC(NC(c3ccn(C(C)C)c3C)=O)C2)c1O 92633,C1(NC(C(COC)(C)OC)=O)CC2(C1)CN(C(=O)C(C)C1CCCC1)C2 92634,N12CC3(CC1CCO3)C2=O.C1(O)(CC#C)CC(NC(=O)C(=O)NCC(F)F)C1 92635,C1(N(CCO)CC)CCC(n2cc(-c3cnn(CCF)c3)nn2)CC1 92636,N1(C(CCC(C)c2ccccc2)=O)CC2(C1)CN(C(C13CC(CO1)C3)=O)C2 92637,C1(C(=O)NCC2CC(OCC)C2)(C(C)C)CCCN(C(=O)C(=O)N(C)C)C1 92638,N1(C(C(COC)(C)C)=O)CCCC(C2(NC(=O)C(F)C(F)(F)C(F)(F)F)CC2)C1 92639,c1(C(C)(C)C)nccc(C(N2CCCC2CCNC(c2cc(Cl)ns2)=O)=O)n1 92640,CC(C)C(O)CCN=c1nc2c(cnn2C)c(NCCc2ccc(N)cc2)[nH]1 92641,C1(CC(=O)NCc2c(C(=O)NC(C)CC3CC3)[nH]cc2)CCC2(CC1)CC2 92642,Nc1c(F)ccc(Cl)c1C(=O)NC1CN(C(c2cc(Cl)c(F)cc2F)=O)CC1F 92643,C=CCCC(C)N=c1[nH]c(=NCCCN2CCOCC2)c2cc(OC)ccc2[nH]1 92644,C1(N(C(c2c(C)sc(Cl)n2)=O)C)CCCN(C(=O)CCOc2ccccc2)CC1 92645,N1(C(c2c(N(C)C)cccn2)=O)CCc2cc(-c3cc(F)ncc3F)ccc2C1 92646,C#Cc1ccc(CC(=O)NC2CCCC2NC(=O)C(C)CCCOC)cc1 92647,C(c1ccccc1)=CCC(=O)N(C)C(N(CC(N1CCCC1CCCO)=O)C)=O 92648,C1(CCC(=O)NC(CC)C(F)(F)F)CCCCN(C(=O)Cc2csnc2C)C1 92649,C#CC1(C(N2CCCN(C)CC2)=O)CCN(C(=O)CC2CCCCO2)C1 92650,C(=O)(CCCCCCCC1CC1)NC(C(CO)NC(c1oc(CC)c(C)c1)=O)C 92651,C1(NC(c2c(C)nccn2)=O)CC2(NC(c3ccc(C(F)F)cc3)=O)COC1C2 92652,CC(CCO)C(=O)N1CCC(CNC(c2ccc(SC(C)C(N)=O)cc2)=O)CC1 92653,CCCC(C(O)C(=O)NCC(C)(C)CC)NC(=O)CCS(N)(=O)=O 92654,N1(C(COCC=C)=O)CC(O)CC1(C)C(N1CCOC2CCC12)=O 92655,C1(C)(C(N2CCN(CCC)CC2)=O)CC12CCN(C(=O)CCN(C)C)CC2 92656,N1(C(CN(C(C)=O)C)=O)CC(NC(c2cnc[nH]2)=O)CC(O)C1 92657,O=S1(=O)CCN(N2CCC23CCCC3)CC1.CO 92658,C(=O)(C1=NOC2COCC12)NCC(C(=O)NC(C=C)(C)C)(F)C(C)C 92659,C1(C2(O)CN(C(C3(CO)CC3)=O)C2)(CNC(C2CN(C)C(=O)N2)=O)CC1 92660,CCC(C)C(C)(O)CNC(=O)CC(C)N(C(=O)CSc1nc[nH]n1)C 92661,c1(C(N(CC(CNC(CC(C)SC)=O)C)C)=O)cc(Br)ccc1N 92662,C1(c2n(C)c(N3CCc4scnc4C3)nn2)Cc2ccccc2CN1 92663,N1(C(=O)CCC2CC(F)(F)C2)CCN2CCN(C(=O)C(F)C(F)(F)F)CC2C1 92664,c12cncc(c1)C(=O)NC1CCN(C1C)C(=O)CCC(=O)NC2.C(C)(C)(C)OC 92665,CC(CCNC(c1ccnn1C)=O)CCNC(c1ccccc1SC1CC1)=O 92666,c1(C(N2CCC(NC(C(c3cc(C)cc(F)c3)C)=O)C2)=O)cnn2c1OCCC2 92667,c1(N(CC(CC)OC)C)ccc(S(=O)(=O)NC(C2CCN(C)CC2)C)cn1 92668,Cc1cc(NC(=O)CC(CN)C2CC2)ccc1OC(F)F 92669,Cc1c(C(=O)NCC2CN(C(C3CCC4CC4C3)=O)CCCO2)cncc1Cl 92670,C12(NC(c3c(C)cc(C)[nH]3)=O)CCN(C(=O)Cc3cncnc3O)CC1C2 92671,C(CCCC(C)C)NC(C(C1CN(C(c2scc(OC)c2)=O)C1)O)=O 92672,c1(C(NOCC(=C)Cl)=O)ccc(OCCN(C)C)cc1 92673,C1(CCOCC)CCCOC1.C1CC(=O)N1.C1(=O)CCN(CC)CC2(CC2)N1 92674,Cc1ncncc1C(=O)NCCC1(O)CCN(C(=O)C(C)O)C1 92675,C(=O)(C(C)(C)C(=O)NCC(C)NC(c1c(C(F)F)cccc1C(F)F)=O)NC 92676,C1(CN(C(C(c2ccccc2)OC)=O)C)CCN(C(c2nc(Cl)sc2C)=O)CC1 92677,c1(C(N2C(CNC(C(CCCC)O)=O)CC(F)(F)C2)=O)cc2c(=O)[nH]ccn2c1 92678,N1(C(c2n(C(C)C)ncc2)=O)CCN(C(=O)Sc2cccc(Cl)c2)CC12CC2 92679,C1(CC(=O)NCCC2(C)CCN(C(=O)CSC(F)F)C2)CCC2(CCC2)O1 92680,c1(NC)scnc1C(N1CCC(C(=O)NCCCOC2CCC2)C1)=O 92681,CC(C(=O)NC1CC(C)(NC(C2COC(=O)N2C)=O)C1)C(F)F 92682,N1(C(C2CCCC(CC)C2)C(=O)NCC2CC2)CCC(S(=O)(=O)CC)C1 92683,c1(N2CC3CC(NC(c4cc(C)n(C(C)C)n4)=O)C3C2)nc2cc(Br)ccc2o1 92684,N1(C(C(CC)O)=O)C2CCC1CC(NC(c1cccc(N)c1C)=O)C2 92685,N1(CC(=O)NC(Cc2cn(CCCCOC)nn2)C)CCCC(C(=O)O)C1 92686,c1(C(N2CC(NC(c3cc(CC)on3)=O)C2)=O)c(Cl)cc(C)cc1Cl 92687,N1(Cc2nc(COC)sc2)CCC2(NC(=O)CC3CCCC(=O)N3)CCCC12 92688,CN=c1nc(N(CC(=O)N(C)C)C)[nH]c(=NCC(CO)C2CC2)[nH]1 92689,c1(OC)ccc(Br)c(C(=O)NCC2CCN(C(C3CNC(=O)C3)=O)CC2)c1 92690,c1(N(CCOCC)C)nnc(C2CCC(=O)N2)n1Cc1sccc1C 92691,C1(NC(C2(COC)CC2(F)F)=O)CCCCC1NC(=O)C(CCO)N(C)C 92692,C(=O)(C(=O)CC(C)C)N1CC(C(C(=O)NC(CCC)c2ccco2)O)C1 92693,CCC(C)C(C(=O)N1CCCC1C1(C)CC1)N(C(=O)C(C)CC1(OC)CCCC1)C 92694,C(=O)(CCCCCCNC(=O)Cc1csc2nc(C)cn12)N1CC(F)(C(=O)OC)C1 92695,c1(C(=O)NCC2(C)CCC2)ccc(CNC(c2csc(Cl)c2)=O)s1 92696,N1(C(C(CSC)(C)C)=O)CCC2(CCN(CCOc3cc(F)ccc3F)C2)C1 92697,c1(C(N(C)CC2CN(C(CC3C(C)CCO3)=O)C2)=O)cccc(=O)n1O 92698,Cc1sc(Cl)nc1C(N1CC(C(C)NC(=O)C(C)Cc2cccnc2)C1)=O 92699,N1(C(c2c(C)n(C(C)C)cc2)=O)CCC2CCC12CNC(c1ccnc(O)c1)=O 92700,C1(NC(C(C)(Cl)Cl)=O)COC2(CCN(C(C3CCn4ccnc4C3)=O)CC2)C1 92701,C1(C)(NC(CCSC)=O)CCN(CCCOc2ccccc2Br)C1 92702,c1(C(=O)NC2CN(C(CC3CCC(OC)CC3)=O)CC2SC)cccc(F)c1O 92703,C1(C(=O)NCC=CCNC(c2cnc(O)s2)=O)(C(F)F)CC(F)(F)C1 92704,Cn1cccc1C(=O)NCCCCCNC(=O)CC1(C)CC1(F)Cl 92705,C(=O)(C(C)(C)C(C)C)NCC(C)(C)CN(C(CC(=O)NCCNC(C)=O)=O)C 92706,CC1(C)C(C(c2nnnn2C2CCCC2)NCCn2ccnn2)C1(C)C 92707,CCN=C(NCCc1ccccc1Br)N1CCC(C(c2cccc(C)c2)=O)C1 92708,c1(CC(=O)NCC2N(C(C(C)(O)C3CC3)=O)CCC2)ccc(CC2CC2)c(F)c1 92709,C1(C2CC2)(C(N2C(C)(CC(C)C)CCC2)=O)CN(C(c2ncn3c2CCC3)=O)C1 92710,c1(C(N2CC(C(N)=O)(CNC(C3(F)C(C)OCC3)=O)C2)=O)scc2c1CCCC2 92711,O=S(=O)(c1c[nH]ccc1=NC1CCN(c2ccc(Cl)cc2)CC1)NCCCO 92712,C1(NC(C(CSC)OC)=O)COCCN(C(=O)Cn2cc(Br)ccc2=O)C1 92713,C1(NC(Cn2cc(CC)nn2)=O)CCCC2CN(C(c3cc(F)n(C)n3)=O)CC12 92714,c1(CC)c(C(N2CCOCC2CNC(c2ccc(F)s2)=O)=O)cnn1C(C)(C)C 92715,C12(C(N3CCC(C(C)NC(c4ccc(F)s4)=O)CC3)=O)CCC(C1)C(C)(C)O2 92716,c1(N2CCN(C(C)=O)CC2)nc2c(F)cc(F)cc2c(=NC(C)c2nc[nH]n2)[nH]1 92717,C(CNC(C1(C(F)F)CCC1)=O)(CC(F)(F)F)NC(CSc1n[nH]c(=N)s1)=O 92718,N1(Cc2cccc(OC)c2C)CC2CN(C(c3ccc(N(C)C)nc3)=O)CC2C1 92719,C12(C(=O)NCC3(CNC(=O)C=Cc4cncs4)CCCC3)OCCCC1C2(F)F 92720,C1(NC(c2n(C)c(Cl)cn2)=O)CCN(C(c2c(F)cccc2Cl)=O)CC12CCC2 92721,c1(N(C)C)ccc(F)c(NC(=O)Nc2cc(OC(F)(F)C(F)Cl)cc(Cl)c2)c1 92722,N1(C(=O)Cc2csnn2)CCCC(c2cn(Cc3ccccc3)nn2)C1 92723,C=C1CC2CCCC(C1)N2C(=O)C(CNC(=O)CCc1cscn1)CC(C)C 92724,C12(C(=O)NCC(CNC(c3c(CC)n(C)nc3)=O)(C)O)CCC(C1)S(=O)(=O)CC2 92725,c1(NC(C2CCCN(CC)C2)=O)ncnc2c1ncn2C1CC(O)C(O)CC1CO 92726,N1(C(CCOC(C)C)=O)CCCC1C=CC(N1CC(F)C1)=O 92727,Cc1[nH]nc(C(N2CCCC(NC(C3CC3c3ccccc3)=O)C2)=O)c1Cl 92728,c1(C(N2CCCC(NC(C3(CC=C)CC3)=O)C2)=O)c[nH]c2cc(Br)ccc12 92729,CC1=CCSC1C(=O)N(C1CCN(C(c2cnc(Cl)[nH]2)=O)C1)C 92730,CCC1=NOC(C(N2CCC(C(C)(C)C(=O)NCCCc3nccs3)C2)=O)C1 92731,c1(C(C)OC)nc(C(=O)NC2CC(CCNC(c3cc(Cl)cs3)=O)C2)cs1 92732,N1(C(C(C)N2CCCC2)=O)CC2C=CC1C(C(=O)NCCc1cn(C)cn1)C2 92733,O=C(C1=CCCOCC1)NC(CO)C(=O)NCCCc1cnn[nH]1 92734,N1(C(C(C2CC2)OC)=O)CCN(C(c2cc(C)nc(C)c2)=O)C(C2CC2)C1 92735,C(=O)(CC(C)CNC(=O)C(C)(C)CC1CC1)NC(c1ccc(C)s1)C 92736,N1(C(C2C(OC)C2)=O)C2CCC1CC(OC1(C(=O)Nc3ccc4c(c3)CCC4)CC1)C2 92737,C1(C)(NC(C(N2CCC(C)C2)=O)=O)CCN(C(C2CCC(F)(F)CO2)=O)CC1 92738,N1(C(CCCCCC#C)=O)CC2CCCC(NC(C3CCNC3=O)=O)C2C1 92739,c1(CC(=O)NC2CC(C)N(C(c3cc4sccc4[nH]3)=O)C2)cccc(F)c1Cl 92740,c1(-c2cn(CCNC(C3CC(c4scc(C)n4)C3)=O)nn2)ccccc1S(C)=O 92741,c1(C(C(F)(F)F)OC(C(c2n(C)cnc2)O)=O)cccc(C(F)(F)F)c1 92742,c1(NC(C=Cc2c(C)n(C)nc2)=O)ccc2c(c1)C1(CCCCC1)C(=O)N2 92743,c1(C2CN(C(=O)CC3CC3c3cc[nH]n3)C2)cc(O)nc(O)n1 92744,c1(CCC(=O)NC(Cc2cn(CCSC)nn2)C(=O)O)ccc2c(c1)CCCO2 92745,c1(N2CCC(N(C)C(C3(C)CCC(=O)N3)=O)CC2)ncc([N+](=O)[O-])c(=N)[nH]1 92746,C(=O)(CCC(C)C#N)NCC1CC(NC(c2c(CC)nn(C)c2)=O)C1 92747,C1(C)(C(=O)NCC(C)NC(C2CC(CC)(CC)C2)=O)CCC(C)C1 92748,C(=O)(CCC(C)(C)NC(=O)C(C)CC#N)N1CCC(OC(C)=O)C1 92749,Cc1ccc(O)nc1CNC(=O)CC(C)(C)CNC(C1OCCC1C)=O 92750,C(C(CC(C)C)C(=O)NCC1COCC(=O)N1C)NC(C(CC=CC)C)=O 92751,CC(C)C(C(=O)N(C)CC1CCN(C(c2ccncc2Cl)=O)C1)NC(N)=O 92752,Cc1cc(C)c(C(N2CCCCCC2CNC(c2nccnc2N)=O)=O)cc1N 92753,c1(C(=O)NCC2CC(OC)CN2C(C2CC(SC)C2)=O)cc(Cl)cc([N+](=O)[O-])c1 92754,c1(C(N(CCN(C(=O)C2=NOC(C)C2)CC)CC)=O)cc(C)nnc1O 92755,c1(OCCC)cc(N)c(F)cc1CNC(CCC1Sc2ccccc2O1)=O 92756,C(=O)(C(C)(C(C)C)OC)N1CCC(CCNC(CC(C)SC)=O)CC1 92757,c1(C(=O)NC2CC(CC(=O)N(C3CN(C(C)C)C3)C)C2(C)C)cc(C#N)cn1C 92758,C1(NC(C(CC)CO)=O)CC2(CCN(C(C3C=C3C)=O)C2)C1 92759,C1(CNC(Cn2c(CCC)nnc2S)=O)CCN(C(=O)C2=CC(C)(C)C2)C12CC2 92760,c1(C(=O)NCC2(O)CCN(C(CCc3nc(C)sc3)=O)C2)cccc2cncn12 92761,C(=O)(C(C)(C)CS(C)(=O)=O)NC(c1c(CC)cccc1)CNC(C1CC1F)=O 92762,c1(NC2CC(C(C)=NO)C2(C)C)ccnc2cc(Br)ccc12 92763,Cn1nc(CNC(C2CCCSCC2)=O)cc1Nc1ccccc1 92764,CC1CN(C(C2(CCF)CCOCC2)=O)CC(C)N(C(=O)Cc2csc(Cl)n2)C1 92765,c1(C(=O)NCC2C(NC(C3(C(N)=O)CCC3)=O)C2)cccc(F)c1F 92766,C=CCCCCC(=O)NC1(CNC(c2cc(CCC)oc2C)=O)CCC1 92767,c1(CC(=O)NCC2OCC(CNC(C3(CC=C)CC3)=O)C2)ccccc1C(N)=O 92768,N1(C(C(CC)F)=O)CCN(C(C2(CO)COC2)=O)CC1c1cnn(C)c1 92769,c1(CC(N2C(CNC(C3CC(O)C3)=O)CCC(C)C2)=O)nnc2n1CCOC2 92770,Cc1cc(CNC(C2CCN2C)=O)oc1C(=O)NCCc1[nH]cnc1C 92771,C1(C(C)C)N(C(C2(CO)CCN(C(c3ccc[n+]([O-])c3)=O)C2)=O)CC1(C)C 92772,N1(CC=C)CCCN(C(=O)CC2C3CN(C(=O)C=C(C)C(F)F)CC23)CC1 92773,C(=O)(C(CC(C)(C)C)OC)NC12C(NC(CNC(=O)OC)=O)CC(CC1)C2 92774,C1(CC(=O)OC)CC(C(N2CC(c3ccccc3)C2(C)C)=O)CCO1 92775,C1(NC(=O)NC2CCN(Cc3ccccn3)C2)CC2(CCC2)CO1 92776,c1(SCC#C)cccc(C(=O)NC(C)CCCNC(=O)C(C)OCC(C)C)c1 92777,N1(C(c2n(C)ncc2)=O)CCC(C2(NC(c3coc(O)n3)=O)CC2)CC1 92778,CC1=CCN(C(C2(N(C)C(c3ccoc3C)=O)CC2)=O)C1 92779,c1(C(=O)NCC2(NC(C3(CC)CCCCO3)=O)CCCCC2)n[nH]c2c1CCC2 92780,c1(C(=O)NCCCC2(NC(COCCCOC)=O)CC2)ncnc2sccc12 92781,Cc1cnc(F)c(CNC(=O)C(c2ccoc2)NC(=O)C2=CCCCC2)c1 92782,N1(C(CN(C2CCC2)C)=O)CCCCC12CN(C(C1(c3ccno3)CC1)=O)C2 92783,c1(NC)cnc(Cl)cc1C(=O)NC(C1CCN(C(C2CCCC(=O)N2)=O)C1)C 92784,c1(SC)nc2nc(C)c(CC(=O)NC3COC4(CCN(CCF)C4)C3)c(C)n2n1 92785,C1(C(N(C)CC2CCSC2)=O)C2CC3C(C2NC(c2cc(=O)n(C)cn2)=O)C13 92786,N1(C(C=C(C)C)=O)CCc2ccccc2C1CNC(=O)CC1NC(=O)NC1=O 92787,c1(NC(=O)NC(CC)COCC(F)(F)F)cc(OC)c(Br)cn1.c1cccc(C)c1 92788,c1(C(CNC(N2CC(NC(C3CCCO3)=O)C2)=O)OC(C)(C)C)cccnc1 92789,Cc1cc(C(N2CCC(NC(c3cc(-c4ccccc4)co3)=O)C2)=O)cs1 92790,N1(C(C2CCC(NC(C3CC(C)(F)C3)=O)C2)=O)CC(CO)C(CO)C1 92791,N1(C(c2c(CC)nco2)C(=O)NC)CCN(Cc2nccs2)C(C)C1 92792,C=CCCCCC(=O)N1CCCOC(CNC(=O)CC(C)(C)C#N)C1 92793,c1(C(=O)Nc2c(CC)ccnc2)cnc2c(-c3csc4ccccc34)cnn2c1 92794,N1(C(CC(=O)OCC)=O)CCCC1(C(N1CC(F)(C(N)=O)C1)=O)CC 92795,C1(O)(C(C)NC(c2cnccn2)=O)CCN(C(c2nn(C)cc2N)=O)C1 92796,C1(CN(C(COCCCC(C)C)=O)C)CN(C(C2CCCCS2)=O)CCO1 92797,Cc1nnc2cc(N3CCCC(CCNC(=O)CC=C(Cl)Cl)CC3)ncn12 92798,c1(OC)cncc(C=CCC(=O)NCc2cn(C)nn2)c1 92799,c1(C(N2CCS(=O)(=O)C(C3CC3)C2)C(=O)NC)ccc(F)c(C)c1Cl.C(C)OC 92800,c1(C(c2nnnn2C2CCOC2)NCC2(COC)CC2)cc(Br)c[nH]1 92801,CC1CCN(C(=O)C=CBr)C1CNC(=O)C=CC1CCOC1 92802,c1(NCc2c(OC)cccc2)nc(N2CCC(NCC(F)CO)CC2)cc(C)n1 92803,Cc1ccc(C(N2CC(CC(F)C(=O)N3CC(O)(c4cnn[nH]4)C3)C2)=O)[nH]1 92804,C1(CC(=O)N(C2CCCC2C(N2CC(N3CCC3)C2)=O)C)CC(O)C12CCC2 92805,C1(C2CCN(C)CC2)(C(=O)NC(CC)CNC(=O)CCC2CC2(F)F)CC1 92806,C(=O)(C1=C(Cl)CCCC1)NC1C2CN(C(C3CC(C(=O)OC)C3)=O)C1C2 92807,O=S(=O)(c1cccc(=NCCC2(C(F)(F)F)CC2)[nH]1)N1CC=CC(O)C1 92808,CC(C)CC(C)C(=O)NCC12CC(CN1C(c1ccnc(Cl)c1O)=O)C2 92809,c1(C(=O)NCC2CN(CCn3ncnn3)CCO2)c(Cl)cccc1[N+](=O)[O-] 92810,C(=O)(C(C)(O)C(C)(C)C)NCC(CN(C(=O)CSc1ccccc1[N+](=O)[O-])C)O 92811,Cc1cc(CC(=O)N(C2CN(C(=O)C(c3cncnc3)C)CC2O)C)c(C)s1 92812,n1(CCC(=O)OCc2cccc(OC)n2)nc(C)c(C)c1C 92813,N1(C(C2N(C(CCc3cn(C)nc3)=O)CC=C2)=O)CCCc2occc2C1 92814,N1(C(C2(CCC)CCNC2=O)=O)CCC(CNC(=O)C(CC)SC)(COC)CC1 92815,c1(NC(N2CCN(CCNC(C3C(=O)NCC3)=O)CC2)=O)cccc(F)c1O 92816,c1(C(=O)NCC2CN(C(C3CCC3)=O)CC2(F)F)c(Br)ccc(F)c1F 92817,N1(C(Cn2ncn(C)c2=O)=O)CCCC1C1CCCN1C(=O)CC1CCC2CC12 92818,c1(C(=O)NCC2(NC(C(CC3CCC3)OC)=O)CC2)ccn(C(C)C)c1C 92819,C1(NC(c2cnc(OCC)s2)=O)CN(C(c2ccn(CCF)n2)=O)CCC1CO 92820,C12(C(N3CC(C(C)NC(=O)CCCN(C)C)C3)=O)CCCCC1C2 92821,Cc1c(CNC(=O)C=CCC(C)(C)NC(=O)Cc2cccnc2O)nnn1C 92822,C1(NC(c2ccc(C(C)C)s2)=O)CCC(NC(=O)CCC2CCCCN2C)CC1 92823,N1(CCN2CCC(C)CC2)CC(NC(C2(c3ccccc3Cl)CC2)=O)CCC1C 92824,N1(C(CC2(C)CCCO2)=O)CC2CCCC2(NC(c2cc[nH]c2)=O)C1 92825,N#Cc1cccnc1-c1csc(Nc2cc(C(F)(F)F)ncn2)n1 92826,c1(CNCC(COC)OC)ccc(-c2cc(C(C)=O)ccc2OC)cc1F 92827,C1(C(C)(C)C)CCC(C(=O)NCC(C2CCC2)NC(c2ccncc2O)=O)CC1 92828,c1(OC)csc(C(c2nnnn2Cc2cccs2)NCCCF)c1OC 92829,C1(CC)CN(C(c2ccsc2C#N)=O)CC1C(N1CCOC(C)C1)=O 92830,C1(C(=O)NCC(C)(C)NC(c2nnc(C)s2)=O)CCCC(F)(F)CC1 92831,c1(N(C(=O)Cc2cc(C(=O)O)on2)C2CC2)nc(Br)ccc1Br 92832,c1(C(N2C(CCCNC(C3(C)CC3(Cl)Cl)=O)CCC2)=O)ncc(F)cn1 92833,C1(CC)CN(C(C23CCC(F)(CO2)C3)=O)CCN1C(c1ccc(NC=O)cc1)=O 92834,c1(OC)cc(O)c(NC(c2ccnn2CC2(C)COC2)=O)cc1C 92835,C1(CC)CCCN(C(C2COCC2(C)C)=O)C1C(=O)NC1CCCCOC1 92836,c1(C(N2CCC(C(C)NC(=O)C3=CCCCC3)C2)=O)nc[nH]c2ncnc1-2 92837,c1(C(N2CC(O)CC(NC(C3(C=C)CC3)=O)C2)=O)ccc2c(OC)ncnc2c1 92838,c1(C(=O)NCCCN(C(C(C)OC)=O)C)c2c(c[nH]c1=N)CCC2 92839,C1(NC(c2n(C)nnn2)c2ncc(-c3ccccc3F)o2)Cc2cscc2C1 92840,c1(C(N2CC(CNC(=O)C3=CCOCC3)OCCC2)=O)cncc2ccsc12 92841,C=CCC(C(=O)NCCCCNC(c1cnn(C)c1Br)=O)NC(C)=O 92842,C1(C(=O)NCCN(C(=O)OC)C)(NC(C2CC(F)C2)=O)CCOCC1 92843,C12(C(=O)NC(CC)CN(C(=O)CSCCOC)C)CCCC1C2Br 92844,C1(NC(C(C)OC)=O)(CNC(c2cnnn2C(C)C)=O)CCC(F)(F)CC1 92845,C(CCCCC(=O)N1CCC(NC(c2cn(C)c(C)n2)=O)CC1C1CC1)SC 92846,N1(C(C(C)C(C)O)=O)CCC2(CC1)CC(NC(=O)Cn1nc(C(F)F)cc1C)C2 92847,c1(C(N2CCN(C(CCC)=O)CC23CC3)=O)nccc2ccncc12 92848,c1(OC)c(C(N2CC3CCC3(NC(=O)CC3(C4CC4)CC3)C2)=O)c(C)nn1C 92849,C1(C(=O)NC2CC(CNC(c3sc(C)c(O)n3)=O)C2)CCCC(F)(F)CC1 92850,c1(C(=O)NCC(C)NC(c2ccc(C3(CC)CC3)cc2)=O)cc(=O)c(Br)c[nH]1 92851,C1(CNC(C(C)c2ccsc2)=O)COCCN1C(c1sccc1Br)=O 92852,C(=O)(CC1=CCOCC1)NCC(CC(C)C)(C)NC(=O)Cn1ncnn1 92853,CC1(NC(=O)C(Cl)Cl)CCCCC1C(=O)NCC1CN(C2COC2)C1 92854,c1(C(C(=O)NC(CC)CN(C(=O)CCc2ncc[nH]2)C)OC)cccc(OC)c1 92855,N#Cc1ccc(C(=O)N(CCCNC(c2cccn(O)c2=O)=O)C2CC2)cc1 92856,Cn1ncc([N+](=O)[O-])c1C(=O)NCCC(C)(C)NC(C1CC1c1cccnc1)=O 92857,N1(C(C=Cc2c(C)ccnc2)=O)CC2CCC1CC2NC(C1CC12CCOC2)=O 92858,C1(Cc2nc(C)[nH]n2)CCN(C(=O)C(=O)NC2CCOC2C(C)C)CC1 92859,c1(COC)ccc(C(N2CC(NC(C3(C4CCCCO4)CC3)=O)C(O)C2)=O)cc1 92860,Cc1ncc(C=CC(=O)NCC2(F)CC(NC(=O)CC(=O)N(C)C)C2)c(O)n1 92861,N1(C(CC2C(=O)NCCC2)=O)Cc2occ(C(N3CCC3C3CCC3)=O)c2C1 92862,C1(C(N)=O)(OC)CC(CC#N)CN(S(=O)(=O)CCCC#N)C1 92863,C1(CNC(CC(C=C)(C)C)=O)CN(C(=O)CCC(C)N(C)C)C2(CCC2)C1 92864,CCCCC(CC(=O)NCC1(C(C)C)CC1)NC(C1(C2(C)CC2)CC1)=O 92865,C(=O)(C(C)(C)CCCNC(C1CCCN(C)C1)=O)NCc1ccc(CC)o1 92866,c1cc(CCNCc2ccccc2)c2c(c1)CN(c1ccc3nnnn3n1)CC2 92867,Cc1c(C2(NC(C3CCC(C)CC3)C(F)(F)F)CC2)cccc1Br 92868,CON1CCC(C(=O)NCC2CC3CN(C(C4CC(N(C)C)C4)=O)CC23)CC1 92869,C1(C(=O)NC2(CC=C)CN(C(=O)Cn3nc(C)cc3N)C2)CC(=O)N(CCC)C1 92870,c1(C(N2CC(OCCNC(CC3(C=C)CCOCC3)=O)C2)=O)ccc2cnoc2c1 92871,c1(C(=O)NCC(CCNC(C2(OC)CCCOC2)=O)O)cnc(C(F)F)c(C)c1 92872,Cn1cccc(C(=O)NCC2CCN(C(C3(CC(F)(F)F)CC3)=O)CC2)c1=O 92873,c1(CC)ccccc1OCCC(=O)N1CC(CNC(=O)C=Cc2csc(C)n2)C1 92874,N1(C(C=CC(C)(C)C)=O)CC2CC(NC(c3ccc4nnnn4c3)=O)CC2C1 92875,c1(CC(=O)NC2(C)CC(NC(CCSCC)=O)C2)ccc(F)cc1F 92876,C1(C#C)(C(=O)NCCOCCCC#C)CCN(C(C2CCC(=O)O2)=O)CC1 92877,c1(CCC(=O)NC(CNC(CNC(C(CC)C)=O)=O)CO)cccc(O)c1 92878,C(c1cnn(C)c1)=CC(=O)NC1(C2N(C(CCOCC)=O)CCC2)CC1 92879,c1(CC)cccnc1C(=O)N(C(C)CNc1cccc(OCCN(C)C)c1)C 92880,CC(C)(C(=O)NCC=CCNC(C1CNC(=O)C1)=O)c1ncco1 92881,c1(CNC(c2c(C(C)C)n[nH]c2)=O)cccc(NC(=O)CCc2cnccn2)c1 92882,c1(C(C)(C)NC(C2CC(NC(=O)OC(C)(C)C)C2)=O)cccc2c(Br)ccnc12 92883,CC(CF)CC(=O)NCC1(CCCNC(=O)C(C)N(C)C)CCCC1 92884,C(=O)(C1CCCc2nc[nH]c21)N1CCCC(NC(c2cccc(F)c2)=O)C1 92885,CCC(CC(=O)N1CCOCC(CNC(c2ccn(C3CC3)c2C)=O)C1)C(C)C 92886,C(CC(C(C)(C)C)NC(C1CC(=O)CC(=O)N1)=O)N(C(=O)C=Cc1ccsc1)C 92887,C(=O)(C#CC1CCOCC1)NCC1(C(C)NC(C2CC(F)(F)C2)=O)CC1 92888,c1(C(=O)O)ccc(S(=O)(=O)NC2CCN(C(=O)CC(F)(F)F)CC2)c(Cl)c1 92889,C1(CCN(C)C)CCN(C(=O)CN(C)C(C2(C)C=CCC2)=O)C1 92890,C(C(C(C)(C)C)NC(C1CC1c1ccsc1)=O)NC(c1cnc(OC)s1)=O 92891,CC1C(NC(c2ccn(CC#N)n2)=O)CCN1C(C1COCCO1)=O 92892,C12(C(N(C)CC3CN(C(=O)CC4=CCCC4)CCO3)=O)CCCC(C)(C1)OC2 92893,N1(CC(=C)Br)CCCC(CN(C(c2cc(OC(C)C)ccn2)=O)C(C)C)C1 92894,C(=O)(CCCC(C)NC(c1[nH]cc(C)c1C)=O)NCC(C)NC(=O)OC 92895,CC1CCC(NC(C2CC(C)(C)C2C(F)(F)F)=O)CN1C(c1cc2c([nH]1)CCC2)=O 92896,C(=O)(C(CC(F)F)C1CCC1)NC(CNC(=O)COc1cccc(F)c1F)CO 92897,C1(NC(CC2C(C)C2)=O)C2CC1N(C(=O)CCOc1ccccc1O)C2 92898,C12(NC(c3snc(O)c3Cl)=O)CCC1CN(C(=O)CCOc1cccnc1)C2 92899,N#Cc1ccc(CCC(=O)NCCc2cccc3sccc23)c(F)c1 92900,CC1=NOC(C)(C(=O)N(C)CC2CN(C(C3COC(C)(C)O3)=O)CCO2)C1 92901,N1(C(c2ccnc(Cl)c2)C(=O)NCC2CC2)CCC2(CC1)OCc1ccncc12 92902,N1(C(C(CC)C(C)C)=O)CCCC2C1CCN2C(c1cc(F)c(F)cc1O)=O 92903,c1(C(N2C3(CNC(CC(C=C)C)=O)CCCC(C2)C3)=O)ccc2oc(C)nc2c1 92904,C(=O)(CS(=O)(=O)CC(C)C)NC(C1(O)CCN(C(C(CC)CC)=O)CC1)C 92905,S(=O)(=O)(c1cnc2nc(O)nc(O)c2c1)NC(c1ccc(Br)cc1)COC 92906,N1(C(c2cnc(CC)[nH]2)=O)CC(C)N(C(=O)Cc2coc3ccccc23)CC1C 92907,Cc1noc(C)c1CCC(=O)NCC1(F)CN(C(=O)COCC2CCCC2)C1 92908,N1(C(C(C)NC(CC)(C)C)=O)C2CCC1C(CNC(=O)COCC(F)F)C2 92909,c1(C(=O)NCCC(=C)CNC(=O)C(C)Oc2ccc(SC)cc2)csc(C#N)c1 92910,C1(NC(C(C)C#N)=O)CS(=O)(=O)C2CN(C(c3nnn4c3COCC4)=O)CC12 92911,C1(=O)C(C)N1C1CCCC1.C1(C(=O)OCC)(NC(=O)COC)CC1 92912,C(CN=c1ccn2c(Br)cnc2[nH]1)C1(OC)CN(C(c2cn(C)nc2OC)=O)C1 92913,N1(C(C(CC#C)C2CC2)=O)C2CCC1CN(C(=O)C(C)C1CCC1)C2 92914,CCCC(O)C(=O)NC(C(N1CCC(CN(C)C)C1)=O)C1(C)CC1 92915,N1(C(C(C=C)OC)=O)CCN(C(=O)Cc2c(C(F)(F)F)coc2C)CC1CCO 92916,c1(OC)ccc(CN2CCC(CC(N3CCCC3C(N)=O)=O)C2)c(Br)c1 92917,C1(CNC(C=CC(C)=O)=O)CCN(C(=O)Cn2cnnn2)C1(C)C 92918,c1(CC(N2CC(NC(C3CCC3)=O)C3C2C3)=O)cc(F)cc(Br)c1 92919,CCC(O)C(C)(C)C(=O)N1CCC(Cn2cc(CN(C(=O)CCCN=[N+]=[N-])CC)nn2)C1 92920,S(=O)(=O)(CC(=O)N1CCCC(N(C(=O)CC2CCCCN2CCF)CC)C1)NC 92921,CC1(C(N2CCC(CNC(C3(CCF)CCOCC3)=O)C2)=O)CC=CCO1 92922,c1(C(=O)OC(C)C)csc(NC(=O)CSc2n[nH]c(O)n2)n1 92923,Cc1ncc(Br)cc1NC(C1CN(C(=O)C(C)S)CCC1O)=O 92924,c1(CNC2CC(C(N3CCN(CC#C)CC3)=O)C2)cccc2nc[nH]c12 92925,Cc1cc(N)cc(C(=O)N(CCCNC(=O)C(c2ccccc2F)C)C)c1F 92926,c1(C(C)C)cccc(C(N2CCCCC2CNC(=O)C(C)(C)c2cscn2)=O)c1 92927,C(CN=c1[nH]c(=NCC2CCCN(CCCO)C2)[nH]c2c1COC2)OCCO 92928,c1(C(N2CC(NC(c3n(C(C)C)ncn3)=O)C2)=O)cccc(OCC(F)F)c1 92929,N1(C(C2CCCC2)=O)CCN(C(=O)C=CC2CCCCC2)C(c2ccncc2)C1 92930,c1(C(=O)NC2CN(C(C3(C#C)CCCC3)=O)CC2O)ccc(Cl)c(C)c1Cl 92931,N1(C(CCSCC)=O)CC(CNC(=O)Cc2ccc(C)c(OC)c2)C(F)(F)C1 92932,C1(C(=O)NC2C(CNC(=O)Cn3cnc([N+](=O)[O-])n3)C2)CCC2(CCCCC2)C1 92933,c1(OC)ccc(O)c(C(=O)NC2CC(CCNC(C3CC3Br)=O)C2)c1 92934,c1(C(=O)NCCC2CC(Nc3c(C)c(Cl)ncn3)C2)c(C)cc(=O)oc1C 92935,N1(C(c2c(C)noc2)=O)C2CCC1CN(C(=O)C(C)CC1CCC1)C2 92936,O(NC(=O)CC(C)N(C(=O)Cc1ccnn1C)CC)CCOCC 92937,N1(C(C2(C)CCCO2)=O)CCCN(C(c2nc(=N)cc[nH]2)=O)C(CO)C1 92938,C1(C(N(C)CC2C3CN(C(=O)CCCCCN(C)C)CC23)=O)CC2(C1)CC(CF)C2 92939,C=C(C)C(CC(=O)N1CCCC(N(C(C)C(=O)N(C2CC2)C(=O)C2CC2)C)C1)OCC 92940,c1(C(=O)NCC2(C)CC(NC(c3ncc(CC)cn3)=O)C2)c[nH]cc(C)c1=O 92941,CCC(CCSC)C(=O)N1CCOC(NC(=O)CNS(N)(=O)=O)C1 92942,c1(NCC2C(NC(c3cc(OC)ns3)=O)CC2)nc(C)ccc1C(=O)OC 92943,Nc1nonc1C(N1CC(OCC(=O)NC2(C3CCCO3)CC2)C1)=O 92944,N1(C(c2cc(C)cc(C)c2)=O)CCCC2(NC(c3ccnnc3C)=O)CC2C1 92945,CC1OCCN(C(=O)CC2CC(NC(C3CC4(CCC4)C3)=O)C2)C1CO 92946,N1(C(CCSCCCC)=O)CC2CCCN(C(c3ncoc3C)=O)C2C1 92947,C1(NC(CC2C(C)(C)C2)=O)CC2(CCCN(C(c3c(Cl)csc3Cl)=O)C2)C1 92948,c1(NC(N(C(C2CCCO2)COC)C)=O)ccc(C(C)C)cn1 92949,c1(C(=O)NC2C=CC(CNC(C3CN(OC)C(=O)C3)=O)C2)ccn2c1CCCC2 92950,Cc1cccc2[nH]cc(C(N3CC(C)(NC(C4CCC(C5CC5)C4)=O)C3)=O)c12 92951,N1(C(c2ccc(OC)nn2)=O)CCCC(F)(CNC(=O)CC2CCC(O)C2)C1 92952,N1(C(=O)CCCN2CCCC2)CCC2(C1)CN(C(=O)C1=COCCC1)C2 92953,C(=O)(C1CSc2ccccc21)N1CC(OCCNC(C2CN3CCN2CC3)=O)C1 92954,C1(CNC(C2(C)CC3CC3C2)=O)CC(C(F)(F)F)CCN1C(=O)CCCN=[N+]=[N-] 92955,C(=O)(C1=NN(C2CC2)C(=O)CC1)N1C(CNC(CCSCC)=O)C(C)(C)CCC1 92956,C(C(C(=O)NCc1nccn1CC)C(C)(C)C)NC(c1oc(CC)c(C)c1)=O 92957,N1(C(c2c(CC)[nH]nc2Cl)=O)CCC(NC(=O)CCn2ccnn2)C(CC)C1 92958,CC(C)(C(=O)Oc1cc(F)cc(F)c1)C(F)F.N1(CCl)C(=O)NC(CC)C1=O 92959,C(=O)(C(C)CCCC(C)C)NC(CC=C)CNC(=O)C=CC(=O)N(C)C 92960,N1(C(C2(COC)C=CCC2)=O)CCC(CF)(NC(=O)CN2C(=O)CNC2=O)C1 92961,c1(C(N2C(CNc3cc(OCC)ncn3)CCCC2)=O)ccc(C#N)nc1C 92962,N1(C(c2cnc(C)nc2C)=O)CCCC2(CCN2C(c2cnc(Cl)c(I)c2)=O)C1 92963,CCC(O)C(C)(C)C(=O)N(CC(O)CN(C)C(c1nccnc1OC)=O)C 92964,c1(C(=O)NCC(CCNC(c2ccc(C#C)cc2)=O)O)c(C)cc(C)cc1C 92965,c1(OCCC(=O)NCC#CCNC(C2(CC#C)CC2)=O)cccc(C(N)=O)c1 92966,C1(CNC(C(C)n2cccn2)=O)(CN(C)C)CCN(C(=O)Cc2cscn2)CC1 92967,N1(C(COCC)=O)CCCCC1C(C)NC(c1cnn(C(C)C)c1F)=O 92968,Cc1cccnc1C(N1CCCC1C1CN(C(=O)CC2CCCN2C(C)C)C1)=O 92969,c1(OC)ccccc1NC(C(=O)NC(CNC(c1cc(Cl)no1)=O)C(C)(C)C)=O 92970,CCCCC(O)C(=O)N1CCCC1(C)CNC(=O)CCSc1n[nH]c(C)n1 92971,c1(CN(C2CCCC2c2ccccc2)C)cc(F)cc(F)c1O 92972,N1(C(c2c(C)cc(C)o2)=O)CCC(NC(=O)C(C)CN2CCOCC2)C12CC2 92973,C1(NC(c2cc(CSCC)on2)=O)CN(C(=O)C(C(C)(C)C)[SH](C)CS)CCC1(C)C 92974,c1(NC2CC3CN(C(CSSC)=O)CC32)cnc(C#N)c(C#N)n1 92975,S(=O)(=O)(c1ccc(C=CC(=O)NC2CCSC3(CCC3)C2)cc1)NCC 92976,C(=O)(CCCC(=O)NC(C)C(CO)NC(C1NC(=O)OC1C)=O)NCCC 92977,c1(CC)nn(C)cc1NC(=O)C(O)CCNC(C1CCCOC1)=O 92978,N(C(=NCC1CNC(=O)C1)NCC1CCCCN1CC(C)C)C(CC)CC 92979,c1(C(N2C3CC(NC(C4CCS(=O)(=O)CC4)=O)C2CC3)=O)ccc2nnnn2c1 92980,C1(Cn2cc(C(CCCCCC)(C)O)nn2)C(F)(F)C12CCOCC2 92981,c1(C(=O)NCC2(COC)CN(C(C3CN(C)C3)=O)C2)cc(Cl)cnc1OC 92982,c1(OCCC(N2CCC(CN(C(=O)CCC3CC3(C)C)C)C2)=O)ccccc1F 92983,C1(C(=O)NCCN(C(=O)CCc2nccs2)C)CC(N(C)C)CCO1 92984,C(=O)(CCC(C)(F)F)NCC(N1CCN(C(C2(CC)CCOC2)=O)CC1)C(F)F 92985,c1(C(N2CCC(N(C(C3CCSC3)=O)CCO)C2)=O)cc2cscc2s1 92986,c1(N(C(CCn2cc(CN3CCN(C)CC3)nn2)=O)C)cc2ccc(Cl)cc2s1 92987,C1(C2CCCC2)(NC(C2CCN(Cc3ccccc3)CC2C2CC2)=O)CCC1 92988,N1(Cc2nccc(OC)c2)CCC2(CCN(C(=O)C(C)S(=O)(=O)C(C)C)CC2)CC1 92989,c1(C(N2CCOCC(CNC(C(C)(O)C3CC3)=O)C2)=O)cccc2scnc12 92990,N1(C(C=CCC)=O)CCC2CCN(C(c3c(C)[nH]c4ccc(O)cc34)=O)CC2C1 92991,C1(C2CC2)(CNC(C(CCCC)C)=O)CCN(C(=O)C(F)OC(F)(F)F)C1 92992,C(=O)(CC(C)(C)CNC(C1(C)CC(=O)C1)=O)NC(C(=O)N(CC)CC)C 92993,C1(NC(C2(CC(=O)OC)CC2)=O)CCN(C(c2ncccc2F)=O)CC1C 92994,CC1OC2(C)CC1(C(=O)NC1(CNC(=O)C(C)OCCN(C)C)CCCC1)C2 92995,c1(C(=O)NCCC(C)NC(=O)C(C)(C)c2cc[nH]n2)nnc(S)nc1O 92996,n1(CC(N2CC(C)N(C(=O)CCCS(N)(=O)=O)CCC2)=O)ncc2ncccc12 92997,Cc1ncc(NC(=O)C(C(CC(=O)C(=O)C=Cc2ccccc2)O)N(C)C)cc1Cl 92998,C(=O)(C(C)(C)Cc1ccc(O)cc1)NCC1(F)CC(CNC(COC)=O)C1 92999,Cc1ccc(C=O)nc1F.C12(CC3CCOC3)CN(C1)C2.OCC 93000,c1(NC(C2C(NC(=O)CCC(F)(F)F)C2)=O)cc(Cl)nn2ccnc12 93001,c1(SC)cncc(C(=O)NCC2(CNC(c3cncc(N)n3)=O)CCCC2)n1 93002,C(=O)(CC1=CCN(C(=O)CN2CCCC2)CC1)NCCc1nccc(C)n1 93003,N1(C(CNC(c2c(C)ccs2)=O)=O)CC(CO)CC1C 93004,N1(C(c2c(C)cccc2C)=O)CC2CCC1C(CNC(C1(C(C)C)CCC1)=O)C2 93005,CC(Cn1ccnc1)C(=O)NC(C1CCCCC1)CNC(=O)CC1(C)CC1 93006,C=C=CCC(=O)NC(C1CC1C(N1CCCC1CC)=O)C 93007,C(=O)(CC(CC(C)C)NC(=O)OC(C)(C)C)NCC1CC(NC(CC(C=C)C)=O)C1 93008,c1(OC(C(N2C(C(C)NC(C(C)(C)OCC)=O)CCC2)=O)C)ccc(Cl)cc1 93009,c1(C(=O)NC2(C)CCC2)ccc2c(c1)COC2(C)C.N12CCC(CCO)(C1)CC2=O 93010,c1(C(N2CCN(C(c3c(OC)ccs3)=O)C(C)C2)=O)cn2nc(OC)ccc2n1 93011,CC1CCc2ncc(C(N3CCC4(CCN4C(c4c[nH]c(=N)o4)=O)C3)=O)n2C1 93012,C(=O)(CS(=O)(=O)c1ccc(Cl)cc1)N(CC(C)NC(C(CC)C#N)=O)C 93013,N1(C(Cc2c(C)cnn2C)=O)CCCN(C(c2ccc(OC(F)F)cc2)=O)CC1 93014,C#CCC(C)(C(=O)NCC1CNC(=O)O1)NC(c1cccs1)=O 93015,c1(OC(C)C)nccc(C(N2CC(NC(=O)CC3CC(F)C3)C3(CC3)C2)=O)c1F 93016,CCC(CNC(=O)C(CCOC)NC(c1ncc[nH]1)=O)(CC)C(N)=O 93017,c1(C(c2n(CC)nnn2)NCCSC2CCCS2)ccc(C#N)cc1F 93018,c1(C(C(=O)NC2CCCN(C(C3C(C(C)(F)F)C3)=O)C2)O)cccc([N+](=O)[O-])c1 93019,C1(C(=O)NCC(C2CC2)NC(C2CCC2)=O)CCc2[nH]nc(O)c2C1 93020,CCC(F)(F)CC(=O)N1CC(C(=O)NC2CC2(C)c2nc[nH]n2)(OC)C1 93021,C1(NC(C(N2CCCCCC2)C)=O)CC2CCC1N(C(=O)CCC(N)=O)C2 93022,C1(NC(COCCC)=O)CCN(C(c2cc(Cl)ccc2OC(F)F)=O)CC1C 93023,c1(C(=O)NCC2N(C(CCn3c(C)cc(C)n3)=O)CCCC2)cc(C)c(C)nn1 93024,C(c1cccc(O)c1)=CC(=O)NC(CNC(C1N(CCC)CCC1)=O)C(C)C 93025,CC(C)(C)S(=O)(=O)CC(=O)NCCC1CN(C(c2csnn2)=O)CCO1 93026,CC1OC2CCC1(C(=O)N(CCCN(C(=O)COCC1(F)CC1)C)C)C2 93027,N1(C(C(c2ccccc2)SC)=O)CC(CO)(NC(=O)Cc2cc(C)no2)C1 93028,N1(C(c2cn(C)c(Br)c2)=O)CC2CC(CNC(=O)C=C3CCOCC3)C2C1 93029,c1(NCC2CCN(C(C3C(CC)C3)=O)C2(C)C)ncnc2c1cnn2CC 93030,C(=O)(C(=O)CC(C)CC)N(C(CNC(C(CCCC)O)=O)CC)C 93031,N1(C(c2c(CC)n(C)nc2)=O)CCC2CCN(C(c3cscc3SC)=O)CC12 93032,c1(C(=O)Nc2c(C)cc(CC)nc2)nc(Br)c2c(F)cccn12 93033,N1(C(c2cn(C3(C(N)=O)CC3)nn2)C(=O)NC2(C)CC2)CCN(CCC#N)CC1 93034,S(=O)(=O)(c1ccc(C(=O)NC2CCC(CNC(c3cncc(N)n3)=O)C2)o1)NC 93035,N1(C(C2(CCC=C)CN(C(c3ccc(C)cn3)=O)C2)=O)CCC(O)C(C)(O)C1 93036,C(=O)(C(CN(C)C)CC)NC1C=CC(CNC(CSCC#C)=O)C1 93037,CC(C)(Cc1nn[nH]n1)C(=O)N1CCOCC1C(=O)OC1CCCCC1 93038,C1(NC(C2C(CC(C)C)C2)=O)CC(CNC(c2ocnc2C2CC2)=O)C1(C)C 93039,CC1(O)CCCN(C(=O)C(Cc2cnc[nH]2)NC(=O)CCN2CCCC2=O)C1 93040,C1(C(NOCCOCC)=O)CN(C(=O)C(C)C2CCC2)CC12CCC2 93041,N1(C(CC2CC(C)C2)=O)CCCN(C(c2ncc(F)cc2F)=O)CC1C 93042,C1(N(C(=O)CC2COC(=O)C2)C)CCCCN(C(C2CS(=O)(=O)C2)=O)C1 93043,c1(NCCCOCCOC)ccc(S(=O)(=O)NC(C)CS(C)(=O)=O)cc1Cl 93044,c1(OC)cnnc(C(=O)NCC(C2CC2)NC(C2(OC)CCOC2)=O)c1 93045,C1(Nc2cc(NC(C)CC3CC(=O)NC(=O)N3)ncn2)CCc2nnc(C)n2C1 93046,c1(C(=O)NCC(C(C)C)NC(C2CC3(C2)CC3(F)F)=O)cccc(C(N)=O)c1N 93047,c1(C(=O)NC2CN(C(C(CC)n3nccc3C)=O)C2)cc(C)cc(Cl)c1 93048,C1(C(CC)CC)CCN(C(=NCc2cccc(NS(C)(=O)=O)c2)NCC(F)F)C1 93049,C1(F)(CNC(C(C)Cn2ccnc2)=O)CCN(C(=O)CN2CCCNC2=O)C1 93050,c1(N(CC(C)NC(c2ccc(OC(C)C)cc2)=O)C)cccc(F)c1[N+](=O)[O-] 93051,C1(N(C)C(C2(NC(=O)C(C3CCOCC3)F)CSC2)=O)CCCCC1O 93052,N1(CC)CCN(CC(N2CCN(C(=O)C(CC(C)(C)C)NC(C)=O)CC2)=O)CC1 93053,c1(C(=O)NC2(CN(C(c3c(CC)oc(C)c3)=O)C)CC2)cnc(OC)c(Cl)c1 93054,C1(CCNC(CC=CC)=O)CC(F)(F)CN1C(=O)COc1ccncc1 93055,C(C(N=[N+]=[N-])C(=O)N1CCOCC(NC(c2ccc(Cl)nc2Cl)=O)C1)OCC 93056,c1(CC)cnc(O)c(C(N2CCC(O)C(NC(C3SCC=C3C)=O)C2)=O)c1 93057,C(=O)(CC(C)(C)CCCCC)N1CCCC(NC(C2C(=C)C2)=O)(COC)C1 93058,c1(C(N2CC=CC(NC(C(C(=O)OCC)F)=O)C2)=O)n[nH]c2c1CCCC2 93059,C1(O)(C(CC)C(=O)NC(CNC(C2CC2F)=O)Cc2ccccc2)CCCCC1 93060,C1(CNC(C=CCOC)=O)CC(C)(C)CN1C(C1CCC(C(C)C)CC1)=O 93061,c1(CC(=O)NCc2cn(CC(C)NC(C3(C(N)=O)CC3)=O)nn2)ncc(Cl)s1 93062,C(=O)(CC(O)CCSC)NCC(CN(C(c1scnc1C(F)F)=O)CC)(C)C 93063,C1(OCC)CCCN(C(=O)Cc2nc(-c3ccc(F)cc3)oc2C)C1 93064,CC1(C)CC(O)C(O)CN(C(C2(c3cc(C(F)(F)F)cc(F)c3)CC2)=O)C1 93065,CC1CCC(NC(C2CC23CCSCC3)=O)CN1C(=O)CCN1CCCCC1 93066,c1(C(N)=O)cc(Cl)ncc1NC(C1(O)CCN(C(=O)Nc2cncnc2)C1)=O 93067,c1(C(=O)NCCN2CCN(C(=O)COC3CCOC3)CC2)cc2c(s1)CCOC2 93068,C1(NC(c2cc(C)[nH]n2)=O)CCCC1(C)NC(c1cnc(C2CC2)o1)=O 93069,c1(CCNC(N(CCCO)C)=O)csc2ccc(Br)cc12 93070,N1(C(c2cc3n(n2)CCO3)=O)CCC2CCN(C(c3csc(F)c3)=O)C2C1 93071,C1(O)(CN(C)C(C2SCCS2)=O)CCN(C(c2ccc(C3(C)CC3)cc2)=O)C1 93072,C1(C(=O)NCC2CCCO2)(CC)CN(C(=O)CCCNC(C)=O)C1 93073,c1(N(C(CNC(c2cc(CCC)[nH]n2)=O)C)C)ncnc(Cl)c1Br 93074,CONc1cccc(C(N2CCCC(C(=O)Nc3nc4ccccc4[nH]3)C2)=O)n1 93075,C=C(C)C1OCCCC1C(N1CCCC1CCNC(c1ccsc1C(F)F)=O)=O 93076,C1(CNC(C2CC3CC3C2)=O)CC2(CCC2)CN1C(C1(O)CCSCC1)=O 93077,c1(OC)nc2ncnc(N(C(=O)OC)C(C3CCc4nccn4C3)=O)c2s1 93078,Cc1cnc(O)c(CNC(=O)CC(C)N(C)C(C2CCCC(=O)CC2)=O)c1 93079,C1(O)(CN(C(CC(C)(C)OC)=O)C)CCCN(C(c2nnn3c2CCC3)=O)C1 93080,c1(C(N2C(C)CC(NC(C=C(C)C)=O)C2)=O)ncnc2c1c(Br)cn2C 93081,N1(C(CCOc2ccc(C)c(Cl)c2)=O)CC2CCCN(C(C3CC3C)=O)C2C1 93082,C1(CC)CN(C(c2cc(C)co2)=O)CCC1NC(=O)C(F)(F)C1CCCC1 93083,N1(C(C2N(C(CCNC(=O)OCC)=O)C(CC)CC2)=O)CC2CCCC(O)C2C1 93084,C1(N(C(C23CC(CCC)(C2)C3)=O)CC)CCCN(C(C2(O)CCSCC2)=O)CC1 93085,N1(C(C(C)N(C(c2ccc(Cl)s2)=O)C2CC2)=O)CC(C(N)=O)CC1(C)C 93086,C1(NC(=O)C=C2CCCC2)CCCCC12CCN(C(C1(CF)COC1)=O)CC2 93087,C(c1cc(F)c(O)c(F)c1)=CC(N1CC2C(N(C(COC(CC)C)=O)C)C2C1)=O 93088,C1(OC)CCCC(CC(=O)NCC(C)(C)CN(C(=O)CC2CC=CCC2)C)C1 93089,N1(C(=O)OC(C)(C)C)CCC2CN(C(C3CC34CCC(=O)CC4)=O)CCC12 93090,c1(C(=O)NCC#CCNC(c2cc(OC)no2)=O)cc(Br)c(C)nc1O 93091,c1(C(N(CC(C)NC(c2c(C(C)C)cco2)=O)C)=O)cc2oc(Br)cc2[nH]1 93092,c1(C(=O)NC(CC=C)CNC(c2[nH]ccc2COC)=O)cncnc1C 93093,N1(C(C(C=C)OC)=O)CCN(C(C2CC3CCCC3C2)=O)CC12CCC2 93094,C=C1CCN(C(c2cc(CC)n(C)n2)=O)C(C(N2CCC(C)CC2)=O)C1 93095,Cc1cc(=NCCCNN(C)C(=O)C2CC2)[nH]c(Cc2ccsc2)n1 93096,C1(NC(CC2CC(=O)NC2)=O)CN(C(=O)CC2C=CCCC2)C2(CCCCC2)C1 93097,Cn1c(=O)oc2cc(CNC(=O)NCCCC3C=CCC3)ccc12 93098,N1(C(C2CCN(C)C(=O)C2)=O)CCC2(CCCN2C(c2ccc(F)c(Cl)n2)=O)C1 93099,C1(CCNC(CC2CCC(=O)O2)=O)CCN(C(=O)CC2COCC2O)CC1 93100,C1(CC2CC2)CCCC1N=c1cc[nH]cc1S(=O)(=O)N(CCC)C 93101,c1(CNC(C(CO)NC(CCCSC)=O)=O)ccc(C)nc1O 93102,C1(CCCNC(CC2(OC)CCC2)=O)CN(C(=O)C(CO)N(C)C)CCO1 93103,CC(CC(N)=O)C(=O)N1CCCCC(NC(c2cc(-c3ccc(Cl)s3)[nH]n2)=O)C1 93104,c1(OC)cc(C(=O)NC2CC(C(=O)NCCn3nncc3C)C2)on1 93105,c1(SCCC)cccc(-c2nc(-c3occc3C)nn2CCC)c1 93106,C1(N(C(=O)OC(C)(C)C)CCO)CCCN(C(=O)NCC2C=CCC2)C1 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93211,C1(CC)CN(C(=O)Nc2ccc(C3CNCC3(F)F)cc2)CC2(CCOC2)O1 93212,c1(C(=O)NC2CC(CNC(c3nn(CC)c(C)c3)=O)C2)cccc(C(C)C)c1N 93213,N1(C(c2cc(C(N)=O)[nH]c2)=O)CCC2(CC2C(N2CCCCC2CF)=O)C1 93214,C(=O)(C(Cn1cncn1)NC(c1ccn(C)n1)=O)NCCCOC(C)C 93215,N1(C(c2ccc(CN=[N+]=[N-])cc2)=O)CCC2(CC1)CC2NC(=O)C(N)=O 93216,C1(CNC(c2cc(COC)no2)=O)C(C)CCN1C(=O)CSc1c(C)n[nH]c1C 93217,Cc1cc(C#N)nc(=NCC2CCNC2=O)[nH]1 93218,C1(CC(=O)N(CC(=O)OC)C(C)C)CN(C(=O)CCCC2CC2)CCC1C 93219,CC(C(O)C(F)F)NC(c1ccc(CNC(=O)C=CC2CCCCC2)cc1)=O 93220,C(=O)(C(CCC)C1CCCCC1)N(C(CCCC)C)C 93221,C1(C2CN(C(=O)CC(C)O)C2)(NC(c2c(CC)n(CC(C)C)nc2)=O)CC1 93222,c1(C(=O)NCC23CC(NC(c4coc(Cl)n4)=O)(C2)C3)nccc(C(F)(F)F)n1 93223,C1(C(=O)NC2CN(C(C3CS(=O)(=O)C3)=O)C2)CCCNC1=O 93224,C1(C)(CC)CC(N=c2[nH]c(=NCc3nnc4ccc(C)cn34)[nH]c3c2CCC3)C1 93225,CS(=O)(=O)c1cccc(CN2CCCC(CNC(c3cccc(Cl)c3Cl)=O)C2)c1 93226,c1(OC)cccc(C(C)C(=O)NCC2CN(C(c3nc(O)sc3C)=O)C2)c1 93227,c1(OC)c(Cl)ccc(C(=O)NC(CNC(=O)CCC2OCCO2)C(C)(C)C)c1F 93228,C1(C(=O)NC(CNC(C(CC)=CCCC)=O)CO)CCC(N(C)C)CC1 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93281,Cc1c(C(=O)NC2CCC(C(N3CCC(CF)CC3)=O)C2)cccc1CO 93282,N1(C(C(CC)(C)O)=O)CC(NC(C2(c3cccs3)CCCC2)=O)CC2(CCC2)C1 93283,N1(C(=O)Nc2c(CC)cccc2)CCN(C(c2cc(C)ccc2C)=O)C(CO)C1 93284,C(=O)(C(CCC1CC1)NC(=O)C=CC(=O)N(C)C)NCC(CC)C#N 93285,N1(C(C(=O)NC(CSC)=O)C(C2CC2)C2CC2)CCN(CC2CCOC2)CC1C 93286,c1(C(=O)OCC)ccc2[nH]cc(C(=O)OC(Cc3ccncc3)C(=O)NC)c2c1 93287,C(=O)(C(C)CC(=O)NC1CC2CC(NC(=O)Cc3cncnc3O)C1C2)OC 93288,C1(S(C)(=O)=O)(C(=O)NC2CCCCN(C(C(C)NC(=O)NC)=O)C2)CCCCC1 93289,c1(CNCc2c(C)c(Br)cnc2)cc2c(cn1)OCCO2 93290,C1(C(=O)NC(CC)CCO)CN(C(=O)C=CC2CC2)CC1OC 93291,O=C(C#CC1CCCOC1)NCC1CCC(NC(C2CCCC3CC23)=O)CC1 93292,C1(NC(C(CC2CCC2)OC)=O)(CNC(c2cc(CO)[nH]n2)=O)CCCCC1 93293,N1(C(C=NOC)=O)CC(NC(C23CCCC2C3(F)F)=O)CC12CCCCC2 93294,n1(CC)ccc(C(=O)NCC2CCC(C)N(C(=O)CC(=O)N(C)C)C2)cc1=O 93295,C1(C(=O)NCC2CCCN2C(=O)CC2(C(F)(F)F)CC2)CCCC2CCCCC12 93296,c1(C(=O)NCCC(=C)CNC(=O)CC(CC)C2CCC2)cc(Cl)c(OC)c(Cl)n1 93297,c1(OC)ccc2c(c1)CC(C)CC2NC(c1ccoc1Br)=O 93298,N1(CC(C)NC(CCC2CC(C)C2)=O)CCN(C(=O)C(O)c2ccsc2)CC1 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93317,CCCC(C)(CCC)C(=O)NCC1CC(O)CN1C(C1CC2(COC(=O)N2)C1)=O 93318,C1(NC(C(CC)NC(N)=O)=O)CC2CC1N(C(c1cnc(OC)c(C)c1)=O)C2 93319,c1(OC)ccc(NC(c2cccnc2-c2cn[nH]c2)=O)cc1O 93320,C1(CNC(COC2C(C)CCCC2)=O)CCC2(CN(C(c3cscc3Cl)=O)C2)O1 93321,c1(C(N2CCC(O)(CNC(c3n(CC)nnc3)=O)C2)=O)c(Cl)ccc(Cl)c1Cl 93322,CCC(O)CC(=O)NC(C(=O)NCc1nc[nH]n1)c1ccoc1 93323,N1(C(=O)NCC(C(C)N(S(C)(=O)=O)C(C)C)(C)C)CCCC1C1CCCCO1 93324,C#CC(CC(C)C)NC(C1CCN(C(=O)CCc2csnn2)C1C(C)C)=O 93325,N1(C(c2cnc(C)[nH]2)=O)C2CCC1CN(C(c1cnnc(C)c1)=O)CC2 93326,CCC(O)C(C)C(=O)NCCN(C(=O)C(n1nnnc1C(C)(C)C)C)CC 93327,CC(C)C#CC(=O)NC(C)(CNC(=O)C(C)NC(C1CCCC1)=O)CO 93328,C1(C(N(CC(C)NC(C(C(=C)Cl)(C)C)=O)C)=O)CCc2nccn2C1 93329,Cc1cc(C(N2CCC(CC(=O)Nc3cccc(F)c3)C2)=O)c(Br)cc1F 93330,c1(C(=O)NC2C(C(=O)NCCC#N)C2)cccc2c(O)nccc12 93331,c1(C(=O)NCC2N(C(c3c(CCC)[nH]cc3)=O)CCC2)ncccc1C(F)F 93332,c1(C(N2C(C(C)C)C(NC(=O)C(C)CN(C)C)CC2)=O)cc(F)cc(F)c1O 93333,N1(C(c2c(C)cc(CC)o2)=O)CCC(C)N(C(=O)C(C)CO)CC1 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93352,C1(CNC(c2cc(CC)c(C)s2)=O)CCCC2(CN(C(C3CCCOC3)=O)C2)O1 93353,C1(NC(C2(SC)CC2)=O)CCCC(NC(c2csc(CC(F)(F)F)n2)=O)C1 93354,Cc1nc(N2CCN(Cc3cc(C(=O)O)cc(F)c3)C3CC23)c2c[nH]nc2n1 93355,c1(C(C#C)NC(=O)CC2CCN(CCC(C)C)C2)cccc(F)c1 93356,c1(C(CC(=O)NCCCN(C(C(COCC)C)=O)C(C)C)O)ccc(F)cc1 93357,C(=O)(C(C(=O)OC)C1CC1)N(C(CCNC(COCC=C)=O)C)C 93358,CP(C)(=O)C1CCCC1C(=O)NC1CC1NC(c1ccc2c(c1)CC2)=O 93359,C1(C(N(CCOC)CCNC(=O)C=Cc2ccoc2)=O)CCCC(C)CC1 93360,c1(C(C)(C)C)ccnc(C(N2CCC(CO)(NC(c3nonc3N)=O)C2)=O)c1 93361,C12(NC(c3cc4ccccn4n3)=O)COCCC1CN(C(=O)Cc1cc[nH]n1)C2 93362,C1(CNC(c2n(CC(=C)C)nnn2)c2cnoc2)Cc2ccccc2C1 93363,C(=O)(CCS(=O)(=O)N(C)C)N1C(CC)C(NC(c2cc(C3(C)CC3)n[nH]2)=O)CC1 93364,C1(C(=O)OCC)C=CCN(C(=O)CSc2nncn2C(C)C)C1 93365,N1(C(CC(CC)C)=O)CC2(C1)C(NC(=O)Cc1ccc(C)cc1)CCS2(=O)=O 93366,CC(C)CCC(=O)N1CCCC1C1CCN(C(=O)COC2CCCC2)CC1 93367,c1(C(c2n(C(C)C)nnn2)NC23CC2CS(=O)(=O)C3)ccc2c(c1)COC2 93368,N1(C(C(CCC)C)=O)CC2CC1CC2N(c1ccc(OC(CN(C)C)C)cc1)C 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93405,Cc1cc(C)nc(CCn2c(N3CC(F)(F)CC3C)nnc2C2CCCCC2)n1 93406,C1(CNC(CCS(=O)(=O)NC)=O)CC2(CO1)CN(C(=O)CC(C)(C)C1CC1)C2 93407,C#Cc1cn(C)nc1C(N1CCC(CC(=O)NCc2ncc(C)cc2C)C1)=O 93408,C1(N(C(C2CCN(CC)CC2)=O)C2CC2)CCCN(C(c2ccnc(F)c2)=O)C1 93409,c1(OC)cc(N)ccc1C(N1CC(NC(=O)Cc2cc(C)on2)C(C)C1)=O 93410,C(=O)(CCCN(C)N=O)N1CC(C)C(NC(=O)CSc2cnn(C)c2)C1 93411,c1(NC(c2c(CC)n(-c3cccc(F)c3)nc2)=O)ccc(=O)n(C2CC2)c1 93412,C1(CNC(=O)CSc2nc[nH]n2)CCN(Cc2ccccc2F)CC1(F)F 93413,c1(C(C(=O)NCCN(C(C2C(OC(C)=O)C2)=O)C)OC(C)C)ccccc1 93414,C1(CC=C)(NC(=O)C(O)Cc2ccccc2)CCN(C(=O)Cc2ccc(Cl)cc2)C1 93415,CC(C)(O)CCC(=O)NCC1CN(C(=O)CCn2cccn2)CC12CC2 93416,c1(CN(CC(=O)N)C(C)C)ccc(OCC(CCCC)=O)c(OC)n1.CC 93417,C12(C(C)(C)C)CC(C(=O)NC3(CO)CN(C(C4COC(=O)O4)=O)C3)(C1)C2 93418,c1(CC)ccc(CC(=O)NCCCCNC(c2cnn(C)c2)=O)cc1F 93419,C(=O)(C1=CCSC1)NC(C(=O)NC(CC=C)CO)CO 93420,Cc1c(C(=O)NCCNC(c2ccc3nn[nH]c3n2)=O)oc2ccccc2c1=O 93421,C1(C(=O)NCC2(NC(C(C)=O)=O)CCCC2)CCCCC1C(=O)N(C)C 93422,C1(C)(NC(C(=O)NC(c2ccc(C(=O)OC)cc2)CO)=O)CCS(=O)(=O)CC1 93423,C=CC1(C)COCCN1c1nnc(-c2cc(C)cc(F)c2)n1CCCOCCO 93424,N1(C(CCC2(C(=O)OC)CCC2)=O)CCC(CC(F)(F)F)C1.C1(C)(C)C=CC(=O)N1 93425,CCC(CCCC(=O)NC(C)CCC(C)(C)C)NC(c1n[nH]cc1C)=O 93426,c12nc(sc1C)C(=O)N1CC3C(C3C1)CO2.CC(=O)CC(C1(CSC)CC1)=O 93427,CC1(C)CC1(C(=O)NCC1CC(=C2CC2)C1)NC(=O)C=CCO 93428,C1(CC(C)(C)C)CN(C(C2CCSCC2)=O)CC1NC(C1CCC(=O)N1)=O 93429,c1(CNC(Cc2c(C)nc[nH]2)=O)ncc(C(N2CCC(CC(F)F)C2)=O)cn1 93430,n1(C(C)C)ccc(CC(=O)NCC(C2CC2)NC(c2csnc2C2CC2)=O)n1 93431,C1(C(=O)NC(C2(O)CN(C(c3ccccc3Cl)=O)C2)C)CCCC(C)(C)O1 93432,C1(F)(C(=O)NC(CC#CC)C)CCN(C(c2cc(CC)sn2)=O)CC1 93433,C1(C(=O)NCCC2N(C(CCCCOCC)=O)CC(OC)C2)CC(=O)NC1(C)C 93434,N1(C(C=CC=CC)=O)CCN(C(=O)C(n2nnnc2C(C)(C)C)C)C(C)C1 93435,c1(C(N(c2c(CC)cccc2F)C)=O)cc(Br)cc(S(C)(=O)=O)c1 93436,c1(C(=O)NC2CCC(NC(COC(CC)(C)C)=O)CC2)ccc(Br)cc1Cl 93437,c1(C(C)=O)ccc(C(=O)N(CC(C)CNC(=O)C(F)C(C)C)C)nn1 93438,c1(C(N2CCOC3CC23)=O)ccc2cccnc2c1.C12(CCC1)CC(=O)N2C1CC1 93439,c1(C(=O)NC(C2CN(C(=O)CC3CCOCC3)C2)C)cccc(C#CC2CC2)c1 93440,N1(C(C2CC(=O)NC(=O)N2)=O)CCN(C(c2csc3nccn23)=O)C2CCCC12 93441,c1(CN(C)CCc2cccs2)cccc2c1CNC2 93442,C1(C)(NC(C(CC)=CC)=O)CCN(C(c2coc(CN3CCOCC3)n2)=O)CC1 93443,Cc1cc(C)c(C(=O)NCC2CCN(C(=O)CC(C)c3cccnc3)C2)c(S)n1 93444,C(N=c1[nH]c(=NCCC2CCCCC2)[nH]c2ccc(Cl)cc12)c1ccc(F)cc1 93445,N1(C(C(C)NC(N)=O)=O)CCC2CCCC12C(=O)NCC#CC(F)(F)F 93446,N1(C(C2CC(=C)C2)=O)CC2(CNC(=O)CS(=O)(=O)N3CCCCC3)CC(F)(C1)C2 93447,CC(C)CS(=O)(=O)CCC(=O)N(CC(O)CNC(=O)C(C)Cc1ccncc1)C 93448,C1(COC)(NC(=O)Cc2cscn2)CN(C(=O)CCNC(C2CC2C)=O)C1 93449,c1(C(=O)NCC(C)NC(c2ccc(CC(F)(F)F)cc2)=O)cc2cc[nH]c2cn1 93450,c1(C(=O)NCC(CNC(CN2CCC(OC)C2)=O)CO)c(C)nc(C)n1O 93451,C#CCCCC(=O)N(CCC(=O)NCC1CC2CCC2C1)C 93452,C(=O)(C1=C(Cl)CCCC1)N(C(C)(C)CC(=O)NCC1CCCC12CC2)C 93453,C1(NC(c2n(CC)ncc2C)=O)CCCCC12CCOCC2 93454,c1(CC(=O)OCC)cc(NCCC2NC(=O)NC2=O)ncn1 93455,S(=O)(=O)(C1CCC(=O)CC1)N1C(CC(=O)Nc2c(C)csc2)CCC1 93456,n1(CC)nc(C(=O)NC2(C(N3CCC(C(=O)OC)CC3)=O)CCN(C)C2)cc1C 93457,N1(c2ccc(C(C)=O)cn2)CCCCC(NC(C2(C3CCCO3)CC2)=O)C1 93458,CC1(CC(=O)NCCC2(CO)CCC2)CCCN1c1cc(-n2ccnc2)ncn1 93459,C1(C(=O)NC(c2nccn2C)C)CC2CC2N1C(=O)C=Cc1cc[nH]n1 93460,N1(C(C(C(C)(C)C)=O)=O)CCn2nc(CNC(C3CCCCNC3=O)=O)cc2C1 93461,CC(C)(CNC(=O)COC1CCCC1)CC(=O)NCc1cncnc1 93462,c1(C(=O)NCC2C(NC(c3cc(OC)ncc3)=O)C2)cc2cc(Cl)ccc2o1 93463,N1(C(c2ncc(C)nc2)=O)CCCC(C)(CNC(=O)C2=NNC(C(F)(F)F)C2)C1 93464,C1(NC(CSc2cccc(C)c2)=O)CC(NC(=O)Cc2cnc(C)[nH]2)C12CCC2 93465,CC(CC(=O)c1ccc(Cl)cc1)C(=O)Nc1ccc(Br)cc1 93466,C(=O)(NNC(=O)c1ccc(C(F)(F)F)o1)c1c(C)ncs1 93467,Cc1csc2ncc(C(N3CCOC(C(C)NC(=O)C(C)(C)CF)C3)=O)n12 93468,N1(C(C2C=CCC2)=O)CCC(C(N2CCCC2CC(c2ccc[nH]2)O)=O)CC1 93469,C(=O)(C(O)CC(F)(F)F)NC1CC(NC(=O)CC(C(F)F)n2ccnc2)C1 93470,C(CC(C(C)(C)C)NC(c1cnc2n1CCS2)=O)N(C(C(C)SCCCC)=O)C 93471,N1(C(C(CC)OCC)=O)CC(N(C)C(c2ccc(=O)oc2)=O)C(C)(C)C1 93472,C1(NC(c2c(C(C)C)ocn2)=O)CC2CN(C(c3cc(C(F)(F)F)on3)=O)CC12 93473,c1(C(=O)NC2C3CN(C(C(=O)NCC(F)F)=O)CC32)csc2cncn12 93474,CN1C=C(I)c2c(NC(c3ccc(OCCF)cc3)=O)ncnc2C(Br)=C1 93475,c1(N2CCC(NC)C(O)C2)nc(Cl)nc2c1ncn2CCc1ccccc1 93476,C1(OC)CC(C)CN(C(=O)C(c2ccoc2)NC(C2CC(F)CN2C)=O)C1 93477,c1(-n2c(C)nnn2)cc(C(=O)Nc2ccc(N(C)C)nc2)ccc1Cl 93478,N1(C(C(C2CCC2)OCC)=O)CCC(F)C(NC(c2noc(C3CC3)c2C)=O)C1 93479,Cc1cn2c(C)c(C(=O)NCC3(CNC(C4OCC4(C)C)=O)CC3)nc2s1 93480,CC1CC(CCNC(=O)CCCCN2CCCC2)CCN1C(=O)CC#N 93481,C1(C(=O)NC(CC2CN(C(C(CCC)=CCC)=O)C2)C)CCc2n[nH]cc2C1C 93482,c1(C(N2C(C(=O)Nc3n(C)ncc3I)C=CC2)=O)cc2ccccc2[nH]1 93483,Cc1ncccc1C(N1CC(CNC(C2CCCN2C)=O)C(C(F)(F)F)C1)=O 93484,c1(NCC(CCC)C)cccc2[nH]nc(C)c12 93485,C(=O)(C1CCCn2ccnc21)NC1CC2(CN(C(C(C)Cc3cnco3)=O)C2)C1 93486,C12(CNC(C(COC)O)=O)CCC(NC(=O)CC(C)C)(CO1)C2 93487,C1(CNC(CNC(C2C(C)C2)=O)=O)(CO)CCN(C(C2CN(C(N)=O)C2)=O)C1 93488,CC(c1ccccc1C)=CC(=O)NCC(C)(C)NC(C1CCCS1)=O 93489,C(=O)(CCCCNC(c1cn[nH]c1)=O)NC(C)CCN(C)C 93490,C1(C(C(=O)OC)NC(=O)COCC(N2CCCC2)C)CCOCC1 93491,c1(CC)sc(C(=O)N(C)CC2CN(C(C3CN(C)C(=O)N3)=O)CCO2)cc1C 93492,c1(C(=O)Nc2ccc(F)cc2CO)cnn2c1CN(C(C1CC1C1CC1)=O)CC2 93493,C=CCC(C(=O)NCC(CC)(CC)NC(=O)C(C)NS(C)(=O)=O)C(C)(C)C 93494,C(=O)(CC(C(=O)OC)OC(=O)CC1CCN(C(c2ccc(=O)oc2)=O)CC1)OC 93495,c1(N2C(CNC(C=CC=CCC)=O)CC3(CCC3)C2)nc(Cl)nc2cnn(C)c12 93496,c1(C(=O)NCC(C)(O)CNC(C2CCCCN2N=O)=O)c(Cl)cncc1Cl 93497,C(N=c1ncc2ccccc2[nH]1)C1CC(NC(=O)COc2ccccc2F)C1 93498,c1(C(=O)NC(C(C)NC(CCCOCC)=O)CO)cnc2c(c1)NC(=O)CN2C 93499,CC1(C)CCN(C(c2csc(Cl)n2)=O)CC1NC(c1csc2ccccc12)=O 93500,C1(CC(=O)NCc2cn(CCNC(C3(CC)CCCC3)=O)nn2)CCC(=O)NC1 93501,c1(C(=O)NCCN(C(C(c2cccc(C)c2)O)=O)C)cccc2nn[nH]c12 93502,C1(C(N(CC(C)O)CCNC(C(C)C)=O)=O)OCC1(C)C 93503,Cc1noc(C)c1NC(=O)CC1CCCCC1NC(c1coc(CO)c1)=O 93504,c1(NC(C(=O)N(C(c2ccccc2C)C(C)C)OCC)=O)ccc2c(c1)CCN2 93505,N1(C(Cc2c(C)n[nH]c2)=O)CCN(C(=O)COC(F)(F)C(F)(F)F)CC12CCC2 93506,c1(OC)cc(OC)c(CN2CCC(C)(NC(c3nc(Cl)sc3C)=O)C2)c(Br)c1 93507,c1(C(N2CC(N(C(C(C)NC(N)=O)=O)C)C2)=O)cnc(O)cc1C(F)(F)F 93508,C1(NC(C#C)=O)CCN(Cc2ccc(-c3ccccc3)cc2)CC1F 93509,N1(C(c2nc(CCC)sc2)=O)CC(CNC(=O)C(CC)OCC)OC(C)(C)C1 93510,c1(C(N(CC=C)CC=C)=O)ncccc1OC(C)=O.c12ccc(nc1)NC2C 93511,c1(C(N2CCCC(CNC(CN(C(C)=O)C)=O)C2)=O)c(Br)ccc(N)c1F 93512,c1(C(=O)NCC2CCN(C(c3c(CC)nccn3)=O)C2)c(C)sc(C)c1C 93513,C1(NC(C2ON=C(C(C)C)C2)=O)CC2CCC1CC2NC(=O)C(C)(C)CO 93514,C#Cc1cccc(C(=O)NC(C2CCN(C(=O)CSCC(F)(F)F)C2)C)c1 93515,N1(CC(=O)NC(C)CN(C(=O)C(O)Cc2ccccc2)C)Cc2ccccc2C1 93516,C1(CCNC(c2c(C)cccn2)=O)CCN(C(C2COCC(C)(C)O2)=O)C(C)C1 93517,N1(C(C2N(S(C)(=O)=O)CCC2)=O)CC2CC(C(=O)Nc3ccc(Cl)cc3)C1C2 93518,c1(OC)cccc(C(N2CCOCC2C(=O)NCc2ccc(Br)c(F)c2)=O)c1O 93519,C1(NC(C2CCS(=O)(=O)C2)=O)CCN(C(C2CC(Cl)(Cl)C2)=O)CC12CCC2 93520,Cc1noc2ncc(C(N3CCN(C(=O)CC(C)CF)C(CO)C3)=O)cc12 93521,c1(C(N(C2CC(SC)C2)C)=O)cccc(-c2cnn[nH]2)c1 93522,C1(CCCNC(C(=O)NC(C(=O)OC(CC)C)C)=O)CCOCC1 93523,C1(NC(c2c(C)cns2)=O)CN(C(c2ccc(NC3CCCC3)cc2)=O)C2CC12 93524,c1(C2C(C(=O)NCCCNC(c3ccc(=N)[nH]n3)=O)C2)nccc2ccccc12 93525,C1(NC(C=CSC)=O)COC2(CNC(c3cnc(N)c(Br)c3)=O)CC1C2 93526,c1(-n2cc(C(=O)NC(CNC(CCSCCC)=O)C3CC3)nc2)cccc(Cl)c1 93527,N1(C(c2cnc(COCC)s2)=O)CC(NC(=O)C(F)(F)CC)CC12CCCOC2 93528,N1(C(C2CC(CCNC(CC3CCN(C)C3=O)=O)C2)=O)CC2(C1)CC1(CCC1)C2 93529,N1(C(C2C(=C)C2)=O)CCCCC(C2CN(C(c3ccc(O)c(F)c3F)=O)C2)C1 93530,C(=O)(C1=CC2(CCOC2)C1)N(CCNC(C(c1cccc(O)c1)C)=O)C 93531,c1(NC(=O)CC2CCc3ccccc3N2)ccc2c(c1)OC(F)(F)O2 93532,CCC(CC)(CCNC(=O)C1=C(C)OCC1)NC(=O)COC(C)(C)C(F)(F)F 93533,C12(C(=O)OC)C3C4C1C1C2C3C41C(=O)Nc1c(C#N)nccc1 93534,C12(NC(c3n[nH]c(C)c3C)=O)CCCN(C(c3cccc(Cl)c3Cl)=O)CC1C2 93535,c1(C(=O)NC(C(CO)NC(c2ccc(C)o2)=O)C)cn2ccnc2s1 93536,C12(C(=O)OC)CCCC1CN(C(C1CN(C(=O)Nc3ccc(F)c(Cl)c3)C1)=O)C2 93537,C=C(C)C(CC(=O)NC1CCC1CNC(=O)Cc1cn2ccsc2n1)OCC 93538,c1(SCC(=O)NC(CC(C)C)CNC(=O)CC2CCOC2)nnc2ccccn12 93539,CC1COC(C)(C)CN1C(=O)CCC1CCCN(C(C23CCCC2CCC3)=O)C1 93540,CC1(CCNC(=O)C(=O)NC2CC2)CCN(C(C2CC2c2ccco2)=O)CC1 93541,C(=O)(CC(C)C(F)F)NC(c1cccc(C)c1)CNC(C1CCN(C)C1)=O 93542,c1(OC)cc(O)ncc1C(=O)NC(C)(C)CNC(C1C2CCCCC12)=O 93543,C(C1CCn2ccnc21)N(C1CCCO1)C(=O)NC(c1cnn(C)c1)COC 93544,C1(NC(c2c(CC)c[nH]c2)=O)C(CNc2ncccc2C#N)CCC12CCC2 93545,N1(C(CCC2C(C)C2)=O)CCOC(C2(NC(=O)C(=Cc3ccccc3)F)CC2)C1 93546,n1(CCN(C(=O)C(C2CCNCC2)F)CCOC)cc(C)cn1 93547,C1(C(N2CC(O)(CN(C(C3C(SC)CCC3)=O)C)C2)=O)CCN(CCF)CC1 93548,c1(C(=O)NCC(=O)NCC(=C)Br)ccc2sc(C(=O)OC(C)(C)C)c(C)c2c1 93549,C1(NC(c2c(C)c(-c3ccccc3)on2)=O)C2CCN(C(=O)C=CCO)CCC12 93550,C1(NC(C2C(C(=O)OC)C=C2)=O)CC2CCCC(C1)N2C(=O)C(C)(C)CF 93551,C1(CNC(=O)CSCC2(CF)CC2)CC2(CCN(C(c3cscn3)=O)C2)CO1 93552,CC(C)CC(O)CC(=O)N1CCC1C(N1CC(c2nc(=O)o[nH]2)C1)=O 93553,C(=O)(C1CCCc2nn[nH]c21)N(C)CC1CCCN1C(C1(O)CC1)=O 93554,N1(CC(=O)NC(C2CCOCC2)CC)CCCC(C(=O)NC(C)(C)C)CC1 93555,c1(C(N(CC(C)NC(C2(C)CC=CCC2)=O)C)=O)ccc2c(c1)n(C)c(=O)n2C 93556,CC(c1ccco1)=CC(=O)N(C)CC1CCCN1C(C1CCC(=O)C1)=O 93557,c1(CC)ccc(C(N2CC(NC(c3ccc(COC)[nH]3)=O)C(C)C2)=O)cc1F 93558,N1(C(C2N(C(c3ccc(C)nc3C)=O)CCCC2)=O)CCn2cnnc2C1C 93559,c1(C(=O)NCC2CCCC(NC(COCCC)=O)C2)cccc(O)c1Br 93560,c1(NC(c2ncc(-c3ccc(OCC)c(F)c3)cn2)=O)cc(C)cc(C#N)c1 93561,c1(C(N2CCC(N(CC#C)C(c3cc(OC)cs3)=O)CC2)=O)cnc(O)cc1O 93562,C(N=C(NCC(C)(C)C)N1CCCC(O)(C(N)=O)C1)c1cccc(CC)c1 93563,CC1(C(=O)NCC2CCCN(C(=O)CCCCC3CC3)C2)CC(F)(F)C1 93564,CC(CC(=O)N(C1CCN(C(c2cccn2C2CCCC2)=O)C1)C)C(F)(F)F 93565,CCCCCCC(=O)NC(c1ccccc1)CNC(=O)CC(C)C(C)C 93566,N1(C(CCOC)=O)CCC2(CCC(NC(=O)Cc3csc(NC=O)n3)C2)CC1 93567,c1(N2C(CNC(c3cnc(C4CC4)nc3)=O)CCCCC2)ccc2nnnn2n1 93568,Cc1coc(C=CC(=O)NCC(CNC(=O)Cn2cccnc2=O)CO)n1 93569,N1(C(C(CC#C)O)=O)C(C(=O)N(CCCCOC)C)C2CC(O)C1C2 93570,c1(CC(=O)N(CC(C)O)CCNC(=O)CCC#N)ccc2ncsc2c1 93571,C1(CN(C(C(CC)OCC)=O)C)CN(C(=O)C(C)NC(N)=O)CCO1 93572,N1(CC(=O)NCC(CNC(C2(C)CC(F)C2)=O)CO)CC(=O)NC1=O 93573,CCC(C)C(O)CC(=O)N1CCCN(C(=O)CCCN2CCCC2)CC1 93574,C1(C(=O)NCCNC(CCn2ncc(C)c2)=O)CCC(O)CN1C 93575,c1(CCN(C(=O)C(=O)NC2CCN(CC(F)F)C2)C)ccccn1 93576,C1(CC(=O)NC2C(NC(Cn3cc(C(C)=O)nn3)=O)C2)NC(=O)NC1=O 93577,c1(OC(C(=O)NCCC2(NC(CC(C)O)=O)CCCC2)C)ccc(Cl)c(Cl)c1 93578,c1(N2CC(C)CN(C(C(CCC)C)=O)C(C)C2)ncc(S(C)(=O)=O)cc1Cl 93579,c1(NC(C)CNC(=O)C(C)Cc2cnc[nH]2)ccc2c(n1)CC(C)(C)CC2=O 93580,N1(C(c2c(CC)n(C)cc2)=O)CC(C(=O)NCC(CC2CC2)CO)CCC1(C)C 93581,C1(CNC(C=CC(CC)C)=O)CCCC2CN(C(c3nc(C)nn3C)=O)CC12 93582,CC1(C)CC(CNC(C2(C)CCC(=O)N2)=O)CN(C(=O)CCCc2ccsc2)C1 93583,CC(C)(CC(=O)NC(CO)C(=O)NCCN1CCCNC1=O)C1CC1 93584,C(C)(CN=[N+]=[N-])NC(C(COC)NC(=O)C=CC1CCOC1)=O 93585,C1(NC(C)Cc2ccc(Cl)cc2Cl)CC2CCC1(C)C2(C)C 93586,C=CCC(C(=O)NCC(C(C)(C)C)NC(c1cnn2c1CCC2)=O)C(C)(C)C 93587,C1(CCNC(CNC(=O)OC)=O)CC(F)(F)CN1C(=O)C(O)C(F)F 93588,CCCCC(C(=O)N(C1CCN(CC)C1)C)NC(C1CCCCNC1=O)=O 93589,Cc1ccc(F)cc1C(N1CCN(C)CC1CNC(C1CCOC(C)(C)C1)=O)=O 93590,c1(C(N2CC(CNC(C3(CO)CCCO3)=O)C2)=O)cc(O)c2ccoc2c1 93591,C(c1cc(C)c(C)cc1C)=CC(=O)NCC1CC(CNC(C(CC=C)(C)C)=O)C1 93592,CCC(C)(C)C(C)NC(=O)C(C)CNC(=O)CN1CCOC1=O 93593,N1(C(=O)OC)C2CCC1C(NC(=O)CCc1nc(C3CC3)no1)C2 93594,C12(C(=O)NCC(CC=C)NC(=O)CCOc3ccc(Cl)cc3)CC1COC2(C)C 93595,N1(C(C2CCC(=O)C2)=O)CCC(C(=O)NCc2cccc(F)c2)(CO)C1 93596,N1(C(c2snc(C)c2Br)=O)CCN(C(=O)C(C)C2CC2)C(C)C1 93597,C12(NC(CC(=C=C)C)=O)CCN(C(=O)CCN3CCOCC3)CC1C2 93598,N1(C(c2c(CC)occ2)=O)CC2(C1)CN(C(=O)CC(c1ccccc1OC)C)C2 93599,N#Cc1cc(S(=O)(=O)N2CC(F)CC2C(=O)NCCCN2CCCC2)ccc1Br 93600,N1(C(C=CC(=O)N(C)C)=O)CC(C(C(=O)NCCC2CC(F)C2)N(C)C)C1 93601,c1(N(CCCN(C(Cn2nnc(C)n2)=O)C)C)ncnc2cc(Br)ccc12 93602,C1(N=c2ccc3nnnn3[nH]2)(CNC(C(C(CC)C)OC)=O)COC1 93603,C(=O)(N=c1ccc(C2CCCCC2)n[nH]1)NCC1OCC(C)(C)C1 93604,c1(C(=O)NCC(C)NC(CC(c2ccc(C)cc2)C)=O)ccc2oncc2c1 93605,CC1(C)CC(CNC(=O)Cn2ncccc2=O)CN1C(C1CCCCNC1=O)=O 93606,N1(C(CCCCCC=C)=O)CCC2(CCN(C(=O)CC3CSCCO3)C2)C1 93607,C1(CNC(CC=CC=C)=O)COC(C)(C)CN1C(=O)C(c1cccc(Cl)c1)C 93608,N1(C(C(C=C)O)=O)CCC(NC(c2c(CC)ncnc2CC)=O)C(F)C1 93609,c1(C(N2CC(N(C(COCCC=C)=O)C)C(O)C2)=O)cc(C(F)F)cc(SC)c1 93610,CC(CC(C)(C)C)C(=O)NC(C)CCCCNC(C1CCCC(C)C1)=O 93611,Cc1ccc(C)c(C(c2nnnn2C2CC(F)(F)C2)NCC(C)(C)C2CCCO2)c1 93612,c12cnn(C)c1S2.C1(C(NOCCOC)=O)CCN(CC(C)(C)C)C1=O 93613,C(CCC(=O)N(C1CCC(NC(=O)Cn2nccn2)C1)C)=CC(C)C 93614,c1(SCC(C)NC(C(C)C)=O)ccccc1-c1cccc(CC(=O)OC(C)C)c1 93615,N1(C(CSCCCC)=O)CC2CC(NC(c3cc(C)c(C)c(C)c3)=O)C(C2)C1 93616,C#CCC(CC#C)C(=O)NCCCN(C)C(c1ccc(C)nc1N)=O 93617,c1(C(N2CCC(NC(CCCOCCC)=O)C2C)=O)cc(C)n(CC)c1C 93618,c1(C(=O)NC2C3CN(C(c4cn[nH]c4)=O)CC23)cnc2ncnn2c1O 93619,C=C(CNC(=O)CC(O)C1CCCC1)CCNC(=O)CC1(C)CC1(Cl)Cl 93620,CC1(C)OCCOC1CC(N1CCN(C(c2[nH]cnc2C#N)=O)CC1)=O 93621,C(=O)(C(CC(C)(C)C)OC)N1CCC(N(C(=O)CN2CCCNC2=O)CC)C1 93622,C=Cn1nccc1C(N1CC(OCCC(=O)N(C2CCCC2)CCOC)C1)=O 93623,C1(C(=O)NCC2CN(C)C(=O)C2)CC2CCCC2N1C(=O)CSC(C)(C)C 93624,C1(C(=O)NCC(C)NC(C2CCS(=O)(=O)CC2)=O)CCc2nc(O)[nH]c2C1 93625,c1(OC)cc(C(N2CCC2CNC(=O)C(n2nc(C)cc2C)C)=O)ccc1F 93626,C1CCCS(=O)(=O)C1.CCCC 93627,Cc1nc(OC(C)(C)C)ccc1-c1ccc(NC(N2CCNC(C)C2)=O)cc1 93628,Cc1nc(C2CC2)ncc1C(=O)NC1CC1C(=O)NC1CC1C 93629,C(CCN=c1[nH]cncc1I)NC(C1N(CC)C(=O)CC1)=O 93630,C(C)(C)(CCCNC(=O)COc1cccc(F)c1)NC(c1ccc(SC)o1)=O 93631,CC(CC(C)(C)C)C(=O)NCC1CCCN1C(C1CCNC1=O)=O 93632,C1(C(=O)NCc2c(C(=O)NC3C(OCC)COC3)c[nH]n2)CN(C)CCO1 93633,C(CC(=O)N1CCN(C(=O)C(F)F)C(CC(F)(F)F)C1)(C1=CCCC1)OCC 93634,c1(CN(CC(CC)OC)C(=O)OC(C)(C)C)c(F)ccc(F)c1OC 93635,c1(C(=O)OC(C2CC(F)(F)C2)C(=O)N(CCOC)C)ccsc1C(F)F.CO 93636,Cc1cc(CCNC(c2nc(C3CC3)oc2C)=O)cc(Br)c1 93637,C(C(CCS(C)(=O)=O)OC)Nc1ccc(C(=O)OC)c(Br)c1 93638,c1(C(N2CC(CCOC)N(C(=O)Cc3cnoc3)CC2)=O)cc2c([nH]1)CCCC2 93639,N1(Cc2onc(C(C)OCC)n2)CCN(C(=O)C(C)(C)CF)CC1 93640,N1(C(C(CN(C)C)(F)F)=O)CC(C2CN(C(c3cccc(C4CC4)n3)=O)C2)C1 93641,CCCCCC(O)CNC(=O)CN(C(=O)C(C1CC1)OCC)C 93642,C1(C(=O)Nc2nnn(CC(=O)OC)c2C)CC(c2ccc(OC)cc2)=NO1 93643,N1(c2nnc(C)n2CC2CC3(CCCC3)CO2)CCc2nc[nH]c2C12CCC2 93644,c1(CC(=O)NC2(CF)CCN(c3nc(SC)c(C)cn3)C2)ccc2ncsc2c1 93645,c1(C(N2CC3C(CNC(=O)C(O)C4CC4)(C3)C2)=O)cnnc2ccccc12 93646,c1(C(=O)NC(c2c(CC(=O)OC)occ2)=O)ncccc1OC(F)F.C1(S)CC1CC 93647,N1(C(CCCN2CC(C)C2)=O)CCCC1C=CC(=O)N(C(C(N)=O)C1CC1)C 93648,C(CN=C(NCc1ccnc(OC)n1)NCC1(C)CCC(=O)N1)OCC 93649,c1(C(N(CCCCCCNC(C2CC2(F)F)=O)C)=O)ccc2c(n1)COCC2 93650,c1(OCC(=O)NCCC(CCNC(C=CC=CC)=O)C)ccc(CO)cc1 93651,C1(CC)C(C(=O)NC2C(C)C2C)CCN1C(c1ccncc1F)=O 93652,C1(CNC(=O)Cc2cscn2)CCCCN(C(C2(F)CCCCCC2)=O)C1 93653,CCCCCCn1cc(C2(C)CN(C(=O)C(C3CCC(=O)N3)C)C2)nn1 93654,Cc1noc2cc(C(N3CCCC3CCCNC(c3ccsc3Cl)=O)=O)ccc12 93655,N1(CC#C)CCOC(C)(CNC(=O)CC(Cc2ccccc2)CC)C1 93656,c1(C(C(=O)NC2(CC)CCN(C(c3cnco3)=O)CC2)C)c(C)nc(O)nc1C 93657,CC1=C(C(=O)NC2CCC(NC(C3CC3c3ccccc3)=O)CC2)CCO1 93658,C1(CNC(c2nnc(CC)s2)=O)CC(C)N(C(=O)C(F)C2CCC2)C1 93659,c1(OC)ccc(C(=O)NC2CC(NC(=O)C=Cc3cccs3)C2)cc1F 93660,c1(OC)ccc([N+](=O)[O-])cc1NNC(=O)C1CCSCC1 93661,N1(C(=O)Nc2c(Cl)cn(CCC)n2)CCC(N(C)CCOCCO)C(C)C1 93662,c1(C(c2nnnn2CCC2CC2)NC(CCC(=C)C)C)ccc(C)cc1[N+](=O)[O-] 93663,C(=O)(CC(C)(C)C)NC(C)C(=O)N(C1CCN(C(=O)CSc2cn[nH]c2)CC1)C 93664,CC12CC(CC(=O)NC3(C)CN(C(=O)CC4CCCOCC4)C3)(CO1)C2 93665,c1(OC)ccc(NC(=O)N(CC(O)CC(F)(F)F)C2CC2)cc1OCC(N)=O 93666,c1(CNC2C(C(N3CC(COC)C3)=O)CCC2)ccc(CO)cc1 93667,C(CCN(C)C(c1ccc(-n2cncn2)cn1)=O)(C(C)C)NC(CSCC=C)=O 93668,CCCCC(CC)CC(=O)NC1CCN(C(c2cc(O)ccc2F)=O)C1 93669,N1(C(CC2(OC)CCCCC2)=O)CC(CNC(=O)C(C)SC)C(C)(C)C1 93670,CC(C)CCC(O)C(=O)NC1(C)CCN(C(c2ccc(C(F)(F)F)s2)=O)C1 93671,c1(CC(=O)NCCN(C(=O)C(O)C(F)(F)F)CC)ccccc1S(C)=O 93672,c1(NC(C(CCC)NC(C2CC=CCC2)=O)=O)cnc2ccnn2c1 93673,Cn1nc(C(N2CC(O)CCC2C(N2CCC3(CC2)CC3)=O)=O)cc1C#N 93674,c1(C(N(CC(CN(C(c2cc(CC)[nH]n2)=O)C)O)C)=O)sc(C)nc1C(F)(F)F 93675,C1(CNC(C(C2CCCC2)OC)=O)CCN(C(C2CCCCS2(=O)=O)=O)CC1C 93676,N1(C(C(Cc2cnn(C)c2O)NC(=O)CCCF)=O)CCNC(=O)CC1 93677,C1(NC(c2cc(C)sn2)=O)CCN(C(=O)Cc2cscn2)CC1(C)C 93678,CCC(COC)S(=O)(=O)NC(=O)CCc1nc(C(C)C)no1 93679,C1(C(N2C(CNC(CCOC)=O)COCC2)=O)CCc2ccc(F)cc2C1 93680,Cc1cc(C(=O)NC(CO)C(C)NC(=O)CC(C)C2CCCCC2)nnc1O 93681,c1(OC)cc(C#N)ccc1C(N1CC(N(C(=O)C(c2ccccc2C)C)C)C1)=O 93682,c1(C(N(C)CC2N(C(c3c(CC)nc[nH]3)=O)CCC2)=O)cc(C)nn1C1CCC1 93683,C1(C(=O)Nc2ccc(Br)nc2)CC12CCN(Cc1ccc(Br)cc1F)C2 93684,N1(c2nc(C)nc(C#N)c2)CCCC(C2(NC(C3C4CC5C(C4)C35)=O)CC2)C1 93685,C1(C(=O)NCC(C)(C)NC(=O)C(c2ccc(Cl)cc2)OC(F)(F)F)CCCC(=O)O1 93686,C=CCC(C(=O)NCC1CC2(CC2)CN1C(c1cnncc1C)=O)C(C)C 93687,c1(C(=O)OCC(=O)N(C2CCCC(C)C2)C(C)(C)CO)cc2scc(Cl)c2[nH]1 93688,C(N=c1[nH]cnc2cc[nH]c12)C1CCC2CN(C(=O)OC(C)(C)C)CC21 93689,n1(CC#C)c(C)cc(C(N2CCCC(NC(c3[nH]ccc3C3CC3)=O)C2)=O)c1C 93690,c1(NC(C2(COC)CC=CCC2)=O)cc(P(C)(C)=O)ccc1COC 93691,C1(O)(CNC(C(C2CCC2)SC)=O)CCN(C(=O)CCC=CC(C)C)C1 93692,c1(C(=O)NC2CC(N(C(C(C=C)(C)C)=O)C)C2)cc(F)c(Cl)c(N)c1Cl 93693,c1(OC)cc(C)c(C(=O)OCCCCN2CCCCC2=O)cc1OC 93694,CC1CC(N=c2[nH]c(C(C)(C)C)nc(=N)[nH]2)CCN1C(c1ccn(CCF)n1)=O 93695,C1(C(=O)NC2CCN(C(C3(c4ccsc4)CC3)=O)C2)CCC(CO)CC1 93696,CC1C(C)N(C(=O)CC(C)c2ccncc2)CCN1C(c1ccc(F)cc1)=O 93697,CCC(C)C(C(=O)NCC1(C)CN(CC=CNC)CCO1)OCc1ccccc1 93698,CC(C)CC(CC(=O)NC(C1CCC1)C)NC(c1ccc(O)cc1)=O 93699,Cc1oc(C(N2CC3CC3(NC(=O)CC3CC4CC4C3)C2)=O)cc1Br 93700,C(C(C)(C)CC(=O)NCC1(CO)CC2CC2C1)NC(c1c(CCC)nco1)=O 93701,N1(C(C(N2CCSCC2)C)=O)CCC2C(C1)CN2C(c1cncc(C(N)=O)c1)=O 93702,c1(NC(C)=O)ccc(N)c(C(=O)NCCN(C)C(C2CC2C)=O)c1 93703,C1(C2CC2)C(=O)NOCC(=O)N1.C#CCCSC 93704,c1(C(=O)NCC(Br)Br)ccc2c(c1)CCOC2 93705,N1(C(COCCC=C)=O)CC2CCC1C(NC(c1ccc(Cl)c(F)c1O)=O)C2 93706,N1(C(C2(C)CCCO2)C(=O)NCCC(=O)OCC)CC2CS(=O)(=O)CC2C1 93707,C12(C(NOCCOCC)=O)CC(CO)(CN1C(=O)CN(C)C)C2 93708,C(=O)(CS(=O)(=O)CC(C)C)NC1(C)CCC(NC(c2ccc(C#C)cc2)=O)CC1 93709,c1(C(N2CCCC(C(C)(C)C(=O)O)C2)=O)ncn2c1CCC2 93710,Nc1c(-c2ccccc2)nsc1C(N1CC(O)C(O)C1)=O 93711,c1(CCC)cc(OC)nc(N2CCCCCC2C)n1 93712,c1(CC)nc(C(=O)NC2CC(F)(CNC(C3CC3OC)=O)C2)c2ccccn12 93713,CCCC(C)(O)C(=O)NCC1(F)CCN(C(=O)CCc2ccc(Cl)nc2)C1 93714,CC1(C)CCCC(CC(=O)NCC2CC(O)CN2C(=O)Cc2csc(Cl)c2)C1 93715,c1(Cn2cc(CNC3CC(C(C)C)SC3)nn2)ccccc1O 93716,c1(C(=O)NC(C(C)(C)C)CNC(C2(CO)CCCC2)=O)ccc2cccnn12 93717,CCC(CCOC)C(=O)N1CCCC(CCNC(C2(O)CCSC2)=O)C1 93718,N1(C(=O)NC(CC#C)C)CCC(CNC(=O)CC2(C)CC2)C(CC)C1 93719,C1(CNC(=O)C2=CCOCC2)CC2(CCC2)CN1C(=O)COc1ccccc1F 93720,C1(O)(C(C)NC(c2ccsc2)=O)CCN(C(c2coc(CO)c2)=O)C1 93721,N1(C(C(C)n2ccnc2)=O)CC2(CCCCN2C(=O)C(N2CCOCC2)C)C1 93722,C1(C(N(CCCCCC)C)=O)CC2(CCC2)CN1C(C1CCCCC(=O)N1)=O 93723,CC1CCn2ncc(C(=O)NCC(C)(CO)NC(c3ccc(N)cc3O)=O)c2C1 93724,C(c1cccc(O)c1O)=CCNC(=O)NC12CC(C1)C2 93725,Cc1c(Cl)c(C(=O)NCC2(C)CCC(NC(C3(C)CCSCC3)=O)C2)nn1C 93726,N1(C(C(=O)NCCOC)C(C)CC2CC2)CCc2c(C#N)cccc2C1 93727,CC(CN=c1nc(N2CCCC3(CCCO3)CC2)c2[nH]ccc2[nH]1)C(C)(F)F 93728,C(N=c1cc[nH]cc1S(=O)(=O)NCC1CCOC1C)c1ccc(C(C)C)cc1 93729,c1(OC)cc(CC2CC2CN2CCOC(C(F)(F)F)C2)c(F)cn1 93730,C1(CNC(CC=C)=O)CCC2(CCN(C(=O)CNC(=O)C3CC3)CC2)CO1 93731,c1(C(N(CCN(C(C(C(C)C)C)=O)C)C)=O)ccc2nnc(C(F)F)n2c1 93732,c1(NC(C2CN(C(c3ccc(O)cc3Cl)=O)CCC2O)=O)cccc(Br)c1 93733,N1(C(C(=O)NC(C(=O)OC)C)C(C2CC2)OC)CC(C)C12CCOCC2 93734,N1(C(C(NC2C(C)(C)COc3ccccc32)=O)=O)CCc2cc(Cl)cc(Cl)c2C1 93735,C1(CNC(C(=O)NC(C)C)=O)CC2(C1)CN(C(=O)COCCCF)C2 93736,N1(C(C(COC)OC)=O)CCC2(CCN(C(C3CS(=O)(=O)C3)=O)C2)C1 93737,C1(CNC(C2(S(N)(=O)=O)CC2)=O)CCC2CN(C(=O)CCNC(N)=O)CCC2C1 93738,Cc1nc2n(c1C(N1CCCC1c1ccn(C)n1)=O)CCCC2 93739,c1(CC)csc(C(=O)NC(c2nccn2C)c2nnnn2C2COC2)c1C 93740,c1(-c2cn(C(C(=O)N(C(C)C(F)F)C3CC3)C)nn2)cccc(F)c1Br 93741,N1(C(CC(C(CC)C)O)=O)CCN(C(c2ccncc2F)=O)CC2(CC2)C1 93742,C1(C(C)NC(C(C2CC2)OCC)=O)CCN(C(=O)C(F)CC2CCC2)C1 93743,NS(=O)(=O)c1n[nH]cc1C(N1CCN(C(=O)C2=NOCC2)C(CC(F)(F)F)C1)=O 93744,N1(C(C2CSCN2S(=O)(=O)CC2(c3nn[nH]n3)CCC2)=O)CCOCC1 93745,N1(C(COCC=C)=O)CCCN(C(c2c(C(F)(F)F)cccc2F)=O)CC1C 93746,CC1=C(C(=O)NC2CC(C(=O)Nc3cccnc3C)C2)CCO1 93747,C(CSC)(C(=O)N(CCC(=O)NCC1CC1(Cl)Cl)C(C)C)OC 93748,CC1CC(C(=O)NC2(CC(=O)N(C3CC4(CC4)C3)C)CCC2)CCS1 93749,CC(C)CC(C(=O)N(C(C)CCNC(=O)CCCN=[N+]=[N-])C)C(C)C 93750,CC1=CCC(C(N2CC3C(C2)N3C(c2cc(Cl)c(Cl)s2)=O)=O)CC1 93751,c1(NC(=O)Nc2cc(CN(C)C)cc(C(F)(F)F)c2)cc(F)c(Br)cc1Cl 93752,C1(NC(COC)=O)CCCCC1C(=O)NC1COCC1CN(C)C 93753,CC1CN(C(C2(n3cnnn3)CC2)=O)CCC1N(C(=O)CC1(C)CCC1)C 93754,c1(C(N2CC(CCNC(c3c(C)nsc3)=O)C(C)C2)=O)cc(N)c(F)c(F)c1Cl 93755,C1(C(=O)OC)CCC(C2CCCCC2)CN1C(=O)NC1CCCC(C(F)(F)F)O1 93756,C12(COC)CC(NC(C3CSCCS3)=O)(CN1C(c1cc(Cl)n(C)n1)=O)C2 93757,C=CC(CCC)CC(=O)N1CC(NC(C2CSC2)=O)C2(CCC2)C1 93758,CC(C)C(F)(CNC(=O)CCCC1CC1)C(=O)N(C(CO)C(C)C)C 93759,N1(C(C=CC2(C)COC2)=O)CCCN(C(c2ccc(Cl)o2)=O)CC1 93760,Cc1ccc(C(C)CNN(C(=O)CN2CCC2C)CCN(C)C)s1 93761,c1(C(C)(F)F)ccc([N+](=O)[O-])cc1C(=O)NC1CC1CNC(c1ccon1)=O 93762,N1(C(c2ccc(C)o2)=O)CCC(NC(c2cc[n+]([O-])cc2)=O)C2(CCC2)C1 93763,C(=O)(C1=CC2CCCCCCC12)NCCOCCNC(CCCCCOC)=O 93764,C1(CNC(C(C)(C)n2ccnn2)=O)CC(C(=O)NCCCCCCF)=NO1 93765,CC(CC(=O)N1CCC(C(N2CCCC(CO)CC2)=O)O1)c1ccco1 93766,C1(CC=C)(N(C2CCC(C)CO2)C(=O)CCC)CCN(C(=O)CC)C1 93767,c1(C(C)NC(C(=O)N(C2C(OC)COCC2)C)=O)ccnc(Cl)c1F 93768,C1(C(=O)NC(CCOC)CNC(C2CC2C)=O)CCN(C2CC2)CC1 93769,c1(CC(=O)NCC2N(C(c3c(CC)occ3)=O)CCC2C)cccc(O)c1F 93770,C12CC3CCC(C1)N3C2=O.c1(OC)ccc(C(C)Nc2cc(F)c[nH]2)cc1 93771,N1(C(c2ncsc2C(C)C)C(=O)NCCOC)CCCC(N(C(N)=O)C)C1 93772,c1(C(=O)NC(CNC(CNS(CC)(=O)=O)=O)C2CCC2)c(S(C)(=O)=O)cnn1C 93773,N1(CC(N2CCC(c3nc(CC)[nH]n3)CC2)=O)C(=O)CCC(N)C1=O 93774,N1(C2C(=O)NCC2)CCC2(CCN(C(C3C4C5CCC(C5)C34)=O)C2)C1 93775,C1(C)(COC)CCCN(C(=O)C(C)N(C(c2csnc2Cl)=O)C2CC2)C1 93776,c1(C(=O)NCC2CC(NC(c3c(C)cc(O)nn3)=O)C2)c(O)ncc2c1CCC2 93777,C1(OC)CC(CNC(C2(C#N)CCC2)=O)N(C(c2c(C)n[nH]c2C)=O)C1 93778,N1(C(c2ncc(CCNC(C3(C)CC3)=O)s2)=O)CCCC2(CCO2)C1 93779,c1(NC2C(C3CCN(C(C(=O)OCC)=O)CC3)OCCC2)cccc2[nH]ncc12 93780,c1(CC(=O)NCCOCCCN(C(=O)CC2CCCO2)C)cncc(F)c1 93781,c1(OC)cnc(F)c(C(=O)NCCCC(CO)NC(C2(C)COCCO2)=O)c1 93782,N1(C(COCC(=C)C)=O)CCC(C)(CC(=O)N(CC(C2CC2)OC)C)C1 93783,N1(C(c2c(C)[nH]nc2Cl)=O)CCN(C(C2CC2F)=O)C(c2cc(F)ccc2F)C1 93784,N1(CC)CCOC(CSCC2C(NC(=O)NC(=O)Cn3nnc(C4CC4)n3)C2)C1 93785,c1(C(N(C)CC2(O)CCN(C(c3nnc(C)s3)=O)CC2)=O)cc2ccccn2n1 93786,N#Cc1cc(C(N2CCN(C(C3(Cl)CC34CCOCC4)=O)CC2)=O)ccc1F 93787,c1(C(=O)NCCCC(C)NC(CC(C(C)C)O)=O)cc2c(Cl)ccnc2s1 93788,Nc1nccnc1C(N1CCC1CNC(c1c(Br)n[nH]c1Br)=O)=O 93789,N1(CC)CC(NC(=O)C(CO)NC(=O)C(C2CCCCC2)C)C(C)C1 93790,C1(NC(c2c(CC)onc2)=O)CCC2(CC1)CC2NC(C12CC3CC1C2C3)=O 93791,N1(C(c2n(CC)nnc2)=O)CC2CCCC1C2CNC(c1cnc(Cl)s1)=O 93792,c1(NC(CCC)C)ccc(S(=O)(=O)N2CCC(CCO)C2)cc1Br 93793,C1(CC(=O)NCC2C3CN(C(C4C(Cl)(C(=O)OC)C4)=O)CC32)COCC(C)(C)O1 93794,c1(C(N2C(C(NOCC=CC)=O)CCC2C2CC2)=O)cccc(O)c1F 93795,N1(C(CCCOC)=O)CC(OC)C(NC(=O)CCCc2nccs2)C1 93796,CCC(C(=O)N(CCC(C)N(C(c1[nH]nnc1C(F)F)=O)CC)C)N(CC)CC 93797,C1(CC)CN(C(c2cc(C)n(C(C)C)c2)=O)CCC1NC(C1CC(F)CN1C)=O 93798,CC(CC(=O)NC1CCCN(C(=O)Cc2nn(C)cc2Br)C1)C(F)F 93799,c1(CN(CCC)Cc2ccc(-c3ccnnc3)cc2C)ccc2cc[nH]c2c1 93800,C=CCC(C(=O)NCC1CCC(NC(c2cc(C3CC3)sn2)=O)CC1)C(C)C 93801,C(=O)(CC(C)CC(C)C)NC1(CCOC)CCN(C(=O)CC=C(Cl)Cl)C1 93802,C1(C(C)(C)NC(=O)CCN2CCC2)CCN(C(c2ccc(OCCF)cn2)=O)CC1 93803,c1(CCC)nnc(C23CC4CC2C3C4)n1C1CC(c2ccccc2)C1 93804,N1(C(C(CCC)CNC(=O)CC(C)CC)=O)CCC(C)(C#N)CC1 93805,C(CCN=c1nc(-c2ccncc2)cc[nH]1)N(C(C(C(C)S(C)(=O)=O)C)=O)C 93806,C1(CC)CC(OC)CN(CC(=O)NNC(=O)c2cccnc2)C1 93807,Cc1cc(CC(=O)NCC(CC(C)C)NC(c2sccc2C)=O)n(C)n1 93808,c1(C(=O)NCCN(C(C2CC(=O)N(O)C2)=O)CC)ccc2cn(C)nc2c1 93809,N1(C(C2C(COC)CC2)=O)CCCC(CO)(NC(=O)CC(CC)C2CCC2)C1 93810,c1(NC(C2OCCN(Cc3cccc(OC)c3Br)C2)=O)c(F)ccc(F)c1OC 93811,c1(SC)cccc(C(=O)N(CCCCNC(c2occc2C2CC2)=O)C)c1 93812,N1(C(C(C)(CO)NC(C)=O)=O)CC2CCCN(C(=O)C(CC(C)C)C(N)=O)C2C1 93813,c1(C(N2CCC(CNC(c3ccccc3NCCO)=O)C2)=O)ccc[n+]([O-])c1 93814,c1(C(N2CCC(CC)(CO)C2)C(=O)NCCSC2CC2)ccnc(P(C)(C)=O)c1 93815,C(N=c1[nH]c(=NC(C)C(C)F)[nH]c2c1SCC2)c1c(Cl)ccc(OC)c1 93816,C1(C(=O)NC(CN(CCCOc2nccc(C)c2)C)C)CCCCNC1=O 93817,c1(CC(=O)NC(CN(C(=O)C=C(C)c2ccsc2)CC)C)cc[nH]c(=N)c1 93818,c1(OC)cc(CCNC(C2C3CCCC3CN2C)=O)cc(OC)c1OC 93819,Cc1ccc(C=CC(=O)N(CC(=O)NCC2CCC2)CC(C)O)o1 93820,N1(C(C(n2ncc(C)c2)C)=O)CC=CC(C(=O)NCCN2CCC(O)C2)C1 93821,N1(C(c2ncc(C(C)(C)C)s2)C(=O)NCCCCCC)Cc2ncsc2C1 93822,N1(C(COC(c2ccn(C)n2)=O)=O)CCCCC1CCCNC1CCO1 93823,CC(CC(=O)NCCCNC(=O)Cc1csc(-c2ncccn2)n1)C(C)(C)C 93824,C(=O)(CC(C)(C)C(=O)N1CC2CC(NC(c3ccnnc3)=O)C2C1)OCC 93825,N=c1[nH]nc(CC(=O)NC2CCC(NC(=O)CCN3CCC(F)C3)C2)s1 93826,C1(c2nnnn2Cc2ccccc2)(NCc2scc(C)n2)CCOC2(CCC2)C1 93827,C(CCCCCC=C)NC(C(CN(C(c1c(C#C)c[nH]n1)=O)C)C)=O 93828,N1(C(c2ccc(F)c(F)c2Br)=O)CCOC2(C1)CN(c1ncncc1I)C2 93829,C1(NC(CC(CC)SC)=O)CCN(C(=O)COc2cccc(F)c2F)C(C)C1 93830,C(CS(=O)(=O)CC(=O)N1CCC(C(C)(C)NC(C2CCCC(F)(F)C2)=O)C1)OC 93831,C1(C(=O)NC2(c3onc(C)n3)CC2)C2CCC(C2)N1C(=O)CC1CCNC1=O 93832,CC1COc2c(C(N3CCNC(C4CCOCC4)C3)=O)cccc21 93833,c1(OC)ccc(C(N2C(C(=O)Nc3nc(C4CC4)cs3)CC3CC23)=O)cc1I 93834,N1(Cc2c(OC)nccc2I)CCC2CN(C(=O)Cc3ccc(O)cn3)CCC12 93835,C(=O)(CS(C)(=O)=O)NCC1N(C(CN(C)C(C2CCC(F)(C(=O)O)C2)=O)=O)CCC1 93836,C1(C)(C(=O)NCC2(OC)CN(C(=O)CCc3cccc(C)c3)C2)CCC(C)C1 93837,C12(C(N3CC(CC=C)(NC(c4cc(C(N)=O)cs4)=O)C3)=O)CCCCC1C2(F)F 93838,C1(NC(Cn2c(C)csc2=O)=O)CCN(C(C2CCCC(C#N)C2)=O)CC1(C)C 93839,Cc1nc(C(=O)N(C)C)ccc1C(N1CC(C2(NC(=O)C(C)N(C)C)CC2)C1)=O 93840,N1(C(c2c(C)ccc(C)n2)=O)CCC2(CCN(C(c3ccncc3)=O)CC2)C1 93841,C1(C(N(C)Cc2nnc(C)o2)=O)CCC2(CC2)N1C(=O)C(O)CC1CCCC1 93842,N1(C(C(C)n2cccc2)=O)CCCC(C(=O)NC2CCCC(O)C2)CC1 93843,C1(COC)(CNC(=O)C(C)(C)SC)CCCN1C(=O)C=Cc1cncs1 93844,Fc1ccc(F)c(-n2cc(C(c3cccc(F)c3F)C3CC3)nn2)c1 93845,c1(C(=O)OC)ncc(Br)cc1NC(C1CCN(C(C2CC(C)(C)C2)=O)C1)=O 93846,c1(C(=O)NC(C(C)C)CNC(=O)C(O)c2ccsc2)ccn2c1CCC2 93847,c1(C(N2CCCC(CN(C)C(C3CC4(C3)CC4F)=O)C2)=O)c(F)cc(O)cc1F 93848,C1(S(=O)(=O)NC2CCN(c3ccccc3OC)C2)(OC)CC1 93849,c1(C(N(C2CN(C(=O)Cn3ncccc3=O)CC2F)C)=O)scc2c1OCCO2 93850,C(=O)(C(C)(C)C(=O)NC(C)C=CC(N1CC2C(CO)C2C1)=O)NC 93851,N1(C(CCNC(=O)OC)=O)CCCCC1CNC(C1OC2CCC1C2)=O 93852,c1(C(=O)NCC2CN(C(C(CC)C(C)C)=O)CC2O)ccc2c(c1)OCCCO2 93853,c1(C(C)CNC(=O)Cc2sccc2Br)cccc(C(F)(F)F)c1 93854,Cc1cc(C(=O)NC2CCCC(CNC(=O)Cc3ccnc(F)c3)C2)nc(C)n1 93855,c1(NC)ccc(C(=O)NCC2CCCCCN2C(c2ccn(CC)n2)=O)cc1F 93856,c1(C2(CNC(C3CCCN(S(C)(=O)=O)C3)=O)CC2)ccc(C#N)c(Cl)c1 93857,CC1OCCOC1C(=O)NC1(c2ccccc2)CCN(C(=O)Cc2ccsc2)C1 93858,CCC(C(=O)NC(C1CCCC1)CNC(c1cn2ccnc2cn1)=O)C(F)(F)F 93859,C=Cn1nncc1C(=O)NCC(CCNC(c1ccsc1Cl)=O)OC 93860,c1(CC(=O)NC2(CCNC(C3(C(=O)NC)CC3)=O)CCC2)cccc(F)c1Cl 93861,C1(CNC(c2scc(OC)c2)=O)CN(C(=O)C=C2CCSCC2)CCN1C 93862,c1(NC(C)CN2CCCC2=O)cccc(OC(C)(C)C)c1 93863,c1(C(c2nnnn2-c2cccc(OC(F)F)c2)NCCCC=C)ccc(F)cc1F 93864,c1(C(=O)NCC(CCNC(CN(C2CC2)CC)=O)O)cccn(C)c1=O 93865,c1(C(=O)NC2CC(C(N3CCN(S(C)(=O)=O)CC3)=O)C2)ccc(I)cc1F 93866,C1(CC)CC(O)CCN1C(C1COCC1NC(c1cnn(C)c1)=O)=O 93867,N1(C(C2C(C)OC(C)C2C)=O)CCCC(C2CCN(CCS(C)(=O)=O)C2)C1 93868,n1(CCCC(=O)NC(C)C(c2ccccc2)NC(=O)C2=CCC2)ccccc1=O 93869,C1(C(N2C(CNC(=O)CCCC3CC3)CC3(CC3)C2)=O)CCc2nncn2CC1 93870,c1(C(N(C2CCN(C(C34CC(CC(F)F)(C3)C4)=O)C2)CC)=O)sc(NC)cc1C 93871,c1(C(N(CCCN(C(C(C2CCCCC2)OCC)=O)C)C)=O)cnn(C(C)C)c1 93872,CCS(=O)(=O)CC(=O)NC(CCC1CC1)C(=O)NC1(CO)CC1.CSC 93873,N1(C(C(C2CC2)OCC)=O)CCC(CNC(c2cc(O)n(C)n2)=O)C(O)C1 93874,C1(CCCCCNC(CCC#C)=O)CCN(C(c2ncn(C)c2C)=O)CC1 93875,N1(C(COCc2cc(C)no2)=O)CC(CNC(=O)C=C2CCCC2)CCC1C 93876,c1(SCC)ccccc1CC(=O)NCC1CC(O)CN1C(=O)COC(F)F 93877,n1(C2CC(=O)C2)cnc2c(N3CCC(CC(=O)O)C(F)(F)C3)ncnc12 93878,C12(C(=O)OC)CCCC1N(C(c1csc3ccccc13)C(=O)NCC(C)C)CC2 93879,C1(NC(C(F)=C(C)C)=O)CC1C1CCN(C(c2nccc3cccnc23)=O)CC1 93880,c1(CC)ccc(C(=O)NC2(C)CCN(c3ccc(OC(C)C)nn3)C2)cc1 93881,C1(C(=O)NCC(C)(O)C(F)F)CC12CCN(C(=O)Cc1cncs1)CC2 93882,Cc1ccc(C(F)F)cc1C(=O)NC1CC(C)(NC(=O)CC2CC=CCC2)C1 93883,c1(C(=O)NC2CC(NC(CC(C=C)C)=O)C2)c(C)nn(CCO)c1C(F)F 93884,S(=O)(=O)(c1cccs1)N.C1(C(c2c[nH]c(C(F)(F)F)c2C2CC2)=O)CCNCC1 93885,C1(NC(CSC(C)C)=O)CCC2(C1)CN(C(C1(C(C)(F)F)CC1)=O)C2 93886,C1(C(=O)NCC2(O)CC(C(=O)NC(CC)C(C)(F)F)C2)CCC2CC1CO2 93887,CC1CCN(C(C2(C)CCOC(C)C2)=O)CC1CNC(c1nccnc1Cl)=O 93888,C(C(C)C(=O)N=c1ccn(C(C)(C)C(=O)OC)[nH]1)OC 93889,C1(C)(C(N2CCC(NC(C3(CCOC)CC3)=O)CC2)=O)CCN(C)C1=O 93890,CCC(CNC(C12CC(CC(F)F)(C1)C2)=O)(CC)NC(c1cn(CCO)nn1)=O 93891,c1(C(=O)OC)sccc1S(=O)(=O)Nc1cc(C(=O)O)cc(C(C)C)c1 93892,C1(NC(C=NOC)=O)(CNC(=O)C(C2CC2)OCC)CCCCC1 93893,CCC(C)(C#N)C(=O)N1CC(NC(c2oncc2C)=O)C(C)C1 93894,Cc1ncc(OCC(N2CCC(NC(c3csc(F)c3)=O)C2)=O)c(C)n1 93895,c1(CC(N2C(CNC(C(CC)C(C)C)=O)COCC2)=O)c[nH]c2cnc(Cl)cc12 93896,c1(SCC)cc(CC(N2CC(C(=O)OC)C2)=O)cs1 93897,c1(C(=O)NCC(C)NC(C(c2ccccc2)NC(CC)=O)=O)cc(O)n(CC)n1 93898,C(=O)(C(CCC(C)(C)C)OC(=O)CCc1cc(O)ccc1Br)OC 93899,N1(C(c2ccc(COC)[nH]2)=O)CC(C)CCC1CNC(c1nccc(C)n1)=O 93900,C1(CC(=O)NCC(C)(O)CNC(c2c(F)cncc2Cl)=O)CCS(=O)(=O)CC1 93901,C1(NC(c2cc(CC)on2)=O)CC(CNC(c2cc(C)c(C)o2)=O)C1(C)C 93902,C(=O)(C(O)CCCNC(c1c(C)ccnc1O)=O)N1CCC(CC=C)C1 93903,N1(C(c2c(CC)cc(N)cc2)=O)CCCC2(NC(c3ccc(OC)s3)=O)CC2C1 93904,c1(CN(C(=O)NCC2(C)CCCC2C)CC)ccc(Br)cc1 93905,C1(n2cc(CCN(C(CC(CSC)OC)=O)C)nn2)CCCCNC1=O 93906,CCCC(O)CN(C)C(c1cn(CCNC(=O)C(O)C2CCC2)nn1)=O 93907,C1(NC(C2(OC)CCSC2)=O)CCCCC1NC(=O)C(c1ccccc1C)(C)C 93908,C1(C(=O)NCCC(C)NC(C(C)Cc2cccc(F)c2)=O)CC(C(C)(C)C)=NO1 93909,c1(C(=O)NCC(CNC(C=Cc2ccc(CC)o2)=O)O)ccc(O)c(C)c1 93910,N1(C(c2cc(OC)ncn2)=O)CCOC(C)(CNC(=O)Cc2cccnc2C)C1 93911,CN1CCC(CC(=O)N(Cc2ccccc2)Cc2ccccc2)C1 93912,CC1(C)CC(CNC(=O)CCc2nc[nH]n2)CCN1 93913,c1(CC)cc(N)ccc1C(=O)NCC1CCCCN1C(=O)CCc1cnc(O)[nH]1 93914,c1(C(N(C2CCCN(C(=O)CSC(F)F)C2)C)=O)cc2cccc(F)c2cn1 93915,S(=O)(=O)(c1ccc(NC(c2ccc(C)cc2)CCO)cc1)C(CC)C 93916,c1(C(=O)OC)cnc(C)[nH]c1=NCCC(C)NC(=O)C1CCCc2n[nH]cc21 93917,CCCC(CNC(=O)C(=O)C(C)(C)C)C(=O)N1CC(N2CCCC2=O)C1 93918,C1(NC(C2N(C(C)=O)CCOC2)=O)CC2(C1)CN(C(C1CC(NC(C)=O)C1)=O)C2 93919,C1(NC(C2CCS(=O)CC2)=O)CCCN(C(=O)CCC2CCCCC2)CC1 93920,N1(C(c2c(SC)cccc2)=O)CC(CNC(C23C4C5C6C4C2C6C35)=O)CC(C)C1 93921,Cc1cc(F)c(C(N2CCCC2CN(C)C(C2CC=CC2)=O)=O)cc1F 93922,n1(CC)cc(CNC(C2CN(C(c3ccc[nH]3)=O)CCO2)=O)c(C)n1 93923,c1(OC)ccc(NC(=O)C2CC2)cc1NC(=O)NCc1ccccc1C(C)C 93924,c1(OC)ccc(C(N2CC3CCC2C3NC(=O)C#CC(=O)N(C)C)=O)c(N)c1F 93925,N1(Cc2cc(COC)no2)CCC(=O)N(CCC(C(F)(F)F)OC)C1=O 93926,C1(NC(=O)C=Cc2cscn2)CC2CCC1(CNC(c1cc(Cl)c[nH]1)=O)C2 93927,c1(C(=O)NC(CNC(C2(COC)CCCO2)=O)C)ccc(Cl)c(N)c1 93928,N1(C(C2(C)CCOC2)=O)C2CCC1C(NC(c1cnc(C3CC3)[nH]c1=N)=O)C2 93929,C(CCc1cccc(C(F)(F)F)c1)(C(N)=O)NC(C(=O)N(CC(F)Cl)C)=O 93930,c1(C(=O)NCC2(NC(C(CC)NC(C)=O)=O)CC2)ncc(F)c(OC)n1 93931,Cc1oc(C2CCOCC2)nc1C(=O)NCCCNC(=O)Cc1nncs1 93932,Cc1nc2ccc(C(=O)OCN3CCCN(C(C(=O)NC4CC4)=O)CC3)cc2[nH]1 93933,CC1CSc2ccc(Br)cc2C1NC(c1c(N)ccc(Br)c1F)=O 93934,c1(C(N2CCCCC(CNC(C3(C4CCC4)CC3)=O)C2)=O)cccn2cncc12 93935,N(C(=NCc1ccn(CCOC)n1)NCCNC(C)=O)C(c1cnc(CC)o1)C 93936,CC(CCc1ccccc1)CC(=O)NCC1(O)CN(C(=O)CC2CCCOC2)C1 93937,n1(C(C)C)nccc1C(=O)NC(C1CCCN1C(C1CCC1C)=O)C 93938,C(=O)(CN=c1cc[nH]cc1)NCC1CCN(C(c2c(CC)noc2)=O)C1(C)C 93939,c1(C(N2CC(CNC(C(CC=C)OC)=O)C(C)C2)=O)cc2ccccc2o1 93940,c1(C(=O)NC2CCC(NC(CSCC(=O)OC)=O)C2)csc2cccnc12 93941,C1(C(N2CC3C(CNC(c4c(C)nco4)=O)(C3)C2)=O)C(O)C(=O)N(C)C1C 93942,N1(C(C2(c3ccccc3)CCCN2)=O)CC2CC23CC13 93943,CC(C)(O)CC(=O)NC1CC1NC(C1(c2ccc(O)nc2)CCC1)=O 93944,c1(CC)ccc(C(=O)NCC2CCCCCN2C(C2CCC(=O)C2)=O)cc1Cl 93945,Cc1snnc1C(N1CC(CCO)(NC(c2cc(C(N)=O)cs2)=O)C1)=O 93946,C(=O)(CS(=O)(=O)c1ccccc1Cl)NC(CNC(C1N2CC(C)N(CC2)C1)=O)C 93947,CCC(CCC(=O)NCCCC(C)NC(=O)CNS(N)(=O)=O)OC 93948,N1(CCC(=O)OC(CN(C(C)=O)CC)OC)c2ccccc2Sc2ccccc21 93949,Cc1nc(O)nc(C)c1C(=O)NCC(C)(O)CNC(C1CC=CCO1)=O 93950,C1(COCc2cccc(NC(CC(C)(C)SC)=O)c2)CCc2ccc(F)cc2O1 93951,Nc1ccc(CCCC(=O)N2CCC(NC(=O)C=CC(F)(F)F)C2)cc1 93952,C1(CNC(CSCC=C)=O)CC2CCC1N(C(c1cc(C)nc(N(C)C)n1)=O)C2 93953,N1(C(C(C)OC)=O)C2CCC1CC(NC(=O)Cc1ccc(O)c(C)c1)C2 93954,c1(C(=O)NCC2C(NC(CCNC(=O)NC)=O)C2)ccc2c(c1)COC2 93955,N1(C(c2ccnc(C)c2N)=O)CC(NC(=O)CCC2CC2)C2CCCC12 93956,C1(NC(C2(CCOC)CC2)=O)C2CC(NC(C3(O)CCC3)=O)CC12 93957,c1(C(=O)NC2(CNC(C(C(C)C)F)=O)CC(F)(F)C2)nccc2n[nH]cc12 93958,c1(N)cn(C(C)C)nn1.c1(C(N(C(C)C)C2CC2)=O)ccnn1CC(F)(F)F 93959,N1(C(c2ccc(C)c(O)c2)=O)CC2CC1CCC2NC(c1cc(Cl)c[nH]1)=O 93960,CCC(C)(C)C(=O)N1CCCC(CC(=O)NCCCNC(=O)OC)C1 93961,c1(C(N(C2CCCN(C(C(C)NC(C)=O)=O)CC2)C)=O)cc2ccc(F)cc2[nH]1 93962,CN1CC(C)(C(=O)NCC2CC(NC(c3cccc(OC(F)F)n3)=O)C2)CC1=O 93963,C1(CNC(C=C2CCC(C)C2)=O)CN(C(=O)CC2(C)CC(F)(F)C2)CC1O 93964,c1(SC)cccc(C(=O)NC(CCNC(=O)Cn2cnnn2)C(C)C)n1 93965,c1(NCCc2ccc(C(=O)NCc3nccnc3Br)cc2)c(F)ccc(Cl)c1F 93966,c1(C(N2CC(c3nnc(C)o3)OCC2)=O)ccc(F)c(N)c1 93967,C(=O)(C(CC)NC(c1cn(C2CC(CC3CCCCC3)C2)nn1)=O)OCC 93968,C1(C)(C(=O)NCCN2CC(OC)C2)CCN(C(=O)CN2CCOCC2=O)C1 93969,C1(=O)C(C)(O)C(C)N1.Cc1c(-n2cc(C3CC3)nn2)cnn1-c1ccccc1Cl 93970,C(=O)(C(C)(C)C(=O)N1CC(C(=O)NCCCCNc2cccc(F)c2C)C1)NC 93971,C#Cc1cccc(CC(=O)NC2CCOCC2C(N2CCOCC2C(N)=O)=O)c1 93972,CC(C)C(C)C(CNC(=O)C=Cc1cncn1C)NC(=O)CCc1cnn(C)c1 93973,N1(C(CCc2cccc(C)c2)=O)CCN(C(=O)COC2CC=CC2)C(C(F)F)C1 93974,N1(C(Cc2c(F)ccc(C)c2)=O)CC2CCN(C(C3CC4CC4C3)=O)C(C2)C1 93975,C(CC(=O)NCC(C)CNC(=O)CCNC(C1CCCO1)=O)NC(C)=O 93976,c1(-c2scc(C(=O)NCC(C)N(C(=O)CC3COC(=O)C3)C)n2)cccc(Cl)c1 93977,c1(C(=O)NC(CCCNC(C(CC)C(C)O)=O)C)ncn2ccccc12 93978,C1(F)(C(N(CCNC(C2CC2c2ccco2)=O)CCOCCO)=O)CCOCC1 93979,Cc1cncnc1NCC1(CC(=O)NCCc2nn[nH]n2)CCCCC1 93980,C1(C(=O)NCCc2c(C)ncs2)CN(C(=O)CCC(F)(F)F)CC1(C)C 93981,C1(CC(=O)NC2CCS(=O)(=O)C2)CN(c2ccncn2)CCO1 93982,CC(CC(=O)NC(CNC(C1CC1F)=O)CO)n1ccnc1 93983,C=CCC(C(=O)N1CCC(CC)CC1C(=O)NCC(F)Br)C(C)C 93984,C1(C(=O)NCC2(CC)CC2)CCC(NC(=O)C(c2ccsc2)N(C)C)C1 93985,C1(C(=O)NCCc2nc(C)sc2)CC(=O)CN1C(c1c[nH]ccc1=O)=O 93986,C1(OC)CC(N=c2[nH]c(=NCCSc3nnc(C)s3)[nH]c3cccc(F)c23)C1 93987,C1(O)(C(N2CC3(C(=O)OCC)C(C2)CCO3)=O)CCc2ccccc2C1 93988,N1(C(c2cc(CCC)nc(O)c2)=O)CC2CCC1CN2C(=O)C=CC1CCOC1 93989,C1(NC(c2c(CC)noc2)=O)CC2CC1CN(C(c1nc(O)sc1C)=O)C2 93990,C1(C(N2C(c3cn(CC4CNC(=O)O4)nn3)CCC2)=O)CCOCC1C(=O)O 93991,c1(C(CN(C(=O)C(F)Br)C(=O)OC)=O)ccccc1C1CCCC1 93992,c1(N(C(CC)=O)C)ccc(N(C)C(c2ccc(NC(=O)C3CC3)cc2)=O)nn1 93993,Cc1cccc(CNC(=O)C(CNC(C2CC23CCC3)=O)C(C)C)c1C 93994,C1(CNC(C=NOC)=O)CN(C(=O)Cc2n[nH]cc2Br)CCO1 93995,C(C(CC(C)C)C(=O)NCCCN(C)C(c1cc(Cl)cc(Cl)c1)=O)OC 93996,C1(NC(c2cnsn2)=O)CC2CC(NC(c3ccn(CCF)n3)=O)C2C1 93997,N(C)(C1CCc2c(Cl)cccc21)C1CCN(c2cc(C)cc(F)c2)C1=O 93998,C1(CNC(CSC)=O)CC2CCC1N2C(C1(c2ccccc2)CCOCC1)=O 93999,CCC(C(=O)N(CC(C)NC(c1cnn[nH]1)=O)C)OC 94000,c1(C(N2CC(C(=O)NC)OCC2)C(=O)NC2CCOCC2)sc([N+](=O)[O-])cc1Cl 94001,N1(C(C(c2n(C)ncc2)O)=O)CCC2(CC1)CC(NC(C1(C)CCC1)=O)C2 94002,CC1CN(C(=O)CCCNC(N)=O)CCCN1C(=O)CCC(=O)Nc1nccs1 94003,N1(C(C(OC)OC)=O)CCC(NC(=O)C=Cc2ccc(C)o2)CC(C)(C)C1 94004,c1(C(=O)NCC(C(C)(C)C)NC(C2(OCC)CCC2)=O)c[nH]nc1[N+](=O)[O-] 94005,O=C1NCCCC12CCN(c1nc(N3CC4C(C3)C4(F)F)c3ncsc3n1)CC2 94006,CC1(C)OC2C3CC(C2O1)N(C(C1CCC(=O)C1)c1ccncc1)C3 94007,N1(C(c2c(OC)cc(C)s2)=O)CCCOC(CCNC(C2CC2[N+](=O)[O-])=O)C1 94008,C1(C(=O)OCC)(NC2CCN2C(c2cc(Cl)ccc2OC)=O)CC2(C1)OCCO2 94009,C(=O)(C(CC=C)C(C)C)NC(CC#C)C(=O)NCc1ccc[n+]([O-])c1 94010,C1(NC(c2cc(Cl)cs2)=O)CCC2CCN(C(C34C5CC(CC35)C4(F)F)=O)C1C2 94011,c1(C(N(CCN(C(=O)CC(C)(C)O)CC)CC)=O)cc(C)c(C)c2ncsc12 94012,N1(C(C(CCC)C#N)=O)CCC(C)(C)CC1C(=O)NC(c1ncc(C)cn1)C 94013,N1(C(c2c(CC)ccs2)=O)CCC2CN(C(c3nnn4ccccc34)=O)CCC12 94014,C1(COC)CN(C(c2ccsc2S(C)(=O)=O)=O)CCN1C(=O)C#CC1(C)CC1 94015,C12CCN(C1)C(=O)C(C)(C)OCCN2.C(=O)(C(SC)SC)N(C)CC 94016,CC1CN(C(C2(F)CCCC2)=O)CC1NC(c1ccnc(CO)c1)=O 94017,C1(O)(CN(C(C(=O)NC(c2ccccc2O)CC)=O)C2CCCC2)CCSCC1 94018,N1(C(C2(CC(C)C)CC2)=O)CCOC(CCNC(=O)CC2CCCCN2C)C1 94019,N1(C(=O)CCN2CCC(O)CC2)CC2OCC(NC(C34CC(CO3)C4)=O)C2C1 94020,C1(NC(c2cc(C)on2)=O)CN(C(=O)CC(C2CC2)C2CC2)CC1C(F)F 94021,C(C(=O)NC1CCCCC1NC(=O)CCOC1CCC1)(C(C)C)OCC 94022,C1(C(=O)OC)C(C(=O)OC)C2CCC1N2Cc1ccccc1Br 94023,C(=O)(C(C)CC(F)(F)F)NCCC1(NC(C(C2CCCC2)OC)=O)CCOCC1 94024,N1(C(C(CC(C)C)F)=O)CC(NC(=O)Cn2cccn2)CC12CCCCC2 94025,C12(C(=O)NCCCCO)CCC(C(=O)Nc3coc(C4CC4)n3)(CC1)C2 94026,Cc1c(NC2CC(F)C(F)C2)ccc(C(=O)O)c1F 94027,C(=O)(CCCCC(C)=O)N1CCC(C(N2CCC(F)(CO)CC2)=O)(CC)C1 94028,c1(C(N2C(C)CC(CNC(CC=CC=C)=O)C2)=O)cc(Cl)ncc1F 94029,c1(C(=O)CSC2CCOC2=O)cc(N2CCCC2=O)ccc1O 94030,c1(OC)c(F)ccc(C(=O)N(CCCNC(=O)C(O)C(F)(F)F)C2CC2)c1F 94031,c1(C(=O)NCCC(CNC(C2N(CC)CC2)=O)OC)cc2nc(Cl)ccc2s1 94032,C1(C(=O)NC(C=C)C)OCCC1CNC(C1(OC)CCC1)=O 94033,Cn1cc(S(N)(=O)=O)cc1CC(=O)NC1(CNC(=O)Cc2ccccc2O)CC1 94034,C1(C#N)(C(N2CC(C(=O)NCCCC(=O)NC)(CC)C2)=O)CCCCC1 94035,C1(C(=O)NCc2c[nH]nc2C2CC2)(CC)CCCN(C(=O)CC2CC2)C1 94036,CNS(=O)(=O)N1CCC(C(N2CC(CCNC(=O)CC(C)COC)C2)=O)CC1 94037,c1(C(N(C2(C3CCCN3C(=O)CCc3cnn(C)n3)CC2)C)=O)cc(F)cc(F)c1 94038,Cc1[nH]c(C#N)cc1C(=O)NC1CN(C(=O)C2=CC(C)(C)C2)CC1C(F)F 94039,CCCCC(C(=O)NC)NC(=O)C(=O)NC1CC(=O)N(c2ccc(Br)cc2F)C1 94040,c1(OC(C)C(=O)NCCC(C)(C)NC(c2coc(Cl)c2)=O)ccccc1Cl 94041,C1(NC(c2nn(CC)c(O)c2)=O)CN(C(=O)Cc2cnccc2C)CC2(CC2)C1 94042,c1(OC)ccn2cc(C(=O)NC3(C)CN(C(=O)C4=CCCCC4)C3)nc2c1 94043,n1(CCC)cccc1C(N1CC(COC)(NC(=O)C(O)CN(C)C)C1)=O 94044,C12(C(=O)NC(c3n(C)ncc3)CO)CCCC1CN(C(C1CCCC1)=O)C2 94045,C1(CC(=O)NCC#CCNC(C2CCN(CC(C)C)C2)=O)COC(C)(C)CO1 94046,C(C)(c1ccccc1F)=CC(=O)NC1CCN(C(c2nccc(CC)c2)=O)C1C 94047,c1(NC(C(c2ccc(CC)cn2)N(C)CC2C(=O)ON=C2C)=O)ccc(Br)cc1C 94048,C1(CNC(CN2CC(CC)C2)=O)(CNC(=O)CSC(C)C)CCCC1 94049,C1(CNC(C(C)(Cl)Cl)=O)CCCCN(C(=O)CC2CCC(=O)N2)CC1 94050,c1(C(=O)NC(CCC)CO)n[nH]c2cc(Cl)c(-c3ccc(C(C)=O)cc3C)cc12 94051,N1(C(C(C)(C2CC2)OC)=O)CCC2(CCCCC2NC(=O)C(C)C2CC2)C1 94052,C12(CC(=O)N(C)CCN(C(=O)C=CC3COC(C)(C)O3)C)CCCCC1C2(F)F 94053,N1(C(C=Cc2n(C)cnc2)=O)CCOCC(C(=O)Nc2ccc(Cl)nc2)C1 94054,c1(C(=O)N(c2ccnc(Br)n2)CCSC2CCCN2)ccc(Cl)cc1 94055,C(c1ccc(Br)o1)=C(C)C(=O)NCC1CC1CNC(c1ccc(=N)[nH]n1)=O 94056,N1(C(c2cn(CCC)nc2)=O)CCN(C(=O)CN(C(=O)C(C)C)C)C2COCC12 94057,C1(C)CCC(=O)N1.c1(SC)ccsc1C(=O)NCCCOCCOCCO 94058,C1(CC)CN(C(=O)CN(C)C)CCC1NC(=O)C(c1cccc(C)c1)(F)F 94059,CCC(C(=O)NC1CC(CO)N(C(C2CNC(=O)N2C)=O)C1)C(C)C 94060,N#CC1(c2ccccn2)CCCC2(CC1)OCCO2 94061,c1(-c2cn(C(CN(C(C(C3CCC3)OC)=O)C3CC3)C)nn2)cn2ccccc2n1 94062,CC(C)CC(CNC(c1cnn(C(C)C)c1)=O)C(=O)NC1CCSCC1 94063,N1(CC)C2CCC1CN(C(C1CCC(CNC(C3CCC(C)(O)CC3)=O)O1)=O)C2 94064,Cc1cccc(C2(F)CCN(C(c3ccc(C(F)(F)C(F)(F)F)cc3)=O)C2)c1 94065,C1(CC)CC(CC(N2CCC(CN(C)C(c3ccc(CO)nc3)=O)C2)=O)CCO1 94066,Cc1cc(Cl)ccc1OCC(=O)NCCC1=CCN(C(C2CCC(C)O2)=O)CC1 94067,c1(NCCC(=O)NC(CNC(CC2(CC=C)CCCC2)=O)C)ccccc1CC 94068,C1(C(=O)NC(C)(C)C(N2CCOCC(O)C2)=O)CC(=O)CC12CCC2 94069,c1(C(N2CC(O)(CNC(CC3C(C)(C)C3)=O)C2)=O)nc(F)ccc1Cl 94070,CC1C(C)N(C(c2ccc[n+]([O-])c2)=O)CCN1C(c1cncc(N)n1)=O 94071,c1(C(=O)NCCc2c(C)n[nH]c2)cn(C)nc1OC(F)F.c12ccccc1N2 94072,C(=O)(C(CCC1CC1)NC(C1CCCN1C1CC1)=O)NCC(C)CC1CCCC1 94073,CC(C(=O)N1CCC(OC2CCCCC2)C1)S(C)(=O)=O 94074,C1(F)(CNC(CC)=O)CCC(CNC(C2CCC(C3CC3)C2)=O)CC1 94075,CC1CN(C(c2cncn2-c2ccccc2)=O)CC1NC(=O)C(F)=C1CCCC1 94076,CCCCCCCCCCN(CCC)Cc1csc(C)n1 94077,N1(Cc2cccc(C(N)=O)c2)CCCC2(C1)CN(c1ncnc3n[nH]c(Br)c13)C2 94078,c1(C(N2CCC3(C(C(=O)NCCCCCO)C3)C2)=O)cccc2[nH]ccc12 94079,C(=O)(C(COC(C)(C)C)OC)NC(C=CC(=O)NCC#C)C 94080,c1(C(N(CCC)CCNC(=O)CC2CC=CC2)=O)coc2c(OC)cccc12 94081,c1(NC(C2C(NC(Cc3cn(CC)nc3)=O)CC2O)=O)ccc(C)cc1COC 94082,Cc1ncc(N)cc1C(=O)NC12CC(NC(=O)CNC(c3cccnc3)=O)(C1)C2 94083,c1(C(N2CCCC2C)C(=O)NCCCSC)cc(C(F)(F)F)ccc1C 94084,N1(C(c2c(C)c(C(N)=O)ccc2)=O)CC2CC(NC(c3n[nH]cc3Cl)=O)C(C2)C1 94085,c1(CC(=O)N(C(c2ccccc2)C(=O)NCC(C)(C)N(C)C)C2CC2)cnn(C)c1 94086,c1(-n2c(-c3cccnc3C)nc(C(C)OC)n2)ccc(C)c(F)c1 94087,c1(C2C(C(=O)OCC)C2C(C)C)ccc([N+](=O)[O-])c(N)c1 94088,Cc1cnccc1CN1CCC(NC(=O)Nc2ccccc2Br)CC1 94089,C1(C(N2CCC(CC(C)NC(=O)C3CC3)CC2)=O)CCCCC1(C)C 94090,Fc1cc(-c2ccc(CNCC3CC4(CCC4)CO3)s2)cc(F)c1F 94091,Oc1ncccc1NCCCN(c1ccccc1)CCC1CC1C1CC1 94092,Cc1cc(C(=O)NCCOCCNC(c2c(C)cccc2C)=O)c(N)c(Cl)c1 94093,Cc1cccc(CC(=O)NCCC2(NC(C3CCCC3C(N)=O)=O)CCC2)c1 94094,c1(NC(C)=O)cccc(C(N2CC(C(C)NC(=O)C(C)c3ccsn3)C2)=O)n1 94095,Cc1cc(N2CCC(C(N3CC(CNC(=O)C(C)C(C)O)C3)=O)C2=O)ccc1F 94096,c1(N(C)C)ncc(C(=O)NC2(CCCN(C(C3CNC(=O)C3)=O)CCO)CC2)cc1Cl 94097,c1(SCN(C(CCC)C)C)ccc(C)c(C)c1F 94098,N1(C(CC2(OCC)CCC2)=O)CCCCC1C(C)NC(C1CC(N=[N+]=[N-])C1)=O 94099,Cc1oc(C(=O)NC2C3CN(C(c4cnco4)=O)CC23)cc1S(C)(=O)=O 94100,N1(C(c2c(Cl)ccc(OC)c2N)=O)Cc2nc(C)nc(O)c2C1 94101,n1(CC(=O)NC(CNC(C2(OC)CCCOC2)=O)(C)C(C)C)ncc(O)nc1=O 94102,c1(C(N(C2CN(C(C3CC(O)C3)=O)C2)C)=O)sc(Cl)cc1Br 94103,S(=O)(=O)(c1ccc(NCCN2CCNC(=O)C2)c(Cl)c1)N(C)CC1N(C)CCOC1 94104,C=C1CCN(C(c2ccc(F)cn2)=O)C(C(=O)NCCN(CCO)CC)C1 94105,c1(C(N2CCC(OCCNC(C3CCC3)=O)C2)=O)cnc(C2CC2)nc1 94106,C1(NC(CCn2ccc(C)n2)=O)CC(O)CN(C(c2occc2C2CC2)=O)C1 94107,n1(CC)nc(C)c(C(=O)N(C)CC2CC(F)CN2C(=O)CC(C)C2CC2)c1Cl 94108,N1(C(c2csc(Br)c2)=O)CCCN(CC(=O)Nc2ccc(OC)cc2)CC1 94109,C1(C2CN(C(c3cnc(C(F)(F)F)cn3)=O)C2)(NC(C(C)c2ccco2)=O)CC1 94110,c1(CN(C)C)ccc(C(=O)N(C2CN(C(=O)CC3CC3C3CC3)C2)C)cc1 94111,N1(C(COc2ccc(C#C)cc2)=O)CC(C)CN(C(C2(C)CC=CC2)=O)CC1C 94112,C1(OC)CC(CNC(c2cc(F)n(C)n2)=O)N(C(c2ccc(C#N)o2)=O)C1 94113,C(=O)(CCS(=O)(=O)C(F)(F)F)NC1C(NC(CC(C)(C)C#N)=O)COC1 94114,C1(CC=C)(C(=O)NCCCOCCSC)CCCN1C(c1n[nH]cc1C)=O 94115,CC1(C(=O)NCC2(NC(C3CCS3(=O)=O)=O)CCCC2)CCC(O)CC1 94116,C1(NC(C(COCC)C)=O)CN(C(c2cc(C)c(Br)o2)=O)CC1SC 94117,CC1(C)CC(C(=O)NCC2CN(C(=O)CCC3CCC3)C(C)(C)C2)CNC1=O 94118,N1(C(CCSCC)=O)CC(NC(C2Cc3nnc(C)n3C2)=O)CC12CCOCC2 94119,C1(CC(=O)OCC)CN(Cc2cnn(Cc3ccccc3)c2C)CC2(CCC2)O1 94120,C1(OC)CC(CNC(c2nncn2C(C)C)=O)N(C(=O)C(C)OC2CCCC2)C1 94121,C(CCCCC(=O)NCC12CCCC(CO1)C2)N(C(=O)CCCCO)C 94122,C1(C(=O)NC(CCC)C(=O)NCC)CCN(C(=O)OC(C)(C)C)C12CC2 94123,C1(F)(CNC(C(C=C)O)=O)CCCN(C(c2ccc(C)cc2Br)=O)C1 94124,Cc1ccc(C(C)CC(=O)NC2CC(CNC(=O)C(C)(C)n3cccn3)C2)cc1 94125,N1(C(C(C=C)(C)C)=O)CCC2(CCCCC2NC(c2cn(CCO)nc2C)=O)C1 94126,N1(C(C(=O)NCCS(=O)(=O)NC)CCSNC2CC2)CCOCC(C(C)(C)C)C1 94127,c1(N(C)Cc2ccnc(-c3ncc[nH]3)c2)cncc(NCc2csc(Br)c2)n1 94128,c1(C(N2CCCCC2C2CCCCC2)C(=O)NCCC)nn(CC)cc1Cl 94129,N1(C(c2c(CC)cco2)=O)CC(CNC(C2CC2C)=O)OC(C)(C)C1 94130,C1(=O)CC(C)CCC=C(C)CN1.c1(OC)ccc(C(N2CC3C(C2)C3(F)F)=O)c(O)c1 94131,c1(OC)ccc(C(=O)NC23CC(NC(C4CC45CCOC5)=O)(C2)C3)cc1O 94132,C1(CN(C(=O)CCCNC(N)=O)C)CCN(C(=O)CCc2cn(C)cn2)CC1 94133,c1(CC2CCN(C(=O)C(C)CSC)C2)ccccc1C(N(C(CSCC)=O)C)=O 94134,C[Si]1(C)CCCCN(C(=O)C(Cc2ccco2)NC(=O)CCCF)C1 94135,c1(CNC(c2cnc(C)s2)=O)cccc(NC(c2csc(Cl)c2Cl)=O)c1 94136,c1(C(=O)NCCC(C)NC(C2OCC2(C)C)=O)cc(C2CC2)oc1C1CC1 94137,CCCCC(CC)CC(=O)NC1CCC(C(=O)NCC2(OC)CC2)C1 94138,N1(C(c2c(C)n(C(C)C)nc2)=O)CCN(C(c2ncc(N)cc2Cl)=O)CC1C 94139,c1(SCC(N2CCC(CC=C)(NC(=O)CC3(C)CC3)C2)=O)ccc2c(c1)CCC2 94140,C1(C(N2CCC2(C)C)=O)(OC)CCN(C(C2CCC(=O)O2)=O)C1 94141,c1(C(C)C)ccc(C(C)NC2CCOC2C)cc1 94142,C(=O)(C(C)(CC)CC)NC(C(=O)NCCCCOCC)CCC1CCC1 94143,C1(CC(=O)N(C(C(C)C)C)C)C=CC(NC(=O)C=CC2CCCC2)C1 94144,C1(CC(=O)NC(C)(C)CNC(=O)CNC=O)CC(C)(C)CN1C(C1CCCC1)=O 94145,N1(C(C2N(C(c3c[nH]c(=O)cn3)=O)CC23CCCC3)=O)CCCC(C2CC2)CC1 94146,c1(C(N2C(CNC(C3=C(C)CCC3)=O)CCC2)=O)cc(Cl)c2ccccc2n1 94147,C(CS(=O)c1ccccc1)NCC1(OCC)CCC(O)CC1 94148,n1(CCC)ncc(C(N2CCOC(C(C)NC(=O)CCn3ccnc3)C2)=O)c1C 94149,c1(C(=O)NCCCN(C(C2(COC)CCCO2)=O)CC)ccc2n[nH]cc2c1 94150,C1(NC(CCCC)=O)CCN(c2ncncc2C)CC1OCc1ccccc1 94151,c1(C(N2CCCC(C)(NC(CC(CC)C)=O)C2)=O)cc(F)cc2c1CCC2 94152,CCC(CC(C)C)C(=O)NC1(C)CC(NC(C2CCOC2C(F)(F)F)=O)C1 94153,N1(C(C2C(OC)C2)=O)CCN(C(=O)Cc2csc(Br)n2)CC(O)C1 94154,N1(c2c(OC)ccc(Br)n2)Cc2c[nH]nc2C(C)(C)C1 94155,Cc1cc(C(=O)NC2CC3CC2N(C(c2oc(Br)nc2C)=O)C3)nc(C)c1 94156,CCC(C)(CCC(C)C)C(=O)N1CC2OCCN(C(=O)C=CC(C)(C)C)C2C1 94157,c1(C(=O)NCC(CNC(c2cnc(OCC)s2)=O)F)cc(=O)c(OC)c[nH]1 94158,c1(COC)cc(CN2CCOCC2C#N)ccc1OC 94159,C1(CNC(=O)C=CCc2cnc[nH]2)C=CC(NC(c2cnc(C3CCC3)s2)=O)C1 94160,N1(C(CCN(CC)CC)=O)CCC2(NC(=O)CCOCC(C)(C)C)CCCCC12 94161,C1(C(=O)OC)(OC(C)=O)CCN(C(=O)C(C)(C)Br)CC1.N12CC(C1)C2=O 94162,c1(-n2c(Cc3cnc[nH]3)nc(C(c3ccccc3)OC)n2)cc(C(F)(F)F)ccc1C 94163,CC(C)(CCCC(=O)N1CC2(CCCCC2)C1)NC(=O)Cn1cccn1 94164,C1(CNC(c2nc(-c3ccc(Br)cc3)ns2)=O)CCCN(c2ncccn2)C1 94165,c1(C(N(C)CC2N(C(CC=C)=O)CCOC2)=O)cnn2c1CCC2 94166,CCC(C#N)(CC)C(=O)NCC(N1CCN(C(c2cc(C)ncc2C)=O)CC1)C 94167,c1(CCCC(=O)NCCNC(C2COCCO2)=O)c[nH]c2ccccc12 94168,C1(C(=O)NCc2cc(OC)ns2)CN(C(=O)C=CC2CCCC2)CCN1C 94169,N1(CC)CC(C(N2CCC(C(C)NC(=O)C(C)(F)F)CC2)=O)CCC1=O 94170,c1(C(N(C)CC2(O)CCN(C(c3cnn(C)c3)=O)C2)=O)ccc(F)c(O)c1F 94171,c1(-n2ncc(C(=O)NCC(CNC(CNC=O)=O)CO)c2)ccc(F)cc1 94172,c1(NC(=O)C(=O)NC2(NC(CC(C)C)=O)CC2)ccc(C#N)c(Cl)c1 94173,N1(C(c2cc(C)oc2)=O)CCC(NCCc2cnn(C)c2)C(C)C1 94174,c1(-n2cc(CN(C(CC(C(CC)(C)C)C)=O)C)nn2)ccc2c(c1)OCCCO2 94175,C(=O)(C1=CCN(C(C2(C#N)CC(=O)C2)=O)C1)NC1CCC(C)(C)C1 94176,C1(N(C(c2c(C)occ2)=O)C)CCCC2CN(C(c3ccc(=O)n(C)c3)=O)CC12 94177,C1(NC(COCC#C)=O)CC2CN(C(=O)C(C)CC3CCCC3)CC2C1 94178,C1(C(=O)OC)CCN(C(=O)CSc2cc(Cl)ncc2OC)CCC1(F)F 94179,c1(CN2CC(CNC(c3cocn3)=O)C2)cccnc1O 94180,C12(OC(C)=O)CC(C(C3(C(N4CCC4)=O)CC3)=O)(C1)C2.c1(OC)ccccc1 94181,O=C1CCc2cc(C(=O)NCCC3(NC(=O)CCC(F)(F)F)CC3)ccc2N1 94182,c1(C(N(C(C)CNC(c2cccc(Cl)c2OC)=O)CC)=O)cc(Cl)cc(C)c1N 94183,c1(C(N(C(=O)C(C)c2nccs2)CC)C2CC2)cccc(Br)c1 94184,N1(CCCNC(N2CC=CC2CO)=O)CCOCC1 94185,Cc1ncsc1CCC(=O)NC1CC(CCNC(C2(CO)CCC2)=O)C1 94186,C(CCC(O)C(=O)NCCOc1ccccc1)NC(Cn1nc(C)oc1=O)=O 94187,CC(C)S(=O)(=O)CC(=O)NC1CN(C(c2ccc(OC(C)C)cc2Cl)=O)C1 94188,C1(CNC(Cc2c(OC)nccc2)=O)CC2(CC(NC(=O)C(C)S)C2)C1 94189,C1(C)C(=O)NNC(=O)Nc2ccc1cc2.c1(OC(C)=O)ccc(OC(F)F)cc1 94190,O(N=C1CCCCCC1)CC(=O)NCCC1(NC(CCCCCOC)=O)CC1 94191,N1(C(C23CC(COC)(OC2)C3)=O)CCC(C(=O)NC2CCCCNC2=O)C(O)C1 94192,N1(C(c2ccc(C(C)=O)cc2)=O)C2CCC1CC(NC(c1cc(Cl)cnn1)=O)C2 94193,C1(NC(C2CC(OC)C2)=O)CCCC2CN(C(=O)CCn3c(C)csc3=O)CC12 94194,c1(C(=O)NCC2(O)CN(C(=O)CC3CCC(O)C3)C2)cnc2c(c1)COCC2 94195,C(=O)(CCCCC(C)(C)OC)NC(CC(=C)C)C(=O)N(C1CC1(C)C)C 94196,C1(NC(c2cc(CC)ncc2)=O)CC2(CCCCN2C(C2CC=C(C)CC2)=O)C1 94197,C1(NC(=O)CN2CCOCC2=O)CC2(C1)CN(C(=O)CN1CCCS1(=O)=O)C2 94198,Cn1ncc2c(NCC3COCC4(CCC4)O3)[nH]c(=NCC3(S(C)=O)CC3)nc12 94199,C12(c3cc(CN(CCCCCCCC)CCC(N)=O)[nH]n3)CC3CC(CC(C3)C1)C2 94200,c1(CCNC(N2CC(C)C(N(C)C)C2)=O)cc(N)ccc1Cl 94201,N1(C(c2cc(OC)ns2)=O)CC2CCC(NC(C3CCc4cnnn4C3)=O)C2C1 94202,c1(C(=O)NCC2C(C)CCN2C(C2CC3(C2)CC3(F)F)=O)cc(N)c(N)cc1F 94203,C1(CC(=O)NCCC(=C)CNC(C2(C(C)C)CNC(=O)C2)=O)CCCC(C#N)C1 94204,c1(CNc2cc(C(F)(F)F)c(Cl)cc2)cccc2sccc12 94205,c1(C(=O)NC(CCCC)CNC(=O)C(COC)CC)cccn2ncnc12 94206,CCCCCCCC(=O)NCC(C)=CC(=O)Nc1ccc(C(C)C)nc1 94207,c1(N2CCC(CC(=O)N(C)C)CC2)nnc(C2CCc3c[nH]nc32)n1CC1CC1 94208,c1(CNC(C(c2cnn(C)c2)NC(CCCCNC(C)=O)=O)=O)cc(C)cnc1F 94209,C(CC(O)C(F)(F)F)NC(C=CCN(C(CCCOCC=C)=O)C)=O 94210,C1(C)(CNC(C(C)SC)=O)CCN(C(c2cncc(CO)c2)=O)C1.C(N)=O 94211,CC(=O)C(C)CC(C)C(=O)N1CCC(C(=O)NCCCNC(=O)C(C)C)C1C 94212,C1(C2(OCC)CCC2)(NC(CCC2CCCN(C(C(CCC)=CC)=O)C2)=O)CC1 94213,N1(C(C)C(=O)NCC(c2ccccc2)NC(=O)CC2CC2)CCC(O)CC1 94214,c1(C(=O)NC2CCN(C(=O)C(F)CC3CC3)CC2O)ccc2cccnc2n1 94215,N1(C(=O)OC(C)(C)C)CCCC1CNC(C1CC(N2CCCC2)C1)=O 94216,c1(C(N(CC(C)NC(=O)CCc2ccc(F)c(F)c2)C)=O)ccc(Cl)c(F)c1 94217,c1(C(N2C(C(C)NC(=O)C(C)(C)N(C)C)CCC2)=O)cnc2[nH]c(O)nc2c1 94218,N1(C(COC)=O)CC(NC(c2sc3cccc(F)c3c2C)=O)CC12CCOCC2 94219,c1(OC)ccc(C(F)(F)F)cc1NC(=O)C(=O)NCC1CC(=O)C12CC2 94220,c1(OC)cc(NC2CCC(NC(=O)CSC)CC2)ncn1 94221,C1(C(N(CCF)CC)=O)CC(NC(C2CC(F)(CF)C2)=O)CCO1 94222,n1(CCN(C)C)nccc1C(=O)NCC=CCNC(c1cc(CF)on1)=O 94223,C(C(O)CC(C)(C)C)NC(C1CC(C)(NC(c2n(CC)nnc2)=O)C1)=O 94224,c1(CN(C)CC2N(C(c3c(C)snc3)=O)CCC2)cnn(C)c1Cl 94225,C(=O)(CC(C)C(C)C(C)C)NC(CC)(CC)CCNC(c1cn(C)ccc1=O)=O 94226,C=CCCC(O)CNC(C12CC1CCN2C(c1ccsc1OC)=O)=O 94227,C(CCCCC(=O)NC1(CF)CCN(C(=O)CC(=O)OCCC(C)C)C1)SC 94228,c1(OC(CC)C)cc(NC(N2CCC(CSC)CC2)=O)ccc1OC 94229,Cc1ccc(S(=O)(=O)CC(=O)N2CCCC(O)CC2)cc1C 94230,CC1CCN(c2cncc(C(N3CCC(C)(NC(c4cnn[nH]4)=O)C3)=O)c2)CC1 94231,N1(C(CC(C=C)C)=O)CC2CC(C1)N(C(=O)CSCc1ccc(F)cc1)C2 94232,N1(C(C2C(OC)CN(C(CCOCC#C)=O)C2)=O)CCCC(C)(F)C1 94233,C(C(COC)C(=O)NC1CCC1C(=O)N(C)CC1CC1(C)C)OC 94234,CC(C)C#CC(=O)NC1CCC(N(C(=O)CC2CCCO2)C)CC1 94235,C(=O)(C(C)(C)C(=O)N1CCC(C)C(NC(c2c[nH]cc2C(F)(F)F)=O)C1)OCC 94236,N1(C(CN(C(=O)OC)C)=O)CCC(C(C)NC(C2CC2C(C)O)=O)CC1 94237,C12(CCC)CCN(CC1)C2=O.C1(=O)CCCN1.C1(COCC)(SC)CCC1 94238,C=CCCCC(=O)N1CCC(N(C(=O)C(C)Cc2cnn(C)c2)C)C1 94239,N1(C(C2C3CCN(C(C(C)(C)O)=O)CC32)=O)CC(C)(C)OC(C)(C)C1 94240,C(=O)(CCC1=NNC(=O)CC1)N1CC2(OCC(NC(C(CCC#C)O)=O)C2)C1 94241,c1(OC)cccc(CCC(=O)NCC(C)CNC(=O)C(C)(C)c2cncnc2)n1 94242,CCCC(CC)C(=O)N(C)CC1CCCN(C(c2ccnc(O)c2)=O)C1 94243,C#Cc1ccc(C(=O)NCC2CCCN2C(=O)C(C)CN2CCOCC2)cc1F 94244,CC1CNC(=O)CC(N2CCOC(c3ccc(Cl)c(Cl)c3)C2)C1 94245,c1(C(=O)NCC(CNC(CN2CCCC(CC)C2)=O)(C)C)cccc2c1CCN2 94246,C1(NC(C(CO)NC(=O)CC2(c3ccon3)CC2)=O)CCCC(CNC(N)=O)C1 94247,Cc1cc(C(=O)NCC2CC2NC(=O)CN2CCCNC2=O)cc([N+](=O)[O-])c1O 94248,C(=O)(C(O)CCC(C)C)N1C(CNC(C=CC(C)(C)SC)=O)COCC1 94249,Cc1ccc(CSCC(N2CC(NC(C3CCCC3(C)C)=O)C(C)C2)=O)cc1 94250,C1(OC)CCC2(C(N3CC(NC(=O)C(C)OCC4CC4)C(C)C3)=O)CC12 94251,C12(NC(c3cncc(OC)c3)=O)CCCN(C(=O)Cc3ccsc3)CC1C2 94252,c1(C(=O)NCCCN(C(=O)CC2CC=CCC2)C(C)C)ccc(Cl)c(N)c1 94253,N1(C(c2ccc(SC)cc2)=O)CC2CC1CCN2C(=O)C=Cc1nc(C)cs1 94254,C#Cc1cncc(C(=O)NC(C)C(c2c(F)cccc2F)O)c1 94255,C(c1ccc(F)cc1)=CC(N1CC2CN(C(C3CCCS3(=O)=O)=O)C2C1)=O 94256,N1(C(C(c2ccn(C)n2)NC(C(c2cc(CO)[nH]n2)C)=O)=O)CC2CCOC2C1 94257,C(=O)(C1=C(C#N)CCC1)N1CCC(C=C)(C(=O)NCC(C)N(C)C)C1 94258,C(=O)(C(C)(C)CC(F)(F)F)NCC1N(C(CCCc2n(C)cnn2)=O)CC1 94259,c1(C2C(C(=O)NC3(CNC(=O)Cc4cnoc4)CCC3)C2)ncnc2ccsc12 94260,Cc1cc(F)cc(C(=O)NC2CCC(NC(=O)C(C)c3ccsc3)CC2)c1C 94261,Cc1cc(F)c(NC(=O)NCC2CCCN(C)C2)cc1Cl 94262,CC(C)(O)CCNC(=O)NCCCC1CCN(Cc2ccccc2)C1 94263,N1(C(c2nc(C)sc2)=O)CCCC(C)(C(=O)Nc2c(Cl)cnnc2Cl)C1 94264,N1(C(C(F)OC)=O)CC2CC1C2NC(c1ccnc(C)c1)=O 94265,C1(C)(CNC(C=NOC)=O)CN(C(=O)COC2CC=CC2)C(C)(C)C1 94266,C1(CN(C(CC(=O)NCC)=O)C)CN(C(=O)C(C)(CC2CCC2)OC)CC12CC2 94267,N1(C(C2(OC)CS(=O)(=O)C2)=O)CC(NC(c2ccccc2)=O)CCC1C 94268,C1(C)(C(=O)NC(C2N(C(c3c(C)snn3)=O)CCC2)C)CCN(C)C1=O 94269,C#Cc1ccc(NC(=O)CC2(c3ccc(OC)cc3)CCC2)cn1 94270,C(C(C)(C)C(=O)NC(c1ccccc1F)CNC(C1CCCO1)=O)N(C)C 94271,S(=O)(=O)(c1ccccc1C(C)C)N1CCC(C2N(c3nccc(C)n3)CCC2)C1 94272,C1(NC(c2c(C)cc(F)s2)=O)CC2CCC(C1C)N2C(c1ccc(CF)cc1)=O 94273,C1(CC(=O)N(CCCNC(=O)C(O)Cc2cnc[nH]2)CCC)CCCCC(=O)N1 94274,C1(NC(CCC(C)=O)=O)CCN(C(c2ccc(C(F)(F)F)nn2)=O)C(C)C1 94275,c1(CC)cc(F)ccc1C(=O)NC1CC2C1CCN2C(c1coc(N(C)C)n1)=O 94276,C12(CNC(C(COC)(F)F)=O)CCCC1N(C(c1c[nH]c(Br)c1)=O)CC2 94277,C#CCC(CC(F)F)C(=O)NCc1ccc(CCNC(=O)CCCOCC)cc1 94278,c1(C(=O)NCC(CC(C)C)NC(=O)C(F)CC2CC2)cccc([N+](=O)[O-])c1 94279,C1(N(C(C(C)C)=O)C)CCCC(NC(c2nnn(C)c2C(F)(F)F)=O)C1 94280,c1(CC(=O)NC(C)(C)CN(C)Cc2ccnc(SC)n2)c[nH]c2ccccc12 94281,CC1CCCN(C(=O)OC(C)(C)C)C1C(=O)Oc1nnc(-c2cccc(Cl)c2)s1 94282,c1(CNCC(CC(C)C)CCO)nc2ccccc2c2ccccc12 94283,c1(C(N(CCC(C)NC(c2cnc(OC)s2)=O)C)=O)cccc2c1CCO2 94284,c1(C(=O)NCCC(C)(C)NC(C=CC=CCC)=O)c(C)oc2nc(Cl)ccc12 94285,c1(C(=O)NCC2C(C)CN(C(=O)Cc3cccc(Cl)c3)C2)ccnc2[nH]cnc12 94286,N1(C(CCCC)=O)CC(NC(=O)C(C)NC(c2ccc(C)s2)=O)C(C)C1 94287,C1(OC)(NC(N2CCC(COCc3ccccc3)CC2)=O)CC(O)C12CCC2 94288,N1(C(Cn2c(C)cc(C)n2)=O)CCCN(C(c2cn(C(F)F)cn2)=O)C(CO)C1 94289,C1(C(N2CC(c3onc(C)n3)C2)=O)CCN(C(c2sccc2C)=O)CC1O 94290,c1(C(=O)NCCC2CCCN(C(=O)C=CCO)C2)cccc2c1CCCC2=O 94291,c1(C(C)NC(C2(F)CN(C(C(C)SC)=O)C2)=O)cncc(F)c1 94292,C(=O)(C1=COCCC1)NCCC(C)O.C12CCC1C(=O)N2 94293,C1(C(=O)NC(c2ccncc2)(C)C)CC(NC(C2CCCC(=O)N2)=O)CCO1 94294,c1(N(CCC(O)C(C)(C)C)C)nc(=N)[nH]c(=NC2CC2c2cnn(C)c2)[nH]1 94295,CC1(C)CCOC1CC(N1C(CNC(C2OCCC2(C)C)=O)CC2CC12)=O 94296,C(=O)(C1=CC2CCCCC12)NC(c1ccccc1)CNC(C(=C(C)C1CC1)F)=O 94297,c1(OC)cnc(Cl)[nH]c1=NC1CCC2CN(C(=O)C(C)n3cnnn3)CC12 94298,C1(NC(c2nc(COC)oc2)=O)CCC(NC(C2CC2(F)Cl)=O)CC1 94299,c1(C(=O)NC2CC2NC(C2CC(=O)N(C3CCCC3)C2)=O)csc2c1CCCC2 94300,c1(N2CC(C(=O)NC)OCC2)nc2c(c(=NCCC3CC3)[nH]1)CCC2 94301,N1(C(C(C(CC)C)OC)=O)CCC(N=c2nc(C(F)(F)F)[nH]s2)C2(CCC2)C1 94302,CC#CCC(C(=O)NCCC(C)CC)NC(=O)C(=O)N(C)C 94303,N1(C(CNS(CC)(=O)=O)=O)CCCC(CCNC(C2CCCO2)=O)CC1 94304,c1(C(=O)NC2CCCCN(C(c3cc[nH]c3)=O)C2)ccc2cccc(Br)c2n1 94305,c1(OC)nc(C)ccc1C(N1CC(NC(=O)Cc2nnc(C)o2)C(C#N)C1)=O 94306,Cn1cnc2c[nH]c(=NC3CC(F)CN(c4ncnc5n[nH]cc45)C3)nc12 94307,N1(C(C2(c3cc(C)no3)CC2)=O)CC2CN(C(C3CCCCC(=O)N3)=O)CCC12 94308,C(=O)(CCCCCCC(C)C)NCC1(F)CC(NC(c2c(C)n[nH]c2)=O)C1 94309,N1(C(c2c(C#C)cn(C)n2)=O)CCCC2(C1)C(NC(c1ccsc1)=O)CCN2C 94310,C1(CC)CCCN(C(=O)CC(C)C2CC2)C1C(=O)NC1CN(C)C(C)(C)C1 94311,c1(COC(N(CCCOc2cccnc2)C)=O)cccc(N)c1Br 94312,CC(C)S(=O)(=O)c1c(C(=O)NCC2CC3(CCN2)CCOCC3)cccc1Cl 94313,CCC1=C(C(=O)NCC2CN(C(=O)C(C)c3ccco3)CCO2)CCCO1 94314,Cc1cc(SCC(=O)NCC(C)(CO)NC(C2CC(C)CCO2)=O)cc(C)c1 94315,C1(S(N)(=O)=O)(C(=O)NCCCN(C(c2cccc(F)c2SC)=O)CC)CCC1 94316,c1(C(N2CCC(n3cc(-c4c(C)nn(C)c4Cl)nn3)C2)=O)cc(S(N)(=O)=O)co1 94317,C(=O)(C(C)CCCOC)N(CC(=O)NC(CCN(CC)CC)C)C 94318,c1(C(=O)NC(CC)(C)CNC(c2ccc(C(F)F)o2)=O)c(C)cc(C#N)cc1C 94319,n1(CC)nc(C)c(C(=O)NC(CNC(c2sccc2C)=O)CO)c1C(F)F 94320,c1(OC)cc[n+]([O-])c(C(=O)NCC(C(C)C)NC(C2CNC(=O)C(C)(C)C2)=O)c1 94321,c1(NC(=O)C(=O)N(C)Cc2cscc2Br)ccc(CCNCC(=O)N(C)C)cc1 94322,C1(C(=O)NCC2CN(C(Cn3nc(C)oc3=O)=O)C2)Cc2ccccc2C(=O)O1 94323,[N-]=[N+]=NC1CC(C(=O)NCCc2cscn2)N(C(=O)C#CC2CCOC2)C1 94324,N1(C(=O)NC(C)Cc2c(Cl)cccc2Cl)CC(=O)N(C)CC1C(C)C 94325,CC1CN(C(C2CN(C(=O)CCC3(C#N)CCC3)CCO2)=O)Cc2c[nH]nc21 94326,c1(C(=O)NC(C(C)C)Cc2ccc(F)cc2)ccc(N2CCCC2=O)c(Cl)c1 94327,Cc1ccc(C(=O)NC(CCC2CC2)C(N2CCCC(C)(F)C2)=O)c(C)c1 94328,CC1(C(=O)NCC2OCCC2C(=O)NCCOCC2CCC2)CC(C#N)C1 94329,Cc1cccc(Br)c1C(C(=O)N(CC(C)C(C)(C)C)C)NC(c1c[nH]c(=N)o1)=O 94330,C=CC(CC)CC(=O)NC12CC(C1)N(C(=O)C(C1CC1)OC)C2 94331,C=CCCCCCC(C)(c1nnnn1CC=C)NC(C)CCC(=O)OC 94332,C(C)(C)(CN=c1[nH]c2ccccc2s1)C1N(C(C2(COC)CC2(F)F)=O)CCCC1 94333,C1(C(=O)NC(C)CCNC(c2cncc(Cl)c2)=O)Cc2nn(C)cc2C(=O)N1 94334,C12(C(=O)NCC3N(C(C(N4CCC(C)C4)=O)=O)CCN(C)C3)CC(C)(C1)OC2(C)C 94335,CCC1=NOC(C(N2CC(F)(C(=O)NC(C(C)C)c3nc[nH]n3)C2)=O)C1 94336,C1(CNC(CCCOCC)=O)CCCC2(CN(C(=O)C(c3cnn(C)c3)=O)C2)O1 94337,Cc1ccc(CO)c(NC(=O)CC2(O)CN(C(C3CC(C(C)C)C3)=O)C2)c1 94338,CN1CCOC(C(=O)NCC2CCCCN2C(C2(O)COC2)=O)C1=O 94339,C1(CNC(C2C(C)OCC2)=O)CN(C(C2(C3CCC3)CC2)=O)CCN1C 94340,Cc1csc(C(N2CCCC(C(C)NC(C34CC(CCO3)C4)=O)C2)=O)c1C 94341,C1(C(N(CCCNC(C=CC=CCC)=O)C)=O)CCOC(C)C1 94342,c1(OC)ccc(C(C)(C)C(=O)N(O)Cc2cn(C(C)C(C)O)nn2)cc1OC 94343,C1(C(=O)NCC(N(C)C)C2CC2)CC2(CC2)CN1C(c1n[nH]c(O)n1)=O 94344,C1(CCC)CN(C(=O)CC(C)CC)CCN1C(=O)CN1CCC(C)CC1 94345,C1(CCC)(NC(=O)CCC2CC2C)CCN(C(C2CC3CCC3C2)=O)CC1 94346,c1cc(OC)c(O)c(OC)c1.C1(C(N(CC=C)CC=C)=O)CCN(N)CC1O 94347,N1(C(C2(CO)CCC2)=O)CCC(Cn2cc(-c3ccsc3)nn2)C(F)(F)C1 94348,CCCC(CC)C(=O)NC1(CO)CCCN(C(c2cc(C(C)C)cnc2C)=O)C1 94349,N1(C(c2cc(C)cc(Cl)n2)=O)CCCC2(CC(NC(c3cc(C#N)c[nH]3)=O)C2)C1 94350,C(=O)(CCC(F)(F)F)N(CC(C)NC(=O)C(C)CC1CC1)CC 94351,C1(CC(=O)NC(C(C)OC)(C)C)CCN(C(=O)C=CC(F)F)CC1 94352,C(=O)(CCCC(=O)OC)NCCCN(C(C(COC)OC)=O)CCO 94353,c1(CN)ccccc1-c1cn(CCC(=O)NC2CC3CC3C2)nn1 94354,C1(NC(c2cnc(C)nc2O)=O)CC2CC(C1)N(C(C1CN(C(N)=O)C1)=O)C2 94355,n1(CS(=O)(=O)NCC(c2ccc(OCC)cc2)(C)C)cccc(C)c1=O 94356,c1(C(=O)NC2C3CN(C(C(=C(C)C4CC4)F)=O)C(C3)CC2)cccn2ccnc12 94357,N1(C(C(C)(C)OC(=O)NCC)=O)CCC(C2CC2)(CNC(=O)C(C)S(N)(=O)=O)C1 94358,C1(C)(CNC(C(C)OCCC=C)=O)CCCN(C(c2cn(C(F)F)cn2)=O)C1 94359,O=C(C1CCCOc2ccccc21)NC1COCC1n1cc(-c2ccsc2)nn1 94360,c1(CNC(c2c(C)cnn2C)=O)ccc2c(c1)CCC2NC(=O)CSC(F)(F)F 94361,c1(C(=O)NC(C2(CNC(C3CC(SC)C3)=O)CC2)C)cc2ccncc2c(O)n1 94362,N1(C(CCSCCCC)=O)CC2CC2(NC(c2oncc2C)=O)C1 94363,C1(SC(C)C)CCN(CC2(CNCc3ccc(N(CC)CC)o3)CCOC2)CC1 94364,N1(C(c2nn(C)c(F)c2)=O)CCCCCC1CNC(C1C2CCCCC12)=O 94365,c1(C(N2C3(CNC(C(CC)F)=O)CC(C2)C3)=O)nc(C(C)C)ncc1Br 94366,C1(C(F)(F)F)CCC(F)(CNC23CC4CC2C3C4)C1 94367,c1(C(=O)NC2(c3ccccc3)CN(C(c3cnn(C4CC4)c3)=O)C2)n[nH]c(O)n1 94368,c1(C(=O)NC2CC3(C(NC(CN4C(C)CCC4)=O)C3)C2)ccnc2[nH]c(O)nc12 94369,n1(CC(N2CCCCCC(NC(C(C=C=C)C)=O)C2)=O)[nH]cc2c(=O)ncnc1-2 94370,C1(C(=O)NCCCCCNC(CC(C)OC)=O)CC(=O)N(c2cnn(C)c2)C1 94371,CCCCC(CC)C(=O)NCC(C)(C)NC(c1sccc1SC)=O 94372,Cc1cc(C(N2CCNC(C(=O)NCC3CC(=O)N(C)C3)C2)=O)cc(C#N)c1 94373,c1(C(=O)NC(CNC(C2CC(C(=O)OC)C2)=O)(C)C(C)C)sc2cncn2c1C 94374,c1(CNC(CC2CCN(CC(C)(C)C(=O)O)CC2)=O)ccc(F)c2[nH]ncc12 94375,c1(OC)ncc(Cl)c(NC2(CNC(=O)CCc3ccc(O)nc3)CCCC2)n1 94376,C1(CNC(C(CC)C)=O)CCCC12CCN(C(c1ccc(F)c(F)c1)=O)CC2 94377,c1(NC(C)=O)cccc(F)c1-c1cnc(F)c(C(N2CC3C(C2)C3(C)C)=O)c1 94378,c1(C(=O)NC(c2cccc(N)n2)C)cnc2n1CCOCC2 94379,C(=O)(C(C)(C)CC(F)(F)F)NCC(CNC(c1c(OC)n(C)nc1)=O)(C)C 94380,CCC(C)(O)C(=O)NC1C=CCN(C(c2cn(C)nc2C)=O)C1 94381,c1(CCCC(=O)N2CC(C(C)NC(c3cnsn3)=O)C2)ccc(O)cc1 94382,CCC(CC)C(F)C(=O)NC(CC1CCCC1)C(=O)N(C1CCC(F)(F)C1)C 94383,C1(C(=O)NC(CN(C(=O)CCCCSC)CC)C)COCCN1C 94384,C12(C(=O)NC3CC(CC(=O)NCCn4ccnn4)C3)CCCC1C2 94385,C1CN=C2NC3=C(C(=NC4CC(C4)S1)N2)SCC3.CN(C1COc2ccccc21)Cn1cccn1 94386,Cc1cc2ncc(C(=O)NC3CC(CCNC(=O)Cn4cc(Cl)cn4)C3)cc2[nH]1 94387,N1(C(CCC=C)=O)CCC(CF)(NC(c2cnn(C3CCCCC3)c2)=O)C1 94388,c1(CNC2(c3n(C)nnn3)CSCSC2)cc(Br)c(C#N)cc1F 94389,C1(CNC(=O)C(O)CN2CCOCC2)CCN(C(c2cc(CF)on2)=O)CC1 94390,N1(C(C(=O)NCCOC)=O)CCC(CF)(NC(=O)CCCC2CC2)C1 94391,c1(C(=O)Nc2ccc(CC(=O)OC)cc2I)cnc2c(c1)c(C)nn2C 94392,C(=O)C1C2CN(C2)C(=O)C2(CC2)CN1.C(C(=O)OCC)N(CCC)C.C1CC1 94393,C1(CNC(CC(CC)OC)=O)CC2COCC2N1c1nnc(CC(C)C)s1 94394,c1(C(CC)NC(=O)NCCCOCC)cccn1Cc1ccccc1 94395,c1(C(N2CCC(Cc3ccccn3)C2)C(=O)NC(C(=O)OC)C)cccc(CO)n1 94396,C1(NC(CN2C(C)CC2)=O)COC2(C1)CN(C(c1cnc(C3CC3)[nH]c1=N)=O)C2 94397,N1(C(CC2(CC)CC2)=O)CCCC1N(C(=O)C1CC1)Cc1nnc(O)o1 94398,c1(C(=O)NC(CNC(c2n(C)c(S)nn2)=O)CC(F)(F)F)nn(C)cc1[N+](=O)[O-] 94399,c1(OC)ncc(C(=O)NCCOCCN(C(=O)CCc2cccnc2)C)s1 94400,c1(C(=O)N(C2CC(C(=O)Nc3c(C)c(Br)cnc3)C2)C2CC2)ccc(F)cc1[N+](=O)[O-] 94401,c1(NC(CC(C)NC(C2CCC3CC3CC2)=O)C)c([N+](=O)[O-])cnn1C 94402,c1(CCN(C(=O)NCc2cnc(C(C)C)[nH]2)C)ccc(F)c(F)c1 94403,n1(CC)nncc1C(=O)N(CCN(C)C(C1(N(C)C)CCC1)=O)C(C)C 94404,C1(CC)CN(C(=O)CC(C(F)F)NC(=O)C(C)=C2CCC2)CCCO1 94405,c1(OC)cccn2ncc(C(=O)N(C3CN(C(=O)CN4CCC4C)CC3O)C)c12 94406,c1(OC)cc(CC(=O)N(CCNC(=O)CCC2CC2(Cl)Cl)CC2CC2)cc(F)c1 94407,c1(C(N2CCC3CN(C(C4CCN(C)C4=O)=O)C3C2)=O)ccc2c(c1)OCCC2 94408,c1(C(=O)NCCN(C(=O)C(c2ccc(F)cc2)C)CC)ccc(F)c2c1OCC2 94409,C12(CNC(c3cn(CCC)nc3)=O)CC1CN(C(=O)CC1CCC1(F)F)C2 94410,C1(C(N2CCN(C(CNC(=O)CC(F)(F)F)=O)CC2)=O)CCc2nc(O)[nH]c2C1 94411,Cc1c(C(=O)NCC2(CC(N3CCCC3C(N)=O)=O)CC2)[nH]ccc1=O 94412,Cc1noc(C)c1C(=O)Nc1ccsc1C(=O)NC1CC1(F)F 94413,c1(-c2n(C)c(C3CCCC(O)CCC3)nn2)ncc2c(Br)cccc2n1 94414,CC1(C(N2CC(CO)C(c3ccccc3)C2)=O)Oc2ccccc2NC1=O 94415,N1(C(C)C)CC2C3CCC(C2C1)N(C(c1ccnc2ccnn12)=O)C3 94416,c1(NC(C2COCCN2C(C2CC2C2CC2)=O)=O)cc(F)ccc1Br 94417,N(C1CCCn2cnnc21)C(=O)CC1CCCN(C(c2c[nH]nc2Br)=O)CC1 94418,C1(O)(CNC(CCCC(=O)N(C)C)=O)CC2CCC(C1)N2C(=O)Cc1cncnc1 94419,C1(CCNC(C(C2CCCN(C(C3C4CN(C)CC34)=O)C2)C)=O)CCCC2CC12 94420,C1(C(=O)NC2C(NC(c3c(C)cc[nH]3)=O)CCCC2)CN2CCN1C(C)C2 94421,C1(CCC)CN(C(c2nc(C)oc2OCC)=O)CCN1C(c1cc(=O)cc[nH]1)=O 94422,c1(C(=O)NC(C)(CNC(c2cn[nH]c2)=O)Cn2cccn2)cccc2scnc12 94423,c1(NC(=O)NC2CC3CC(C(=O)O)CC23)cc2cc(Br)ccc2s1 94424,c1(CN(C(=O)CC(C)C)C(c2cccnc2)C)ccc(F)c(F)c1 94425,c1(C(=O)NCC(=C)CCNC(=O)Cc2occc2C)ccccc1SCC 94426,C1(C(=O)NCCC2CSCCN2C(=O)C(C)N=[N+]=[N-])(CC)CC(C)(C)C1 94427,N1(C(c2c(C)ncc(N)c2)=O)CC(C)CN(C(c2cc(Cl)ncc2Cl)=O)C(C)C1 94428,C(=O)(C(C)(C)C(=O)N1CCOC(CC(=O)Nc2ccccc2N(C)C)C1)OC 94429,c1(C(C(=O)NCC)N(CC(=O)OCC)C)ncc(Cl)n1C 94430,c1(SCC)ccc(C(=O)NC2CN(C(=O)CCCN(C)C(=O)OC)CC2O)cn1 94431,c1(C(=O)NC(CC)(CNC(=O)C(F)(F)COC)CC)ccc2cccnc2n1 94432,c1(OC)nc(C(=O)NCC2CCN(C(c3sc(OC)nc3C)=O)C2)ncc1F 94433,C(C)(C)(CCNC(=O)Cc1cc(C(C)C)no1)NC(COCC(=O)NC)=O 94434,CC(=O)CCC(=O)N1CCC(c2ccccc2)(NC(c2cccs2)=O)C1 94435,C1(NC(c2ncn(-c3cn(C)nc3)c2)=O)CN(C(=O)CN2CCOCC2)C2CC12 94436,c1(C(N2CC(NC(c3c(C)ncc(C)n3)=O)C(F)C2)=O)cc2cccc(F)c2s1 94437,C(C(C(=O)NOCCCC)NC(c1ccc(C)nn1)=O)SCC 94438,c1(OC)c(Cl)ccc(C(=O)NCC2CC(C)CCN2C(C23CC(OC)C2C3)=O)c1F 94439,N1(C(C(CCC)(C)CC)=O)CC2(C1)CN(C(c1csnc1C)=O)CC2CO 94440,Cc1cc(C(N2CC3(C2)SCCC3NC(=O)CCc2cn[nH]c2)=O)c(Cl)cc1F 94441,c1(C(C)C)ccc(C2(C(N3CCC(NC(=O)CSCC#N)C3)=O)CCCC2)cc1 94442,c1(C(N2CCC(c3nncs3)C2)C(=O)NCCSC)cccc(CO)n1 94443,C1(C)(C(=O)NCC2(OC)CN(C(C3CC34CCC4)=O)C2)CC2CCC1O2 94444,c1(C(=O)OC)cc(C(=O)NCC(C)(F)C(C)C)cc(Cl)c1C 94445,c1(C(N2CCCC(C3N(C(CC=C)=O)CCC3)C2)=O)ccc(CC)cc1Cl 94446,CCCCC(O)CC(=O)NC(CCC1CCC1)C(N1CCC2(CCCO2)C1)=O 94447,c1(C(=O)OC)ccc(NC(C2CC(O)CN2Cc2ccsc2)=O)cc1Cl 94448,c1(C(=O)NCC2(F)CCN(C(CSCCOC)=O)C2)ccc2occ(C)c2c1 94449,N1(C(=O)Oc2ccccc2)CCCC2C1CCN2CCOc1cccc(Br)c1F 94450,C(=O)(C1=CCSC1)NC(C1CCCN1C(=O)C=Cc1cncnc1)C 94451,C1(NC(CCC(C)NC(=O)CCP(C)(C)=O)=O)C2CCCC1CC2 94452,c1(C(N(C)CC2CCCN(C(c3c(C)cn(C)n3)=O)C2)=O)cc2cccnc2s1 94453,N1(C(Cc2nc(CC)sc2)=O)CCCC(C)(NC(=O)CN2CC(C)OC(C)C2)C1 94454,C1(NC(C2C(OC)CC2)=O)CCCC(NC(c2nc(OC)c(C)s2)=O)C1 94455,C=CC(C)(O)C(=O)N1CC(NC(=O)CCOCC)C(C(F)(F)F)C1 94456,CN1CCN(C(=O)C(C)(C)n2cnnn2)CC1CNC(=O)C(F)CC1CCC1 94457,C=C(C)CC(C(=O)NC(c1cccc(F)c1)C)NC(=O)C(=O)NCC(F)F 94458,c1(SC)ccc(C(=O)NC2CCN(C(=O)Cn3cc(C(C4CCOC4)C)nn3)C2)o1 94459,c1(C(C)(C)C)nc(=NC2(CNC(C3CCC4(CC3)CC4(F)F)=O)COC2)s[nH]1 94460,c1(N2CCC(CCF)CC2)nc(N2CCC3C(C2)C3(F)F)c2[nH]ccc2n1 94461,C1(OC)(CNC(C2CC2C)=O)CCN(C(c2sccc2CC#N)=O)C1 94462,c1(C(N(C(CNC(C2CCN(C(CC)=O)C2)=O)C)C)=O)cc([N+](=O)[O-])cc(C)n1 94463,C1(NC(c2ccc(OC)s2)=O)CN(C(c2ccc(CO)nc2)=O)CC1C(F)F 94464,c1(N2CC(CN(C)C(c3c[nH]cc3Br)=O)C2)nc(Cl)nc2c1ncn2C 94465,c1(N(C2CCN(C(CC(CCC)C)=O)CC2)C)ccc(S(=O)(=O)N2CCC2)cn1 94466,c1(C(=O)Nc2c(C)n(-c3ccc(OC(F)F)cc3)nn2)cn2cc(F)ccc2n1 94467,CC1SCCN(C(=O)C(C)(C)C2CCN(C(=O)C#CC3CC3)C2)C1C 94468,CC1=C(C(=O)N2CCCCCC2C(=O)NCCC2(C)CCCC2)COCC1 94469,c1(C(N2CCN(C(C(CC)CC)=O)C(C(C)(C)C)C2)=O)ccc2c(c1)COCO2 94470,C(=O)(CCC(=O)N(CC(N1CCC(CC2CC2)C1)=O)CCC)NCCC 94471,Cc1cc(N)c(C)nc1C(=O)NCC1CCN1C(=O)Cc1nc(C(C)OC)no1 94472,CN1CCN(C(=O)CC2CCCCO2)C(CNC(C2C(C)(C)C2(C)C)=O)C1 94473,c1(C(=O)NCC=C2CCN(C(c3cnc(C)n3C)=O)CC2)cnn2c1N(C)CC2 94474,n1(CC(=O)NCC(CN(C(C2CCCC2O)=O)CC)(C)C)nnc2ccccc12 94475,N1(C(c2ccc(C)c(F)n2)=O)CC2(CCCC2NC(C23CC2COC3(C)C)=O)C1 94476,c1(C(=O)NC(C(=O)OC)Cc2cn(-c3cnn(C)c3)nn2)cccc2nccn12 94477,C1(CNC(C=CS(C)=O)=O)CN(C(=O)C=Cc2cccc(F)c2)CCCO1 94478,C(CCCCCNC(c1cccc(C(N)=O)n1)=O)NC(c1c(C(C)C)c[nH]c1)=O 94479,c1(C(=O)NCc2c(C)c(Cl)ncc2)n[nH]c2c1CN(C(C1CC1C)=O)CC2 94480,c1(C(N(CCN(C(CCCN(C(C)C)C)=O)C)C)=O)cc(O)c2ccsc2c1 94481,c1(N(CC=C)C)ncnc2c1ncn2CC(C)(Cc1ccccc1)CO 94482,C1(CNC(C2CCCO2)=O)CC2CC2N1C(=O)CC1CC(n2cnnc2)C1 94483,C(=O)(CC(C)CC(C)C)N1C(C(=O)NCC2(CC)CC2)CSCC1 94484,N1(C(C(OC)OC)=O)CCN(C(=O)CCCSC)CC(CO)C1 94485,C(=O)(C(CNC(=O)CC1CC=CCC1)C(C)C)N1C(C2(OC)CC2)CCC1 94486,C=C1CC(C(=O)NC2CCCSC2)(CNC(=O)C(C)c2ccco2)C1 94487,O=C1CCOC(C(=O)NCC2CC(F)(CNC(=O)C(F)n3ccnc3)C2)C1 94488,C1(C(=O)NCCC2CCCN(C(C(=O)N(CC)CC)C)C2)CC(=O)NC(=O)C1 94489,N1(C(C(=O)NCCC2(C)CC2)CC2(C)CC2)CCC2(CCCCO2)C1 94490,CCC(CCC(=O)N(C1CC1(C)C)C)NC(c1cn(CC)nn1)=O 94491,C1(OC)CC(Nc2csc3cc(F)ccc23)C12CCOCC2 94492,c1(C(N(CC(C)(C)NC(C2CCC=CCC2)=O)C)=O)ccc2scnc2c1 94493,N1(CC(=O)NCC2(O)CC(NC(c3ccc(CC)o3)=O)C2)CCCCCC1=O 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95041,c1(C(=O)NC(CCCCNC(C(CSC)C)=O)CO)cc(S(=O)(=O)NC)cs1 95042,N(C(=NCc1cccs1)NC1CC1c1ccc(F)cc1)C(CC=C)CO 95043,C1(C(=O)NC2CCCC2NC(c2cnc(C)[nH]2)=O)(OC)CCCCC1 95044,c1(CC(N2C(CNC(CC3CCN(C)CC3)=O)CCC2)=O)n[nH]c2ccccc12 95045,C1(Nc2ccc(OCC(=O)OCC)cc2)CCC2CCCC2C1 95046,c1(CC(=O)NCC#CCNC(Cc2nnn(C(C)(C)C)n2)=O)c(F)cccc1Cl 95047,C1(CC(N2CCC(O)(CC)C2)=O)CCN(C(c2ncc(F)cc2F)=O)C1(C)C 95048,c1(C(=O)NC(CC)CNC(C2CC3OC2C2CC32)=O)ccc2nnnn2c1 95049,c1(OC)nc(NC2CC(F)(CNC(=O)CCN3CCOCC3)C2)nc(C)c1F 95050,C1(N(C(C2(C)CCCS2)=O)CC)CCCN(C(c2c[nH]nc2OC(C)C)=O)CC1 95051,c1(C(=O)NC2CN(C(C3CC(=C)C3)=O)CC2F)csc2c1CCCC2 95052,c1(NC)ccc(C(=O)NCC(C)(C(C)C)NC(=O)Cc2ccc(O)nc2)cc1F 95053,C1(C(N2CCC(OC(C)=O)C2)=O)CCCCCN1C(C1COCCC1C)=O 95054,C1(N(C(C(C)OCCOC)=O)C)CCCN(C(c2ccc(C#N)o2)=O)CC1 95055,N1(C(c2c(Cl)cc(C)nc2)=O)CCC2CCN(C(=O)CC3CC3C3CC3)C2C1 95056,c1(NC(c2ccc3nccnc3c2)=O)ccc2c(c1)CN(CCF)C2 95057,c1(C(=O)NC(C2CCCCN2C(=O)Cn2cncn2)C)ccc(C(F)F)cc1F 95058,c1(C(N2CCC(C)(CNC(C(C)NC=O)=O)CC2)=O)c2c(nn1C)CCOC2 95059,CCC(F)(F)C(=O)NC(C1CC(NC(=O)CC2CCC(=O)NC2)C1)C 95060,N1(C(c2cc(OC)ncn2)=O)CCCC(CO)(NC(=O)CN(C)C(=O)C2CC2)C1 95061,c1(C(=O)NCCCCCC(=O)N(C2CCCC2C#N)C)cc2ccccc2[nH]1 95062,c1(C(N2C(C(=O)NC(CC)C)CC(F)C2)=O)ccc2cc[nH]c2c1Br 95063,n1(CCNC(C2CC2c2cncs2)=O)cc(CNC(C2(Cl)CC2)=O)nn1 95064,C1(C(=O)Nc2cccc(-c3ccccc3)n2)(OC)CCS(=O)(=O)CC1 95065,Cc1nn(C)c(Cl)c1CN1CCCC(NC(c2cccc(OCC(C)C)c2)=O)C1 95066,N1(C(CC(C(=O)OC)(C)C)=O)CCCC2C1CCCN2C(c1ncn(C)c1C)=O 95067,C123C(C4CC1C2C4)CNC(=O)N1CCC3C1.N1(S(C)(=O)=O)CCCC1C(F)(F)F 95068,N1(C(c2cccc(C)c2)=O)CC(CNC(C2OCCCC2(C)C)=O)CC(C)C1 95069,C1(C(=O)NC(CCC)C(N)=O)CCC2(CC2)CN1C(=O)OC(C)(C)C 95070,CC(C)S(=O)(=O)C(C)C(=O)NCC1(C(=O)Nc2cnccc2C(C)(C)C)CC1 95071,N1(C(=O)C(C2CCC2)NC(C23CC(CO)(C2)C3)=O)CCCC(O)C1 95072,C1(NC(c2n[nH]c3c2COC3)=O)CN(C(c2cc(O)ncc2F)=O)C2CCCC12 95073,c1(C(C)(C)C(F)F)ccc(COC(=O)C(Cl)Cl)cc1 95074,N1(C(c2cccc(C)c2Cl)=O)CCN(C(=O)C(C)(O)CC(F)(F)F)CC12CCC2 95075,c1(C(N(CCC(C(C)C)NC(C=CC)=O)C)=O)cc2cc(Cl)sc2[nH]1 95076,c1(CC)ncc(C(=O)NC2CC(C)(NC(=O)Cc3ccc(SCC)cc3)C2)cn1 95077,C1(C#N)(C(=O)NCCCC(CNC(c2cccc(COC)c2)=O)C)CCCCC1 95078,c1(C(=O)Nc2c(C)ncc(Br)c2)cc2oc(C)cc2[nH]1 95079,c1(-c2cn(CC(=O)NC(c3ccc(C)[nH]3)CC)nn2)c(C(=O)O)cnn1C 95080,C(=O)(C(C)C(C)(C)O)NCC(C1CC1)NC(c1nn(CC)c(C(F)(F)F)c1)=O 95081,c1(C(N2CCC(NC(C(C)CC3CCC3)=O)(CF)C2)=O)cnn2c(=O)cc[nH]c12 95082,c1(CC(=O)NC2C(NC(CC=CC=C)=O)CCCC2)ccc(C)c(Cl)c1 95083,C1(C(N(C(C)C(=O)N(C)C)C)=O)CCCN(C(=O)Cn2cncn2)C1 95084,c1(-c2nnc(C)o2)ccc(C(=O)NCC(CO)NC(=O)CCC=CC(C)C)cc1 95085,c1(CNC(C(=O)N(CC(C)C)C(c2cc[nH]c2)=O)=O)ccc(Cl)c(C(F)(F)F)c1 95086,O=C1NCCC12CCCN(C(=O)C(c1ccc(I)cc1)O)C2 95087,C1(NC(=O)CC2CC3CC3C2)CC2CC1N(C(C1(N3CCOCC3)CC1)=O)C2 95088,n1(CCCOC)nnnc1C(c1nncn1C(C)C)NC(COC)C(C)C 95089,C1(CC(=O)NCC(CCNC(C(CC)=CCCC)=O)O)CCCOCC1 95090,C1(NC(=O)C=Cc2cncs2)COC2(CCN(C(=O)Cc3cnns3)C2)C1 95091,Cc1cc(C(=O)NC(CNC(=O)C(C)Cc2ccc(F)cc2)C(C)C)nc(O)c1 95092,c1(NCc2ccc(C)nc2Cl)ccc(S(=O)(=O)NC2COC(C3CC3)C2)cc1Cl 95093,c1(C(=O)NC2C(NC(C(C3CCC3)OC)=O)C2)sccc1Cl 95094,C1(CNC(c2csnc2Cl)=O)CCN(C(=O)CCc2nncs2)CC1O 95095,Cc1coc(C(N2CCC(C(C)NC(=O)CC3CC(=O)C3)C2)=O)c1C 95096,n1(C(c2cccc(Br)c2)C)c(-c2cn(C)nn2)csc1=Nc1ccc(O)cc1 95097,C(c1cncnc1O)=CC(=O)NC(CCC)CNC(=O)CC1CN(C)C1 95098,C(CCCCCO)c1cn(CCOCCNC(CC2C(C)C2)=O)nn1 95099,N1(C(c2cc(C)oc2)=O)CCCC(NC(=O)CC(C2CC2)C2CC2)C1C 95100,C1(CC(=O)N(C2CCCCC2)C)C2CN(C(=O)CC(F)F)CC12 95101,O=C(C1CCCn2nccc21)NC1CCN(C(c2cc(F)c(F)cc2Cl)=O)C1 95102,c1(C(N(C)CC2CCN(C(CC3(OC)CCC3)=O)C2)=O)cc(C)ccc1C 95103,c1(NC2C(SC)CCC2)nc2ccccc2nc1NCC(C)C(C)C 95104,c1(C2(C(=O)NC3C(NC(=O)CO)CCC3)CCC2)ccc(Br)cc1 95105,c1(C(N(CCC(=O)NCCCCF)C(C)C)=O)nn(C)cc1Cl 95106,C1(CNC(c2c(OC)csc2)=O)CN(C(=O)CCc2c[nH]c(=N)[nH]2)CC1C 95107,C(=O)(C1=C(F)CN(C(c2ccc3occc3c2)=O)CC1)NC(C)C(O)C(F)F 95108,N1(C(C(CCSC)NC(N)=O)=O)CCCC(CNC(=O)C=C(C)C)CC1 95109,Cn1ncc2c(N)c(C(=O)NC(CNC(=O)CC3CC=CC3)CO)cnc12 95110,N1(C(COC(CC)C)=O)CC(C2CN(C(c3cc(C)c(OC)c(C)c3)=O)C2)C1 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95128,C(=O)(C1CCc2snnc21)N1CCC(CN(C(C2(C)CNC(=O)C2)=O)CC)CC1 95129,C1(C(=O)NCC(CN(C(=O)CCCc2cccs2)C)(C)C)CC2CCC1O2 95130,C=CCN=C(NCC1CN(C)CCN1C)NCC1CCN(CC)C1 95131,C1(NC(CCOCCC)=O)CCSC12CN(C(=O)C(C(C)C)n1cnc(C)c1)C2 95132,C(=O)(CC1=CCCCC1)NC1CN(C(C2CC3(CC(C)C3)C2)=O)CC12CC2 95133,C1(C(N2CCC(F)(C(=O)N(CCCO)C3CCC3)C2)=O)CC2(CCCO2)C1 95134,c1(CC(=O)NCCC2N(C(c3c(C)csc3)=O)CCOC2)c(C)nc(O)nc1C 95135,C=CCC(C)C(=O)NC1COCCC1C(=O)NCC(C)(O)C1CCC1 95136,Cc1ccc(C2CCCC2NC(c2nnnn2C(C)C)CCC2CCCO2)cc1 95137,C1(C)(CNC(C2(C(=O)OC)CCO2)=O)CC(OC)CN1C(c1cncn1C)=O.C1(C)CC1 95138,N1(C(c2ccc(SCC)cc2)=O)CC2(C1)CN(C(=O)CN(C)CCOC)CCO2 95139,Nc1ccc(Cl)cc1C(=O)NCC1(F)CC(NC(=O)CC2CCC(O)C2)C1 95140,C1(NC(CCCC(=O)OCC)=O)COC2(CCN(S(C)(=O)=O)C2)C1 95141,CC1(C)CCN(C(C2OCCC2(C)C)=O)CC1C(=O)NC1(CC(N)=O)CC1 95142,CN=C(NS(=O)(=O)Cc1ccns1)NC1CCCC1COC(C)(C)C 95143,c1(CC(=O)NCC(C2CC2)NC(c2c(C(N)=O)coc2)=O)cnc2cccnn12 95144,C1(C(N2CC(N(C(=O)C(CO)NC(=O)C(F)(F)F)C)C2)=O)CC2(C1)CC2F 95145,CC1(C)CCN(CCNC(C2C=CCCN2C(=O)CC2OCCO2)=O)C1 95146,Cc1c(CC(=O)NCC=C2CCN(C(=O)CCCCN(C)C)CC2)cnn1C 95147,CC1CCC(C(=O)NC2CC2CNC(c2ccnnc2O)=O)CC1 95148,c1(CC(=O)NCC2C(CNC(C3CCN(C)C3)=O)C2)c[nH]c2ccncc12 95149,Cc1cc(N2CC(C(C)NC(=O)CC(C)c3ccccc3)C2)c(Br)cc1[N+](=O)[O-] 95150,Nc1cc(C(N2CC(C(N3CCNCC3)=O)C2)=O)c(F)c(F)c1F 95151,c1(C(N2CCCC(C)(NC(=O)CCC3CCC3)C2)=O)ccc([N+](=O)[O-])cc1 95152,N1(C(C(C)(C)NS(C)(=O)=O)=O)CC2CCN(C(c3cc(F)cc(Cl)c3N)=O)C2C1 95153,c1(C(=O)NCc2nc(C(=O)NCC3CC3)co2)cnc(O)c(F)c1 95154,C(=O)(C(F)C(CC)CC)N1C(CNC(CN(C2CC2)CC)=O)CCCCC1 95155,Cc1cnccc1C=CC(N1CCC(CNC(=O)Cc2ccc(O)cc2Cl)C1)=O 95156,c1(CCC(=O)NCC2N(C(c3occ(C)c3C)=O)CC2)c(Cl)cncc1Cl 95157,C1(NC(CSCC#C)=O)C2CC3CN(C(=O)CC(n4nc(C)cc4C)C)C1C3C2 95158,c1(C(=O)NCC(CNC(CCNS(CC)(=O)=O)=O)(C)C)cc(Cl)nnc1O 95159,c1(C(=O)NCCCOCCN(C)C(C2CC23CCOC3)=O)cn2cccnc2n1 95160,c1(C(N(C(C(=O)NC(C(=O)OCCC)(C)C)C)CCC)=O)ccc(CC)c(F)c1 95161,CCCC(C(O)C(=O)N1CCC(N(C)CC)C1)NC(=O)CCn1cnc(=N)[nH]1 95162,CC(C)(F)C(C)(F)C(=O)N1CCCN(C(=O)CCC2CCC(O)CC2)CCC1 95163,C(=O)(C1=CCCN(C(C2C=CC=CC=C2)=O)C1)NCC=CCCC 95164,C1(NC(COC(C)C)=O)CCOC(C(=O)NC2(CO)CC2)C1 95165,CC1C(NC(=O)CC(C)(C)C)NCCN1CC=CCN 95166,C12(C(N3C4C(NC(CC5(OCC)CC5)=O)CC(C4)C3)=O)CCC(CO)(CC1)CC2 95167,n1(CC(=O)NC(CNC(C2(OC)CC2)=O)C(C)(C)C)c(O)nc2ccccc12 95168,C1(CC)COC(C)CN1C(c1nc(F)ccc1Br)C(=O)NCCCC1CC1 95169,C12(NC(c3cnc(C)[nH]3)=O)CCCCC1N(C(c1csc(S(C)(=O)=O)c1)=O)CC2 95170,N1(CC(=O)NCC(CNC(CCOC(C)=O)=O)C)CCCCC1C 95171,CC1OC2(C)CC1(C(N1CC(C(N)=O)(CNC(c3ccc(C#N)cn3)=O)C1)=O)C2 95172,C1(CCC)CN(C(=O)CC2CCN(C(c3cc[nH]c(=N)n3)=O)C2)CCO1 95173,C(=O)(C(O)CC(F)(F)F)N1CC(C(C#C)OC)(NC(=O)Cc2ccccc2)C1 95174,c1(OC)ccc2c(ccn2CC(=O)NC2CCCC2CNC(=O)C(F)C(C)C)c1 95175,c1(C(=O)NCC2N(C(C3CCC3)=O)CCN(C)C2)nnc(O)c(Br)c1O 95176,C1(C(=O)NC2C(C)(C)C(Nc3ncc(Br)cn3)C2)CC2CCCCCCC12 95177,CC1CC(C(N2CC(NC(C3(C)CC3(F)Cl)=O)C2)=O)CCS1 95178,O=C1CC(C(N2CCC(CNC(=O)CCN3CCOCC3)CC2)=O)NCN1 95179,C(=O)(C(=O)N=S(C)(C)=O)N1CC(C)(c2cn(C3CC4OC(=O)CC34)nn2)C1 95180,C1(CC)CCN(C(=O)C(O)C(C)CC)C(C(N2CCCN(C(N)=O)CC2)=O)C1 95181,c1(CCS(=O)(=O)NC(c2c(CC#N)n[nH]c2)=O)c[nH]c2ccccc12 95182,C1(CC)CCCC1C(=O)NC1(CNC(=O)CC2(NC(C)=O)CCCC2)CCOC1 95183,C1(NC(C2CC(NC(C3CNC(=O)N3)=O)C2)=O)CC2CC(O)C1C2 95184,C1(C(=O)NC2CC(n3cccn3)C2)(CC)CCCN(C(=O)CCCC#N)C1 95185,N1(C(C(n2nnnc2C(C)(C)C)C)=O)CC(NC(=O)C(C)C(C)(F)F)C(C)(C)C1 95186,CC(C)CCC(C(=O)N(CCN=[N+]=[N-])C)NC(=O)CCCC1CCCC1 95187,C(CC(N)=O)(C(=O)NC(c1ccccc1O)C)NC(CC(C)OC)=O 95188,CC1(C)Cc2ccc(S(=O)(=O)N3CCCC(c4ccno4)C3)cc2C1 95189,C1(OC)CN(C(=O)CN2CSCC2=O)CC1NC(C12CC1CNC2=O)=O 95190,c1(OCC)cccc(CC(=O)NC2CC(CO)N(C(=O)CCC3CC3C)C2)n1 95191,c1(C(=O)NCCC2CC(NC(C3N(CC)CCC3)=O)C2)cccc2sccc12 95192,C(=O)(C1CCCc2nn[nH]c21)N1CC2CCN(C(=O)CC34CC(C3)C4)CC2CC1 95193,c1(C(=O)NC2(C)CC(NC(c3cnn(CC)c3Cl)=O)C2)sc2cncn2c1C 95194,c1(-c2ccc(C)cc2)cn2cnc(C(=O)Nc3nc(C)ccc3C#N)c2s1 95195,C(=O)(CC1=CCN(C(c2n[nH]c(O)n2)=O)CC1)N(CC(C)C)C1CC1 95196,C1(C(N2CCC(c3ccnn3C)C2)C(=O)NCC(=C)C)CCOC2(CCC2)C1 95197,c1(COC)cccnc1C(=O)NCCC1CCCN(C(c2cc(C)co2)=O)C1 95198,FC(F)(F)CCCCN=c1[nH]c2c(c(=NCc3cccc(C4CC4)c3)[nH]1)COCC2 95199,c1(C(=O)NCCNC(c2cc(C(C)(C)C)n[nH]2)=O)cccc2c1CCC2 95200,C1(NC(CCCSC)=O)CC2CCC(C1)N2C(=O)C=Cc1ccc[nH]1 95201,N1(C(CCCOCC)=O)CC2(CC(NC(=O)C(F)(F)c3ccccn3)C2)C1 95202,C1(CC(=O)N(C2CC2)CC2CC2)(OC)CN(C(C)=O)C1.C1(C)CCN1 95203,C1(C(=O)NC(CNC(CC(CC)C2CC2)=O)C(C)(C)C)CCn2c(O)nnc2C1 95204,N1(C(c2cnc(COC)s2)=O)CC2C(CNC(=O)Cn3ccnn3)C2C1 95205,CCCC(C(F)(F)F)NC(=O)CC=CCNC(c1ccc(OC)s1)=O 95206,C=C(C)CCCC(=O)NCC(C)N(C)C(C1CCCCN1C(c1ccco1)=O)=O 95207,N1(C(CC(C)C)=O)CCCC2(CCN(C(c3ccc(N)cc3)=O)C2)C1.CC=CCN 95208,c1(NC(=O)NC(c2cccc(C)c2)C)cccc2c1CC(=O)N2 95209,C1(NC(C2CC(C(F)(F)F)(OC)C2)=O)CN(C(=O)CC(C)(C)O)CCC1F 95210,c1(OC)cc(C)nc(C)c1NC(=O)NC1CC2CNC1C2 95211,C(=O)(C1CCc2ccccc21)N1C(CNC(Cn2nc(C)c(Cl)c2)=O)CC1 95212,C12(C(=O)NC3C(C)N(C(c4ccc(F)nc4)=O)CCC3)CCC(CC1=O)C2(C)C 95213,N1(C(C(C(=O)OCC)F)=O)CC2(CCN(C(c3ccc(F)cc3O)=O)C2)C1 95214,c1(C(=O)NC2C(C(N(C)C)=O)C3CCC2C3)cnc2[nH]cc(C#N)c2c1 95215,N1(C(c2cc(C(C)=O)[nH]n2)=O)CCC2(CCN(C(=O)CN3CCCCC3C)C2)C1 95216,C#CCC(O)C(=O)N1CCOCC1CC(N1CCOCC1CCC)=O 95217,c1(C(N(CCCCNC(C2CC2(C)C)=O)C)=O)ccc(OCC(F)F)nc1 95218,C1(Cn2c(N(C(c3ccccc3)C)CC)nnn2)CCN(C)C1 95219,C(=O)(C(O)CCCCC)N1C(C2(NC(CC=CCC)=O)CC2)CCC1 95220,CC(C)(C)S(=O)(=O)CC(=O)NC12CC(C1)N(C(=O)CCc1ccc(F)cc1F)C2 95221,C1(CNC(CCCC(C)O)=O)CN(C(c2ccc3[nH]ccc3c2)=O)CC12CCC2 95222,c1(OC)ccc(C(=O)NCC(CNC(c2ccc(C)o2)=O)OC)c2ccccc12 95223,N1(C(C(c2cnn(C)c2)C)=O)CC(CC(N)=O)OC(C)(C)C1 95224,C(=O)(NNC(=O)CCN1CCCCC1)NC1CCN(CC(CC)C)C1 95225,C1(N(C(CN(C)C(N)=O)=O)C)CCC2CN(C(=O)COc3ccsn3)CC12 95226,C1(C(C)NC(CCSC)=O)CN(C(=O)CNC(=O)C2CC2)CCO1 95227,C1(CCNC(CNS(N)(=O)=O)=O)CCC(NC(=O)COCC2CCCO2)C1 95228,C(=O)(C1CCc2c[nH]nc21)N(C(CC)CC(=O)N1CC(N2CC(O)C2)C1)C 95229,c1(OC)ccc(F)c(C(=O)NCCC2CCN(C(=O)CC3(OC)CC3)C2)c1F 95230,Cc1ccc(C(=O)NC2CCC(CNC(=O)CCC(=O)N(C)C(C)C)C2)nc1C 95231,c1(CCCC(=O)NC2CCCC(CNC(C=CCOC)=O)C2)c(F)cccc1F 95232,CC1(C)CC(CNC(C2CCCC2O)=O)CN(C(c2ccc(O)c(F)c2F)=O)C1 95233,c1(C(=O)NC2C(CNC(C(N3CCC(C)C3)=O)=O)C2)ccn2nccc2n1 95234,N1(C(CCCOC(C)=O)=O)CCN(C)CC1C(N1CC(CCO)C1)=O 95235,N1(C(c2c(C)nc(Cl)cc2)=O)CCC2(CC1)CCN(C(c1ccc(Br)cn1)=O)C2 95236,C(CCSCCO)(C(=O)NC)NC(C1(N=[N+]=[N-])CC1)=O 95237,N1(C(=O)NC(c2nc(CC)sc2Br)C)CCCN(S(C)(=O)=O)CC1 95238,C1(OC)CN(C(=O)C(C)Oc2cccc(Br)c2)C(C)(C)C1 95239,c1(-n2cnc(C(N(C)C)=O)n2)ncc(Cl)cn1.c12ccc(o1)C(=O)NOC2 95240,N1(C(COCCNC(c2ccc(C)cc2)=O)=O)CC(C)CCCC1C 95241,c1(C(=O)NCC2N(C(C3C(COC)C3)=O)CC2)cnn(CC(F)F)c1C 95242,N1(C(C(C)n2cccc2)=O)CCCC(CC(=O)NCCCc2cc[nH]n2)CC1 95243,C1(F)(CNC(C2(CC#C)CC=CCC2)=O)CCN(C(=O)C=C(C)Cl)CC1 95244,C(C(=O)N1CC(c2ccccc2)(NC(=O)Cc2cnns2)C1)(C(C)(C)C)SC 95245,c1(CC)nc2n(n1)CC(NC(=O)NCC1CCCN(C)C1=O)CC2 95246,C1(C(N2CC(N(OC)C)C2)=O)COCC2(CCN(CC(C)C)C2)O1 95247,C(=O)(C(CNC(C12CCCC(CO1)C2)=O)C(C)C)NCCC(C)C 95248,N12CCC3CCN(CC13)C(=O)C1(C)CCN2C1.c1(CCC)ncoc1C=O.CC 95249,C1(CN(C(c2cc(C)oc2)=O)C)CCN(C(C2CCOC(=O)N2)=O)CC1 95250,C(N=c1cc(C)[nH]c(=NCc2cocn2)[nH]1)C1(SC)CCCCC1 95251,N1(C(C2(SC)CN(C(c3nn(CC)c(O)c3)=O)C2)=O)CC2CC2C2CC12 95252,CC1CCN(C(=O)C(C2CC2)NC(c2csc(O)n2)=O)CCS1 95253,CN1C(=O)OCC1C(N1CCC(CNC(C23CC(C)(CO2)C3)=O)C1)=O 95254,c1(C2OCCN(C(C3COCC4(CCC4)O3)=O)C2)c(F)cc(Br)cc1F 95255,c1(C(=O)NC(CNC(C2C(F)(C(=O)OC)C2)=O)(C)C(C)C)cc(C)c(C)cc1N 95256,c1(C(=O)NC2CC(C(C)NC(c3cnc[nH]3)=O)C2)ccc(Br)c2ccncc12 95257,C1(C(=O)NCCCC#C)(CF)CCN(CC(=O)NCc2cc(CC)oc2C)C1 95258,CCC(CC)C(C(=O)N1CCC(N(C(=O)CCn2ccnc2C)CCO)C1)OC 95259,c1(C(=O)NCCCCC(=O)NC2(CO)CN(C(N)=O)C2)cccc(C=C(F)F)c1 95260,C1(C(N2CCCCCC2CCO)=O)(OC)CCN(Cc2cnc(F)c(Cl)c2)CC1 95261,C12(C(N3CCCN(CCC#C)CC3)=O)CCCCC(CNC1)C2(F)F 95262,N1(C(C(c2ccoc2)NC(c2cc(CC)on2)=O)=O)CCn2cnnc2C1 95263,N1(C(c2cc(OC)c(Br)s2)=O)CCCC12CCCN(C(=O)C(C)O)C2 95264,N1(C(C(CC(=O)OCC)C)=O)CCC(C)N(C(=O)CCc2cn[nH]c2)CC1 95265,c1(OC)noc(C)c1S(=O)(=O)NN(C)CC(C)CC(C)C(C)(C)C 95266,c1(C(=O)NCc2cccc(-c3ccc(NCC4CC4)nc3)c2)ccc(O)cc1F 95267,C1C(=C(C(=O)OCC)C(C)C)C(C#C)(F)CCN1C 95268,C(=O)(C1=CC(O)C(NC(=O)CCc2cnoc2)C1)N1CC(C#N)(SC)C1 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95286,C1(O)(CC(=O)NC(C(C)NC(Cc2ccn(CC(C)C)n2)=O)(C)C)CCOCC1 95287,c1(NCC2(OC)CCC(C)(C)C2)ccc(C#N)c(C)c1 95288,C(c1ccccc1Br)=CC(=O)NC1CN(C(c2ccc(C(N)=O)[nH]2)=O)C1 95289,c1(C(N(CCN(C(=O)C(C)NS(C)(=O)=O)CC)CC)=O)nn(C)nc1C 95290,c1(C(N2CCC(N(C(CC(COC)C)=O)C)CC2)=O)c(OC)cccc1O 95291,CC1CC(C(=O)NCC(F)C2CCC2)CCN1C(c1occ2c1CCC2)=O 95292,C1(CC(=O)NCCCC2CCCCN2C(=O)CSC2CCCC2)CCCOCC1 95293,C(=O)(CC(C(F)F)NC(C1OCCO1)=O)N(CC=C)CC 95294,C1(NCC(C)(N)C2CCC2)CCC(CCc2ccncc2)CC1 95295,Cn1cc(C#CCNC(=O)CNC(c2ccns2)=O)cn1 95296,C(CC(=O)N(CCCCN(C(=O)CCSCCC)C)C)OCC#C 95297,C1(C(=O)NC(C(=O)NC)(C)C)CN(Cc2cn(C)nn2)CCC1O 95298,CC(C)CC(CNC(c1csc(C2CC2)c1)=O)NC(C1CC(OC(F)F)C1)=O 95299,Cn1cnc2c1C(C(=O)NCCCNC(=O)CCCc1ccncc1)CC(=O)N2 95300,c1(C(=O)OCc2c(C)sc(Br)n2)c(Cl)sc(Cl)c1C 95301,C(C1=CCN(C(C2CC3C=CC2C3)=O)CC1)NC(C(c1cnn(C)c1)OC)=O 95302,C1(CC(=O)NC(c2ccnc(F)c2)C)CCN(C(=O)CC2CCCC2)CC1 95303,O=C(CCCn1cc(CCC(=O)CS(=O)(=O)CC(F)(F)F)nn1)N=c1cco[nH]1.N 95304,Cn1nc(C(=O)NCCC2(NC(c3cc[nH]n3)=O)CCC2)cc1C(F)(F)F 95305,C(=O)(C1=C(C#N)CCC1)N1CC(OC)C(C(=O)NC2(S(C)(=O)=O)CCCC2)C1 95306,C1(C(=O)NCC(=C)CCNC(c2cnn(C3CC3)c2)=O)(CC)CCC(C)(C)CC1 95307,CC1CN(C(C2CCC(C)(O)CC2)=O)CCC1NC(C1SC2C=CC1CC2)=O 95308,C(=O)(CC(O)C(C)(C)C)N(CCN(C(c1ccnc(OC)c1F)=O)C)C 95309,Cn1cnnc1CCC(=O)NCc1ocnc1Cn1cc(C2(C)CC2)nn1 95310,CC1Oc2c(C(=O)NCCCOCC(=O)O)cccc2NC1=O 95311,N1(C(C2(CC=C)CCCN2C(C2CC(C)CCO2)=O)=O)CCC2CN(C)CC2C1 95312,C(CCC(C)(C)NC(=O)Cc1cnc(C2CC2)[nH]1)NC(C(C)OCCCC)=O 95313,CCC(CCC(=O)N1CCC(C(=O)NCc2cc(F)ccc2O)C1)OC 95314,C(C)(C)(CC(F)C(=O)N1CC(CO)C1)NC(CC(C)(C)C)=O 95315,Cc1cnc2c(CN3CC4CN(C(=O)Cc5cnn(C)c5)CC4C3)cnn2c1 95316,c1(C(=O)NC(CNC(c2cc(C)c(N)cn2)=O)C2CC2)ccc2sc(C)nc2c1 95317,C1CCCCC(=O)N1C.C1(C(=O)NC2(CC(=O)OC)CC2)CCCCC1F 95318,c1(OC)coc(C(N2CC(C)CCC2CNC(=O)C(C)(C)CN(C)C)=O)cc1=O 95319,c1(C(=O)NCC2CN(C(C3CCCCCC3)=O)CCO2)ccc2ocnc2c1 95320,N1(C(c2ncn(C(C)(C)C)c2)=O)CC(NC(c2ocnc2C(F)F)=O)C(CO)C1 95321,C#CCCCCCCC(=O)N1CCC(C(C)C(=O)N(C(C)C(=O)OC)C)CC1 95322,N1(C(CCOC(C)=O)=O)CCCC2(C1)CN(C(c1ncn3c1CCC3)=O)CCO2 95323,C1(C(N2C(CN(C)NC(c3cn(CC4CC4)nn3)=O)CCC2)=O)CC2CCC2C1 95324,c1(CC(=O)NC2(CNC(c3cc(CCO)on3)=O)CC2)nc2ncccn2n1 95325,Cc1ncc(C(=O)NCC2CCCCN2C2CC2=CC(F)(F)F)n1C 95326,C(CNC(C1CN(C(C)=O)C1)=O)(C(C)(C)C)NC(C(CC1CCC1)OC)=O 95327,C#CC1(C(N2CC(O)(C(F)C(=O)Nc3ccc(COC)cc3)C2)=O)CC(=O)C1 95328,c1(OC)cc(C(C(=O)NC2(C)CC2)N(C(C)C)C)c(Br)cn1 95329,c1(CC)c(Cl)nc(C2CCCC2)[nH]c1=NCCN(C(=O)CC(C)(C)C)C1CC1 95330,C1(C(=O)NCC(CCC)O)CCN(C(=O)C(C(=O)OC)OC)C12CC2 95331,c1(C(N2CC(N(C(c3scc(C)c3C)=O)C)C2)=O)ccc2c(c1)CCC=C2 95332,CCC(O)C(C)C(=O)NC1CC(c2ccccc2)(NC(c2cc[nH]c(=N)c2)=O)C1 95333,C1(C2CCN(C(C3CCNC3=O)=O)CC2)(NC(C2=NOC(C)C2)=O)CC1 95334,n1(CC)nc(C(F)(F)F)cc1C(N1CCCC(N(C(=O)C2=CCC2)CCO)C1)=O 95335,c1(OC)cc(CCC(=O)N(C2CCC(NC(=O)C(C)(C)C)C2)C)ccc1F 95336,Cc1ccccc1CCCN1CCC(N(C(=O)C(CO)c2ccccc2)C)C1 95337,c1(C(=O)NC(CN(C(c2c(OC)cc(Cl)cc2)=O)C)C)ccc2c(C)noc2c1 95338,Cc1ccc(CCC(N2CCC(C)C2CNC(=O)Cc2ccsc2)=O)cc1 95339,N1(C(C(C)C2CCC2)=O)CCC2C(C1)NC(=O)CN2C(=O)C(=O)N1CCCC1 95340,c1(CN(CCCOC)C(C)C)cc(C(=O)O)ccc1I 95341,c1(C(=O)NCC2(C(F)F)CCN(C(C(CCC)O)=O)C2)cc2ccc(C)cc2[nH]1 95342,C(CCCCCNC(=O)C1CC1)NC(C(n1cc(Br)cn1)C)=O 95343,C1(c2c(C)cccc2C)CCN1N1CC2CCC(CO)(CC2)C1 95344,CC12CCCC1N(C(C1C3CC3CN1C(=O)CC#N)=O)CCC2 95345,C1(C(=O)NCC(C)N(C(CCC=CC)=O)C)CCCC(OC)C1 95346,c1(C(N2CCC(O)(C(C)NC(=O)CN(C)S(N)(=O)=O)C2)=O)cc(Cl)cc(Cl)c1 95347,c1(CC)cnc(Cl)[nH]c1=NCC(C)(C)NC(C1CCC2CC(C)CN2C1)=O 95348,C(=O)(C1=NN(C)C(=O)CC1)N(C1CCN(C(c2c(C(C)C)ccc(Cl)c2)=O)C1)C 95349,C(=O)(CC(F)(F)C(C)C)N(CC)CC1CCCN1C(=O)C=Cc1c(C)noc1C 95350,N1(C(c2c(CC)ncs2)=O)CC2(CCN(Cc3cc(C)nc(C)n3)C2)C1 95351,c1(OC)cc(O)c(CNC2CC2C(=O)Nc2ccc(Br)cc2CO)c(Br)c1 95352,N1(C(C2(SC)CN(C(C3CCC(F)C3)=O)C2)=O)CCC(C2(C)CC2)C1 95353,CCC(C(C)(F)F)NC(=O)CN(C1CC(C#N)C1)C(c1cc(C)c(C)[nH]1)=O 95354,c1(OC)cc(C(N2CCCC2CNC(=O)C(C)C(C)C)=O)cc(Br)c1 95355,Cc1c(-n2cc(CC3CCN(C(c4ccc(CO)cc4)=O)C3)nn2)cccc1Cl 95356,O=C(N=c1ccn(CCO)[nH]1)C1CCCN1C(c1cc(C(=O)NC)[nH]n1)=O 95357,c1(CNC(C(CC)C)c2nnnn2CC(F)F)ccc(F)c(F)c1C 95358,CC1(CN(C(C)(C)C)C(C2(C)CN(C(=O)CC34CC(C3)C4)C2)=O)CCOCC1 95359,C1(NC(c2coc(Cl)n2)=O)CCC2CCN(C(C3CCC(=O)N(C4CC4)C3)=O)C12 95360,c1(CC)nn(C)c(CC(=O)NC2CCN(C(=O)COCC(=O)OC)C2CC)c1Cl 95361,n1(C(C(=O)NC2CCN(C(C(C(C)O)C)=O)C(C)C2)C)cc2ccccc2n1 95362,c1(C(=O)NC2C(CNC(Cc3scc(C)n3)=O)CCCC2)cc2ccccc2o1 95363,N1(C(CCC=C=C)=O)CC(NC(=O)Cn2ccccc2=O)C2(CCC2)C1 95364,C1(C(=O)NC(CCNC(c2c(C)snc2)=O)C(C)C)CC2(CCOC2)C1 95365,C(=O)(CC(C)(O)CC(=O)O)NC1CCCN(C(c2ccc(C)cc2C(C)C)=O)C1 95366,c1(CC(C)C)cc(C(=O)NCC(F)CNC(=O)C(F)CC2CC2)cc(O)n1 95367,c1(CC(=O)NCCN(C)C(C2(CCF)CC2(F)F)=O)ccccc1CO 95368,Fc1ccc(C2(C)CCCCC2)cc1Cl.c1(CNC2CC2)nnnn1C1CCOC1 95369,c1(C(=O)NC2(C)CCN(C(CCCC)=O)C2)cccn2c(CC)nnc12 95370,C(=O)(C1OCC(C)c2ccccc21)NCCOC(c1cc(OCC)no1)=O 95371,N1(CCC(N2CC(CNC(C(C=C)(C)CC)=O)OCC2)=O)Cc2ccccc2C1 95372,C1(CNC(C(c2ccc(F)cc2)OC)=O)N(C(=O)C2=CCOC2)CCCC1(C)C 95373,C1(C(=O)NCCNC(C2CC3(C2)CC32CCC2)=O)CCCC12OCCO2 95374,C1(C(=O)NC2CCC(NC(C=Cc3ccc(C)o3)=O)C2)CCCC(C#N)C1 95375,N1(C(c2cc(C)c(C)nn2)=O)CC(C)CN(C(c2ccn(C)c(=O)c2)=O)C(C)C1 95376,C1(NC(CCCOCCOC)=O)CC(O)CN(C(=O)CCS(=O)(=O)N(C)C)C1 95377,N1(C(Cc2c(C)cc(C)s2)=O)CCN(C(C2(C)CCCNC2=O)=O)CC12CCC2 95378,CCCC(C)(O)C(=O)N1C2CCC1C(CNC(c1cc(Br)cnc1N)=O)C2 95379,C(=O)(C1CCCn2ncnc21)NC1CCN(C(c2c(CC)noc2)=O)C1C 95380,C(=O)(C1=CCCC1P(C)(C)=O)N1C(C(C)NC(CCOC)=O)CCC1 95381,N1(C(C2C3(CC(NC(c4cnc(CC)o4)=O)C3)C2)=O)CC2CC(C)C2C1 95382,C#Cc1ccc(CN(c2cc(-c3ccc(F)nc3F)ccn2)c2ccccc2)cc1 95383,c1(N(C)Cc2scc(C)c2)cc(NCc2ccc(N3CC=CC3)cc2)ncn1 95384,C1(C(NNC(=O)NCC(C(C)C)(C)C)=O)Sc2ccccc2NC1=O 95385,C1(CNC(c2cnc(C3CCCO3)s2)=O)(Cc2cccc(Br)c2)CCCCC1 95386,Cc1cc(C#N)cc(C)c1C(=O)NC(CNC(=O)C=Cc1cncn1C)C1CC1 95387,CCCCCC(O)C(=O)N1CC(F)(C(=O)NCC2(C)CC(C)=NO2)C1 95388,CC1=C(C(=O)NCCCCCN(C(=O)C(n2ccnc2C)C)C(C)C)CCC1 95389,c1(C(=O)NC(C)CN(C(=O)CC(C)c2cccnc2)C)ccsc1S(N)(=O)=O 95390,c1(SC)ccc(NC(=O)NCCc2cncc(C)n2)c(Br)c1 95391,N1(C(C2C3(CCN(Cc4n(C)ncc4)C3)C2)=O)CCC2(CCNC(=O)CC2)CC1 95392,O=C1CCCCC(C(=O)NC2(CCC(=O)NC3CC4CCC3O4)CCCC2)C1 95393,CCC(O)C(F)(F)C(=O)NCc1cc[nH]c1C(=O)NC(C)CCO 95394,C1(C(N2CC(C#C)(N(C)C)C2)=O)CC(F)(F)CN1C(C1OCCC1C(C)C)=O 95395,C1(COC)(CNC(=O)CC=CCc2ccccc2)CCN(C(c2cnns2)=O)C1 95396,C12(C(=O)NC(CCOC)CNC(c3ncc(C)cn3)=O)COCC1C2(F)F 95397,C12(NCc3ccc(CCCCC)cc3)CCC(CO)(CC1)OC2 95398,c1(C(N2CCC(C(=O)NC3(C)CC3)C(O)C2)=O)ccc(C#N)c(F)c1 95399,c1(C(C)=O)ccc(O)c(NC(=O)C=CC2CCCN2C(=O)COCC(C)C)c1 95400,N1(C(C2N(C(C3CCC3)=O)CCN(C)C2)=O)CCC2CC1C(=O)N2C 95401,Cc1ccc(C#N)cc1C(N1CCC(NC(C2(C)CC(C)(C)C2)=O)C(C)C1)=O 95402,N1(C(C(N(C)C)C2CC2)=O)CC(NC(c2ccc(C(C)(F)F)cc2)=O)C(C)(C)C1 95403,C(=O)(CC(C)(C)C(C)(F)F)NC(CNC(C1(C)CCN(C)C1)=O)(C)CO 95404,C(C(C(C)C(C)C)NC(=O)C1=NOCC1)NC(c1n(C=C)ncc1)=O 95405,N1(C(C(C)(C)O)=O)Cc2ccccc2CC1CNC(=O)Cc1c[nH]nc1O 95406,CCCCCC(C)(C)CNC(=O)C(C1CCN(C(c2sc(F)cc2C)=O)C1)C 95407,c1(C(N2CC(CN(C(CC(=O)NCC#C)=O)C)C2)=O)cncc2sccc12 95408,N1(C(c2ccc(C)s2)=O)CCc2sc(CNC(=O)C=CC3CCCN3C)nc2C1 95409,CCCCC(O)C(=O)NCC(CO)NC(c1cncc(NCC)c1)=O 95410,CN1CCCC(CCNC(=O)CC2CCCC(NC(=O)Cc3ccsc3)C2)C1 95411,C(=O)(CC(C(C)(C)C)NC(=O)CC1=CCOCC1)NCc1c(C)noc1 95412,c1(C(N2CC(N(C(CC(n3ccc(C)n3)C)=O)C)C2)=O)n[nH]c2c1CN(C)CC2 95413,c1(CC(=O)NCC(C2CCOC2)NC(CCC#C)=O)cccnc1OC 95414,n1(CC)cc(CN(C)C(=O)NCCC2(CO)CCOC2)nn1 95415,C1(NC(C2OCCN(CC)C2)=O)CC2CC1CC2C(=O)NC1CN(C)CC1C 95416,C1(C)(CC)CC(NC(C2CC(F)(CO)C2)=O)CN1C(c1cnc(SC)s1)=O 95417,C1(CC=C)(NC(c2cnc(CC)[nH]2)=O)CCN(C(=O)Cn2cnc(C#N)n2)C1 95418,N(S(=O)(=O)N1Cc2ccccc2C1)C(C(c1ccccc1)N(CC)CC)=O.C(C)(=O)O 95419,c1(C(=O)NCC(CCOC)NC(=O)C(C)OCC(C)C)cnc2c(c1)nnn2C 95420,N1(C(c2c(C)nccc2)=O)CCN(C(=O)C#CC(C)(C)O)C(CC(C)(C)C)C1 95421,S(=O)(=O)(c1cc(Br)c2c(c1)OCCO2)N(C1CCNC1)CC 95422,N#CC1CCC(C(=O)NC2CC(CNC(=O)CCc3cnc[nH]3)C2)CC1 95423,C1(NC(CC(CCC)O)=O)CCC2CN(C(c3ccc(O)c(N)c3)=O)CCC2C1 95424,C1(C(c2cccc(Cl)n2)NC(c2n(CC)ncn2)C)CC12CCC(F)(F)CC2 95425,N1(C(CCC)=O)C(C)C2CC1C2NC(=O)CCCc1ccc(Cl)c(C)c1 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95740,c1(C(C(=O)NCC(F)F)N(C2CC2)CC)ccc([N+](=O)[O-])c(O)c1 95741,N1(C(c2cnn(CC)n2)=O)CC2CCC(NC(=O)Cc3c(C)noc3Cl)CC2C1 95742,C=C(C)c1cccc(NC(C2C=CCN2C(=O)CC2CCC(=O)NC2)=O)c1 95743,C(C(C)(O)C(F)(F)F)NC(CC(CNC(CCCNC(=O)OC)=O)C)=O 95744,C1(C(=O)NC(C(C)Oc2ccccc2)=O)COCCN(C(=O)C=CC2CCC2)C1 95745,CC1(C)OCCCC1CNC(=O)CC1CCN(C(=O)Cc2ccccn2)CC1 95746,N1(C(CC)=O)CCC(NC(=O)C(C)n2cncn2)C1.C1(=O)CC2(CC2)N1 95747,c1(CCCC(=O)NCC(CNC(CN(C2CCC2)C)=O)F)csc2ccccc12 95748,C1(CC(=O)NCC(CCC)C)CCCN(C(C2CC(F)C2)=O)C1 95749,CC1CN(C(=O)CN(C)C(N)=O)CC(CCNC(=O)C(c2ccccc2F)O)O1 95750,c1(C(N2CC(N3CCN(C(C(CCSC)O)=O)CC3)C2)=O)cc2n(n1)CCO2 95751,c1(CCCC(=O)NC2C=CCN(C(CNC(COC)=O)=O)C2)ccc(C)c(C)c1 95752,Cn1cc(C(N2CCC(C(=O)Nc3c(O)cccc3F)CC2)=O)n(C)c1=O 95753,N1(C(C2(F)C(C)OCC2)=O)CCCC2(CCN(C(=O)CC3CCC=CCC3)C2)C1 95754,c1(C(=O)NCCCCNC(C2COC(=O)O2)=O)ccc2cncnc2c1 95755,c1(C(=O)NCC(C)(O)CNC(=O)C2=CCSC2)c[nH]c2cccc(C#N)c12 95756,N1(C(c2cc(C(F)(F)F)ccc2I)=O)CCC2(CCN(Cc3cccnn3)C2)C1 95757,N1(C(COCCC=C)=O)CCN(C2CCC(NC(=O)C(C)(C)C3CC3)C2)CC1 95758,C1(C(=O)NCC(c2ccc(F)cc2)NC(=O)C(F)C2CCC2)CCCCS1(=O)=O 95759,c1(C(C)(C)CNC(=O)OCc2nc[nH]n2)ccc(F)cn1 95760,C(=O)(C(CC(F)F)C1CCC1)NCCN(C(C1(C)ON=C(C)C1)=O)C 95761,CC(C)(C(=O)NCC(CO)NC(C1CCOC1)=O)C1CCC1 95762,C1(NC(C2(C(=O)OC)CC23CCC3)=O)C2CC3CC1CC(O)(C3)C2 95763,CNS(=O)(=O)N1CCC(C(=O)NCCNC(C2CN3CCC2(C)CC3)=O)CC1 95764,C1(c2ccccc2)(NC(C2C(C=C)C2)=O)CCN(C(=O)C=Cc2nccs2)C1 95765,CC1CCC(Cl)=C(C(=O)N2CCCCC2CNC(=O)CC2CCCOC2)C1 95766,N1(C(c2c(C)csc2)=O)CC2CC(C1)CN(C(C1CC(C)(C)C(C)(C)C1)=O)C2 95767,c1(C(N2CCOCC(NC(C3C(COC)C3)=O)C2)=O)cc2ccc(F)cc2cn1 95768,c1(C(N2C(CNC(c3ccc(OC)nc3)=O)CC2)=O)ccc(F)c2ccsc12 95769,C1(N(C(c2cc(C(C)C)no2)=O)C)CCCC(NC(C2CN(C(C)C)C2)=O)C1 95770,c1(C(=O)NCC(CC)(C)NC(C2CNC(=O)O2)=O)nc2ncccn2n1 95771,Cc1cccc(F)c1C(=O)NCCC1CN(C(C2CC(=O)NC(=O)C2)=O)C1 95772,N=c1cc[nH]cc1CNC(=O)NC1CCN(c2cccnn2)CC1 95773,C1(CNC(Cc2cccc(OCC)c2)=O)CN(C(c2scnc2C)=O)CC12CC2 95774,CN(CCCC(=O)N1CCC(C(C2CCC2)NC(=O)C(O)C(F)(F)F)CC1)N=O 95775,c1(SC)cccc(C(=O)NC2CN(C(c3cccnc3O)=O)CC2C)c1O 95776,O=C1CCC(C(=O)NC(C2CCCC2)CNC(c2cc(F)c(F)cc2O)=O)=NN1 95777,Cc1onc(C(N2CCCC(NC(c3cc(Br)no3)=O)C2)=O)c1[N+](=O)[O-] 95778,c1(C(=O)NCCC2(CO)CN(C(c3ccc(OC)o3)=O)C2)ccnc(SCO)c1 95779,c1(N2CC(C)(C)OCC2)nc2cccnc2c(=NC2CCC(CC(N)=O)C2)[nH]1 95780,N1(C(C2C(C(C)C)CCC2)=O)CC(N(C)C(C2CCC(=O)O2)=O)C(C)(C)C1 95781,C1(C)(CC)CC(NC(=O)CC2(C)CCCC2)CN1C(=O)CSc1n[nH]c(O)n1.C1(C)CC1 95782,C12(CC(=O)N(C)Cc3cnccn3)CC(CCO1)N(C(=O)CC1COC(=O)C1)C2 95783,c1(SC)cccc(-c2nnc(N(CCCC(C)C)C)n2CC2CCCCO2)c1 95784,N1(C(C(CC(C)C)ONC(C2CCOCC2(C)C)=O)=O)CCc2c(nnn2C)C1 95785,c1(C(N=c2nnn(C)[nH]2)=O)oc2ccccc2c1CO.c12cc(Br)ccc1N2CCO 95786,C1(C(N2CC3C(NC(C(C)N(C(C)=O)C)=O)C3C2)=O)CCC([N+](=O)[O-])CC1 95787,c1(CNC(=O)CCc2ncc[nH]2)ccc(CNC(c2cc(Cl)ns2)=O)cc1 95788,C(CC(=O)N1CC2CCC(C1)N2C(=O)C=Cc1ncc[nH]1)(C(F)(F)F)OC 95789,C1(C(=O)NCC2(C)CC(C)C2)CCC(C2CC2)N1C(C1CC(F)C(=O)N1)=O 95790,N1(C(c2cnc(COC)s2)=O)CC2(CCC2NC(=O)C(C)=C(C)C)C1 95791,c1(C(=O)NCC(CC)NC(c2csc(C(C)OC)n2)=O)ccc(O)c(Cl)n1 95792,N1(C(C2(C)COC2)=O)CCCC2(CCCCC2NC(C2CC3CC3C2)=O)C1 95793,Cc1cc(C(N2CCC(CN(C)Cc3conc3C)C2)=O)cc(C)c1 95794,N1(C(C(C)NC(COC)=O)=O)CC2C(N(C(=O)CN3CCC(O)CC3)C)C2C1 95795,N1(C(CC(C)(C)NC(c2c(C)nn(C)c2)=O)=O)CC2CCCCCC2C1 95796,CN1C(=O)C(=O)N(CC(N2CCC(C)(C)C2CNC(=O)CC2CCC2)=O)C1=O 95797,C(=O)(CC(C)(C)C)N1CC(N(C2CCC(Oc3ccncc3)C2)CC)C1 95798,CC(C)(C)CC(O)C(=O)N1CCCC1C(C)(C)NC(c1ncc2[nH]ncc2n1)=O 95799,N1(C(C2(C3CCCO3)CC2)=O)CCCCC1C(=O)N(C1(SCC)CC1)C 95800,C(CC(C(=O)N(CC(N1CCCC(CC(C)C)C1)=O)C1CCC1)OC)OC 95801,c1(C(N(C(C)C(N2CCCC(C)(C)C2C)=O)CC)=O)ccc2[nH]ccc2c1 95802,CCC(CC(=O)NC1CN(C(c2[nH]cc(C)c2C)=O)CC(C)(C)C1)CC(F)(F)F 95803,c1(C(N2C3(CNC(CC4(C)CCCO4)=O)CC(C2)C3)=O)cccc2c[nH]nc12 95804,N1(C(c2c(COC)ccs2)=O)CCN(C(=O)C=Cc2cscn2)C(CC(F)F)C1 95805,c1(C(N2CCC(C(C)(C)NC(CS(=O)(=O)NC)=O)C2)=O)cc(C)ccc1N 95806,Cc1nc(NC2CC2)sc1C(=O)NC(C)CN(C)C(C1CC2CC2C1)=O 95807,C(CC(C)(C)C)(C(=O)NOCCC(C)O)NC(c1c(C)n(C)nn1)=O 95808,c1(OC)ccc2c(c1)C(C(=O)Nc1ccc(N(C)C)cc1)C(C)N2 95809,c1(CC)cc(C(N2CCCC2C(C)NC(c2cc(F)cc(F)c2)=O)=O)ccc1C 95810,c1(C(=O)NC2C(C)CN(C(=O)CCCN(C)N=O)C2)noc2c1CC(C)(C)CC2 95811,C#CCC(C)(C)C(=O)NC1CC(N(C(=O)CCC=CC(C)C)C)C1 95812,c1(OC)cnnc(C(=O)NC(C2CN(C(=O)CCOc3ccccc3Cl)C2)C)c1 95813,O=C(CN1C(=O)C(F)(F)Oc2ccccc21)OC(C(F)(F)F)c1nccs1 95814,C1(NC(=O)Nc2cccc(C)c2)CCN(Cc2cscn2)CC1(C)C 95815,CC(CC(N)=O)C(=O)NCC(N=c1[nH]nc(-c2ccccc2)o1)c1ccccc1 95816,C1(CNC(C2CC(F)(CO)C2)=O)C2CN(C(=O)CSc3ccc(F)cc3)CC12 95817,C(=O)(NNc1cc(Cl)cc(Cl)c1)C(Cn1cc(-c2c(C)ccc(C)c2)nn1)=O 95818,n1(CCC(C)C)nc(-c2ccc(N)cn2)nc1CCc1nc(-c2cccs2)no1 95819,C1(C2C(NC(=O)CCSC3CC3)C2)CCCN(C(c2cncc(C3CC3)c2)=O)C1 95820,N1(C(C=CC=CC)=O)CCCC(C)(C)C1CNC(=O)C(CC)C(F)(F)F 95821,C1(NC(CC(C)F)=O)CN(C(=O)CCOc2cccnc2)C2(CCCC2)C1 95822,C(CCC(O)CO)SC.C12CC(CO1)NC(=O)C1(CCC1)CC(=O)NC2 95823,C1(NC(c2cc(OC)c(Br)nc2)=O)CCC2CN(CC(=O)N(C)C)CC2C1 95824,c1(C(C)NC(C2OCCN(C(c3c(C)nn(C)c3)=O)C2)=O)cccc([N+](=O)[O-])c1 95825,c1(SC)ccc(Cl)c(C(N2CCN(Cc3cn(CCF)nn3)CC2)=O)c1 95826,CC(C)C(C)CC(=O)N1CC(O)CC1CNC(=O)COc1ccon1 95827,N1(C(CC2CCCC(C)(C)O2)=O)CCN(C(=O)CC(F)(F)F)CC12CCC2 95828,N1(C(C2CC(=O)N2)=O)CC2CN(C(c3cccc(F)c3Cl)=O)CC12 95829,C1(NC(C2CC(CC)(CC)C2)=O)C=CCN(C(=O)C(N2CCOCC2)C)C1 95830,c1(-c2n(-c3c(CC)cccc3)nc(CCOC)n2)ccc(S(C)(=O)=O)c(F)c1 95831,Cc1c(C(N2CC3CC3(CNC(=O)CCOC3CC3)C2)=O)cccc1C(F)(F)F 95832,N1(C(C(C)(C)OCC)=O)CCCC(N(CCO)C(c2coc(C)n2)=O)C1 95833,c1(OCCC)cc(CNCCCNC(C2CCN(C(C)=O)C2)=O)ccn1 95834,c1(C(=O)NCC2C(CNC(C(F)=CC)=O)C2)ccc(-c2cccnc2)s1 95835,c1(C(=O)NCCn2cc(C(=O)NC(COC)C3CCC3)nn2)cncc(C)n1 95836,c1(NC(C(C)n2ccnn2)=O)cccc(CNC(c2ccoc2Br)=O)c1 95837,c1(OC)c(F)c(CN(C)Cc2ccc(Br)cn2)cc(OC)c1F 95838,C1(C(=O)NCc2c(C(=O)NC3CCN(C)C3)occ2)CC1C1CCCC1 95839,N1(C(C=CC)=O)CCOCC(C(=O)Oc2ccccc2OCC)C1 95840,C1(CC(=O)N(C2CCCN(C(CN(C(=O)OCC)C)=O)C2)C)CCC(C)(C)CO1 95841,C(=O)(CC(C)(C)CC(F)F)NC1CC(C)N(C(C2CCN2C2CCCC2)=O)C1 95842,Cc1cccc(C(=O)NCC2(C)CCC(NC(c3cnccn3)=O)C2)c1 95843,C1(C#N)(C(=O)NCC2CC(OC)CN2C(C2CCC2(C)C)=O)CCOCC1 95844,C1(C(=O)NCCSCCC=C)CCC(O)CN1C(c1cccc(OC)n1)=O 95845,C12(NC(CN(CCC)C)=O)CC(CNC(=O)CCC(C)(C)OC)(C1)OC21CCC1 95846,c1(CCN)ccn(C2CC2)c1.C1(CC(C(C(=O)N(C)C)=O)=O)CCCOC1 95847,N#Cc1cc(Br)ccc1CN1CC2CN(C(c3cc(Cl)sc3Cl)=O)CC2C1 95848,N1(C(C2(C)C(C)C2)=O)CCOCC(CNC(c2ccc(Cl)c(Cl)c2)=O)C1 95849,n1(C(C)C)ccc(CCN2CCCC2c2cncn2C)n1 95850,N1(C(C(=O)NC(CC)CN(C(=O)C=C2CCC2)C)C)C(=O)NC2(CCCC2)C1=O 95851,N1(C(CCCC(=O)NCC)=O)CC2C3CCC(C2C1)N(C(c1cn(C)nn1)=O)C3 95852,C(C(=O)N=c1ccn(C(C)C)[nH]1)(c1cccs1)NC(c1c(C)cns1)=O 95853,c1(C(=O)Oc2cccc(C3CC3)c2)ccc2nccn2n1 95854,CN=c1[nH]c(=NCCCN2CCOC2=O)[nH]c(=NC2CC(=O)N(C)C2)[nH]1 95855,C#CC(C(C)(C)C)NC(c1cccc(CNC(=O)COCC(=C)C)n1)=O 95856,C(=O)(C(C)Cc1cccnc1)NC(c1cn(C(C2(CSC)CC2)C)nn1)CCC 95857,C(CC1C(=O)Nc2ccccc21)NC(=NCC)NCC1(C)CCC(=O)N1 95858,C1(NC(C2(OCC)CCCC2)=O)COC2(C1)CN(C(=O)C(CC1CC1)OC)C2 95859,C1(CCC)CN(C(C2CCCCN2CCC)=O)CCN1C(=O)C1=CCC1 95860,C(=O)(C1=NOC2(CCN(C(c3ccc(F)c(F)c3F)=O)C2)C1)NCCCC(C)C 95861,c1(CCC(=O)NCC(C2CC2)NC(CCC(=C)Cl)=O)nc(O)c2cnn(C)c2n1 95862,c1(OC(C)C)cnccc1C(N1CCC(CNC(C2(CO)CCCCC2)=O)C1)=O 95863,c1(C(C(C)NC(=O)CCc2cnc[nH]2)NC(c2ccon2)=O)ccccc1 95864,C1(CNC(CCC(CC)C)=O)CC2(CO1)CN(C(=O)CCC1CCCCC1)C2 95865,N1(C(=O)CC2CCC2(F)F)CC(CO)C2(C1)CN(C(=O)C(F)F)C2 95866,C=CCN(OC)C(=O)C(C(C)O)NC(=O)CCC(C)NC(C)=O 95867,c1(C(c2n(C(CC)(C)C)nnn2)NC2(c3ccncc3)CC2)cnc(OC)c(F)c1 95868,C(=O)(C(C)CCCOC)NC1CC(C)(CNC(c2c(CC)cno2)=O)C1 95869,C1(CNC(C2N(C(c3cccc(C)c3)=O)CCC2)=O)CC2CC1CC2CO 95870,CCN=c1[nH]c(C(=O)NCCC(C)(C)CNC(c2cnc(O)cc2OC)=O)cs1 95871,C#CCCCCC(=O)NCC12CC(NC(C3CCCC3(F)F)=O)(C1)C2 95872,C1(CC(N2CCCCC2CNC(c2cc(C)c(C)[nH]2)=O)=O)(COC)CCOCC1 95873,c1(C(=O)NC2CCN(CCCNC(C(C=C)OC)=O)C2)cc(O)cc(=O)o1 95874,C(=O)(CC(CCCC)NC(=O)Cc1nc(=N)[nH][nH]1)NCCC=CC=C 95875,c1(SCC(=O)NCCCC2CN(C(C3(F)CCOC3)=O)CCO2)ccc(F)cc1 95876,CC1CCN(C(c2cc[nH]n2)=O)CCN1C(C1(c2ccccc2)CC(O)C1)=O 95877,N1(C(C2(C(F)F)CCCC2)=O)CC(Nc2ncnc3scnc23)CC2(CCC2)C1 95878,c1(C(=O)Nc2cc(C)c(O)cc2)cn2c(n1)CN(Cc1cccc(F)c1I)CC2 95879,CC(=O)CCCC(=O)N1CCCC1CN(C(=O)C(C)Cc1cccc(Br)c1)C 95880,C1(C(N2CC(CNC(=O)CCCCCO)C(F)(CO)C2)=O)Cc2ccncc2C1 95881,Cc1nc2c(s1)CCCC2CNC(c1nc(Br)sc1C1CC1)=O 95882,c1(C(N2CCC(C(C)NC(c3cscc3F)=O)C2)=O)c(F)ccc2c1OCC2 95883,N1(C(C(c2ccccc2F)C)=O)CCC2C(NC(=O)CSc3ccc(Cl)cc3)C12 95884,c1(C(=O)NCC=CCNC(c2cc(C)nn2CC(F)F)=O)c(Cl)ccc(C)c1O 95885,C1(C(=O)NC2C(OC)CN(C(C=CC=CCC)=O)C2)CC(=O)CC(=O)N1 95886,c1(C(=O)NC)ccc(C(=O)NC(CNC(c2ccn(CCOC)n2)=O)CO)s1 95887,N12CCN(CC1)c1ccc(o1)C2.Cc1c[nH]cc1CNS(=O)(=O)CCCl 95888,C12(O)CCN(CC1)C(C)(C)C=CC(=O)NCC2.C1(NC(N)=O)COC2COCC12 95889,c1(C(=O)NC2CCN(C(C(CSC)C)=O)C(C)C2)cn2cnnc2cn1 95890,C1(C(N(OC)CC2CCCCC2)=O)CC(O)CN1C(c1cc(F)n(C)n1)=O 95891,CC(C(C)(C)CO)NCc1n[nH]c(C(C)(C)C)n1 95892,N1(C(C(C)CC(N)=O)=O)C2CCC1CC(N(C)C(c1cccc(C(N)=O)c1)=O)C2 95893,c1(C(=O)OCCc2ccc(OC)c(Br)c2)ccc2c(c1)C(=O)OC2 95894,N1(C(C(CC)N(C)C)=O)CCN(C(=O)CCN2CCCS2(=O)=O)C(CO)C1 95895,C1(C(=O)NCCCN(C(c2c(CC)con2)=O)CC)CCSC(C)C1 95896,N1(C(=O)Cn2cc(C(F)(F)F)cn2)CCC2CN(C(=O)CC3CC3)CC2C1 95897,C1(CNC(Cc2[nH]c(=N)sc2)=O)CCN(C(C2CC3C=CC2C3)=O)CC1C1CC1 95898,c1(C(=O)NCC(CN(C2CC2)OCC)(C)O)nc(Cl)ccc1N.c12nc(cs1)CC2 95899,c1(NC(c2ncn(CC)n2)=O)ccc(N)cc1.C(C)(C)(CC(=O)OCC)N(CC)CC 95900,c1(C(N(CCN(C)CC2CCCC2)C)=O)cc(-c2ccoc2)on1 95901,Cc1cnc(C(=O)NC2CN(C(c3c(O)cccc3F)=O)C3CC23)c(C)c1 95902,c1(C(=O)NC(C(CO)NC(CN(CC)CC)=O)C)ccc(F)cn1 95903,CC(C)C(C(C)NC(c1cscn1)=O)NC(c1ccc(CO)o1)=O 95904,C=CCCC(C)NC(=O)C(C)N(C(=O)C(=O)NC1CC1)CC 95905,c1(NC)ccc(Cl)c(C(=O)NCC(C(C)(C)C)NC(=O)C(C)c2ccon2)c1 95906,C1(NC(C2CC(=O)NC2)=O)CN(C(c2cnc(Cl)c(Cl)c2)=O)CCC1(F)F 95907,CCCS(=O)(=O)c1ccc(C(=O)NC(CC)(CC)CCNC(=O)CCOC)cc1 95908,C1(CC(=O)NC(C#C)(C)C2CC2)C2CCC(C2)N1C(C1CCOC1C(=C)C)=O 95909,C1(N(C)C(C2CCCS2)=O)CCCC2CN(C(=O)CC3CCS(=O)(=O)CC3)CC12 95910,C=CCC(CC(=O)NCC#CCOC)NC(c1cccc(C#N)c1C)=O 95911,c1(C(=O)NC2C(NC(=O)CCN3CCCCC3=O)CC2)ccc2nc[nH]c2c1F 95912,C=CCC(C)(C)CC(=O)NCC(CC)(CC)NC(=O)CCC(C)C#N 95913,c1(OC)cc(OC)c(C(N2CC(C)(NC(=O)C(O)Cn3cncn3)C2)=O)c(N)c1 95914,c1(C(=O)NC2C(C)CCN(C(=O)CCOC3COC3)C2)cc2cccc(Cl)c2[nH]1 95915,c1(C(N(CC(C)O)CCNC(=O)Cc2cc(C3CC3)no2)=O)cnc2c[nH]nc2c1 95916,N1(Cc2c(C)n[nH]c2C)CC2(CN(C(=O)COc3ccccc3)CCO2)C1 95917,C1(CC)(CO)CCN(C(=O)C(O)CNC(c2cc(Cl)no2)=O)C1 95918,C1(n2ccnc2)(C(=O)NC(CCNC(C=CCC)=O)C)CCCC1 95919,Cc1cc(C(C)(C(=O)NCCCC(C)CO)NC(=O)OC(C)(C)C)ccc1Cl 95920,c1(OC)ccc2[nH]nc(C(=O)NC(C)CNC(c3c(F)cc(C)cc3F)=O)c2c1 95921,C=Cc1cccc(CN2CC3CC2CN3C(c2nc(Cl)sc2Cl)=O)c1 95922,CC1CN(C(c2cccn3ncnc23)=O)C(C)CN1C(c1ccc(O)nc1Cl)=O 95923,CCCC(CCC)CC(=O)NCC1(F)CC(CNC(=O)CC(CC)OC)C1 95924,C(CN=[N+]=[N-])(C(=O)NC1CC2CCCC2C1)NC(c1n[nH]c(C)c1O)=O 95925,c1(C(=O)NC2CC3CN(C(c4ccc(F)cc4F)=O)CC23)cccc2nc[nH]c12 95926,C(=O)(C(C)CS(C)=O)Nc1cccc(NC(c2sc(C)c(O)n2)=O)c1 95927,c1(C(=O)NCC#CCNC(c2nncc(OC)c2)=O)cc2ccc(Cl)c(F)c2o1 95928,c1(C(N(C)CC2C3CN(C(COC)=O)CC32)=O)ccc2ncccc2c1F 95929,c1(NC(C(C)Cn2ccc3ccccc23)=O)cc(S(C)(=O)=O)ccc1F 95930,C1(NC(CSS(C)(=O)=O)=O)COCCC1Cc1ccco1 95931,C1(NC(C(CCC)O)=O)CCCN(C(=O)CCc2ccc(F)nc2)CC1 95932,C1(CNC(c2c(OCC)ccs2)=O)C2CC1N(C(=O)C=CC1CCC1)C2 95933,C(CC(=O)NC1CC(C)N(C)CC1C)(C(C)(C)C)NC(c1n[nH]c(C)c1Cl)=O 95934,c1(-c2c(C)occ2)nc(CC2CCC(O)C2)n(C2CCCCC2)n1 95935,c1(C(=O)NC(CC=CC)C(=O)NCC=CC2CC2)cnc2ccccn12 95936,C(=O)(C1=CCOCC1)NCC1(C)CCN(C(=O)CCC2CCCCC2)C1 95937,N1(C(C2C(C(N)=O)C2)=O)CC2CCC(C1)N2C(c1ccc(F)c(N)c1)=O 95938,CC1COCC(C(N2CCC(C(=O)NCC(C)(O)C(F)F)C2)=O)O1 95939,c1(NCC(CC)N(c2ccccc2)C)nccc(=NC(C)c2cccnc2)[nH]1 95940,c1(OC)ccc(C(N2CC(NC(C3CCCOC3)=O)C3CC3C2)=O)cc1[N+](=O)[O-] 95941,c1(CCC(=O)NC2CC3CCC2N3C(c2ccnnc2)=O)ccc(O)c(F)c1 95942,CC(C)C(C(=O)N(CC(C)O)C1CCC1)n1cncn1 95943,C1(NC(CCc2cc(C)sc2C)=O)CCCCN(C(C2CC2C(F)(F)F)=O)C1 95944,c1(C(=O)OC)ccc(C)cc1CC(N1CCC(Cn2cc(CSC)nn2)CC1)=O 95945,N1(C(C2CCN(C(c3cscc3Br)=O)C2)=O)CCC(O)(CO)CC1 95946,CCC(CN(C)C)CC(=O)NCC(C)(C)CN(C)C(c1ccc(CC2CC2)cc1)=O 95947,c1(C(N2c3cccc(C(=O)OC)c3CC2)=O)ccc2c(F)cc(F)cc2n1 95948,C(=O)(CC(C)P(C)(C)=O)NCCC(CNC(C1C2CCCC12)=O)OC 95949,C1(C(=O)NCC(=O)OCC)(NC(CC(N(CC)CC)C2CC2)=O)CC(F)C1 95950,C1(COC)CCC(C2COCCN2C(=O)C(=O)N(C)CC2CCCCC2)O1 95951,N1(C(C)=O)Cc2ccccc2CC1C(=O)NCC(C)OC(F)F 95952,c1(C(=O)NC(C2CCN(C(CS(CC)=O)=O)C2)(C)C)cc(F)cc(C)c1C 95953,C1(CNC(C2C(OCC)C2)=O)CN(C(=O)CCCC(N)=O)CCC1C 95954,N1(C(c2n[nH]c(C)c2O)=O)CC(=O)NCC1C(=O)NC1CCOC1(C)C 95955,C1(CNC(CNC(N)=O)=O)CN(C(c2cccn2Cc2ccccn2)=O)CCO1 95956,CC(C)(C#N)CC(=O)NCCC1CCN(C(c2cncc(C(N)=O)c2)=O)CC1 95957,C(=O)(CC(C)c1ccco1)N(C1CCCCC1)CCNC(CSCC#C)=O 95958,Cc1sc(Cl)c(C(=O)NCC(=O)NC2CC(NC(C)CCCC(C)C)C2)c1C 95959,C(=O)(C(C(C)C)C(=O)OC)NC1C(C(=O)Nc2cccc(C(=O)NCCC)c2)C1 95960,C1(C(N(CCCCC2CCCC2)C)=O)CCCN1C(=O)C(=O)NC1CCCCO1 95961,N1(C(COCC(=O)NC)=O)CCCC(NC(c2cc(N)cc(F)c2)=O)CC1 95962,C1(NC(c2c(SCC)cccn2)=O)CC2CC1CN(C(=O)CC1CC3CC3C1)C2 95963,C1(CCCNC(c2scc(C)c2)=O)CN(C(c2sccc2C#N)=O)CCO1 95964,c1(C(=O)NC2C(CNC(c3c(OC)nn(C)c3)=O)C2)cccc2c1OCCC2 95965,c1(OC(C(=O)NCC=CCNC(CCC)=O)(C)C)ccc([N+](=O)[O-])cc1 95966,c1(CC(N2CC(NC(C=CCN(C)CC)=O)C(C)CC2)=O)ccc(Cl)c(Cl)c1C 95967,C1(NC(C(C)c2cccs2)=O)CCN(C(c2c[nH]c(C(F)(F)F)c2)=O)CC1F 95968,c1(NC(Cc2cccc(NC(CC(C)C)=O)c2)=O)ccc(O)cc1[N+](=O)[O-] 95969,C(N(C(=NCCCCCCS(N)(=O)=O)NCCCCC(C)C)S(=O)(=O)C)C(C=C)C 95970,C1(C(=O)NCc2cc(C(N(CCO)CC)=O)n(C)n2)CCC(=O)C(C)C1 95971,c1(C(N(C)CC)=O)cc2ccc(OCCN(C(COC(CC)C)=O)C)nc2[nH]1 95972,N1(C(c2c(C)ccc(F)c2)=O)CCC(F)(F)C(NCc2cc(Br)c(Br)s2)C1 95973,C1(NC(C2(CC#C)CCCCC2)=O)COC2(C1)CN(C(=O)C(C)N1CCC1)C2 95974,N1(C(c2ccnc(C(=O)OC)n2)C(=O)NCCCSC)CCC(S(N)(=O)=O)CC1 95975,N1(C(C(C2CCOC2)OCCOC)=O)CC(CNC(=O)C(CC)(CO)OC)C(C)C1 95976,C1(C)(C(=O)NC(C)CCN(C)C(c2cncc(Cl)c2)=O)CCc2ccccc2C1 95977,C1(C(N(CC(O)CNC(c2coc(CO)c2)=O)C)=O)CC12CC(C)(C)C2 95978,N1(C(C2N(C(C)=O)CC=C2)=O)CC2CCC(C1)C2C#N.C1C(=O)N1C 95979,c1(C(N2CCC(OC(F)F)CC(C)(C)C2)=O)cnc2ccccc2c1 95980,C1(C)(CC)CC(NC(C23CC(CO)(C2)OC3C)=O)CN1C(=O)CSC(F)F 95981,C1(NC(C2CC2F)=O)CN(C(c2cnc(S)nc2)=O)CC2(CCC2)C1 95982,C1(n2cc(C3CCN(C(C4CC45CCC5)=O)C3)nn2)CCOCC1O 95983,c1(C(=O)NC2CC(N(C(CCCOCCC)=O)C)C2)ccc(CC)cc1O 95984,C1(C)(CC)CCC(NC(=O)C(C)(C)C2CCCN2C(C2CCC(=C)CC2)=O)CC1 95985,N1(C(Cc2c(C)scc2)=O)CCCC2(CC(NC(c3ncccc3F)=O)CO2)C1 95986,c1(C(=O)OC)nc(C)n2c1N(C(C1CCC1c1ccccc1)=O)CC2 95987,C(C(CCO)C(C)(C)C)NC(C(=O)NC1C(C)(C)C1)=O 95988,N1(C(C(=O)Nc2c(C)c(Br)c(Br)cn2)=O)CC2(COC(C)(C)C2)C1 95989,c1(C(N2C(CNC(C(C3CC3)OCC)=O)CC2)=O)nc(C(=O)O)cn1C1CC1 95990,Cn1cc(Cl)c(C(=O)NCc2occc2C(=O)NCc2cc(O)ns2)n1 95991,C1(NC(=O)NCc2ccc(CO)cc2)CCN(C(=O)C=C(C2CC2)C2CC2)CC1 95992,C1(CCC(=O)N(C(C(C)SC)C)C)CCN(C(c2cnc(O)o2)=O)CC1 95993,c1(N2C(CC(=O)OCC)CCCC2)ncnc(OC)c1Br 95994,N1(C(CC(CCCC)O)=O)CC2(CCN(C(c3cc(C)nc(O)c3)=O)CC2)C1 95995,C1(C)(CNC(C2(F)CC(C(=O)OCC)C2)=O)CCN(C(C2CN(C)C(=O)N2)=O)C1 95996,C1(F)(C(=O)NCC2N(C(c3c(CC)nco3)=O)CC=C2)CCCN(C)C1 95997,c1(-c2nc(CSC)nn2-c2ccn(C3CCOCC3)n2)cnn2c(C)ccnc12 95998,Cn1cc(C(N2CCC(F)(CNC(=O)C(O)C(F)F)C2)=O)c(Cl)n1 95999,N1(C(C2N(Cc3c(C)cc(Br)cn3)CC3(CC3)C2)=O)CCC(C)(CO)C(O)C1 96000,C#CCCC(O)CCNC(C1CSCN1C(c1cccnc1C)=O)=O 96001,C1(C(N2CC(SC)C(n3cc(C(C)(C)CO)nn3)C2)=O)CCCCN1N=O 96002,Cc1cnc2nccc(C(=O)NC3(CN(C)C(c4cnn(C)c4C)=O)CC3)c2c1 96003,c1(NC(C2C(NCc3ccc(OCC)c(C#N)c3)C2)=O)nccc2scc(Br)c12 96004,N1(C(Cc2ncc(CC)[nH]2)=O)CCC2CN(C(C3CCc4c[nH]nc4C3)=O)C2C1 96005,N1(C(CC)(C)C)CCN(C(=NC2CC2)NCc2ncccc2Br)CC1 96006,C(=O)(C(O)P(C)(C)=O)N1CC2C(C(N3C(C)(C(=O)NC)CC3)=O)C2C1 96007,C1(NC(c2c(NC)snc2C)=O)CCCN(C(=O)C(C)CC(C)C)CC1 96008,c1(C(N2CCC(C(=O)NCCCOC)(CO)C2)=O)cc(C#N)[nH]c1C 96009,C1(C(=O)NC(c2cnn[nH]2)C)CC(O)CN1C(C1CN(C(N)=O)C1)=O 96010,C1(CNC(C(C)N(C(Cc2c(C)scc2)=O)C2CC2)=O)CC2(CCC2)C1 96011,c1(CC)ccc(CC(=O)NC2CCC(C)N(C(c3[nH]c(C)cc3C)=O)C2)cc1F 96012,C(=O)(C1=NOCC1)N1C(C(=O)NC2CCC(CO)C2)CCCC1 96013,C(=O)(C#CC1CCCOC1)N1CC(C(C)NC(CC(C)C)=O)OCC1 96014,Cc1ccc(C2CC2NC(c2c[nH]cc2C(=O)O)=O)cc1 96015,c1(C(C)C)cc(C(=O)N(C2CN(C(=O)CC(C)N(C)C)CC23CC3)C)cc(F)c1 96016,C1(NC(C(F)OC)=O)CN(C(=O)Cc2cncn2C2CC2)CC1O 96017,c1(C(N2CCC(C)(CNC(C3(CC)CCOCC3)=O)C2)=O)cc(C#N)ccc1F 96018,c1(C(N2CCCCC(CNC(C3CC3F)=O)C2)=O)ccc2c3c(cccc13)CC2 96019,N1(C(c2c(C(C)C)cccc2F)=O)CC2CCC(NC(=O)CN3CCC3C)(C2)C1 96020,Cc1ccc(C(=O)N(C2CCN(C(c3cc(Cl)no3)=O)CC2C)C)nc1O 96021,CCC(F)(C(=O)OC)C(=O)N1CC(O)(C(C)NC(C2CN(S(=O)(=O)CC)C2)=O)C1 96022,CC1CN(C(=O)C=Cc2cnccn2)CC(C)CN1C(C12CC1C2)=O 96023,Cn1ccc(C(=O)NC2CC2C(=O)Nc2ccc(C(N)=O)cc2F)cc1=O 96024,C1(OC)CCCN(C(=O)C(CNC(=O)C(COC)N(C)C)CCC)CC1 96025,C12(CNC(CC3(COC)CC3)=O)CCCC(CN1C(c1cncc(C)c1)=O)C2 96026,c1(NC(C2CCCC(C(=O)OC)C2)=O)nn(C)c2ccccc12 96027,c1(OC)ccc(NC(=O)NC2CN3CCC2(C(F)(F)F)C3)c(OC)c1 96028,C1(C(=O)NCCN2CC=CC2)CCN(C(C2CC23CCC3)=O)C12CC2 96029,C1(C(C)(C)O)(CNC(C2CCCO2)=O)CN(C(=O)C(N2CCOCC2)C2CC2)C1 96030,C1(CC(=O)NCC(C(C)C)NC(C2CCC(C(=O)OC)C2)=O)CCCC(C)(C)O1 96031,C(CC(=O)N1CC2(CCOC2=O)C1)(C(C)(C)C)NC(C(CCC)F)=O 96032,C=CCC(F)(F)C(=O)NC1CN(C(c2cc(CC)ccn2)=O)CC1OC 96033,N1(C(c2c(CC)c(C)sc2)=O)CCCCC(CNC(=O)CCC2(C)CC2(F)F)C1 96034,CC1CN(C(c2ccnn2CCF)=O)CCC1CNC(C1CC2(CCOC2)C1)=O 96035,CC1CN(c2nnnn2C)CC2(CCN(C(c3cccc4c[nH]nc34)=O)CC2)O1 96036,Cn1ccc2ccc(C(=O)NC(C)(CNC(C3CC(O)C3)=O)C3CC3)cc12 96037,c1(C(C(=O)NCC2CC2)N(C(C(=O)OCC)CC)C)ccc(C)c(OC)n1 96038,c1(CN(C(C(=O)NCC(c2cccc(Br)c2)C)=O)C)cc(F)c(Br)cc1F 96039,N1(C(C(C(C)C)OCC)=O)CCCC(O)(CN(C)C(c2nc(C)ccc2F)=O)C1 96040,Cc1nn(-c2ccccc2)nc1Cn1cc(C2CN(C(=O)CC3CCC3)C2)nn1 96041,C(C(C(C)(C)C)N(C)C)NC(=O)NCC1(C(C(C)C)O)CC1 96042,c1(C(=O)OC)ccc(C#N)c(Cl)c1.C12CCN(CC1)C(=O)CCC1CCN(C1)C2 96043,C(CCC(C)CC(=O)NC1(CF)CCN(C(=O)CN(C)CCO)C1)=C(C)C 96044,n1(CC)cc(CCNC(=O)C(Cc2cn[nH]c2)NC(=O)CNC(C)=O)nn1 96045,CC(C)CCC(=O)N(CC(O)CN(C(=O)CNS(=O)(=O)Cc1ccon1)C)C 96046,C1(NC(C2CCC(C(F)F)CC2)=O)COC2(C1)CN(C(C1(F)CCCC1)=O)C2 96047,N=c1c(C(=O)NC2CCCC2C#N)c[nH]n1-c1ccccn1 96048,N1(C(Cc2nc(CC)sc2)=O)C2CCC1C(CNC(C1CCOCC1(C)C)=O)C2 96049,C(=O)(C(C)(C)C(=O)N1CCCCC1C(=O)NCC1C2CCCOC12)OCC 96050,Cc1ccc(C2CC2C(=O)NCC(C2CCC2)NC(c2cocn2)=O)o1 96051,C(=O)(CC(F)(F)F)NCC(C)CNC(=O)CNC(=O)Nc1ncccn1 96052,c1(C(N2CCCCC(CNC(C3C(C)C3)=O)C2)=O)ccc2nn[nH]c2c1 96053,Cc1ncc(Br)c(N2CCCCC2C(N2CC3CNCC3C2)=O)n1 96054,CC(C)(CCNC(C1CC12CC2)=O)NC(=O)CNC(C1CCC1)=O 96055,C(=O)(C1=C(C#N)CCC1)NCCCC(C)(C)NC(C1C(CC)OCC1)=O 96056,CC1=NOC(=O)C1CCC(N1CC(COC)(NC(=O)CCc2cc(C)on2)C1)=O 96057,C1(C(N(CCC(=O)NCC2C3COCC23)C)=O)OC2CCC1C2 96058,CC1CC(NC(c2ncccc2Cl)=O)CN1c1cc(C(N)=O)ncn1 96059,N1(C(Cc2scc(C)c2)=O)CCCC(CN(C(=O)CCC(=O)N(C)C)C)C1 96060,CC(C)C(O)C(=O)NC1CCC1CNC(c1ccccc1C(N)=O)=O 96061,c1(NC(COC)=O)ccc(SC(C)(C)C(C)NC(=O)CCNC(=O)CO)cc1 96062,C1(CC=C)(C(=O)N(C)Cc2cc(-c3ccccn3)no2)CCCNC1 96063,N1(C(c2c(C)cno2)=O)CCN(c2nc(C(C)C)ns2)C(CCO)C1 96064,c1(CN=C(NC(COC)C)NC(c2c(C)cccc2C)C)cc(F)c(C)cc1F 96065,C1(C)(C(=O)NCCCNC(C)=O)CCN(C(C2CC(=C3CC3)C2)=O)CC1 96066,c12nc(ncc1F)N(c1ccc(C#N)cc1)C2=O.C1(SC)CCNCC1(C)C 96067,C1(C(N(C(C(N)=O)C2CC2)C)=O)CCC1NC(=O)C=CCON 96068,N1(CC)CCC(NC(C2(CCNC(=O)Cc3ccc(C)o3)CC2)=O)C(C)C1 96069,N1(C(c2ncn(C)c2)=O)CCCC(C2(NC(c3cnc(Cl)c(F)c3N)=O)CC2)C1 96070,c1(OC)nc(N2CCN(Cc3ccc4ccccc4c3)CC2)c2ccccc2n1 96071,c1(OC)ccncc1C(=O)NC(c1nocc1C(=O)N(C1CC1(C)C)C)C 96072,CC(C)CC(C)(O)C(=O)N1C2CCC(C(=O)NCc3cnns3)C1CC2 96073,N1(C(C2CN(C)C2)=O)CCC2(NC(=O)Cc3cc(O)nnc3O)CCCCC12 96074,c1(OC)cc(C=CC(=O)Nc2ccc(F)c(C(F)F)c2)c(OC)c(OC)c1 96075,N1(C(CC(COC)(C)O)=O)CCC(N=[N+]=[N-])(C(=O)NOCC(N)=O)C1 96076,Cn1ccc2[nH]c(C(N3CCC(NC(C4(n5cccn5)CC4)=O)C3)=O)cc12 96077,c1(CNC(CC2N(C)CCC2)=O)ccc(C(=O)NCC(N2CCCC2)C)nc1 96078,C(C(=O)N=c1cc(C)n(C2CC2)[nH]1)=CC1CN(C(C2C(CC)CCCC2)=O)C1 96079,N1(C(CCC)=O)CCC2(CCCN2C(=O)CCc2ccc(OC)cc2)C1 96080,Cc1cccnc1CC(N1CCC(C(F)F)(CNC(c2cc(CF)on2)=O)C1)=O 96081,c1(C(N2C3(CNC(C(CCOC)C)=O)CCC2CC3)=O)cc(Cl)cc(Cl)c1OC 96082,c1(OC)cc(C(=O)NC(C)C(C)NC(=O)CCc2ccnc(C)n2)cc(F)n1 96083,c1(C(=O)NCCCn2cncn2)ccc(CO)nc1.C12(CC1)C(=O)N2 96084,CN1CCC(CC(=O)NC(C)(C)CCCCNC(=O)C2=CCCCC2)C1=O 96085,c1(NC(C(C)NC(=O)NC)=O)cc(NC2CCOC2)c(F)cc1F 96086,Cc1nc(NCCC2(CO)CC2)cc(=NC(C)c2ccc(Cl)c3c2CCCC3)[nH]1 96087,c1(NC(C2CC2NCc2cscn2)=O)cccc(Cl)c1I 96088,c1(C(=O)NC2CCCC(C(C)C)CC2)nc2c(s1)C(CCCN)CCCC2 96089,N1(C(COCCOC)=O)CCC2(CNC(=O)C3=NNC(=O)CC3)CCCCC12 96090,c1(OC)ncnc(OC)c1C(=O)N(C)CC1(NC(C2CCC3CC23)=O)CC1 96091,c1(CN2CCCC(C(N3CCOC4CC34)=O)C2)cnc(Cl)cc1Cl 96092,c1(C(=O)NC2(CC)CN(C(c3ccc(CF)cc3)=O)C2)cccc(NC)n1 96093,Cc1c(C(N2CC(C)(NC(C3OC4CCC3C4)=O)C2)=O)[nH]c2c(Cl)cccc12 96094,c1(C(=O)NCC2CN(C(C3(CC(C)=O)CC3)=O)CC2C)cccc(Cl)c1F 96095,N1(C(CC2(C=C)CCC2)=O)CCC(C2(NC(=O)C(C)O)CC2)C1 96096,c1(ONC=O)cc(O)ccc1O.c1(CC)c(C(=O)NOC(C)(C)C)cnn1C 96097,c1(CC)nn(C)cc1C(N1CCC(C)C1CNC(c1ccn(C(F)(F)F)n1)=O)=O 96098,N1(C(c2cnn(C)c2C#N)=O)CCC2(CCN(C(=O)CC3CC(F)C3)C2)C1 96099,c1(C(=O)NCC(CN(C(c2c(O)ccc(CC)c2)=O)C)C)cc(S(N)(=O)=O)co1 96100,c1(OC)cc(C(=O)CN2CCC(S(N)(=O)=O)C2)cc(Br)c1OC 96101,C1(OC)CCC(CC(=O)N(CCCNC(=O)C(C2CCCCC2)N(C)C)C)CC1 96102,Cc1ccc(Cl)c(N)c1C(N1CCC(CNC(=O)C(C)(F)F)C(C)C1)=O 96103,C=CCCC(C(=O)N(CCNC(=O)CC(=C)Br)CCOCCO)c1ccccc1 96104,C1(c2c(C)cccc2)CCCC(N=c2[nH]c(N(C)CC3CC3)nc3c2CSC3)C1 96105,c1(C(=O)OC(c2ccc(F)cc2F)C(=O)OC)cccc2nsnc12 96106,C1(COC)(CNC(C2(C)CC(F)C2)=O)CCCN1C(=O)CCCCn1ccnn1 96107,CCC(C)(C#N)C(=O)NC1CCCN(C(=O)CCC(C)c2ccccc2)C1 96108,C1(NC(c2cnn(C)c2Cl)=O)CCC2CC1CN2C(c1cc([N+](=O)[O-])c[nH]1)=O 96109,c1(C(=O)NCC(=O)NCCNC(C2ON=C(CC)C2)=O)n[nH]c2ccc(Cl)cc12 96110,Cc1cc(NC(C2CCCCCN2C(c2cccs2)=O)=O)ccc1O 96111,CCCCCCCCN(C(=O)C(CC1CCC1)OCCNC(=O)C(C)OC)CC 96112,C1(C(N(C)CC2(O)CN(C(C(C)n3cnnn3)=O)C2)=O)CCC2(CCC2)C1 96113,N1(C(C(C(C)C)S)=O)CCn2cnc(C3=CCC(C)(C)CC3)c2C1 96114,Cc1cc(N2CCC(NCC3CCN(c4ccccc4)C3)C2=O)ccc1F 96115,N1(C(C(C)OCC#C)=O)CC2(CCN2C(c2ccccc2CO)=O)C1 96116,CCC(C)(CC)C(=O)NCCCCCNC(C1CCCC(C)CC1)=O 96117,C(=O)(C(F)(F)C(O)C1CC1)NCC(C)(C)CNC(c1cc(Cl)ccc1F)=O 96118,C1(C(N2CC3CC(OCC(=O)NCCCOC(C)(C)C)C3C2)=O)CN2CCCN1CC2 96119,CC(C)CN=C(NCC1(c2ccon2)CCC1)N1CC(C)S(=O)(=O)C(C)C1 96120,CCC(CC(C)C)C(C(=O)NCCCCCCl)N1CCCCC1C(=O)NC 96121,C(CC(C)C)(C(=O)N1CCC(CNC(c2ccc(Cl)cc2C)=O)C1)NC(=O)OC 96122,C1(CNC(CC(C)N(C)C)=O)CN(C(c2n[nH]c3c2COCC3)=O)CC(C)(C)O1 96123,CCCC(C(C(=O)NCc1ccccc1)N1CC(O)C2(CC2)C1)OC 96124,c1(CC(N2CC(=C(CNC(C(CC)n3ccnc3)=O)F)C2)=O)ccc(F)cc1C 96125,C(CC(C)(C)C(=O)NCC(C)(C)CCNC(=O)CC1CCCNC(=O)C1)OC 96126,N1(C(C(CC)n2cccn2)=O)CC(N(C(=O)CC2CC(C(=O)OC)C2)C)C(O)C1 96127,N1(C(C2CC=C(C)CC2)=O)CC2(CCCC2NC(C2(C3CCC3)CC2(F)F)=O)C1 96128,c1(C(N2CCC(=CC(N3CCC34CCCCC4)=O)CC2)=O)c(F)cc(F)cc1Cl 96129,C1(CN(C(=O)C(C)COC)CC)CCN(C(c2cnn(C)c2SC)=O)CC1 96130,C1(C(N(C)CC2(O)CCC2)=O)CCN(C(c2ccccc2)=O)CC1 96131,CC(C(=O)N1CCC(n2cc(-c3ccccc3F)nn2)CC1)C(F)F 96132,N1(C(C(CCC)O)=O)CC2(CCN(C(=O)Cc3ccc(Br)cc3F)CC2)C1 96133,N1(C(COc2c(Cl)ccc(C)c2)=O)CC2CN(C(C3CCCCO3)=O)CCC12 96134,N1(C(C=CC=CCC)=O)CCCC2(NC(=O)OCC(F)(F)F)CCCC12 96135,c1(C(N2CC=CC(NC(COCC(C)C)=O)C2)=O)cn2ccncc2n1 96136,N1(C(Cn2cnc(=N)[nH]2)=O)CCC2(NC(c3ccc4nc[nH]c4n3)=O)CCCC12 96137,c1(C(N)C(=O)NC2(CC(=O)O)CC2)ccc(Br)c(F)c1 96138,c1(C(=O)NC2C(C(N(C(CC(C)C)CO)C)=O)OCC2)ccc([N+](=O)[O-])[nH]1 96139,c1(C(=O)NC(CN2CC(C)CC(C)C2)C)nc(Cl)c(Br)cc1[N+](=O)[O-] 96140,c1(C(N2CCC(CCOC)C2)=O)n[nH]c2c1CN(C(=O)CCc1cccnc1)C2 96141,N#Cc1ccc(F)cc1C(=O)NCC1CCN1S(=O)(=O)CC1CCC1 96142,CC1C(NC(=O)CC2=CCN(C)CC2)CC2CCC1N2C(C1CCCOC1C)=O 96143,C12(CNC(c3cccc(C)n3)=O)CCCCC1N(C(c1ccc(O)cc1)=O)CC2 96144,c1(C(N)=O)cc(Cl)ccc1S(=O)(=O)N1CCC(Cc2ccc(Cl)cc2)C1 96145,CN1CC(C(=O)NC(c2nc[nH]n2)Cc2ccccc2)c2ccccc21 96146,c1(OC)ccccc1C(F)(F)C(=O)N(C)CCNC(c1cc(Cl)ncn1)=O 96147,CCCS(=O)(=O)CC(=O)NC1CC2(C1)CN(C(=O)C(C)(O)C1CCOCC1)C2 96148,C1(C(N2CCC(OC)(CNC(=O)C(C)n3cccn3)C2)=O)CC(=O)CC(=O)C1 96149,c1(C(=O)NC(CNC(c2c(C(C)C)c[nH]n2)=O)(C)C)ccc2c(c1)C(C)C(C)O2 96150,C1(CNC(CC2(CSC)CC2)=O)CC12CCN(C(c1c(C)nsc1Cl)=O)CC2 96151,CN1CCOCC1CNC(C1(NC(C2CCCOCC2)=O)CCCCC1)=O 96152,C1(NC(CCOC)=O)CCCCC12CCCN(c1nnco1)C2 96153,N(C(=NCCOC(F)F)NCC(Cc1ccccc1)C(C)C)CC(CC)(C)C 96154,c1(NC(CC2N(C(c3c(C)nc[nH]3)=O)CCC2)=O)cc(F)cnc1Br 96155,C1(C(=O)NCC(C)NC(c2c(CCC)n[nH]c2)=O)CC12CCC1(CC1)CC2 96156,Cc1cc(C(N2CC(C(O)C(N3CCCC(CCCO)C3)=O)C2)=O)nc(C)n1 96157,c1(CCC)ccc(N)c(NC(=O)COC2CCN(C(=O)C3=CCCC3C)C2C)c1 96158,CC(F)(Cc1ccccc1)C(=O)NCC1CCN1C(c1nc(=N)cc[nH]1)=O 96159,N(C(=NCC(C)C)N1CCN(Cc2ncoc2C)CC1)C(COC)C 96160,C1(C(=O)NCCCN(C)C2CC2)CC=CCN1C(=O)CC1CCOC1 96161,C1(NC(COCCNC(C(n2c(C)ccn2)C)=O)=O)CCC(C(C)C)CC1 96162,CC(CC(N)=O)C(=O)NC(CC(N)=O)C(=O)NC(C)CCO 96163,N1(C(CC=C=C)=O)CCN(C(=O)C=Cc2ccc(-c3ccccc3)s2)C(CO)C1 96164,c1(N(C2CNCC(C)C2)C(CCc2cccc(C)n2)=O)nccc(C#N)n1 96165,C1(C(N(C2CCN(C)CC2)CCO)=O)CC2CCN(C(=O)Cn3cccc3)CC12 96166,C1(C(=O)Nc2c(COC)nn(C)c2)N(C(C2CC=C(C)CC2)=O)CCC1(C)C 96167,N1(C(c2c(CNC(CC(C)C3CCCO3)=O)n[nH]c2)=O)CCC2(CCN(C)C2)C1 96168,c1(C(N)=O)ccc(S(=O)(=O)NC2(Cc3nccs3)CCC2)cc1C(=O)O 96169,c1(C(=O)Nc2ccc(CN(C)CC)cc2)cc(Br)cc(Cl)c1Cl 96170,C1(C)(C(N2CCC(C(=O)NC(CCC(C)C)C)CC2)=O)CCC2CC2C1 96171,c1(C(=O)NC(C2COCCN2C(=O)CC2CCOC2)C)cccc(Br)c1 96172,N1(C(C2N3CC(C)N(CC3)C2)=O)CCCC2(CCCN2C(C2CC23CC3)=O)C1 96173,c1(NC(c2n(C)cc(Nc3ncc(Br)cn3)n2)=O)c(F)cccc1I 96174,C1(C(=O)NC2(C)CC(C(=O)NC3CC3c3ccsc3)C2)CN2CCN1CC2 96175,N1(C(CCC(=O)NC)=O)CC(C)CN(C(c2cnccn2)=O)C(C)C1 96176,C(c1csc(C)n1)=CC(=O)NC(CCNC(c1n(CC)cnn1)=O)C 96177,c1(NC)cnccc1C(=O)N(C1CCN(C(=O)CC2(C)CCOCC2)CC1)C 96178,c1(CC(C(=O)NCCNCC)NC(=O)OC(C)(C)C)cc(Cl)sc1Cl.CCOC 96179,c1(C(C)NC(CN(C(CCCN(C(C)=O)C)=O)CC(C)C)=O)cccnc1C 96180,N1(C(CCn2cc(-c3cc(C)c(N)cc3)nn2)=O)CC(N=[N+]=[N-])CC1CO 96181,C1(CNC(CC=CC)=O)CN(C(C2CCCC2CC)=O)CC1C 96182,c1(C(=O)NC2CCCN(C(c3cnc(CC)[nH]3)=O)C2)c(C)ccc(C)c1N 96183,c1(C(=O)NC(CNC(CSCC#C)=O)CCOC)cnc2c(C)cccc2c1 96184,CC(CCNS(=O)(=O)Cc1ccnc(Cl)c1F)P(C)(C)=O 96185,N1(C(CSCC)=O)CC(C)(C)OC2(C1)CN(C(C1C3CS(=O)(=O)CC13)=O)C2 96186,C1(C)(C(N(CC(C)O)CCNC(=O)Cc2ccno2)=O)CCC(=O)N1 96187,c1(CC)nc(CC(=O)NCC2CCCC2NC(=O)COc2ccsn2)n[nH]1 96188,N1(C(=O)CCOc2ccccc2C(F)F)CC2(CCN2C(C2CC2Cl)=O)C1 96189,C(c1scnc1C)=CC(=O)N(CC(C)(C)NC(c1c(CCC)occ1)=O)C 96190,c1(C(=O)NC2C(NC(c3cc(Cl)cs3)=O)COCC2)ccc(F)c2c1CCC2 96191,C(=O)(CC1=CCOCC1)N1CCC(O)(C(C)NC(=O)Cc2c[nH]nc2O)C1 96192,Nc1ccc(C(=O)NCC2CCN(C(C3CC(F)C(=O)N3)=O)C2)cc1F 96193,C1(CNC(c2cccc(NCC(F)(F)F)c2)=O)OC(=O)C2(C(=O)O)CC12 96194,n1(CC(=O)NC(CC(C)NC(=O)CSCC(F)(F)F)C)nc2n(c1=O)CCOC2 96195,CC1CC=C(C(=O)N(CCCN(C)C)CCNC(=O)CCCc2ncco2)CC1 96196,Cc1ncc2cc(C(N3CCC(c4nc(C5CC5)no4)CC3)=O)c(O)nc2n1 96197,c1(COC)nn[nH]c1C(=O)N(CCC(C)NC(C1(OC)CC1)=O)C 96198,CCC(C)CCCCC(=O)N1CCC(NC(c2cnc(N(C)C)cn2)=O)CC1C 96199,N1(c2snc(C(C)(C)OC)n2)CCOC(CNC(C2CC(=O)N2)=O)C1 96200,c1(C(=O)OC)nc(=NCC(CO)NC(=O)C(O)C2CC2)c2c([nH]1)CCC2 96201,C1(C(N(CC(CC)NC(=O)CCNC(N)=O)CC)=O)OCC2COCCC12 96202,Cc1nc(C(C)C)nc(O)c1C(=O)NC1CCCCC1NC(C1CC2(CC2)C1)=O 96203,C1(CCNC(COCCN(C)C)=O)CN(C(=O)Cc2cncnc2)CCO1 96204,C1(NC(CCCN(C(=O)CCC(F)(F)F)C)=O)CC2CCC(C1)N2C 96205,C1(C2CCOCC2)(C(N2CC3(CN(C(C4CC4F)=O)C3)OCC2)=O)CCOCC1 96206,CC1CCc2onc(C(=O)N(CC(C)NC(c3ccc(Cl)cn3)=O)C)c2C1 96207,C(C(N=[N+]=[N-])C(=O)NCC1(C(=O)NCC(C2CC2)OCC)CCCC1)OCC 96208,c1(CN(CCC)CCO)cncc(-c2ccc(CN(C)C)cc2)c1 96209,C=CCCC(O)CN(C(=O)C(c1ccco1)NC(c1cnc(O)o1)=O)C 96210,C#CCC(C)(C)C(=O)N1CC(N(C)C(c2cc(C#N)ccn2)=O)C2(CC2)C1 96211,C1(CC=C)(NC(COCCC=C)=O)CN(C(c2cc(Br)cs2)=O)C1 96212,C(C(C)N(C)N1CCCC1C1CCCCN1CC(F)F)c1c(C)cccc1 96213,O(N=C1CCCCCC1)CC(=O)NCC#CCNC(c1csc2ccccc12)=O 96214,c1(C(N2C(CNC(CCC)=O)C(C)CC2)=O)ccc(F)c(OC)c1F 96215,c1(NC(C)CCNC(C2CC2(F)F)=O)nnccc1C#N 96216,N1(C(CCCOC(C)C)=O)CC(C)C(C)(CNC(c2ncc(CO)[nH]2)=O)C1 96217,c1(C(=O)NC2CC(NC(CCc3c(OC)cccc3)=O)C2)nc(Cl)ccc1N 96218,N1(C(C(c2cccc(Cl)c2)C)=O)CC2CC(C1)N(C(=O)C(O)CCN(C)C)C2 96219,N1(CC(=O)NC(C)C)CCC(NC(c2ccsc2C(F)F)=O)C(C)C1 96220,C1(C(=O)NC2CC(C(C)C)OC2)CN(C(C2CCCSC2)=O)CC1F 96221,C1(C(=O)NC23CC(NC(C(C)c4ccco4)=O)(C2)C3)CN2CCN1CC2.C12CC1C2 96222,Cc1nc2cc(C(=O)NC3CN(C(=O)CC4CC4)CC(C)(C)C3)cc(O)c2[nH]1 96223,C1(C(N2CCC(C)(C(N3CC(C(C)C)OCC3)=O)C2)=O)CC2CC(=O)C1O2 96224,O=C(NNC(=O)c1ccc(N2CCCC2=O)nc1)C1CSCN1C(=O)C(F)(F)F 96225,CC(C)CCCC(C)C(=O)NCC1CN(C(c2ccc(SC)o2)=O)CCCO1 96226,N1(C(C(CCC)N(C)C)=O)CC2CN(C(c3cnc(OC)nc3OC)=O)CC12 96227,c1(C(=O)NC2CCC(C)(NC(C3CCCCO3)=O)CC2)cc(F)c(F)c(F)c1 96228,C12(NC(C3CCS3(=O)=O)=O)CCCN(C(c3cc4ccsc4s3)=O)CC1C2 96229,c1(N2CC(CC=C)(NC(c3cc(C4(C)CC4)on3)=O)C2)nc2ccc(Br)cc2o1 96230,C1(NC(C2(COC)CC=CC2)=O)CC(O)CN(C(c2c(OC)ccnc2O)=O)C1 96231,CCCC(C(=O)N(C)CCNC(=O)C=CC1CCCO1)S(N)(=O)=O 96232,C(=O)(CC(C)C(C)C(C)C)N1CCC(NC(c2cn(CCC=C)nn2)=O)C(C)C1 96233,C(CC(C)C)(C(N)=O)NC(c1n(CC=C)nnn1)c1cnc(-c2ccccc2)s1 96234,CC(C)CC(CC(=O)NC(C(N)=O)C1CC1)NC(C1COCCC1C)=O 96235,C(=O)(CCC(=O)c1cccnc1)NCCCC(C)NC(=O)C(F)n1cccn1 96236,CC(C)(C#N)C(=O)NCCCOCCCNC(C1CC(O)(c2ccccc2)C1)=O 96237,N1(C(CCCC(=C)C)=O)CC2(CCN(C(=O)C(C(C)(C)C)N(C)C)CC2)CC1C 96238,C12(F)CCN(C1)C2=O.c1(N(CC(=O)NC)CC)ccc(Oc2cccnc2)cc1 96239,C12CCCCN(C1)C2=O.C(CCCC(=O)NCC1(C2CC2)CCC1)N(C)C 96240,N1(C(CCCN(C(C)=O)C)=O)CCOC(CNC(C2COCCN2C(C)=O)=O)C1 96241,C1(NC(CCC(C)C)=O)CN(C(C2CCCN(S(C)(=O)=O)C2)=O)CCC1C 96242,c1(C(=O)NCC2(NC(=O)C=CI)CCCCC2)ccc2nc(O)[nH]c2c1 96243,c1(C(N2CCC(OC)(CNC(c3ccc(C)nc3O)=O)C2)=O)ccc(N)c(O)c1 96244,C12CCCC(C1)CNC2=O.C(C(=O)N)(c1cccs1)N(C)C.C1(NC(N)=O)CC1 96245,C(=O)(C1CCCc2nn[nH]c21)NCCC1CC(NC(=O)C=CCF)C1 96246,C(CN=C1NC2COCC2N1)NC1c2cc(Br)sc2CC1 96247,N1(C(COC)=O)C2CCC1CN(C(c1ccnc(N(C)CC3CC3)c1)=O)C2 96248,N1(C(c2n(CC)ncc2)=O)CC(CCNC(=O)C(=O)NCC(F)F)OC(C)C1 96249,C1(N(C)C(C2CCC(=O)C2)=O)CCCN(C(=O)CCCN2C(=O)CNC2=O)CC1 96250,C1(CNC(C(C)C)=O)CCCCN(C(c2ccc(O)nc2Cl)=O)C1 96251,C1(C2CCC2)(C(=O)NCC2C(NC(c3cccc(C(F)F)n3)=O)CC2)CC1 96252,c1(C(=O)NC2CC(CNC(C(C=C)(C)C)=O)C2)sc2ccc(C(C)=O)cc2c1C 96253,C1(CCNC(CC2(CC)CCC2)=O)(NC(c2cnc(OC)s2)=O)CCCC1 96254,c1(OC)ccc(F)cc1CC(=O)NCC1CC(C)N(C(c2cnncc2O)=O)C1 96255,Cc1cccc2[nH]c(C(=O)NCCC3CCCCN3C(C3(C)CCCS3)=O)cc12 96256,C1(NC(c2n(CC)ccc2)=O)CC2CC(C1)N(C(=O)C(Br)=C(C)C)C2 96257,C(c1nc2ccccc2s1)=CC(=O)OCC(c1cc(C(N)=O)c(O)cc1)=O 96258,C1(C(N(C)Cc2c(C)nn(C)c2)=O)CCN(C(=O)C(C)n2cncn2)C12CCC2 96259,N1(C(c2cc3cc(Cl)ccc3o2)C(=O)NCCOC)CCOc2ccccc2C1 96260,Cc1nn2c(c1CNC(C1(n3nccn3)CC1)=O)CN(C(c1ccco1)=O)CC2 96261,N1(C(c2ccc(OC)c(C)c2)C(=O)NC2CCCC2)CCC2(CC(=O)N(C)C2)C1 96262,c1(OC)ccc(CC(N2CCCC2CC(N2CCC(F)C2)=O)=O)c(OC)c1 96263,Cc1cc(C(=O)NC2CCN(Cc3cncc(C(F)(F)F)c3)C2)c(F)c(Br)c1 96264,N1(C(c2[nH]cc(C)c2C)=O)CC(NC(=O)CC2CCCOC2)CC1(C)C 96265,CC1CCC(C(N)CN(C(=O)OCC=O)Cc2cnnn2C)CC1.C(C)(C)C 96266,c1(C(N2CCC(NC(c3cc(Cl)cc(F)c3F)=O)C2)=O)cccc2cc[nH]c12 96267,CC1=C(C(=O)NCCNC(=O)C(C)N(CC(F)(F)F)C)S(=O)(=O)CCO1 96268,C1(CN(C)C(C2CCC3CC23)=O)CCCN(C(=O)CN(C2CCS(=O)(=O)C2)C)C1 96269,C1(NC(C(C2CCOC2)OC)=O)CCC2CC1CN2c1ncnc2[nH]cnc12 96270,C(=O)(C1COc2ccc(Cl)cc21)C(N1CCn2c(C)nnc2C1)=O 96271,c1(C(c2nnnn2C)NC(c2cccc3cc[nH]c23)C)nc2c(s1)CCCCC2 96272,S(=O)(=O)(c1ccc(Cl)cc1F)N1C2CN(Cc3ccc(C)o3)C(C2)C1 96273,c1(C(N(C2CN(C(C3(C)CCCCO3)=O)C2)C)=O)coc(S(C)(=O)=O)c1 96274,N1(C(c2c(OC)nsc2)=O)CCN(C(=O)CCN2CCCC2)C(CC(C)(C)C)C1 96275,c1(C(=O)NCC(C)(CO)NC(C(CC=C)CC=C)=O)cccc2cccc(C)c12 96276,c1(C(C(=O)NCC2CC(NC(CSCC(N)=O)=O)C2)=O)ccc(Cl)cc1Cl 96277,C1(CC(=O)NCCOC(C)=O)C=CC(NC(=O)C=Cc2ccsc2)C1 96278,c1(CC)cc(OC)ccc1C(=O)NC1CCN(C(=O)C(C)C(C)C)C1.C(C)(=O)O 96279,C#CCCCCCCCC(=O)NCC1CC(CNC(=O)CC(C)C(C)(C)C)CO1 96280,c1(OC)nccnc1CNC(c1csc(C(=O)NCCc2ccncn2)n1)=O 96281,Cc1ccc(C)c(CC(=O)NC2CN(C(C34CC(CO)(C3)OC4C)=O)C2)c1 96282,C#CCC(C(=O)NC1CC1NC(C1CN(C(=O)N(C)C)C1)=O)C1CC1 96283,C1(CC=C)(NC(=O)CCCC(C)=O)CCN(C(=O)CSCCN(C)C)CC1.C(N)=O 96284,C1(CCC)(NC(=O)CCOCCCOC)CCN(C(=O)C(C)CC(C)C)CC1 96285,CC1(C)CC(C(=O)NC2CCN(CCF)C2)CN1C(=O)CCC(=O)c1ccc[nH]1 96286,c1(C(N2CCCC(CC)(NC(=O)NC(C)(C)C)C2)=O)ccc2ccc(O)cc2c1O 96287,c1(OC)ccc(C(N2CCCC(CNC(=O)CCc3ccoc3)C2)=O)c(Br)c1 96288,c1(C(N2C(CNC(C(c3ccc(Cl)cc3)SC)=O)C=CC2)=O)ccncc1SC 96289,N1(C(Cc2c(C)noc2C)=O)CCCN(C(=O)Cc2c(F)cccc2F)C(C)C1 96290,c1(C(N(CCNC(C2C(C)C2)=O)CC2CC2)=O)cnn(CCc2ccccc2)c1 96291,CC1(C)OC(=O)CC1C(N1CCC12CN(C(=O)Cc1ccc(Br)cc1)C2)=O 96292,C1(N2CC2=O)CCN(C(c2ccnnc2)=O)CC1.C12CC(C1)N2C.C(C(C)C)S.CO 96293,c1(CC)oc(C)cc1C(N1CC2CC2(CNC(c2sc(C)cc2OC)=O)C1)=O 96294,C1(OC)CCCC1n1cc(C(CC)NC(c2csc(C(F)(F)F)n2)=O)nn1 96295,C1(C(C(=O)O)NC(C(COC(C)=O)C)=O)C2CC3CC(C2)CC1C3 96296,c1(C(=O)NC2(C)CC(NC(c3ccc(CO)o3)=O)C2)cnc2scnc2c1 96297,CC(CC(F)F)C(=O)NCCC=O.c1(CC(=O)NCCO)sc(O)nc1O 96298,C(=O)(CCCCC(N)=O)NCC(S(C)(=O)=O)CNC(C1CC1Cl)=O 96299,Cc1cccc2ncc(C(N3CCC(C)CC3CNC(c3c[nH][nH]c3=N)=O)=O)n12 96300,C1(CNC(CC(=C)C)=O)CCC2(CO1)CC(NC(=O)C=CC1CCC1)C2 96301,N1(C(=O)OC(C)(C)C)CC(C(=O)Nc2ccc(Cc3cncs3)cc2)C2CC12 96302,CCCC(C)(CC)NC(C1(NC(=O)CNC(=O)CC(C)C)CCN(C)C1)=O 96303,C(C(F)(C(=O)NC1(C(=O)NC(C)C)CC1)C(C)C)NC(C(CC)(C)C#N)=O 96304,C(=O)(C1CCCc2c[nH]nc21)NC1C(CC)N(C(=O)C(C)C(C)(C)C)CC1 96305,Cn1nccc1C(F)=CC(N1CCC(NC(=O)Cc2ccon2)C1(C)C)=O 96306,C1(NC(=O)C=Cc2cnc[nH]2)CC2(C1)CC(C(=O)NCC1CCC(F)(F)C1)C2 96307,c1(C(=O)NCC(CNC(c2c(CC)nc(C)[nH]2)=O)F)cc(O)cc(F)c1 96308,c1(CNC2C(OC(C)C)CCCCC2)cn(C)[nH]c1=NC(=O)OC(C)(C)C 96309,N1(C(CC2CCN(C(C(C)Oc3ccccc3)=O)C2)=O)CC2COC(=O)C2C1 96310,N1(C(C2CC23CC(OCc2ccc(O)cc2)C3)=O)CCC(F)(F)C(O)C1 96311,N1(C(c2noc(CC)c2C)=O)Cc2occ(C(=O)NCCC3CC(F)(F)C3)c2C1 96312,Cc1cc(F)c2nc(O)cc(C(=O)NC3CCCN(CC(F)F)C3)c2c1 96313,c1(C(=O)NC2C(F)CCN(C(CCC(C)=O)=O)C2)ccc(Cl)c(C)c1F 96314,C(=O)(NN1CCCN(C)CC1)c1c(C)ccnc1 96315,c1(CC(=O)NC2CC(C)N(C(=O)COCC3CCCOC3)C2)csc2nccn12 96316,c1(C(=O)NC2CC(NC(C3(C(F)(F)F)CC3)=O)C(O)C2)cnc2c(F)cccn12 96317,N1(C(c2cc(CC)oc2C)=O)CCC(C2CC2)C1CNC(c1ccc(=O)oc1)=O 96318,c1(C(N2CCCCC(C(N3CC(CC)N(C)CC3)=O)C2)=O)cccc2[nH]ncc12 96319,C1(OC(c2n(C)nc(Br)c2)=O)C2CC3C(=O)OC1C3O2 96320,C1(NC(CC(=C)C)=O)CC2C(NC(C3CC(=O)N(C(C)C)C3)=O)C2C1 96321,C(C(C)(C)C(=O)N1CCC(C)C1)NC(C1(CC(=O)OCC)CC1)=O 96322,c1(C(=O)NC(CC=C)CNC(=O)C(C)CCC)cccc([N+](=O)[O-])c1O 96323,c1(C(=O)NCC2CN(C(C3N(C(C)C)CCC3)=O)CC2O)onc2c1CCCC2 96324,c1(OC)ncc(F)cc1C(=O)NC1CC1NC(=O)CSC(C)(C)C 96325,N1(C(Cn2c(C)ncc2)=O)CCn2cc(C(N3CCC4(CCCO4)C3)=O)nc2C1 96326,N1(C(=O)NCc2nc(C3OCCO3)cs2)CCOc2c(F)cccc21 96327,N12CCN(CC1)C1CCN(C1)CC2=O.CC(Cc1ccccc1)C(=O)OCC#N 96328,C1(O)(CCNC(C(=O)NC(C)C)=O)CN(C(=O)C(C)CC2CCCCC2)C1 96329,N1(C(c2c(Cl)cnc(C)n2)=O)CC2(CCC2)CC1CNC(=O)CCc1ccon1 96330,C1(NC(c2cnccn2)=O)CCC2(CC1)CN(C(c1ccoc1Cl)=O)CCO2 96331,c1(CNC(Cn2cc(C3(C)CC(OC)(OC)C3)nn2)=O)ccc2nsnc2c1 96332,n1(CC(=O)NCCCN(C(C2C(CC)CC2)=O)CC)ncccc1=O 96333,C1(SC)CN(C(=O)Cn2cnc(=N)[nH]2)CC1NC(C1(C)CCCO1)=O 96334,C12(CNC(CSCC=C)=O)CC1CN(C(c1cc(C3CC3)nn1C1CC1)=O)C2 96335,N1(CC(COC(COC)C)O)CC2C3CCC(C2C1)N(C(C1COCCO1)=O)C3 96336,C#CCCCC(=O)N(CCCCCNC(=O)C(CC)NC(N)=O)CC 96337,C1(NC(C(C)c2ccco2)=O)CCC2CC1CN2C(=O)CC1(C)CCOCC1 96338,c1(NC(N2CCC(CCC)(CO)C2)=O)cc(O)nc2cnccc12 96339,C(=O)(CC(O)C(Cl)(Cl)Cl)N1CCC(OCC(=O)N(c2ccn(C)n2)CC)C1 96340,C1(CC(=O)NCCCCCCN(C(=O)C=Cc2cnccn2)C)CCC(=O)NC1=O 96341,O=C1CN(C(=O)CCc2nc(O)n[nH]2)C(C(=O)NC2CCC3(CC3)C2)CN1 96342,C(=O)(C1CSc2ccccc21)NC(CNC(c1cccc(S(C)=O)c1)=O)(C)C 96343,C1(C(=O)NC2CC3(C(NC(CSCCOC)=O)C3)C2)CCc2nn[nH]c2C1 96344,c1(OC)ccc(F)c(C(=O)NC2CN(C(=O)COC3CCC3)CCC2CO)c1Cl 96345,C1(C(=O)OC)CCC(CC(=O)NCCCNC(c2cccn2C)=O)CC1 96346,CC1(C(=O)NCCC2(O)CCN(C(=O)CC3CSC3)C2)CCC(F)(F)CC1 96347,C1(C)(CC(=O)NC2(CC(=O)NC3CC(OC)C3)CCC2)CCCCC1 96348,C1(C(=O)NCCCC(C)(C)NC(CN(CCOC)C)=O)CCC2(CC1)CC2(F)F 96349,c1(-n2cc(C(C)N(C)C)nn2)ccccc1C(=O)N(C(C)CCO)C 96350,CCC(C(=O)OC)C(=O)N1CCCCC1CCNC(=O)CSc1n[nH]c(C)n1 96351,C(C)(c1ccc(F)cc1F)=CC(=O)N(CC)CC1CCN(C(=O)C(C)OC)CC1 96352,C#CCCCCC(=O)NCc1ccc(C(=O)NC(CCC)C(F)(F)F)cn1 96353,C12(CC(N3CC(C)C(CNC(C4CCCOC4)=O)C3)=O)CCC(CC1)OC2 96354,C1(OC)CC(C(=O)NCC2(n3ccnn3)CC2)N(C(=O)CCc2cn[nH]c2)C1 96355,c1(C(=O)NNC(c2cc(F)ccc2F)=O)cc(F)c(Br)c(F)c1 96356,N1(C(C2CC(C)=C(C)CC2)=O)CCC(C)(C)CC1C(=O)NCc1ccnc(O)c1 96357,C1(NC(C)=O)CC(NC(c2ccc(OC(F)F)cn2)=O)C1(C)C 96358,c1(C(=O)NC2C(NC(C3(C#N)CCCO3)=O)COC2)cc2ccncc2s1 96359,S(=O)(=O)(CCCCF)NC(C1(N)C2CCC12)=O 96360,CC#CCC(C)N=c1[nH]c(=NC)[nH]c(=NCc2sccc2S(C)(=O)=O)[nH]1 96361,c1(NC(=O)NCc2ccc3nonc3c2)cc2cccnc2c(Br)n1 96362,N1(C(C2CC3CC2C2CC32)=O)CC2CCC1CN2C(C1CCS(=O)(=O)N1)=O 96363,C1(C(N(CCF)CC)=O)C2CCCC2CN1C(c1cnn2c1CCC2)=O 96364,N1(CCC(=O)NC(CC(C)NC(Cc2ccn(CC)n2)=O)C)CCN(C)CC1 96365,N1(C(c2n(CC)ncc2Cl)=O)CCC(C2CCN(C(=O)C(C)=C3CC3)C2)C1 96366,Cc1coc(C(C)C)c1C(=O)NCC1CN(C(=O)C(C)OCCC(C)C)CCO1 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96456,CCC(CC)CC(=O)NC1CCCCC1NC(=O)C(C1CCCC1)OC 96457,c1(CCCC=C)cn(C2CC2CNC(C2CCC2c2ccccc2)=O)nn1 96458,C1(CNC(Cc2cc(C)sc2)=O)(NC(=O)CC2CCCN(C)C2)CCN(C)C1 96459,c1(C(=O)NCCN(C(C(=O)NC)=O)CC(C)O)cnc(-c2ccccc2)[nH]1 96460,C1(CC(=O)N)CCCCN1C.C(C(=O)N)=CC=CCC.C1CCN(C)CCOCC1 96461,c1(C(=O)NCCC(C)N(C(CC(CC)O)=O)C)[nH]nc2ncnc(O)c12 96462,N1(C(CN(C(CO)C2CCC2)CC)=O)CCCCC1CC(=O)NCC(C)C 96463,N1(C(Cc2ncn(C)c2)=O)CC=C(C(=O)NCCC2CCCC3CC23)C1 96464,CC(CC(=O)N1CCCCC1CCNC(C12CC(CC(F)F)(C1)C2)=O)C(C)(C)C 96465,c1(N(C)Cc2ccccc2)nc(=NCC2COCC(C)(C)O2)[nH]c2c1CCCC2 96466,C(C(=O)NCC(C)(Cl)CC)(C(C)O)NC(C1C(=C)C1)=O 96467,CC(C)CC(=O)N(CC(=O)NC(C)CCC1CCCO1)CC1CC1 96468,NC(=O)CC(O)C(=O)NCCC1(NC(=O)COC2CCCCC2)CCC1 96469,CC1CCn2ncc(C(N3CCC(C)C(NC(=O)C(F)C(C)(C)O)C3C)=O)c2C1 96470,C(=O)(C(F)(F)C1(O)CCC1)NCCCCN(C(C(N1CC(C)C1)C)=O)C 96471,c1(C(N2CC(C(=O)OC)OCC2)=O)cnc2[nH]cnc2c1 96472,CCCCC(O)C(C)C(=O)NC1CC(N(C)C(c2c[nH]nc2Cl)=O)C1 96473,N1(C(CC(CC)C)=O)CC2CC(NC(=O)CC3CC(C(F)F)C3)CC2C1 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96526,c1(CC(=O)NC2CCCCC2NC(C2CC3C=CC2C3)=O)cccnc1Br 96527,C1(OC)CC2CC(C(=O)Nc3cccc(CNC(=O)C=CCF)c3)CC12 96528,c12n[nH]c3cc(ccc13)NC1CN(c3cc(ncn3)C(=O)NC2=O)C1.CC=CC 96529,c1(-n2ccc(C(=O)NCC3CC(NC(C=NOC)=O)C3)n2)cccc(F)c1 96530,Cc1ccc2c(Nc3ccc(C(N4CCC(F)CC4)=O)nc3)ncnc2c1 96531,C(c1ccc(S(C)(=O)=O)o1)=CC(=O)NCCC(CCNC(C1(C#C)CC1)=O)C 96532,CC1CN(C(c2ccc(=O)[nH]n2)=O)CC(CCNC(c2ccnc(O)c2F)=O)O1 96533,c1(-n2c(Cc3onc(C)n3)nc(C3CCC(C)CC3)n2)cccc2ccccc12 96534,c1(NC(c2cc(NC(=O)C(=O)NC3CC3)cc(F)c2)=O)cccc2c1OC(F)(F)O2 96535,n1(CCC)cc(C(=O)N(CCN(C(=O)C(C)n2cccc2)CC)CC)c(C)n1 96536,C1(C(=O)NCC2CCCC(NC(c3ccncc3F)=O)C2)(SC)CC(F)(F)C1 96537,CCCC(CCC)CC(=O)NC1CC(CCNC(=O)CNC(=O)C(C)(C)C)C1 96538,CP(C)(=O)CCC(=O)N1CCCCC(CCC(=O)NC2CC3(CCC3)C2)C1 96539,CCC(C)(F)C(=O)NCCN(C(=O)CNC(c1ccncc1)=O)CCOCCO 96540,N1(C(CSCC(C)C)=O)CCC(CC(=O)N(C)CC2CC2C)C1(C)C 96541,c1(CCC(=O)NC2C(CNC(Cc3cc(C)sc3)=O)C2)cnc2ccccc2c1 96542,N1(C(CC2(C=C)CC2)=O)CCOCC(CNC(c2c(C(C)C)cccc2C)=O)C1 96543,C(=O)(C1CC(=O)Nc2ncn(C)c21)N1CC(C)N(C(c2ccc(F)s2)=O)CC1 96544,c1(C(=O)NCC(C2CCC2)NC(C2CCOC2)=O)cc(Cl)cc(C(F)(F)F)n1 96545,C1(C(N2CC(CCNC(=O)C(C)N(C)C(C)=O)(OC)C2)=O)CCNC(=O)C1 96546,c1(SC)ncc(C(=O)NCC2CCCC2NC(=O)C(F)C(C)(C)O)c(O)n1 96547,c1(CC)ccc(C(N2CCC(C(=O)NCC3CCC(F)(F)C3)C2)=O)cc1 96548,N1(C(CN(C(C)=O)C)=O)CCCCC(CNc2ncc(C)c(C)n2)C1 96549,C(=O)(C1OCCn2ccnc21)NCCCN(C(C(CC)(C)O)=O)C 96550,C=CCCC(C(=O)NC1CC(C)OC1=O)NC(c1ccc(C)nn1)=O 96551,c1(C(N2CC(NC(C3CCN(C(C)=O)C3)=O)C(C)C2)=O)cc2cc(Cl)cnc2o1 96552,CS(=O)(=O)c1cc(C(N2CCC3C(C2)CN3C(=O)Cc2csnn2)=O)cs1 96553,N1(C(CCC(C)=O)=O)CC2CC(C1)N(C(c1cccc(C(=O)N(C)C)c1)=O)C2 96554,c1(C(N2CC(C)C(NC(c3ccc(CC4CC4)s3)=O)C2)=O)coc2c1CSC2 96555,N1(CC)CCCCC1C(=O)NC(C)C(=O)NCCOCCN(C)C 96556,C=CC(C)(CCOC)C(=O)NCC(C)C(F)C(=O)N1CC(C)=C(C)C1 96557,c1(CC)nc[nH]c(=NCC(C)(C)NC(C2C(C)C2C)=O)c1F 96558,c1(N2CC=CC(NC(CNC(CC)=O)=O)C2)cc(C)ncc1C#N 96559,C12(C(=O)NCC(CNC(=O)CN3CCCC3=O)F)CC(C1)C(C(F)(F)F)O2 96560,c1(C(N2CCCCC(NC(C(CC=C)(C)C)=O)CC2)=O)cnn2c1CC(C)CC2 96561,C#CCCCC(=O)NC1(CCNC(c2cc(C(F)(F)F)n[nH]2)=O)CC1 96562,CCC(C(=O)N(C(C)CCNC(c1cn(C)cn1)=O)C)NC(C)=O 96563,C1(C(C)NC(C2(SC)CCC2)=O)CCN(C(c2cc(CC3CCC3)on2)=O)CC1 96564,c1(OC)cc(C(=O)NC2CN(C(C3CCC4CC34)=O)CC2OC)ccc1C 96565,c1(C(=O)NC2C(NC(C(C)O)=O)C2)cc2ncccc2[nH]1 96566,C(=O)(C(CC1CC1)c1ccccc1)NCCN(C(=O)C(C)(C)SC)CCC 96567,C(=O)(CC1OCc2ncccc21)NCC(CNC(CCC=CC)=O)(C)O 96568,C1(C(=O)NCC2(C)CCN(C(C)=O)C2)CC2(CCOCC2)CN1 96569,N1(C(C2CCC(CC)O2)=O)CCC2CN(C(=O)C(c3ccc(C)cc3)F)C(C)C12 96570,CC(C)CCCCC(=O)N1CCN(C(=O)CCCCc2cnn[nH]2)C2CC12 96571,C(=O)(C1CCc2nnc(C)n21)Nc1cccc(NC(CCCCCC=C)=O)c1 96572,C1(C(=O)OC)(C(=O)NCCCC(C)NC(=O)Cn2ccnn2)C=CCC1 96573,Cc1ccc(C=CC(N2CCC(O)(C(C)CNC(=O)CCc3ccco3)C2)=O)s1 96574,N1(C(CC2(N(C(C(c3cncnc3)C)=O)C)CC2)=O)CC(F)(CO)C1 96575,CCCCCC(O)CC(=O)NC(CCC)CC(N1Cc2ccccc2C1)=O 96576,C1(CC)CN(C(=O)Cn2ccc(O)nc2=O)CCN1C(C1CCN(C)C1=O)=O 96577,C(=O)(C(O)CC(F)(F)F)NC1CC(C)(CC(=O)NC(C)Cc2ccnn2C)C1 96578,C(=O)(CCCCC(C)(C)OC)N1CCCCC(CNC(CS(CC)(=O)=O)=O)C1 96579,c1(-c2cc(C(N(C)CCN(c3cccc(Cl)n3)C)=O)n[nH]2)ccc2c(c1)OCO2 96580,C(=O)(C1CCCc2nncn21)NCCC(C)N(C(C(C(CC)C)O)=O)C 96581,CC1(C)CCCC(C(N2CCCC2CNC(C2(C(N)=O)CC2)=O)=O)C1 96582,CON(C(=O)C(C)=CCNC(C1CC1C1CCC1)=O)C1CCCC1 96583,C(=O)(C(C)(CC)C(=O)NCC1(CNC(C2CNC(=O)N2)=O)CC1(F)F)OCC 96584,C(=O)(C(CCc1ccc(F)cc1)C(C)(C)C)NCC1N(C(CC=C)=O)CC(O)C1 96585,n1(CC)cc(Cl)c(=NC(=O)c2ccnn2CCC(F)(F)F)[nH]1 96586,C(=O)(CCC(C(C)C)NC(=O)C1=C(C)OCC1)N1CC=C(COC)CC1 96587,CCS(=O)(=O)CC(C)NC(=O)C(N1CCCC(C(F)(F)F)CC1)=O 96588,C1(CC(=O)N(C(C)C)CCN(C(=O)C=Cc2ccco2)C)CC2(CCC2)CCO1 96589,c1(C(=O)NCC2(NC(CC(CCC)O)=O)CCOC2)c2c(c[nH]c1=N)CCC2 96590,c1(C(N(CC(CNC(CC2C(CC)C2)=O)(C)C)CC)=O)cc(=O)cc[nH]1 96591,c1(OCC)cccc(C(c2nnnn2C2CC2)NCCC(O)COC)n1 96592,Cc1noc(C(=O)N(CCC(C)NC(=O)C(C)Cc2c(C)n[nH]c2C)C)c1C 96593,c1(OCC(=O)NC2(CCCNC(C3(CO)CC3(F)F)=O)CC2)cccnc1 96594,N1(C(CC2(OCC)CCC2)=O)CCOC(CNC(c2nnc(S)n2C)=O)C1 96595,C12(C(N3CC(Cn4ncc(C)c4)OCC3)=O)CCCCC(=O)N1CCC2 96596,c1(OC)cc(C(=O)O)ccc1CNc1ccc(-c2nncs2)cc1 96597,C1(CC(=O)NC(C(=O)NCCCn2cnnc2)C2CCCC2)CCC(O)C1 96598,C1(COC)(CNC(c2sccc2Cl)c2nnnn2Cc2ccccc2)CCCO1 96599,C1(Cn2cc(-c3ncc(C)s3)nn2)CCCN(C(=O)CC2CCC(=O)N2)C1 96600,c1(CN(C(c2csnc2C)C(=O)NCCOCC2CC2)CC)ccccc1Br 96601,CCCCCC(C)(CC)C(=O)N1CC2(CCC2NC(=O)CSC(F)(F)F)C1 96602,n1(-c2ccc(OC)cc2)[nH]nnc1=NCC(CSC)C1CC1 96603,N1(C(CC)C(=O)NCCO)CCN(CCNC(=O)Cn2ncnn2)CC1 96604,C1(C(=O)NC2C=CCN(C(c3cc(F)ccc3Cl)=O)C2)CCn2c(O)nnc2C1 96605,c1(CNC)cccc(N)c1.c1ccc(OC2CCCC2)nc1 96606,Cc1cc([N+](=O)[O-])c(S(=O)(=O)N2CCC(c3c(C)cnn3C)CC2)cc1F 96607,C1(CC(=O)NC)CN(C(C23CC(C#N)(C2)C3)=O)CCN1C(c1coc(Cl)n1)=O 96608,c1(C(=O)NCC2(NC(=O)CCCN3CCCC3)CCC2)c[nH]c2nc(Cl)ccc12 96609,N1(C(c2cc(CC)on2)=O)CCC(NC(C2(C)CCCOC2)=O)C(F)C1 96610,C(=O)(CC(C(F)(F)F)N1CCOCC1)NCC(C)NC(c1cc(Cl)ns1)=O 96611,CC1CCN(CC(=O)N(CCC(C)(C)NC(=O)C(F)CC2CCOC2)C)C1 96612,C=CC(C)(C)CC(=O)NC(C)CCNC(c1cc(Cl)ncc1NC)=O 96613,C(CCCCCC(=O)N(CCC(C)NC(c1cc2cnccc2[nH]1)=O)C)SC 96614,N1(C(Cc2cc(C)[nH]n2)=O)CCOCC1CNC(=O)CNC(=O)Cc1ccco1 96615,Cn1ccnc1C(=O)NC(C(=O)NCC1(O)CCSC1)C1(C)CC1 96616,C(CCCC(=O)NCC#CCNC(=O)C(c1ccccc1)SC)SC 96617,CC(O)C(C(=O)NCC=CBr)NC(C1CC(=O)C1(C)C)=O 96618,Cc1nc(NCC2CC2NC(=O)C(C)NC(=O)CC(C)(C)C)c(C)c(C)n1 96619,N1(C(c2ccc(C)c(NS(C)(=O)=O)c2)=O)CCC2(CC1)CC2(C)NCC(N)=O 96620,CC(C)(CNC(=O)OC(C)(C)C)CNC(c1ccsc1I)=O 96621,C1(CNC(CCC(C)(F)F)=O)CN(C(c2cnc3c[nH]nc3c2)=O)CCC1(C)C 96622,C1(OC)=NC=C1C(=O)N(CCn1cc(C(=O)O)nn1)CC1CCCO1 96623,c1(NC(COC(C)=O)=O)ccc(N)c(C(=O)NCC(C)CN2CCCC2)c1 96624,C(=O)(CC(C)(C)C(=O)N1CC(C(=O)NC(C2(O)CCC2)C)C(C(C)C)C1)OCC 96625,C1(CNC(COCC(=C)C)=O)CCC(C)(C)CN1C(C1CCCCS1)=O 96626,CCCCN=C(NCc1cc2c(s1)CCCC2)NCC1(C#N)CC1 96627,C1(CNC(C2(C(C)C)CNC(=O)C2)=O)CCCN(C(C2CCNC(=O)C2)=O)CC1 96628,C(C)(C)(CCC(=O)N1CCCC(N(C(=O)C(N2CCCCC2=O)C)C)C1)OC 96629,N1(C(c2c(C#C)c[nH]n2)=O)CCC(F)CC1C(N1CC(C(N)=O)C(C)C1)=O 96630,C(=O)(C(C)CC(F)(F)F)NCC(=C)CCNC(=O)C(CCCC)N(C)C 96631,C=C(C)CCCC(=O)NCC(C)(C(C)C)NC(=O)CCOc1ccccc1C 96632,CC1CN(C(=O)C(C)(C)C)CCN1C(=O)CC1(C)CCN1C(C1CCC1)=O 96633,C(=O)(CC(C)CC(F)(F)F)NCC1N(C(c2cnc(SC)s2)=O)CC(O)C1O 96634,N1(C(C2C(CC)OCC2)=O)CC(C)(C)CCC1CNC(c1cc(C)nc(O)n1)=O 96635,C1(C)(C(N2CC(NC(C3SCCS3)=O)CC(C)(C)C2)=O)C2Cc3ccccc3C12 96636,N1(C(c2cc(C3CC3)oc2)=O)CCC(NC(C2CCC(NC)CC2)=O)CC1.CS 96637,N1(C(c2cccc(C)c2C)=O)CC2CCC1(CNC(c1[nH]c(O)nc1C)=O)CC2 96638,c1(CC(N2CC(NC(CCOC)=O)C(C(F)F)C2)=O)ccc(OC(F)F)c(F)c1 96639,CC1(C)C2CC(C(=O)NC3(C)CN(C(=O)C=CCCc4ccccc4)C3)CC12 96640,c1(C(=O)OCC)nc(C(=O)NCC2C(O)CC2O)cs1 96641,N1(C(c2nccc(N)c2Cl)=O)CCC(NC(=O)Cc2nccs2)C(CO)CC1 96642,C1(NC(C=C(COC)C)=O)COC2(C1)CN(C(c1cc3sc(C)nc3[nH]1)=O)C2 96643,C1(CNC(CC2N(C(C)=O)CCC2)=O)(OC)CCN(C(=O)C=CC(N)=O)CC1 96644,N1(C(c2c(OC)ccs2)=O)CCN(C(=O)C(O)CC(C)C)C(C2CC2)C1 96645,c1(N2CCN(C(CCC)=O)CC2)nc(N(CCC(C)(C)CC)C)nc2c1CCC2 96646,CCC(C)(C)C(C(=O)N(C)CC1(CNC(c2ncc3ccccn23)=O)CC1)OC 96647,Cc1ccc2nc(C)c(C(=O)NC3CC3CNC(c3ncccc3Cl)=O)cc2c1 96648,c1(NC)c(C(=O)NCCCNC(c2cc(F)c(F)c(F)c2)=O)sc2nccnc12 96649,N1(C(C(C)N(C)C(c2ccc(=O)n(C)n2)=O)=O)CCC(C2CCC2)C1 96650,C1(C(=O)NCC(CC(=O)Nc2ccc(OC)cc2)OC)CCCCCN1C 96651,C1(C)(CNC(C(C)NC(N)=O)=O)CCCN1C(C1CCOC(=O)N1)=O 96652,C1(NC(C=C(CCC)C)=O)CC2CC1N(C(=O)CC1(O)CCCCC1)C2 96653,c1(CC(C(N2C(CNC(c3cnc(C)[nH]3)=O)C=CC2)=O)C)cccc(Br)c1 96654,c1(NC(CC)C(OC)OC)ncc(S(=O)(=O)NC2CS(=O)(=O)CC2O)cc1Cl 96655,C#CC1(O)CC(C(N2CC(NC(c3scnc3C)=O)C(O)C2)=O)C1 96656,C(=O)(C1=COCCC1)N1C(CN(C(c2ccc(OC)nn2)=O)C)CCCC1 96657,CCC1=NOC(C(=O)NC23CC2CN(C(=O)CCOC2CCCC2)C3)C1 96658,Cc1cc(-c2cn(CC(N3CC(COCC4CCCO4)C3)=O)nn2)n(C)n1 96659,CC1(C(N2CCN(C3CCCN(C(C4(C(N)=O)CC4)=O)C3)CC2)=O)CCNC1=O 96660,c1(C(=O)NCC(C2CCOC2)NC(c2n(C(C)C)nnc2)=O)cnc2n1CCC2 96661,N1(C(C(C)Oc2ccc(SC)cc2)=O)CC(C2(NC(=O)CC=C(Cl)Cl)CC2)C1 96662,C1(NC(Cc2c(C)cccc2)=O)CCN(C)C12CCCN(C(=O)C(F)C(C)C)C2 96663,c1(C(N(CC(C)N(C(C(F)=C(C)C)=O)C)C)=O)cnc(O)n(C2CC2)c1=O 96664,C1(C)(NC(c2n(CCC)nnn2)C2CC2(Br)Br)CCC(=O)N(C)C1 96665,CC1(C(=O)NCc2ccoc2C(=O)NC2CC(O)C2)CCC2CC2C1 96666,c1(-c2cc(C(=O)NCC3(NC(c4cscn4)=O)CCCC3)n[nH]2)ccc(O)cc1 96667,c1(C(N(CCCNC(C23CCCCC2C3)=O)C)=O)cc2c(cc1Cl)NC(=O)C2 96668,O(NC(=O)C1(NC(=O)COCCOCCOC)CC1)C(c1nn[nH]n1)COC 96669,C1(C(=O)Nc2c(C(=O)OCC)cno2)CC2(CC2)CN1Cc1cccc(O)c1Cl 96670,C(=O)(C(C)(O)CCN(C)C)NCC(CC)NC(c1cc(C)cc(Br)c1)=O 96671,c1(OCc2ccc(SC)o2)cccc(C)c1C 96672,N1(C(c2c(C)nc(C3CC3)[nH]2)=O)C2CCC1(CNC(=O)C(C)c1ccco1)CC2 96673,c1(C(N2C(CNC(CC(=O)NCC)=O)CC(OC)C2)=O)cc2c(=O)[nH]ccn2n1 96674,c1(C(=O)NC2C(C)N(C(=O)Cn3cccn3)CC2)nc(F)ccc1Cl 96675,C1(C(=O)NCCCOC=C)C2CCCC2CN1C(=O)CN1CCCCC1=O 96676,N1(CC(=O)N(C(C)CNC(=O)CN(C2CCCC2)C)CC)CCC(C)C1 96677,c1(NCCc2c(C)nn(-c3c(C)cccc3)c2C)c(Br)cc(Br)c2ccc(C)nc12 96678,Cc1cc(C(F)(F)F)nn1CC(=O)NC1CCCCC1NC(c1ccc[nH]1)=O 96679,N1(C(CCCOCC)=O)CC2(CCN(C(=O)C(C)CCO)CC2)C1C(C)C 96680,CC1=C(C(=O)N2CC(NC(c3ccsc3C(F)F)=O)C(C)C2)CCO1 96681,CCC(C(=O)NC1CC(C)(CNC(=O)C=CC(=O)NC(C)C)C1)C1CCC1 96682,N1(C(C=C(CC)C)=O)CCC2(CCCN2C(c2cnc(C(C)(C)C)nc2C)=O)C1 96683,c1(CC(=O)OCC(C2CCCC2)OC)ccc(Br)cc1Br 96684,N1(C(CC(CCC)C)=O)CC(CNC(c2ccnnc2C)=O)OC(C)(C)C1 96685,Cc1ccc(CNC(c2cc(F)cs2)=O)c2c1CCCC2 96686,c1(CC(=O)NC2CC(F)(CNC(=O)Cc3ccncc3Cl)C2)ccc(Cl)cn1 96687,CC(C)C(CCN(C(=O)CC1CCSC1)C)NC(=O)CC1CCC(=O)N1 96688,Cc1cc(=NCC2CCSC2(C)C)[nH]cc1S(=O)(=O)N1CCOC(CCO)C1 96689,C(=O)(C1=CC2CCCC12)NCC1(CN(C)C(C2CCN(CCO)C(=O)C2)=O)CC1 96690,c1(C(=O)NCC2(NC(c3ccc(C#C)cc3C)=O)CC2)ccc(P(C)(C)=O)cc1 96691,CC1CCC(CC(N2CCC(Cc3cn(CC(C)(C)OCCO)nn3)C2)=O)OC1 96692,Cc1nn(C)c2nc(C(=O)NC3CN(C(=O)COC4CCOC4)C3)cc(O)c12 96693,C1(C(=O)NC2C(O)C3CCCC23)CCN(C(=O)CCC2CC2)O1 96694,CCC(CCC(=O)N(C(CC(=O)NC)C1CC1)C)NC(=O)C(C)(C)N(C)C 96695,C12(C(=O)NC3CC(CNC(c4c(CCC)nns4)=O)C3)CC3CC(C(=O)N1)C2C3 96696,N1(C(C=C2CCC(C)(C)CC2)=O)CCC2(CCC(NC(C3CCCO3)=O)CC2)C1 96697,CCCCCC(O)C(=O)NC(C1(O)CN(C(c2cncc(Cl)c2)=O)C1)C 96698,c1(C(N(C2(c3ccccc3F)CC2)C(=O)OCC(N)=O)=O)ccnc(Cl)c1 96699,N1(CCN(CC(C)C)C(c2cc(C)c(C)s2)=O)CCCN(C(N)=O)CC1 96700,N1(C(C(F)=CC)=O)CC(NC(=O)CC2COCCO2)CC2(CCC2)C1 96701,N1(C(c2csc(CO)n2)=O)CCN(C(=O)Cn2cccc2)C(CF)C1 96702,c1(NC(c2n(CC(=C)C)nnn2)c2cc(C(C)(F)F)on2)cc(F)cc(F)c1 96703,N1(C(=O)NCC2CCCC(C)C2)CCCc2occc2C1 96704,c1(C(C)=O)ccc(NC(=O)C(=O)NCC(Cc2ccc(Cl)cc2)C(=O)O)cc1 96705,Cc1ccc(CCC(=O)NC2C=CCN(C(C3(C(F)F)CC3)=O)C2)cn1 96706,C1(NC(c2cn(CC)nc2C)=O)(CO)CCN(C(c2csnc2Cl)=O)CC1 96707,C1(NC(c2cn[nH]c2)=O)CCOCC1NC(c1cc(-c2ccncc2)on1)=O 96708,C(=O)(CCC(CC)NC(=O)C1=C(C)CC1)N1CCC(CCCC)C1 96709,c1(OC)ccc(CCCC(=O)N2CC(CCNC(=O)C(O)C3CC3)C2)cc1OC 96710,c1(OC(C)C(F)(F)F)ccccc1-n1cc(C2CCCC2O)nn1 96711,C1N=C2NC(=NC=C2Cl)NC(=O)N2CC1C2.c1(OC)ccc(SC)cc1OC 96712,c1(C(N(C2CC3(C2)CC(N)C3)Cc2c(OC)c(Br)ccc2)=O)c(F)ccc(F)c1Cl 96713,C1(C)(C(=O)NC(c2nn[nH]n2)CC)CC(NC(=O)CC(C)=C(C)C)C1 96714,c1(C(=O)NCC=Cc2c(OC)cc(Br)cc2)c(Cl)ccc2c1OCO2 96715,N1(C(CCSC)=O)CC(NC(c2cc(-c3ccncc3)no2)=O)CC12CCOC2 96716,C1(NC(CC2CCC(C)(C)CO2)=O)CC2CN(C(=O)C3=CCCOC3)CC2C1 96717,c1(CC)cc2c(N3CC(C)(C)CC3CNC(=O)C(C)(C3CC3)OC)nc(C)nc2s1 96718,c1(OC)nsc(C(C(=O)Nc2ccccc2)N(C)CC2CC(F)(F)C2)c1Cl 96719,c1(C(c2n(C)nnn2)NC(C2CCCOC2)(C)C)cc(C2CC2)n(C)n1 96720,c1(C(N2CCN(C(Cc3cncc(OC)c3)=O)C3C2C3)=O)cncc2sccc12 96721,C(=O)(C1CCCc2ncnn21)NC12CC(CNC(=O)COc3ccsn3)(C1)C2 96722,C1(C)(NC(C2C(=C)C2)=O)CCN(C(=O)CCn2c(C)c(C)sc2=O)CC1 96723,C(CO)(CCF)NC(C=CCN(C(=O)Cn1cncn1)C)=O 96724,C(=O)(C1CCOc2ccccc21)N(CCCCCCNC(C(CC(C)C)=O)=O)C 96725,c1(C(=O)NCC(CC)NC(c2ccccc2S(C)=O)=O)cccc(C#CCO)c1 96726,CC1(C)OC2(C(=O)NCC3CN(C(=O)CC4CCCCO4)CC3(F)F)CCC1C2 96727,N1(C(c2nc(CC)sc2Br)=O)CC2(CCC2NC(C2CC=CCC2)=O)C1 96728,S(=O)(=O)(C1CN(C(=O)OC(C)(C)C)C1)NC(C)CC1CCC(C)(C)CC1 96729,N#Cc1[nH]c(=NCC(C2CCCCC2)NC(C2(O)CCSCC2)=O)sc1Cl 96730,c1(N(C(C)COc2ccccn2)C)ccncc1S(=O)(=O)NCC1CC1(F)F 96731,C1(CNC(c2c(C)cnn2C)=O)CN(C(c2c(C)ncn2C)=O)CCC1C 96732,C1(NC(c2cnc(C)nc2)=O)CCCN(C(C2CCCC(F)(F)C2)=O)C1C 96733,c1(NC)cnc(C(=O)NCC(C)(C)OCCNC(=O)CCOCCC(C)C)cn1 96734,N1(C(CCC(CC)C)=O)CC2CC(C1)CN(C(=O)CCC1CNC(=O)N1)C2 96735,CC(C)C(C(=O)NC1CC(NC(=O)C(C)N(C)C)C1)N1CCCCC1 96736,C(CCN=C(NCC1CCOC1)N1CCc2sc(Cl)cc2C1)OCC(C(F)F)(F)F 96737,C=C1CCN(C(=O)C(c2ccccc2)NC(c2cccn2C)=O)C1 96738,O=C(C#CC1CCOC1)NC1CCOCC1NC(=O)Cc1nc2ncccn2n1 96739,c12cnc(nc1)OCC1CCCN1C2=O.CCC(=O)NC(C)(C)C1CCC1 96740,c1(OC)cc(C(N2CCC(CC(=O)NC3CCCNC3=O)C2)=O)cc(C)c1 96741,c1(CC(=O)N(C2CN(C(c3ccc(F)s3)=O)C2)CC)cccc2cccnc12 96742,N1(c2nc(C)nc(O)c2)CC(C2CCCCN(C(C3CCCN3C=O)=O)C2)C1 96743,C1(O)(C(=O)NCC2C(NC(C(CCC)O)=O)CCCC2)CCc2ccccc2C1 96744,CC1CCN(C(=O)CCc2ccc(Cl)cc2F)CC1CNC(=O)CN(C)C(N)=O 96745,C1(CC(=O)NC2CC2c2ccccc2)CCN(Cc2ccccc2Br)CC1 96746,C(=O)(C(F)(F)CCn1cccn1)NC(CC(C)C)CNC(=O)CC12CC(C1)C2 96747,C(CC(C)(C)CC(=O)N(C1CC(=C2CC2)C1)C1CC1)OC 96748,C(N=c1[nH]c(=N)[nH]c(=NC2CCCCC2N(C)C)[nH]1)c1ccc(CC)cn1 96749,CC(CC(=O)N1CC(O)(CN(C(=O)CCCn2cccn2)C)C1)CC(F)(F)F 96750,CC1OCCCC1C(=O)NCCn1ccc(C(=O)Nc2ccsc2)c1 96751,c1(C(=O)NC2CC(CCNC(C=CC(C)C)=O)C2)cc2c(s1)CCS(=O)(=O)C2 96752,C1(C(=O)NC(c2nncs2)C)CN(C(C2CC2Cl)=O)CC12CCC2 96753,c1(CCCN(C(C2CCCN(CCCOC)C2)=O)C(C)C)nnc2ccccn12 96754,c1(C(CC)C)ccc(C(C(=O)NCCC2(C)CC2)N(C2CCCCCC2)C)cc1 96755,N1(C(C(C)(C)OCC)=O)CCC(N(C(c2sccc2F)=O)CC)CC1 96756,Cc1cc([N+](=O)[O-])c(Cl)cc1NC(c1ccc(NCc2ccn(C)n2)cn1)=O 96757,C1(CCC(N2CCCC2Cc2ccccn2)=O)CCc2ccccc2N1 96758,c1(SC(COC)(C)COC)nc(C)nc2sc3c(c12)CCC3 96759,C1(CNC(=O)C(c2ccc(Cl)cc2)=O)COCCN1C(c1cc[n+]([O-])cc1)=O 96760,Cc1ccc(O)c(C(=O)N(C)CC2CC(F)CN2C(C2CN3CCC2CC3)=O)c1 96761,N1(C(C(N2CCCCCC2)C)=O)C2CCC1CN(C(=O)C(N)=O)C2 96762,C1(NC(C=NOC)=O)CCCCC1NC(=O)C(CO)c1ccccc1 96763,C1(NC(CCc2n(C)cnn2)=O)CCN(C(=O)CCn2cccn2)CCC1CO 96764,c1(C(=O)NC2(CNC(CC(CCCC)O)=O)CC2)cccc2c(C)ccnc12 96765,C(CC(=O)NCC1CN(C(C)C)C1)(C(F)(F)F)NC(C=C(C)C)=O 96766,C(=O)(C1=Cc2ccccc2C1)N(CC(C)NC(CC(C)c1ccccc1)=O)C 96767,N1(C(C(CN(C)C)O)=O)CCC2C(C1)CN2C(c1cnn2cccnc12)=O 96768,C1(NC(C(CC)C)=O)CCCN(C(C2CC(O)(C#N)C2)=O)C1C 96769,Cn1ncc2c(N3CCC(NC(=O)CCOCC4CCCO4)CC3)c(C#N)cnc12 96770,c1(C(=O)NC2CN(C(=O)C(O)Cc3ccccc3)CC2F)c(F)cc(F)cc1F 96771,N1(C(=O)CCc2nc(O)n[nH]2)CCC2CCN(C(C3CCCC(F)C3)=O)C2C1 96772,N1(C(c2n(CC)ncc2Cl)=O)CCOC(C)(CNC(C2(F)CCCCC2)=O)C1 96773,O=C(C1=CCCC1)NCCc1ccc(Oc2cccnc2)cc1 96774,C1(CC)CN(C(C2CC2[N+](=O)[O-])=O)CCN1C(=O)C#CC1(C)CC1 96775,CCCS(=O)(=O)CC(=O)NCC1(CNC(c2cncc(NCC(C)C)c2)=O)CC1 96776,N1(C(Cc2c(C)c(Cl)c(Cl)cc2)=O)CCC2CCN(C(=O)C(C)(F)F)CC2C1 96777,C1(C(C)C)CN(C(=O)C(C(C)C)N(C)C)CCN1C(c1cccc(C2CC2)n1)=O 96778,c1(CCNC(C2(C(=O)NCC)CC2)=O)cc(NC(=O)C(C)OC)no1 96779,Cc1ccnc(C(C)(C)NC(=O)CC2CCCN2C(=O)CC(=O)NCC2CC2)c1 96780,N1(C(C(COC)O)=O)CCCC(NC(=O)C(O)CCn2cncn2)C1C 96781,Cc1cc(Br)cc(SSC(C2(C#N)CC2)C)c1 96782,C1(CCNC(c2c(-c3cccc(OC)c3)ncc(Cl)c2)=O)C2CCCCCCC12 96783,c1(C(N(C2CCCN(C(C3CC4(CCC4)CO3)=O)C2)CC)=O)cc2sccc2s1 96784,O=C1CSc2cc(C(N3CCCN(C(=O)CCC(F)F)CC3)=O)ccc2N1 96785,Cc1cccc([N+](=O)[O-])c1NC1CCCC(C(=O)N=c2cc(C3CC3)[nH][nH]2)C1 96786,CCC(C)C(O)CC(=O)NC(C(=O)NC1CCCC1(C)N(C)C)C1CCOC1 96787,C1(C(=O)NC(CCCNC(CSCC#C)=O)CO)Cc2ccncc2N1 96788,N1(C(C=C(CSC)C)=O)CC2CCC(C1)N2C(=O)COCC1CCC1 96789,N1Cc2c([nH][nH]c2=NC(=O)C2CC2F)C1(C)C.c1(OCC)ccc(COCCl)cc1Cl 96790,Cc1c(NC(C2C3CC2N(C(=O)C(CO)c2ccccc2)C3)=O)ccnc1Cl 96791,C(C)(C)(C(C)CC(=O)N1CC(O)(CO)C1)NC(CCC#CC)=O 96792,C1(CN)CC(F)CN1C(=O)CC1CCCC(NC(c2cnn[nH]2)=O)C1 96793,c1(CCN(C)C)nc(-c2cnc(CCSC(C)(C)C)[nH]2)n(CCN(C)C)n1 96794,C1(C(N(C2CCCN(C(c3cnc(C(F)(F)F)nc3)=O)C2)C)=O)CC2(C1)CC2F 96795,c1(C(=O)Nc2cccc(CNC(c3cscn3)=O)c2)ncc2ccccn12 96796,CCC(C)(C(=O)NCCCOCCNC(=O)C(C(C)C)n1cccc1)C(F)F 96797,C(=O)(C(F)CC(C)(C)NC(=O)CC(C(=C)C)OCC)NCC(=O)NCC#C 96798,Cc1ccc(O)c(C(=O)NCC2CC(NC(=O)CC(C)C)C23CCC3)c1 96799,C(=O)(CC(F)(F)CC(F)(F)F)Nc1c(COC)nn(-c2ccccc2)c1 96800,c1(C(CNC(c2occc2CN(C)C)=O)NC(C2CC(=C)C2)=O)ccc(F)cc1 96801,N1(C(c2n(C)ncn2)=O)CC(NC(=O)Cc2ccc(Br)cc2Cl)CC(F)(F)C1 96802,C1(CCC(=O)NCCn2cc(CNC(C(C)O)=O)nn2)NC(=O)NC1=O 96803,C=CC(C)CC(=O)NCCC1CCN(C(=O)CCCc2cc(C)no2)C1 96804,C1(CN(CCC(C)C)C)CCCCN1C(=O)CCN1CCCC1 96805,C#CCC(CC(F)F)C(=O)NC1CN(C(c2nn(C)cc2C)=O)CC12CC2 96806,N1(C(C=CC(C)NC(c2ccc(CC)s2)=O)=O)CCCC1(C)C(C)C 96807,c1(C(=O)NCC2(C(F)F)CCN(C(C(C)(C)C(N)=O)=O)C2)ccc2ccsc2c1 96808,CC(C)(C)CCC(F)C(=O)NC1CCCC1C(=O)NCc1cccnc1 96809,CN(C)S(=O)(=O)N(C)CC(N1CC(NC(C2CC3CCCC23)=O)C1)=O 96810,C1(NC(c2ccc(C(F)F)nc2)=O)CCCC(CNC(C2CCCC23CC3)=O)C1 96811,CC1CCN(C(=O)C(F)(F)F)CC1C(=O)Oc1c(C(=O)OC(C)(C)C)cccc1 96812,c1(C(=O)NCCCC(C)NC(C2CCC(=O)N2)=O)ccnc(C(F)(F)F)c1F 96813,CCCCCC(O)C(=O)N1CC(CNC(=O)C(C)NC(=O)CC(C)(C)C)C(C)C1 96814,C1(C(=O)NC(c2nccn2C)CC)CC(NC(C2CC2Cl)=O)CCO1 96815,N1(C(CCSCC(C)C)=O)CC(CNC(=O)CCNC(=O)NC2CC2)C2CC12 96816,C12(C(NOCC)=O)CCN(C(=O)CCc3ccccn3)CCC1C2 96817,c1(C(C(=O)NC(C(C)NC(C2(C(=O)N(C)C)CC2)=O)C)C)cccc(C#N)c1 96818,C1(CNC(c2cn(C)nc2Cl)=O)CC2OCCC2N1C(c1cc[nH]c(=N)c1)=O 96819,c1(C(N2CCCC(C(N3CCCC34CC4)=O)C2)=O)cccc2c(O)ncnc12 96820,C=C(C)CC(C(=O)N1CC(c2ocnc2CNC(C2CC2C2CC2)=O)C1)OCC 96821,C(=O)(C(C)(C)CCCNC(C1CCCC(O)C1)=O)NC(CCC)CCC 96822,c1(CNC(C(C)OCCCC)=O)ccc2c(c1)CCN(C(c1c[nH]c(=N)s1)=O)C2 96823,O=C1CCCc2ccc(NC(=O)CC3CCN(Cc4cccnc4Cl)C3)cc2N1 96824,c1(C(=O)NCCN(C)C(c2cnn(-c3ccncc3)c2)=O)nscc1Br 96825,C1(C(N(C(CSC)C)C)=O)C2CCN(C(=O)C3=CCOCC3)CC12 96826,S(=O)(=O)(c1ccc(NCc2nc(Cl)ccc2Br)cc1Br)NC(CC)C1CCC1 96827,Cc1[nH]nc(C(=O)N(C(C)CCNC(=O)CC2(C)CCCCC2)C)c1C 96828,c1(C(CNC(c2ccnc(Cl)c2)=O)NC(c2c(C)cco2)=O)ccc(F)cc1F 96829,Cn1cnn(CCC(N2CCC(OCCNC(C3CCC4(CC4)C3)=O)C2)=O)c1=O 96830,c1(OCC)ccc(C(F)(F)F)cc1NC(=O)NC1CCCC(SC)C1 96831,C(C(C(=O)N(CCC(C)NC(C1(C(C)(C)O)CCC1)=O)C)OC)OC 96832,c1(OC)cc(F)ccc1CN1CCCC1CNC(c1ccoc1)=O 96833,S(=O)(=O)(c1cccs1)NCCC(=O)N(CCNC(c1c(CC)occ1C)=O)C1CC1 96834,c1(CNC(=O)CC2CC(F)C2)n[nH]cc1C(=O)NCC#CC1CC1 96835,C(C(C(=O)NC(c1ccoc1)C)NC(=O)C(C)c1cc[nH]n1)OCC 96836,c1(C(=O)NCCC2N(C(C(C)C(F)F)=O)CCC2)csc2ccc(F)cc12 96837,N1(C(c2c(CC)noc2)=O)CC(C2CCN(C(c3ccnn3C3CC3)=O)CC2)C1 96838,N1(C(CS(=O)(=O)NC)=O)CCC(NC(=O)C(C)=C2CCCC2)C(F)C1 96839,Cn1cnc2[nH]c(=NCc3cscc3Cl)nc(N3CCC(C(O)CO)CC3)c12 96840,C(=O)(C(=O)N=S(C)(C)=O)NCC(CC)(CC)NC(=O)C(=O)C(C)(C)C 96841,C1(C)(C(N(CC(C)O)CCNC(C2(CCCC)CCC2)=O)=O)CCOC1 96842,N1(C(C(C2CN(C(c3ccc(O)cc3)=O)C2)OC)=O)CC2(CCC(=O)O2)C1 96843,c1(OC)ncccc1C(=O)NC(C)CNC(c1[nH]c(C2CC2)nc1C)=O 96844,CCC(CC(=O)NCC(C)(F)CNC(=O)CCc1csnn1)C(F)F 96845,C12CCCN(C1)CC(=O)N2.C(C(C)(C)C)N(C(CN(CCC)C)=O)C 96846,Nc1cccc(C(=O)NCCC2CCC(NC(=O)CC(C3CC3)C3CC3)C2)c1F 96847,n1(CC=C)cccc1C(=O)NC1CC(N(C)C(c2ccc(C(F)(F)F)s2)=O)C1 96848,N1(C(CSCC(C)C)=O)CCCCC(NC(C2COC2)=O)C1 96849,c1(N2CCC(CNC(Cc3nc(C(C)C)on3)=O)C2)cccc(F)c1F 96850,c1(C(=O)NC(C2CCCC2)CO)cc(CCNC(c2ccc[nH]2)=O)on1 96851,Cc1ccc(=O)n(CC(=O)NC2CC(C)(NC(C3CC(CF)C3)=O)C2)n1 96852,c1(C(N2CC(C)C(CNC(=O)C3=CCCCO3)C2)=O)cc2c(Cl)c(F)ccc2[nH]1 96853,C=CC(C)(C)C(=O)N(CC(C)N(C)C(c1ccc(CO)cc1)=O)C 96854,Cc1cc(Br)cnc1C(=O)OC(C)(C)C.c1(N2C3CC(C3)C2)cncnc1C(N)=O 96855,C1(CNC(C(C2CC2)OC)=O)CN(C(=O)C(C(C)C)NC(=O)CC(C)C)CC1C 96856,C1(C)(C(=O)NC2CN(C(C(C(=O)OC)(C)C)=O)CC2O)CCc2ccccc2C1 96857,CC(C#N)CCC(=O)N1CCC(CCCNC(=O)CCC2CCCCC2)CC1 96858,C(=O)(C1=CCCCC1)N(C)CC1CN(C(CC2(OCC)CCC2)=O)C1 96859,C(=O)(C(CC)C(F)(F)F)NCC(CC(=O)NC(C#C)(CC)CC)C 96860,N1(CCc2c(C)non2)CCCC12CCOCC2 96861,N1(C(CCc2cnc(C)o2)=O)CC2C(CNC(=O)C(C3CCOCC3)F)C2C1 96862,C12(NC(CCCOC)=O)CC(CNC(C3CCN(C)C3C)=O)(C1)OC2(C)C 96863,C1(NC(c2cnc(OCCO)cn2)=O)CCCN(C(=O)COCCO)C1 96864,C(C(O)CC(F)(F)F)NC(CC1CN(C(CCOC)=O)C(C)C1)=O 96865,C1(NC(COC(C)C)=O)CCC(N(C(=O)CCNC(=O)OC(C)(C)C)C)CC1 96866,c1(C(=O)NC(CC(C)NC(C)=O)C)cc(Br)c2[nH]c(C)nc2c1 96867,C(CCC(O)C(=O)NCC1CC2(CCC2O)C1)NC(Cc1cnc(C)s1)=O 96868,Cc1c(C(=O)NCCCNC(=O)C(C)c2ccco2)c(C)n2ccncc12 96869,c12ccc(cc1)C(=O)N1CCC(CC1)NC2.C1(NC(c2cc[nH]n2)=O)CCCC1 96870,c1(CNC(c2nncs2)=O)cccc2sccc12.C12CCCC(C1)CNC2=O 96871,C1(NC(C2C(CNC(Cc3cc(OC)no3)=O)CCCC2)=O)CC2CCCC2C1 96872,C1(C(N2CCC(N(C)C(c3occc3Cl)=O)C2)=O)CN(C)C(=O)N1 96873,c1(C(N2CCCC(C(F)F)C2)C(=O)NCc2nccs2)cc2cc(Br)ccc2o1 96874,c1(NC2CC(C)N(C(=O)C3=CCC3)C2)c(C#N)nnc2ccccc12 96875,C(CC(C)(C)C(=O)N1CC(C(=O)NC(C)C(C)(C)C#N)C2(CC2)C1)OC 96876,C1(N(C(c2c(C)nsc2)=O)C)CN(C(c2cn(C3CC3)nc2C)=O)CC12CC2 96877,N1(C(Cc2c(C)ccs2)=O)CCC(C)C(NC(=O)CCOc2ccc(F)cc2)C1 96878,C1(CNC(c2c(C(C)C)onc2)=O)CCCC2(CN(C(c3cnnn3C)=O)C2)O1 96879,C1(N(C(c2cn(C)nc2C(F)(F)F)=O)CC)CCN(C(=O)CNC(=O)OC)CC1 96880,N1(C(c2cc(C(C)C)on2)=O)CCC12CN(C(=O)CSCCN(C)C)C2 96881,c1(C(=O)NC2(c3cnccn3)CCC2)nccc2nc[nH]c12.C12CC1CNC2=O 96882,CC1CC(=O)NCCN1C(C1C2CCC(C2)N1C(=O)C=Cc1ccsc1)=O 96883,c1(OCC(=O)NCCC2CC(NC(CN3C(C)CC3)=O)C2)ccc(Cl)nc1 96884,O=C1CCNc2cc(C(N3CC4C(NC(=O)C(F)(F)C(F)F)C4C3)=O)ccc2N1 96885,N1(C(C2C(C3CN(C(c4n(C)cc(Cl)c4)=O)C3)C2)=O)CCC2(CNC(=O)N2)C1 96886,C1(CC)CN(C(=O)Cc2c(C)cccc2Br)CCN1C(C1CN(C)C1)=O 96887,N1(C(CCC=C(C)C)=O)CC(NC(=O)Cc2ccsc2)C(Cc2ccccc2)C1 96888,c1(C(N2CCN(C(CN(CC)CC)=O)CC2C(C)C)=O)onc2cc(C)ccc12 96889,N#CCCCC(=O)NCC(O)CNC(c1cnc(Cc2ccccc2)cn1)=O 96890,C1(C)(C(=O)NC(C(C)C)CCNC(=O)Cc2cccn2C)CCOC(C)C1 96891,c1(C(=O)NC2CC=C(C(=O)N3CCC(C=C(C)C)CC3)C2)cc2cccnc2[nH]1 96892,C12CCN(C(C)C1)C(=O)CNC2=O.c1(NC(C(CC)=CC)=O)cccc(C)c1 96893,Cn1cc(NC(=O)C(CN(C)C)NC(=O)CCC(N)=O)c(C(N)=O)n1 96894,CCCCC(O)CC(=O)NC1CN(C(c2c(F)cc(N)cc2F)=O)CC2(CC2)C1 96895,N1(C(CC=CC)=O)CC2CCC(C1)N(C(c1cnn(-c3ccccn3)c1N)=O)C2 96896,NC12CN(C(=O)C(C3CCCCC3)Sc3ccccc3)CC1CS(=O)(=O)C2 96897,C1(CNC(=O)Cc2cscn2)CC(O)CN1C(C1CC(=O)N(c2nccs2)C1)=O 96898,C(=O)(CC(C)(C)C=C)NC(CC=C)CNC(=O)C(c1cccc(F)c1)O 96899,c1(N(C(=O)NC(c2ncc[nH]2)CC)CC)n[nH]c2c1COCC2 96900,O=C1Nc2cccc(-c3ccc(F)c4occc34)c2CO1 96901,C(=O)(C1=CCC(NC(C2CC3C=CC2CC3)=O)C1)NCC1(C)CCCC1O 96902,N1(C(c2ccc(CNC(CC(C=C)C)=O)nc2)=O)CCC(N(C)C)C(C)C1 96903,c1(C(=O)NC(C(=O)NC(CCCC)CO)Cc2cc[nH]n2)cc(C)n(C)c1C 96904,C(CC(C)C)(C(=O)N(C1C=CC(C)(C)CC1)CCC(=O)OC)OC 96905,Cc1cc(C(N2CCC3(CC3C(=O)Nc3ccc(F)c(O)c3)C2)=O)cnc1C 96906,c1(OC)cc(OC)c(C(N2CCC(NC(C3CCC3(F)F)=O)C2C)=O)cn1 96907,C(CCCCC(=O)N(C)C(c1ccco1)C)N(C(c1n(CC#C)ccc1)=O)C 96908,c1(C(=O)NCCC(CNC(C=CS(C)=O)=O)O)cc(F)c(N)c(F)c1 96909,C(C)(CC(C)(C)CO)NC(CC1(CNC(C(CC)C#N)=O)CC1)=O 96910,c1(CC)[nH]c(=NCC2C(C)CCCN2C(=O)CN2CC3CC3C2)sc1C 96911,N1(C(C2C(CC)CCCC2)=O)CCC(NC(=O)C(C)CC2CCCC2)C(C)(C)C1 96912,c1(C(=O)NC2(C)CC(NC(C(CO)N(C)C)=O)C2)cccc(F)c1Br 96913,CC1(NC(=O)CC=CCNC(c2coc(C3CC3)c2)=O)CCOC1C1CC1 96914,N1(C(C(COC)OCc2ccccc2)=O)CCOC(CSC2CC2)C1 96915,c1(OCC)cc(C(C)=O)ccc1Sc1nnnn1C1CCCCCC1 96916,c1(CC(=O)NCC2C3CN(C(CCCC(=C)C)=O)CC32)ccc2[nH]ccc2c1 96917,C=CC1CCCN(C(C)=O)C1.c12ccc(cc1Cl)NC(=O)CCCn1cc-2nn1 96918,N1(C(CCCC#N)=O)CCN(C(=O)CC2CC(c3cccc(F)c3)C2)CC1CF 96919,c1(CC)sc(C(=O)NCC(C)(C)CNC(c2ccc(C(=O)OC)nc2)=O)cc1C 96920,N1(C(C(CC)NC(C)=O)=O)CCC2(CCC(NC(c3cnccc3Cl)=O)CC2)C1 96921,CCC(C)CCC(=O)NCCC1(NC(c2sccc2OC)=O)CCC1 96922,C12(CNC(Cn3c(C)nnn3)=O)CCCCC1N(C(c1ccnnc1)=O)CC2 96923,c1(CN2CCCCC2C)cc(N2CCN(CC3CCC(SC)C3)CC2)nc(C)n1 96924,C1(NC(=O)C(c2ccccc2)F)COC2(C1)CN(C(c1scnc1Cl)=O)C2 96925,N1(C(c2ccc(N(C)C)cn2)C(=O)NC2COC2)Cc2nc(Br)sc2C1 96926,N1(C(C2CC(CC)C2)=O)CC(O)(CNC(C2C3COCC23)=O)C1 96927,C(=O)(C1CCCc2nnn(C)c21)NCC(C)(C)OCCNC(CCOCCC)=O 96928,C(=O)(CCC(=O)NN(C)C)N1C(CN(C(C2C(CN(C)C)C2)=O)C)CCC1 96929,N1(C(C)C(=O)NCC2CCCN2C(c2cnn(CCO)c2N)=O)CCN(C)CC1 96930,c1(C(N(C2CC(NC(C3(CO)CCCC3)=O)C2)C)=O)cncc2ccc(F)cc12 96931,C1(C)(CN(C)C(c2ccoc2)=O)CCCC1NC(=O)CNC(C1CCOCC1)=O 96932,C1(Cn2cc(CC(C)(C)O)nn2)CN(C(c2cnncc2O)=O)CCO1 96933,CC1CN(C(=O)C(c2cccnc2)O)CCC1CNC(c1ccc(Cl)c(O)c1)=O 96934,CC1CN(C(C2(CF)COC2)=O)CC1NC(=O)C(F)(F)c1nccs1 96935,c1(C(=O)NCc2ccc(-c3cn(C)nc3)cc2)cc(O)cc(O)c1 96936,C(=O)(Nn1cnnc1C)C1CN(C(C(N2CC(C)C2)C)=O)CC1C 96937,c1(CCN2CC(C(F)(F)C(=O)OC)C(F)C2)c(C)nn(C)c1C 96938,N1(C(c2c(C)nn(C)c2)=O)CCOC2CN(C(=O)C(C)(O)c3ccccc3)CC12 96939,C=CC1(C(=O)NCC(C2CC2)N(C)C(c2cccc(F)c2)=O)CCCCC1 96940,c1(C2(CNC(C3CCCO3)CC)CC2)ccccc1C(=O)O 96941,N1(C(=O)NCC2CSCCS2)CCc2n[nH]cc2C1 96942,C1(C(=O)NCCCN(C(=O)C(c2ccc(F)cc2)(F)F)C)CCCC(F)C1 96943,C=CC(C)(CCOC)C(=O)N(CC(O)CNC(c1cc(C(F)F)cc(C)c1)=O)C 96944,c1(C(N(CCCNC(c2cnnn2-c2ccccc2)=O)C)=O)snc(O)c1Cl 96945,c1(C(N2CCC(C)(CNC(C(CSC)C)=O)C2)=O)ccnc2ccsc12 96946,c1(C(c2nnnn2C)OC)c(F)ccc(Br)c1NC(CSC)C(C)C 96947,C1(NC(C2SCCS2)=O)CCC2(CCCN(C(c3cccnn3)=O)C2)C1 96948,Cc1nc(C(=O)NCC(=O)NC(C(=O)O)C(C)C)[nH]c1C 96949,C1(N(CCNCC(C(C)(C)C)OC)CC)CCS(=O)(=O)C1 96950,C12(C(=O)NC(C3(NC(C(CC)n4ccnc4)=O)CCC3)C3CC3)COCC1C2(F)F 96951,c1(CNC(=NCCOCC)NCC2CCCC(C3CC3)O2)nc2ccccc2s1 96952,CC1=C(C(=O)N2CC(NC(=O)C(C)S(C)(=O)=O)C3(CCC3)C2)COCC1 96953,CC1=NS(=O)(=O)N(C)C=C1C(=O)NCC1C=CC(NC(=O)C(C)CC2CC2)C1 96954,C1(C(N2CC(NC(CSCC)=O)C2)=O)CCC2CCC1O2 96955,C1(CN(C)C(C2(NC(=O)C3CC3)CC2)=O)CN(C(=O)CSC(F)(F)F)C(C)(C)C1 96956,c12ccc(cc1Br)s2.N1(C(=O)OCC)CCC2C(O)CC12 96957,N1(C(C(CC)CC)=O)CC(C)(C)C(NC(=O)CC2CCOC(CC)C2)C(C)(C)C1 96958,CN1CC(C(=O)NCC2CC(F)CN2C(=O)Cc2ccoc2)CC1=O 96959,N1(C(CCC(=O)NCCC)=O)CC2CN(C(=O)CCN3CCN(C)CC3)C2C1 96960,c1(C(CCOC)NC(C2(c3ccccc3)CC2(Cl)Cl)=O)ccc(C)cc1 96961,C1(OC)CC(NC(=O)N(CCCOCC2CC2)C2CC2)C12CCCO2 96962,c1(C(=O)NC(C2CCOC2)CNC(c2ccc[nH]2)=O)cc2c(s1)CCCC2 96963,c1(C(=O)NCC2CC2NC(C23CCC2CC3)=O)cc2c(s1)CCCC2 96964,C(C(CC(F)(F)F)NC(=O)C(C)Oc1ccccc1F)NC(CCC=C=C)=O 96965,N1(C(C(CC(F)F)N(C)C(c2ccncc2O)=O)=O)CCCN(C)CCC1 96966,c1(C(C(=O)NCC(C)N(C(C2CCCO2)=O)CC)(C)C)cccc2ccccc12 96967,c1(C(N2C(C)C(NC(=O)C3CC3)CC2)=O)cc2c(cc1[N+](=O)[O-])OCCCO2 96968,c1(C(N2C(CN(C(CCC3C(C)C3)=O)C)COCC2)=O)cc(N)cnc1Cl 96969,N1(C(C(C2CCCC2)OCC)=O)CC2CCC1CN2C(=O)C(c1ccccc1)O 96970,c1(C(=O)NCC(CNC(=O)Cn2cnnc2O)O)cc2cccc(F)c2s1 96971,c1(C(N2C(Cn3cc(CCSCC)nn3)CCC2)=O)ccc(C)c(Br)c1 96972,C1(C(=O)NCC=C=C)(CNC(=O)CCc2conc2C)CCCCC1 96973,c1(CC(=O)NCC2CC2NC(C2CC(F)C2)=O)ccc2c(c1)OCO2 96974,C1(NC(CCC(=O)NCC)=O)CCN(C(=O)CCP(C)(C)=O)C(C)C1 96975,c1(CNC(CC(CCC)CC)=O)cccc2c1CN(C(=O)C(F)(F)CC)C2 96976,C(=O)(C1Cc2ccc(Cl)cc21)NC1(CO)CCCN(C(c2c(CC)cno2)=O)C1 96977,CC1(C)CCC(CC(=O)NCC(O)C(=O)NCC2(C(O)C(C)C)CC2)C1 96978,Cc1cc2ccc(C(N3CCC(NC(=O)C(C)C4CC4)C(F)C3)=O)cn2c1 96979,C1(C(C)NC(=O)CCc2cncn2C)CCN(C(c2ccccc2F)=O)CC1 96980,c1(Cn2cc(CNC(C(CC)C)c3ccccc3)nn2)ccc2c(c1)oc(=O)n2C 96981,Cc1nc(CCC(=O)NC2CCN(C(c3ccc(C)n3C)=O)C2C2CC2)[nH]c1C 96982,Cc1ccn2ncc(C(=O)NC3(C)CCCN(C(C4CCC4(F)F)=O)C3)c2n1 96983,c1(C(=O)NC2C(CNC(C(C)OCCCC)=O)CC2)cccc2nccnc12 96984,C1(CNC(=O)CC2CCCCC2)CCN(C(C2C3CCCC23)=O)CC1O 96985,N1(C(C=CC(CC)=CC)=O)CCC(NC(c2cc(C)[nH]n2)=O)CC1C 96986,c1(CC(N2CCC(C3N(C(=O)OC(C)(C)C)CCC3)C2)=O)ccc(F)c(Cl)c1 96987,c1(C(N(C)CC2CCN(C(C(C3CCOCC3)OC)=O)C2)=O)cccc(=O)o1 96988,C1(CCNC(CC=C=C)=O)CCCN(C(c2cncc(N)n2)=O)CC1 96989,C12(C(=O)NC3(CC#C)CCC3)CCC(CN(C(=O)C(C)(O)C3CCC3)C1)C2 96990,Cc1cc(Cl)c(C(=O)NC2CC(C)N(C(C3CC(CF)C3)=O)C2)s1 96991,c1(C(=O)NCCN(C(=O)COC2CCCC(C)C2)CC)cncc2[nH]ccc12 96992,C1(C(N(C2CCN(C(c3cnns3)=O)C2)CCC)=O)CCC(C(F)(F)F)O1 96993,CC1CN(C(c2ccc(CN3CCCC3)cc2)=O)CCCN1C(=O)COCCF 96994,c1(C(N2C(=O)NC(C)(c3cccc([N+](=O)[O-])c3)C2=O)=O)ccc(O)cc1[N+](=O)[O-] 96995,c1(CNC(=O)NC2CC(C)SC2)ccccc1CCO 96996,N12CCn3ncc(c3C1)OCC2=O.N1(C(=O)OC(C)(C)C)CC(F)C1 96997,N1(C(C2N(CC)C(=O)CC2)=O)CCC2(C1)CN(C(C1CCCCC1O)=O)CCO2 96998,C1(NC(C(CCOC)C)=O)C2CCN(C(=O)C(C)(C)COC(C)C)CC12 96999,C1(C(=O)NCC2(CN(C)C(c3cc(C#N)cs3)=O)CC2)CCc2ccccc2C1 97000,C1(NC(c2nccs2)=O)CN(C(c2ccns2)=O)CCC12CCOCC2 97001,C1(CNC(C(CC)n2ccnc2)=O)CCN(C(=O)Cn2nnc(C)n2)CC1 97002,N1(C(c2[nH]ccc2CNC(C2(O)CCSC2)=O)=O)CCC2CCC(C2)C1 97003,c1(CNS(C)(=O)=O)cc(-c2ccc(Nc3nccs3)cc2)cc(S(N)(=O)=O)c1 97004,C12(C(=O)NC(CCN(C)C)CO)CC(CO)(CN1C(C1CCCC(=O)N1)=O)C2 97005,c1(C(=O)NC2C(=O)N(c3cccc(Br)c3)CC2)cc(I)c(Cl)cc1Cl 97006,c1(C(=O)NC2C(NC(C(C)OCC#C)=O)CC2)cc(N)ccc1O 97007,CC(CNC(=O)OC(C)(C)C)C(=O)NCCN(C)C(c1conc1C(C)C)=O 97008,Cc1cc2c(cc1C)C(C(=O)NCC(C)NC(=O)CC1(C#N)CC=CC1)CO2 97009,C(=O)(C1=C(C)N(C)c2nnnn2C1)NCCCCNC(COCCSC)=O 97010,N1(C(C(C)C2CC2)=O)CCOC2(CCN(C(c3csc(C(C)(C)C)n3)=O)C2)C1 97011,c1(C(=O)NCC(CC(=O)Nc2c(OC)nn(C)c2)OC)cc(C)cc(O)n1 97012,c1(CC(=O)NCC2N(C(C34CC(OC)C3C4)=O)CCC(C)C2)c[nH]c2cccnc12 97013,c1(CC(=O)NC(CC(C)NC(C(CC)N(C)C)=O)C)coc2c(C)c(Cl)ccc12 97014,CC1CC(C(=O)N(C)Cc2nc[nH]n2)N1C(c1nocc1Cl)=O 97015,C(CCC(CCC)NC(c1nc(C)ccc1C)=O)NC(C(CCC)NC(C)=O)=O 97016,C(=O)(C1CCc2snnc21)N1CCCC(NC(CSCC#C)=O)CC1 97017,C1(NC(c2cncc(OC)c2)=O)CCCN(C(C2C=CCS2)=O)C1C 97018,Cc1cn2c(n1)C(C)CC1CCC(C2)N1C(=O)C(N1CCOCC1)=O.C12CCC1C2 97019,CCC(C)(O)C(=O)NCC1CN(C(=O)Cn2ccc(C3CC3)n2)CCO1 97020,N1(CC(CC)C(C)C)C(=O)CN(CCCc2nccs2)C1=O 97021,c1(NC(C(=O)NC2(COC)CCOCC2)=O)ccc2c(c1)N(C)C(=O)CO2 97022,c1(CCN=C(NCC(COC)C)NCCC(C)(C)C)ccc2[nH]ccc2c1 97023,C(=O)(C(CC(C)C)C(C)C)NC(CNC(c1occ(OC)c(=O)c1)=O)CO 97024,C(=O)(CC(C)(C)C)N1CC(NC(C2CCN(C(C)=O)C2)=O)(CO)C1.C1(=O)C(C)N1 97025,C12(C(=O)NCC3(F)CCC(CNC(Cc4ccn(C)n4)=O)C3)CC1COC2(C)C 97026,c1(C(=O)NCC2(C(C)NC(C3C(CC)C3)=O)CC2)cnc(C)o1 97027,c1(CC(=O)NC(C)CNC(C2COC2)=O)ccc2ccncc2c1 97028,N1(C(c2nc(C)oc2C)=O)C2CCC1CC(CNC(=O)C(C)Cc1ccco1)C2 97029,C1(NC(C(CC)c2ccccc2)=O)CC2(NC(=O)COC3CCCC3)COC1C2 97030,Cc1cc(O)ncc1C(N1CC(CO)(NC(c2ccc(C(F)F)cn2)=O)C1)=O 97031,c1(NC(C2C(NC(C=CC=CC)C=O)CCCC2)=O)cc(Cl)ccc1I 97032,CC(C)C(O)C(C)C(=O)N1CCCC(N(C)C(c2ccnc(OC3CC3)c2)=O)C1 97033,CC(CC(=O)NC1CC1NC(=O)Cc1ccoc1)N1CCCC1=O 97034,N1(C(c2cn(C)nc2)=O)CCC2CN(c3ccc(Cl)cc3[N+](=O)[O-])CC2C1 97035,Cc1cc(C(F)(F)F)nc(=NCCc2ccc(CC(C)C)cc2)[nH]1 97036,c1(C(=O)NC(C=CC(=O)NC2C(OC)C3(C2)CCC3)C)cccc2cncn12 97037,C(=O)(C1=CCN(C(=O)C(C)(C)C2CCCO2)C1)NC(C)CC1CCCO1 97038,Cc1nsc(N)c1C(=O)NCC1(O)CCN(C(c2ccoc2Cl)=O)C1 97039,CC1C(NC(=O)C(F)C(C)(C)O)CC2CCC1N2C(=O)Cc1ccsc1 97040,C1(C)(CC)CC(C(=O)NCCCC(CO)NC(=O)CN2CCCC2=O)CCO1 97041,CN1CCN(C(C2CCOCC2)=O)CC1C(N1CC(C(N)=O)C1)=O 97042,C(=O)(CC(F)(F)C(F)(F)F)NCC(C)(C1CC1)NC(CCN(C)CCO)=O 97043,C1(NC(C(N2CCN(C)CC2)C)=O)CC2C(NC(=O)C(C)(C)O)C2C1 97044,N1(C(c2c(C)cncc2)=O)C2CCC(C2)C1CNC(=O)C=CC(=O)NC1CC1 97045,C1(C)(CC(=O)N(C)CCNC(c2csc(C3CC3)n2)=O)CCS(=O)(=O)N1 97046,C(CO)(CO)(CO)NC(C1(CCNC(C(C)C2CCCC2)=O)CC1)=O 97047,N1(C(C(N2CCN(C(C(=O)OCC)=O)CC(C)C2)=O)=O)CCC2(CC1)CNC(=O)C2O 97048,N1(C(C(C)c2cc[nH]n2)=O)C2CCC1CC(CNC(C1(CF)CCC1)=O)C2 97049,N1(c2ncnc(N(C)Cc3cccc(SC)c3)c2C)CCC(C)C(C)(C)C1 97050,C(=O)(CC(F)(F)C(F)F)NCC1N(C(c2ccc(CC)c(Cl)c2)=O)CCC1CC 97051,c1(SC)ccc(O)c(C(=O)NCC2CCCC2NC(C2CC2C(F)F)=O)c1 97052,N1(C(c2c(CNC(C3(CSC)CCC3)=O)n[nH]c2)=O)CCC(O)CC(C)C1 97053,C1(CNC(CC2CC(NC(C3(OC)CCSC3)=O)C2)=O)CC(=O)N(C)C1=O 97054,C1(CNC(C=C(CCC)C)=O)C(C)CCCN1C(C1CN2CCC1CC2)=O 97055,C12(C(=O)NCC3(CNC(C=CC(CC)C)=O)CCC3)CCCC1(C(N)=O)C2 97056,c1(C(=O)NC(CC=C)CNC(=O)CN(S(C)(=O)=O)C)cccc2oc(C)nc12 97057,CCN=c1[nH]c(C(N2CCN(C)CC2CNC(c2c(C)ccn2C)=O)=O)cs1 97058,N1(C(CCOCCCC#C)=O)CC(OC)CC1CNC(c1cn(C)nc1CC)=O 97059,c1(CN2C(CC(=O)Nc3cnn(C4CC4)c3)COCC2)ccc([N+](=O)[O-])cn1 97060,N1(C(c2cccc(CC)c2)=O)CCOCC(C)(CNC(c2nc(C)oc2C)=O)C1 97061,C1(NC(c2csc(C)c2N)=O)CC2CCCC(C1)N2C(=O)C(C)(C)CC1CC1 97062,C1(C(N(CCC(N2C(CCC)COCC2)=O)C)=O)CCC(C)(O)CC1 97063,C(CCCCOC(C)=O)(C(=O)NC)N1CC(CC(C#C)C)C1 97064,C1(CNC(CCC(=C)Cl)=O)CC2CCCCC2N1C(=O)CCc1ccn(C)n1 97065,C12(NC(C=C(CCOC)C)=O)CC(CNC(C3CC3C(N)=O)=O)(C1)C2 97066,C(=O)(C1=CC(O)C(NC(=O)C(O)CC(F)(F)F)C1)N1CCCC(C(N)=O)C1 97067,C1(NC(c2cc(C(C)C)n(C)n2)=O)CCCCC12CCN(C(=O)C(F)F)CC2 97068,CC1(C)C(CC(=O)NCC2(O)CCSC2)CCN1C(c1cn[nH]c1)=O 97069,CC12CN(C(c3ccc[nH]3)=O)CC1CN(C(C1(C3CCCO3)CCC1)=O)C2 97070,N1(C(c2c(OC)c[nH]n2)=O)CCCC(C)(C(=O)NCCCn2nccn2)C1 97071,c1(N(C)C(=O)OC(C)(C)C)ncncc1I.C1(C)(CO)CC12CCC2 97072,CC1(C)NC(=O)N(CC(=O)NCC(CO)NC(=O)C(C)(C)NS(C)(=O)=O)C1=O 97073,Cc1cc(N2CCC(C)(CO)CC2)ncc1S(=O)(=O)NC1CCCOC12CCC2 97074,c1(OCC)cccc(CC(=O)NCC2(OC)CCN(C(c3cc[nH]c3C)=O)C2)n1 97075,N1(C(CCCC(=C)C)=O)CC(NC(c2cscc2CC)=O)CCC(O)C1 97076,c1(C(N2CCN(C(C3(COC)CC=CC3)=O)CC2C)=O)cc(N)c(C)cc1Cl 97077,N1(C(=O)OC(C)(C)C)CCc2[nH]nc(C(N3CCC(F)(F)C(O)C3)=O)c2C1 97078,c1(OC)c(Cl)cc(C(=O)NC2CC(NC(c3nccc(C)n3)=O)CC2O)nc1Cl 97079,N1(C(CCC#CC)=O)CC2CCC1C(CNC(=O)Cc1c(C)nc(O)nc1O)C2 97080,C(=O)(C(CC1CC1)NC(=O)COC1CCN(C(=O)CN(C)C2CC2)C1)OC 97081,C1(CNC(CC2C(C)CCC2)=O)CN(CCCC(C)(C)C)CCC1C 97082,CC1(C(=O)NCC2CCC(F)(CNC(c3ccc(C(N)=O)o3)=O)C2)CCC(=O)N1 97083,Cc1cc(C)c(C(N2CC(N(C(=O)C(O)CN(C)C)C)C(O)C2)=O)cn1 97084,c1(C(=O)NC2CCN(C(c3cnc(CCC)s3)=O)C(C)C2)cc(F)c(C)cc1Cl 97085,C=C=C(C)CC(=O)NCCN(CC(C)O)C(=O)CN(C1CC1)CC 97086,c1(NC(c2n(CC=CC)ncc2)=O)cnc2c(c1)CN(S(=O)(=O)CC(C)C)CC2 97087,C1(NC(CCc2cc(OC)no2)=O)(CO)CCN(C(C2COCCO2)=O)C1 97088,N1(C(CCCCC#N)=O)CC2CCCCN2CC1CNC(=O)C=CC(F)(F)F 97089,N1(C(COCCOCC#C)=O)CCC2CN(C(c3sc(C)cc3Cl)=O)C2C1 97090,C1(OC)(COc2ccc(F)cc2F)CCN(C(=O)CS(=O)(=O)N2CCCC2)CC1 97091,N1(C(c2ncn(C(C)C)n2)=O)CC(F)(F)CC1C(N1CCNC(=O)C1C)=O 97092,C1(NCCNC(C2(CCC)CC2)=O)CCCN=C1 97093,c1(C(=O)NCC2C(NC(C(C#C)(C)C)=O)COC2)ccc(Cl)c(CC)c1 97094,CC(C)C(O)CC(=O)NCC1(NC(c2ccc(C3OCCO3)cc2)=O)CCCC1 97095,N1(C(C=CCOC)=O)CCCC(C)(NC(c2cn3ccsc3n2)=O)C1 97096,C1(CC(=O)NCC(C2CC2)NC(=O)CCOCCOCCCO)CCOC1 97097,c1(OC)cccc(C(N2CCN(C(c3cnc(C)[nH]3)=O)C3CC23)=O)c1[N+](=O)[O-] 97098,c1(OCC)ccc(C(=O)NCCC2CN(C(=O)CCC(N)=O)CC2C)cc1OC 97099,C#Cc1ccc(C(=O)NC2CCCC2NC(C2(COC)CCNC2=O)=O)cc1 97100,CCC(C)(COC)C(=O)N(N1CCN(C(=O)CCC(C)OC)CC1)C 97101,Cc1cccnc1C(=O)NC1CCCC1n1cc(C(C)(C)OC(=N)O)nn1 97102,C1(n2cc(CNC(C(C)C3CC3)=O)nn2)CCCN(C(=O)CC2CCCCC2)C1 97103,N1(C(c2n(C)nc(C)c2F)=O)C2CCC1CN(C(=O)COc1ccccc1F)C2 97104,c1(C(=O)NCCN(C(CC)C)C)ncccc1CNC(=O)CC1CN(C)C(=O)N1 97105,C1(NC(CCC(C)NC(c2c(C)n(C)cn2)=O)=O)CCNC(=O)CC1 97106,C1(CNC(C=CCN(CC)CC)=O)CN(C(=O)CS(N)(=O)=O)CCCO1 97107,c1(N(C(c2ccnn2CC)C(=O)NC(CC)C)C)ccc(C)c(F)c1 97108,C1(C2CCN(C(=O)CN(C)C(=O)OC(C)(C)C)CC2)(NC(C=CCCC)=O)CC1 97109,CC1(C)CCC(F)(F)CC1C(=O)NC1CN(C(=O)Cc2nc[nH]n2)CC1N=[N+]=[N-] 97110,C1(CC(=O)NC2CCCC(N(C(=O)C=C3CCCCC3)C)C2)(OC)CCCCC1 97111,C(=O)(C1=COCCO1)N1C(CC(C)(C2CC2)NC(c2cc(C)c(Cl)s2)=O)CCC1 97112,N1(C(c2c(CCC)nco2)=O)CCCC2CN(C(c3cccc(C)c3)=O)CCC12 97113,CS(=O)(=O)c1ccc(C=CC(N2CC3CN(C(=O)C=CBr)CCC23)=O)o1 97114,c1(C(CNCc2cn(CC(CC)O)nn2)O)ccc(OC(F)(F)F)cc1 97115,CON(C(=O)C=CC(C)NC(=O)CC1CCCC(C)O1)CC1CC=CCC1 97116,C1(CNC(CCNC(C=CC(C)(C)SC)=O)=O)C(C)(C)C1(C)C 97117,N#CC1CCC(C(=O)NCCCCC(=O)NCCN2CCC(O)CC2)C1 97118,C1(NC(c2scc(C(C)=O)c2)=O)CC(NC(c2cncc(C(F)F)c2)=O)CC1O 97119,C1(C)(CN(C(=O)CC2(O)CCC2)C)CCCC1NC(c1sccc1Cl)=O 97120,C(CC(C(=O)N1CC(N2CCCC2=O)C1)NC(=O)Cn1cnnc1)OC 97121,N1(C(C)C)Cc2ccc(NC(=O)Nc3cc(O)nc(=O)n3C)cc2C1=O 97122,c1(OC)ccc(C(N2CC(N(C(=O)Cc3ccc(O)nc3)C)C(F)C2)=O)cc1F 97123,c1(CC2CCN(C(C(C)OCCN(C)C)=O)C2)c(I)ccnc1F 97124,N1(C(C=C2CCC(C)CC2)=O)CC2CCC(CNC(C3CC3(Cl)Cl)=O)C2C1 97125,N(C(=S)N1CCC(CC(C)C)(CO)CC1)c1ccc(OC)cc1 97126,c1(OCC)ccccc1C1(C(=O)NCC(O)CNC(=O)C(C)NC(C)=O)CC1 97127,c1(C(N2CCCC(C)(NC(C(C)c3ccsn3)=O)C2)=O)ccc2[nH]ccc2c1 97128,N1(C(C2CC(=C)C2)=O)CCC(C(=O)NCCC(O)COC)CC1 97129,C1(C2CC2)(CC2N(C(COc3onc(C)n3)=O)CCC2)CCC1.C12(CC1)C(=O)NC2 97130,c1(C(N2CCCCC2C)C(=O)NCCCCCC)cc(OC)ccc1Cl 97131,C(c1cn[nH]c1)=C(C)C(=O)NCCCNC(=O)Cn1cc(CSCCO)nn1 97132,C(=O)(C(F)(F)C1=CCOCC1)N1C2C(NC(c3cc(C)c(C)[nH]3)=O)C(C2)C1 97133,N1(C(C)=O)CCCC1C(=O)NC(C1(O)CN(C(c2coc(N(C)C)n2)=O)C1)C 97134,C(=O)(C(CCNC(=O)C(O)CCSC)OC)NCCC1C(C(=O)OC)C1 97135,c1(C(=O)NCC(C2CC2)NC(C(COC)O)=O)ccc(OC)c(C2CC2)c1 97136,c1(C(=O)NC2C(CNC(c3c(C)c[nH]n3)=O)CCCC2)cc(Cl)ncc1Cl 97137,C1(CNC(CC2CC(=C)C2)=O)CC2(CCN(C(=O)CCc3cc(C)on3)C2)CO1 97138,C1(SCC)CCCN(C(c2cc(N(C3(C(COC)C4CC4)CC3)C)cnn2)=O)C1 97139,Cc1cnsc1C(N1CCCC1CCCNC(=O)Cc1cnn(C)c1)=O 97140,c1(C(=O)NCC2CCCN(C(C(C)OC)=O)C2)ccnc(P(C)(C)=O)c1 97141,c1(NC(C(C2CC(NC(c3ccc(C)s3)=O)C2)F)=O)ccccc1N=[N+]=[N-] 97142,C(=O)(CC(C1CC1)NC(C1CCCN1C(C1CCCO1)=O)=O)NC 97143,c1(OC)ccc(C(=O)NCCC2CN(C(C3C(C)(C)C3(C)C)=O)CCO2)nc1N 97144,N1(C(c2c(CC)cno2)=O)CCOCC1CC(=O)N(C1CCN(C)C1=O)C 97145,c1(C(=O)NCC(C2CC2)NC(c2n(CCC)ncc2)=O)cc(OC)ccc1OC 97146,C1(OC)CN(C(=O)CC(C)SC)CC1NC(=O)CCC1CCCCCC1 97147,N1(C(COCCC#C)=O)CCN(C(C2CC(C)OC(C)C2)=O)C(CS(C)(=O)=O)C1 97148,n1(CC)ncnc1C(C)NC(=O)C(C1CC1)N(C)C(=O)NC1CCCC1 97149,N1(C(CC2(C)CC2(Cl)Cl)=O)CC2CCC1C1CN(C(=O)Cn3cccc3)CC21 97150,N1(C(c2nc(C(=O)O)co2)=O)CCC(O)C12CCSC2 97151,C(=O)(C1CCCc2cccnc21)NCC1CN(C(C2C(C)C2C)=O)CC(C)(C)O1 97152,N1(C(C2(CC=C)CC2)=O)CC(C(=O)NCC2CC(C(C)(C)C)C2)C(F)(F)C1 97153,N1(C(c2n[nH]c(=N)s2)=O)CCC2(CC1)COC(CNC(=O)COCC(F)F)C2 97154,C1(C(N2CCCC(CN(C(=O)CCF)CC)C2)=O)CCC2(CCC2)CO1 97155,c1(C(=O)NC2C(NC(c3cc(OC)ncc3)=O)C2)cc2cc(Cl)ccc2s1 97156,C(=O)(CC1=NN(C)C(=O)C1)NC12CC(CNC(C(CC=C)(C)C)=O)(OCC1)C2 97157,S(=O)(=O)(c1ccc(N2CCC(n3ccnn3)C2)c(Br)c1)N(CCOC)CC1CC1 97158,N1(C(C2C(=C)C2)=O)CC2CCCC(CNC(c3c(CC)noc3C)=O)C2C1 97159,Cc1cccc(C(C(C)C)NC(=O)NCCc2nc(C(C)(C)C)no2)c1 97160,C1(C(C(=O)OCC)CC(=O)OC)CCC(C)CN1C(=O)C=Cc1cccc(F)c1 97161,CCC(CC(C)C)C(=O)NCC1CCCC1C(=O)OC.C12(CC1)C(=O)N2 97162,N1(C(c2cc(C)no2)=O)CCCC(C(=O)NCC23CCCC2C3)C1 97163,C1(CNC(C(CC)OC)=O)CN(C)CCN1C(=O)CCOCC(C)C 97164,c1(OC)ccc(C(N2CCC(NC(c3cnc(C)nc3C)=O)C2)=O)cc1OC 97165,Cc1ccc(F)c(C(N2CC3CCC2(CNC(c2ccoc2C)=O)C3)=O)c1 97166,Nc1cc(C(N2CCN(C(=O)CCc3cnccn3)C3CC23)=O)c(F)c(F)c1F 97167,C1(C(=O)NCC(CO)NC(=O)CCc2cncnc2O)CCC12CCOCC2 97168,N1(C(C2CCN(OC)CC2)=O)CCC2CN(C(=O)C(O)C(F)(F)F)C(C)C12 97169,C1(CC#C)(C(N2CC(O)C(O)C2)=O)CCN(C(c2cc(CC)oc2C)=O)C1 97170,N1(C(C(C)NC(N)=O)=O)CC(NC(=O)C(F)(F)c2nccs2)C(C)C1 97171,C1(OC)(CNC(C2CC(O)C2)=O)CN(C(C2(c3ccccc3)CC2(Cl)Cl)=O)C1 97172,CCC(CC)C(=O)NCC(C)(C1CCC1)NC(=O)Cc1c[nH]nc1O 97173,c1(N(CCn2c(C)ncc2)C)nc(N(C)CCF)c2c(n1)c(C)nn2C 97174,c1(C(=O)NCC(CC)(C)NC(=O)CCCSC)cnc2ncccn12 97175,C1(CCC(=O)NCCN(C(CNC(CCC)=O)=O)CC2CC2)CCCC(O)C1 97176,C(C(N)CC(C)(C)C(=O)N1CCC(N(C)Cc2cccnc2)C1)OC 97177,c1(C(N(C)CC2CN(C(C3CC(N=[N+]=[N-])C3)=O)CCO2)=O)ccn2nccc2n1 97178,c1(OC(N2CC3C(C(=O)NCCC#C)C3C2)=O)ccc(C(=O)O)c(F)c1 97179,c1(C(C(CN)=O)=O)ccc(F)cc1F.C1(=O)CCCC2(CCC2)N1.C1(C)CC1 97180,CCCCC(CC)CC(C(=O)NC)N(C1(C(=O)OCC)CCOCC1)CC 97181,CC(CC(C)(C)C)C(=O)N1CC(NC(=O)C(C)(C)CC2CC2)C(C)C1 97182,c1(C(=O)OC)ccc(NCC=Cc2ccccc2OC)cc1O 97183,c1(C(C(N2CC(NC(CCNC(=O)OC)=O)C2)=O)C)c(F)cccc1F.C1CO1 97184,C1(N(C(C(CSCC)NC(=O)C(F)=CC2CC2)=O)C)CCCC(C)C1C 97185,c1(C(=O)NCC(CCNC(CN(CCC)C)=O)O)c(F)c(F)cc(F)c1F 97186,CC(C)P(=O)(CC(=O)NCC(CNC(=O)CCCF)CO)C(C)C 97187,C1(C(N2C(C(C)NC(c3cc[nH]n3)=O)CCCC2)=O)CNC(=O)CC1(C)C 97188,C1(NC(C2(COC)CC2)=O)CC(C)N(C(=O)C=Cc2c[nH]nc2C)C1 97189,C1(O)(CNC(C=CCOC)=O)CCCN(C(=O)C(C)NC(c2ccccc2)=O)C1 97190,Cc1ccccc1OCCCC(=O)NC1CCCC1NC(C1(O)CC(CF)C1)=O 97191,N1(CCCCOCCC)CC(c2ccccc2)C1COC1CC1 97192,N1(C(c2ccc(C)cc2)C(=O)NCC)CC(C)C(N=[N+]=[N-])C1 97193,C(C(C)(C)C(=O)NCC1CCCC1N)NCC.c1(SC)ccncn1.OC 97194,Cc1cccc(O)c1C(=O)NCC1(CNC(=O)CC2CCOC2)CC12CCC2 97195,c1(C(N2CCC(N(C(C(CC=C)OC)=O)CCOC)C2)=O)cc2n(n1)CCCN2 97196,CCCC(CNC(C1(CC)CCN(C(=O)C(C)=C2CCCC2)C1)=O)CCO 97197,Cc1ccc(C(C)C(=O)N(CC(O)CN(C)Cc2cn(C(C)(C)C)nn2)C)cc1 97198,N1(C(C=CCC)=O)CCCC1C(C)(C)CNC(C1CC(F)C1)=O 97199,C#CCC(C(=O)N1CCN(C(=O)Cc2ncnn2C)CC1)C1CC1 97200,c1(C(=O)NCCC(C)NC(c2ncc(F)cc2N)=O)cc(Cl)cc(Cl)c1 97201,N1(C(CCC2CC(OC)C2)=O)CC2(CCN2C(=O)CSS(C)(=O)=O)C1 97202,C1(CNC(=O)CCOC2COC2)(NC(c2cc[n+]([O-])cc2)=O)CCOCC1 97203,Cc1cn(C)nc1C(N1CC(n2cc(CCn3cncn3)nn2)C(O)C1)=O 97204,C1(CNC(c2c(OC)oc(C)n2)=O)CN(C(=O)CSC(C)C)CCC1C 97205,c1(CC)ccc(C(N2CCOCC2CNC(=O)CC(C)COC)=O)nc1 97206,C1(CC(=O)NC(C)C(C)(C)NC(c2cccc(C(F)(F)F)c2)=O)CCC(=O)N1C 97207,N1(C(c2nccc(C)c2)=O)CCN(C(c2cnc3[nH]cncc2-3)=O)C2CCC12 97208,CC1C=C(C(=O)N(C(C)CCNC(c2ccccc2C(=O)N(C)C)=O)C)CC1 97209,c1(C(=O)NC(CNC(c2c(C)nc(OC)s2)=O)C)cnc(O)c(C(F)(F)F)c1 97210,c1(CC(=O)OCC)cnc(N2CCN(Cc3ccccc3)C(=O)C2)nc1C 97211,c1(C(N(CCCN(C(=O)CC2CCCC3(CC3)C2)C)C)=O)ccncc1N=[N+]=[N-] 97212,C1(CC(=O)NCCOC2CCN(C(c3c(C)cno3)=O)C2)CCC(C)(C)CC1 97213,c1(C(=O)NC2CCN(C(c3cc(OC)cc(Cl)c3)=O)C2C)cccc2cnnn12 97214,c1(NC(C2(CC#C)CCCCC2)=O)cnn2c1N(C)CCC2C 97215,O=C(C(O)CC(F)(F)F)N1CCC2(C1)CN(C(c1ccc(C3CC3)s1)=O)C2 97216,N1(C(C(C=C)(C)C)=O)CC2CCCC(N(C)C(c3nn(C)cc3Cl)=O)C2C1 97217,N1(C(C(CC)COC)=O)CCCC(F)(CNC(=O)Cc2ccccc2OCC)C1 97218,CC1CN(C(C2CC2(Cl)Cl)=O)CC1CCNC(C1CCCCCC1)=O 97219,c1(N2CC(C(C)NC(c3c(OC)cccc3)=O)OCC2)ncc2ncn(C)c2n1 97220,c1(C(C)C)nccn1CC(=O)N(C)CCN(C(=O)CN1CCC1C)C(C)C 97221,C1(CC(N2CC(CNC(c3c(C)onc3)=O)OCC2)=O)CCC2(CCC2)CO1 97222,C(=O)(CC(C)(C)C)NC1CC(C)(CNC(C2C(OCC)C2C)=O)C1 97223,c1(SCCC(=O)NC(COC)CNC(=O)COCC2CCCS2)ccccn1 97224,CC(C(=O)N1CCN(C(c2ccc(C(N)=O)nc2)=O)C(CC2CC2)C1)C(C)(C)C 97225,C(CC(C)C(=O)N1CC(NC(=O)C(c2ccc(O)cc2)=O)C(C)C1)OC 97226,c1(C(=O)NCC2CC(NC(C(c3cccc(Cl)c3)OC)=O)C2)ncccc1F 97227,c1(C(C(=O)NCC2CC(NC(C=CC=CC)=O)C2)C)ccc([N+](=O)[O-])cc1 97228,c1(NC(C(CC)n2cnc(-c3nn[nH]n3)n2)=O)ccc(Br)c2c1CCO2 97229,C=C(C)C1CN(C(=O)C(C2CCOC2)NC(=O)C=CC(=O)NC2CC2)CCO1 97230,c1(OC)cc(OC)nc(N2CC(C)(NC(=O)C(O)C(C)C)C2)n1 97231,C(CC(C)C)(C(=O)NCCC(F)(F)C(C)C)ONC(C1C(CC)N(C)CC1)=O 97232,c1(NC(c2ccc(F)cc2Cl)C)ccc(C=NO)cc1 97233,CC1CCCC1(C)C(N1CCOC(C(C)NC(=O)Cn2cc(N)cn2)C1)=O 97234,c1(OC)cc(OC)c(CNC(=O)C(=O)N(C)Cc2ccc3ncoc3c2)c(F)c1 97235,C1(CCNC(c2cnc(C)nc2C)=O)CCN(C(=O)C(C)CC(F)F)CC1(F)F 97236,CCCCC(O)C(C)C(=O)NCC(F)CNC(C1(COC)CC1)=O 97237,C1(NC(c2ccc(F)c(F)c2)=O)CCN(Cc2nnc(COC(C)C)o2)CC1C 97238,CC(CN=c1[nH]c(=NCc2ccccc2CCO)[nH]c2c1CCCC2)CC(C)O 97239,C1(NC(N(CCCO)CCC)=O)CCCCC1OCC1COC1 97240,C1(NC(=O)Cc2ccco2)COCCN(C(C2CCN(C3CC3)C2=O)=O)C1 97241,C(CCO)(C(=O)N1CCOCC1CCC1CCCN1C(C1CCSC1)=O)N(C)C 97242,C#Cc1cc(NC(=O)C(c2ccco2)NC(=O)Cc2cc[nH]n2)cc(F)c1 97243,c1(OC)ncc(C(=O)NC(C)C(C)NC(c2ccc(F)cc2C2CC2)=O)cc1C 97244,c1(CCC(=O)NCCNC(CCNC(C)=O)=O)ccc(Br)nc1 97245,c1(N2CCN(C(=O)C=Cc3ccc(Cl)cc3Cl)CC2)ncnc2ccc(Cl)cc12 97246,c1(OC)ccccc1C(=O)NC1CC(CNC(=O)CC2(O)CC2)C1 97247,C1(C(=O)NCCNC(c2ccc(CC)cc2F)=O)CC(=O)N(C)C(=O)N1 97248,Cc1ccc(C(N2CCN(C(C3CC4(CCC4)CO3)=O)C(C)C2)=O)cc1Cl 97249,Cc1cc(C(=O)NCC(C2CC2)NC(c2cnn(CCF)c2)=O)n[nH]1 97250,CCC(C#N)C(=O)N1CCN(C(CNC(c2cccn2C(C)C)=O)C(F)F)CC1 97251,C1(CN2CCN(CCn3cc(-c4n(C)ncn4)nn3)CC2)CCc2nnnn2C1 97252,c1(OC)cc(CC(N2CCC(NC(C3CC3C)=O)C2(C)C)=O)ccc1Cl 97253,C(=O)(C(CCc1ccccc1)N1CCOC(CNC(=O)C2CC2)C1)NCCOC 97254,N1(C(C(C)(C)OC(C)C)C(=O)O)Cc2cc(Br)ccc2CC1C(F)F 97255,N1(CCOCC)CC(C(=O)OCCn2cc(C=CSC(C)(C)C)nn2)CC1=O 97256,c1(NC(N2CC(COC)N(CC(F)F)CC2)=O)cc2cc(OC)ccc2s1 97257,c1(CNc2nnc(CC)n2CC(=O)OC(C)(C)C)cccc(S(F)(F)(F)(F)F)c1 97258,CC(C)CC(C)(O)C(=O)N1CCC(N(C(=O)Cn2cnnn2)CCO)C2(CC2)C1 97259,C1(NC(c2ccc(CC(=O)NC)cc2)=O)CCN(C(C2CCCN(C)C2)=O)CC1O 97260,C12(C(=O)NC3CC(CNC(c4cnc(C5CC5)o4)=O)C3)CCCN1CCC2 97261,N1(C(c2cnc(C3CCCCC3)s2)C(=O)NCC=C)CCC(O)CC(C)(C)C1 97262,Cc1nc(NCCC2=CCCC2)cc(N2CCCN(S(C)(=O)=O)CC2)n1 97263,c1(C(=O)NC(C2(O)CN(C(CCCSC)=O)C2)C)ncc(C)cc1[N+](=O)[O-] 97264,C=C(C)CC(C(=O)NCC(=O)NCc1ccco1)NC(=O)CC1(O)CCCCC1 97265,C(C(=O)Nc1noc(C)n1)(C(C)C)NC(CCC)=O 97266,C=C=C(C)CC(=O)NCCN(CC(C)O)C(=O)CC1CC(OC)C1 97267,C(Cc1cc[nH]n1)(C(=O)N(CCCF)CC)NC(C=CC=CC)=O 97268,Cc1cc(Br)ccc1CC(=O)NC1CC1NC(C1(C)CC(C)(C)C1)=O 97269,CCCC(C)(O)CC(=O)NCCN(C(=O)C(c1ccc(SC)cc1)=O)C 97270,Cc1cc([N+](=O)[O-])cc([N+](=O)[O-])c1NC(C)CNC(c1n[nH]cc1Cl)=O 97271,CC(C)C(C)CC(=O)NC1CN(C2CN(C(C3(C)CC=CC3)=O)C2)C(=O)C1 97272,c1(C(=O)NC2CCCCC2C(=O)Nc2ccc(Cl)cc2Br)c(Br)cccc1[N+](=O)[O-] 97273,c1(C(N2C(CNC(CC)=O)CC(C(F)(F)F)C2)=O)cc2c(cc1F)NC(=O)CC2 97274,c1(C(C)(N)C(=O)NCc2ccsc2Cl)cccc(I)c1 97275,CCC(C)CC(C(=O)N(CC(C1CCC1)OC)C)NC(c1cnn(C2CC2)c1)=O 97276,c1(OC)cc(C(=O)NCCC2=CCN(C(=O)CC(C)O)CC2)cc2cnn(C)c12 97277,CC(C)C(C)CC(=O)N(C1CC(C(=O)NCC(O)(C2CC2)C2CC2)C1)C 97278,c1(C(N2CC(CNC(C3CCc4nn[nH]c4C3)=O)C2)=O)cc2n(n1)CC1(CC1)C2 97279,Cc1ccc(C(N2CCOC(C)(CNC(=O)Cc3sccc3Cl)C2)=O)cc1Cl 97280,CC(CN(C)C)CCC(=O)N(CC(C)(C)NC(C1CCC(=O)C1)=O)C 97281,C(CC(C)(C)C)(C(=O)NCC1(O)CCN(C)C1)NC(C=CC(C)(C)SC)=O 97282,C1(C)(C(=O)NC(CC)C(F)(F)F)CCCN(C(c2cc(C)oc2C)=O)C1 97283,C(C)(CC(C)(C)C)(c1ccccc1)NC(C1CCC(F)(F)C1)(c1n(C)nnn1)C 97284,c1(C(=O)NCCN(C)C(c2ccc(Cl)c(Cl)c2)=O)cc2sccc2[nH]1 97285,c1(-c2cccc(OC(C)=O)c2)nc2c(s1)CCN(C(C1C3COCC13)=O)C2 97286,C1(C(N2CCC(CNC(=O)CN3CC4CC4C3)(OC)C2)=O)(COC)CCOCC1 97287,Cc1cc(=NC2CCCn3ccnc32)[nH]c(N2CC3C(CO)C3C2)n1 97288,N1(C(C2C(c3c(C)cccc3)C2)=O)CCN(C(c2nc(O)c(C)s2)=O)CCC1C 97289,C1(C(=O)NC(CNC(c2c(C(=O)OC)scc2)=O)C(C)(C)C)CCCC2(CC2)C1 97290,C#Cc1cccc(C(N2CC=CCC2C(N2CCCC(C(C)(C)C)C2)=O)=O)c1C 97291,Cc1cnn(C)c1C(=O)NCC(CC(=O)NC(C)(C)CC(C)C)C1CCC1 97292,c1(C(N2C(CC=C)(C(=O)NCC3CC(F)(F)C3)CCC2)=O)cc(C)cc(C#N)c1 97293,c1(CCC(=O)NC(C(C)NC(C2(C(=O)N(C)C)CC2)=O)C)ccc2ncccc2c1 97294,c1(C(N2CCC(CNC(c3ccc(CO)o3)=O)C2)=O)snc(Cl)c1Cl 97295,c1(C(=O)NC(C(C)C)CCNC(c2cccc(O)n2)=O)ccc2c(c1)CCOC2 97296,C1(C(=O)NCC2C(NC(c3c(C)cncc3)=O)CCC2)CCC(C2CCCO2)O1 97297,C(=O)(C1=COCCC1)N(C)CC1CCN(C(C(CC2CCC2)OC)=O)C1 97298,C(=O)(C1=COCCC1)N1C(C)CC(NC(=O)Cc2nnn(C(C)(C)C)n2)C1 97299,C(=O)(C1OCCn2ccnc21)N(CCCCNC(C1(C(=O)NC)CCC1)=O)C 97300,C1(CNC(Cn2c(C)ccn2)=O)CCC2CN(C(=O)CCc3nncs3)CC12 97301,c1(-c2onc(-c3cccc(OC)c3)n2)cccc2cc(OC)ccc12 97302,C12(NC(Cc3cccc(COC)c3)=O)CCC(C1)N(C(=O)C(C)NS(C)(=O)=O)C2 97303,CC(F)(F)CCCC(=O)NC1CC(F)CN(C(=O)Cc2c(F)cccc2F)C1 97304,CC1=C(C(=O)NCCN(CCCN(C)C)C(=O)CN2CCNC(=O)C2)CCO1 97305,C1(C(N2C3C(CNC(C(C(C)O)C)=O)CC(CC3)C2)=O)CCc2cnn(C)c2C1 97306,N1(C(C(C)(C)O)=O)CC2CCC1CN2C(C1(C#N)CCC1)=O 97307,C1(C(=O)NC(CCCNC(c2c(Cl)cc(C)s2)=O)C)CCCC2(CCC2)O1 97308,C1(C)(C(=O)NC23CC(NC(CCSC)=O)(C2)C3)C2CCC(C2)C1(C)C 97309,N(C1C(=O)Nc2ccc(F)cc21)C(C1=C(C)OCC1)=O 97310,N1(C(C(N2C(C)CN(c3ccncc3)CC2)=O)=O)CCC(C2(O)CCC2)CC1 97311,CN1CCC1C(N1CCC1C(N1CCC1)=O)=O 97312,CCC(C(=O)OC)C(=O)N1CC(CO)(NC(=O)C=CC2CCCCC2)C1 97313,C1(C(=O)NCC(=O)NCC2CC2)(CC)CCN(C(=O)C(C)CC#N)C1 97314,C(=O)(C1CC(C)(C)Oc2ccccc21)N1CCC(NC(c2n(C)cnc2)=O)C1 97315,N1(C(C(=O)NCC(c2cn(C)nc2)(C)O)=O)CCc2c(ncn(C)c2=O)C1 97316,O=C(C1CCCn2cncc21)NC1CN(C(=O)CC2CCCCC2O)C1 97317,Clc1ccc(-c2nc(CN3CC4CC4C3)n(-c3cccnc3)n2)cc1Cl 97318,N1(C(CCNC(COC)=O)=O)CC(CNC(=O)Cc2ccc(C)s2)C2CC12 97319,Cc1ccc(C(=O)NC23CC2CN(C(c2ncncc2F)=O)C3)c2ccccc12 97320,c1(C(=O)NCC(C)(C2CCC2)NC(CC(CC)C)=O)cnn2c(Cl)cccc12 97321,c1(C(N2C(CNC(=O)C(O)CC3CCCC3)CC(O)C2)=O)c[nH]c2ncccc12 97322,Cc1ccc([N+](=O)[O-])cc1C(N1CC(O)CC1C(=O)Nc1cnc(Br)c(Cl)c1)=O 97323,C1(CC(=O)NC2CC(CNC(C=CC=CC)=O)C2(C)C)CCC(C)(C)CC1 97324,c1(C(=O)NC(CC)(C)CNC(=O)CC2CCC23CCC3)nsc2ccccc12 97325,Cc1[nH]nc(C(=O)NC2CN(C(=O)C=CCF)CC2C(F)F)c1C 97326,N1(C(C(C(=O)OCC)(C)C)=O)CCc2ccccc2C(NC(=O)CCC2CC2)C1 97327,CON(C(=O)C=CC(C)NC(=O)C(CO)N(C)C)C1CCC1 97328,CC1(C)CCOC1C(N1CCCCC1C1CCN(C(=O)C(O)C2CCCC2)C1)=O 97329,C(=O)(CC(O)CC(C)C)NCC(C1CCCCC1)NC(C(CC)(CO)OC)=O 97330,N1(C(CC(C=C)C)=O)CCC2CCCC12C(=O)NCCCC(=C)Cl 97331,C(=O)(C1=NOC(C)(C)C1)N1C(C(C)N2CC(O)C2)CCC1.c1(O)ccccc1 97332,Cc1cc(C(N2CCCN(C(=O)CCN3CCC3)CC2C)=O)cc2c1CCC2 97333,CCC(C)(C(=O)NC(C1CCN(C(=O)C(C)=CC2CC2)CC1)C)C(N)=O 97334,Cc1noc(C)c1CC(C)NCc1cnc(-c2ccccc2F)s1 97335,c1(C(=O)NC(CCCC)CNC(=O)CC(C)C2CC2)cc(C)c(C)c(Br)c1 97336,c1(NC(C)CN(C(=O)CC2CCS(=O)(=O)C2)C)cc2nn[nH]c2cc1[N+](=O)[O-] 97337,N1(CCNC(C2CC(C3CC3)C2)=O)CCN(C(=O)C(O)C2CCC2)CC1 97338,C1(C(=O)OCC)CCCC(NC(=O)C(c2ccc(Cl)s2)C)CC1 97339,c1(OC)cc(C(N2CCC(CO)(NC(=O)CN(C)C)C2)=O)cc(F)c1F 97340,C1(N(C(C=Cc2occ(C)n2)=O)C)CC2CCC(C1)N2C(=O)C(F)(F)C(C)O 97341,c1(CC)c(C(=O)NCC(C)N(C)C(c2cnn(CCO)c2)=O)cnn1CC 97342,c1(CC(=O)NC(CC(C)NC(C(C)(C)OCC)=O)C)c(C)noc1C 97343,C(C)(CO)(CC(C)C)NC(CC1(CNC(C(COCC)C)=O)CC1)=O 97344,Cc1cc(Cl)cc(Br)c1NC(C1CC(C)CN1C(c1cnc(O)cc1O)=O)=O 97345,C(=O)(CS(N)(=O)=O)CCSC(CC1CN(C(CCN(C(=O)OCC)C)=O)C1)C 97346,N1(C(c2ccc(C(C)=O)s2)=O)CCC2CN(C(C3CC(CF)C3)=O)CC12 97347,N1(C(C2(C)CC2(Cl)Cl)=O)CCC(C)(NC(=O)CN2CCS(=O)CC2)C1 97348,N1(C(c2occ(C)c2)=O)CC2(NC(c3c(-c4ccsc4)noc3C)=O)CCC1C2 97349,CCC(C)(O)C(=O)NCCCN(C(=O)CC1CCCS1(=O)=O)CCO 97350,C123CC4CCC(C1C2)N4C3=O.C1(NC(=O)CO)Cc2nnsc2S1.N1CCOCC1 97351,C(=O)(C1CCCc2nncn21)N1C(CNC(C(C)S(N)(=O)=O)=O)CCC1 97352,n1(CCC)cc(C(=O)NCC2CCCC2NC(=O)C(C)SC(F)(F)F)cn1 97353,c1(NC(C2(F)CCN(Cc3ccc(O)c(F)c3F)CC2)=O)c(Cl)cc(F)cc1Cl 97354,c1(C(=O)NCC2C(C)CCN2C(c2ccc(C3CC3)o2)=O)cc(O)nc(O)n1 97355,c1(C(=O)NCCC2CC(NC(C3ON=C(C)C3)=O)C2)ccccc1-n1ccnn1 97356,c1(C(c2cc(C(F)F)no2)=O)ncn(CC2CCCN2)n1 97357,C1(C(=O)NCC(CO)NC(C=COCC)=O)CC2(C1)CC(O)C2 97358,CCCCC(CNC(C1OC(C)CC1C)=O)NC(=O)CNC=O 97359,CC1=C(C(=O)N2CCC(NC(C3CCCC(F)(F)C3)=O)C(F)C2)C(=O)OC1(C)C 97360,N=S1(=O)CCN(C(c2cc(F)c(C(=O)O)cc2F)=O)CC12CCC2 97361,c1(C(=O)NC(CC=C)CNC(=O)CC(C)P(C)(C)=O)ccc2c(O)ncnc2c1 97362,CC(C(=O)NCC1(F)CN(C(c2ccc(Cl)cc2O)=O)C1)C1=CCCC1 97363,c1(C(N2C(C(N3CCCC(C)CC3)=O)CC2)=O)ccc(C#N)cc1Cl 97364,Cc1cc(C(=O)N(CC(O)CN(C)C(C2(O)CCCC2)=O)C)ccn1 97365,CCC(CCC(=O)N1CCC(C(N)=O)C1)NC(=O)C1=CCCC1 97366,Cc1nc(C(C)NC(=O)CC2CCN(C(c3c[nH]c(C(N)=O)c3)=O)CC2)c(C)o1 97367,S(=O)(=O)(c1ccc(C(N2CCCC2C(N2CCCC(F)C2)=O)=O)cc1)NC 97368,CCCCCC(F)C(=O)N(C(C)C(N1CCOC2(CC2)C1)=O)C 97369,N1(C(c2nn(CC)nc2C)=O)CC(C)OC2(CCN(C(=O)C(C)(C)C3CC3)C2)C1 97370,N1(C(C2CC(=C)C2)=O)CC2CC(C1)CN(C(=O)COC1CCC1)C2 97371,C1(C(=O)NC(CCO)C2CCC2)C2CCC(C2)N1C(=O)CC1CSCCO1 97372,N1(C(C(C)Oc2ccccc2C)=O)CCCC(C)(NCCN2CCCC2=O)C1 97373,N1(C(CC2CCN(C(C(C)CC3CCCC3)=O)C2)=O)CCC2(CCCCC2)C1 97374,c1(OC)ccc(C=CC(=O)N(CCCNC(=O)CC2CCCC(C)C2)C)cc1Cl 97375,C(CC(C(=O)N=c1ccn(CCF)[nH]1)NC(=O)C(C)NC(=O)CC)OC 97376,c1(NC(C(N2CC(N(C)C)C2)=O)=O)cc2c(s1)CCC2C(=O)OC(C)(C)C 97377,C(=O)(C1=CCN(C(=O)C(c2ccccc2)F)C1)NC(C#C)CC 97378,c1(C2CCCN(C(=O)NCCC(CC)CO)C2)cc(OC)c(OC)c(F)c1 97379,C(=O)(CCCCC(F)(F)F)N(C1CCCC(NC(COCCOCC#C)=O)C1)C 97380,C1(NC(C(CC)CC(C)C)=O)CCCC2CN(C(c3csc(C(C)=O)c3)=O)CC12 97381,c1(-c2n(CCCOC)nc(-c3cccc4c3CCC4)n2)ccc2nnc(C)n2c1 97382,C(=O)(C(C)C(C)C(C)(C)C)N1CC(CCNC(c2c(OC)cc(F)cc2)=O)C1 97383,CC1(C)CC(CC(=O)NCCOC2CN(C(C3C4CCC(F)C34)=O)C2)C(=O)O1 97384,CC(C)(Cc1ccccc1)CN=c1[nH]c(N2CCC(CF)CC2)nc2c1CSC2 97385,N1(C(c2cn(C(C)C)c(=O)cc2)=O)CCC2CN(C(C3(O)CCOC3)=O)CC12 97386,N1(C(CSc2ccc(C)cc2)=O)CCC(NC(=O)CN2CC(C)C2)CC1C 97387,c1(CC(=O)N(CCCNC(CC(C)OC)=O)C)cccc(OC(F)F)n1 97388,c1(CNC2(c3ccc(C)cc3)CCOCC2)ccc2c(c1)NC(=O)NC2 97389,C1(NC(C#CCNC(C(C(C)C)N(C)C)=O)=O)CCCCNC1=O 97390,c1(N(CCCN(C(=O)COC(F)(F)F)C)C)cc2c(cn1)C(=O)CCC2 97391,C1(CNC(=O)NC2CC2)CCN(C(=O)NC(c2c(Cl)cc(Cl)cc2Cl)C)CC1C 97392,CC1CN(C(c2cnccc2N(C)C)=O)CC2(CCN(C(=O)CSC3CC3)C2)O1 97393,Cc1cc(C(=O)NCCN(C(C2CCC(=O)NC2)=O)C(C)C)cc(C)c1O 97394,C1(C(=O)NCC(C)(O)CO)C2CN(C(=O)Cn3nccn3)CC12 97395,C1(C(N2CCN(C(c3c[nH]cc(Cl)c3=O)=O)CC2)=O)OC2CCC1CC2 97396,N1(C(C2CC(=C)C2)=O)CC2(CNC(c3cc(Cl)ncc3OC)=O)CC1(COC)C2 97397,c1(N(C(CC(CC)C)=O)C2CNCCOC2)nc(C(F)(F)F)cc(C)n1 97398,C=C(C)CCCC(=O)N1CC(C(=O)NC(C)CCCCCC)OC(C)C1 97399,C1(C(=O)Nc2cc(C)no2)CCC2(CN(Cc3csc(N4CCOCC4)n3)C2)O1 97400,CC(C)(CCNC(=O)CN1CC2CC2C1)CN=c1[nH]c2cc(Br)cnc2s1 97401,C1(NC(CC2N(CC)CCC2)=O)CN(C(c2ccc(N)cc2O)=O)CC12CCC2 97402,C1(C(N2C(CCNC(C(C3CCCCC3)OC)=O)CCC2)=O)CCCC1C1CC1 97403,N1(C(c2nc(CC)oc2)=O)CC2(C1)CN(C(=O)C(=O)NOC)C2 97404,Cn1cnc(CC(O)C(=O)NCC(C)(C)NC(=O)CCc2cnoc2)c1 97405,C(CN=c1[nH]n(C)cc1[N+](=O)[O-])C1(C(C)NC(C23CCC(CC2)C3(C)C)=O)CC1 97406,c1(C(=O)NCCCN2CCN(C(C(CC#C)C)=O)CC2)cnn2cccc(C)c12 97407,C(=O)(CCCC(=O)N1CCOCC1C(=O)NCC1(C)CC(O)C1)OCC 97408,c1(C(=O)NCC2CN(C(CN(C)S(N)(=O)=O)=O)C2)cc2n(n1)CCCCO2 97409,C(=O)(C(O)CC(C)C)NC1CC2C(NC(CC(CC)OC)=O)C2C1 97410,CC(=O)C(C(C)C)NC(=O)CN(C(=O)C(C)Oc1cccnc1)C(C)C 97411,c1(C(N2CC(C(C)NC(c3cccn3C)=O)C2)=O)ccc(Br)cc1O 97412,c1(C(C)C)nnc(C=CC(=O)NCCC2(CNC(C3CC4(C3)CC4F)=O)CC2)o1 97413,O=C1COc2cc(NC(c3nc(C(=O)Nc4cncs4)cs3)=O)ccc2N1 97414,c1(C(N(C=O)Cc2ccccc2)=O)cc(=NCCC2CC2)[nH]cc1Br 97415,C#CCC(C(=O)NCC(C)CNC(c1ccn(CC(F)(F)F)n1)=O)C1CC1 97416,C1(CNC(CN(C(=O)CSc2ccccc2C)CC)=O)(CO)CC2CCCC12 97417,C1(C(=O)NCC2(C#C)CCCC2)CCC2(CC2)N1C(c1ccc(C)n1C)=O 97418,C1(CNC(c2cn(C(C)C)c(=O)cc2)=O)CC12CCN(C(=O)C(=O)N(C)C)CC2 97419,C1(C(N(CC(=O)OCC)C)=O)(CNC(=O)CN2CCCC2=O)CC12CCC2 97420,C(=O)(N=c1[nH][nH]c2c1CN(C(c1cn3ccccc3n1)=O)C2)c1c(C)onc1 97421,c1(C(C(=O)OCC(c2cncc(C(=O)OC)n2)=O)(F)F)cc(Cl)nc(Cl)c1 97422,c1(C(=O)NC(C2CCN(C(c3ccc(F)nc3)=O)C2)C)cc2cc[nH]c(=O)c2s1 97423,C(C(CC)(CC)N(C)Cc1ccccc1)NC(C1C(CC(=C)C)COC1)=O 97424,C(=O)(C(C)(C)C(N)=O)NCC1C(NC(C2N(C(=O)NC)CCC2)=O)CCCC1 97425,N1(C(C(C(=O)OCC)OC)=O)CCC(CC)CC1C(=O)Nc1ccc(C)cc1 97426,C1(C(=O)OCC)CCN(C(c2coc(C)n2)C(=O)NC2CCC2)C1 97427,C(=O)(CC1CCNc2ccccc21)NC1(CO)CCCN(C(C2(C#C)CC2)=O)C1 97428,C1(C(C(c2nnnn2C2CC2)NCc2cnc(CC)[nH]2)C)CCCCCC1 97429,c1(C(=O)NC(CC)C)cnc2ncc(-c3cc[nH]c(=NC)c3)cn12 97430,CCC1CC(=O)NC(C)Cn2cc(nn2)COCc2ccccc2C1CCC 97431,N1(C(c2c(C)nc(C(C)C)s2)=O)CCN(Cc2ccncc2C#N)C2CC12 97432,N1(C(C(C(CC)C)N(C)C)=O)CCC=C(C(=O)N2CCC(C)C(CO)C2)C1 97433,C1(C)(NC(C2C(CCC)C2)=O)CCN(C(c2ncoc2-c2ccccc2C)=O)C1 97434,c1(OC)cc(C)c2cc(C(=O)Nc3nnc(C(C)C)s3)[nH]c2c1 97435,C1(C(N(C)CC2CCCCN2C(=O)CN2CCNC2=O)=O)CC2(CC2)CN1C 97436,C(=O)(C1=CCOC1)NC(C1CN(C(=O)Cn2nccn2)CCO1)C 97437,c1(CC(=O)N(CC(C)CNC(=O)C=C2CCOCC2)C)ncn2c1CCCC2 97438,N1(C(c2nc(C)sc2)=O)CC2(CC2)CC1C(=O)Nc1c(F)cccc1Br 97439,C1(C(=O)NC(C2CCN(C(c3cnco3)=O)C2)C)CCCC(=O)N1C 97440,Cc1cnc(F)cc1CN1CCC(N(c2nccn(C)c2=O)C)C1 97441,NC(=O)CCC(=O)NCC1CCCCN1C(C1(F)CCOCC1)=O 97442,CN1CCC(N(C)C(C2COCCC2NC(c2cncc(Cl)c2)=O)=O)CC1 97443,C(C(C)(C)C#CC(=O)NCc1cccs1)NC(c1c(CC)ccc(F)c1)=O 97444,N1(C(C(n2cc(C(C(OC)OCC)C)nn2)C)=O)CC(C)(C)OC(C)(C)C1 97445,N#Cc1ccc(NC(=O)C(=O)NC(C2CCCCC2)Cc2ccccn2)cc1F 97446,C(=O)(C#CC1CCC1)N1CCC(N(C(c2ccc(OC)nn2)=O)C)C1 97447,c1(C(N2CCCN(C(c3cccnc3)=O)CCC2)=O)cc(Br)c2occc2c1 97448,C1(C(=O)NCC2(C(C)C)CC2)CC(N=[N+]=[N-])CN1C(=O)Cn1ncnn1 97449,C1(NC(c2c(C)c[nH]n2)=O)C(C)(C)CN(C(C2CCNC(=O)C2)=O)CC1(C)C 97450,C1(C)(CNC(CC(C)OC)=O)COCCN(C(c2csc(-c3ncc[nH]3)n2)=O)C1 97451,CC1(C)CC(CO)CN1CC(C1CCOC1)F 97452,c1(COC)cc(C(N2CCCC(NC(=O)CC3(CSC)CC3)C(F)C2)=O)cc(Cl)c1 97453,C12(NC(C(CCC(C)C)O)=O)CCCC(CN(C(=O)CNC(=O)C3CC3)C1)C2 97454,c1(SCCN(c2ncc(F)cn2)C(C2CCC(N)C2)=O)cc(Cl)cnc1F 97455,c1(C(N2C(C)CC(CNC(=O)CC3CCC(=O)N3)C2)=O)cnc2c(c1)CCC2 97456,C1(C(N(CCCCNC(C(C2CC(F)(F)C2)OC)=O)C)=O)CCC2CC1CO2 97457,C12(CNC(CCC(=O)N(C)C)=O)CCCC1CCN2C(C1CCCC1)=O 97458,N1(C(=O)NC2(C)CC(C(=O)OCC)C2)CC(c2ccc(OC)cc2)OCC1(C)C 97459,c1(C(=O)NCC(CCNC(c2ccc(F)c(F)c2F)=O)O)cccc2c[nH]nc12 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97566,c1(OC)ccc(CNCc2cc(C(=O)Nc3ncc(Br)nc3I)ccn2)c(Cl)n1 97567,N1(C(CCC(=C)C)=O)CC2(CC(NC(C3CC(O)CN3C(N)=O)=O)CO2)C1 97568,C(C(C)(CSC)CN=c1[nH]c(=NCC(CSC)CO)[nH]c2c(F)cc(F)cc12)OC 97569,C(CC1=CCN(C(=O)Cc2cnccn2)CC1)NC(CN(C)C1CC1)=O 97570,C1(OC)CC2(C1)CC(C(=O)NC1COCCN(C(=O)CSCC3CCCO3)C1)C2 97571,C1(NC(c2c(C)sc(-c3nc[nH]n3)n2)=O)CC2CCC(C1)N2C(C1(SC)CC1)=O 97572,C(=O)(C(C(C)(C)C)N(C)C)NCCSCC(=O)N(C1CN(C)CC1O)C 97573,N1(C(COC(C)C)=O)CCC2CCN(C(c3nc(=O)n(C)[nH]3)=O)C2C1 97574,C(c1c(Cl)cccc1Cl)=CC(N1CCN(C(C2CC2F)=O)C(CF)C1)=O 97575,N1(C(C(C)(C)C)=O)CC(NC(=O)CNC(c2ccncc2)=O)CC(O)C1 97576,c1(C(C)=O)c(NCCCCC(C)NC(=O)CCc2ccc(C)s2)ncnc1Cl 97577,c1(C(N2CC(CCNC(CC3C(CC)C3)=O)C2)=O)ccnn1CC.C(C(F)(F)F)N 97578,c1(C(=O)NC(CNC(C(C2CC(F)(F)C2)OC)=O)C)cnc2c(c1)NCC(=O)N2 97579,c1(OCC)c(C(=O)NC2CCN(C(C3(CF)CC(F)(F)C3)=O)C2)cccc1F 97580,C12(C(=O)NC3CCN(C(CC(CC)C)=O)CC3)CCC(=O)N1CCS2 97581,CN1CCc2cc(C(=O)NC3CC(NC(c4cc(C5CC5)[nH]n4)=O)C3)ccc21 97582,Cc1ccc(C(N2CC(NC(=O)Cc3n[nH]cc3Br)C(C)(C)C2)=O)cc1C#N 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97600,c1(C(=O)NC(CC)CN(C(=O)Cc2cc(C)[nH]n2)C)cccn(C(C)(C)C)c1=O 97601,N1(C(CCC#CC)=O)CCc2ccccc2C1CNC(=O)CCN(C)C(C)=O 97602,N1(C(C2C(C(N)=O)C2)=O)CCCC(CC(N2CC(COC)CC2CO)=O)C1 97603,c1(C(=O)NC2CC(C)(C(N(C)CC3(CC)CCC3)=O)C2)ccc(C)nn1 97604,C1(C(N2CCC(CNC(C3(CC(C)C)CCC3)=O)C2)=O)C2CCCCC12 97605,C1(CC)C(C(N2CC(O)C2)=O)CCN1C(c1cc(C)no1)=O 97606,C1(C(=O)N(CC(O)CNC(C2(CSC)CCOC2)=O)C)(COC)CCCC1 97607,C(=O)(C(CC)C(F)(F)F)NC1CC(CC(=O)NCC2C(C(=O)OC)C2)C1 97608,CCC(CC(F)F)C(=O)N1CCC(C2(NC(c3ccc(CC4CC4)s3)=O)CC2)C1 97609,c1(CC)cc(C(=O)NC2C=CC(CNC(=O)C(F)=CC3CC3)C2)ccn1 97610,c1(C(N(CCCNC(C2CCCC23CC3)=O)CC)=O)ccc(F)c(CO)c1 97611,Cc1coc(C)c1C(=O)NCC1CCN1C(C1(c2ccc(Cl)cc2)CCCCC1)=O 97612,c1(C(=O)NC(CC(=C)C)C(=O)NC2(C)CC2(C)C)cccc2[nH]ncc12 97613,C1(C(=O)NCCNC(c2c(SCCOC)cccn2)=O)Cc2ccc(C)cc2S1 97614,Cc1cnccc1CC(=O)NCCCCC1CCN(C(=O)CCCF)CC1 97615,c1(NCCOC)ccc(C(=O)NC2CCCCC2NC(c2cocc2C)=O)cc1 97616,c1(C(=O)NC23CC(C(=O)NCc4c(C)cccn4)(C2)C3)ccc2c[nH]nc2c1 97617,N1(Cc2ccc(-c3c(CC)ccnc3Cl)s2)CC2CCCC2(CO)C1 97618,c1(NCC)cc(NC(c2n(CC(=C)C)nnn2)CCSC)ccc1C 97619,C=CCC(CNC(=O)C(C#N)C(C)C)C(=O)NC(c1cncn1C)CO 97620,Nc1cncc(C(N2CC(CO)(NC(C3CC3c3cn[nH]c3)=O)C2)=O)c1 97621,C1(NC(C(c2ccccc2)C)=O)CCN(Cc2c(O)cccc2F)CC1O 97622,C(=O)(CC(C)CN(C)C)NCC(=CC(N1CC(F)(CC)C1)=O)C 97623,CCCCC(C(=O)N1C2CCCC1CN(C(C1(C3CCCO3)CC1)=O)C2)C(C)C 97624,Cc1c(C(=O)NCC(C)(C)NC(C2CC(=O)N(C)C2)=O)oc2ccccc2c1=O 97625,C1(C(=O)NCC=CC)CCN(C(=O)C2=CCCC2C)CCO1 97626,C(=O)(CCCn1cncn1)NC(CC)CNCCC(C)(C)C 97627,C=C1CC2(C1)C(=O)NC(C)CCCNC(=O)C1(CC1)NC2=O.C(C)(C)(C)O.C(F)F 97628,CCC(CNC(=O)CNC(=O)OC)(CC)NC(c1cc(C2CCC2)[nH]n1)=O 97629,C#CC1CCC(C(N2CCCC(NC(=O)CCOC(C)C)C2)=O)CC1 97630,C1(NCCSC)CC2CC(NC(C3CC3c3ccc(F)c(F)c3)=O)C2C1 97631,N1(C(C2N(C(C)=O)CC(O)C2)=O)CCC2C(NC(c3ncsc3C(C)C)=O)CC12 97632,CC(C(=O)NC(CC1CC1)C(=O)N(CCS(N)(=O)=O)C)S(C)(=O)=O 97633,C1(NC(CCC#C)=O)CC(OC)CN(C(=O)CCS(N)(=O)=O)C1 97634,CC1CCCC1(C)C(=O)NCc1cccc(CN(C(=O)Cn2cnc(=N)[nH]2)C)c1 97635,c1(C(=O)NC2CC3CC(NC(=O)CN4CCCC4=O)C3C2)occ2c1CCOC2 97636,CC1CN(C)CCN1C(=O)C1=CCCOCC1.C1CCC(F)(F)CC1F 97637,c1(OC)ccc(CC(N2CCC(CNC(C3CC4CCCC34)=O)(OC)C2)=O)cc1 97638,c1(OC)cc(-c2cnc(Cl)c(C(=O)N(CC#N)CC#N)c2)c(F)cn1 97639,O=c1c2ccccc2ncn1SC1CCc2c(F)cccc21 97640,C1(c2cn(C)nc2)CC1C1CC1C(=O)OCc1ccccc1CF 97641,n1(CC)nc(C(=O)NCCC2(NC(=O)Cn3cnc(Br)c3)CC2)cc1C 97642,C(=O)(C(C)(C)C(N)=O)NCC(C(=O)NCC(O)C(F)F)OC 97643,CN1CCOC(CNC2CCC(CNC(c3cnccc3Cl)=O)CC2)C1 97644,C1(C(N2CCCC2)=O)CC=CCC1C(=O)NC1CC2CC2N1S(=O)(=O)CCCCl 97645,c1(C(=O)NC(C(C)NC(c2c[nH]c(Br)c2)=O)C)ccc(F)cc1OC(F)F 97646,c1(OC)ccc2nc(NC(=O)C3=CCCN(CC4CCCCO4)C3)[nH]c2c1 97647,Cc1ccc(C(=O)NCCn2ccc(C(=O)N(C3COCC3(C)C)C)c2)n1C 97648,C1(c2ccccc2)(C(=O)NCC(CCNC(c2c(C)scn2)=O)O)CC(F)(F)C1 97649,c1(OC)cnc(Cl)[nH]c1=NC1CC2CN(C(=O)CCc3ccc(F)cc3F)CC12 97650,Cc1cnc2n1C(C(=O)N1CCC(C)(NC(c3csnc3Cl)=O)CC1)CCC2 97651,C#CCC(C)(C)C(=O)NCC(CNC(c1ccnn1C1CCC1)=O)C(F)(F)F 97652,S(=O)(=O)(c1cccc(Cl)c1)NCC(=O)NCC12N(C(CCC=C)=O)CC(CC1)C2 97653,C12(C(=O)OC(C)(C)C)CCCN(C(=O)O)CC1C2.CCC(C=O)C(C)C 97654,C1(NC(c2[nH]cc(CC)n2)=O)CC2CC1N(C(=O)Cc1cccc(C)c1Cl)C2 97655,N1(C(C(C)N(CC)CC)=O)CC(C2CN(C(C3CC3(C)C(F)(F)F)=O)C2)C1 97656,N1(C(C(C)NC(COC)=O)=O)CC2CC(C)N(C(c3ccccc3)=O)C2C1 97657,O(NC(=O)CCN(C(=O)CC1CCC(C#N)C1)CCO)CCCC 97658,C1(CCCC)CN(C(=O)C(C)CC2CC2)CCN1C(=O)C=Cc1ccccc1 97659,N1(C(CC=CCC)=O)CC(NC(=O)CCC2C(=O)NN=C2C)CC(C)C1 97660,Cc1cc(Cl)ccc1NC(=O)C(C)(C1CCC1)NC(C1CC(CF)C1)=O 97661,N1(C(c2c(C)c(Br)no2)=O)CCC(C)(NC(C2CC(CF)C2)=O)CC1 97662,c1(C(=O)NCCN(C(c2csc(-c3csc(C)n3)c2)=O)CC)nc(C2CC2)cs1 97663,N1(C(C(F)=CC)=O)CCN(C(c2cnc3n2CCS3)=O)C(C2CCCC2)C1 97664,N1(C(Cc2cn(C(=O)OCC)nn2)=O)C(NC(=O)CC(=O)NC)CC2COCC12 97665,N1(C(CCc2cn(C)nc2)=O)CCC2(CCC2NC(=O)C=CBr)CC1 97666,Cc1cc(=NC(C)C2CN(C)CCN2C)[nH]c(=NCc2ccoc2C)[nH]1 97667,c1(C(=O)NC2(C)CCN(C(C(C)NC(C)=O)=O)C2)cc2cc(Cl)cnc2[nH]1 97668,c1(C(N2C(C(N3CC(C#C)C(O)C3)=O)COCC2)=O)cccc2c[nH]nc12 97669,C(=O)(C1CCc2c[nH]nc21)NCCC(C)NC(COCCOCC#C)=O 97670,C(=O)(C(C)C(C)C)NC(C(C)NC(c1n(CC)ncn1)=O)CO 97671,C(CCC(C)(C)C(=O)NCC(C#N)CC)NC(CSCCC)=O 97672,CCCCCCCCC(=O)NC(CC(C)(C)C)C(=O)N1CCOC2CCC12 97673,C1(CNC(CC(C=C)C)=O)CC2CCC1N2C(c1ccc(CO)s1)=O 97674,Cc1cccc(Cl)c1C(N1CCC(N(C(=O)C(C)SC(C)C)CCO)C1)=O 97675,C(=O)(C#CC1CCCCC1)N1C(C(N2C(COC)CCCC2)=O)CC(O)C1 97676,CCC(C)C(C(=O)NCCCCC1CN(C(=O)CC(F)(F)F)C1)OC 97677,C1(C(=O)NC2CCCC2)CCCN1C1CC1.C12(CC1)N(C)C2=O 97678,n1(CC(=O)NCC2(F)CC(NC(Cc3cn(CC)nc3)=O)C2)nc(O)ccc1=O 97679,C1(C(=O)NCC2(O)CN(C(C(C)Cc3ccc(N)cc3)=O)C2)CCC2(CCC2)O1 97680,c1(C(=O)NCC(C2N(C(C(COCC)C)=O)CCC2)(C)C)c(OC)cccc1Cl 97681,c1(NC(C(=O)Nc2cn(CCOC)nc2)=O)ccc(NC(C)=O)cc1 97682,CCCCCC(=O)NC(CC1CC1)C(=O)NC1CC1c1cnn(CC)c1 97683,c1(OC)cc(N)c(Cl)cc1C(=O)NC1(C)CC(NC(=O)C(C)CC2CCCC2)C1 97684,C=C1CCN(C(=O)C(N)=O)C(C(=O)NCC=Cc2ccccc2)C1 97685,C(N=c1nc2sccc2c(NCC2CC(=O)NC(C)C2)[nH]1)c1nc(C)c(C)s1 97686,N1(C(C=CC(=O)OCC)=O)CCC(NC(=O)C=CCOC)C1Cc1ccncc1 97687,CCS(=O)(=O)CC(C)N=c1[nH]c(=NC(C)c2ccccc2Br)[nH]c2ncn(C)c12 97688,CON(CCC(=O)N(C)C)C(=O)NC(CO)CC(C)(C)C 97689,Cn1nccc1C1CC1NC(C1(NC(C2CC2Cl)=O)CC(CO)C1)=O 97690,C1(NC(C=C(C)C2CC2)=O)CC(CNC(c2cc(CO)c(C)o2)=O)C1(C)C 97691,N1(C(c2n(CC)ncc2Cl)=O)CC2CC(C1)N2C(=O)CCN(C)C 97692,CCCC(C(O)C(=O)NCCC1CCC(C)(C)C1)NC(c1cc(C)nnc1C)=O 97693,CCC(C)(C(=O)NCC1(C)CC(F)(F)CN1C(c1ccc(F)cc1)=O)C(N)=O 97694,C12(C(=O)NC3CN(C(C(F)=CC)=O)CC(O)C3)CCC(C)(CC1)OC2 97695,N1(C(C(C)CCO)=O)CCCC(C2CN(C(=O)C(F)(F)C(C)O)C2)C1 97696,O=C(NN1CCOCC1)N1CC2CC(NC(=O)OCc3ccccc3)C(C2)C1 97697,c1(-c2ccc(N(C)C)nc2)ccc(CC(=O)NCc2ccn(C)c2)cc1F 97698,C(=O)(CC(CC)C(F)F)N(CC(=O)NCc1cccnc1)CCC 97699,N1(C(c2oc(CC)c(C)c2)=O)CC2(CC)CC1(CNC(c1sccc1F)=O)C2 97700,C1(CC(=O)NCCSCCC=C)CN(C(c2nnsc2C)=O)C(C)(C)C1 97701,c1(SCC(=O)NC2C3CC2CN(C(=O)CC2(CO)CC2)C3)cc(Cl)ccc1Cl 97702,C1(NC(C2N(CCC)CCC2)=O)CCCN(C(C2(CC)COC2)=O)C1 97703,c1(C(=O)OC)nc(Cl)[nH]c(=NCCNC(=O)Cc2c(C)nc(O)nc2C)c1OC 97704,Cc1cc(=NCCCCC2(C)OCCO2)[nH]cc1S(=O)(=O)N(C)C(C1CCC1)C 97705,CCS(=O)(=O)c1ccc(C(=O)NCC2CN(C(=O)C(C)C(C)O)CCCO2)cc1 97706,C1(C(=O)NC(C(=O)N(CC)CC)C)CN(C(=O)Cc2scnc2C)CC1C1CC1 97707,C(=O)(CC(C)(C)C#N)NCC1CN(C(c2ccc(C(C)C)cc2)=O)CC1C 97708,Cc1ncc(C(N2CC(NC(=O)C3=CCCC3)C(CO)C2)=O)n1C 97709,N1(C(CC2N(C(c3c(C)nc(C)o3)=O)CC2)=O)CC(C)(C)CCC1CO 97710,C1(C2CCC2)(C(=O)NCCCC(C)NC(C2CCCN2C)=O)CCC1 97711,CC(C)CC(C(=O)N1CCC(NC(=O)CCN2CCC(N(C)C)CC2)C1)N(C)C 97712,C1(COC(C)C(N2CC(COC)(NC(C3CCC(=O)O3)=O)C2)=O)CCCCO1 97713,C(=O)(CCCCC(=O)NCC1CCN1C(C1(O)CC1)=O)NC 97714,C1(NC(N2CCC(C(=O)NC)CC2)=O)CN(C(=O)CSC(F)F)C2CCCCC12 97715,c1(C(N2C(CNC(C(C=C)OC)=O)CCC2)=O)cc(C)cc(O)n1 97716,c1(NC(C(c2ccc(SC)cc2)N(C(COC)C)C)=O)ccc(F)cc1 97717,c1(C(=O)NCC=CC)n[nH]cc1CNC(=O)C(C)n1cccn1 97718,c1(C(C)CC(=O)NC(C)CNC(C2(n3ccnn3)CC2)=O)cccc(F)c1 97719,CC1CNC(=O)CN1C(C1(NC(C2CC2C2CCCO2)=O)CC(CO)C1)=O 97720,c1(CC(=O)NCC(CC)(C)NC(=O)C(C)CC(N)=O)sc2ccccc2c1C 97721,c1(C(=O)NC2CN(C(C(c3ccc(OC)cc3)O)=O)CC2C)cc(F)cc(Cl)c1 97722,CC1(C)CC(CNC(c2ccc(-n3cnnn3)cc2)=O)N(C(=O)CCC2CC2)C1 97723,N1(C(C=CC(C)OC(C)=O)=O)CCC(O)(CO)C1.C1(C)(C)C(=O)N1 97724,N1(C(CCNC(C(C)(C)C)=O)=O)CCCC(O)(CNC(=O)CSCCC#N)CC1 97725,C1(CC(=O)NC2(COC)CCN(C(=O)C=CBr)C2)OCCCC1(C)C 97726,c1(CC(=O)NCC(C2CCCC2)NC(CC=C)=O)ccc(Br)cc1 97727,C1(CC)(NC(=O)CCCc2cccs2)CCN(C(=O)C(C)COC)C1 97728,N1(c2nnn(C)n2)CCCCC1CNC(C1COC(=O)N1C)=O 97729,Cc1ncnc(C)c1CC(=O)NCC1CC1CNC(=O)CC#N 97730,CC1CN(C(=O)CC2CC=CC2)CC1C(=O)NC1CC1F 97731,c1(C(N(C(C)CNC(=O)Cc2ccc(OC(C)C)cc2)CC)=O)cn(C)c(O)n1 97732,C1(C(=O)NCC2C(C(F)(F)F)CN(C(CC=C=C)=O)C2)Cc2nnc(C)n2C1 97733,C1(C(=O)NCC(C(=O)OC)O)CCCCN(C(C2(O)CCOCC2)=O)C1 97734,N1(Cc2ccc(OCCCC)cc2)CCC(C2CC(OC)C2)CC1 97735,n1(CC(=O)NCCN(C(C(CC)c2ccccc2)=O)C)c([N+](=O)[O-])cnc1C 97736,c1(OC)cccc(SCCC(N2CC3CC2C3NC(c2cccc(F)n2)=O)=O)c1 97737,C1(c2nc(C)[nH]n2)COCCN1C(c1ccc(Br)cn1)C(=O)NCC(C)C 97738,Cc1ccc(F)c2oc(C(=O)N(CCCNC(=O)C(C)(C)CO)C)cc12 97739,c1(C(=O)NC)ccc(C(=O)NC2CCC2NC(c2cc(O)ccc2Cl)=O)cc1F 97740,C1(CC(C)C)CCN(C(=O)C(CCC2CCC2)NC(=O)COCC2CCOC2)CC1 97741,n1(-c2ccc(C)o2)cc(S(=O)(=O)NC2=NCCCC2)cn1 97742,C1(NC(c2c(C)nc(C)o2)=O)CCC(C)N(C(C2CCN2C)=O)C1 97743,CCCC(C#N)C(=O)NC1(C(=O)NCCCCCC(C)C)CSC1 97744,c1(C2CC(C(N3CCC(OCCNC(CC)=O)C3)=O)C2)cccc(F)c1 97745,O=C(C1CSc2ccccc21)NCc1ccc(OC(F)F)cc1 97746,N1(C(CC2(OC)CCC2)=O)CCCCC1C(=O)N(C1CCC1C)C1CC1 97747,CCC(C(=O)N(CCCN(C(=O)CC1CC(F)C1)C)C)NC(N)=O 97748,N1(C(CCCN(C)C)=O)CC2CCCC(C1)C2C(=O)Nc1n[nH]c(C(F)(F)F)n1 97749,C1(CC)C(=O)NCCN1C(=O)C(F)C(C)CNC(=O)COc1cnn(C)c1 97750,c1(C(=O)COC(Cc2nc(C3C(C)N(C)CC3)on2)=O)c[nH]c2cccnc2c1=O 97751,C(=O)(C1=NOC2COCC12)NC1CCC(C(N(C(C)C(C)(C)C)C)=O)C1 97752,CCCCC(C)C(=O)N1CC(C(C)NC(=O)COCCCNC(N)=O)C1 97753,c1(C(=O)NC(=O)NCCc2c(C(N3C(CC)CCC3)=O)c[nH]n2)cncc(C)c1.C.N 97754,N1(C(C(C)C(F)F)=O)CC(NC(=O)CC2CC(C)(C)C(=O)N2)CC12CCCCC2 97755,N1(C(C2CCN(C)C2=O)=O)CC(C2CCN(C(c3ncn4c3CCC4)=O)CC2)C1 97756,c1(OC)cccc(C(CNC(C2CC2CF)=O)NC(=O)Cc2ccnn2C)c1 97757,C1(CC)CN(C(=O)CCOCC(C)(C)C)CCN1C(c1cnn(C)c1OC)=O 97758,CN1CCC2CCC(C1)N2C(=O)CC1CC(O)CN1C(=O)C1=C(Cl)CC1 97759,Cc1noc(C2CN(C(=O)CC(C)N(C(=O)C(C)OCCN(C)C)C)C2)n1 97760,Cc1cc[nH]c(=N)c1C(=O)NCC1(C)CCN(C(c2c(C)cnn2C)=O)CC1 97761,C1(NC(C2CC(CCC)C2)=O)CC2CC(NC(=O)C(C)Cn3ccnc3)CC2C1 97762,C1(CN(CCOC(c2n[nH]c(O)n2)=O)CC)CCC2CC2C1 97763,C(=O)(CCC(=O)NC(C)C)NC(C(c1ccccc1)NC(c1cnc(C)s1)=O)C 97764,c1(NC(N2C(C)(CC(=O)OC)CC2)=O)cncc(-c2cc[nH]n2)c1 97765,N1(C(CSCC(C)C)=O)CCC(C)C(CN(C(=O)C(C)(C)CC2CC2)C)C1 97766,c1(OC)cccc(C(F)F)c1C(N1CCC(C(C)NC(=O)C(C)C#N)C1)=O 97767,n1(CC)nccc1C(=O)NCC1CC1CNC(=O)CNC(c1cnn(C)c1)=O 97768,c1(C(C)CNC(=O)C(=O)Nc2cnn(-c3nccs3)c2)cccc(O)n1 97769,C=C=CC(C)C(=O)NCC(C)(C)OCCNc1ccc(O)nc1 97770,CN1CCC2(CCN2NC2CC(C(=O)O)C2(C)C)C1 97771,CC(C)C(O)C(=O)NCCCCC1CN(C(=O)C(=O)NCCO)C1.C1(C)CC1 97772,C1(C(=O)NCCCN(C(=O)C=C2CCC(C)C2)C(C)C)CC2(CCOCC2)CO1 97773,n1(CC(=O)NCC(CO)NC(c2n(CC#N)ncc2)=O)nc(C(F)(F)F)cc1Cl 97774,c1(CC)cnc(C(N2CC(NC(c3ccc(OC(C)C)cn3)=O)CC2C)=O)cn1 97775,c1(CC=C)ccccc1C(=O)NCc1nc(CNC(C2CC=CCC2C)=O)cs1 97776,CC(C)C(C(C)NC(c1ccc(Cl)s1)=O)NC(c1cnc(S)[nH]1)=O 97777,C1(C(N(C2CC2C(F)F)CC)=O)CCN(C(=O)COCC(C)C)C1 97778,c1(C(N2CCC(NC(C3CC(C)=C(C)CC3)=O)C2C)=O)cnn2c(C)ccnc12 97779,C1(C)(C(=O)NC(c2cccnc2O)C)C=CCN1C(c1cc(C2CC2)[nH]n1)=O 97780,C(=O)(CCC(N)=O)N(C1CCN(C(=O)C(CCSC)N(C)C)C1)CC 97781,c1(C(=O)NC(C2CCN(C(=O)CSc3ccccc3)C2)C)ccc2scnc2c1 97782,c1(OC)ccc2cnn(CC(N3Cc4ccc(OC(F)F)cc4C3)=O)c(=O)c2c1 97783,CC1CC=CCC1C(=O)NC(c1cnn(C)c1)C(=O)NC1CCC(F)CC1 97784,N1(C(C(CC)C)=O)CCCC12CCN(C(c1ccccc1[N+](=O)[O-])=O)C2 97785,N#CC1(C(N2CCCCC2C(=O)NC2CC(NC(N)=O)C2)=O)CC2CC2C1 97786,c1(C=O)ccc(F)cc1.N1(C(CCC)c2cccs2)CCC(c2cnc(C)s2)C1 97787,N1(C(C=C)=O)CCC2(CCC2)C(NC(C2CCc3cncn3C2)=O)C1 97788,Cc1noc(NC(=O)C(=O)NCc2ccc(CN3CCOCC3)cc2)c1C 97789,c1(NC(C(=O)NCC2CCC(NC(=O)CSC3CC3)C2)=O)ccc(Cl)cc1 97790,N1(C(C(C)O)=O)CCc2nc[nH]c2C12CCN(C(=O)C(F)Cl)C2 97791,C=CCC(Cc1ccccc1)N=c1nc2c(ncn2C)c(NC2C=CCCC2)[nH]1 97792,C(=O)(C#CC1CCCCC1)N(CCCC(=O)NC1(CCNC(C)=O)CCC1)C 97793,N1(C(C2(OC)CCOC2)=O)CC(C)N(C(C2CCCC2c2nn[nH]n2)=O)C(C)C1 97794,c1(C(=O)NC(C)Cn2cc(CCCC(C)O)nn2)ccc2nccn2c1 97795,c1(OC)ccc(C)c(C(=O)NC2(CN(C(=O)CC3CCOC3C)C)CC2)c1 97796,N1(C(C2(CC=C)CC=CC2)=O)CCN(CC(=O)NC(c2nn(C)cc2O)C)CC1 97797,CC(C)(C(=O)NCC(C1CCCC1)NC(=O)Cc1cnc[nH]1)Oc1ccccc1 97798,C12(C(=O)NC3C(CNC(C(C)OCCCC)=O)C3)CC3CC1C2C3O 97799,C1(C2CCOCC2)(C(N2CC(CNC(=O)CCc3ccccn3)C2)=O)CC1(F)F 97800,S(=O)(=O)(c1cc([N+](=O)[O-])ccc1C(=O)O)Nc1c(C(C)(F)F)nccn1 97801,c1(OC)cc(C(=O)NC(C2CCN(C(=O)Cc3sccc3C)CC2)C)ccc1F 97802,C1(CC)CCCC(N(C(=O)CCNC(C)=O)OC(=O)Cc2cccnc2O)CC1 97803,C1(NC(C2(CO)CCCC2)=O)CCCCN(C(C2CN3CCC2CC3)=O)CC1 97804,N1(C(c2nc(COC)sc2)=O)CC2CC1C2CNC(c1n[nH]cc1F)=O 97805,Cc1ccc(F)c(CNC(C2(C)CCCN2C(=O)CCN2CCCC2=O)=O)c1 97806,c1(NC(C=C(C)c2ccco2)=O)c(O)cccc1O.C1(CN)CC1C(=O)N.C12CC1C2=O 97807,c1(OCC)cccc(CC(N2CCC(CCNC(C3(C)CC(O)CN3)=O)C2)=O)c1 97808,c1(OC)c(C(=O)NCC(C)(C)CNC(=O)CCCc2ncc(C)o2)cccc1F 97809,n1(CC)cnc2c(NC3CC(NC(=O)CSCC(=O)OC)C3)ncnc12 97810,C1(C2(C3C(c4ccc(C)cc4)C3)CCC2)CN(C2CC2)CC1(C)C 97811,C1(C(C)C)CN(C(=O)CC(F)(F)F)CCN1C(=O)C(C)OCC(F)(F)F 97812,c1(C(C(=O)NC(CC)(C)CNC(c2n[nH]cc2Br)=O)C)ccc(F)c(F)c1 97813,c1(C(N(C2CCCC2)CCNC(C(C)N(CC(F)(F)F)C)=O)=O)ccc(=O)n(C)n1 97814,C1(C(N2CC3CCC(CC)(C2)C3)=O)Cc2c[nH]nc2CN1C(=O)OC(C)(C)C 97815,Cc1cc(C(=O)NC(Cn2cccn2)C(=O)Nc2cccc(Cl)c2)c(C)o1 97816,C1(NC(C=CCOC)=O)CCC(N(C)C(c2cn(-c3ncccn3)cn2)=O)CC1 97817,N1(C2CCC(NC(C3(C(N)=O)CC3)=O)C2)CCN(C(=O)C=Cc2cnc[nH]2)CC1 97818,C#CC1(C(N2CC(C)(C)C2C2CC2)=O)CCN(C(=O)C=C2CCCCC2)C1 97819,N1(C(CNC(C(CC)C)=O)=O)CC2C(NC(=O)CCCCN3CCCC3=O)C2C1 97820,c1(CC)c(C(=O)NC2CC(N(C(=O)CC3CC(C)=NO3)C)C2)cccc1C 97821,C1(NC(c2c(C)nn(C3CC3)c2)=O)C2CC3CN(C(=O)C(C)(F)F)C1C3C2 97822,c1(C(=O)NC2(CN(C(=O)Cc3cn[nH]c3)C)CC2)cc2cccc(Br)c2o1 97823,c1(CC(=O)OC(C)(C)C)cc(C(=O)NC2CCC2NC(c2csnn2)=O)no1 97824,C(=O)(C(C#N)CC1CC1)NCC(C)(C)NC(C1CC(CCC)C1)=O 97825,c1(CC(=O)NC2C(NC(Cc3cc(C)ns3)=O)COC2)cccc(C(C)C)c1 97826,C1(NC(c2c(OC)cc(C)cc2)=O)C(C)CCN(C(=O)C(C)C2CCOC2)C1C 97827,C1(CNC2CCCCC2)CCN(C(c2nn(C)cc2C)c2n(CC)ncn2)CC1 97828,c1(C(=O)NCCC2CC(NC(=O)C=CCO)C2)ccc2c(n1)OCCO2 97829,C1(C(N(CC(CC)NC(c2cscc2C2CC2)=O)CC)=O)CCC(C)(C)C1 97830,Cc1cccc(F)c1CNC(C1CCCN(C(C2CC2C)=O)C1)=O 97831,CCC(C)(CO)C(=O)NCCC1(NC(C2CC3(C2)CC3(F)F)=O)CC1 97832,c1(C(N2C(Cn3cc(CNC=O)nn3)CCC2)=O)ccc(S(F)(F)(F)(F)F)cc1 97833,CC1CC2(CCN(C(c3ccc(Br)cc3Cl)C(=O)NCc3ccco3)CC2)CO1 97834,N1(C(C(C)CF)=O)CC2CC(NC(=O)CSCc3ccccc3Cl)C1C2 97835,N1(C(CC(C)C)=O)CCCN(C(=O)COCCCF)C(c2ccccc2)C1 97836,C(=O)(C(=O)N(O)C(C)C)NCCCN(C(c1c(C)ccc(C)n1)=O)C1CC1 97837,CC(c1ccccc1)=CC(N1CCC(F)(CNC(C2CC(C)(C)CN2C)=O)C1)=O 97838,c1(CNC2CCC(NC(=O)Nc3cccc(C)c3)C2)cccc2c1OCC2 97839,C(=O)(CCC(=O)CCC(=O)N1CCC2OCCCC2C1)OC(C)(C)C 97840,C12(CNC(C3CC(C)(O)C3)=O)CCC1CCN2C(=O)CCc1ccccc1Cl 97841,C1(N(C=O)Cc2cnc3ccccc3c2)CCCCC(F)(F)C1 97842,CC1CN(C(C2(CNC(=O)CCC3CCCN3C)CCC2)=O)CCN(C)C1 97843,S(=O)(=O)(c1ccc(NCC2(C)CC2(F)F)c(Cl)c1)N1CCCC2(CC(OC)C2)C1 97844,C1(N(C(c2c(CC)ncs2)=O)C)CCC(NC(C2CC23CC3)=O)CC1 97845,c1(C(=O)NC(CNC(c2c(C)ocn2)=O)C(C)C)cnc(OCC2CC2)c(Cl)c1 97846,C12(CNC(c3ccc(F)c(C4CC4)c3)=O)CCC1CCN2C(c1coc(Cl)n1)=O 97847,CC(=O)CCCC(=O)N(CC(=O)NCc1noc2c1CCC2)CC(C)C 97848,c1(C(=O)NCCN(C(=O)C(C)(CC)CO)CCC)ccc(Cl)nc1OCC 97849,N1(C(=O)OC(C)(C)C)CCC2(CCCCN(C(=O)NC3CCCS3(=O)=O)C2)C1 97850,c1(OC)cc(N2CC(C(C)NC(C3(C(F)F)CCCC3)=O)C2)nc(OC)n1 97851,c1(C(N(C(C)CNC(c2cccn2C)=O)C)=O)ccc2oc(O)nc2n1 97852,C1(C(N2CC(CC)(CC)C2)=O)(CF)CCN(C(=O)CC2CC2COC)C1 97853,C1(CC=C)(NC(=O)CCCNC(C)=O)CC2CCC(C1)N2C(c1cnn(C)n1)=O 97854,CC(C)C(F)(F)CC(=O)N1CCN(C(C2CC(CC(F)(F)F)C2)=O)C(C)C1 97855,N1(C(=O)CCn2cccn2)CCN2C(=O)NCCC2C1 97856,C1(=O)CCN=C(NCCF)NC2CC(C2(C)C)N1.c1(C(NC)=O)cccc(C)c1 97857,CC1CN2CCN1C(C(N1CC3CC3(NC(=O)Cn3cccn3)C1)=O)C2 97858,C(=O)(CCC(CC)OC)NC(CCCNC(C1(COCC)CCC1)=O)C 97859,c1(CC)ccc(OC)cc1C(N1CCC(CO)(NC(c2cnc(O)s2)=O)CC1)=O 97860,N1(C(CCCC2(C)N=N2)=O)CC2CCC(C1)C(NC(=O)CC1CC3CC3C1)C2 97861,Cc1ccc(-c2cn(CC3CCCN3C(=O)CSc3cc(C)nn3C)nn2)cc1 97862,c1(C(C)C)ncncc1C(N1CCN(CC(C)NC(=O)CC2(C#N)CC2)CC1)=O 97863,C1(CNC(c2cn(C(C)C)nn2)=O)C2CN(C(=O)C(CO)N(C)C)CC12 97864,C1(NC(CC(C)C)=O)CC(NC(c2ccc(O)c(C(C)C)c2)=O)C12CCOCC2 97865,C1(NC(=O)CCN2CCOCC2=O)CN(C(C2CC3(C2)CC32CC2)=O)CC12CC2 97866,c1(C(=O)NC2CN(C(c3c(C)cc(N)cc3)=O)CC2F)cccc2c[nH]nc12 97867,C1(CNC(C(=O)NC(C)C)=O)CCN(C(=O)CCc2nncn2C)CC1(F)F 97868,c1(NC(N2CC(N(CCCNS(N)(=O)=O)C)C2)=O)ccc(N=NC(N)=O)cc1 97869,CC(C)C(C(=O)NCCOCCO)C(C)NC(C1CC(F)(CF)C1)=O 97870,C=CCC(C)(C)CC(=O)NCC1(O)CC(CNC(C2CCCC23CC3)=O)C1 97871,N1(C(C(=O)Nc2c(COC)noc2)=O)CCOC2(CCc3ccccc32)C1 97872,C1(C(N(C(C)C(=O)NCCCC(C)CO)C2CC2)=O)CCC(=O)N(C)C1 97873,C(C)(CC(=O)N(CC(C)C(=O)NC1(CO)CC=CC1)CCO)OC 97874,CC(C)C(F)(CNC(c1cccc(O)c1F)=O)C(=O)Nc1ccc(F)cc1F 97875,N1(C(CC(C(C)C)C)=O)CCC(CNC(=O)CCCc2ncco2)C(F)(F)CC1 97876,C1(CN=C(NC2C(C)C2)NCc2cccnn2)CCc2ccccc2C1.SC(F)(F)F 97877,CC(=O)CCC(=O)N1CC(NC(C2(c3ccccc3Br)CC2)=O)CC1C 97878,c1(C(c2n(CC)nnn2)NCc2csc(C)n2)cncc(-c2cccc(F)c2)c1 97879,C1(C(=O)NCC2N(C(C(C)(C)C(N)=O)=O)CCC2)CN2CCCC2CO1 97880,C1(C(=O)NCc2c(C)cc(F)cc2)CCC2CN(C(=O)CCN3CCCC3)CC12 97881,N1(C(C(CC)NC(N)=O)=O)CCC(OCCCNC(=O)C=CC(C)CC)CC1 97882,C(=O)(C1CCCn2nccc21)NCC(CNC(c1ccc(=O)oc1)=O)CO 97883,N1(C(C=C(C)C)=O)CC(CO)(NC(C2(C3CCCCO3)CC2)=O)C1 97884,C1(NC(C(CNC(c2nnc(O)nc2O)=O)O)=O)CNC(=O)C12CC2 97885,N1(C(c2c(C(C)C)con2)=O)CCC(CNC(C2OCCCC2(C)C)=O)CC1C 97886,CC(CCNC(C1CCCCC1)=O)CCNC(=O)CCN(c1ccc(Cl)cc1)C 97887,c1(C(C)C)cc(N2CCCC(C3CCCCN3CC3(C(=O)OC)CC3)C2)ncn1 97888,N1(C(C2C(OCC)C2)=O)CC2CCC1CN2C(=O)CCc1cncn1C 97889,Cc1noc2ncc(C(N3CC(NC(c4c(O)cccc4O)=O)C(C)C3)=O)cc12 97890,C12(C(=O)NCC3CN(C(C4C(OC)CC4)=O)CC3C)CCC(N(C)C)(CC1)CC2 97891,C1(C(=O)NC2(CC)CC2)CN(C(=O)Cc2cccs2)CC(C)(C)C1 97892,C1(C(N2C(C(OC)OC)CCC2)=O)C(C)OCCN1C(C1CCNC(=O)C1)=O 97893,N1(C(c2c(C)cc(CO)o2)=O)CC2(CNC(=O)C(C3CCOCC3)O)CCC1C2 97894,c1(CC)nc(C(=O)N(CC(C)O)CCNC(C2C=C(C)CS2)=O)co1 97895,N1(C(=O)Cc2cnsc2)CCC2(CCOC2)C(CNC(C23CCC(C2)C3)=O)C1 97896,N1(C(C23CCCC2C3)=O)Cc2cc(Cl)ccc2CC1CO 97897,C1(CC=C)(C(=O)NC2CC23CC(NCCCc2ccccc2)C3)CCCNC1 97898,c1(C(=O)Nc2cccc(CNC(=O)CCc3nncs3)c2)c(F)ccc(F)c1Cl 97899,O=C1OC(CNC(=NCCc2cccs2)NCC2CC(CF)C2)CC12CC2 97900,c1(C(=O)NCCC(N2CC(O)(CN(C(C(C=CC)O)=O)C)C2)=O)cccc(C)c1 97901,C1(NC(c2n(C(C)(C)C)ncc2)=O)(CO)CCN(C(=O)Cc2ccnc(O)c2)C1 97902,C(=O)(CCC(F)(F)Cn1cc(CC(O)C2CC2)nn1)N(C)Cc1cc(Cl)sc1Cl 97903,C12(CNC(Cn3c(C)nc(C)n3)=O)CCCC1N(C(c1cnc[nH]1)=O)CCC2.C1CC1 97904,C1(C(=O)NC(CC(=O)NC)C2CC2)CCCN(C(=O)CNC(C)=O)CC1 97905,C=CC1(C(N2CCC(O)(CC(C)C)C2)=O)CCN(C(c2ccc(Cl)o2)=O)C1 97906,c1(C(=O)NCCCNC(=O)C=CCN2CCCC2)c(Cl)csc1Cl 97907,CC1(C)CC(CNC(=O)C=CC2CC2)N(C(C2CCC(C)(C)O2)=O)C1 97908,C1(C(N2CCC(NC(C(C)=C3CCC3)=O)C2C)=O)CCOC2(CCC2)C1 97909,C(CCNC(=O)C(C)CC1CCCC1)(C(=O)NC1COCCC1O)OC 97910,CCCC(CCCNC(=O)Cn1nc(C)n(C)c1=O)NC(c1cc(C)[nH]c1C)=O 97911,c1(C(=O)NC)cc(=N)[nH][nH]1.C(C(C)(C)O)N(C(=O)CC1(C)CC1)C 97912,C(=O)(C(C)C(F)(F)C(F)F)NCC(CNC(c1ccc(C(C)C)nc1)=O)(C)O 97913,c1(C(N2CCC3(C(NC(C(COC)O)=O)C3)CC2)=O)ccc(O)c2c1CCCC2 97914,c1(C(C(=O)NCC)NCC)ccc(S(=O)(=O)N(C)C)cc1 97915,N1(C(c2cc(CNC(C(c3cncnc3)C)=O)no2)=O)CC2CCC(CC2)C1 97916,N1(CC2N(C(C(n3cc(C(C4CCOCC4)C)nn3)C)=O)CC2)CCCCCC1 97917,C1(NC(C(N2CCC(C)CC2)=O)=O)CC2CC1N(C(=O)C(C)C#N)C2 97918,CCC(C)(C)C(C)CC(=O)N1CC(NC(c2cc(C(F)(F)F)n(C)n2)=O)C(F)C1 97919,C(=O)(CCCN(C)N=O)N1C(C(C)NC(C2CC3C(C2)C3(F)F)=O)CCC1 97920,CC(C)(CN=c1ccnc(C2CC2)[nH]1)NC(=O)CCCCc1cnn[nH]1 97921,c1(N(c2ccc(Cn3cccn3)cc2)C(C2(C)SCCCS2)=O)ccc(Cl)c(Cl)c1 97922,O(S(=O)(=O)c1cc(Br)ccc1Br)c1ccc(OCC)c(Br)c1 97923,N1(C(C2C(C)(C)CC2)=O)CC2CCCCC2(CNc2ccnc(CO)n2)C1 97924,N1(C(C(C2CCOC2)OC)=O)CCCC1C1CCN(C(C2(OC)CC2)=O)C1 97925,Cc1c(Br)noc1C(=O)NC(c1ccc(-n2cccn2)cc1)C 97926,S(=O)(=O)(c1c[nH]ccc1=NCC1CCS(=O)(=O)N1C)NC(C)Cn1ccnc1 97927,C1(C(=O)NC(C)CF)C2CCC(C2)N1C(c1ncccc1Cl)=O 97928,c1(CC(C)C)cc(C(=O)NC(C2CCOC2)CNC(C2CC(O)C2)=O)no1 97929,C1(C(=O)NC2C(CC)CN(C(C3CCCN(C)C3)=O)CC2)CCC2CCCCN12 97930,C1(C(=O)NCC(CNC(C=C(C)Cl)=O)C)CCCN1C(c1ccccn1)=O 97931,c1(C(N2CCOCC(CN=c3nnn(C)[nH]3)C2)C)ccc(Cl)c(Cl)c1F 97932,c1(C(=O)NCC(C)CN(C)C(C2CC(F)(CF)C2)=O)c(C#N)ncn1C 97933,C1(NC(c2cc([N+](=O)[O-])c[nH]2)=O)CC2CCC1N(C(=O)Cc1ccno1)C2 97934,c1(C(N(CCC(C)NC(c2ccc(C3CC3)o2)=O)C)=O)ncccc1Br 97935,C(C(C)NC(=O)Cn1nc(C)cc1C)(C(C)C)NC(CCC#C)=O 97936,c1(OC(C)C(=O)NC2CC(NC(C3CS(=O)(=O)C3)=O)C(O)C2)cccc(F)c1 97937,C1(CC(N2CCC(CCNC(=O)CN3CCCNC3=O)C2)=O)CC2C=CC1CC2 97938,N1(C(CCOCC#C)=O)CCCC(CCNC(c2cc(CC)[nH]n2)=O)C1 97939,Cc1nc(-c2ncccn2)sc1C(=O)N(CC1CCC(C)CC1)Cc1nccs1 97940,C=CC1(CC(N2CC(CO)(CF)C2)=O)CN(C(C2CCC(C)C2)=O)C1 97941,C1(CN(C(=O)Cn2cccn2)C)CCCN1C(C1(CF)CC1)=O 97942,Cn1ncc2c(NCC3CC3(F)F)nc(N3CC4C5CCC(C5)C4C3)nc12 97943,C#CCCCC(=O)NC1CC=CCC1C(=O)NCc1nnnn1C1CC1 97944,c1(C(=O)NC2C(C)N(C(=O)Cc3cnn(C)c3)CC2)cc2cccnc2nc1N 97945,c1(CNC(C(CC=C)C)=O)ccc(CNC(C2CC(C)N(C)C2)=O)c(F)c1 97946,Cc1cc(CNC2CC3(C2)CC(Nc2cc(Cl)nc(C)n2)C3)cc(O)n1 97947,CC1CC=C(C(=O)N2CC(C)(C)CC2CNC(c2sccc2C(C)(C)C)=O)CC1 97948,C1(CNC(C2C(C)(C)C2)=O)CCC2(CN(C(=O)C=CCCc3ccccc3)C2)O1 97949,N(C(=NCC(C)(C)C1(O)CCC1)N1CCC2(C)C(C1)C2(Cl)Cl)CCSC 97950,C1(CNC(C2(C)C=CCCC2)=O)CC2(CO1)CN(C(C1CSC1)=O)C2 97951,C1(C(=O)NC2(N=[N+]=[N-])CC2)CCC2(CCN(C(=O)COC3CCCC3)CC2)C1 97952,N1(CC(=O)NC(CC)CNC(=O)CCOC(C)C)CCC(C)C1 97953,N1(C(c2c(C(C)C)onc2)=O)CC(C)CN(c2ncnc3c2cnn3C)C(C)C1 97954,C1(CNC(=O)C=Cc2cc(Cl)sc2Cl)CCCCCN1C(c1cnn[nH]1)=O 97955,C1(C(=O)NCC(C)CN(C)C(c2cnc3occc3c2)=O)CCc2nnnn2C1 97956,c1(NC(c2ncccc2Br)c2n(CCSC)nnn2)ccc(C)c(C)c1 97957,CC1CC2(CO1)CN(C(c1coc3c1CN(C(=O)C(C)(C)OC(C)(C)C)C3)=O)C2 97958,c1(C(=O)Nc2cccc(NC(C=CS(C)=O)=O)c2)cc2ccoc2cc1F 97959,c1(C(N2CCCC(NC(CCCC#C)=O)C(F)C2)=O)c(C)nn2c1CCCC2 97960,c1(C(N(C2CCOC2)C)=O)nc2ccccc2cc1[N+](=O)[O-] 97961,C=CCCC(C)(C)C(=O)N1CC2CC2(CNC(c2ccnc3[nH]nnc23)=O)C1 97962,c1(CC(=O)OC(c2ccc(OC)cc2)CC)c(F)cccc1F 97963,c1(C(=O)NCC2C(CNC(c3ccc(SC)cc3)=O)C2)cc(C2CC2)nc(Cl)c1 97964,C1(CC=C)CCCCC1(c1nnnn1CCCF)NC1COCCOC1 97965,C(=O)(CC(C)C(C)(C)C)NC(C1CCCC1)CNC(c1nc(CC)sc1N)=O 97966,c1(OC)cc(C(N2CC(CNC(c3cc(Cl)ccc3O)=O)C2)=O)cc(Cl)n1 97967,C1(CC(=O)OC)C(C(=O)OCC(c2ccccc2)(C)F)C1(C)C 97968,CC1CC(C(=O)N(C2CCCCCC2)CCNC(c2cncc(F)c2)=O)C(=O)O1 97969,N(C1CC(C)n2ncnc21)C(C1CCCN(CCCOCC)C1)=O 97970,C1(NC(Cc2nc(C(C)C)on2)=O)CC(F)CN(Cc2ncccc2CO)C1 97971,c1(-c2ccc(CCCC)cc2)cnc2ccc(C(N3CCCC(CO)C3)=O)cn12 97972,N1(C(C(C(C)C)OC)=O)CC(CNC(=O)C=CS(C)(=O)=O)CCC1C 97973,CC(CN(C)C)CC(=O)NC1(CNC(c2cnc(C3CCC3)s2)=O)CCC1 97974,N1(C(CCC#CC)=O)CCC(CCNC(=O)CSS(C)(=O)=O)C(F)(F)CC1 97975,N1(C(C(COC)OC)=O)CCn2nc(CNC(C34CCCC3C4(F)F)=O)cc2C1 97976,C(C(C)(CO)NC(=O)CCC1(C)CN(C(C2CCN(C(C)C)C2)=O)C1)OC 97977,c1(CC)ncncc1C(N1CCN(C(CNC(C2CC(O)C2)=O)C(F)F)CC1)=O 97978,c1(SCC)ccc(Cl)cc1.C(=O)(CCCOC(=O)C1n2c(cnc2)C(=O)O1)OC 97979,C(CCCC(=O)NC(CN=[N+]=[N-])C(=O)NC(c1ccccn1)C)OC 97980,C(C(=O)Nn1cnn(C)c1=S)N1CC(NC(CCCC#CC)=O)C1 97981,N1(C(CC=CC)=O)CCC2(CCC2NC(=O)COCC)CC1 97982,CC1CN(C(C2(O)CC3CCC2C3)=O)CCC1CNC(=O)CC1CCCCC1O 97983,C1(C(=O)NCCCN(C(C2N(CCC)C(=O)CC2)=O)C)CC2(CCCCC2)CO1 97984,C1(CC(=O)N(CCN(C(c2c(CC)noc2)=O)C)C(C)C)NC(=O)NC1=O 97985,c1(CC)nnc(N2CCC(OCCNC(=O)Cn3cnnn3)C2)o1 97986,N1(C(C(CCC2CC2)NC(C(C(CC)C)N(C)C)=O)=O)CCOC(C)(C)CC1 97987,C(C)(CO)(C(=O)NC1CCN(CCNC(=O)CC2CCC(=O)NC2)CC1)OC 97988,C1(O)(C(=O)NCC(C)(C)NC(c2cnc(CC(C)C)s2)=O)CCCCCC1 97989,CC1(C#N)CC2(CC(NC(=O)NC3COCCC3c3ccccc3)C2)C1 97990,C1(NC(CCCC(=O)NCC)=O)CCN(C(c2ncc(F)cn2)=O)C12CCC2 97991,CCOC(C)(C)c1ccc(NC(=O)NCC(=O)OC(C)C)cc1 97992,N1(C(C(C)CC2CCC2)=O)CCOC2(CCN(C(=O)C(C)(C)c3cc[nH]n3)C2)C1 97993,C=CCCC(C)(C)C(=O)NCC#CC(=O)NCCc1ccsc1 97994,c1(C(=O)NC2C(NC(CCc3ccn(C)n3)=O)C2)cc(N2CCCCC2)ncn1 97995,N1(C(C(F)=CC)=O)CCC(C2CCN(C(=O)CC3C=CCCC3)C2)CC1 97996,C1(N(C(=O)CCC2CCC2)C)CCCN(C(C2(CSC3CC3)CCC2)=O)CC1 97997,C(=O)(CCC(=O)c1ccc(Cl)s1)N1CCC(C(C)NC(=O)C=CC2CCOC2)C1 97998,C(=O)(C1CCc2c[nH]nc21)N1CC(CC(=O)NCCCc2cnn[nH]2)(OCC)C1 97999,CC(C(C)(C)C)=CC(N1CCCC1C(C)(C)CNC(C1OCCC1C)=O)=O 98000,N1(C(c2cccc(CC=C)c2)=O)CC2(C(=O)N(CC(C)C(F)(F)F)C)CC1CO2 98001,Cc1cc(C(N2C(C(=O)NCC3(CO)CC4CC4C3)CCC23CC3)=O)nc(C)c1 98002,CC1=C(C(=O)NC2CCC2NC(c2cnoc2C)=O)CCCC1 98003,c1(NCC2(NC(C3N(C(C)=O)CC3)=O)CCC2)c(C#N)cnc2c(C)cccc12 98004,C1(CCNC(C2(CC(=O)OC)CC2)=O)CCCN(C(=O)Cc2nocc2C(C)C)C1 98005,C1(C(=O)NCC2C(NC(C(C#C)(C)C)=O)CCC2)CCc2nncn2C1 98006,Cc1csc2cc(C(=O)NC3CC3NC(c3cc(F)cc(F)c3)=O)[nH]c12 98007,Cc1cc(Cl)c(NC(C2CC2C(=O)Nc2ccc(C(F)(F)F)nc2)=O)cc1O 98008,c1(C(=O)NCC(=O)NCC(C)CNC(c2ccc(F)nc2)=O)ccc(N)cc1 98009,N(C1CCCc2n[nH]cc21)C(C(c1ccoc1)NC(CC(C(CC)C)O)=O)=O 98010,c1(C(=O)NC2CN(C(C3C(C)(COC)C3)=O)C2)ccc(S(N)(=O)=O)nc1 98011,N1(C(C(C)=C(C)C)=O)CCN(C)CC1CNC(=O)C(O)C(F)(F)F 98012,c1(C2(C(=O)NCC3CCN(S(C)(=O)=O)C3)CCCC2)cc(F)ccc1F 98013,C12(C(N3CC(C(=O)N(C)Cc4cc[nH]n4)(CC)C3)=O)CCCC1C2(F)F 98014,c1(C(N2CCC(NC(C3(C=C)CCOCC3)=O)C2)=O)cc(F)c(F)c(O)c1F 98015,N1(C(CCCC#N)=O)CCCCCC1CNC(=O)CCCn1ccnn1 98016,C(c1ccc(Cl)cc1)(C(F)(F)F)=CC(N1CCN(C(C(C)O)=O)C2(C1)CCC2)=O 98017,C1(NC(C(C2CCC2)OCC)=O)CCCCCN(C(c2cncc(CC)c2)=O)C1 98018,CCC(CNC(c1cccnc1CNC(C1(C)CCCN(C)C1)=O)=O)(CC)CO 98019,N1(CC(C)NC(c2ncnn2-c2ccccc2)=O)CCN(CCCC2CC2)CC1 98020,C1(C(=O)NCc2ocnc2C(=O)N(C2CCCCC2O)C)(CC)CCCCC1 98021,c1(N(C)C)cncc(C(=O)NC2CN(C(c3ccsc3)=O)C3CC23)c1 98022,C1(C(N2CCC(CCNC(C3CN(C(N)=O)C3)=O)C2)=O)Cc2cccnc2C1 98023,c1(NC2(CNC(C(CC)CC(F)F)=O)CCCCC2)nc(O)c2c(ncn2C)n1 98024,Cc1csc2c(C(=O)NC3CCC(CCNC(c4cnc(O)o4)=O)C3)ncnc12 98025,CC1CN(C(C2COC(=O)N2C)=O)CC(C)CN1C(=O)C(=O)Nc1ccccc1 98026,c1(C(N(CCCCNC(Cn2c(C)ncc2)=O)C)=O)cc(F)cc([N+](=O)[O-])c1 98027,Cc1ccc(N)c(C(=O)NCC(C)(C)CN(C(=O)Cc2c(F)cncc2Cl)C)c1 98028,Cc1ccc(SC(C)C(=O)NC2COCC2CNC(=O)CCC#N)cc1 98029,C1(NC(CC=C)=O)CCCN(C(=O)C=Cc2cncc(C)c2)C1C 98030,Cc1nccnc1CNC(=O)CCCN(C(=O)C(C)CC#N)C 98031,c1(C(N2CCC(F)(CNC(C3(COC)CCC3)=O)C2)=O)cccc2[nH]c(=N)oc12 98032,C(CCC(C)CC(C(=O)NCCC1CC1)N(C)CCc1ccccc1F)=C(C)C 98033,CC(CC1CC1)CC(=O)N(C)CCNC(c1cccc(-c2cccs2)n1)=O 98034,CCC(C(=O)NCC(C1CCC1)NC(=O)CCCNC(N)=O)N(C)C 98035,C1(C(=O)NC2C(CC)N(C(=O)CN3CCC(F)CC3)CC2)CC2CC(=O)C1C2 98036,CCC(CO)(C(=O)N1CC(C(N)=O)(CNC(=O)CC2CCC3CC23)C1)OC 98037,C1(NC2(COC)CC(C)SC(C)C2)CCCC1C1CCCC1 98038,C(C(=O)N1CCCC(CNC(C2(C(F)(F)F)CC2)=O)C1)(C(C)O)NC(C)=O 98039,C1(C(N2CC(NC(N)=O)C2)=O)(CNC(C2C(C)(CC)C2)=O)CC(C)(C)C1 98040,C1(NC(c2c(C)ncnc2)=O)C2CCCN(C(c3nccn3C)=O)C2C1(C)C 98041,Cc1cc(NC(C2CN(C(=O)CCc3cc(F)cc(F)c3)CCO2)=O)cc(F)n1 98042,c1(CC)ccnc(C(N2CC(N(C)C(c3cc(Cl)c(Cl)s3)=O)C2)=O)c1 98043,C12(NC(c3c(CC)oc(C)c3)=O)CCN(C(=O)Cn3nc(C)cc3C)CC1C2 98044,C1(NC(C(c2cccc(F)c2)C)=O)CC(F)(F)CC1NC(c1cc(C#N)c[nH]1)=O 98045,N1(C(CC2CCCN(C(C3(C)CCCCC3)=O)C2)=O)Cc2n[nH]cc2C1CO 98046,C=CCC(C(=O)NC1CC2(CCN(C(=O)CN3CCSCC3)C2)C1)C(C)(C)C 98047,N1(C(c2c(Cl)cc(C)s2)=O)CCC(NC(C2SC3C=CC2CC3)=O)C(CO)CC1 98048,C1(C(F)F)(OC)CC(C(=O)NCCC2CN(C(=O)CC3CC3C)C2)C1 98049,c1(C(=O)NC2(C)CN(C(C3CCCCC3C3CC3)=O)C2)cccc2[nH]ccc12 98050,N1(C(C(CCC)C)=O)CC(C)(C)OC2(C1)CN(C(c1nccn3nccc13)=O)C2 98051,c1(CCC(=O)NCC(C)(C)OCC(=O)N(CCCC)C)cccn1C 98052,C1(NC(=O)CC2CCCNCC2)CCCC(NCc2ccccc2)C1 98053,N1(C(c2c(CC)ccc(F)c2)=O)CC2CCC(C1)N2C(c1cc(Cl)c(Cl)s1)=O 98054,Cc1nn(CC(C)C)c(Cl)c1C(=O)NCC(C1CC1)NC(C1CCC(O)CC1)=O 98055,c1(C(N2CCCC(N(CC(CC)C)C)C2)=O)c(O)cc(=O)n2c1COCC2 98056,C1(NC(C(C)N2CCC2)=O)CC(C)CN(C(c2cccc(Br)c2F)=O)C1 98057,c1(CCC(=O)NC2(C)CC2C(F)(F)F)ccc(O)cc1 98058,C(=O)(C(C)CS(C)(=O)=O)NCCCC(C)NC(c1ccccc1[N+](=O)[O-])=O 98059,n1(C(C)C)cnc2cc(NCC3CCC4(CCOCC4)C3)ccc12 98060,N1(C(c2cn(C)c(O)n2)=O)CCC2CCCC12C(=O)N(C)C 98061,c1(C(=O)NC2CCC(CNC(C3(C=C)CCC3)=O)CC2)c(C)ccc(Br)c1F 98062,c1(CC(=O)NCC(CC=C)NC(=O)Cc2cncn2C)ccc(Cl)c(C)c1 98063,Cc1cccc(C2(N(S(C)(=O)=O)C)CC2)c1.c12nnc(n1CCC#N)C2 98064,c1(C(=O)NCC2(C)CN(C(=O)C(F)Cl)C2)cccc2c1OC(F)(F)O2 98065,C1(CC=C)(C(=O)NC2CCC(CNC(C3(O)COC3)=O)C2)CCOCC1 98066,C=CC1CCCN(N2CCOCC2c2cccc(C)c2C)C1 98067,N1(C(C2CC(O)(CC#C)C2)=O)CCOCC1CNC(c1c[nH]nc1F)=O 98068,CN1CC=CCC1CC(=O)NC1CCCCC1NC(c1ccsc1C(F)F)=O 98069,c1(C(N2CCC(C)CC2C(=O)NOC(C)(C)CO)=O)c[nH]c2ccccc12 98070,c1(C(=O)NC2CC(NCc3cc(C)[nH]c3C)C2)c(F)c(F)c(O)c(F)c1F 98071,c1(NC(C2CCN(Cc3ccc(N4CCCCC4)cc3)C2)=O)ncc(F)cc1O 98072,NC1COC2(C(=O)NCC3CN(CCCO)CCO3)CC1C2 98073,C1(OC)CCn2cc(C(=O)NCC3CC3NC(=O)Cn3ncnn3)nc2C1 98074,C=C(C)C(CC(=O)N1CCCC1CN(C(=O)CC1(O)CCC1)C)OCC 98075,c1(CC)nc[nH]c1C(=O)NC(C)CCN(C(=O)CC1(N(C)C)CCC1)C 98076,C12(C(=O)NCC3OCCN(C(c4ncn(C(C)(C)C)n4)=O)C3)CC(C1)S(=O)(=O)C2 98077,C1(C(NOCCC(=C)C)=O)CCN(C(=O)Cc2cccnc2)CC1O 98078,C(=O)(CS(=O)(=O)CCC(F)(F)F)NCC(C)(C1CC1)NC(C1ON=C(CC)C1)=O 98079,N1(C(C(C=C)O)=O)CC2CCC(C1)N2C(=O)CSc1nnc(S)s1 98080,C(=O)(CC(C)(C)CNC(=O)C=CC1CCCCC1)N(CC)Cc1ccn(C)n1 98081,CC(CN(C)C)C(=O)NC(C1CCCN1C(=O)C=CCO)C 98082,N1(C(c2cc(C)oc2)=O)CC2CCCC2(Nc2ncncc2I)C1 98083,c1(C(=O)NCCCN(C(C2C(CCC)CCC2)=O)C(C)C)c(C)n[nH]c1C 98084,CC1(C)C(CNC(=O)CCCCCNC(=O)CCCC2CCCC2)CC1(F)F 98085,C1(NC(c2cncc(C)n2)=O)CCSC12CN(C(c1cc(C(F)F)ccn1)=O)C2 98086,C12(C(=O)Oc3cn(COC)nn3)CC(C(N3CCC(N(C4CC4)CC)C3)=O)C1C2 98087,C1(C(=O)NCCC(CCC)C2CC2)CN(C(=O)C(C)(C)C(C)O)CC1(F)F 98088,C(C(C)(C)CN=c1cccc(S(=O)(=O)NCC2CCCSCC2)[nH]1)OC 98089,N1(C(C2CCCN(Cc3cc(B(O)O)co3)C2)=O)CCCC2(CCNC2=O)C1 98090,C(=O)(C(C)(C)C)NCCC(=O)NCCN(C(CSCC=C)=O)C1CC1C 98091,c1(C(=O)NCCCNC(c2nc(CCC)oc2)=O)cncc(C(C)=O)c1 98092,c1(C(N2C(CN(C)C(c3cc(Cl)no3)=O)CCC2)=O)cnc(Cl)cc1N 98093,c1(C(=O)NC(CSCC)C(N2CCC(NC(N)=O)CC2)=O)cnc(F)cc1C 98094,C(C(C)CN=c1[nH]c(=NCCS(=O)(=O)CCO)[nH]c2cc(C)ccc12)OCC 98095,Cc1ccc(C(=O)N(CC(C)O)CCNC(C2CCCO2)=O)nc1 98096,S(=O)(=O)(c1ccc(NCC(Cc2ccccc2Br)OC)cc1Cl)N(CC=C)CC 98097,CN1CCN(C(=O)CC2CCCN2C(=O)CCc2ccoc2)CC1C1CC1 98098,c1(N2CC(C(N)=O)(CNC(c3ccc(-c4cnco4)cc3)=O)C2)ccnc(C#N)n1 98099,C1(O)(C(N2CCC(N(C(=O)C(C)O)CCOC)CC2)=O)CCC(C)CC1 98100,N1(C(C(=O)N(C)C)=O)CCOC2CCN(C(C3SCCCS3)=O)CC12 98101,Cc1ccc(C(N2CC(CNC(=O)C(C)NC(C)(C)C)C2)=O)c2cccnc12 98102,c1(C(N2CCN(C(C3C(C)(C)C(=O)C3)=O)CC2CCO)=O)cnn2cccnc12 98103,N1(C(C(C=C)OC)=O)CC2(C=C(C(=O)N3CC(CO)C(C)(C)C3)CO2)C1 98104,C1(CNC(c2ccnc(S)c2)=O)CC12CCN(C(=O)CS(=O)(=O)C1CC1)CC2 98105,C(=O)(CC(C)C(C)(C)NC(=O)CCc1cc(C)[nH]n1)N(CCOCCO)CC 98106,Cc1cc(N2CCOC2=O)ccc1N=c1[nH]c(N(C)C)nc2c1CCCCCC2 98107,C1(CCNC(CC=C=C)=O)CCCN(C(=O)CC2(C#N)CCOCC2)CC1 98108,C(=O)(CC(C)(C)C(C)(F)F)N1CCC(N(C(CCC(C)C#N)=O)C)CC1 98109,C1(CNC(C2(N(C)C(C3(C4CC4)CC3)=O)CCC2)=O)CCCC1(C)C 98110,C1(C(=O)NC2CCNC2=O)CN(C(c2ccc(Br)c(F)c2F)=O)CC(F)(F)C1 98111,C1(C(=O)NCC2C3CN(C(c4cnn(CC)c4Cl)=O)CC32)COCCN1C=O 98112,C#Cc1ccc(CC(N2CC(NC(=O)C(C)CC(C)C)C2)=O)cc1 98113,C1(C(N(CCNC(COCC)=O)C)=O)(NC(=O)OC(C)(C)C)CCN(C)CC1 98114,C(C1CCCCC1)=CC(=O)NCC1C(NC(c2cc(C(C)C)no2)=O)CCC1 98115,CCCCC(F)C(=O)N1CCC(C(=O)N(CCOC(F)F)CC)(CC)C1 98116,CC(CN=c1[nH]c(=NCc2ccnn2CC(F)F)[nH]c2cc[nH]c12)S(C)(=O)=O 98117,c1(C(=O)NC(CCCNC(C=CCCC(C)C)=O)C)cc2scnc2[nH]1 98118,C1(C(=O)NC2(COC)CN(C(C3(SC)CCC3)=O)C2)CC2CC1CC2O 98119,c1(-c2cnc(C(=O)Nc3c(OCC)nccc3C)nc2)ccc2nc(C)oc2c1 98120,c1(C(=O)NCCN(C(C(C=C)(C)C)=O)CC)cc(=O)n2nccc2[nH]1 98121,C1(C(=O)NCCOCCN(C)C(c2cc(C(F)(F)F)nn2C)=O)CCC12CCCO2 98122,CCCC(C(=O)NCCCCCN(C(=O)C(C)OC(C)(C)C)C)OC 98123,C1(O)CCCC(OC)C1.c1(C2(C(C(CC(C)OC)=O)=O)CCC2)ccc(Br)nc1 98124,C(C(CCO)C(C)(C)C)ONC(=O)Oc1c(C)scc1 98125,c1(C(N(C2CCN(C(=O)CN(C)CCO)C2)CC)=O)ccc(Cl)nc1OC.N(C)(C)C 98126,C=C(C)CC(C(=O)NC(C1CN(C(c2cccn2C)=O)CCO1)C)NC(C)=O 98127,C1(CNC(C2CC(CC)C2)=O)CN(C(c2cc[nH]c2C)=O)CC12CCC2 98128,c1(CC(=O)NCCC(C)N(C(=O)C(c2ccccc2)O)C)cccc2c1OCO2 98129,Cn1cc(Br)cc1C(=O)NCC1CCN1C(=O)CC1(O)CCCCC1 98130,c1(C(=O)NC(CC)CNC(=O)C2=C(C)OCC2)cc2c(Cl)c(F)ccc2[nH]1 98131,c1(C(N2CCC(O)(CN(C(CCSC)=O)C)CC2)=O)ccc(F)c2c1OCC2 98132,C1(C(=O)NC(CC)CN(C)C(c2cc(C3CC3)[nH]n2)=O)OCC2CCCC12 98133,C(=O)(CS(=O)(=O)C1CCCC1)NC(C(CO)NC(C(C(CC)CC)C)=O)C 98134,C1(NC(CC(C)(C)SC)=O)CC(O)CN(C(c2cccc(O)c2Cl)=O)C1 98135,C1(NC(c2c(C)nc(O)[nH]2)=O)CC2CCC1CN(C(c1csc(=N)[nH]1)=O)C2 98136,c1(C(=O)NC2CCOC2C(N2CC(SC(F)F)C2)=O)cncc(O)c1 98137,Cc1nc2cc(C(=O)NC3CN(C(=O)C(C)N(C)C)CC4CCCC34)cnc2[nH]1 98138,c1(C(=O)NCCN(C(=O)C(F)(F)C2CC2)CCOC)c[nH]cc(C)c1=O 98139,C=C=CC(C)C(=O)NC1(C(N2CC(N3CCCCC3)C2)=O)CC1(C)C 98140,c1(C(N2C(CNC(Cc3c(C)n(C)cn3)=O)C(C)CC2)=O)cnc(Cl)cc1N 98141,c1(C(=O)NCCC2(CNC(CC(C)c3ccco3)=O)CC2)nccc2ccsc12 98142,Cc1cc(=O)c(NC(=O)C(C(C)NC(c2csc(Cl)c2)=O)C(C)C)c(C)[nH]1 98143,C12(CCOC1)C(=O)NCCN(C)C2=O.c1(C(C)OC)nc(C=O)co1.C1CC1 98144,c1(CC)noc2ncc(C(=O)NCC(F)CNC(c3cscn3)=O)cc12 98145,c1(C(C(=O)N(CC(CN(C)C(c2cnc(O)o2)=O)O)C)(C)C)ccc(O)cc1 98146,c1(NC(C(Cc2cc[nH]n2)NC(C(C)=C2CC2)=O)=O)ccc2c[nH]nc2c1 98147,N1(C(C(C2CN(C(CCNc3cc(C)[nH]n3)=O)C2)O)=O)CC2C(C1)C2(F)F 98148,c1(C(N2CCC(N(C(CC=C(C)C)=O)CCO)C2)=O)cc2ccsc2n1C 98149,Cc1cc(O)ccc1C(N1CCC(NC(=O)C(=O)Nc2c(F)cccc2F)C1)=O 98150,C(=O)(CCCCCCNC(=O)Cn1ccccc1=O)NC(C)C(C)(C)O 98151,N1(C(COC(c2nccn2C)C)=O)CCN(C(=O)CC2C=CCC2)CC(C)(C)C1 98152,N1(C(CCN(C(C(C)OCC=C)=O)CC2CC2)=O)CCC(O)(CN(C)C)C1 98153,C1(OC)CC(NC(=O)Nc2ccnn2C2CNC2)CC1OC 98154,c1(C2C(=O)N3CCC(C3)CO2)ccccc1.c1(O)ccccc1.CC(C)O 98155,c1(C(C)C)ccc(Cl)cc1C(=O)N(C(C)CNC(=O)Cc1cnoc1)C 98156,C1(C(=O)NCC2CCCN(C(C=C(C)C(F)F)=O)CC2)CCC2(CCOCC2)O1 98157,C(=O)(C1=CCCCO1)NCC1C(C)CCN1C(=O)C(C)(C)OCC(F)(F)F 98158,N1(C(c2n(C)cnc2)=O)CCN(C(=O)CCC2CC(C)(C)CO2)CC(C)(F)C1 98159,C1(C(=O)NC(c2ccccc2)CNC(CCSC)=O)CC(=O)C12CCCC2 98160,c1(NC(C(C2CCN(C(c3c(C)csc3C)=O)C2)C)=O)cccc(F)c1C 98161,O(NC(=O)CCc1cnc(C)s1)CC(=O)NC(CCC)C1CC1 98162,c1(CC(=O)N(CCCNC(=O)CCc2ncccn2)C(C)C)cn(C)nc1Cl 98163,O=C(CS(=O)(=O)N1CCOCC1)NCC1CC(O)CN1C(=O)C=CC1CCCO1 98164,C(=O)(CCC(C)(C)F)N1CC(C2N(C(c3cc(C)n(C)c3)=O)CCC2)(O)C1 98165,N1(C(c2n(C(C)C)ncn2)=O)CC(NC(c2ccccn2)=O)C(CC(C)(C)C)C1 98166,Cc1cc(S(=O)(=O)NCC(C)(C)CN)cnc1C(F)(F)F 98167,C=CCC(CNC(=O)CC1CC(C)(O)C1)NC(=O)Cc1coc(-c2cccs2)n1 98168,N1(CCOC)CC(C(=O)NCC2CCC2NC(c2cc(C)ns2)=O)CC1=O 98169,c1(C(N(CCN(C(Cc2cc(C)[nH]n2)=O)C(C)C)C)=O)cc(C)c(N)cc1F 98170,N1(C(CN(C)C(C2CCC3(CC3)C2)=O)=O)CCC2(C=CCO2)C1 98171,CC1(C)CCc2nc(Cl)nc(N3CCC(C4CCCN4)C3)c2C1 98172,n1(CC(N2CCC(CN(C(C3C(C)OCC3)=O)C)C2)=O)nc2ccccn2c1=O 98173,C(=O)(C(C(C)CC)N(C)Cc1ccccc1Br)NCC(=C)C 98174,N1(C(C2CC3CC3C2)=O)CCC2CN(C(=O)CC3CC3Cc3ccccc3)C2C1 98175,C(CC(C)(C)C(=O)N(C)Cc1ccccn1)NC(C(C(C)C)C)=O 98176,C1(C#N)(C(=O)NC2CCN(C(c3c(Cl)nc(OC)s3)=O)C2)CC12CCC2 98177,N1(C(CC(CC)(C)C)=O)CCC2(CC1)CC2CNC(=O)CCn1nc(C)nc1C 98178,C1(NC(CC2N(CCCC)CCOC2)=O)CCN(C(=O)OC(C)(C)C)C(C)C1 98179,C1(C(=O)NC(CC)C)C2CCN(C(C3CCN(C(N)=O)CC3)=O)CC12 98180,c1(C(N2CC(OC)C(NC(=O)C3=COCCC3)C2)=O)ccc2[nH]c(=N)[nH]c2c1 98181,c1(C(N2C3(CN(C(C4CCCN(C)C4)=O)C3)CCC2)=O)c(O)cccc1[N+](=O)[O-] 98182,c1(CCNC(C(CC)O)=O)ccc(CNC(c2cscc2C)=O)cc1 98183,C1(CNC(c2c(C(C)C)nns2)=O)C2CN(C(C3CCCN3S(C)(=O)=O)=O)CC12 98184,C(=O)(C(CC)C(C)O)NC1(CC=C)CCN(C(=O)CCc2ccc(O)nn2)C1 98185,CCCC(C(=O)N1CC(F)(CNC(c2nccnc2C)=O)C1)NC(N)=O 98186,C1(NC(C(CC)C)=O)CCCCCC1C(=O)NCc1ccc(Cl)cc1 98187,N1(C(C2C(=C)C2)=O)CCC2CN(C(=O)CCCOc3ccccc3Cl)CC2C1 98188,C1(C(N2CC3CC3(C(=O)NC3CCC3)C2)=O)CCC(C(F)(F)F)CC1 98189,C(=O)(C1CCCc2nc[nH]c21)N1CCC(C)(NC(c2cccc(N)c2O)=O)C1 98190,C1(C)(C(=O)NC2CN(C(C3CCCC(C)(C)C3)=O)CC23CC3)CCCCNC1=O 98191,N1(C(Cc2c(C)ocn2)=O)CC(NC(C2CC3CC3C2)=O)CC(C)C1 98192,C(=O)(C#CC(C)(C)CNC(C1COCCN1C)=O)NCC1(C)ON=C(C)C1 98193,c1(NC(c2[nH]cc(C#N)n2)=O)ccc(F)cc1F 98194,C1(CC(=O)NCc2n(CC)ncn2)CCN(C(c2ncc(C)cc2F)=O)C1(C)C 98195,N1(C(COCCCC)=O)CCN(C(=O)CC2COC(C)(C)CO2)C(C2CCC2)C1 98196,C1(C2CCC2)(C(N(CCCNC(C(C(C)C)CO)=O)C)=O)CC1(F)F 98197,c1(C2C(NC(=O)NC3(C)CCOC3)C2)ccnc(F)c1 98198,c1(N2CC(C)(COC)C2)ncc(C(F)(F)F)cc1Cl.C12(CC1)C(=O)N2C.C=O 98199,c1(C(=O)NCC2C(C)CN(C(=O)C3=CCCCO3)C2)occ2c1CCCC2 98200,c1(CN2CCC(CC(=O)N(CC=C)CC3CCOC3)C2)c(F)cccc1F 98201,C1(C(=O)Nc2c(CC)n(CC(C)C)nc2)CCC2(CC1)CCC2N 98202,c1(C(N2C(CNC(c3cncc(C)c3)=O)CC(C)(C)C2)=O)cncc2nc[nH]c12 98203,CCC1=C(C(=O)NC2C=CC(CC(=O)NCCC(C)(O)C3CC3)C2)CCCO1 98204,c1(C(N(CCCNC(=O)CCCc2cnn[nH]2)C)=O)ccc2oc(O)nc2n1 98205,N1(C(c2ccc(CC)o2)=O)CCCN(C(c2ccsn2)=O)CC1CO 98206,C1(CC)CN(C(c2cn(CCC(C)C)nn2)=O)CCN1C(=O)C(=O)NCC(F)F 98207,c1(NC(C2CC(NC(C3N(C)CCCC3)=O)C2)=O)c(C#N)ccc2ccccc12 98208,Cc1nc(C(=O)NC(C2CCOC2)CNC(=O)C=CCOC(C)(C)C)cn1C 98209,CC1(NC(c2cn(Cc3ccccc3)nn2)=O)CN(C(c2cscc2F)=O)C1 98210,C(=O)(C1CCCc2c[nH]nc21)N1CC(CCNC(C2CCCC(C)(C)CC2)=O)C1 98211,C1(CNC(COC2(C)CN(C(c3c[nH]c(C#N)c3)=O)C2)=O)CCCC(F)C1 98212,CCCN=C(NCCN1CCCCC1)NC1CCCC1c1ccccc1.C1CS1 98213,c1(OC)cc(CCC(=O)NC2CCCN(C(C3CCOC3C)=O)C2)ccc1Cl 98214,Cc1cc(C(=O)NCc2c[nH]nc2C2CCN(C(C3(O)CCOC3)=O)C2)sc1C 98215,c1(C(=O)NC(CNC(C=CSC)=O)(C)C)cnc(O)c(Cl)c1 98216,c1(C(=O)NCC(C(C)C)NC(C(CC)N(C)C)=O)cc2ccccc2n1C 98217,CCC(CC)C(=O)NCC1CN(C(=O)C(n2ccc(C)n2)C)CC1O 98218,C=CC(C)CC(=O)NCC(CC1CCCC1)C(=O)NCCOC(=O)NC 98219,c1(C(C(=O)N(CCNC(COCCC)=O)CC2CC2)O)cccc(C)c1 98220,C1(NC(C2(C#N)CCCC2)=O)CCN(C(C2CCS(=O)(=O)N2)=O)CC1CO 98221,c1(NCCN(C)C(c2cccc(F)c2F)=O)nc(Cl)nc2nc(Cl)n(C)c12 98222,N1(Cc2c(Br)ccc(C)c2)CC2CC(NC(=O)Cc3c(C)noc3C)CC2C1 98223,C1(C(=O)NCc2nnn(CC)n2)C(C2CC2)CCN1C(C1CN2CCC1C2)=O 98224,C1(C(=O)NCC(CC)N(C(=O)CCC2CCC(C)O2)C)CC(F)(CF)C1 98225,C1(NC(c2c(C(C)(C)OC)cccc2)=O)CC(O)CN(C(=O)C(C)=CC2CC2)C1 98226,Cc1c(Br)ccc(F)c1NC(=O)COC(C12CCC(N=[N+]=[N-])C1C2)=O 98227,c1(CC(N2CCN(C(=O)C(O)C(F)(F)F)CC(O)C2)=O)cncc2ccccc12 98228,CCC(CC(=O)N1CC(NC(=O)CCc2nncn2C)C(C(F)(F)F)C1)C(C)C 98229,C1(NC(CC2OCCN(C(C(C)OCC(C)C)=O)C2)=O)CC2CC1CC21CC1 98230,C12(NC(=O)COC3CCC3)CCCN(C(=O)CCCC(F)(F)F)CC1C2 98231,Cc1cc(S(=O)(=O)NCC2CC(c3ccc(F)cc3)C2)cnc1Cl 98232,C(C(C)(C)CC(=O)N1CCC(F)(C(N)=O)C1)NC(c1c(C)cnnc1)=O 98233,c1(CC)nc(=N)[nH]c(=NC2CC(C)(C)OC3(CCC3)C2)[nH]1 98234,C1(C(N(CCOC)CC)=O)(CNC(=O)C(C)n2cccc2)CCCC1 98235,c1(C(C)C)ncc(C(=O)NCCCN(C)C2CC2)cn1.C1C(=O)N1 98236,C1(CC)(CC)CC(C(=O)NCC2(F)CC(NC(=O)CSC3CC3)C2)C1 98237,C(=O)(C(C)(C)CS(N)(=O)=O)N(CCN(C)C(c1ccc(F)cc1C(F)(F)F)=O)C 98238,Cc1cc(C)n(CC(N2CCC(C)(CNC(=O)C(C)C(C)(C)C)C2)=O)c(=O)n1 98239,N1(CC(CCCC)CC)CCc2sccc2C1CC 98240,c12ccc(c(F)c1)C(=O)NCC1(CC1)CN2.c1(CCC)nnnn1CCC(C)C 98241,C1(CNC(c2csnn2)=O)CCN1C(=O)Cc1nc[nH]n1 98242,C1(C)(NC(C2N(C(CS(CC)(=O)=O)=O)CCOCC2)=O)CCCCC1(C)C 98243,c1(OC)cc(C(N2CCCCC2CNC(C2CCS(=O)(=O)N2C)=O)=O)cc(C)n1 98244,n1(CC)cc(Cl)c(C(=O)NC(C)(C)CNC(=O)CSC2CCS(=O)(=O)C2)n1 98245,C1(C)(CC(=O)NCCOC2CCN(C(C3(C(C)C)CC3)=O)C2)CCS(=O)(=O)N1 98246,N=c1[nH]c2c(s1)CCCC2C(=O)OCCCCC(=O)Nc1c[nH]c2ccccc12 98247,CCCC(C(=O)N1CC2CC1(CNC(=O)C(C1CCOCC1)F)C2)S(N)(=O)=O 98248,C1(CCNC(C(C)NC(=O)Cn2cnnn2)=O)CCCCN1C(=O)CNC=O 98249,C(C(C)CN=c1nc(N2CCCC3(CCSCC3)C2)c2sccc2[nH]1)OC 98250,CCCCC(C(=O)NCC(C)(C)NC(c1cnnc(O)c1)=O)C(C)C 98251,C(=O)(C1CCCc2c[nH]nc21)N(CC(C)NC(C1Cc2cc(Cl)ccc2O1)=O)C 98252,c1(C(C)C)cc(C(=O)NC(C2CCOC2)CNC(C2CC(=C3CC3)C2)=O)nn1C 98253,c1(C(=O)NC2CC(CNC(c3cc[nH]n3)=O)C23CCC3)c[nH]c2cnccc12 98254,N1(C(C(C(=O)OCC)F)=O)CC2CCC1C1CN(C(=O)C(C)(F)C(C)(C)F)CC21 98255,C(C(C(C)C(C)C)NC(=O)CSC)NC(CCc1cncc(OC)c1)=O 98256,C1(c2n(CC=C)nnn2)(NCc2cc(C3CCCC3)on2)CC2CC1CC21CC1 98257,n1(CCCCC2C(C)(O)CCC2)cnc2c(N3CC(CF)C3)ncnc12 98258,c1(N2CC(C)(CCO)OCC2)ccncc1S(=O)(=O)NCC(C)(C)c1cccs1 98259,c1(C(NOCC(=O)N(C(CC#C)C)C)=O)ccc(O)nn1 98260,N1(CC)CC2COCC(CO)(C1)C2O.N1(C(C(=O)N)=O)CCN(c2cccnn2)CC1 98261,CC(O)(Cn1ccccc1=O)C(=O)NCC1CC(NC(C2CC=CCO2)=O)C1 98262,Cc1ccc2c(=NCC3CCOCC3)[nH]c(=NCCC(C)(C)CO)[nH]c2c1.CCC 98263,c1(NCC(COC)(C)CO)[nH]c(=NCCc2ncccc2C)nc2scnc12 98264,N1(C(C(=O)NC(C)C)=O)CCC(C)(CCNC(C2C=CCCC2)=O)CC1 98265,O=C1CNc2cc(C(N3CC4CC3CN4C(=O)CC3C=CCC3)=O)cnc2N1 98266,N1(C(C2C(COC)C2)=O)CCN(C(=O)C(O)CCc2ccccc2)C(C)C1 98267,N1(C(C(CC)NC)=O)CC2(C1)CN(C(=O)C(CC(C)C)NC=O)CC2CCl.C(C)(C)N 98268,N1(C(CCC2(CCC#C)N=N2)=O)CCC2C1CCN2C(C1C2C=CSC12)=O 98269,C1(CNC(CSCCN(C)C)=O)(NC(=O)CSC2CCCCO2)CCCCC1 98270,CC(C)C(C)C(=O)NCc1ccc(OC(F)F)cc1.C12CCN1OC2=O 98271,C(C(=O)NCC(C)NC(=O)C(c1cscn1)N(C)C)(OCC)OCC 98272,c1(C(=O)NC2CN(C(=O)C(F)CC3CCCCC3)CC2O)ncc(Cl)cc1O 98273,N1(C(C2(CC#C)CCN(C(=O)CCN(C)CC)C2)=O)CCN2CC(O)CC2C1 98274,Cc1cc(NC(=O)C(=O)NCCC(C)O)sc1NC(c1ccccc1)C 98275,C1(C(N(C2(CC(=O)NCCC3(C)CCOC3)CC2)C)=O)CCCC(=O)N1 98276,C1(CC)CCCN(CC(=O)NC2CN(C(=O)CC3(C#N)CC3)CC2O)C1 98277,n1(CC)ncc(C(=O)NC2CC(NC(=O)CCC3CCCCN3C)C(O)C2)c1C 98278,C1(CNC(c2cc(SC)c(F)cc2)=O)CN(C(C2CNC(=O)O2)=O)CC12CCC2 98279,N1(C(c2cn(CCOC)nc2)=O)CCC(CCNC(=O)C(C)SC(C)C)CC1 98280,C(CCN=c1nc(N2CCC(C)C3(CCCCC3)C2)cc(C)[nH]1)OCC 98281,C#CC1(C(=O)NCC(O)CN(C)C)CCN(C(C23CC(CO)(C2)C3)=O)CC1 98282,c1(C(N2CC(C(=O)C(F)F)OCC2)=O)cc(F)ccc1SCO.c1(C2(O)CC2)ccno1 98283,c1(OCC)ccc(-n2nc(-c3cccc(Cl)c3)nc2Cn2ccc(C)n2)cc1 98284,CC1CN(C(C2CN(C(c3sccc3C#N)=O)CCN2C)=O)CC(=O)N1C 98285,C1(NC(C2(C=C)CC2)=O)CCN(C(=O)CCc2c(C)nc(S)nc2C)CC1(C)C 98286,CCC(CC(=O)NC(CN(C)C(c1ccn(CC)c(=O)c1)=O)CC)C(F)F 98287,c1(C(C(=O)NCC2N(C(CSCC#C)=O)CC=C2)(C)C)ccc(COC)cc1 98288,c1(C(=O)NC(CN(C(c2cnc(O)o2)=O)CC)C)cc2nc(Cl)ccc2s1 98289,c1(C(=O)NCC(C)=CC(=O)NCCC(C)CC)nnn(C)c1N 98290,C1(C(N2CC(CNC(C(C)=C(CC)C)=O)C2)=O)C2Cc3cc(Cl)ccc3C12 98291,N1(C(=O)COCC(F)F)CCOC(CNC(C2(c3cccs3)CCCC2)=O)C1 98292,C1(C(=O)Nc2ccc(OCC(=O)OC)cc2)CCCCC1(OC)OC 98293,N1(C(Cn2c(C)nc(C)n2)=O)CCC(C(=O)NCCc2nncn2C)CC1(C)C 98294,N1(C(C2OCCC(C)C2)=O)CC2CN(C(c3cc4cnccc4o3)=O)CC2(C)C1 98295,C1(NC(CC=C)=O)CCN(C(c2occc2C)=O)C1C(C)(C)C 98296,C1(C(=O)NCCCC(C)NC(c2cc(C)sn2)=O)CCC(=O)N(CC(F)(F)F)C1 98297,c1(NC(=O)CC2CSC2)cccc(CNC(C2CCC(C(=O)O)CC2)=O)c1 98298,CC(CC(=O)N1OCC(F)(F)C(=O)NCC(C)C1)C(C)(C)C 98299,CC(CC(=O)N1CC(NC(c2cccc(Cl)c2)=O)C1)C(=O)c1ccccc1 98300,c1(NC(C(CCC)N(C)Cc2cn3ccsc3n2)=O)cnc(C)c(C#N)c1 98301,CCCCCCCCCCCCCCCCCN1CCC1(C(=O)OC)CC 98302,c1(C(N2CCC(C(=O)NCCC(C)(C)OC)C2)=O)c(C)nsc1N 98303,c1(C(N(CCNC(C(CC)N(C)C)=O)CCOC)=O)nc(C)ncc1Br 98304,C1(NC(c2n[nH]c(C)c2O)=O)CN(C(=O)C2=C(Cl)CCOC2)C2(CCOC2)C1 98305,C1(NC(CSCC#C)=O)CCCC12CCN(C(c1cc(Cl)cc(F)c1N)=O)CC2 98306,c1(Nc2ccc(-c3c(OC)nccc3)cn2)ccn2nccc2n1 98307,N1(C(C(C2(O)CCC2)NC(=O)CCN2CCOCC2)=O)CC(F)(C2CC2)C1 98308,N1(C(CCCNC(C)=O)=O)CCOCC1Cc1cn(NC(=O)CS(N)(=O)=O)nn1 98309,C1(C(=O)NCCN(C(c2ccc(C)c(C)n2)=O)CC)CC2(CCOC2)C1 98310,N1(C(C(c2scc(C)n2)C)=O)CCC2(CCC(CNC(C34CC3C4)=O)OC2)CC1 98311,c1(C(=O)NCC(CNC(C(CC)=CCCC)=O)O)cnc(C(F)(F)F)nc1 98312,C(=O)(N=c1nc(C2(CC(=O)N(C)C)CCC2)[nH]s1)c1c(C)n[nH]c1 98313,Cc1cc(=O)n(CCC(=O)NCCN(C(c2ccccc2)=O)C2CC2)cn1 98314,c1(OC)c(NC(C2CCN(Cc3c(F)ccc(C)c3Br)CC2)=O)ccc(F)c1F 98315,N1(C(c2c(CC)n(C)nn2)=O)CC2(C=C(C(=O)NCC(C)=CCO)CO2)C1 98316,N1C(CC(=O)NCCC2(C(=O)NCc3cnns3)CCC2)CCOCC1=O 98317,C1(C)(C(=O)NC(COCCOCCOCC#C)=O)CN2CCC1CC2 98318,c1(N(c2n(C)nnc2)C(C2CNC2)=O)ccn2ncc(Br)c2n1 98319,C(=O)(C1=CCCCC1P(C)(C)=O)NC1(CNC(C(C)(C)c2ccccc2)=O)CC1 98320,c1(C(=O)NC2C(CNC(c3ccnc(C(F)F)c3)=O)C2)cncc2cnccc12 98321,N1(C(c2c(C)cco2)=O)CCC(C(=O)NCCc2ccncn2)C12CCC2 98322,C1(NC(=O)COC)CCCC(NC(C2CCCO2)=O)C1.c1nccc(O)n1 98323,N12CCC3CCCC13NCC(O)CC2=O.N1(C(=O)OC(C)(C)C)CC(CO)C1 98324,N1(C(CCCCOC)=O)C2CCC1CC(NC(=O)C(C(C)(C)C)NC(C)=O)C2 98325,CCC(CC)CC(=O)N1CC=CC(C(=O)NCC=CC(=O)OCC)C1 98326,N1(C(c2n(C)nc(C(F)F)c2)=O)CCC(NC(C2CC2(C)C)=O)C12CCC2 98327,N1(C(CCCC(=C)C)=O)CCCC(C2CCN(C(C3CN4CCN3CC4)=O)C2)C1 98328,c1(C(=O)NCCCn2cc(C3CCCC3O)nn2)cnn2cccc(Cl)c12 98329,c1(N(C(=O)OCC)C)ccc(NC(C2(c3ccccc3Cl)CCOCC2)=O)cc1 98330,c1(C(=O)OC)c(C)sc(Br)c1O.n12cc(nn1)NCC2 98331,CC1CCCN(C(=O)CCCn2ccnn2)C1CNC(c1cnc(Cl)n1C)=O 98332,C(C(C)CC(F)(F)F)NC(C(c1ccnn1C)NC(C(C)SCCOC)=O)=O 98333,c1(CCC(=O)NC2(C)CC(NC(C(C)=CC)=O)C2)ccc(F)cc1Cl 98334,Cc1cc(Br)cc(CN2CCC(O)(C(=O)NC3CCC(O)C3O)CC2)n1 98335,c1(CC(N2C3C(NC(COCCOC)=O)C(C3)C2)=O)ccc([N+](=O)[O-])cc1Cl 98336,c1(C(=O)OC)cccnc1C(=O)NC1C(CNC(C2(n3cccn3)CC2)=O)CC1 98337,O(N(C)C(=O)CNC(N1CC(CO)C(c2ccccc2)C1)=O)CC 98338,C1(NC(c2ncn(C(C)C)c2)=O)CCOCC1NC(=O)CC(=O)NC1CC1 98339,C1(C(C)NC(=O)C(C)n2cccn2)CCN(C(c2ccnnc2Cl)=O)CC1 98340,c1(C(C)C)ccc(F)cc1C(N1CCC(NC(=O)C(O)C2CC2)C(O)C1)=O 98341,C#Cc1cccc(CC(=O)NCC2(NC(c3cnncc3C)=O)CCCCC2)c1 98342,C1(C(=O)NC(C2CCN(C(C(CC)C)=O)C2)C)CCn2c(cnc2C)C1 98343,O=c1c2ccccc2[nH]cc1N1CCCCC12CCCC2 98344,c1(OC)ccc2c(c1)OCC(CNC(c1sc3cccnc3c1Br)=O)O2 98345,N1(C(c2cnc(C(C)(C)C)s2)C(=O)NC)CCN(C(=O)OC(C)(C)C)CC1C 98346,c1(CC)cc(N)ccc1C(N1CC2C(NC(=O)CCN3CCC(F)C3)C2C1)=O 98347,O=C1NC(=O)C2(CCN(C(=O)NC(c3ccc4ccccc4c3)C(F)(F)F)C2)N1 98348,O=C(C1=CCCC1)NC1CN(c2cc(-n3cncn3)ncn2)CC1F 98349,C(c1c(F)cccc1F)=CC(N1CC(OCCNC(C(C(C)OC)O)=O)C1)=O 98350,c1(CNC(C(CC)=CCCC)=O)ccc(CNC(=O)CCc2cnccn2)cc1 98351,Cc1cc(C(N2CCCC(CNC(=O)C(C)CF)C2)=O)cc(I)c1 98352,c1(OC)ccc2c(c1)CCN(c1nc(N(CC(C)C)C)c3ncccc3n1)C2 98353,N1(C(C(CC)Oc2ccccc2)=O)CCC2CN(C(c3ccn(C)c3)=O)C2C1 98354,C1(C(N(CCCCCNC(C(COC)OC)=O)C)=O)OCCOC1(C)C 98355,c1(C(=O)NC2CC3(C(NC(c4c(N)cc(Cl)nc4)=O)C3)C2)n[nH]c2c1CCSC2 98356,C1(C(=O)Nc2cccc(CNC(CCCC#C)=O)c2)CCn2c(C)cnc2C1 98357,c1(C(N2CC(N(C)C(C3CCC(C(F)F)CC3)=O)C2)=O)cc(C#N)ccc1F 98358,C(CCCCCC(=O)N1CCC(O)C(F)(F)C1)NC(=O)CC1CC2CCC1O2 98359,CCCCC(C)CCC(=O)NCC1(NC(c2ccc(O)cn2)=O)CCOCC1 98360,n1(C(C)C(=O)NCCC2(O)CCN(C(=O)C(F)F)C2)c(=O)oc2ccccc12 98361,C(N=C(NC1CC1)NC1CC(C)(C)CCc2ccccc21)c1c(C)ncs1 98362,C1(NC(COCCOCCOC)=O)CCCC2CN(C(C3CC4CC4C3)=O)CC12 98363,n1(CC(N2CCC(CN(C(c3c(OC)scc3)=O)C)C2)=O)nc(C)c(Cl)c1C 98364,C(=O)(CCC(C)(C)F)NCC1C(C(=O)NC(CC=C)C2CC2)CCO1 98365,CC1(C)CN(C(=O)CCOc2ccccc2F)CC1NC(=O)C=CC1CCOC1 98366,CC(C)(C)CC(C)(C)C(=O)NCC(CO)NC(=O)CC1CCCCCC1(F)F 98367,Cc1ccc(NC(=O)C(C)OC(c2sccc2S(N)(=O)=O)=O)c([N+](=O)[O-])c1 98368,Cc1cccc(COC(C)C(=O)NC2COCC2NC(=O)C#CC2CC2)c1 98369,CCC(C)CCC(=O)NC1CCCCC1NC(=O)Cn1ccc(C(=O)OC)n1 98370,C1(C(N(C(CSC)C)C)=O)CCCCC(C)(C)C1 98371,c1(C(=O)NC(CC)CNC(=O)C(C(C)C)OC)c(Cl)nc2ccccn12 98372,c1(C(N2C(CCCNC(CCSCCC)=O)CCC2)=O)coc2c1CS(=O)(=O)C2 98373,C1(C(N2C3C(NC(COCCCCOC)=O)C(C3)C2)=O)CCCC2(CCOC2)O1 98374,N(C(=NCCN1CCOCC1(C)C)NCCSc1cccc(C)c1)CC(CC)OC 98375,C(=O)(CC(C1CC1)NC(=O)CC1CCC(O)C1)NCC=C 98376,N1(C(c2cc(SC)oc2C)=O)CCC2(CCC2NC(c2occc2C)=O)CC1 98377,C=CCC(C)C(=O)NC(C)Cn1cc(CNC(c2ccnn2C(C)(C)C)=O)nn1 98378,Cc1nn(CCO)c(C)c1C(=O)NCCCNC(=O)Cc1ccccc1Cl 98379,C1(COC)(NC(c2ccc(OC)cn2)=O)CCCN(C(c2cc(C)oc2C)=O)C1 98380,c1(OCC(=O)N(CC(CNC(C(CCC)N(C)C)=O)O)C)c(C)cccc1C 98381,C(=O)(C(O)CC(C)C)NC(c1nc(C(=O)NCc2nc(C)cc(C)n2)co1)C 98382,C12(NC(c3c(COC)ncs3)=O)CCN(C(=O)CCOC3CC3)CCC1C2 98383,c1(NC(=O)NC2C(C(C)(C)C)OCCC2)nccc(Br)c1F 98384,C1(NC(C2CC(C)(CC)C2)=O)CN(C(C2C3CCC(=O)C23)=O)CCC12CCC2 98385,C=CCCC(C(=O)NCCCC(N)=O)NC(=O)CC1C=CCC1 98386,N1(C(C2N(CC)CC2)=O)CC2CC(C1)N(C(=O)CCC1CCC(C)O1)C2 98387,C(C)(C)(C(=O)NC(CNC(=O)COc1cnn(C)c1)C(C)C)NC(=O)OC 98388,N1(C(=O)COCC2CCCCO2)CCN(C(=O)C(F)(F)C2CC2)CC2(CC2)C1 98389,C(C1=CCN(C(=O)CC(F)(F)F)CC1)NC(C(C)Sc1nncn1C)=O 98390,C(=O)(CCCC(F)(F)C(F)(F)F)NCC1(NC(c2nc(C#C)sc2)=O)CC1 98391,C1(NC(C(=O)N(C)CC2CCCCO2)=O)CCCOC1c1ccccc1 98392,N1(CCC)CCCCC1CN=C(NC(CC)CC)NC1CCS(=O)(=O)C1 98393,C1(C(N2C(CC(C)=O)CCCC2)=O)CC2CCN(C3CC(=O)NC(C)C3)CC12 98394,c1(C(=O)NC2CC3CN(C(c4c(CC)nccc4)=O)C2C3)cc2cccnn2c1 98395,C1(SC)CN(C(C2(O)CC(F)(F)C2)=O)CC1NS(=O)(=O)CC1(C)CC1(F)F 98396,C1(NCc2cccc(-c3nnc(C)o3)c2)CCC(C)(C)CC1CN=[N+]=[N-] 98397,Cc1oc(C)c(C(N2CCC(NC(=O)CN3CC(C)(C)C3)CC2)=O)c1C 98398,C(c1cccc2cccnc12)=CC(=O)NC1CN(C(C2CC(C)(O)C2)=O)CC1O 98399,Cc1ccc2oc(C(=O)N(C(C)CN(C)C(c3cn(C)c(O)n3)=O)C)cc2n1 98400,c1(C(N(c2cc(C(C)(C)C)ccn2)C(C)C2CC2)=O)cc(C2CC2)ncc1Br 98401,c1(NC(=O)OC)cccc(C(=O)NCC(C)CN(C(=O)COC(C)CC)C)c1 98402,CCCC(C)(O)C(=O)NC1CC(Nc2ccc(NS(C)(=O)=O)cc2)C1(C)C 98403,N1(C(c2cnc(C(C)C)o2)=O)CCOCC1CC(=O)NCC1(C)CCCC1O 98404,N1(C(C(CC(F)F)N(C)C(c2cc(=N)[nH][nH]2)=O)=O)CCC2(C1)CN(C)C2 98405,CC(F)(F)CCCC(=O)N1CCCCC(NC(=O)C=Cc2cncc(F)c2)C1 98406,C1(C(=O)OC)CCC(n2nnnc2C(CC)(c2nccs2)NC(C)COC(F)F)C1 98407,c1(C(N2CC(NC(c3c(CC)ccs3)=O)C(F)C2)=O)ccc2ccnn2c1 98408,N1(C(CC(CC(C)(C)C)O)=O)CCCC(C2CN(C(=O)CCn3cncn3)C2)C1 98409,c1(C(N(C2CCN(CC)C2)C)=O)cnc(CNC(=O)C(n2ccnc2C)C)nc1 98410,CC(C)C(CCN(C(=O)Cc1cnoc1)C)NC(c1cnn(C2CCCC2)c1)=O 98411,c1(OC)cc(OC)cc(C(O)C(=O)NCC(C)CCSC)c1 98412,c1(NC(C2CC23CC(NC(C2CCC2)=O)C3)=O)ccccc1CCO 98413,N1(CC)CC(C(N2CCOCC2CN(C)C(C2(C(=O)NC)CCC2)=O)=O)NC1=O 98414,CN1CCN(C(C2(C)CC2(C)C)=O)CC1C(=O)NCc1ccc(F)cc1 98415,N1(C(C2C(C=C)OCC2)=O)CCCN(C(c2nc(C)n(C)c2C)=O)C(C)C1 98416,c1(C(N2CC(N(C(=O)C3=COCCO3)C)C(C)(C)C2)=O)ccnc2ccncc12 98417,c1(C(N2CC(NC(=O)C=CCOCC(F)(F)F)C3C2C3)=O)ccc(C(F)F)cn1 98418,CS(=O)(=O)c1cccc(S(=O)(=O)N2CCC3CN(C(=O)C)CC23)c1.C1CC1 98419,C1(OC)CCn2cc(C(=O)N(C)CCN(C(=O)C(C)C#N)C)nc2C1 98420,N1(CC)C(C)CN(C(=NCc2ccc(C#N)s2)NC(C)C2CC2)CC1C 98421,O=C(C1CCc2nccn21)NCCC1CCCCN1C(c1cnc(C2CC2)[nH]1)=O 98422,CC(C)CC(O)C(=O)N(C(CNC(=O)CCC(=O)c1ccc(Cl)cc1)C1CC1)C 98423,N1(Cc2cc(C)cc(F)c2)CCCC(C)C1CNC1CCC(NC)CC1 98424,N1(C(CS(CC)=O)=O)CCC2(CCCCN(C(C3(c4ccncc4)CC3)=O)C2)C1 98425,C(=O)(C(C)CS(C)=O)N1C(CNC(c2c(NC(C)=O)c[nH]c2C)=O)CC(F)C1 98426,c1(OC)ccc(CCC(=O)NCC(C)N(C)C(c2ccc[nH]2)=O)cn1 98427,C(CC(=O)N(C(C)CNC(=O)C=C(C)C(C)C)C)N(CCC)C 98428,Cc1nc(C(=O)NCC2(CNC(C3CC34CCCC4)=O)CCC2)cn1C 98429,C1(CC)(CC)CC(NC(=O)Cn2nccc2C)CN1C(=O)CSC1CC1 98430,C(=O)(C(O)CC(C)(C)C)NCCCCNC(C(c1c(C)n[nH]c1C)C)=O 98431,Cn1ncc2c(C(N3CCC3CNC(c3ccc4c(n3)CCO4)=O)=O)cccc12 98432,CC12CC(NC(c3csc(O)n3)=O)(C1)C1(CN(C(=O)CC3=NNC(=O)C3)C1)O2 98433,Cc1cc(Br)cc(C(N2CC(N(C(=O)C#CC(C)(C)C)C)C(F)C2)=O)c1C 98434,C(C)(CNC(=O)C(=O)NCC(C)OC(F)F)(CO)OC 98435,C1(CC)CCCC(N(CC(F)F)CC2CC2)C1 98436,c1(C(=O)NC2CCC(NC(C(CC=C)CC)=O)CC2)ccc(S(=O)(=O)NC)nc1 98437,C(CC(C(=O)N1CC(C(C)C)C1)NC(C1CC=CCC1)=O)OCC 98438,c1(CNC(Cn2ncc(C)c2)=O)cccc(-n2cc(C3CCNC(=O)C3)nn2)c1 98439,c1(C(N2C(CNC(c3ncc[nH]c3=O)=O)CC(OC)C2)=O)ccn2cccc2c1 98440,N1(C(CCC)=O)CCC2(NC(=O)C=CC3CCCO3)CCCC12 98441,N1(C(c2ncc(C)nc2)=O)CCC(O)CC1C(N1CCOCC1C(C)C)=O 98442,N1(C(=O)OC(C)(C)C)CC2CCCC(C1)N2C(c1cc(C(F)F)ccn1)=O 98443,c1(NC(C(C)C)=O)cc(CNC(=O)NCCCN(C)C)nn1C 98444,c1(C(CNC(=O)CC2CC3CC3C2)NC(Cc2c(C)ocn2)=O)cccc(Cl)c1 98445,c1(OCc2onc(C)n2)cncc(C(=O)NCCSC2CCN(C)C2=O)c1 98446,c1(CCC(=O)NCC(CC)NC(c2cn(CC(=O)OC)nn2)=O)ncccc1C 98447,CC1CC(NC(c2ccn(CCNC(c3cc(C(N)=O)[nH]n3)=O)c2)=O)CCS1 98448,c1(CC)cc(N2CC3C(CNC(c4n[nH]cc4Cl)=O)C3C2)nc(CC)n1 98449,CCC(O)CC(=O)NCC(C)(F)CNC(c1c(C)nsc1C)=O 98450,N1(C(C=CC)=O)CC2CN(C(C3CCN(C4CC4)CC3)=O)CCC2(CO)C1 98451,N1(C(c2c[nH]c(=NC)s2)=O)CCC(NC(=O)CN2CCCNS2(=O)=O)C(F)C1 98452,Cc1ccn(CC(=O)NCC#CCNC(c2sc(C(C)(C)C)nc2C)=O)c(=O)c1 98453,C1(CNC(CSCCC)=O)CCCCN1C(c1csc(C2CCCCC2)n1)=O 98454,CCCCS(=O)(=O)NC(C)C(=O)NC1(CNC(c2nnn(C(C)C)c2C)=O)CC1 98455,N1(C(C2C(=C)C2)=O)CCN(C(=O)CC(C)(C)c2ccccc2)C2(CCC2)C1 98456,C1(C(N2C(C(C)CNC(c3ccc(F)cc3)=O)CCCC2)=O)CC(C)(C)CN1C 98457,C1(C(=O)NC(C2CN(C(=O)CCCC(N)=O)C2)C)CCC2(CCOC2)O1 98458,N1(C(c2cnc(CC)s2)=O)CC(C)CCC1CNC(=O)CNS(=O)(=O)NC 98459,C1(CNC(=O)C(F)Cc2ccccc2)CN(C(C2(F)CC2)=O)CCCO1 98460,C(CN=c1[nH]c(C)cc(=NCC(CO)c2ccccn2)[nH]1)c1cncc(C)n1 98461,N1(C(c2c(SC)snn2)=O)CCCCC1CCCNC(C1CCS1(=O)=O)=O 98462,c1(C(=O)NCC2(C)CCCN2C(c2cccc[n+]2[O-])=O)ccc2scnc2c1 98463,C1(C(=O)OC)COC(CCC(=O)NC(C)CCNC(=O)C(N)=O)C1 98464,CCCCCCC(C)(CCC)C(=O)N1CC2CCC(C1)N2C(=O)Cc1ccco1 98465,C(=O)(C(CC(C)(C)C)OC)NCC(CNC(C1CCC(=C)CC1)=O)OC 98466,c1(C(N2CCC(O)(C(N3CCOC(CO)C3)=O)C2)=O)c(F)cncc1F 98467,C#CCC(CC#C)C(=O)NCC1CCN(C(C2(C)CCN(C)CC2)=O)C1 98468,CC1CN(CC(=O)CCc2c(F)cccc2F)CC2(CCCOC2)O1 98469,CCC(O)CC(=O)N1CC(CC(C)NC(c2cc(-c3cccs3)on2)=O)C1 98470,C1(C(=O)NCCN(C(=O)CCCc2ccncc2)C(C)C)CCC2(CCC2)OC1 98471,C1(C(=O)NCC(C(C)C)NC(CC(C(F)(F)F)OC)=O)COc2ccccc2O1 98472,N1(C(c2ccc(N(C)C)cc2)=O)CCN(C(=O)CNC(=O)NC2CC2)C2CC12 98473,CN1CCOc2ncc(C(=O)NC3CCN(C(C45CCC4C5)=O)C3C3CC3)cc21 98474,CC1CC(C(=O)NCC(C)(O)C2CC2)N(C(C2CC(CF)C2)=O)C1 98475,C(CC(F)F)(C(=O)NCC1(C)CCCO1)N(C)C(C1CC(C2CC2)=NO1)=O 98476,N1(C(C(C)NC(N)=O)=O)CCC(NC(c2scnc2Br)=O)C1(C)C 98477,C1(c2cn(CC3COCCO3)nn2)(NC(=O)CC2CC2(Cl)Cl)CCCOC1 98478,C(=O)(CCCC(C)(C)NC(=O)C=Cc1ccnn1C)N1CCC(CC=C)C1 98479,C1(CNC(C(COC)(C)O)=O)CCCCN(C(=O)CC(C)C2CCCCC2)C1 98480,N1(C(C=C2CCC(C)C2)=O)CCOC(C(C)NC(C2CCCN(C(N)=O)C2)=O)C1 98481,C(=O)(C(CNC(c1csc(F)c1)=O)CC1CC1)NCC1C(CC)C1 98482,C1(CNC(C(CC)NC(C)=O)=O)CN(C(=O)C(C)(C)COCC)CC1CC(C)C 98483,c1(CN2C(CNC(c3cc(CC)[nH]c3)=O)CC2)cc(Br)ccc1OC(F)(F)F 98484,C1(N(C(=O)C=Cc2ccoc2)C(c2c(C)snc2)=O)CCN(c2nncs2)CC1 98485,N1(C(C(C=C)(C)C)=O)C(CNC(=O)CCOC)CC2COCC12 98486,N1(C(C2(C#N)CC2)=O)C2CC1CN(C(C1CC1C1CCCO1)=O)C2 98487,O=C(CCCCCCNC(C1CCOC(=O)CC1)=O)NC1CCC=CCC1 98488,C(CCN=c1[nH]c(N2CCOC(C(C)(C)C)C2)nc2c1SCC2)OCCOC 98489,CCCC(C)(CC)C(=O)NC(CNC(=O)C(c1ncccc1C)(F)F)CO 98490,c1(-c2c(OCC(=O)OC)ccc(Br)c2)ccc2c(c1)C(C)C(C)O2 98491,C1(C(N(C2CCN(C(c3cc(C(C)(C)C)on3)=O)C2)C)=O)CCCS(=O)(=O)N1 98492,C1(C(=O)NC(CC)C(=O)N(C)C)CC(NC(C2(C)CC(C)=NO2)=O)C(O)C1 98493,c1(C(=O)NC(CC(C)NC(c2nc(C)[nH]n2)=O)C)cn2cc(Cl)cnc2n1 98494,c1(-n2cc(C(N(CCNC(C(CC)(C)O)=O)C3CC3)=O)nn2)cc(C)cc(F)c1 98495,Cc1cc(C(F)F)n(CC(=O)NCC(C2CC2)NC(=O)C(C)Cc2ccco2)n1 98496,N1(C(C(=O)NCC)=O)CCOC2(CCN(C(c3cc(C)nc4c3cnn4C)=O)C2)C1 98497,CC1CN(c2nnc(-c3cc(CC(N4CCCCC4)=O)[nH]n3)n2C)CC(C2CC2)O1 98498,c1(CC(=O)NCC23N(C(CCNS(C)(=O)=O)=O)CC(C2)C3)c[nH]c2cccnc12 98499,CCCCCC(C)CC(=O)NCCN(C(=O)C(F)CC1CCCC1)C 98500,N1(C(c2cccc(C(C)C)n2)=O)CC(CNC(=O)COC2CC2)N2CCC1C2 98501,C(CC(F)F)(C(=O)NCc1cc(O)cc(F)c1)N(C)C(c1ccnc(CO)c1)=O 98502,C12CCC(CC1)N2.C(=O)(C(C(C)O)N(C)C)N(CCC(=O)N1CCCC1)C(C)C 98503,n1(CC(=O)NC2C3N(C(c4c(C)cn(C)c4)=O)C(CC3)C2)cc2ccccc2n1 98504,N1(C(CC(CC(C)C)C)=O)CCC2CN(C(C3CC34CC4)=O)C(C)C12 98505,C1(CNC(C2N(C(N)=O)CC(O)C2)=O)CC2(CC2)CN1C(=O)CCC1CC1 98506,C1(CCC)CN(C(=O)Cn2ccnc2C)CCN1C(c1cccc(Cl)c1)=O 98507,c1(C(=O)NCC(c2ccc(OC)cc2)NC(CC)=O)ccc2ncccc2n1 98508,N1(C(c2cc(F)c(C(F)(F)F)c(F)c2)=O)CCN(C2CCNC2=O)CC(O)C1 98509,c1(C(=O)NC(C2(O)CN(C(Cn3ncc(C)c3)=O)C2)C)nc(C2CC2)ncc1Cl 98510,N1(C(C=C(C)Cl)=O)CCN(CC(C)(C)C)CC1.C1C(C)NC(=O)O1 98511,Cc1cc(C(N2CCCC2CCCNC(C2CC23CCSCC3)=O)=O)nc(C)c1 98512,CC(C)CC(C(=O)NC1C=CCN(C(=O)C=CBr)C1)C(N)=O 98513,c1(C(=O)NCCN(C)C(c2ccc(C(F)C(F)(F)F)cc2)=O)ccnc(Cl)c1N 98514,c1(C(=O)NCC#CC(=O)NCC2CN(C(C)=O)C2)c[nH]c(=S)cn1 98515,c1(C(=O)NC2CCN(C(C3N(C)C(=O)OC3)=O)C2)cncc2c1CCCC2 98516,C(=O)(NNC(=O)c1ccc(I)cc1)N1C(CC(C)C#N)CC1 98517,Cc1c(Cl)ccnc1C(N1CCC(C)(NC(C23CCC(CC2)OC3)=O)C1)=O 98518,C(=O)(CC(C)CC(C)(C)C)N1CCC(CNC(c2ccc(C=C)cc2)=O)(CO)C1 98519,c1(COC)csc(C(=O)N(CCNC(C2CCCC2O)=O)C2CC2)c1 98520,N1(C(C#C)=O)C2CCC1CN(C(c1ccc(Cl)nc1F)=O)C2 98521,C12(C(N3CC(O)CC(NC(c4ccncn4)=O)C3)=O)CCCC(CCC1)C2O 98522,C(C)(CCC(F)(F)F)(C(F)(F)F)NC(CNc1ccc(OC)cc1)=O 98523,C(=O)(CCC(C)(C)F)N(CC(Cc1ccccc1)NC(C1CCSC1)=O)C 98524,CC1CCC(NC(c2c(C(F)F)cccc2F)=O)CN1C(c1cccc(N)n1)=O 98525,C1(NC(c2c(CNC(c3cnncc3O)=O)cc[nH]2)=O)CC12CCCCCC2 98526,c1(C(N2CCC(N(C(C(C)=C3CCCC3)=O)C)C2)=O)c(C)c[nH]c1CC(N)=O 98527,C1(C#N)(C(N2CC(NC(c3ccc(COC)s3)=O)C(SC)C2)=O)CC12CCCC2 98528,C(=O)(CCS(C)(=O)=O)NCC(C)(CO)NC(=O)CSCCCc1ccccc1 98529,N1(C(C=C(CC)CC)=O)CC(O)(C2(CNC(=O)CC3COCCN3CC)CC2)C1 98530,c1(CN(C)CC2CCCN(C(=O)CCc3ccccn3)C2)cccc(F)c1C#N 98531,c1(CNC(Cn2cc(CNC(C3(C)C(C)(C)C3)=O)nn2)=O)ccncc1F 98532,c1(C(=O)NCC(C)N(C(=O)C(c2ccc(C(F)(F)F)cc2)C)C)cc(Cl)cn1C 98533,C1(CNC(Cc2c(C)nc[nH]2)=O)CN(C(=O)CC2CCC(C)C(C)C2)CCCO1 98534,Cc1nc2c([nH]1)C(C(=O)N1CCC(N(C)C(C3CC3C)=O)C1)CCC2 98535,CC(C)CC(CNC(c1cnn[nH]1)=O)C(=O)N(C)CCc1ncon1 98536,N1(C(c2cc(SC)oc2)=O)CC(CNC(c2cc(C(F)(F)F)cs2)=O)C(C)C1 98537,c1(-c2cncc(C(=O)NCc3ccnc4[nH]ccc34)n2)cccc(F)c1[N+](=O)[O-] 98538,C1(C(N2CC(OCCNC(=O)C=Cc3cnccn3)C2)=O)CC2CCCCC2O1 98539,C1(C(N2CCCC(N(C(COCCCC#C)=O)CC)C2)=O)CCCCC12CC2 98540,c1(C(=O)NCCCCN(C(Cc2cc(C)sc2C)=O)C)cc(O)nc(O)n1 98541,c1(C(=O)OC)cc(C)nc(N(C(C)CNC(=O)Cc2cc(C)ns2)C)n1 98542,C1(NC(C=C(C)C(C)(C)C)=O)CCC(NC(=O)CC(O)c2ccccc2)CC1 98543,Cc1c(C(=O)NCC2(CNC(C3CC4C(C3)C4(C)C)=O)CCCC2)cccc1N 98544,Cc1cc(C(=O)NC2CC2NC(c2nccnc2C)=O)cc(C)c1Cl 98545,C1(NC(=O)CC2COCCO2)CCOC12CCN(c1ncc(O)cn1)CC2 98546,C(=O)(C1=CC(C)(C)C1)N1CCC(CC(C)NC(=O)CCC2CCCCO2)CC1 98547,c1(C(C)=O)c(C(=O)NCC2(F)CN(C(=O)CC(F)(F)F)C2)cccc1C 98548,CC1(C)Cc2c(cnn2-c2ccccc2)CN(C(c2cc(I)cs2)=O)C1 98549,C1(CC(C)NC(CCCNC(C)=O)=O)CCN(C(C2CCOCC2)=O)CC1 98550,O=C(C1=CC2C=CC(C1)C2)NCCC1CC(NC(c2cc3n(n2)CC(F)C3)=O)C1 98551,CCCCS(=O)(=O)CC(=O)N1CC2C(CN(C(=O)Cc3cn(C)cn3)C)C2C1 98552,n1(CCC(N2CC(NC(c3cnco3)=O)C(O)C2)=O)ncc2c1CCCC2 98553,N1(C(C=CC)=O)CCC(C(C)NC(C2(CCS(N)(=O)=O)CCC2)=O)CC1 98554,C1(NC(c2ccc(C)o2)=O)CC2CCC1CC2NC(=O)CC1C=CCCC1 98555,N1(C(C2C(NC(CN(C(C3C(C)C3)=O)CCO)=O)CCO2)=O)CCC(CCF)CC1 98556,C1(CC)CN(C(c2nc(O)cs2)=O)CCN1C(=O)Cc1ccnc(Br)c1 98557,C1(CNC(CCCOCC)=O)CCC(C)(C)CN1C(=O)CC1CC(OC)C1 98558,N1(C(CC2C(C)CCCC2)=O)CC2CN(C(=O)CCNC(=O)CO)CC(C1)O2 98559,N1(C(C2C(C=C)C2)=O)CC2CCC1C(NC(=O)COc1cccc(F)c1)C2 98560,C(=O)(C(CC)(CC)C(C)C)NC(CC(N1CCC(=CCC)C1)=O)C1CC1 98561,c1(C(=O)NC2(CC)CCN(C(=O)CCF)CC2)cccc2c1C(=O)NC2=O 98562,c1(N2CCC(CC)CC2)nc(=NCCC(F)(F)C(F)F)[nH]c2c1CCC2 98563,C=CC1CCC1C(=O)NCC1(NC(=O)Cn2ccc(C)n2)CCC1 98564,N1(C(c2scc(OC)c2)=O)CCC(C=CC(=O)NC(C)CC2CCC2)CC1 98565,C1(C(N2C(C(=O)NC(COC)C3(C)CC3)COCC2)=O)CC2(C1)CC2(F)F 98566,c1(C(=O)NCC(C)NC(c2c(CC)nc[nH]2)=O)ccc(F)c(Cl)c1N 98567,N1(C(C2(C)CC(F)(F)C2)=O)CCC(O)C(NC(C2CC23CCC3)=O)C1 98568,c1(C(=O)OC)ccnc2c1CCC2NCC(c1cc(F)cc(F)c1)C 98569,c1(CC(=O)N(CC(C)NC(=O)CCNC(N)=O)C)cccnc1Br 98570,c1(CNC(C(C2CC2C)N(C(C)C)CC)=O)cccc(C)c1F 98571,C12(CNC(C3N(CC)CC3)=O)COCCN1C(=O)CN(C(c1cnc(S)[nH]1)=O)C2 98572,c1(C(=O)NC(C(=O)NC2CC(C)OC2=O)Cc2ccoc2)occ2c1CCC2 98573,C12(NC(C(CC)CC)=O)CC3CCC(C1C2)N3C(=O)Cc1cn(C)nn1 98574,c1(N2C3CN(C(C4(CC)CCOCC4)=O)CC2CC3)ncnc2cc(C#N)ccc12 98575,N1(C(Cc2c(C)ncnc2C)=O)CCC2CN(C(=O)CC3NC(=O)NC3=O)C2C1 98576,c1(N2CCCC(C#N)CC2)nc2c(c(=NC3CCc4nn[nH]c4C3)[nH]1)COC2 98577,C(=O)(C(C)(C)C(C)O)NC1CC(N(C(c2nc(CCCCC)sc2)=O)C)C1 98578,c1(-n2cc(C3N(C(C4CCC4(F)F)=O)CC3)nn2)cc(C(F)F)on1 98579,C(C)(C)(CC(=O)N1CC(C)(CCC(N2CCOCC2C(C)C)=O)C1)OC 98580,N1(CC)CCOC(C(N2CCC(CNC(C3(COC)CC3)=O)C2)=O)C1 98581,Cc1cc(C(N2CC(NC(c3c(C4CC4)cccc3F)=O)C(F)C2)=O)c(C)n1C 98582,C1(C(C(=O)NC2COC2)N(C(C2(O)CCC2)C)C)CCOC(C)(C)C1 98583,C1(NC(C2C(C(=O)OC)C2)=O)CCN(C)C12CCCN(C(c1sccc1Cl)=O)C2 98584,c1(C(c2nnnn2C(C)(C)C)NCCCCC2C(C)C2)cc(Cl)n(C)n1 98585,c1(C(=O)NCC2C3CN(C(C(CC(C)C)OC)=O)C2C3)cnn2cccc(Cl)c12 98586,C1(CNC(c2ccn(CC)n2)=O)CCC2CN(C(=O)C(C)C3CCC3)CCC2C1 98587,C1(C(N(CCNC(=O)C(C)(C)c2ccno2)CC)=O)CC12CCc1ccccc12 98588,c1(C(=O)NC2C(NC(c3c(OCC)ccs3)=O)C2)cc(C(C)(C)C)nn1C 98589,n1(CC(C)C)nccc1C(=O)NC1CC1NC(c1csc(NC=O)n1)=O 98590,CC(CCN(C)C)C(=O)NCC1CC(F)CN1C(=O)Cc1cc(C(F)(F)F)co1 98591,C1(CCNC(c2n(CC)nnc2)=O)COCCN1C(c1cc(CCCO)on1)=O 98592,C#CCC(CC#C)C(=O)N(C1CCCN(C(c2snnc2C2CCC2)=O)C1)C 98593,C(=O)(CC(CC)NC(=O)C(O)C1CC1)NCC(=O)OCC=C 98594,C1(NC(Cc2ccc(C)o2)=O)CC2CC1N(C(=O)CC1COCC(C)(C)O1)C2 98595,c1(CC)nc(C(=O)NC(C2CCN(C(=O)CC3(N(C)C)CC3)C2)(C)C)cs1 98596,N1(C(COCCCOC)=O)CCCC(C2CCN(C(=O)COCCF)CC2)C1 98597,C=CCCCC(=O)NCC1CCCC(CNC(c2cnc(C3CC3)o2)=O)C1 98598,C1(C)(NC(CC2(C)CCC2)=O)CCCN(C(C2CC(C)(F)C2)=O)C1 98599,C=CC1(NC(=O)C(F)CC2CN(C(c3cccc(CC)c3)=O)C2)CCOCC1 98600,c1(CNN)cc(S(=O)(=O)NCCCNS(NC)(=O)=O)ccc1C#N.C1(C)CCCC1 98601,CC#CCC(C)NC(=O)CN(CCC)C(c1cccnc1)=O 98602,C1(CNC(c2nc(CCC)sc2)=O)CCC(C)N(C(c2cc(C(N)=O)c[nH]2)=O)C1 98603,C(=O)(C(CN=[N+]=[N-])NC(=O)CCc1cc(C)[nH]n1)NCC1(CC(=O)OC)CC1 98604,N1(Cc2ccc(C(=O)NC(N3CCC(C=C)C3)=O)cc2)CC(O)CCC1=O 98605,CN=c1ncc(-c2cnc(NCc3ncc(C)cc3F)nc2)c[nH]1 98606,CCC1=C(C(=O)N(C)CC2CCCN(C(c3cnncc3NC)=O)C2)CCCO1 98607,N1(CCC(=O)NC23CC(C2)N(C(c2cnoc2C2CCC2)=O)C3)C(=O)CCC1=O 98608,c1(C(=O)NCCN(C(=O)CC2C(=O)NN=C2C)CC)ccc(P(C)(C)=O)s1 98609,CC1CN(C(=O)C=Cc2nccs2)CCN(C(C2CC=CC2)=O)C1 98610,c1(C(=O)NC2CCCCN(C(C3N(CC)CCC3)=O)C2)c(C)c(C)nn(C)c1=O 98611,c1(CCNC(c2cnn(C)c2OC)c2n(CCOCC)nnn2)ccccc1C 98612,c1(C(C(=O)NC)N(C)CC2(C)CCCO2)cn(C)c(=O)n(C)c1=O 98613,C(=O)(C#CC1CCOC1)NCCN(C(c1cnc(C(C)C)s1)=O)CCOCCO 98614,N1(C(c2n(CC)cnn2)=O)CCCC(CO)(CNC(=O)C#CC2CC2)C1 98615,c1(CCC)cc(C(=O)NC2(CF)CN(C(c3cc(C(N)=O)co3)=O)C2)n[nH]1 98616,c1(NCC(=O)NC2CN(C(C3CC4(C3)CC4F)=O)C2)ccccc1Cl 98617,C1(C(C)(C)C)CCCC1C(=O)NCC1(NC(=O)Cc2cscn2)CCC1 98618,c1(C(C)O)ncc(C(=O)N(C2CN(C(=O)COCc3nccs3)C2)C)s1 98619,CC(N=c1nc(N2CCC(C#N)CC2)c2c([nH]1)CCC2)c1cc(Cl)ccc1Cl 98620,N1(C(=O)Cc2cc(F)ccc2Br)CC2(CCCN2C(=O)CN(CCO)CCO)C1 98621,c1(CNC(c2nnnn2C2CCCS(=O)(=O)C2)=O)cccc2c1OCCCO2 98622,N1(C(C2CN(C)C(=O)C2)=O)CC2(CCCC(CNC(=O)C=CCF)O2)C1 98623,c1(N(C)C)cc(-c2cn(CC(F)(F)CNC(c3cc(Br)nn3C)=O)nn2)ccn1 98624,c1(NC(C(N2C(CCC=C)CCC2)=O)=O)cccc(F)c1C 98625,C(=O)(CS(=O)(=O)C1CCCC1)NCC1CN(C(C(CSC)OC)=O)C2(C1)CCC2 98626,N1(C(C(C=C)OC)=O)CC2CC2(NC(C2C3CCC(=O)C23)=O)C1 98627,C#CCC(CC(=O)NCCOC1CCOC1)NC(C1CC1Cl)=O 98628,C1(C(N2CCCC(CC3CC3)C2)C(=O)NCC(=C)C)C2CCOCC12 98629,C(c1c(C)cccc1C)=CC(=O)NCC(CCC)NC(C1(n2cccn2)CC1)=O 98630,c1(C(=O)NC(CC=C)CNC(C2CCCCCN2C)=O)cc2cc(C)ccc2o1 98631,C1(C)(CCNC(C2N(CC)CCC2)=O)CCN(C(=O)CCc2cccn2C)C1 98632,c1(C(=O)NCC2(O)CN(C(C=C(CCC)C)=O)C2)sccc1OC 98633,C1(CC(F)F)C(=O)N1.C12(NC(c3cccc(C)c3)=O)CCC(CC1)CC2 98634,Cc1nc2cc(C(N3CCC(NC(=O)C=C(Cl)Cl)CC3)=O)cc(O)c2[nH]1 98635,C1(C(=O)NCCN(C(C2(COC)CCCCO2)=O)C)CC(=O)N(OC)C1 98636,c1(C(=O)NC(c2cc(C3CC3)on2)C)cn(C)nc1SCC(=O)N(C)C 98637,c1(NC(=O)NC(CCCC)CN2CCOCC2)ccc2c(Br)ccc(C)c2n1 98638,c1(CNCC2(F)CCCN(C(C3CC3F)=O)C2)sc(Br)c2c1OCCO2 98639,c1(C(N2C(CCC(=O)Nc3c(O)ncnc3O)CCC2)=O)ccn2nccc2c1 98640,C(C(C(=O)NC(C(=O)N(C)Cc1ccn(C)n1)C1CCC1)OC)OC 98641,c1(C(N(C)CCN2CCN(C(C3CC3CF)=O)CC2)=O)cnc2[nH]ccnc1-2 98642,c1(OC)ccc2[nH]cc(-c3ccc(Nc4cccc(Br)c4O)c(F)c3)c2c1 98643,c1(CC(=O)NCCCN(C(C(C)SCC)=O)CC)c(C)oc2ccccc12 98644,CC(CC(=O)N1CCOC(CC(=O)NCC(F)Cl)C1)C(C)(C)C 98645,CC1(C)CC(C(=O)NC(C)(CO)C2CC2)CN(C(C2(C3CCCC3)CC2)=O)C1 98646,Cn1nc(-c2nnc(C(F)F)o2)c(Br)c1CN1CCC(C(C)(O)C(F)(F)F)CC1 98647,Cc1nc(C2CCCC2)nc(O)c1CC(N1CCCC(C)(NC(=O)C2CC2)C1)=O 98648,C(=O)(C(C(C)(C)C)N1CCCC1=O)NC1CCN(C(c2ccc(OC)cn2)=O)C1 98649,N1(C(C2C(CC)CC2)=O)CC(CC(=O)NCCCOC2CC2)C(C)C1 98650,N1(C(CCCC=C)=O)CCC(CC)CC1C(=O)N(CC)CC1CCC1 98651,Cc1ccc(C(N2CC(NC(c3ncoc3C(C)C)=O)CC(C)C2)=O)c(N)c1C 98652,N1(C(CC2CC(SC)C2)=O)C(C)CN(C(=O)CC2CCC(=O)N(C)C2)CC1C 98653,C(=O)(C#CC1CCOCC1)NCC(CN(C(C(Cc1c(C)noc1C)C)=O)C)O 98654,C1(C(C)(C)NC(CN(CCSC)CC)=O)CCN(C(=O)C(C)NC(C)(C)C)C1 98655,C#Cc1cccc(C(c2nnnn2CC)NCCC2CC(C(C)C)C2)c1F 98656,C=CCCCCC(=O)NC(C)CCN(C(=O)C=C1CCCCC1(C)C)C 98657,C(=O)(C(C)(C)CC(C)(C)C)N1CC(O)(CCNC(C(C)C(C)(C)C)=O)C1 98658,c1(CN2CCC3(C(C(=O)Nc4ncc(C#N)cn4)C3)C2)ccc([N+](=O)[O-])c(Br)c1 98659,c1(C(=O)NCC2N(C(c3cc(CC)c(Cl)cc3)=O)CC2)ccc(N)c(C)c1C 98660,c1(C(N2CCCCC(NS(CC=C)(=O)=O)C2)=O)cccc(C(F)(F)F)c1O 98661,c1(C(=O)NC2CCN(C(C(CC)(C)O)=O)CC2CO)cccc2c1CCO2 98662,N1(C(c2ccc(OC)cc2)=O)CCN(C(=O)Nc2cc(Br)ccc2OC)CC1C 98663,c1(C(=O)NCC2(O)CCN(C(Cc3ncc(CC)[nH]3)=O)C2)cccc(N)c1C 98664,N1(C(=O)NCC2CCCC(C(C)C)C2)CCC2(CC1)OCC(C)O2 98665,c1(C(=O)NCC(CNC(=O)C(C)(O)C2CCC2)OC)cc(F)c(Cl)cc1Cl 98666,c1(C(N2CCN(C(CS(CC)(=O)=O)=O)CC2)=O)ccc2c(=O)n(C)c(C)cc2n1 98667,c1(C(CN(CC(C)Cc2ccc(Cl)cc2)C(C)=O)=O)cc(C(=O)O)cc(Br)c1 98668,C1(C(=O)NCC2CCN(C(CCC=CCC=C)=O)CC2)Cc2ccccc2C1 98669,N1(C(C=C(C)C(C)(C)C)=O)CC(O)CC1CNC(=O)C(O)C1CCC1 98670,c1(C(=O)NCC(C(=O)NC(CCC)C(=O)N(C)C)O)cc(C)c(C)nn1 98671,N1(C(c2cccc(CC)c2)=O)CC2(C1)OC1(C)CC2(NC(C2CCCO2)=O)C1 98672,Cc1cnn(C)c1CC(=O)NCC1C(C)CCN1C(=O)CC(C)(C)C 98673,C1(CC#C)(C(=O)NCc2cc(C)ns2)CCN(C(c2ccnn2C=C)=O)C1 98674,N1(C(CCOCCNC(c2cc(C)nnc2)=O)=O)Cc2ccc(O)cc2C1 98675,CCCC(C)CCCC(=O)N(CC(O)CNC(=O)Cc1csc(C(C)(C)C)n1)C 98676,C1(CC)CN(C(=O)C(O)CN(C)C)CC1C(=O)NCC1(CC2CC2)CCC1 98677,C(C)(C(=O)NCC1CN(C(=O)C(F)C(F)(F)F)CCCO1)(C(C)C)NC(C)=O 98678,C1(C(=O)NCCN(C(c2nc(OCC)oc2)=O)C2CC2)CCCC12CC2 98679,C1(C(=O)NCCCCNC(c2cn(C)c(=O)n2C)=O)CCn2cnnc2C1 98680,N#Cc1cnc(N2CC3CC(NC(c4c[nH]cc4Br)=O)CC3C2)c(Cl)c1 98681,N1(C(c2sc(C)c(Br)c2)=O)CCC2CN(C(c3c(F)cccc3Br)=O)CC12 98682,Cc1cn2ccnc(C(=O)NC3CCCC3CNC(c3cn(C)nn3)=O)c2n1 98683,CC(=O)CCCCC(=O)NCC(CNC(=O)CCc1cc(Cl)no1)CO 98684,CONC(=O)C(=O)NCCC1CCC(NC(C2C3CCCCC23)=O)C1 98685,C1(C(N(CC(C)NC(=O)Cn2cnc(C(N)=O)n2)C)=O)C(C)(C)C1(F)F 98686,c1(C(C)(C)C)cc(C(N2CCCC(NC(=O)CC3(O)CC3)CC2)=O)ccc1O 98687,C(=O)(CN1C(=O)Cc2ccccc21)NC1CCCC(OCCC)CC1 98688,C1(NC(c2c(OC)cccc2)=O)COC2(CCN(C(c3coc(CO)c3)=O)C2)C1 98689,c1(C(=O)NC2C(F)CCN(C(C(C)OCC=C)=O)C2)c[nH]c2cc(Br)ccc12 98690,c1(CC(N2CCC(NC(Cc3c(C)cccn3)=O)C2)=O)ccc2oc(O)nc2c1 98691,C1(C(=O)NC(CC2CN(C(C(C)OC)=O)C2)C)CCC(C(C)(C)C)O1 98692,N1(C(C(C(C)C)C)=O)CCC2(CCCC2NC(=O)C=CC2COC(C)(C)O2)CC1 98693,C1(C(=O)NC2C(C)OCC2)CCC(O)CN1C(c1cc(F)n(C)n1)=O 98694,c1(C(=O)NC2CCC(CNC(C3C(=C)CC3)=O)C2)cccc(-c2ccccn2)c1 98695,C1(C(N(C2CCCCC2O)C)=O)(CO)CCN(C(C2CCC(C(N)=O)C2)=O)C1 98696,C12(NC(=O)CCC3CCCO3)CC3CCC(C1C2)N3C(=O)C(O)c1ccsc1 98697,N1(C(C(C)N2CCCC2)=O)CCCC(CC(=O)NC2CCC(C3CC3)C2)CC1 98698,c1(C(N(C)CC2(NC(c3cc(C(=O)OC)[nH]n3)=O)CC2)=O)noc2c1CCCC2 98699,c1(C(=O)NC(CN(C(=O)CCC(C)SC)CC)C)cccc2c1NCCC2 98700,c1(CCC(=O)NC2CCC(NC(C(CC)OCC)=O)C2)ccc(OC)cc1F 98701,C(=O)(CCS(C)(=O)=O)NCCC1CCN(C(c2c(C)onc2)=O)CC1 98702,c1(C(=O)NCCN(C(=O)C(F)C(F)(F)F)CCOC)cc(OC)cc(F)c1 98703,n1(C(=O)CCCCc2ccccc2)ncc2c([nH]c3cc(F)ccc23)c1=O 98704,C1(C(=O)NCc2n(CC)ncn2)CC2CC1CC2NC(c1cc(C)nnc1C)=O 98705,C1(C2CCN(C(=O)CC3CCCOCC3)CC2)(NC(C(C(C)C)NC(C)=O)=O)CC1 98706,C(=O)(CS(=O)(=O)CC(F)(F)F)N(C1CCN(C(C(C2CC2)OCC)=O)C1)CC 98707,C(=O)(C1c2c[nH]nc2CN1C(=O)CC(=O)N(C)C)N(CCC)C(C)C 98708,C1(CNC(CC2CCCN(C)C2)=O)CN(C(=O)Cc2cccnc2)C(C)(C)C1 98709,c1(C(N(CCC)CCNC(C2(F)CCC2)=O)=O)cc(C)c2c(c1)CCC2 98710,C1(CC)CN(C(c2cnns2)=O)CC1NC(c1ccc(C(C)(C)CC)cc1)=O 98711,CC1C(C(N2CCC(C(=O)N(C)CC#N)C2)=O)C(O)C(=O)N1C 98712,C#Cc1cnn(C)c1C(N1CCC(C(C)NC(=O)C(CCC)OCC)CC1)=O 98713,c1(SC)cccc(C(N2CCC(NC(c3cncc(C)n3)=O)C2)=O)c1O 98714,N1(C(C2(C)CSC2)=O)CCC2(COC(CNC(C3(C)CCSCC3)=O)C2)C1 98715,c1(C(=O)NC(CNC(c2cc(CC)n(C)n2)=O)C)c[nH]cc(Br)c1=N 98716,c1(C(N(CCNC(C2CCC(COC)O2)=O)CC)=O)c(Cl)ccc(OC)c1N 98717,c1(C(=O)NC2CC(F)CN(C(C3CN4CCC3CC4)=O)C2)c(Cl)ccc(Br)c1F 98718,C1(NC(c2ccc(SCC(N)=O)cc2)=O)CCNCC1(F)F 98719,C1(C(C(=O)OCCCNCC)C)CCNCC1 98720,C(=O)(C1=C(C)CCOC1)N1CC2C(C(=O)NC(c3ccncc3)CC)(COC2)C1 98721,c1(C(N2CC(CCNC(C3CC(C)(CC)C3)=O)C2)=O)cc(C)ccc1[N+](=O)[O-] 98722,CC(C)C(F)(F)CC(=O)NC1CCC(C)N(C(c2ccoc2C2CC2)=O)C1 98723,C1(CC(=O)NCCC(CNC(=O)CC2OCCC2C)OC)CCCN(C)C1 98724,c1(C(=O)OC)cc(CNC(=O)N(C)Cc2ccc(Cl)s2)cc(Br)c1 98725,c1(CC(=O)NCC(CNC(C(CC(C)C)O)=O)C)coc2c(Cl)c(Cl)ccc12 98726,C1(NCC(COC)N)C(C)N(C)CCN1C 98727,c1(CC)cccc(C(N2CCC(CCNC(C3(C)C=CCC3)=O)C2)=O)c1N 98728,c1(NC(CN(C(COCCCC#C)=O)C)=O)ccc(C)cc1.C1(=O)CCN1 98729,C1(C(=O)NCC(CCNC(CC2(C)CC(F)(F)C2)=O)O)COC2(CCC2)CO1 98730,c1(CC)cc(C(=O)NCCCNC(=O)C(c2ccc(C)cc2)C)cn(C)c1=O 98731,c1(C(N2CC(C)N(C)C(C)C2)=O)ccc(S(=O)(=O)NCC2CCOCC2)cc1 98732,N1(C(C(C)CN(C)C(c2cnoc2C2CC2)=O)=O)CC2CCN(C)C2C1 98733,C(S(=O)(=O)C(C)C(=O)N(C(C)C(N)=O)C1CC1)c1n(COC)c(C2CC2)nn1 98734,Cc1c(C(N2CC3C(NC(=O)CCCCC4CC4)C3C2)=O)oc2c(Cl)cccc12 98735,c1(C(N(C(C)CNC(c2conc2C)=O)CC)=O)cc(F)ccc1N 98736,c1(C(C)=O)cc(=NCC2CN(C(C3CC(C)CO3)=O)CCO2)[nH]cn1 98737,N1(C(C2CC=C(C)CC2)=O)CCCC(C2CC2NC(=O)C(C)(C)C(F)F)C1 98738,CC1C(=O)N(C)CN1C(=O)NC1CCn2ncnc2C1 98739,c1(NC(C(C(C)NC(C(C)Cn2cccn2)=O)(C)C)=O)cccc([N+](=O)[O-])c1 98740,C12(C(N3CC(CC(C(=O)N(C(CCC)C)C)O)C3)=O)CCC(OCC)C1C2 98741,c1(OC)cc(NC(C2CN(C(c3ccn(C)n3)=O)CCO2)=O)ccc1O 98742,C(C)(C)(CC(F)C(=O)NCC(C1CCOC1)O)NC(C1CCN(C)C1=O)=O 98743,c1(C(N2CC3C(CNC(C(C)CC(F)F)=O)C3C2)=O)nnc2ccccc2c1N 98744,CN=c1[nH]cc(C(N2CCCC(NC(=O)C(C)CSc3ccc(F)cc3)C2)=O)s1 98745,C1(CNC(C2CC3CC3C2)=O)COCCN(C(c2ccncc2F)=O)C1 98746,Cc1cc(C(N2CC(N(C(=O)Cc3cnoc3)C)C3(CC3)C2)=O)nc(N(C)C)n1 98747,C1(S(C)(=O)=O)(C(=O)NC2CC(C)(NC(CC3C(C)C3(F)F)=O)C2)CC1 98748,N1(C(Cc2c(C)nc[nH]2)=O)CCC(C)(C)C1CNC(c1cnc(O)s1)=O 98749,c1(C(=O)NCC(CC)NC(CSCC=C)=O)cn2c(Br)cnc2s1 98750,c1(N(C)C)ccnc(C(=O)NCCC2CCCN2C(=O)C=Cc2ccco2)c1 98751,C1(NC(C2CC(C(C)C)C2)=O)CCC(O)CN(C(=O)Cc2ccc(Cl)cc2F)C1 98752,c1(OC)ccc(C=CC(=O)NC(C)(C)CN(C)C(C2CCCC(O)C2)=O)cc1F 98753,c1(CC(N2CCC(N(C(C=C(COC)C)=O)CCO)C2)=O)cccc2nsnc12 98754,Cc1cc(-c2cnccc2C(=O)Nc2cnn(-c3ccccn3)c2)ccc1N(C)C 98755,N1(C(=O)NC(C)Cc2cccc(F)c2F)CC(C)(C)CCC1CO 98756,C1(CNC(c2c(C)snn2)=O)CCN(C(c2cnn3ccn(C)c23)=O)CC1(F)F 98757,Cc1sc(COc2ccc(N3CCCC3=O)cc2)c(C)c1Br 98758,c1(NC(=O)NC2CCCN(CCC(=O)OC)C2)ccc(F)cc1C 98759,C(C(C(=O)N1CCC(CN(C)C)C1)n1cc(-c2csnn2)nn1)OCC 98760,CC(C(=O)NCc1cccc(CN(C2CCOCC2)C)c1)C(C)(C)C 98761,C(=O)(CCCCSC)N(C(=O)CN(CC(c1ccccc1)C)C(C)C)CC 98762,C1(C)(CNC(=O)OC(C)(C)C)CC(NC2CSCC2c2ccccc2)C1 98763,C1(NC(=O)C(O)C2CC2)CCC2CN(C(c3cc4c(s3)CCC4)=O)CC2C1 98764,C1(C(NOCC=C(C)C)=O)CCCN(C(=O)CCC(C)N(C)C)C1 98765,Cc1c(NC(c2csc(C(=O)NCC3CCOCC3)n2)=O)cc(F)cc1Br 98766,N1(C(C(C)OCC=C)=O)CC(NC(c2nc(O)c(C)s2)=O)C(n2ccnn2)C1 98767,C1(COC)CCCC1NC(=O)CC1(C)CCN1C(C)=O 98768,CCC(CC(=O)NC1CCC12CN(C(=O)Cc1cc[nH]n1)C2)C(C)C 98769,c12cc(cc(C)c1)CC(=O)NCC(OC)c1noc-2n1.C(CO)OCC 98770,C1(CNC(c2c(C(C)C)csc2)=O)CCCCN(C(=O)COc2ccsc2)C1 98771,C(C(C)CC(=O)N=c1ccn(C(C)C)[nH]1)NC(CCC(CCC)CC)=O 98772,N1(c2cc(NCc3cc(Br)cn3C)nc(C)n2)CCC(C)C2(CCC2)C1 98773,C1(F)(CNC(c2c(COC)cco2)=O)CCC(CNC(=O)C(F)=CCCF)CC1 98774,C1(NC(c2c(C)n(C)nc2)=O)CC12CCN(C(C1CC3CCC3C1)=O)CC2 98775,c1(NC(C2COC3(CCNC3)C2)=O)cc2c(cc1Cl)CCCC2 98776,C1(C)(C(=O)Nc2c(CC)noc2)CCCN1C(=O)CCCn1ccnn1 98777,c1(OC)cc(C(=O)NCC=CCNC(C2(CC)CCCC2O)=O)cnc1C 98778,C1(CNC(c2cc(OC)no2)=O)N(C(=O)Cc2cc(C)cc(F)c2)CCC1(C)C 98779,N1(C(C=NOC)=O)CC(F)CC1C(=O)NCc1cnc(S)nc1 98780,c1(OC)ncccc1C(=O)NCC(C)(C1CC1)NC(c1ccoc1Cl)=O 98781,CCCCCC(O)CC(=O)NCCN(C(=O)CC(C)C)Cc1ccccc1 98782,c1(CC(=O)N(CCOCCCC#C)CC)coc2cc(F)ccc12 98783,C12(c3onc(CC(C)S(C)(=O)=O)n3)COCC(C(C)(C)O)(C1)C2 98784,C(=O)(C(C(C)C)n1cc(C)cn1)NC1(CNC(CCCNC(C)=O)=O)CCCC1 98785,c1(CNC(C(CC)n2ccnc2)=O)cnn2c1CN(c1nnc(C3CC3)o1)CC2 98786,Cc1ccc(NC(=O)C(=O)NCC(C)CNC(=O)CSC(F)F)cc1 98787,C1(N(C(=O)Cc2cscn2)C)CN(C(=O)C(F)(F)c2ncccn2)CC1(C)C 98788,N1(C(C)C)CCCC(CN2CCCC2c2cc(Br)cs2)C1 98789,S(=O)(=O)(c1c(C)noc1C)NCC(=O)NCC1C(NC(CCCCCC=C)=O)C1 98790,c1(NC(C2CC3(CCN(C(=O)CCBr)CC3)C2)=O)cc2c(Cl)cccc2s1 98791,c12nc(cc(N3CCCC3)n1)NC2.c1(C(C(C)OC)C)cccnc1 98792,N1(C(C(CCCC)O)=O)CC2(C1)C(NC(=O)C(CC)C(C)C)CCS2(=O)=O 98793,N1(C(CCCC=C)=O)CC(N=[N+]=[N-])CC1C(N1CCCCC(CO)C1)=O 98794,C(=O)(CCC1=NNC(=O)CC1)N1CCC(CCOC)(NC(c2sccc2F)=O)C1 98795,CC(C)(C)C(O)C(=O)NC1CN(C(C23CC2CNC3=O)=O)CC12CC2 98796,N1(C(C(=O)NC(C(=O)N(CCC#C)C)C2CC2)C)CCOCC1 98797,C1(C(=O)NCC(C)CNC(C2(CO)CCOCC2)=O)(COC)CCCOC1 98798,N1(C(c2c(C)cc(=N)[nH]c2)=O)CCCCC1C1CCCN1C(=O)CCS(C)(=O)=O 98799,C(=O)(CCCCSC)NC(C1CN(C(c2ccc(COC)o2)=O)C1)C 98800,c1(OC(C(C2CCOCC2)OC)OC)cccc(S(F)(F)(F)(F)F)c1 98801,CCCC(CCC)=CC(=O)N(C(CNC(=O)C(C)(C)n1cnnn1)CC)C 98802,CC(=O)C(C)CC(C)C(=O)NC1CCC(CNC(C2CC2Cl)=O)CC1 98803,C1(NC(C(CCSC)NC(C)=O)=O)C2CCC1N(C(c1ccsc1Cl)=O)C2 98804,O=C(CC(C(F)F)NC(c1nc[nH]n1)=O)NCc1conc1C(F)(F)F 98805,N1(C(CC(C)(C)O)=O)CCN(C(c2cc(C#N)cs2)=O)CC1CC#N 98806,C1(NC(C2N(C)CCCC2)=O)CCC12CCCN(C(C1COCCN1C=O)=O)C2 98807,c1(C(C(=O)OCC)N(C(=O)Cn2cc(C3CC3)cn2)C)ccc(C)cc1 98808,C1(C(N2CCN(C3CC3)CC2)=O)CC(=O)N(OCc2ccc(Br)cc2)C1 98809,N1(C(C(C)NC(C)(C)C)=O)CC2CC(NC(c3coc(C(F)F)n3)=O)C1C2 98810,c1(N2CCC(CCC)C2)[nH]c(=NCc2cn(C3CCOC3)nn2)nc2sccc12 98811,C1(NCC(N)=O)CN(C(C2CCCO2)Cc2ccccc2)CCO1 98812,C1(C)(C(N2CCC(NC(C(F)(F)C3(OC)CCC3)=O)C2)=O)CNC(=O)C1 98813,C(=O)(CCC(=O)C1CC1)N1CC(COC)(NC(c2cc(C(C)C)oc2C)=O)C1 98814,C(=O)(C(C)(C)CC#N)NCCCOCCCN(C(C1(N(C)C)CC1)=O)CCO 98815,c1(CNC2(C)CN(CS(CC(=O)OC)(=O)=O)C2)cc(OC)c(OC)cc1O 98816,C1(F)(CNC(c2n(CC)nnc2)=O)COCCN(C(=O)CS(=O)(=O)NC)C1 98817,C=C(C)CC(C)(c1ccccc1)NC(c1cc(CNC)cs1)=O 98818,C(=O)(CC(C)c1cccnc1)NCC(CNC(CN(C(C(C)C)=O)C)=O)C 98819,C1(CNC(c2cc(C)n(C)n2)=O)(CO)CCCN(C(C2CCN(C)C(C)C2)=O)C1 98820,N1(c2ncon2)CCCN(C(=O)CCN2CCCC2=O)CC1.C(=O)OCC 98821,C1(NC(CCC=C)=O)COC2(CCN(C(=O)Cc3cn4c(C)cncc4n3)C2)C1 98822,N1(C(C2C(c3ccc(OC)cc3)C2)=O)CC2CC1CN2c1cc(F)ncn1 98823,C(=O)(C1=CC2C=CC(C1)C2)N1CCC(NC(C2(CC)CC2)=O)C(C)C1 98824,c1(CNCCCn2ncc(C)c2)ccc(C(=O)NCC23CC(CO)(C2)C3)cc1 98825,N1(C(C(CC)CO)=O)CCCC(C)(NC(c2cc(-c3ccco3)on2)=O)C1 98826,c1(CC)cnn2ccc(C(N3CCC(C)N(C(=O)C(C(C)C)C(C)C)CC3)=O)nc12 98827,c1(C(C(N2CC(C(=O)O)C(CO)CC2)=O)(F)F)cccc2ccccc12 98828,N1(C(c2c(C)n[nH]c2)=O)CCCC(c2cn(Cc3ccc(Cl)cc3)nn2)C1 98829,C1(C(N2C(C)CC2)=O)CCCC(NC(=O)COCC2CC2)C1 98830,C1(C2(O)CCC2)(CNC(CC2N(C(C=Cc3ccc(C)o3)=O)CCCC2)=O)CC1 98831,CC1=NS(=O)(=O)N(C)C=C1C(=O)N1CCOc2cc(CN)ccc21 98832,N1(C(CC(C)SC)=O)CC2CC(NC(c3ccnc(F)c3)=O)C2C1 98833,CCCC(C(=O)N(C(C(=O)NCCOCCO)C1CC1)C)NC(N)=O 98834,C(=O)(C(O)CC(F)(F)F)N1CCC(N(C(=O)COCCOC)CC#C)CC1 98835,c1(OC)ccc(C(N)=O)cc1C(=O)N(C)CCNC(=O)Nc1cc(F)cs1 98836,Cc1nn(C)c(=O)c(C(N2C3CCC2CC(NC(c2cnccn2)=O)C3)=O)c1C 98837,c1(C(N2CC(CNC(CC3C(CC)C3)=O)C(C)C2)=O)cn2c(n1)CCC2 98838,N1(C(C2(O)C(C)(C)C2)=O)CCC2(CCCN(C(c3cc([N+](=O)[O-])n[nH]3)=O)C2)CC1 98839,S(=O)(=O)(c1ccccc1CN)NCC(=O)NCC(COC)(C)OC 98840,C(CCCCC(=O)N1CC(C(N2CCOC(CF)C2)=O)(SC)C1)OCC 98841,C=CCCCCCC(=O)NCC=CCNC(C1CNC(=O)N1C)=O 98842,CC1CCCC(C)N1CC(=O)N(C1CN(C(=O)C(c2ccn(C)c2)C)C1)C 98843,C1(C(N2CC(NC(c3c(C)cc(F)cn3)=O)CC2(C)C)=O)CC2(CCC2)CCO1 98844,C1(CNC(CCCCC2CC2)c2n(CC(=C)C)nnn2)CCC2C1C2(F)F 98845,c1(C2(F)C(NC(=O)NCc3ccc(-n4ccnc4)cc3)C2)ccccc1Br 98846,C1(NC(CN(C(C(COCC)N(C)C)=O)CC2CC2)=O)CC(=O)N(O)C1 98847,C=CC(C)(C)CC(=O)NCCC1(C(=O)NC(C(C)(C)O)C2CC2)CCCC1 98848,C=CC(CCC)CC(=O)NC1CN(C(=O)Cn2ccc(=O)cc2C)CC(F)(F)C1 98849,C(=O)(C(O)C1=CCCCC1)NCCC1CCN(C(c2n(C)nc(C)c2Cl)=O)C1 98850,C(=O)(C#CC1CCCOC1)N(C1CCN(C(CC2(OCC)CCCC2)=O)C1)C 98851,C1(C(=O)NC(CC(C)NC(C2N(CC)CCCC2)=O)C)CCC2CC(C)CN2C1 98852,N1(C(C=CCCCC(C)=O)=O)CC(CNC(c2ccnc(C)c2)=O)N2CCC1C2 98853,c1(CC)cc(C(=O)NCCC2CCN(C(=O)CCC3(C)CC3)C2)c(C)o1 98854,c1(NC(C(C2CCC2)NC(c2c[nH]ccc2=O)=O)=O)cnn2c1OCCC2 98855,n1(C(CC)CC)nc(CC(C)CC)nc1-c1ccn(-c2ccc(C(F)F)cc2)n1 98856,c1(N2CCCC(OCC#C)C2)cc(Br)cc([N+](=O)[O-])c1C#N 98857,c1(OC)ccc(C(C)C(N2CCCC2C(C)NC(=O)CC2(CO)CC2)=O)cc1F 98858,c1(C(N2CC3CC(NC(C4(CCN(C)C)CC4)=O)C3C2)=O)ccc2ncnn2c1 98859,c1(C(N(C(CNC(CCCOC)=O)C)C)=O)sc(C(c2ccccc2)C)nc1C 98860,c1(CCCC(=O)NCC(O)CNC(c2ccccn2)=O)ccccc1F 98861,C(=O)(C(CC(C)C)OC)NCC(CCCC)NC(C1CC(CF)C1)=O 98862,C(=O)(C(C)(C)CCCF)NCC1(C)CCC(NC(CN(C2CC2)CC)=O)C1 98863,C(=O)(C1CC(=O)Nc2ncccc21)N(CCCNC(=O)C1CCc2nccn21)C 98864,C(CC(C(C)C)NC(=O)CCc1cncc(O)c1)NC(c1c(C)cns1)=O 98865,C(=O)(CCC(C)(C)F)NCCCC(C)NC(=O)C1=NOC(C(C)(C)C)C1 98866,C1(NC(c2ccn(C3CC3(F)F)n2)=O)CN(C(=O)COC2CC2)CC12CCC2 98867,C1(C#N)(C(=O)NCC(CC)NC(C2(CC)CCC2)=O)CCC1 98868,c1(C(=O)Nc2occ(C(=O)OC)c2C(C)=O)c(F)c(F)c(N)c(F)c1F 98869,c1(C(=O)NCC(CN(C)C(C23CC(CO)(C2)C3)=O)O)ccnc(Br)c1N 98870,C1(NC(=O)OC(C)(C)C)(CNC(c2cc(C(F)F)on2)=O)CCCS(=O)(=O)C1 98871,c1(C(=O)NC2CCC(N(C(CC)=O)C)C2)nnn(C2CC2)c1-c1ccccc1 98872,CC1CC(=O)NCC1C(=O)NCC1CCCN1C(c1cc(CC2CCC2)c[nH]1)=O 98873,c1(NC(C(C(C)C2CC2)N(C(C)(C)C(F)F)C)=O)ccc2c(c1)CCC2.CC=C 98874,N12CCC3CC13NC(=O)C1CC(C1)C2=O.C1CC(CO)(CO)C1.CC(C)(C)C=O 98875,C1(C(=O)OC)CNC(=O)CC12CCN(C(=O)NCC13CCCCC1C3)CC2 98876,c1(C(C(=O)NCCN(C(CC(C)OC)=O)C2CC2)(C)C)ccc(Cl)nc1 98877,C1(NC(C2CC23CC3)=O)C2CC(O)C1N(C(c1ccccc1-c1cc[nH]n1)=O)C2 98878,c1(C(=O)NC(C(C)C)CNC(=O)CC2CCC(=O)N2)cnc(N)c(O)c1 98879,C1(CNC(CN(C(C(C=C)OC)=O)CCOC)=O)CCCC12CCC2 98880,C(=O)(C(C)(C1CCCCC1)NCCCOC(=O)C1CC1)OC 98881,N1(c2n(Cc3cc(C)oc3C)c(C3CCC(=O)N3)nn2)CC2COCC2C1 98882,C1(CN(C(CC(C)c2ccccc2)=O)C)CCCN(C(=O)CCc2ccc[nH]2)C1 98883,C12(C(N3C(C(N(CCCC)C)=O)CC=CC3)=O)CCC(C1)C2(C)C 98884,C1(CC(=O)NC2CC(NC(c3ccc(C(=O)OC)o3)=O)C2)C(=O)NN=C1C 98885,c1(C(N(CC(C)NC(c2ccc(C)nc2)=O)C)=O)n[nH]c2c1CCOC2 98886,Cc1cnccc1C=CC(=O)NC1CCCC(NC(c2c(C)nn(C)c2Cl)=O)C1 98887,Cc1oc(Br)cc1C(=O)NC1CC2(C1)CC2NC(=O)CN1CCCOC1=O 98888,N1(C(c2ccc(CC)cn2)=O)CC(CNC(=O)CCCc2cccs2)CC1(C)C 98889,CC1C(NC(=O)C=CCN(C2CCCC2)C(=O)CCNC(N)=O)CCCN1C 98890,C(c1c(Cl)nc2sccn12)=CC(=O)NC1C2CCN(C(=O)C(O)CC(F)(F)F)C12 98891,C(C)(CN=c1[nH]c(Cl)ncc1C(F)(F)F)NC(c1c(CC)occ1C)=O 98892,c1(C(N2CCN(C(c3cc(CCO)on3)=O)C3CC23)=O)cccc2c1COCC2 98893,C1(CNC(c2ccsc2F)=O)CCC(NC(c2[nH]nnc2C2CC2)=O)C1 98894,C(CNC(=O)CSc1nnnn1C)(CC(F)(F)F)NC(C(C)CSC(F)(F)F)=O 98895,c1(C(=O)NCCn2nccc2C(=O)NCC=CCOC)ccncc1Cl 98896,CC1CCN(C(C2(CO)COC2)=O)CC1NC(=O)CC(F)(F)Br 98897,c1(OC)ccc(C)c(C(=O)N(C2CCN(C(=O)CCC(C)SC)C2)C)c1 98898,c1(CC)ccc(F)cc1C(=O)NCCCC1CCCCN1C(c1[nH]ccc1C)=O 98899,C1(CCC(=O)NCC(C2CCOC2)NC(C(C)SCC)=O)(N(C)C)CCCCC1 98900,c1(C(N2CCC(C(C)(C)NC(CC3N(CC)CCC3)=O)C2)=O)ccc(CO)cn1 98901,c1(C(C)C)ccc(C=CC(=O)NC2COCCN(C(=O)CCC3CC3)C2)cc1 98902,c1(CC(=O)NCCC2N(C(C(C)SC)=O)CCOC2)coc2ccc(F)cc12 98903,CN1CCN(C(=O)Cc2cc(Cl)ccc2Cl)C(CNC(C2CCCN2C)=O)C1 98904,C1(N(C(CCC)=O)C)CCN(C(c2cc(Cl)ncc2OC)=O)CC1C 98905,C1(NC(C2(SC)CN(C(C(CCC)CC)=O)C2)=O)CC(C)(C)OC1(C)C 98906,CC(C)(O)C(C(=O)NC1CCCC1O)NC(c1cnn(C2CC2)c1)=O 98907,C(C(C)CC(=O)NCC1(C(N)=O)CN(C(=O)C=CCn2cncn2)C1)OC 98908,N1(C(CC=CC=C)=O)CC(C2CC2)(C(=O)Nc2ccc(F)c(CO)c2)C1 98909,C(C(C(=O)NCCN1CCC1)NC(c1ccn(C(F)F)n1)=O)OC 98910,N1(C(C(COCC)C)=O)CC(NC(c2csc(=N)[nH]2)=O)CC1C 98911,C1(CC)(NC(=O)C=CC(=O)NC)CCN(C(C2CC2c2ccco2)=O)CC1 98912,C1(=O)CCCNC(=O)C2CC(C2)N1.C1(CCOC)CCCN1C(C)=O 98913,c1(COC)ccc(C(=O)NC23CC(NC(=O)CC(=O)Nc4nccs4)(C2)C3)o1 98914,N1(C(C2CCC3CC23)=O)CCOC2(CCCN(C(c3ocnc3C(F)F)=O)C2)C1 98915,c1(C(=O)NC2C3CN(C(CCC(C)SC)=O)C2C3)ncc(Cl)cc1F 98916,C12(CC(=O)N(CCCCN(C)C(C3C4CCC(=O)C34)=O)C)CCCCC1C2(F)F 98917,Cc1n[nH]c(C)c1C(=O)OC(=O)CNC(=O)CNC1CCC(C(F)(F)F)CC1 98918,C(=O)(CC(O)CC(C)(C)C)N1CC(C(=O)Nc2c(SC)c(F)ccc2)C(F)C1 98919,c1(C(N(C(C)C)CCNC(C2CCCCO2)=O)=O)c(Cl)c([N+](=O)[O-])nn1C 98920,C12(C(=O)NCC3C4CN(C(C5C(C#C)C5)=O)CC43)CCC(CC)(CC1)OC2 98921,N1(C(c2nn(CC)c(C)c2)=O)CCC(N(C)C(c2cc(OC)nn2C)=O)C(C)C1 98922,N1(C(C2(COC)C(C(=O)OC)C2)=O)CCN(C(C)Cc2cccc(C)c2)CC1C 98923,C1(C(=O)NCC2CNC3CC23)CSC(c2ccccc2O)=N1 98924,N1(C(C=COCC)=O)CCC2(CCCC2NC(=O)CCc2cccc(C#N)c2)C1 98925,Cc1ccc2c(C(=O)NCC3(F)CC(NC(C4CCSC4)=O)C3)cnn2c1C 98926,c1(C(=O)NCC(CC)NC(=O)OC(C)(C)C)ccc2occc2c1 98927,c1(C(=O)NCC(CNC(C2CCC(=O)N2)=O)CO)c[nH]c(=O)c2ccncc12 98928,c1(NC(N2CCC(N(C)CC)C2)=O)ccnc(S(C)(=O)=O)c1 98929,C1(N(C(CN(CCOC)C)=O)C)CN(C(c2cc(F)n(C)n2)=O)CC1F 98930,c1(OCC(N2CCCC2CNC(C23CSCC2C3)=O)=O)ccccc1 98931,c1(NC(C)=O)ccc(C(=O)N(CC(O)CNC(=O)C(F)n2ccnc2)C)nc1 98932,c1(C(=O)NC2CN(C(c3nn(CC)c(C)c3)=O)CC2F)cc(Br)ccc1O 98933,c1(CC)cnc(C(=O)NCC2CC2NC(c2cccnc2C)=O)cn1 98934,c1(SCC=CCNC(c2cn(C(COCC)C)nc2C)=O)ccc(F)cc1Cl 98935,N1(CC2(C(N)=O)CN(C(c3ccoc3)=O)C2)CCC(F)CC1.CC(C(=O)N)N(C)C 98936,c1(C(=O)Nc2ncc(-c3c(F)cccc3F)s2)cccc2scnc12 98937,N1(C(c2cn(C)[nH]c2=N)=O)CCCC(NC(c2nocc2Cl)=O)CC1 98938,N1(C(Cc2c(C)ccnc2)=O)CC(F)(F)CC1CCNC(C1CCCOC1)=O 98939,c1(C(=O)NCC2(F)CCN(C(C(=CC3CCCC3)C)=O)C2)cccn2cncc12 98940,c1(C(=O)NCC2(N(C(=O)C(c3ccccc3)F)C3CC3)CC2)cnc2sccn12 98941,C1(F)(C(=O)Nc2nccnc2Br)CCN(C(c2occc2Br)=O)CC1 98942,N1(C(C(F)OC)=O)CC(O)(CCNC(c2ccncn2)=O)C1 98943,C1(C(=O)NCCCN(C)C(C2C(Cl)(Cl)C23CC3)=O)CCc2ccccc2C1 98944,N1(C(=O)Nc2c(CC)ccc(C(F)(F)F)c2)Cc2ccccc2SCC1C 98945,c1(NC(CC(C)F)C)nc2ccccc2nc1NCCN1CCCOCC1 98946,N1(C(c2c(C)n(C)cc2)=O)CCN(C(C2(C)CC(F)C2)=O)C2(CCC2)C1 98947,C(=O)(CC1CCc2ccccc21)NC(C1CCCCC1)CNC(C=CSC)=O 98948,N1(c2cc(NCC3CCOC3)nc(COC)n2)CC2CC(F)CC2C1 98949,c1(N2CCC(O)(NCCNC(CC)=O)CC2)nc(C(F)(F)F)nc(C)c1Br 98950,C1(C(=O)NCc2cnc(C)s2)CN(C(c2csnc2C)=O)CCN1 98951,C1(C(N2CC(CNC(c3n(C)c(=O)ccc3)=O)C(C)C2)=O)CCc2nn[nH]c2C1 98952,C(=O)(CCC(C)(F)F)NC1CCC(NC(C(C)NS(CC)(=O)=O)=O)CC1 98953,N1(C(c2cncc(N)c2)=O)CCCC(C2(NC(c3ccsc3)=O)CC2)C1 98954,C1(C(N2CCC(NC(C3CCCS3)=O)CC2)=O)CCC12CCNCC2 98955,c1(C(=O)NCC2(OC)CN(C(C(CC)O)=O)C2)nc2n(c1C(C)C)CCCC2 98956,C(=O)(CCCCC1CCCCC1)N(C)CCNC(C12CC(O)C1C2)=O 98957,C(CCCCC(=O)NCC1CCN1C(c1ncccc1O)=O)=CC 98958,Cc1ccc(F)c(C(=O)NC2CCC(N(C)C(c3cccnc3)=O)CC2)n1 98959,C(=O)(CCCCC1CC1)N(C1(CC(=O)N(C(c2cc[nH]n2)C)C)CC1)C 98960,c1(C(N2CC3C(CNC(CCCC#N)=O)C3C2)=O)cc2ccccn2n1 98961,S(=O)(=O)(c1cc(C)ccc1C)NCCC(=O)N(C1CCNCC1F)CCCC 98962,N1(CCC)CCCCC1C(=O)N(C)CC1(NC(=O)Cc2ccc(O)nc2)CC1 98963,C=CCS(=O)(=O)NC1CCN(Cc2c[nH]nc2C)C1 98964,C(=O)(CCC(C)(C)C)N1C(C2CCN(C(CCCc3c(C)ccs3)=O)C2)CCC1 98965,c1(N(C2(C)CCNC2=O)C(C2CC3(CSC3)C2)=O)c(Br)cncc1[N+](=O)[O-] 98966,N1(C(C2N(C)CCC2)=O)Cc2ccccc2C1CNC(C1CCCO1)=O 98967,c1(C(=O)NC2CC3(C(C(=O)NC4(CC#C)CC4)C3)C2)cc(C#N)cn1C 98968,CC1C(NC(=O)C(C)(O)C2CC2)CC2CCC1N2C(c1cc(Br)co1)=O 98969,Cc1ccc(C(C)(C)C(N2CCC(C)(NC(=O)CC(C)O)C2)=O)cc1 98970,CCC(C)(CO)C(=O)N1CC(C(=O)NCc2oc(C)nc2C)C(F)C1 98971,Cc1[nH]nc(C(N2CCCC2C2(NC(C3CSCCS3)=O)CC2)=O)c1[N+](=O)[O-] 98972,CN1CCCC1CC(=O)NC1CC(NC(C2(C(=O)NC(C)(C)C)CCCC2)=O)C1 98973,C(=O)(CCCC(C)(C)CC)N1CCC(C(F)F)(CNC(C2CCN(CC)C2)=O)C1 98974,N1(C(c2c(OC)ccs2)=O)CC2(CCC(CNC(=O)COC3CC=CC3)O2)C1 98975,C(=O)(C(O)CCC(C)C)NCC1CCN(C(CCOCCC)=O)CC1O 98976,CCC(CC(=O)NC1(CCNC(=O)CCSC)CCC1)c1ccccc1 98977,c1(OC)ccc(OC)c(C(=O)NCC2CCN2C(=O)Cc2c(F)cccc2F)n1 98978,CC1CCCN(C(c2ncccc2C2CC2)=O)C1CCNC(c1cnc(Cl)s1)=O 98979,C(C(CC(=O)NC1CCC2(CC2)C1)NC(c1c[nH]c(C(N)=O)c1)=O)OC 98980,C(=O)(CC(O)CC(C)(C)C)NC1CCC(F)(CNC(C(CC#C)C)=O)C1 98981,c1(CNC(C)=O)ccc2c(c1)CN(C(c1cc3c(cc1O)OCO3)=O)C2 98982,c1(C(=O)NC(CC(N)=O)C(N2CCC3C(C2)C3(F)F)=O)ccn2cncc2c1 98983,C1(CNC(CC2(N(C(=O)CCc3cncnc3)C)CC2)=O)CC12CCOCC2 98984,Cc1ccccc1-n1ccc(C(=O)NC(C)CCNC(=O)C(C2CC2)N(C)C)n1 98985,c1(C(=O)NCC(CNC(C2C(C(N)=O)C2)=O)F)ccsc1Cl 98986,C1(NC(CN2C(CC)C(=O)NCC2)=O)CCc2nc(N(C)C)ncc2C1 98987,N1(C(c2cc(OCC)cc(F)c2)C)CCn2c(cnc2C(F)F)C1.c1(C)nnnn1C 98988,c1(C(N(CC(C)NC(c2cc(O)nc(Cl)c2)=O)CC)=O)cnc2n1CCCC2 98989,N1(C(c2cncc(C=C)c2)=O)CC2CCC1CN2C(c1cccc(C)n1)=O 98990,N1(C(C2C(NC(C(CCCC)O)=O)C2(C)C)=O)CC2CCCC(C2)C1 98991,c1(CC(N2CC(CCNC(CCC(C)SC)=O)C2)=O)cc(C(F)(F)F)cc(F)c1 98992,C1(SC)CN(C(=O)C=C(C)c2cccs2)CC1NC(=O)Cc1ccsc1Cl 98993,N1(C(c2n(C)ncn2)=O)CCCC2(NC(c3cccc4cnnn34)=O)CCCC12 98994,c1(C(=O)NC2C3(CC(NC(C(CCOC)C)=O)C3)C2)c(F)cncc1Cl 98995,CCCC(C)(O)CC(=O)NCCOCCOCCCNC(C1CCN(C)C1=O)=O 98996,N1(C(C2CCN(C(Cc3cn(C)nc3)=O)C23CCC3)=O)CCC2(CCOC2=O)C1 98997,c1(C(=O)NC(c2nc[nH]n2)C)conc1CNC(=O)CCc1cncn1C 98998,C1(CCCN(C)C)CNC(=O)CN1C(c1ccc(OCc2cccnc2)cc1)=O 98999,C(c1ccc(C)cc1C)=CC(=O)NCC1CC(NC(C2CN(CC)C(=O)C2)=O)C1 99000,c1(CNC(c2ccccc2Br)C)c(Br)nnn1C 99001,C(CC(C(=O)NC(C1CCN(C(c2ncc[nH]2)=O)CC1)C)NC=O)SC 99002,c1(OCC)cncc(C(=O)NCC(F)CNC(c2c[nH]cc2Br)=O)c1 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99302,c1(C(N2CCC(OC(C)=O)C2)=O)cn(CC(F)(F)F)nc1C 99303,CC1CN(C(c2cscc2Cl)=O)CCCN1C(C12CC(C)(C1)OC2C)=O 99304,N1(C(CC2(C)CCN(C(c3cnn(C(F)F)c3)=O)C2)=O)CCCC(O)(C2CC2)C1 99305,C1(C2CCCN(C(=O)C3=COCC3)C2)(NC(c2c(OC)ccs2)=O)CC1 99306,c1(C(N2C(CN(C(CC=C)=O)C)CCC2)=O)ccc(C2CC2)cc1 99307,Cc1sccc1C(c1cnn(C)c1)NC(=O)NC1COCC1C(F)F 99308,CC(N=c1nc2sccc2c(NCc2csc(Br)n2)[nH]1)c1cnccn1 99309,CC(CC(=O)NCC(C12CCC(CC1)C2)NC(=O)C(F)n1ccnc1)C(F)(F)F 99310,c1(SC)cc(=NC(=O)C2N(C(=O)Cn3ccnc3)CCCC2(C)C)[nH]n1C 99311,Cc1c(CC(N2CCC(CCC(=O)NC(CO)CCF)C2)=O)ncn1C 99312,C1(CC#C)CCN(C(CSCC)C(=O)NCCC2CC2)C1 99313,c1(CC(=O)N(CCC(C)NC(=O)C(C2CCOCC2)C)CC)c[nH]ccc1=O 99314,C1(NC(C(CCC)CCC)=O)COC2(CCN(C(=O)CCCCC(C)C)C2)C1 99315,c1(C(=O)NC(C(C)C)CCN(C(=O)C(=O)N(C)C)C)cc2n(c1)CCOC2 99316,Cc1c(-n2cc(C3(C)CCCN3C(C3CCOC3C)=O)nn2)cccc1Br 99317,C(=O)(CCCC(=O)N1CCN(C(=O)C(C)C)C(c2ccccc2)C1)NCCC 99318,C1(C)(C(=O)NCC(C2CCC2)NC(C(C)N(C)C)=O)CCCCC1 99319,C1(NC(C2CCN(CC#C)CC2)=O)CN(C(C2(CC)CC2(F)F)=O)CC2(CC2)C1 99320,Cn1c(C(=O)NCC2(C(N3CC(OCF)C3)=O)CCCO2)cnc1Cl 99321,N1(C(c2cc(Br)no2)=O)CCOCC1CCNC(C1(CO)CCC1)=O 99322,C1(NC(C2N(CC)CC2)=O)C=CC(C(=O)N(CCC(O)CO)C)C1 99323,C(CN=c1cc[nH]cc1S(=O)(=O)NC1CC(O)C(F)C1)C1N(C)CCCC1 99324,Cc1ccc(F)c(C(N2CC=CC(NC(=O)CC(C)C3CC3)C2)=O)n1 99325,c1(-n2cc(CCCNC(c3csc(-c4ccccc4)n3)=O)nn2)cccc(F)n1 99326,Cc1[nH]nc2ccc(C(=O)NCC(CO)NC(=O)CCCn3ccnc3C)cc12 99327,c1(CC)cscc1C(=O)NCC1CC1N(C(c1ccncc1)=O)C(C)C 99328,N1(C(CCCCC)=O)CC2(C1)CN(C(c1ccc(C3CCCO3)nn1)=O)C2 99329,Cc1ccc2[nH]nc(C(=O)NCC3(NC(c4cc(C)n(C)c4)=O)CCOC3)c2c1 99330,C(=O)(C(F)C1=CCCCC1)N(C(CNC(c1c(C)nc(C(C)C)nc1O)=O)C)C 99331,Cc1cccn2nc(C(=O)NCC(O)CNC(=O)C(C)Cc3ccncc3)cc12 99332,c1(COCC(N2CC(N(C(c3cc(OCC)n[nH]3)=O)C)C2)=O)cc(C)cc(C)c1 99333,C(=O)(C(C)(C)CS(N)(=O)=O)NCC(CN(C(=O)Cc1cc2ccccc2o1)C)O 99334,n1(C(C)C)ncc(C(=O)NCC(C(C)(C)C)NC(C2(Cl)CC2(F)F)=O)c1C1CC1 99335,c1(C(N2CC(CNC(c3[nH]cc(CC(C)C)c3)=O)C2)=O)ccc2c(c1)CCO2 99336,N1(C(CCc2ccc(C)s2)=O)CCC(CNC(C2CCCCCC2)=O)CC1C 99337,N1(C(C2(CC)CCCC2O)=O)CC=C(C(=O)Nc2ccn(C3CC3)n2)CC1 99338,C1(C(=O)OCC=C)CCC(CCC(=O)N(C(=O)CCc2cncn2C)C2CC2)C1 99339,C(=O)(C(C(C)CCC=C(C)C)N(c1ccc(CC)cc1)C)NCCC(=O)OCC 99340,c1(NC)cc(C(N2CC(C)(NC(=O)C(C)NC(C3CCC3)=O)C2)=O)cc(Cl)n1 99341,C#Cc1cccc(SCC2C=CCC(C(=O)Nc3cnc(CC=C)nc3C)C2)c1 99342,c1(C(N2C(C(CNC(CC(COC)C)=O)(C)C)CCC2)=O)cc2occc2[nH]1 99343,CCS(=O)(=O)CC(=O)NCC1CCCCN1C(C1CCCN(C(N)=O)C1)=O 99344,C1(NC(c2c(CC)[nH]nc2Cl)=O)COCCN(C(=O)COCC2CCC2)C1 99345,c1(C(=O)NCC2CCN(C(=O)C=CC3CC3)C2)ccnc(Br)c1F 99346,c1(C(=O)NC(COC)CC(=O)NCc2cccnc2F)ccc2cc[nH]c2c1 99347,Cc1c(CNCCN2CCN(C(=O)Cn3cccn3)CC2)cnn1C 99348,c1(C(=O)NC2CC(CCNC(CNC(C)=O)=O)C2)c[nH]nc1C(F)(F)F 99349,C1(NC(CCOC(C)C)=O)CCCC(NC(=O)CCN2CCCCC2)C1 99350,c1(C(=O)NCC(CC=C)NC(c2cnn(C3CC3)n2)=O)ccc(=NCC2CC2)[nH]c1 99351,C1(C(=O)NC(CNC(CCc2onc(C(C)C)n2)=O)(C)CO)CCN(C)C1C 99352,C1(N(C(=O)CONC(C2CCCCC(=O)N2)=O)C)CCCCCC1CO 99353,c1(CCC)cc(C(=O)N(CCC(C)NC(=O)C(C)Cc2ccncc2)C)n[nH]1 99354,C#CC1(C(N2CCCC(C(C)NC(C3COCCN3C)=O)C2)=O)CCCC1 99355,CCC1=C(C(=O)NCCC(C)(C)NC(=O)CCc2ccc[nH]2)CCCO1 99356,C1(CC(=O)NCCCCCn2cc(C(C)(C)OC(C)=O)nn2)C(=O)N(C)N=C1C 99357,Cc1cc(C(N2CC(NC(c3nc(O)c(C)s3)=O)C3CC23)=O)n2nc(C)cc2n1 99358,N#CCC(=O)NNC(=O)Cc1cc(Cl)ccc1Cl 99359,c1(N(CC)CC)ccc(C(=O)NCC2CCCC2NC(C2(CF)COC2)=O)cc1 99360,C1(NC(CCN(CC)CC)=O)CCC2CCN(C(c3ccc[nH]3)=O)C1C2 99361,C1(C(N2CCC(CCNC(C(C)Nc3scc(C)n3)=O)C2)=O)(CO)CCCCC1 99362,c1(C)sc(CO)nc1C.CCC(C)(CNC(=O)C(C)NC(c1cccs1)=O)OC 99363,C1(C(N2CC(N(CC=C)C)C2)=O)CC12CCN(C(=O)C1=CCCC1C)C2 99364,N1(C(C=CCN(C(C(C(=O)OC)OC)=O)C)=O)CCC(F)(CO)CC1 99365,Nc1cccc(C=CC(N2C3CCC2C(CNC(=O)COC2CC=CC2)C3)=O)c1 99366,C(=O)(C1Cc2ccccc21)N1CCC(C(=O)NCC(C)CO)CC1(C)C 99367,c1(NC)ccc(C(=O)NCC(C)(O)CNC(C2CCCCC2O)=O)cc1 99368,c1(C(=O)NCC(CCCC)NC(C2CC2(C)C)=O)cnc2c(F)ccc(F)c2c1 99369,CC(C)(C)CC(=O)N1CC(NC(c2cnn(C3CC3)c2)=O)C2CC12 99370,N1(C(c2ccc(C(=O)NC)cc2)=O)CC(N(C)C(c2conc2C)=O)C2(CC2)C1 99371,N1(C(Cc2cccc(COC)c2)=O)CCN(C(c2nc(O)sc2C)=O)C2CC12 99372,N1(C(CC(C)SC2CCCN2C(=O)OC(C)(C)C)=O)CCCCC1C1CC1 99373,c1(C(=O)NCC2CC(NC(CN3C(C)CC3)=O)C2)cc(F)ccc1N1CCOCC1 99374,Cc1cccc(C2=CCN(C(=O)NCC3CN(C)CCO3)CC2)c1 99375,C(CN=c1nc(O)c(Cl)c[nH]1)N(C(C(c1ccc(C)s1)C)=O)C(C)C 99376,N1(C(CC2C=NN(C)C2=O)=O)CCC(C(=O)Nc2cnc(Cl)nc2)CC1(C)C 99377,CC1COc2c(C(=O)NC3(CNC(=O)C=CS(C)=O)CC3)cccc21 99378,c1(C(N2CCCN(C(CC(C)C3CCCO3)=O)CC2)=O)ncccc1N=[N+]=[N-] 99379,C(CC(=O)Nc1cccc(NC(=O)C(=O)NCC)c1)(C(C)C)OCC 99380,C(=O)(C1=C(Cl)CCOC1)NCC12CN(C(c3c(OC)cccn3)=O)C(C1)CO2 99381,C1(NC(CCOCC)=O)CCCC(NC(=O)C(C)(C2CC2)NC(C)=O)C1 99382,c1(C(=O)NCC(CNC(C2(CCC)CC2)=O)C)cc(OC)c(OC)cc1O 99383,N(C(=NCCc1ccc(Cl)cc1)NCC1CCC(C)O1)Cc1c(CC)nn(C)c1 99384,c1(N2CCC3(C(NCc4c(F)cccc4Br)C3)CC2)ccnc2cc(Br)nn12 99385,CCC(CC(F)F)C(=O)N1CCCC1C1(NC(=O)Cc2ccc(F)cc2)CC1 99386,CS(=O)(=O)CC(F)(F)CCNC(=O)Nc1nn[nH]c1C(F)(F)F 99387,N1(C(C2CC(C#C)(O)C2)=O)CCC(C)(C)C1CNC(c1cc(C)nn1CC)=O 99388,c1(C(N2CCC(NC(C3CCCS3)=O)C2)=O)cc(F)c2cc[nH]c2c1 99389,N1(C(c2c(C(C)=O)cccc2)=O)CC(NC(c2cnn3c2SCC3)=O)CCC1C 99390,c1(COC)nn(C)cc1C(=O)NC12CC(NC(c3cc(C)n(C)c3)=O)(C1)C2 99391,N1(CC(=O)NCCCN2CCN(C(C(CC)(C)O)=O)CC2)C(=O)NC(C)(C)C1=O 99392,C(=O)(C1=CC2(CCOC2)C1)N(CC(C)(C)CNC(=O)CCCn1ccnc1)C 99393,CC(C)(CCCCNC(C1CC(C2CC2)=NO1)=O)NC(C1CC2CCC(C1)S2)=O 99394,CC(C)CC(C)C(=O)NCC1CC2CCC1N2C(C1CC=CCC1)=O 99395,S(=O)(=O)(c1ccc(Br)cc1NCC1CCCCCCC1)N1C2CC(=C)CC1CC2 99396,c1(C(N2CC(NC(C(CCOC)C)=O)(COC)C2)=O)cc(C)c(F)cc1F 99397,N1(C(C(CCC#C)O)=O)CCCN(C(c2cccc(C)c2N)=O)C(C(C)C)C1 99398,CC(C)(O)C(F)CNC(C1(C2CCCN2C(=O)CC2CCCO2)CC1)=O 99399,CC1CC(C(C)NC(C2C=CC(N(C3CC3)C(=O)OC(C)(C)C)C2)=O)CC(C)C1 99400,CC1C(NC(c2cnccc2Cl)=O)C(C)CCN1C(c1cc(N(C)C)ccn1)=O 99401,c1(OCC)ccc2c(c1)C(NC(=O)N(CCCc1nc(C)cs1)CCO)CCO2 99402,N1(CC(=O)NCCCN(C(=O)C(C)Sc2ccccn2)CC)CCCCS1(=O)=O 99403,c1(C(=O)NCC2CCCN2C(c2cnn(C3CCOC3)n2)=O)cnn2c1CCC2 99404,c1(CNCC2(C)CCN(S(=O)(=O)CC3CC(N)C3)CC2)ccc(Cl)c([N+](=O)[O-])c1 99405,C1(C(=O)NCc2cc(C)oc2)CCCCN(C(C2CC(N(C)C)C2)=O)C1 99406,CCC(C)(O)C(=O)N(CCCNC(C1C(C(F)F)C1(C)C)=O)CCO 99407,CC(C)CCCC(C)C(=O)NC1CC(C(F)C(=O)NCCc2c[nH]nc2O)C1 99408,N1(C(c2c(OC)cc(Cl)c(Cl)c2)=O)CCCC2(CCC2O)C1 99409,c1(-n2c(C(c3cccs3)NCc3n(C(C)C)ccn3)nnn2)ccc(Cl)cc1F 99410,Cc1ncc(Br)c(N2CCOC(C(=O)Nc3ccnc(-c4ccccn4)c3)C2)n1 99411,c1(C(=O)NCCN(C(=O)COc2cc(F)cc(Br)c2)C)ccc(OCF)c(F)c1 99412,Cc1csc(Cl)c1C(=O)NCCNC(=O)CCn1ccnc1-c1ccc(Cl)cc1 99413,N1(C(c2cc(CNC(CC(CC)O)=O)no2)=O)CCOC(C)CC1 99414,c1(NC)cncc(C(=O)NCC(C)(C(C)C)NC(=O)CN(C)S(N)(=O)=O)c1 99415,c1(CC)cc(C(=O)NCC(C)(C2CC2)NC(c2cc(C)[nH]n2)=O)ccc1O 99416,CC1SCCCC1C(N1CCC2CC12C(=O)NCCNC(=O)CO)=O 99417,Cc1cn2ccc(C(N3CCC(NC(=O)COc4ccsc4)C3C)=O)cc2n1 99418,N1(C(C2C(C)(C)C2)=O)CCN(C(c2ccnc(C3CC3)c2)=O)C(c2cccs2)C1 99419,Cc1nc(Cl)ccc1C(=O)NCCC1CCCN1C(=O)C(F)C1CCOC1 99420,N1(C(C(C)S(N)(=O)=O)=O)CC(NC(=O)C(F)(F)C2CC2)CC12CCCCCC2 99421,C(c1ccccn1)=C(C)C(=O)NC1CCC(C)(CNC(c2ccncc2)=O)C1 99422,c1(C(=O)NCCC2CC(NC(C(C)O)=O)C2)sccc1C(C)(C)C 99423,CC1CCN(C(c2ncsc2C2CC2)=O)CC1NC(=O)CSc1cn[nH]c1 99424,C(CC(C(C)C)NC(c1nnnn1C1CCOCC1)c1cncs1)OC 99425,C=C(C)CC(C(=O)NCC1(C)COCCO1)NC(=O)CC1CCCN1C 99426,N1(C(COCCOC)=O)CC(C(C)(C)O)(CNC(C2CCCN2C(C)=O)=O)C1 99427,C1(CNC(c2cnn(C)c2Cl)=O)CCN(C(=O)C(C)(O)C2CCC2)CCC1(F)F 99428,c1(C(N2CCC(CC)C2C(=O)NCC(c2ccncc2)C)=O)cnc(O)cc1C 99429,C1(NC(C=CCN(C(=O)CCOC2CCCC2)C)=O)CCC(F)(F)C1 99430,C1(CNC(C(COC)N(C)C)=O)CCCC2(CN(C(=O)C(CC(C)C)OC)C2)O1 99431,S(=O)(=O)(c1c[nH]ccc1=NC(C(C)(C)C)C(C)C)NCCC(CC)C 99432,C(=O)(C1c2c[nH]nc2CN1C(C1CCC1C)=O)N1CCCC(C)(OC)C1 99433,N1(C(C(=CC2CCCC2)C)=O)CC2CCC(C1)N(C(=O)CN1CC(C)C1)C2 99434,N1(C(C(C)C(C)(F)F)=O)CCC2(CCC2)C(CNC(=O)CCCCC2CC2)C1 99435,N1(C(CCc2[nH]c(=N)sc2)=O)CCC2(CCCN2C(=O)CC2CCCC(O)C2)C1 99436,c1(OCC)cc(C(=O)N(CC(C)O)CCOCCO)[nH]n1.C1(=O)C(C)N1.O 99437,C1(C(=O)NCC2(O)CC(NC(c3cc(F)c[nH]3)=O)C2)CC2C=CCC(C1)C2 99438,O=C1NC(=O)C(CNC(C2CC23CC(NC(c2[nH]nnc2C2CC2)=O)C3)=O)N1 99439,C1(N(c2cccnc2OCC(F)F)C(C)=O)CCN(C(=O)C(C)(C)CO)CC1C 99440,CCC1=NOC(C(=O)N(C2(C(=O)NC3CCNC(=O)C3)CCC2)C2CC2)C1 99441,C(CC(C)NC(=O)CNC(=O)OC1CCCC1)OCC 99442,N1(C(C(F)OC)=O)C2CCC1CC(NC(C1CC3CCC(C1)C3)=O)C2 99443,C(=O)(CC(COC)NC(C12CCC(NC(C)C(F)(F)F)C1C2)=O)OC 99444,C1(N(C(CC2(CSC)CC2)=O)CC(C)C)CCN(C(c2cncnc2)=O)CC1 99445,C(=O)(CCC(C(C)O)NC(c1ccc(Br)cc1F)C(c1ccccc1)=O)OC 99446,c1(C(N2CC(C(C)NC(=O)C(C)SC(F)(F)F)C2)=O)coc2c1C(=O)CCC2 99447,CC1CN(C(C2CC(C)(F)C2)=O)CCCN1C(c1cnc(C(F)(F)F)nc1)=O 99448,Cc1ccc(S(=O)(=O)Nc2cccc3c2CCO3)cc1NC(c1ccco1)=O 99449,N1(C(CN(C(C(C)C)=O)C)=O)CCC(CNC(=O)C(C(C)C)N(C)C)C12CC2 99450,C(=O)(CCCC(C)(C)C)N1CC(COC)N(C(=O)C(C#N)C(C)C)CC1 99451,C1(C(C)NC(C(CC)SC)=O)CCCN1C(C1(CO)CCCCC1)=O 99452,c1(C(N(CC(CC)NC(c2nc(=N)cc[nH]2)=O)C)=O)ccc(N(C)C)c(F)c1 99453,Cc1nc(Cl)nc(N2CC3CC2(C(=O)NCCC2CCC(C)(C)CO2)C3)c1[N+](=O)[O-] 99454,Cc1c(C(=O)NCC2CC2NC(=O)CCn2cnc(=N)[nH]2)[nH]c2c1CCCC2 99455,c1(C(N(C2CN(C(C(N3CC(C)C3)C)=O)C2)C)=O)nc(C(C)C)ncc1Br 99456,C(C)(C(C)C(=O)NC1CCC(C(C)O)CC1)NC(c1c(C)snn1)=O 99457,c12ccc(cc1)CNC(=O)N1CCCC1C2.N1(CCC#N)CCCC1 99458,c1(C(NOCC(=O)NC)=O)c(CCc2c(C)ncs2)cccc1C 99459,CC(C)C(C)(Cc1cncn1C)C(=O)NC(C)CCc1ccccc1 99460,c1(CC)cnc(C(=O)NC(c2cccc(C)c2)CNC(=O)C(=O)C(C)C)nc1 99461,n1(CCNC(C(C2CC2(C)C)N(CCOC)C2CC2)=O)ncn1C 99462,Cc1cc(Cc2nc(-c3cncnc3)nn2C(C)C(C)C)ccc1Br